C[C@@H]1CN(C(=O)Nc2ccc3ccccc3n2)CC[C@H]1NC(=O)OC(C)(C)C ZINC000880500045 GI On-Demand Anodyne SMO 37 43 C[C@H]1CN(C(=O)Nc2ccc3ccccc3n2)CC[C@H]1NC(=O)OC(C)(C)C ZINC000880500047 GI On-Demand Anodyne SMO 37 43 C[C@H]1CN(C(=O)Nc2ccc3ccccc3n2)CC[C@@H]1NC(=O)OC(C)(C)C ZINC000880500049 GI On-Demand Anodyne SMO 37 43 C[C@@H]1CN(C(=O)Nc2ccc3ccccc3n2)CC[C@@H]1NC(=O)OC(C)(C)C ZINC000880500052 GI On-Demand Anodyne SMO 37 43 CCOC(=O)[C@H](C)N1CC[C@@]2(CN(Cc3ccccc3)C[C@H](C)O2)C1 ZINC000880500071 EE On-Demand Anodyne SIGMAR1 32 43 CCOC(=O)[C@H](C)N1CC[C@@]2(CN(Cc3ccccc3)C[C@@H](C)O2)C1 ZINC000880500073 EE On-Demand Anodyne SIGMAR1 32 43 CCOC(=O)[C@H](C)N1CC[C@]2(CN(Cc3ccccc3)C[C@@H](C)O2)C1 ZINC000880500075 EE On-Demand Anodyne SIGMAR1 32 43 CCOC(=O)[C@H](C)N1CC[C@]2(CN(Cc3ccccc3)C[C@H](C)O2)C1 ZINC000880500077 EE On-Demand Anodyne SIGMAR1 32 43 Cc1ccccc1[C@H](CC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C)NC(N)=O ZINC000880500079 GD On-Demand Anodyne CTSA 49 34 Cc1ccccc1[C@H](CC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C)NC(N)=O ZINC000880500082 GD On-Demand Anodyne CTSA 49 34 Cc1ccccc1[C@H](CC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C)NC(N)=O ZINC000880500084 GD On-Demand Anodyne CTSA 49 34 Cc1ccccc1[C@H](CC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C)NC(N)=O ZINC000880500086 GD On-Demand Anodyne CTSA 49 34 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCNS(C)(=O)=O)C2)O1 ZINC000880500098 FC On-Demand Anodyne SIGMAR1 55 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCNS(C)(=O)=O)C2)O1 ZINC000880500101 FC On-Demand Anodyne SIGMAR1 55 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCNS(C)(=O)=O)C2)O1 ZINC000880500102 FC On-Demand Anodyne SIGMAR1 55 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCNS(C)(=O)=O)C2)O1 ZINC000880500104 FC On-Demand Anodyne SIGMAR1 55 40 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880500167 DE On-Demand Anodyne NPY5R 18 53 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880500167 DE On-Demand Anodyne SMO 29 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H]3CNC(=O)C3)C2)O1 ZINC000880500247 ED On-Demand Anodyne SIGMAR1 45 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H]3CNC(=O)C3)C2)O1 ZINC000880500248 ED On-Demand Anodyne SIGMAR1 45 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H]3CNC(=O)C3)C2)O1 ZINC000880500249 ED On-Demand Anodyne SIGMAR1 45 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H]3CNC(=O)C3)C2)O1 ZINC000880500250 ED On-Demand Anodyne SIGMAR1 45 38 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880500255 FG On-Demand Anodyne SMO 43 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cnns3)C2)O1 ZINC000880500256 EE On-Demand Anodyne SIGMAR1 41 37 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cnns3)C2)O1 ZINC000880500257 EE On-Demand Anodyne SIGMAR1 41 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cnns3)C2)O1 ZINC000880500258 EE On-Demand Anodyne SIGMAR1 41 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cnns3)C2)O1 ZINC000880500259 EE On-Demand Anodyne SIGMAR1 41 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3nc(C#N)cs3)C2)O1 ZINC000880500272 FF On-Demand Mild SIGMAR1 32 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3nc(C#N)cs3)C2)O1 ZINC000880500273 FF On-Demand Mild SIGMAR1 32 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3nc(C#N)cs3)C2)O1 ZINC000880500274 FF On-Demand Mild SIGMAR1 32 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3nc(C#N)cs3)C2)O1 ZINC000880500275 FF On-Demand Mild SIGMAR1 32 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H](O)C(C)(C)C)C2)O1 ZINC000880500383 EF On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H](O)C(C)(C)C)C2)O1 ZINC000880500384 EF On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H](O)C(C)(C)C)C2)O1 ZINC000880500386 EF On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H](O)C(C)(C)C)C2)O1 ZINC000880500388 EF On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H]3CCC(=O)O3)C2)O1 ZINC000880500481 EE On-Demand Anodyne SIGMAR1 51 43 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H]3CCC(=O)O3)C2)O1 ZINC000880500482 EE On-Demand Anodyne SIGMAR1 51 43 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H]3CCC(=O)O3)C2)O1 ZINC000880500483 EE On-Demand Anodyne SIGMAR1 51 43 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H]3CCC(=O)O3)C2)O1 ZINC000880500485 EE On-Demand Anodyne SIGMAR1 51 43 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCS(C)(=O)=O)C2)O1 ZINC000880500570 FD On-Demand Anodyne SIGMAR1 53 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCS(C)(=O)=O)C2)O1 ZINC000880500572 FD On-Demand Anodyne SIGMAR1 53 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCS(C)(=O)=O)C2)O1 ZINC000880500575 FD On-Demand Anodyne SIGMAR1 53 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCS(C)(=O)=O)C2)O1 ZINC000880500577 FD On-Demand Anodyne SIGMAR1 53 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3nccs3)C2)O1 ZINC000880500590 EG On-Demand Anodyne SIGMAR1 42 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3nccs3)C2)O1 ZINC000880500592 EG On-Demand Anodyne SIGMAR1 42 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3nccs3)C2)O1 ZINC000880500594 EG On-Demand Anodyne SIGMAR1 42 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3nccs3)C2)O1 ZINC000880500596 EG On-Demand Anodyne SIGMAR1 42 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500641 ED On-Demand Anodyne CHRM2 16 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500641 ED On-Demand Anodyne DRD4 38 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500641 ED On-Demand Anodyne CHRM3 17 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500641 ED On-Demand Anodyne SIGMAR1 61 49 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500643 ED On-Demand Anodyne CHRM2 16 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500643 ED On-Demand Anodyne DRD4 38 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500643 ED On-Demand Anodyne CHRM3 17 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500643 ED On-Demand Anodyne SIGMAR1 61 49 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500645 ED On-Demand Anodyne CHRM2 16 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500645 ED On-Demand Anodyne DRD4 38 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500645 ED On-Demand Anodyne CHRM3 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500645 ED On-Demand Anodyne SIGMAR1 61 49 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500648 ED On-Demand Anodyne CHRM2 16 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500648 ED On-Demand Anodyne DRD4 38 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500648 ED On-Demand Anodyne CHRM3 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC3CC3)C2)O1 ZINC000880500648 ED On-Demand Anodyne SIGMAR1 61 49 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500664 EF On-Demand Anodyne CHRM2 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500664 EF On-Demand Anodyne CHRM3 16 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500664 EF On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500666 EF On-Demand Anodyne CHRM2 18 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500666 EF On-Demand Anodyne CHRM3 16 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500666 EF On-Demand Anodyne SIGMAR1 62 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500668 EF On-Demand Anodyne CHRM2 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500668 EF On-Demand Anodyne CHRM3 16 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500668 EF On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500669 EF On-Demand Anodyne CHRM2 18 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500669 EF On-Demand Anodyne CHRM3 16 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)C3CC3)C2)O1 ZINC000880500669 EF On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC3(O)CCOCC3)C2)O1 ZINC000880500671 FD On-Demand Anodyne SIGMAR1 43 38 CNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500672 ED On-Demand Anodyne SIGMAR1 56 39 CNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500672 ED On-Demand Anodyne NPFFR1 42 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC3(O)CCOCC3)C2)O1 ZINC000880500674 FD On-Demand Anodyne SIGMAR1 43 38 CNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500676 ED On-Demand Anodyne SIGMAR1 56 39 CNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500676 ED On-Demand Anodyne NPFFR1 42 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC3(O)CCOCC3)C2)O1 ZINC000880500677 FD On-Demand Anodyne SIGMAR1 43 38 CNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500681 ED On-Demand Anodyne SIGMAR1 56 39 CNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500681 ED On-Demand Anodyne NPFFR1 42 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC3(O)CCOCC3)C2)O1 ZINC000880500682 FD On-Demand Anodyne SIGMAR1 43 38 CNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500686 ED On-Demand Anodyne SIGMAR1 56 39 CNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500686 ED On-Demand Anodyne NPFFR1 42 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@@H]3CCCN3C)C2)O1 ZINC000880500722 FF On-Demand Anodyne SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@@H]3CCCN3C)C2)O1 ZINC000880500722 FF On-Demand Anodyne CHRNA10 43 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@H]3CCCN3C)C2)O1 ZINC000880500727 FF On-Demand Anodyne SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@H]3CCCN3C)C2)O1 ZINC000880500727 FF On-Demand Anodyne CHRNA10 43 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@H]3CCCN3C)C2)O1 ZINC000880500733 FF On-Demand Anodyne SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@H]3CCCN3C)C2)O1 ZINC000880500733 FF On-Demand Anodyne CHRNA10 43 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@@H]3CCCN3C)C2)O1 ZINC000880500738 FF On-Demand Anodyne SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@@H]3CCCN3C)C2)O1 ZINC000880500738 FF On-Demand Anodyne CHRNA10 43 37 COc1coc(CN2CC[C@@]3(C2)CN(Cc2ccccc2)C[C@H](C)O3)cc1=O ZINC000880500800 GF On-Demand Anodyne SIGMAR1 36 40 COc1coc(CN2CC[C@]3(C2)CN(Cc2ccccc2)C[C@H](C)O3)cc1=O ZINC000880500804 GF On-Demand Anodyne SIGMAR1 36 40 COc1coc(CN2CC[C@@]3(C2)CN(Cc2ccccc2)C[C@@H](C)O3)cc1=O ZINC000880500810 GF On-Demand Anodyne SIGMAR1 36 40 COc1coc(CN2CC[C@]3(C2)CN(Cc2ccccc2)C[C@@H](C)O3)cc1=O ZINC000880500814 GF On-Demand Anodyne SIGMAR1 36 40 C=CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500842 CF On-Demand Mild SIGMAR1 55 45 C=CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500844 CF On-Demand Mild SIGMAR1 55 45 C=CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880500845 CF On-Demand Mild SIGMAR1 55 45 C=CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880500846 CF On-Demand Mild SIGMAR1 55 45 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)N1CCCCC1 ZINC000880500847 FD On-Demand Anodyne SAP2 24 41 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)N1CCCCC1 ZINC000880500848 FD On-Demand Anodyne SAP2 24 41 Cc1ccccc1CN1CCC(NC(=O)CN[C@@H]2CCC[C@@]23CCCO3)CC1 ZINC000880500862 GF On-Demand Anodyne SIGMAR1 15 43 Cc1ccccc1CN1CCC(NC(=O)CN[C@@H]2CCC[C@]23CCCO3)CC1 ZINC000880500863 GF On-Demand Anodyne SIGMAR1 15 43 Cc1ccccc1CN1CCC(NC(=O)CN[C@H]2CCC[C@]23CCCO3)CC1 ZINC000880500864 GF On-Demand Anodyne SIGMAR1 15 43 Cc1ccccc1CN1CCC(NC(=O)CN[C@H]2CCC[C@@]23CCCO3)CC1 ZINC000880500865 GF On-Demand Anodyne SIGMAR1 15 43 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cc(=O)c(O)co3)C2)O1 ZINC000880500889 FE On-Demand Anodyne DAO 18 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cc(=O)c(O)co3)C2)O1 ZINC000880500891 FE On-Demand Anodyne DAO 18 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cc(=O)c(O)co3)C2)O1 ZINC000880500892 FE On-Demand Anodyne DAO 18 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cc(=O)c(O)co3)C2)O1 ZINC000880500894 FE On-Demand Anodyne DAO 18 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500904 EC On-Demand Mild SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500904 EC On-Demand Mild NPFFR1 41 35 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500905 EC On-Demand Mild SIGMAR1 48 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500905 EC On-Demand Mild NPFFR1 41 35 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500907 EC On-Demand Mild SIGMAR1 48 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500907 EC On-Demand Mild NPFFR1 41 35 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500908 EC On-Demand Mild SIGMAR1 48 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC#N)C2)O1 ZINC000880500908 EC On-Demand Mild NPFFR1 41 35 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC3OCCCO3)C2)O1 ZINC000880500913 FF On-Demand Anodyne SIGMAR1 45 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC3OCCCO3)C2)O1 ZINC000880500915 FF On-Demand Anodyne SIGMAR1 45 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC3OCCCO3)C2)O1 ZINC000880500916 FF On-Demand Anodyne SIGMAR1 45 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC3OCCCO3)C2)O1 ZINC000880500917 FF On-Demand Anodyne SIGMAR1 45 38 CCCCCCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880500929 CF On-Demand Anodyne LUXR 29 42 CCCCCCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880500929 CF On-Demand Anodyne LASR 57 42 CCCCCCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880500931 CF On-Demand Anodyne LUXR 29 42 CCCCCCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880500931 CF On-Demand Anodyne LASR 57 42 CCCCCCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880500932 CF On-Demand Anodyne LUXR 29 42 CCCCCCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880500932 CF On-Demand Anodyne LASR 57 42 CCCCCCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880500934 CF On-Demand Anodyne LUXR 29 42 CCCCCCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880500934 CF On-Demand Anodyne LASR 57 42 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)N1CCCCCC1 ZINC000880501081 GD On-Demand Anodyne SAP2 24 41 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)N1CCCCCC1 ZINC000880501082 GD On-Demand Anodyne SAP2 24 41 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCC1 ZINC000880501083 FD On-Demand Anodyne DRD4 15 40 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCC1 ZINC000880501083 FD On-Demand Anodyne SIGMAR1 38 48 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCC1 ZINC000880501084 FD On-Demand Anodyne DRD4 15 40 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCC1 ZINC000880501084 FD On-Demand Anodyne SIGMAR1 38 48 CN(C)C(=O)Nc1cccc(C(=O)N[C@H]2C[C@@H](N3CCOCC3)C2(C)C)c1 ZINC000880501085 FE On-Demand Anodyne EPHX2 15 41 CN(C)C(=O)Nc1cccc(C(=O)N[C@@H]2C[C@@H](N3CCOCC3)C2(C)C)c1 ZINC000880501086 FE On-Demand Anodyne EPHX2 15 41 CN(C)C(=O)Nc1cccc(C(=O)N[C@H]2C[C@H](N3CCOCC3)C2(C)C)c1 ZINC000880501087 FE On-Demand Anodyne EPHX2 15 41 CN(C)C(=O)Nc1cccc(C(=O)N[C@@H]2C[C@H](N3CCOCC3)C2(C)C)c1 ZINC000880501088 FE On-Demand Anodyne EPHX2 15 41 O=C(Nc1ccc2ccccc2n1)N1CCN2C(=O)OC[C@H]2C1 ZINC000880501120 DD On-Demand Anodyne SMO 54 41 O=C(Nc1ccc2ccccc2n1)N1CCN2C(=O)OC[C@@H]2C1 ZINC000880501121 DD On-Demand Anodyne SMO 54 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)N3CCOCC3)C2)O1 ZINC000880501126 GD On-Demand Anodyne SIGMAR1 40 36 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)N3CCOCC3)C2)O1 ZINC000880501127 GD On-Demand Anodyne SIGMAR1 40 36 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)N3CCOCC3)C2)O1 ZINC000880501128 GD On-Demand Anodyne SIGMAR1 40 36 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)N3CCOCC3)C2)O1 ZINC000880501129 GD On-Demand Anodyne SIGMAR1 40 36 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CC1 ZINC000880501130 EC On-Demand Anodyne SIGMAR1 42 50 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CC1 ZINC000880501131 EC On-Demand Anodyne SIGMAR1 42 50 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc2ccccc2n1 ZINC000880501132 GG On-Demand Anodyne EPHX2 22 47 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc2ccccc2n1 ZINC000880501132 GG On-Demand Anodyne SMO 36 42 O=C(Nc1ccc2ccccc2n1)N1CCC(CCCO)CC1 ZINC000880501152 DG On-Demand Anodyne SMO 43 42 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880501174 FG On-Demand Anodyne CCR8 48 31 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880501174 FG On-Demand Anodyne SMO 42 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(C)(C)O)C2)O1 ZINC000880501176 EF On-Demand Anodyne SIGMAR1 54 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(C)(C)O)C2)O1 ZINC000880501177 EF On-Demand Anodyne SIGMAR1 54 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(C)(C)O)C2)O1 ZINC000880501178 EF On-Demand Anodyne SIGMAR1 54 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(C)(C)O)C2)O1 ZINC000880501179 EF On-Demand Anodyne SIGMAR1 54 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccnc3)C2)O1 ZINC000880501180 EF On-Demand Anodyne SIGMAR1 45 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccnc3)C2)O1 ZINC000880501181 EF On-Demand Anodyne SIGMAR1 45 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccnc3)C2)O1 ZINC000880501182 EF On-Demand Anodyne SIGMAR1 45 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccnc3)C2)O1 ZINC000880501183 EF On-Demand Anodyne SIGMAR1 45 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCc3cccnc3)C2)O1 ZINC000880501198 FF On-Demand Anodyne SIGMAR1 42 43 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCc3cccnc3)C2)O1 ZINC000880501199 FF On-Demand Anodyne SIGMAR1 42 43 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCc3cccnc3)C2)O1 ZINC000880501200 FF On-Demand Anodyne SIGMAR1 42 43 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCc3cccnc3)C2)O1 ZINC000880501201 FF On-Demand Anodyne SIGMAR1 42 43 C#CCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501202 DF On-Demand Mild SIGMAR1 49 38 C#CCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501203 DF On-Demand Mild SIGMAR1 49 38 C#CCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501204 DF On-Demand Mild SIGMAR1 49 38 C#CCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501205 DF On-Demand Mild SIGMAR1 49 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C/C=C/Cl)C2)O1 ZINC000880501230 DG On-Demand Anodyne SIGMAR1 50 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C/C=C\Cl)C2)O1 ZINC000880501231 DG On-Demand Anodyne SIGMAR1 50 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C/C=C/Cl)C2)O1 ZINC000880501232 DG On-Demand Anodyne SIGMAR1 50 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C/C=C\Cl)C2)O1 ZINC000880501233 DG On-Demand Anodyne SIGMAR1 50 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@H](C)C(=O)NC(N)=O)C2)O1 ZINC000880501242 FC On-Demand Anodyne NPFFR1 40 35 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@H](C)C(=O)NC(N)=O)C2)O1 ZINC000880501244 FC On-Demand Anodyne NPFFR1 40 35 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501256 GE On-Demand Anodyne SIGMAR1 33 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501256 GE On-Demand Anodyne MAP1 76 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501259 GE On-Demand Anodyne SIGMAR1 33 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501259 GE On-Demand Anodyne MAP1 76 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501261 GE On-Demand Anodyne SIGMAR1 33 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501261 GE On-Demand Anodyne MAP1 76 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501263 GE On-Demand Anodyne SIGMAR1 33 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3nccs3)C2)O1 ZINC000880501263 GE On-Demand Anodyne MAP1 76 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCO)C2)O1 ZINC000880501265 DE On-Demand Anodyne SIGMAR1 78 44 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCO)C2)O1 ZINC000880501267 DE On-Demand Anodyne SIGMAR1 78 44 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCO)C2)O1 ZINC000880501269 DE On-Demand Anodyne SIGMAR1 78 44 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCO)C2)O1 ZINC000880501271 DE On-Demand Anodyne SIGMAR1 78 44 CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501272 DD On-Demand Anodyne SIGMAR1 64 40 CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501272 DD On-Demand Anodyne NPFFR1 43 38 CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501274 DD On-Demand Anodyne SIGMAR1 64 40 CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501274 DD On-Demand Anodyne NPFFR1 43 38 CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501276 DD On-Demand Anodyne SIGMAR1 64 40 CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501276 DD On-Demand Anodyne NPFFR1 43 38 CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501277 DD On-Demand Anodyne SIGMAR1 64 40 CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501277 DD On-Demand Anodyne NPFFR1 43 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCCO)C2)O1 ZINC000880501291 EF On-Demand Anodyne SIGMAR1 72 44 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCCO)C2)O1 ZINC000880501293 EF On-Demand Anodyne SIGMAR1 72 44 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCCO)C2)O1 ZINC000880501295 EF On-Demand Anodyne SIGMAR1 72 44 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCCO)C2)O1 ZINC000880501297 EF On-Demand Anodyne SIGMAR1 72 44 C#CCN1CCC[C@H]1C(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501300 DC On-Demand Mild HSD11B1 44 35 C#CCN1CCC[C@H]1C(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501302 DC On-Demand Mild HSD11B1 44 35 C#CCN1CCC[C@H]1C(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501305 DC On-Demand Mild HSD11B1 44 35 C#CCN1CCC[C@H]1C(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501307 DC On-Demand Mild HSD11B1 44 35 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880501309 GB On-Demand Anodyne SIGMAR1 29 40 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880501309 GB On-Demand Anodyne NPFFR1 42 38 CC(C)(C)OC(=O)N1CC[C@H](CCN[C@H]2CCC[C@]23CCCO3)C1 ZINC000880501320 EG On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CC[C@H](CCN[C@@H]2CCC[C@]23CCCO3)C1 ZINC000880501321 EG On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CC[C@H](CCN[C@@H]2CCC[C@@]23CCCO3)C1 ZINC000880501322 EG On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CC[C@H](CCN[C@H]2CCC[C@@]23CCCO3)C1 ZINC000880501323 EG On-Demand Anodyne GPR119 21 41 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880501344 GB On-Demand Anodyne SIGMAR1 29 40 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880501344 GB On-Demand Anodyne NPFFR1 42 38 CC(C)(C)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880501352 EH On-Demand Anodyne EPHX2 39 44 O=C(Nc1ccc2ccccc2n1)N1CCCC2(C1)OCCO2 ZINC000880501431 DF On-Demand Anodyne SMO 41 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N3CCOCC3)C2)O1 ZINC000880501438 FD On-Demand Anodyne SIGMAR1 43 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N3CCOCC3)C2)O1 ZINC000880501440 FD On-Demand Anodyne SIGMAR1 43 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N3CCOCC3)C2)O1 ZINC000880501443 FD On-Demand Anodyne SIGMAR1 43 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N3CCOCC3)C2)O1 ZINC000880501445 FD On-Demand Anodyne SIGMAR1 43 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501448 EC On-Demand Anodyne SIGMAR1 51 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501448 EC On-Demand Anodyne NPFFR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501452 EC On-Demand Anodyne SIGMAR1 51 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501452 EC On-Demand Anodyne NPFFR1 46 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501454 EC On-Demand Anodyne SIGMAR1 51 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501454 EC On-Demand Anodyne NPFFR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501456 EC On-Demand Anodyne SIGMAR1 51 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(N)=O)C2)O1 ZINC000880501456 EC On-Demand Anodyne NPFFR1 46 38 C[C@@H]1CN(CCN2CC[C@@]3(C2)CN(Cc2ccccc2)C[C@@H](C)O3)CCO1 ZINC000880501517 FE On-Demand Anodyne SIGMAR1 49 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCN3CCO[C@H](C)C3)C2)O1 ZINC000880501518 FE On-Demand Anodyne SIGMAR1 49 39 C[C@@H]1CN(CCN2CC[C@]3(C2)CN(Cc2ccccc2)C[C@@H](C)O3)CCO1 ZINC000880501519 FE On-Demand Anodyne SIGMAR1 49 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCN3CCO[C@H](C)C3)C2)O1 ZINC000880501520 FE On-Demand Anodyne SIGMAR1 49 39 CCCCCCCCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501521 DG On-Demand Mild LUXR 29 42 CCCCCCCCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501521 DG On-Demand Mild LASR 57 42 CCCCCCCCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501522 DG On-Demand Mild LUXR 29 42 CCCCCCCCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880501522 DG On-Demand Mild LASR 57 42 CCCCCCCCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501523 DG On-Demand Mild LUXR 29 42 CCCCCCCCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501523 DG On-Demand Mild LASR 57 42 CCCCCCCCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501524 DG On-Demand Mild LUXR 29 42 CCCCCCCCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880501524 DG On-Demand Mild LASR 57 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cncc(F)c3)C2)O1 ZINC000880501525 FG On-Demand Anodyne SIGMAR1 41 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cncc(F)c3)C2)O1 ZINC000880501526 FG On-Demand Anodyne SIGMAR1 41 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cncc(F)c3)C2)O1 ZINC000880501527 FG On-Demand Anodyne SIGMAR1 41 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cncc(F)c3)C2)O1 ZINC000880501528 FG On-Demand Anodyne SIGMAR1 41 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCCCO)C2)O1 ZINC000880501618 EF On-Demand Anodyne SIGMAR1 72 44 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCCCCO)C2)O1 ZINC000880501624 EF On-Demand Anodyne SIGMAR1 72 44 CCN(C)C(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501627 ED On-Demand Anodyne SIGMAR1 48 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCCCO)C2)O1 ZINC000880501629 EF On-Demand Anodyne SIGMAR1 72 44 CCN(C)C(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501630 ED On-Demand Anodyne SIGMAR1 48 42 CCN(C)C(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501632 ED On-Demand Anodyne SIGMAR1 48 42 CCN(C)C(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501634 ED On-Demand Anodyne SIGMAR1 48 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCCCCO)C2)O1 ZINC000880501635 EF On-Demand Anodyne SIGMAR1 72 44 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3ccc(O)cc3)C2)O1 ZINC000880501696 GF On-Demand Anodyne SIGMAR1 40 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3ccc(O)cc3)C2)O1 ZINC000880501700 GF On-Demand Anodyne SIGMAR1 40 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)Nc3ccc(O)cc3)C2)O1 ZINC000880501702 GF On-Demand Anodyne SIGMAR1 40 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)Nc3ccc(O)cc3)C2)O1 ZINC000880501706 GF On-Demand Anodyne SIGMAR1 40 38 COc1cccc(OC)c1OCCCCN[C@H]1CCC[C@@]12CCCO2 ZINC000880501718 EH On-Demand Anodyne ADRA1A 15 40 COc1cccc(OC)c1OCCCCN[C@H]1CCC[C@]12CCCO2 ZINC000880501723 EH On-Demand Anodyne ADRA1A 15 40 C#CCOc1ccc(C(=O)N[C@@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501731 ED On-Demand Mild MMP13 15 41 C#CCOc1ccc(C(=O)N[C@@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501731 ED On-Demand Mild ADAM17 39 41 C#CCOc1ccc(C(=O)N[C@@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501737 ED On-Demand Mild MMP13 15 41 C#CCOc1ccc(C(=O)N[C@@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501737 ED On-Demand Mild ADAM17 39 41 C#CCOc1ccc(C(=O)N[C@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501738 ED On-Demand Mild MMP13 15 41 C#CCOc1ccc(C(=O)N[C@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501738 ED On-Demand Mild ADAM17 39 41 C#CCOc1ccc(C(=O)N[C@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501740 ED On-Demand Mild MMP13 15 41 C#CCOc1ccc(C(=O)N[C@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880501740 ED On-Demand Mild ADAM17 39 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCn3cccn3)C2)O1 ZINC000880501742 EE On-Demand Anodyne SIGMAR1 44 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCn3cccn3)C2)O1 ZINC000880501744 EE On-Demand Anodyne SIGMAR1 44 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCn3cccn3)C2)O1 ZINC000880501745 EE On-Demand Anodyne SIGMAR1 44 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCn3cccn3)C2)O1 ZINC000880501747 EE On-Demand Anodyne SIGMAR1 44 38 C[C@H](C(=O)N1CCCCCC1)N1CC[C@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880501748 GE On-Demand Anodyne DPP7 48 35 C[C@@H](C(=O)N1CCCCCC1)N1CC[C@@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880501749 GE On-Demand Anodyne DPP7 48 35 C[C@@H](C(=O)N1CCCCCC1)N1CC[C@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880501750 GE On-Demand Anodyne DPP7 48 35 C[C@H](C(=O)N1CCCCCC1)N1CC[C@@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880501751 GE On-Demand Anodyne DPP7 48 35 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCC(C)(C)C#N)C2)O1 ZINC000880501762 FH On-Demand Mild CCR1 26 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCC(C)(C)C#N)C2)O1 ZINC000880501765 FH On-Demand Mild CCR1 26 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCC(C)(C)C#N)C2)O1 ZINC000880501768 FH On-Demand Mild CCR1 26 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCC(C)(C)C#N)C2)O1 ZINC000880501772 FH On-Demand Mild CCR1 26 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)N3CCCCC3)C2)O1 ZINC000880501778 GF On-Demand Anodyne SIGMAR1 47 37 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)N3CCCCC3)C2)O1 ZINC000880501780 GF On-Demand Anodyne SIGMAR1 47 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)N3CCCCC3)C2)O1 ZINC000880501781 GF On-Demand Anodyne SIGMAR1 47 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)N3CCCCC3)C2)O1 ZINC000880501783 GF On-Demand Anodyne SIGMAR1 47 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501788 FF On-Demand Anodyne CYP11B1 16 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501788 FF On-Demand Anodyne TBXAS1 20 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501791 FF On-Demand Anodyne CYP11B1 16 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501791 FF On-Demand Anodyne TBXAS1 20 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501793 FF On-Demand Anodyne CYP11B1 16 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501793 FF On-Demand Anodyne TBXAS1 20 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501794 FF On-Demand Anodyne CYP11B1 16 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCn3ccnc3)C2)O1 ZINC000880501794 FF On-Demand Anodyne TBXAS1 20 41 C[C@@](CO)(NC(=O)Nc1ccc2ccccc2n1)C1CC1 ZINC000880501799 CF On-Demand Anodyne MTTP 40 35 C=CCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501809 DF On-Demand Mild SIGMAR1 51 46 C=CCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501810 DF On-Demand Mild SIGMAR1 51 46 COc1cccc(OC)c1OCCCCN[C@@H]1CCC[C@]12CCCO2 ZINC000880501811 EH On-Demand Anodyne ADRA1A 15 40 C=CCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501812 DF On-Demand Mild SIGMAR1 51 46 C=CCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501813 DF On-Demand Mild SIGMAR1 51 46 COc1cccc(OC)c1OCCCCN[C@@H]1CCC[C@@]12CCCO2 ZINC000880501814 EH On-Demand Anodyne ADRA1A 15 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@@H]3CCCO3)C2)O1 ZINC000880501859 EF On-Demand Anodyne SIGMAR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@@H]3CCCO3)C2)O1 ZINC000880501861 EF On-Demand Anodyne SIGMAR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC[C@H]3CCCO3)C2)O1 ZINC000880501863 EF On-Demand Anodyne SIGMAR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC[C@H]3CCCO3)C2)O1 ZINC000880501866 EF On-Demand Anodyne SIGMAR1 46 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCNC(=O)C(F)(F)F)C2)O1 ZINC000880501910 GE On-Demand Anodyne SIGMAR1 41 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCNC(=O)C(F)(F)F)C2)O1 ZINC000880501912 GE On-Demand Anodyne SIGMAR1 41 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCNC(=O)C(F)(F)F)C2)O1 ZINC000880501914 GE On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCNC(=O)C(F)(F)F)C2)O1 ZINC000880501916 GE On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCc3cccnc3)C2)O1 ZINC000880501965 GE On-Demand Anodyne NAMPT 58 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCc3cccnc3)C2)O1 ZINC000880501967 GE On-Demand Anodyne NAMPT 58 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCc3cccnc3)C2)O1 ZINC000880501970 GE On-Demand Anodyne NAMPT 58 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCc3cccnc3)C2)O1 ZINC000880501972 GE On-Demand Anodyne NAMPT 58 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3ncccn3)C2)O1 ZINC000880501974 EE On-Demand Anodyne SIGMAR1 49 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3ncccn3)C2)O1 ZINC000880501977 EE On-Demand Anodyne SIGMAR1 49 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3ncccn3)C2)O1 ZINC000880501979 EE On-Demand Anodyne SIGMAR1 49 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3ncccn3)C2)O1 ZINC000880501981 EE On-Demand Anodyne SIGMAR1 49 40 C#CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501993 ED On-Demand Mild SIGMAR1 44 38 C#CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501993 ED On-Demand Mild NPFFR1 40 35 C#CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501994 ED On-Demand Mild SIGMAR1 44 38 C#CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880501994 ED On-Demand Mild NPFFR1 40 35 C#CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501995 ED On-Demand Mild SIGMAR1 44 38 C#CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501995 ED On-Demand Mild NPFFR1 40 35 C#CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501996 ED On-Demand Mild SIGMAR1 44 38 C#CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880501996 ED On-Demand Mild NPFFR1 40 35 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502017 ED On-Demand Anodyne DRD4 24 46 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502017 ED On-Demand Anodyne OPRM1 15 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502017 ED On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502018 ED On-Demand Anodyne DRD4 24 46 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502018 ED On-Demand Anodyne OPRM1 15 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502018 ED On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502019 ED On-Demand Anodyne DRD4 24 46 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502019 ED On-Demand Anodyne OPRM1 15 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502019 ED On-Demand Anodyne SIGMAR1 62 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502020 ED On-Demand Anodyne DRD4 24 46 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502020 ED On-Demand Anodyne OPRM1 15 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N(C)C)C2)O1 ZINC000880502020 ED On-Demand Anodyne SIGMAR1 62 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne CHRM2 15 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne OPRM1 21 57 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne OPRD1 17 52 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne OPRK1 23 57 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne CHRM3 21 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne SIGMAR1 55 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne MCHR2 52 33 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502035 GF On-Demand Anodyne NPFFR1 47 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne CHRM2 15 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne OPRM1 21 57 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne OPRD1 17 52 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne OPRK1 23 57 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne CHRM3 21 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne SIGMAR1 55 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne MCHR2 52 33 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502036 GF On-Demand Anodyne NPFFR1 47 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne CHRM2 15 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne OPRM1 21 57 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne OPRD1 17 52 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne OPRK1 23 57 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne CHRM3 21 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne SIGMAR1 55 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne MCHR2 52 33 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502037 GF On-Demand Anodyne NPFFR1 47 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne CHRM2 15 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne OPRM1 21 57 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne OPRD1 17 52 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne OPRK1 23 57 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne CHRM3 21 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne SIGMAR1 55 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne MCHR2 52 33 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cccc(C(N)=O)c3)C2)O1 ZINC000880502038 GF On-Demand Anodyne NPFFR1 47 37 NC(=O)c1ccc(CN2CC[C@@]3(C2)CN(Cc2ccccc2)C(=O)CO3)cc1 ZINC000880502057 GD On-Demand Anodyne SIGMAR1 42 39 NC(=O)c1ccc(CN2CC[C@@]3(C2)CN(Cc2ccccc2)C(=O)CO3)cc1 ZINC000880502057 GD On-Demand Anodyne NPFFR1 48 40 NC(=O)c1ccc(CN2CC[C@]3(C2)CN(Cc2ccccc2)C(=O)CO3)cc1 ZINC000880502058 GD On-Demand Anodyne SIGMAR1 42 39 NC(=O)c1ccc(CN2CC[C@]3(C2)CN(Cc2ccccc2)C(=O)CO3)cc1 ZINC000880502058 GD On-Demand Anodyne NPFFR1 48 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCO)C2)O1 ZINC000880502075 DD On-Demand Anodyne SIGMAR1 74 45 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCO)C2)O1 ZINC000880502076 DD On-Demand Anodyne SIGMAR1 74 45 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCO)C2)O1 ZINC000880502077 DD On-Demand Anodyne SIGMAR1 74 45 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCO)C2)O1 ZINC000880502078 DD On-Demand Anodyne SIGMAR1 74 45 c1ccc(CN2CC[C@H](N[C@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502186 DF On-Demand Anodyne DRD4 35 42 c1ccc(CN2CC[C@H](N[C@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502186 DF On-Demand Anodyne SIGMAR1 54 41 c1ccc(CN2CC[C@H](N[C@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502187 DF On-Demand Anodyne DRD4 35 42 c1ccc(CN2CC[C@H](N[C@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502187 DF On-Demand Anodyne SIGMAR1 54 41 c1ccc(CN2CC[C@H](N[C@@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502188 DF On-Demand Anodyne DRD4 35 42 c1ccc(CN2CC[C@H](N[C@@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502188 DF On-Demand Anodyne SIGMAR1 54 41 c1ccc(CN2CC[C@H](N[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502189 DF On-Demand Anodyne DRD4 35 42 c1ccc(CN2CC[C@H](N[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502189 DF On-Demand Anodyne SIGMAR1 54 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC[C@@H]3CCCO3)C2)O1 ZINC000880502225 GD On-Demand Anodyne PDE8B 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC[C@@H]3CCCO3)C2)O1 ZINC000880502226 GD On-Demand Anodyne PDE8B 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC[C@H]3CCCO3)C2)O1 ZINC000880502227 GD On-Demand Anodyne PDE8B 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC[C@H]3CCCO3)C2)O1 ZINC000880502228 GD On-Demand Anodyne PDE8B 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(C)(C)C)C2)O1 ZINC000880502237 FE On-Demand Anodyne SIGMAR1 50 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(C)(C)C)C2)O1 ZINC000880502238 FE On-Demand Anodyne SIGMAR1 50 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(C)(C)C)C2)O1 ZINC000880502239 FE On-Demand Anodyne SIGMAR1 50 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(C)(C)C)C2)O1 ZINC000880502241 FE On-Demand Anodyne SIGMAR1 50 41 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1ccccc1 ZINC000880502251 GD On-Demand Anodyne SIGMAR1 32 40 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1ccccc1 ZINC000880502251 GD On-Demand Anodyne NPFFR1 43 37 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1ccccc1 ZINC000880502252 GD On-Demand Anodyne SIGMAR1 32 40 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1ccccc1 ZINC000880502252 GD On-Demand Anodyne NPFFR1 43 37 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N3CCC3)C2)O1 ZINC000880502304 ED On-Demand Anodyne SIGMAR1 53 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N3CCC3)C2)O1 ZINC000880502305 ED On-Demand Anodyne SIGMAR1 53 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)N3CCC3)C2)O1 ZINC000880502306 ED On-Demand Anodyne SIGMAR1 53 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)N3CCC3)C2)O1 ZINC000880502307 ED On-Demand Anodyne SIGMAR1 53 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502325 FC On-Demand Anodyne SIGMAR1 50 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502325 FC On-Demand Anodyne NPFFR1 43 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502364 FC On-Demand Anodyne SIGMAR1 50 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502364 FC On-Demand Anodyne NPFFR1 43 38 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502365 FC On-Demand Anodyne SIGMAR1 50 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502365 FC On-Demand Anodyne NPFFR1 43 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502366 FC On-Demand Anodyne SIGMAR1 50 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCC(=O)NC(N)=O)C2)O1 ZINC000880502366 FC On-Demand Anodyne NPFFR1 43 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502384 GE On-Demand Anodyne SIGMAR1 43 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502384 GE On-Demand Anodyne NPFFR1 40 35 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502385 GE On-Demand Anodyne SIGMAR1 43 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502385 GE On-Demand Anodyne NPFFR1 40 35 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502386 GE On-Demand Anodyne SIGMAR1 43 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502386 GE On-Demand Anodyne NPFFR1 40 35 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502387 GE On-Demand Anodyne SIGMAR1 43 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NCC(F)(F)F)C2)O1 ZINC000880502387 GE On-Demand Anodyne NPFFR1 40 35 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC(=O)NC1CC1 ZINC000880502388 GC On-Demand Anodyne SIGMAR1 31 44 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC(=O)NC1CC1 ZINC000880502389 GC On-Demand Anodyne SIGMAR1 31 44 C[C@@H](C(=O)N1CCCCC1)N1CC[C@@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880502394 GD On-Demand Anodyne DPP7 48 35 C[C@H](C(=O)N1CCCCC1)N1CC[C@@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880502395 GD On-Demand Anodyne DPP7 48 35 C[C@@H](C(=O)N1CCCCC1)N1CC[C@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880502396 GD On-Demand Anodyne DPP7 48 35 C[C@H](C(=O)N1CCCCC1)N1CC[C@]2(CN(Cc3ccccc3)C(=O)CO2)C1 ZINC000880502397 GD On-Demand Anodyne DPP7 48 35 CCOCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502407 DE On-Demand Anodyne SIGMAR1 58 41 CCOCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502408 DE On-Demand Anodyne SIGMAR1 58 41 CCOCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502409 DE On-Demand Anodyne SIGMAR1 58 41 CCOCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502410 DE On-Demand Anodyne SIGMAR1 58 41 C#CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502425 CD On-Demand Mild SIGMAR1 58 41 C#CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502426 CD On-Demand Mild SIGMAR1 58 41 C#CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502427 CD On-Demand Mild SIGMAR1 58 41 C#CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502428 CD On-Demand Mild SIGMAR1 58 41 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(F)(F)F)C2)O1 ZINC000880502435 EF On-Demand Anodyne SIGMAR1 59 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(F)(F)F)C2)O1 ZINC000880502436 EF On-Demand Anodyne SIGMAR1 59 41 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(F)(F)F)C2)O1 ZINC000880502437 EF On-Demand Anodyne SIGMAR1 59 41 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(F)(F)F)C2)O1 ZINC000880502438 EF On-Demand Anodyne SIGMAR1 59 41 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCN3CCCC3=O)C2)O1 ZINC000880502447 FD On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCN3CCCC3=O)C2)O1 ZINC000880502448 FD On-Demand Anodyne SIGMAR1 41 38 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCN3CCCC3=O)C2)O1 ZINC000880502449 FD On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCN3CCCC3=O)C2)O1 ZINC000880502450 FD On-Demand Anodyne SIGMAR1 41 38 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H]3CCCCO3)C2)O1 ZINC000880502459 EF On-Demand Anodyne DRD4 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H]3CCCCO3)C2)O1 ZINC000880502459 EF On-Demand Anodyne SIGMAR1 42 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H]3CCCCO3)C2)O1 ZINC000880502460 EF On-Demand Anodyne DRD4 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H]3CCCCO3)C2)O1 ZINC000880502460 EF On-Demand Anodyne SIGMAR1 42 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H]3CCCCO3)C2)O1 ZINC000880502461 EF On-Demand Anodyne DRD4 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H]3CCCCO3)C2)O1 ZINC000880502461 EF On-Demand Anodyne SIGMAR1 42 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H]3CCCCO3)C2)O1 ZINC000880502462 EF On-Demand Anodyne DRD4 18 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H]3CCCCO3)C2)O1 ZINC000880502462 EF On-Demand Anodyne SIGMAR1 42 42 CCOc1ccccc1OCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880502468 FE On-Demand Anodyne HCN1 51 36 CCOc1ccccc1OCC(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880502468 FE On-Demand Anodyne HCN4 43 33 CCOc1ccccc1OCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880502469 FE On-Demand Anodyne HCN1 51 36 CCOc1ccccc1OCC(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880502469 FE On-Demand Anodyne HCN4 43 33 CCOc1ccccc1OCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880502470 FE On-Demand Anodyne HCN1 51 36 CCOc1ccccc1OCC(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880502470 FE On-Demand Anodyne HCN4 43 33 CCOc1ccccc1OCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880502471 FE On-Demand Anodyne HCN1 51 36 CCOc1ccccc1OCC(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880502471 FE On-Demand Anodyne HCN4 43 33 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCCC1 ZINC000880502548 GD On-Demand Anodyne SIGMAR1 35 47 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NC1CCCCC1 ZINC000880502549 GD On-Demand Anodyne SIGMAR1 35 47 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@H](C)C(N)=O)C2)O1 ZINC000880502550 DD On-Demand Anodyne NPFFR1 40 34 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@H](C)C(N)=O)C2)O1 ZINC000880502551 DD On-Demand Anodyne NPFFR1 40 34 C[C@@H](C(N)=O)N1CC[C@@]2(CN(Cc3ccccc3)C[C@@H](C)O2)C1 ZINC000880502552 DD On-Demand Anodyne NPFFR1 40 34 C[C@@H](C(N)=O)N1CC[C@]2(CN(Cc3ccccc3)C[C@@H](C)O2)C1 ZINC000880502553 DD On-Demand Anodyne NPFFR1 40 34 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC#N)C2)O1 ZINC000880502554 CD On-Demand Mild SIGMAR1 56 44 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC#N)C2)O1 ZINC000880502555 CD On-Demand Mild SIGMAR1 56 44 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC#N)C2)O1 ZINC000880502556 CD On-Demand Mild SIGMAR1 56 44 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC#N)C2)O1 ZINC000880502557 CD On-Demand Mild SIGMAR1 56 44 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)Nc1ccccc1 ZINC000880502572 GE On-Demand Anodyne NPFFR1 44 38 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)Nc1ccccc1 ZINC000880502573 GE On-Demand Anodyne NPFFR1 44 38 CCOC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502595 ED On-Demand Anodyne SIGMAR1 54 49 CCOC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502597 ED On-Demand Anodyne SIGMAR1 54 49 CCOC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502598 ED On-Demand Anodyne SIGMAR1 54 49 CCOC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502600 ED On-Demand Anodyne SIGMAR1 54 49 CC(=O)OC1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880502639 DF On-Demand Anodyne HTR1F 40 33 CC(=O)OC1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880502639 DF On-Demand Anodyne SMO 47 45 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(N)=O)C2)O1 ZINC000880502644 DC On-Demand Anodyne SIGMAR1 67 42 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(N)=O)C2)O1 ZINC000880502644 DC On-Demand Anodyne NPFFR1 44 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(N)=O)C2)O1 ZINC000880502645 DC On-Demand Anodyne SIGMAR1 67 42 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(N)=O)C2)O1 ZINC000880502645 DC On-Demand Anodyne NPFFR1 44 37 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(N)=O)C2)O1 ZINC000880502646 DC On-Demand Anodyne SIGMAR1 67 42 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(N)=O)C2)O1 ZINC000880502646 DC On-Demand Anodyne NPFFR1 44 37 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(N)=O)C2)O1 ZINC000880502647 DC On-Demand Anodyne SIGMAR1 67 42 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(N)=O)C2)O1 ZINC000880502647 DC On-Demand Anodyne NPFFR1 44 37 O=C1NC2(CCN(C(=O)Nc3ccc4ccccc4n3)CC2)CO1 ZINC000880502650 EE On-Demand Anodyne NPY5R 21 50 O=C1NC2(CCN(C(=O)Nc3ccc4ccccc4n3)CC2)CO1 ZINC000880502650 EE On-Demand Anodyne SMO 35 41 CC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502790 DE On-Demand Anodyne SIGMAR1 71 43 CC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502793 DE On-Demand Anodyne SIGMAR1 71 43 CC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502795 DE On-Demand Anodyne SIGMAR1 71 43 CC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502796 DE On-Demand Anodyne SIGMAR1 71 43 O=C(CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1cccs1 ZINC000880502801 GD On-Demand Anodyne SIGMAR1 18 42 O=C(CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2)NCc1cccs1 ZINC000880502802 GD On-Demand Anodyne SIGMAR1 18 42 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502805 GC On-Demand Anodyne SIGMAR1 50 46 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502805 GC On-Demand Anodyne NPFFR1 42 39 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502806 GC On-Demand Anodyne SIGMAR1 50 46 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502806 GC On-Demand Anodyne NPFFR1 42 39 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502807 GC On-Demand Anodyne SIGMAR1 50 46 COC(=O)CNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502807 GC On-Demand Anodyne NPFFR1 42 39 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502808 GC On-Demand Anodyne SIGMAR1 50 46 COC(=O)CNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502808 GC On-Demand Anodyne NPFFR1 42 39 CC(=O)NCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502817 ED On-Demand Anodyne DRD3 25 40 CC(=O)NCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502817 ED On-Demand Anodyne SIGMAR1 56 38 CC(=O)NCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502818 ED On-Demand Anodyne DRD3 25 40 CC(=O)NCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502818 ED On-Demand Anodyne SIGMAR1 56 38 CC(=O)NCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502819 ED On-Demand Anodyne DRD3 25 40 CC(=O)NCCCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502819 ED On-Demand Anodyne SIGMAR1 56 38 CC(=O)NCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502820 ED On-Demand Anodyne DRD3 25 40 CC(=O)NCCCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502820 ED On-Demand Anodyne SIGMAR1 56 38 C=CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502837 ED On-Demand Mild SIGMAR1 43 39 C=CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502837 ED On-Demand Mild NPFFR1 40 36 C=CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502838 ED On-Demand Mild SIGMAR1 43 39 C=CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880502838 ED On-Demand Mild NPFFR1 40 36 C=CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502839 ED On-Demand Mild SIGMAR1 43 39 C=CCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502839 ED On-Demand Mild NPFFR1 40 36 C=CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502840 ED On-Demand Mild SIGMAR1 43 39 C=CCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880502840 ED On-Demand Mild NPFFR1 40 36 c1ccc(CN2CCCO[C@H](CN[C@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502878 EF On-Demand Anodyne DRD4 21 44 c1ccc(CN2CCCO[C@H](CN[C@@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502880 EF On-Demand Anodyne DRD4 21 44 c1ccc(CN2CCCO[C@H](CN[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880502882 EF On-Demand Anodyne DRD4 21 44 c1ccc(CN2CCCO[C@H](CN[C@H]3CCC[C@@]34CCCO4)C2)cc1 ZINC000880502884 EF On-Demand Anodyne DRD4 21 44 COCCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503005 EE On-Demand Anodyne ADRB2 37 55 COCCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503005 EE On-Demand Anodyne ADRB1 58 55 COCCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503006 EE On-Demand Anodyne ADRB2 37 55 COCCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503006 EE On-Demand Anodyne ADRB1 58 55 COCCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503008 EE On-Demand Anodyne ADRB2 37 55 COCCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503008 EE On-Demand Anodyne ADRB1 58 55 COCCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503010 EE On-Demand Anodyne ADRB2 37 55 COCCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503010 EE On-Demand Anodyne ADRB1 58 55 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@@H]3CCOC3)C2)O1 ZINC000880503073 EE On-Demand Anodyne SIGMAR1 45 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@H]3CCOC3)C2)O1 ZINC000880503075 EE On-Demand Anodyne SIGMAR1 45 37 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(C[C@H]3CCOC3)C2)O1 ZINC000880503076 EE On-Demand Anodyne SIGMAR1 45 37 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(C[C@@H]3CCOC3)C2)O1 ZINC000880503078 EE On-Demand Anodyne SIGMAR1 45 37 CCOC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503079 EE On-Demand Anodyne SIGMAR1 52 49 CCOC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503081 EE On-Demand Anodyne SIGMAR1 52 49 CCOC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503082 EE On-Demand Anodyne SIGMAR1 52 49 CCOC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503084 EE On-Demand Anodyne SIGMAR1 52 49 Cn1ccnc1[C@H](O)C1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880503098 FF On-Demand Anodyne SMO 42 40 Cn1ccnc1[C@@H](O)C1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880503099 FF On-Demand Anodyne SMO 42 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503100 EF On-Demand Anodyne SIGMAR1 51 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503100 EF On-Demand Anodyne SLC18A3 56 43 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503101 EF On-Demand Anodyne SIGMAR1 51 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503101 EF On-Demand Anodyne SLC18A3 56 43 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503102 EF On-Demand Anodyne SIGMAR1 51 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503102 EF On-Demand Anodyne SLC18A3 56 43 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503103 EF On-Demand Anodyne SIGMAR1 51 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN([C@@H]3CCCC[C@H]3O)C2)O1 ZINC000880503103 EF On-Demand Anodyne SLC18A3 56 43 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCc3cnn(C)c3)C2)O1 ZINC000880503116 FF On-Demand Anodyne SIGMAR1 49 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCc3cnn(C)c3)C2)O1 ZINC000880503117 FF On-Demand Anodyne SIGMAR1 49 40 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCCc3cnn(C)c3)C2)O1 ZINC000880503118 FF On-Demand Anodyne SIGMAR1 49 40 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCCc3cnn(C)c3)C2)O1 ZINC000880503119 FF On-Demand Anodyne SIGMAR1 49 40 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cscn3)C2)O1 ZINC000880503122 EG On-Demand Anodyne SCN5A 42 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(Cc3cscn3)C2)O1 ZINC000880503123 EG On-Demand Anodyne SCN5A 42 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cscn3)C2)O1 ZINC000880503124 EG On-Demand Anodyne SCN5A 42 39 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(Cc3cscn3)C2)O1 ZINC000880503125 EG On-Demand Anodyne SCN5A 42 39 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA2 48 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA1 50 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA7 31 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA5B 32 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA4 26 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA5A 30 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA14 24 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA12 38 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CA9 43 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne CYNT 18 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880503362 DD On-Demand Anodyne A6YCJ1_9METZ 23 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA2 48 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA1 50 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA7 31 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA5B 32 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA4 26 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA5A 30 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA14 24 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA12 38 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CA9 43 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne CYNT 18 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880503363 DD On-Demand Anodyne A6YCJ1_9METZ 23 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA2 48 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA1 50 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA7 31 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA5B 32 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA4 26 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA5A 30 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA14 24 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA12 38 41 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CA9 43 44 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne CYNT 18 40 NS(=O)(=O)c1ccc(CCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503364 DD On-Demand Anodyne A6YCJ1_9METZ 23 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA2 48 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA1 50 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA7 31 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA5B 32 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA4 26 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA5A 30 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA14 24 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA12 38 41 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CA9 43 44 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne CYNT 18 40 NS(=O)(=O)c1ccc(CCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880503365 DD On-Demand Anodyne A6YCJ1_9METZ 23 40 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCc3ccncc3)C2)O1 ZINC000880503418 FF On-Demand Anodyne SIGMAR1 58 39 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCc3ccncc3)C2)O1 ZINC000880503419 FF On-Demand Anodyne SIGMAR1 58 39 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CCc3ccncc3)C2)O1 ZINC000880503420 FF On-Demand Anodyne SIGMAR1 58 39 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CCc3ccncc3)C2)O1 ZINC000880503421 FF On-Demand Anodyne SIGMAR1 58 39 NC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503422 DB On-Demand Anodyne SIGMAR1 37 40 NC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503422 DB On-Demand Anodyne NPFFR1 42 36 NC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503423 DB On-Demand Anodyne SIGMAR1 37 40 NC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503423 DB On-Demand Anodyne NPFFR1 42 36 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503448 GD On-Demand Anodyne DRD4 26 48 C[C@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503448 GD On-Demand Anodyne SIGMAR1 46 43 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503449 GD On-Demand Anodyne DRD4 26 48 C[C@@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503449 GD On-Demand Anodyne SIGMAR1 46 43 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503450 GD On-Demand Anodyne DRD4 26 48 C[C@@H]1CN(Cc2ccccc2)C[C@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503450 GD On-Demand Anodyne SIGMAR1 46 43 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503451 GD On-Demand Anodyne DRD4 26 48 C[C@H]1CN(Cc2ccccc2)C[C@@]2(CCN(CC(=O)NC(=O)NC3CC3)C2)O1 ZINC000880503451 GD On-Demand Anodyne SIGMAR1 46 43 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880503596 EG On-Demand Anodyne CSNK1D 45 47 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880503597 EG On-Demand Anodyne CSNK1D 45 47 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880503598 EG On-Demand Anodyne CSNK1D 45 47 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880503599 EG On-Demand Anodyne CSNK1D 45 47 Cn1c(=O)c(CN[C@H]2CCC[C@]23CCCO3)cc2ccccc21 ZINC000880503845 DF On-Demand Anodyne NPSR1 33 44 Cn1c(=O)c(CN[C@@H]2CCC[C@@]23CCCO3)cc2ccccc21 ZINC000880503847 DF On-Demand Anodyne NPSR1 33 44 CCNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503849 ED On-Demand Anodyne SIGMAR1 50 38 CCNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503849 ED On-Demand Anodyne NPFFR1 42 38 Cn1c(=O)c(CN[C@@H]2CCC[C@]23CCCO3)cc2ccccc21 ZINC000880503850 DF On-Demand Anodyne NPSR1 33 44 Cn1c(=O)c(CN[C@H]2CCC[C@@]23CCCO3)cc2ccccc21 ZINC000880503852 DF On-Demand Anodyne NPSR1 33 44 CCNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503854 ED On-Demand Anodyne SIGMAR1 50 38 CCNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503854 ED On-Demand Anodyne NPFFR1 42 38 CCNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503859 ED On-Demand Anodyne SIGMAR1 50 38 CCNC(=O)CCN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503859 ED On-Demand Anodyne NPFFR1 42 38 CCNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503867 ED On-Demand Anodyne SIGMAR1 50 38 CCNC(=O)CCN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503867 ED On-Demand Anodyne NPFFR1 42 38 COCCCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503967 GD On-Demand Anodyne ADRA1A 15 40 COCCCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503967 GD On-Demand Anodyne SIGMAR1 39 41 COCCCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503970 GD On-Demand Anodyne ADRA1A 15 40 COCCCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503970 GD On-Demand Anodyne SIGMAR1 39 41 COCCCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503971 GD On-Demand Anodyne ADRA1A 15 40 COCCCNC(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880503971 GD On-Demand Anodyne SIGMAR1 39 41 COCCCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503972 GD On-Demand Anodyne ADRA1A 15 40 COCCCNC(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880503972 GD On-Demand Anodyne SIGMAR1 39 41 C[C@H]1CCCCN1C(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503973 GD On-Demand Anodyne CPT1A 62 33 C[C@@H]1CCCCN1C(=O)CN1CC[C@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503974 GD On-Demand Anodyne CPT1A 62 33 C[C@H]1CCCCN1C(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503975 GD On-Demand Anodyne CPT1A 62 33 C[C@@H]1CCCCN1C(=O)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C(=O)CO2 ZINC000880503976 GD On-Demand Anodyne CPT1A 62 33 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880503977 GE On-Demand Anodyne PAPA1_CARPA 18 44 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](N2CCOCC2)C1(C)C ZINC000880503978 GE On-Demand Anodyne PAPA1_CARPA 18 44 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880503979 GE On-Demand Anodyne PAPA1_CARPA 18 44 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](N2CCOCC2)C1(C)C ZINC000880503980 GE On-Demand Anodyne PAPA1_CARPA 18 44 N#CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880504058 EE On-Demand Mild ADRB1 33 41 N#CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880504059 EE On-Demand Mild ADRB1 33 41 N#CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880504060 EE On-Demand Mild ADRB1 33 41 N#CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880504061 EE On-Demand Mild ADRB1 33 41 C=C(C)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880504173 DF On-Demand Mild SIGMAR1 59 41 C=C(C)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880504174 DF On-Demand Mild SIGMAR1 59 41 C=C(C)CN1CC[C@]2(C1)CN(Cc1ccccc1)C[C@@H](C)O2 ZINC000880504175 DF On-Demand Mild SIGMAR1 59 41 C=C(C)CN1CC[C@@]2(C1)CN(Cc1ccccc1)C[C@H](C)O2 ZINC000880504176 DF On-Demand Mild SIGMAR1 59 41 c1cncc(CCN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880504225 BE On-Demand Anodyne CHRNA7 15 40 c1cncc(CCN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880504226 BE On-Demand Anodyne CHRNA7 15 40 c1cncc(CCN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880504227 BE On-Demand Anodyne CHRNA7 15 40 c1cncc(CCN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880504228 BE On-Demand Anodyne CHRNA7 15 40 Cn1ccnc1[C@@](O)(CCNC(=O)Nc1ccc2ccccc2n1)C(F)(F)F ZINC000880504363 GF On-Demand Anodyne KCNJ11 40 34 Cn1ccnc1[C@](O)(CCNC(=O)Nc1ccc2ccccc2n1)C(F)(F)F ZINC000880504364 GF On-Demand Anodyne KCNJ11 40 34 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880504854 EF On-Demand Anodyne P2RY12 45 35 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccc3ccccc3n2)C1 ZINC000880504854 EF On-Demand Anodyne SMO 41 38 Cc1cccc(C(=O)NNC(=O)CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880504884 ED On-Demand Reactive KCNK3 45 35 Cc1cccc(C(=O)NNC(=O)CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880504885 ED On-Demand Reactive KCNK3 45 35 Cc1cccc(C(=O)NNC(=O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880504886 ED On-Demand Reactive KCNK3 45 35 Cc1cccc(C(=O)NNC(=O)CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880504887 ED On-Demand Reactive KCNK3 45 35 N#C[C@H](c1cccs1)N1CCN(C(=O)CN[C@H]2CCC[C@@]23CCCO3)CC1 ZINC000880505073 GE On-Demand Mild PTAFR 35 41 N#C[C@H](c1cccs1)N1CCN(C(=O)CN[C@H]2CCC[C@]23CCCO3)CC1 ZINC000880505074 GE On-Demand Mild PTAFR 35 41 N#C[C@H](c1cccs1)N1CCN(C(=O)CN[C@@H]2CCC[C@]23CCCO3)CC1 ZINC000880505075 GE On-Demand Mild PTAFR 35 41 N#C[C@H](c1cccs1)N1CCN(C(=O)CN[C@@H]2CCC[C@@]23CCCO3)CC1 ZINC000880505076 GE On-Demand Mild PTAFR 35 41 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505232 FG On-Demand Anodyne NPY5R 18 40 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505232 FG On-Demand Anodyne EPHX2 20 42 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505232 FG On-Demand Anodyne SFRP1 47 31 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505232 FG On-Demand Anodyne SMO 29 43 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505233 FG On-Demand Anodyne NPY5R 18 40 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505233 FG On-Demand Anodyne EPHX2 20 42 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505233 FG On-Demand Anodyne SFRP1 47 31 C[C@@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505233 FG On-Demand Anodyne SMO 29 43 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505234 FG On-Demand Anodyne NPY5R 18 40 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505234 FG On-Demand Anodyne EPHX2 20 42 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505234 FG On-Demand Anodyne SFRP1 47 31 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@H]1c1ccccc1 ZINC000880505234 FG On-Demand Anodyne SMO 29 43 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505235 FG On-Demand Anodyne NPY5R 18 40 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505235 FG On-Demand Anodyne EPHX2 20 42 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505235 FG On-Demand Anodyne SFRP1 47 31 C[C@H]1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C[C@@H]1c1ccccc1 ZINC000880505235 FG On-Demand Anodyne SMO 29 43 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](CF)C2)nc1 ZINC000880505282 DD On-Demand Anodyne GPR119 50 39 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@H](CF)C2)nc1 ZINC000880505283 DD On-Demand Anodyne GPR119 50 39 CN1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CCC1(C)C ZINC000880505284 ED On-Demand Anodyne NPY5R 30 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne DRD4 34 48 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne ACHE 21 42 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne SIGMAR1 35 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne CCR3 25 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne MCHR1 24 46 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505289 FE On-Demand Anodyne BIRC2 69 49 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne DRD4 34 48 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne ACHE 21 42 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne SIGMAR1 35 43 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne CCR3 25 41 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne MCHR1 24 46 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880505290 FE On-Demand Anodyne BIRC2 69 49 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne DRD4 34 48 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne ACHE 21 42 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne SIGMAR1 35 43 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne CCR3 25 41 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne MCHR1 24 46 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505291 FE On-Demand Anodyne BIRC2 69 49 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne DRD4 34 48 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne ACHE 21 42 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne SIGMAR1 35 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne CCR3 25 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne MCHR1 24 46 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880505292 FE On-Demand Anodyne BIRC2 69 49 O=C(NCc1ccc(N2CCC(O)CC2)c(F)c1)Nc1ccc2ccccc2n1 ZINC000880505344 GH On-Demand Clean NPY2R 43 36 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCCCC2)nc1 ZINC000880505492 FF On-Demand Anodyne DGAT1 38 41 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCCCC2)nc1 ZINC000880505494 FF On-Demand Anodyne DGAT1 38 41 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCCCC2)nc1 ZINC000880505496 FF On-Demand Anodyne DGAT1 38 41 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCCCC2)nc1 ZINC000880505497 FF On-Demand Anodyne DGAT1 38 41 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCc1ccc2c(c1)OCO2 ZINC000880505498 ED On-Demand Anodyne NOS2 100 41 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCc1ccc2c(c1)OCO2 ZINC000880505499 ED On-Demand Anodyne NOS2 100 41 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCc1ccc2c(c1)OCO2 ZINC000880505500 ED On-Demand Anodyne NOS2 100 41 O=C(CN[C@H]1CCC[C@]12CCCO2)NCc1ccc2c(c1)OCO2 ZINC000880505501 ED On-Demand Anodyne NOS2 100 41 O=C(CCN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505506 FF On-Demand Anodyne MTOR 48 33 O=C(CCN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505506 FF On-Demand Anodyne STAT6 41 30 O=C(CCN[C@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505507 FF On-Demand Anodyne MTOR 48 33 O=C(CCN[C@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505507 FF On-Demand Anodyne STAT6 41 30 O=C(CCN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505508 FF On-Demand Anodyne MTOR 48 33 O=C(CCN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505508 FF On-Demand Anodyne STAT6 41 30 O=C(CCN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505509 FF On-Demand Anodyne MTOR 48 33 O=C(CCN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880505509 FF On-Demand Anodyne STAT6 41 30 COc1ccc2c(CN[C@H]3CCC[C@]34CCCO4)cc(=O)oc2c1 ZINC000880505546 EF On-Demand Anodyne MAOB 26 44 COc1ccc2c(CN[C@@H]3CCC[C@@]34CCCO4)cc(=O)oc2c1 ZINC000880505548 EF On-Demand Anodyne MAOB 26 44 COc1ccc2c(CN[C@@H]3CCC[C@]34CCCO4)cc(=O)oc2c1 ZINC000880505550 EF On-Demand Anodyne MAOB 26 44 COc1ccc2c(CN[C@H]3CCC[C@@]34CCCO4)cc(=O)oc2c1 ZINC000880505552 EF On-Demand Anodyne MAOB 26 44 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880505578 FD On-Demand Anodyne NPY5R 23 40 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)nc1 ZINC000880505753 GE On-Demand Anodyne MLNR 28 44 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)nc1 ZINC000880505753 GE On-Demand Anodyne S1PR2 24 43 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)nc1 ZINC000880505753 GE On-Demand Anodyne EPHX2 31 43 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)nc1 ZINC000880505753 GE On-Demand Anodyne GPR119 76 41 Cc1cncc([C@@H]2CCCN2C(=O)Nc2ccc(S(C)(=O)=O)cn2)c1 ZINC000880505768 FF On-Demand Anodyne GCK 19 41 Cc1cncc([C@H]2CCCN2C(=O)Nc2ccc(S(C)(=O)=O)cn2)c1 ZINC000880505770 FF On-Demand Anodyne GCK 19 41 O=C(NC1CCN(C(=O)CN[C@@H]2CCC[C@@]23CCCO3)CC1)c1ccccc1 ZINC000880505772 GE On-Demand Anodyne C3AR1 40 39 O=C(NC1CCN(C(=O)CN[C@@H]2CCC[C@]23CCCO3)CC1)c1ccccc1 ZINC000880505774 GE On-Demand Anodyne C3AR1 40 39 O=C(NC1CCN(C(=O)CN[C@H]2CCC[C@@]23CCCO3)CC1)c1ccccc1 ZINC000880505776 GE On-Demand Anodyne C3AR1 40 39 O=C(NC1CCN(C(=O)CN[C@H]2CCC[C@]23CCCO3)CC1)c1ccccc1 ZINC000880505778 GE On-Demand Anodyne C3AR1 40 39 O=C(CCN[C@@H]1CCC[C@@]12CCCO2)Nc1cccnc1 ZINC000880505785 CE On-Demand Anodyne NAMPT 23 41 O=C(CCN[C@H]1CCC[C@@]12CCCO2)Nc1cccnc1 ZINC000880505787 CE On-Demand Anodyne NAMPT 23 41 O=C(CCN[C@H]1CCC[C@]12CCCO2)Nc1cccnc1 ZINC000880505789 CE On-Demand Anodyne NAMPT 23 41 O=C(CCN[C@@H]1CCC[C@]12CCCO2)Nc1cccnc1 ZINC000880505791 CE On-Demand Anodyne NAMPT 23 41 CS(=O)(=O)c1ccc(NC(=O)NCC2(CC3CC3)CC2)nc1 ZINC000880505823 DE On-Demand Anodyne SLC6A9 20 41 c1cn(CCCN[C@H]2CCC[C@]23CCCO3)cn1 ZINC000880505879 BD On-Demand Anodyne TBXAS1 15 40 c1cn(CCCN[C@H]2CCC[C@]23CCCO3)cn1 ZINC000880505879 BD On-Demand Anodyne QPCT 30 40 c1cn(CCCN[C@@H]2CCC[C@]23CCCO3)cn1 ZINC000880505880 BD On-Demand Anodyne TBXAS1 15 40 c1cn(CCCN[C@@H]2CCC[C@]23CCCO3)cn1 ZINC000880505880 BD On-Demand Anodyne QPCT 30 40 c1cn(CCCN[C@H]2CCC[C@@]23CCCO3)cn1 ZINC000880505881 BD On-Demand Anodyne TBXAS1 15 40 c1cn(CCCN[C@H]2CCC[C@@]23CCCO3)cn1 ZINC000880505881 BD On-Demand Anodyne QPCT 30 40 c1cn(CCCN[C@@H]2CCC[C@@]23CCCO3)cn1 ZINC000880505882 BD On-Demand Anodyne TBXAS1 15 40 c1cn(CCCN[C@@H]2CCC[C@@]23CCCO3)cn1 ZINC000880505882 BD On-Demand Anodyne QPCT 30 40 CCOC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880505940 EF On-Demand Anodyne P2RY12 93 38 CCOC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880505940 EF On-Demand Anodyne SSTR5 49 37 CCOC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880505940 EF On-Demand Anodyne EPHX2 48 50 CCOC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880505940 EF On-Demand Anodyne CCR8 75 44 CCOC(=O)N1CCC(NC(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880505940 EF On-Demand Anodyne SMO 44 39 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](F)(c3ccccc3)C2)nc1 ZINC000880505992 GF On-Demand Anodyne NPY5R 27 43 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](F)(c3ccccc3)C2)nc1 ZINC000880505992 GF On-Demand Anodyne EPHX2 19 43 CC(=O)C1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880506027 ED On-Demand Anodyne NPY5R 25 40 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880506035 FE On-Demand Anodyne NPY5R 28 44 O=c1cc(CN[C@H]2CCC[C@]23CCCO3)occ1O ZINC000880506098 CD On-Demand Anodyne PPO2 15 44 O=c1cc(CN[C@@H]2CCC[C@]23CCCO3)occ1O ZINC000880506099 CD On-Demand Anodyne PPO2 15 44 O=c1cc(CN[C@H]2CCC[C@@]23CCCO3)occ1O ZINC000880506100 CD On-Demand Anodyne PPO2 15 44 O=c1cc(CN[C@@H]2CCC[C@@]23CCCO3)occ1O ZINC000880506101 CD On-Demand Anodyne PPO2 15 44 CCCOc1ccc(OCC(=O)N[C@@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506215 GE On-Demand Anodyne MMP13 17 45 CCCOc1ccc(OCC(=O)N[C@@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506215 GE On-Demand Anodyne PLA2G4B 53 32 CCCOc1ccc(OCC(=O)N[C@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506216 GE On-Demand Anodyne MMP13 17 45 CCCOc1ccc(OCC(=O)N[C@H]2C[C@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506216 GE On-Demand Anodyne PLA2G4B 53 32 CCCOc1ccc(OCC(=O)N[C@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506217 GE On-Demand Anodyne MMP13 17 45 CCCOc1ccc(OCC(=O)N[C@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506217 GE On-Demand Anodyne PLA2G4B 53 32 CCCOc1ccc(OCC(=O)N[C@@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506218 GE On-Demand Anodyne MMP13 17 45 CCCOc1ccc(OCC(=O)N[C@@H]2C[C@@H](N3CCOCC3)C2(C)C)cc1 ZINC000880506218 GE On-Demand Anodyne PLA2G4B 53 32 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1[N+](=O)[O-] ZINC000880506244 EF On-Demand Bother COLA 45 35 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccccc1[N+](=O)[O-] ZINC000880506246 EF On-Demand Bother COLA 45 35 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccc(N2CCOCC2)cc1 ZINC000880506254 FF On-Demand Anodyne MTOR 56 37 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(N2CCOCC2)cc1 ZINC000880506257 FF On-Demand Anodyne MTOR 56 37 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880506286 EG On-Demand Anodyne EPHX2 26 43 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880506288 EG On-Demand Anodyne EPHX2 26 43 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880506290 EG On-Demand Anodyne EPHX2 26 43 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880506292 EG On-Demand Anodyne EPHX2 26 43 O=C1OCC[C@@H]1N[C@@H]1CCC[C@@]12CCCO2 ZINC000880506294 BC On-Demand Anodyne LUXR 44 34 O=C1OCC[C@@H]1N[C@@H]1CCC[C@@]12CCCO2 ZINC000880506294 BC On-Demand Anodyne TRAR 68 34 O=C1OCC[C@@H]1N[C@@H]1CCC[C@@]12CCCO2 ZINC000880506294 BC On-Demand Anodyne LASR 42 31 O=C1OCC[C@@H]1N[C@H]1CCC[C@@]12CCCO2 ZINC000880506298 BC On-Demand Anodyne LUXR 44 34 O=C1OCC[C@@H]1N[C@H]1CCC[C@@]12CCCO2 ZINC000880506298 BC On-Demand Anodyne TRAR 68 34 O=C1OCC[C@@H]1N[C@H]1CCC[C@@]12CCCO2 ZINC000880506298 BC On-Demand Anodyne LASR 42 31 O=C1OCC[C@@H]1N[C@H]1CCC[C@]12CCCO2 ZINC000880506300 BC On-Demand Anodyne LUXR 44 34 O=C1OCC[C@@H]1N[C@H]1CCC[C@]12CCCO2 ZINC000880506300 BC On-Demand Anodyne TRAR 68 34 O=C1OCC[C@@H]1N[C@H]1CCC[C@]12CCCO2 ZINC000880506300 BC On-Demand Anodyne LASR 42 31 O=C1OCC[C@@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880506301 BC On-Demand Anodyne LUXR 44 34 O=C1OCC[C@@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880506301 BC On-Demand Anodyne TRAR 68 34 O=C1OCC[C@@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880506301 BC On-Demand Anodyne LASR 42 31 Fc1ccccc1-n1ccc(CN[C@@H]2CCC[C@]23CCCO3)n1 ZINC000880506511 DG On-Demand Anodyne NPY5R 23 40 Fc1ccccc1-n1ccc(CN[C@@H]2CCC[C@@]23CCCO3)n1 ZINC000880506512 DG On-Demand Anodyne NPY5R 23 40 Fc1ccccc1-n1ccc(CN[C@H]2CCC[C@]23CCCO3)n1 ZINC000880506513 DG On-Demand Anodyne NPY5R 23 40 Fc1ccccc1-n1ccc(CN[C@H]2CCC[C@@]23CCCO3)n1 ZINC000880506514 DG On-Demand Anodyne NPY5R 23 40 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1nccs1 ZINC000880506572 CD On-Demand Anodyne MAP1 88 38 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1nccs1 ZINC000880506574 CD On-Demand Anodyne MAP1 88 38 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1nccs1 ZINC000880506576 CD On-Demand Anodyne MAP1 88 38 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1nccs1 ZINC000880506578 CD On-Demand Anodyne MAP1 88 38 CS(=O)(=O)c1ccc(OCCCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880506848 FF On-Demand Anodyne MMP13 16 42 CS(=O)(=O)c1ccc(OCCCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880506849 FF On-Demand Anodyne MMP13 16 42 CS(=O)(=O)c1ccc(OCCCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880506850 FF On-Demand Anodyne MMP13 16 42 CS(=O)(=O)c1ccc(OCCCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880506851 FF On-Demand Anodyne MMP13 16 42 C#CC[C@H](CCOC)NC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880506890 ED On-Demand Mild GCK 22 41 C#CC[C@@H](CCOC)NC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880506892 ED On-Demand Mild GCK 22 41 O=C(CN[C@H]1CCC[C@]12CCCO2)NCC#Cc1cccc(C(F)(F)F)c1 ZINC000880506902 GF On-Demand Mild CCR2 64 37 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCC#Cc1cccc(C(F)(F)F)c1 ZINC000880506903 GF On-Demand Mild CCR2 64 37 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCC#Cc1cccc(C(F)(F)F)c1 ZINC000880506904 GF On-Demand Mild CCR2 64 37 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCC#Cc1cccc(C(F)(F)F)c1 ZINC000880506905 GF On-Demand Mild CCR2 64 37 CN1CCN(C2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)CC1 ZINC000880506983 GC On-Demand Anodyne CHRM2 41 35 CN1CCN(C2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)CC1 ZINC000880506983 GC On-Demand Anodyne HTR1F 42 33 CN1CCN(C2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)CC1 ZINC000880506983 GC On-Demand Anodyne L3MBTL3 73 40 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)nc1 ZINC000880507010 FF On-Demand Anodyne OXTR 55 34 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)nc1 ZINC000880507010 FF On-Demand Anodyne NPY5R 43 55 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)nc1 ZINC000880507011 FF On-Demand Anodyne OXTR 55 34 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)nc1 ZINC000880507011 FF On-Demand Anodyne NPY5R 43 55 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1nc2ccccc2s1 ZINC000880507093 EF On-Demand Anodyne CSNK1D 39 47 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1nc2ccccc2s1 ZINC000880507094 EF On-Demand Anodyne CSNK1D 39 47 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1nc2ccccc2s1 ZINC000880507095 EF On-Demand Anodyne CSNK1D 39 47 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1nc2ccccc2s1 ZINC000880507096 EF On-Demand Anodyne CSNK1D 39 47 O=C(CN[C@H]1CCC[C@@]12CCCO2)NOCc1ccccc1 ZINC000880507113 DD On-Demand Anodyne SLC12A5 46 36 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NOCc1ccccc1 ZINC000880507114 DD On-Demand Anodyne SLC12A5 46 36 O=C(CN[C@H]1CCC[C@]12CCCO2)NOCc1ccccc1 ZINC000880507115 DD On-Demand Anodyne SLC12A5 46 36 O=C(CN[C@@H]1CCC[C@]12CCCO2)NOCc1ccccc1 ZINC000880507116 DD On-Demand Anodyne SLC12A5 46 36 Cc1cc(CN[C@@H]2CCC[C@]23CCCO3)c2ccccc2n1 ZINC000880507146 CH On-Demand Anodyne ADAM17 67 40 Cc1cc(CN[C@H]2CCC[C@]23CCCO3)c2ccccc2n1 ZINC000880507147 CH On-Demand Anodyne ADAM17 67 40 Cc1cc(CN[C@H]2CCC[C@@]23CCCO3)c2ccccc2n1 ZINC000880507148 CH On-Demand Anodyne ADAM17 67 40 Cc1cc(CN[C@@H]2CCC[C@@]23CCCO3)c2ccccc2n1 ZINC000880507149 CH On-Demand Anodyne ADAM17 67 40 CCCOc1cccc(CNC(=O)CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880507179 EF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CNC(=O)CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880507180 EF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CNC(=O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880507181 EF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CNC(=O)CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880507182 EF On-Demand Anodyne HRH2 26 40 O=c1cc(CN[C@@H]2CCC[C@]23CCCO3)c2ccc(O)cc2o1 ZINC000880507242 DF On-Demand Anodyne HSD17B3 33 47 O=c1cc(CN[C@H]2CCC[C@@]23CCCO3)c2ccc(O)cc2o1 ZINC000880507243 DF On-Demand Anodyne HSD17B3 33 47 O=c1cc(CN[C@@H]2CCC[C@@]23CCCO3)c2ccc(O)cc2o1 ZINC000880507244 DF On-Demand Anodyne HSD17B3 33 47 O=c1cc(CN[C@H]2CCC[C@]23CCCO3)c2ccc(O)cc2o1 ZINC000880507245 DF On-Demand Anodyne HSD17B3 33 47 O=C(Nc1ccc2ccccc2n1)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880507268 FI On-Demand Anodyne SMO 45 47 O=C(Nc1ccc2ccccc2n1)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880507269 FI On-Demand Anodyne SMO 45 47 O=C(CN[C@H]1CCC[C@@]12CCCO2)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880507274 GD On-Demand Bother SSTR1 48 46 O=C(CN[C@H]1CCC[C@]12CCCO2)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880507275 GD On-Demand Bother SSTR1 48 46 O=C(CN[C@@H]1CCC[C@]12CCCO2)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880507276 GD On-Demand Bother SSTR1 48 46 O=C(CN[C@@H]1CCC[C@@]12CCCO2)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880507277 GD On-Demand Bother SSTR1 48 46 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1cccnc1Cl ZINC000880507279 DF On-Demand Anodyne G2YM83_BOTF4 71 36 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1cccnc1Cl ZINC000880507280 DF On-Demand Anodyne G2YM83_BOTF4 71 36 COC(=O)c1cccc(NC(=O)CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880507282 EE On-Demand Anodyne HIF1A 15 45 COC(=O)c1cccc(NC(=O)CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880507283 EE On-Demand Anodyne HIF1A 15 45 COC(=O)c1cccc(NC(=O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880507284 EE On-Demand Anodyne HIF1A 15 45 COC(=O)c1cccc(NC(=O)CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880507285 EE On-Demand Anodyne HIF1A 15 45 CS(=O)(=O)c1ccc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)nc1 ZINC000880507295 FF On-Demand Anodyne RBP4 41 35 CS(=O)(=O)c1ccc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)nc1 ZINC000880507295 FF On-Demand Anodyne SMO 26 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2ccccc2n1 ZINC000880507575 GH On-Demand Clean CASR 45 38 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2ccccc2n1 ZINC000880507575 GH On-Demand Clean MTTP 40 36 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2ccccc2n1 ZINC000880507575 GH On-Demand Clean EPHB4 44 32 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2ccccc2n1 ZINC000880507575 GH On-Demand Clean STAT6 58 36 CCC1(N2CCCCC2)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880507576 GF On-Demand Anodyne NPY5R 25 41 N#Cc1c(NC(=O)CCN[C@@H]2CCC[C@]23CCCO3)sc2c1CCC2 ZINC000880507585 FG On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN[C@H]2CCC[C@]23CCCO3)sc2c1CCC2 ZINC000880507586 FG On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN[C@H]2CCC[C@@]23CCCO3)sc2c1CCC2 ZINC000880507587 FG On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN[C@@H]2CCC[C@@]23CCCO3)sc2c1CCC2 ZINC000880507588 FG On-Demand Mild VIPR1 30 48 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1nc2c(s1)CCCC2 ZINC000880507624 EF On-Demand Anodyne SLC27A1 32 42 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1nc2c(s1)CCCC2 ZINC000880507625 EF On-Demand Anodyne SLC27A1 32 42 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1nc2c(s1)CCCC2 ZINC000880507626 EF On-Demand Anodyne SLC27A1 32 42 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1nc2c(s1)CCCC2 ZINC000880507627 EF On-Demand Anodyne SLC27A1 32 42 CCOc1ccccc1NC(=O)CCN[C@H]1CCC[C@]12CCCO2 ZINC000880507709 EG On-Demand Anodyne HCN1 44 34 CCOc1ccccc1NC(=O)CCN[C@H]1CCC[C@]12CCCO2 ZINC000880507709 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)CCN[C@@H]1CCC[C@@]12CCCO2 ZINC000880507710 EG On-Demand Anodyne HCN1 44 34 CCOc1ccccc1NC(=O)CCN[C@@H]1CCC[C@@]12CCCO2 ZINC000880507710 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)CCN[C@@H]1CCC[C@]12CCCO2 ZINC000880507711 EG On-Demand Anodyne HCN1 44 34 CCOc1ccccc1NC(=O)CCN[C@@H]1CCC[C@]12CCCO2 ZINC000880507711 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)CCN[C@H]1CCC[C@@]12CCCO2 ZINC000880507712 EG On-Demand Anodyne HCN1 44 34 CCOc1ccccc1NC(=O)CCN[C@H]1CCC[C@@]12CCCO2 ZINC000880507712 EG On-Demand Anodyne HCN4 44 34 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507717 EG On-Demand Anodyne ERBB4 43 32 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507717 EG On-Demand Anodyne MCHR1 27 46 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507718 EG On-Demand Anodyne ERBB4 43 32 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507718 EG On-Demand Anodyne MCHR1 27 46 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507719 EG On-Demand Anodyne ERBB4 43 32 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507719 EG On-Demand Anodyne MCHR1 27 46 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507720 EG On-Demand Anodyne ERBB4 43 32 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880507720 EG On-Demand Anodyne MCHR1 27 46 CS(=O)(=O)c1ccc(NC(=O)NOCC2CCC2)nc1 ZINC000880507794 CD On-Demand Anodyne GCK 23 41 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)nc1 ZINC000880507834 FE On-Demand Anodyne GPR119 75 43 O=C(CCN[C@@H]1CCC[C@]12CCCO2)OCc1ccccc1 ZINC000880507847 DF On-Demand Anodyne SLC12A5 63 38 O=C(CCN[C@H]1CCC[C@@]12CCCO2)OCc1ccccc1 ZINC000880507848 DF On-Demand Anodyne SLC12A5 63 38 O=C(CCN[C@@H]1CCC[C@@]12CCCO2)OCc1ccccc1 ZINC000880507849 DF On-Demand Anodyne SLC12A5 63 38 O=C(CCN[C@H]1CCC[C@]12CCCO2)OCc1ccccc1 ZINC000880507850 DF On-Demand Anodyne SLC12A5 63 38 C#CCC1(O)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880508041 EC On-Demand Mild NPY5R 28 42 C#CCC1(O)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880508041 EC On-Demand Mild S1PR2 25 42 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880508043 GF On-Demand Anodyne CNR2 19 42 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880508044 GF On-Demand Anodyne CNR2 19 42 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880508045 GF On-Demand Anodyne CNR2 19 42 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880508046 GF On-Demand Anodyne CNR2 19 42 COc1ccc([C@@H]2CN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CCO2)cc1 ZINC000880508055 GE On-Demand Anodyne MMP13 40 38 COc1ccc([C@@H]2CN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CCO2)cc1 ZINC000880508055 GE On-Demand Anodyne MMP3 40 37 C#CC[C@@H](COC)NC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880508154 DC On-Demand Mild GCK 20 42 C#CC[C@H](COC)NC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880508155 DC On-Demand Mild GCK 20 42 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1nc2c(s1)CCC2 ZINC000880508308 DE On-Demand Anodyne SLC27A1 31 40 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1nc2c(s1)CCC2 ZINC000880508311 DE On-Demand Anodyne SLC27A1 31 40 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1nc2c(s1)CCC2 ZINC000880508314 DE On-Demand Anodyne SLC27A1 31 40 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1nc2c(s1)CCC2 ZINC000880508317 DE On-Demand Anodyne SLC27A1 31 40 C#CC1(F)CN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880508348 CC On-Demand Mild NPY5R 27 45 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)nc1 ZINC000880508543 GE On-Demand Anodyne NPY5R 28 44 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)nc1 ZINC000880508543 GE On-Demand Anodyne EPHX2 15 44 C[C@@H]1CN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CCN1c1ccncc1 ZINC000880508560 GD On-Demand Anodyne GPR119 26 44 C[C@@H]1CN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CCN1c1ccncc1 ZINC000880508560 GD On-Demand Anodyne GCKR 49 37 C[C@H]1CN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CCN1c1ccncc1 ZINC000880508562 GD On-Demand Anodyne GPR119 26 44 C[C@H]1CN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CCN1c1ccncc1 ZINC000880508562 GD On-Demand Anodyne GCKR 49 37 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1nccs1 ZINC000880508641 CE On-Demand Anodyne MAP1 92 37 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1nccs1 ZINC000880508644 CE On-Demand Anodyne MAP1 92 37 CCOC(=O)N1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880508651 EF On-Demand Anodyne P2RY12 174 43 CCOC(=O)N1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880508651 EF On-Demand Anodyne CYSLTR1 23 40 CCOC(=O)N1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880508651 EF On-Demand Anodyne FAAH 19 50 CCOC(=O)N1CCN(C(=O)Nc2ccc3ccccc3n2)CC1 ZINC000880508651 EF On-Demand Anodyne SMO 42 40 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCc1cccnc1 ZINC000880508664 CD On-Demand Anodyne NAMPT 55 42 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCc1cccnc1 ZINC000880508666 CD On-Demand Anodyne NAMPT 55 42 O=C(CN[C@H]1CCC[C@]12CCCO2)NCc1cccnc1 ZINC000880508668 CD On-Demand Anodyne NAMPT 55 42 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCc1cccnc1 ZINC000880508669 CD On-Demand Anodyne NAMPT 55 42 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880508762 FE On-Demand Anodyne PROC 55 31 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880508763 FE On-Demand Anodyne PROC 55 31 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880508764 FE On-Demand Anodyne PROC 55 31 COC(=O)c1ccc(CNC(=O)[C@H](C)N[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880508765 FE On-Demand Anodyne PROC 55 31 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne CHRM2 21 43 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne CHRM1 15 43 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne DRD2 16 46 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne DRD4 38 47 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne ACHE 35 47 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne CHRM3 25 43 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne SIGMAR1 54 49 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne SSTR5 51 38 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne CCR3 22 41 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne C3AR1 40 38 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne MCHR1 43 45 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne CACNA1G 15 46 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508799 GF On-Demand Anodyne BIRC2 46 42 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne CHRM2 21 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne CHRM1 15 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne DRD2 16 46 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne DRD4 38 47 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne ACHE 35 47 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne CHRM3 25 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne SIGMAR1 54 49 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne SSTR5 51 38 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne CCR3 22 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne C3AR1 40 38 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne MCHR1 43 45 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne CACNA1G 15 46 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880508802 GF On-Demand Anodyne BIRC2 46 42 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](CF)C2)nc1 ZINC000880508813 DD On-Demand Anodyne GCK 22 41 COc1cccc(OC)c1OC[C@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880508820 FE On-Demand Anodyne ADRB2 21 43 COc1cccc(OC)c1OC[C@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880508820 FE On-Demand Anodyne ADRB1 24 43 COc1cccc(OC)c1OC[C@H](O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880508822 FE On-Demand Anodyne ADRB2 21 43 COc1cccc(OC)c1OC[C@H](O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880508822 FE On-Demand Anodyne ADRB1 24 43 COc1cccc(OC)c1OC[C@H](O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880508824 FE On-Demand Anodyne ADRB2 21 43 COc1cccc(OC)c1OC[C@H](O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880508824 FE On-Demand Anodyne ADRB1 24 43 COc1cccc(OC)c1OC[C@H](O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880508826 FE On-Demand Anodyne ADRB2 21 43 COc1cccc(OC)c1OC[C@H](O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880508826 FE On-Demand Anodyne ADRB1 24 43 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1cccnc1Cl ZINC000880508828 DE On-Demand Anodyne G2YM83_BOTF4 70 35 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1cccnc1Cl ZINC000880508829 DE On-Demand Anodyne G2YM83_BOTF4 70 35 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1cccnc1Cl ZINC000880508831 DE On-Demand Anodyne G2YM83_BOTF4 70 35 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1cccnc1Cl ZINC000880508833 DE On-Demand Anodyne G2YM83_BOTF4 70 35 COc1ccc(NC(=O)[C@H](C)N[C@@H]2CCC[C@@]23CCCO3)cc1OC ZINC000880508840 EF On-Demand Anodyne ENPP1 65 32 COc1ccc(NC(=O)[C@H](C)N[C@@H]2CCC[C@]23CCCO3)cc1OC ZINC000880508842 EF On-Demand Anodyne ENPP1 65 32 COc1ccc(NC(=O)[C@H](C)N[C@H]2CCC[C@]23CCCO3)cc1OC ZINC000880508844 EF On-Demand Anodyne ENPP1 65 32 COc1ccc(NC(=O)[C@H](C)N[C@H]2CCC[C@@]23CCCO3)cc1OC ZINC000880508847 EF On-Demand Anodyne ENPP1 65 32 CS(=O)(=O)c1ccc(NC(=O)NCCC2CCC2)nc1 ZINC000880508886 CD On-Demand Anodyne GCK 23 41 CS(=O)(=O)c1ccc(NC(=O)NCCC2CCC2)nc1 ZINC000880508886 CD On-Demand Anodyne PRMT3 17 40 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508893 EF On-Demand Anodyne ADRB2 16 68 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508893 EF On-Demand Anodyne ADRB1 24 68 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508895 EF On-Demand Anodyne ADRB2 16 68 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508895 EF On-Demand Anodyne ADRB1 24 68 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508896 EF On-Demand Anodyne ADRB2 16 68 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508896 EF On-Demand Anodyne ADRB1 24 68 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508897 EF On-Demand Anodyne ADRB2 16 68 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880508897 EF On-Demand Anodyne ADRB1 24 68 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508941 GD On-Demand Anodyne HCN1 40 31 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508941 GD On-Demand Anodyne HCN4 40 31 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508942 GD On-Demand Anodyne HCN1 40 31 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508942 GD On-Demand Anodyne HCN4 40 31 O=C(CN[C@H]1CCC[C@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508945 GD On-Demand Anodyne HCN1 40 31 O=C(CN[C@H]1CCC[C@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508945 GD On-Demand Anodyne HCN4 40 31 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508947 GD On-Demand Anodyne HCN1 40 31 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880508947 GD On-Demand Anodyne HCN4 40 31 CS(=O)(=O)c1ccc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)nc1 ZINC000880508980 GE On-Demand Anodyne SLC6A9 44 51 CS(=O)(=O)c1ccc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)nc1 ZINC000880508980 GE On-Demand Anodyne FAAH 20 40 CS(=O)(=O)c1ccc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)nc1 ZINC000880508980 GE On-Demand Anodyne NPY5R 23 40 CS(=O)(=O)c1ccc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)nc1 ZINC000880508980 GE On-Demand Anodyne S1PR2 21 42 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)nc1 ZINC000880509071 GE On-Demand Anodyne NPY5R 26 43 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)nc1 ZINC000880509071 GE On-Demand Anodyne EPHX2 18 50 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@]3(C2)CC3(F)F)nc1 ZINC000880509108 EE On-Demand Anodyne NPY5R 19 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccc2c(c1)OCCO2 ZINC000880509222 FE On-Demand Anodyne NOS2 60 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1ccc2c(c1)OCCO2 ZINC000880509224 FE On-Demand Anodyne NOS2 60 40 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509272 FE On-Demand Anodyne MTOR 57 34 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509272 FE On-Demand Anodyne STAT6 51 31 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509273 FE On-Demand Anodyne MTOR 57 34 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509273 FE On-Demand Anodyne STAT6 51 31 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509274 FE On-Demand Anodyne MTOR 57 34 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509274 FE On-Demand Anodyne STAT6 51 31 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509275 FE On-Demand Anodyne MTOR 57 34 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880509275 FE On-Demand Anodyne STAT6 51 31 CCOc1ccccc1OCCN[C@@H]1CCC[C@]12CCCO2 ZINC000880509354 DG On-Demand Anodyne HCN1 41 32 CCOc1ccccc1OCCN[C@@H]1CCC[C@]12CCCO2 ZINC000880509354 DG On-Demand Anodyne HCN4 42 32 CCOc1ccccc1OCCN[C@@H]1CCC[C@@]12CCCO2 ZINC000880509355 DG On-Demand Anodyne HCN1 41 32 CCOc1ccccc1OCCN[C@@H]1CCC[C@@]12CCCO2 ZINC000880509355 DG On-Demand Anodyne HCN4 42 32 CCOc1ccccc1OCCN[C@H]1CCC[C@]12CCCO2 ZINC000880509356 DG On-Demand Anodyne HCN1 41 32 CCOc1ccccc1OCCN[C@H]1CCC[C@]12CCCO2 ZINC000880509356 DG On-Demand Anodyne HCN4 42 32 CCOc1ccccc1OCCN[C@H]1CCC[C@@]12CCCO2 ZINC000880509357 DG On-Demand Anodyne HCN1 41 32 CCOc1ccccc1OCCN[C@H]1CCC[C@@]12CCCO2 ZINC000880509357 DG On-Demand Anodyne HCN4 42 32 CC(=O)c1cccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880509630 EE On-Demand Anodyne ADRB2 25 43 CC(=O)c1cccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880509630 EE On-Demand Anodyne ADRB3 19 40 CC(=O)c1cccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880509631 EE On-Demand Anodyne ADRB2 25 43 CC(=O)c1cccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880509631 EE On-Demand Anodyne ADRB3 19 40 CC(=O)c1cccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880509632 EE On-Demand Anodyne ADRB2 25 43 CC(=O)c1cccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880509632 EE On-Demand Anodyne ADRB3 19 40 CC(=O)c1cccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880509633 EE On-Demand Anodyne ADRB2 25 43 CC(=O)c1cccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880509633 EE On-Demand Anodyne ADRB3 19 40 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880509708 FF On-Demand Anodyne HRH3 18 42 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880509711 FF On-Demand Anodyne HRH3 18 42 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880509713 FF On-Demand Anodyne HRH3 18 42 O=C(CN[C@H]1CCC[C@]12CCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880509715 FF On-Demand Anodyne HRH3 18 42 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](CO)CC2)nc1 ZINC000880509834 ED On-Demand Anodyne GCK 19 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H](C)c1ccccc1 ZINC000880509949 DF On-Demand Anodyne BIRC8 44 33 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H](C)c1ccccc1 ZINC000880509952 DF On-Demand Anodyne BIRC8 44 33 CCOc1ccccc1NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880509987 DF On-Demand Anodyne HCN1 44 35 CCOc1ccccc1NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880509987 DF On-Demand Anodyne HCN4 45 35 CCOc1ccccc1NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880509988 DF On-Demand Anodyne HCN1 44 35 CCOc1ccccc1NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880509988 DF On-Demand Anodyne HCN4 45 35 CCOc1ccccc1NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880509989 DF On-Demand Anodyne HCN1 44 35 CCOc1ccccc1NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880509989 DF On-Demand Anodyne HCN4 45 35 CCOc1ccccc1NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880509990 DF On-Demand Anodyne HCN1 44 35 CCOc1ccccc1NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880509990 DF On-Demand Anodyne HCN4 45 35 O=C(CN[C@H]1CCC[C@@]12CCCO2)OCc1ccccc1 ZINC000880510086 CE On-Demand Anodyne SLC12A5 68 39 O=C(CN[C@@H]1CCC[C@@]12CCCO2)OCc1ccccc1 ZINC000880510087 CE On-Demand Anodyne SLC12A5 68 39 O=C(CN[C@H]1CCC[C@]12CCCO2)OCc1ccccc1 ZINC000880510088 CE On-Demand Anodyne SLC12A5 68 39 O=C(CN[C@@H]1CCC[C@]12CCCO2)OCc1ccccc1 ZINC000880510089 CE On-Demand Anodyne SLC12A5 68 39 O=C(c1ccc(CN[C@H]2CCC[C@@]23CCCO3)cc1)N1CCCC1 ZINC000880510178 EG On-Demand Anodyne L3MBTL3 74 40 O=C(c1ccc(CN[C@H]2CCC[C@]23CCCO3)cc1)N1CCCC1 ZINC000880510179 EG On-Demand Anodyne L3MBTL3 74 40 O=C(c1ccc(CN[C@@H]2CCC[C@]23CCCO3)cc1)N1CCCC1 ZINC000880510180 EG On-Demand Anodyne L3MBTL3 74 40 O=C(c1ccc(CN[C@@H]2CCC[C@@]23CCCO3)cc1)N1CCCC1 ZINC000880510181 EG On-Demand Anodyne L3MBTL3 74 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne MME 60 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne TIMP3 81 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne CAPN1 45 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne ACE2 53 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne PSMB8 50 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510202 ED On-Demand Anodyne BRCA1 50 30 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne MME 60 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne TIMP3 81 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne CAPN1 45 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne ACE2 53 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne PSMB8 50 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510203 ED On-Demand Anodyne BRCA1 50 30 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne MME 60 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne TIMP3 81 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne CAPN1 45 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne ACE2 53 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne PSMB8 50 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510204 ED On-Demand Anodyne BRCA1 50 30 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne MME 60 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne TIMP3 81 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne CAPN1 45 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne ACE2 53 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne PSMB8 50 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510205 ED On-Demand Anodyne BRCA1 50 30 O=C(NCc1cc(O)nc(S)n1)c1cccc(N2CCCC2)c1 ZINC000880510208 EE On-Demand Anodyne DRD4 43 33 N#Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510211 DD On-Demand Mild ADRB1 30 40 N#Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510212 DD On-Demand Mild ADRB1 30 40 N#Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880510213 DD On-Demand Mild ADRB1 30 40 N#Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880510214 DD On-Demand Mild ADRB1 30 40 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)c1cccc(Cl)c1 ZINC000880510307 CG On-Demand Anodyne ADRB3 39 46 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)c1cccc(Cl)c1 ZINC000880510307 CG On-Demand Anodyne CYP3A4 46 37 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880510308 CG On-Demand Anodyne ADRB3 39 46 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880510308 CG On-Demand Anodyne CYP3A4 46 37 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)c1cccc(Cl)c1 ZINC000880510309 CG On-Demand Anodyne ADRB3 39 46 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)c1cccc(Cl)c1 ZINC000880510309 CG On-Demand Anodyne CYP3A4 46 37 O[C@H](CN[C@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880510310 CG On-Demand Anodyne ADRB3 39 46 O[C@H](CN[C@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880510310 CG On-Demand Anodyne CYP3A4 46 37 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1cc(O)nc(S)n1 ZINC000880510355 ED On-Demand Anodyne PPARD 39 40 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1cc(O)nc(S)n1 ZINC000880510355 ED On-Demand Anodyne MTNR1A 32 40 Cc1c(NC(=O)[C@H](C)N[C@H]2CCC[C@@]23CCCO3)c(=O)n(-c2ccccc2)n1C ZINC000880510365 GF On-Demand Anodyne FPR2 39 41 Cc1c(NC(=O)[C@H](C)N[C@@H]2CCC[C@@]23CCCO3)c(=O)n(-c2ccccc2)n1C ZINC000880510366 GF On-Demand Anodyne FPR2 39 41 Cc1c(NC(=O)[C@H](C)N[C@@H]2CCC[C@]23CCCO3)c(=O)n(-c2ccccc2)n1C ZINC000880510367 GF On-Demand Anodyne FPR2 39 41 Cc1c(NC(=O)[C@H](C)N[C@H]2CCC[C@]23CCCO3)c(=O)n(-c2ccccc2)n1C ZINC000880510368 GF On-Demand Anodyne FPR2 39 41 O=C(NCc1cc(O)nc(S)n1)c1cccn(C2CC2)c1=O ZINC000880510381 DC On-Demand Anodyne POLR1A 65 34 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880510426 EG On-Demand Anodyne CCR2 60 37 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880510427 EG On-Demand Anodyne CCR2 60 37 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880510428 EG On-Demand Anodyne CCR2 60 37 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880510429 EG On-Demand Anodyne CCR2 60 37 COC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880510516 ED On-Demand Anodyne ADRB2 33 43 COC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880510516 ED On-Demand Anodyne ADRB1 48 40 COC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510517 ED On-Demand Anodyne ADRB2 33 43 COC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510517 ED On-Demand Anodyne ADRB1 48 40 COC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880510518 ED On-Demand Anodyne ADRB2 33 43 COC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880510518 ED On-Demand Anodyne ADRB1 48 40 COC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510519 ED On-Demand Anodyne ADRB2 33 43 COC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880510519 ED On-Demand Anodyne ADRB1 48 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880510574 DE On-Demand Anodyne ANPEP 15 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880510574 DE On-Demand Anodyne AMP1_PLAFQ 22 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880510576 DE On-Demand Anodyne ANPEP 15 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880510576 DE On-Demand Anodyne AMP1_PLAFQ 22 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510581 EF On-Demand Anodyne XIAP 30 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510581 EF On-Demand Anodyne BIRC3 59 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510581 EF On-Demand Anodyne BIRC2 30 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510582 EF On-Demand Anodyne XIAP 30 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510582 EF On-Demand Anodyne BIRC3 59 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510582 EF On-Demand Anodyne BIRC2 30 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510583 EF On-Demand Anodyne XIAP 30 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510583 EF On-Demand Anodyne BIRC3 59 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880510583 EF On-Demand Anodyne BIRC2 30 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510584 EF On-Demand Anodyne XIAP 30 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510584 EF On-Demand Anodyne BIRC3 59 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880510584 EF On-Demand Anodyne BIRC2 30 40 O=C(CCCc1ccc2c(c1)OCCCO2)NCc1cc(O)nc(S)n1 ZINC000880510694 GE On-Demand Anodyne NOS2 72 33 COC(=O)c1sccc1NC(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510705 EE On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510706 EE On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510707 EE On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510708 EE On-Demand Anodyne FAS 36 44 C[C@H](NC(=O)CN[C@@H]1CCC[C@@]12CCCO2)c1ccc(Cl)cc1 ZINC000880510723 EG On-Demand Anodyne PRCP 15 41 C[C@H](NC(=O)CN[C@H]1CCC[C@]12CCCO2)c1ccc(Cl)cc1 ZINC000880510724 EG On-Demand Anodyne PRCP 15 41 C[C@H](NC(=O)CN[C@H]1CCC[C@@]12CCCO2)c1ccc(Cl)cc1 ZINC000880510725 EG On-Demand Anodyne PRCP 15 41 C[C@H](NC(=O)CN[C@@H]1CCC[C@]12CCCO2)c1ccc(Cl)cc1 ZINC000880510726 EG On-Demand Anodyne PRCP 15 41 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCC1(c2ccccc2)CCOCC1 ZINC000880510774 FF On-Demand Anodyne KCNA3 43 35 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCC1(c2ccccc2)CCOCC1 ZINC000880510775 FF On-Demand Anodyne KCNA3 43 35 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCC1(c2ccccc2)CCOCC1 ZINC000880510776 FF On-Demand Anodyne KCNA3 43 35 O=C(CN[C@H]1CCC[C@]12CCCO2)NCC1(c2ccccc2)CCOCC1 ZINC000880510777 FF On-Demand Anodyne KCNA3 43 35 C[C@@H]1CCCCN1C(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880510814 CE On-Demand Anodyne DPP7 17 40 C[C@@H]1CCCCN1C(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880510815 CE On-Demand Anodyne DPP7 17 40 C[C@@H]1CCCCN1C(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880510816 CE On-Demand Anodyne DPP7 17 40 C[C@@H]1CCCCN1C(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880510817 CE On-Demand Anodyne DPP7 17 40 O=C(NCc1cc(O)nc(S)n1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880510832 FF On-Demand Anodyne C3AR1 42 42 O=C(NCc1cc(O)nc(S)n1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880510833 FF On-Demand Anodyne C3AR1 42 42 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510906 DE On-Demand Anodyne ADRB2 26 41 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510906 DE On-Demand Anodyne ADRB1 35 40 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510906 DE On-Demand Anodyne ADRB3 19 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510907 DE On-Demand Anodyne ADRB2 26 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510907 DE On-Demand Anodyne ADRB1 35 40 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccc(F)cc1 ZINC000880510907 DE On-Demand Anodyne ADRB3 19 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510908 DE On-Demand Anodyne ADRB2 26 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510908 DE On-Demand Anodyne ADRB1 35 40 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510908 DE On-Demand Anodyne ADRB3 19 41 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510909 DE On-Demand Anodyne ADRB2 26 41 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510909 DE On-Demand Anodyne ADRB1 35 40 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880510909 DE On-Demand Anodyne ADRB3 19 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)C[C@H]1C1CC1 ZINC000880510915 GE On-Demand Anodyne SIGMAR1 16 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)C[C@H]1C1CC1 ZINC000880510915 GE On-Demand Anodyne PDE8B 40 31 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne SSTR2 51 37 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne EDNRB 18 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne TACR1 21 44 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne CCKAR 34 41 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne BRS3 27 42 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne NMBR 86 36 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne GRPR 95 36 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne ECE1 46 36 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne CCKBR 38 40 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne MMP9 15 44 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510961 FF On-Demand Anodyne PSMB8 24 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne SSTR2 51 37 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne EDNRB 18 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne TACR1 21 44 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne CCKAR 34 41 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne BRS3 27 42 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne NMBR 86 36 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne GRPR 95 36 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne ECE1 46 36 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne CCKBR 38 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne MMP9 15 44 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880510962 FF On-Demand Anodyne PSMB8 24 40 CCC[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880511107 GF On-Demand Anodyne PDE8B 42 37 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@]12CCCO2 ZINC000880511113 DH On-Demand Anodyne PPARG 51 42 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@]12CCCO2 ZINC000880511113 DH On-Demand Anodyne PPARA 54 42 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@]12CCCO2 ZINC000880511113 DH On-Demand Anodyne PDE8B 61 36 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880511114 DH On-Demand Anodyne PPARG 51 42 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880511114 DH On-Demand Anodyne PPARA 54 42 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880511114 DH On-Demand Anodyne PDE8B 61 36 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@]12CCCO2 ZINC000880511115 DH On-Demand Anodyne PPARG 51 42 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@]12CCCO2 ZINC000880511115 DH On-Demand Anodyne PPARA 54 42 Cc1oc(-c2ccccc2)nc1CN[C@@H]1CCC[C@]12CCCO2 ZINC000880511115 DH On-Demand Anodyne PDE8B 61 36 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@@]12CCCO2 ZINC000880511116 DH On-Demand Anodyne PPARG 51 42 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@@]12CCCO2 ZINC000880511116 DH On-Demand Anodyne PPARA 54 42 Cc1oc(-c2ccccc2)nc1CN[C@H]1CCC[C@@]12CCCO2 ZINC000880511116 DH On-Demand Anodyne PDE8B 61 36 O=C(CN[C@H]1CCC[C@]12CCCO2)NCCCc1ccccc1 ZINC000880511129 DE On-Demand Anodyne CRTM 34 41 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCCCc1ccccc1 ZINC000880511130 DE On-Demand Anodyne CRTM 34 41 Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511138 DE On-Demand Anodyne ADRB2 29 50 Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511138 DE On-Demand Anodyne ADRB1 35 40 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511139 DE On-Demand Anodyne ADRB2 29 50 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511139 DE On-Demand Anodyne ADRB1 35 40 Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511140 DE On-Demand Anodyne ADRB2 29 50 Cc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511140 DE On-Demand Anodyne ADRB1 35 40 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511141 DE On-Demand Anodyne ADRB2 29 50 Cc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511141 DE On-Demand Anodyne ADRB1 35 40 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCCCc1ccccc1 ZINC000880511211 DE On-Demand Anodyne CRTM 34 41 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCCCc1ccccc1 ZINC000880511212 DE On-Demand Anodyne CRTM 34 41 CCCCCCCC[C@@H](C)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511277 EG On-Demand Mild NOD1 62 34 CCCCCCCC[C@H](C)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511278 EG On-Demand Mild NOD1 62 34 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880511365 DE On-Demand Anodyne ADRB2 24 43 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880511365 DE On-Demand Anodyne ADRB1 24 41 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1F ZINC000880511366 DE On-Demand Anodyne ADRB2 24 43 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1F ZINC000880511366 DE On-Demand Anodyne ADRB1 24 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1F ZINC000880511367 DE On-Demand Anodyne ADRB2 24 43 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1F ZINC000880511367 DE On-Demand Anodyne ADRB1 24 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880511368 DE On-Demand Anodyne ADRB2 24 43 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880511368 DE On-Demand Anodyne ADRB1 24 41 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880511373 GE On-Demand Anodyne L3MBTL3 54 36 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880511374 GE On-Demand Anodyne L3MBTL3 54 36 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880511375 GE On-Demand Anodyne L3MBTL3 54 36 O=C(CN[C@H]1CCC[C@]12CCCO2)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880511376 GE On-Demand Anodyne L3MBTL3 54 36 O=C(CN[C@H]1CCC[C@@]12CCCO2)NCC1(c2ccccc2)CC1 ZINC000880511418 EF On-Demand Anodyne KCNA3 45 37 O=C(CN[C@H]1CCC[C@]12CCCO2)NCC1(c2ccccc2)CC1 ZINC000880511420 EF On-Demand Anodyne KCNA3 45 37 O=C(CN[C@@H]1CCC[C@]12CCCO2)NCC1(c2ccccc2)CC1 ZINC000880511422 EF On-Demand Anodyne KCNA3 45 37 O=C(CN[C@@H]1CCC[C@@]12CCCO2)NCC1(c2ccccc2)CC1 ZINC000880511424 EF On-Demand Anodyne KCNA3 45 37 O=[N+]([O-])c1cccc(CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880511464 CF On-Demand Bother CACNA1D 67 34 O=[N+]([O-])c1cccc(CN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880511466 CF On-Demand Bother CACNA1D 67 34 c1csc(-c2noc(CN[C@@H]3CCC[C@]34CCCO4)n2)c1 ZINC000880511479 DF On-Demand Anodyne ETHR 24 40 c1csc(-c2noc(CN[C@@H]3CCC[C@@]34CCCO4)n2)c1 ZINC000880511480 DF On-Demand Anodyne ETHR 24 40 c1csc(-c2noc(CN[C@H]3CCC[C@@]34CCCO4)n2)c1 ZINC000880511481 DF On-Demand Anodyne ETHR 24 40 c1csc(-c2noc(CN[C@H]3CCC[C@]34CCCO4)n2)c1 ZINC000880511482 DF On-Demand Anodyne ETHR 24 40 CCCc1ccc(C(=O)NCc2cc(O)nc(S)n2)s1 ZINC000880511487 DE On-Demand Anodyne FOLR1 49 36 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880511509 EG On-Demand Anodyne EPHX2 28 40 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880511511 EG On-Demand Anodyne EPHX2 28 40 C[C@@H](CCc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511516 EE On-Demand Anodyne PSMB5 15 41 C[C@@H](CCc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511516 EE On-Demand Anodyne LEF 40 35 C[C@H](CCc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511517 EE On-Demand Anodyne PSMB5 15 41 C[C@H](CCc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880511517 EE On-Demand Anodyne LEF 40 35 C[C@@H]1CN(Cc2ccccc2)C[C@H](C(=O)NCc2cc(O)nc(S)n2)O1 ZINC000880511532 FD On-Demand Anodyne PDE8B 43 34 O=[N+]([O-])c1cccc(CN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880511539 CF On-Demand Bother CACNA1D 67 34 O=[N+]([O-])c1cccc(CN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880511540 CF On-Demand Bother CACNA1D 67 34 N#Cc1cccc(OCCN[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880511549 CF On-Demand Mild CHRNA10 16 43 N#Cc1cccc(OCCN[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880511550 CF On-Demand Mild CHRNA10 16 43 N#Cc1cccc(OCCN[C@H]2CCC[C@]23CCCO3)c1 ZINC000880511551 CF On-Demand Mild CHRNA10 16 43 N#Cc1cccc(OCCN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880511552 CF On-Demand Mild CHRNA10 16 43 CC[C@H](N[C@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccc(OC)cc1 ZINC000880511606 EG On-Demand Anodyne TIMP3 70 43 CC[C@H](N[C@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(OC)cc1 ZINC000880511607 EG On-Demand Anodyne TIMP3 70 43 CC[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(OC)cc1 ZINC000880511608 EG On-Demand Anodyne TIMP3 70 43 CC[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccc(OC)cc1 ZINC000880511609 EG On-Demand Anodyne TIMP3 70 43 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1C(F)(F)F ZINC000880511614 FH On-Demand Anodyne RBP4 51 34 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccccc1C(F)(F)F ZINC000880511616 FH On-Demand Anodyne RBP4 51 34 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC(F)F ZINC000880511673 FD On-Demand Anodyne DRTS_TRYCR 44 30 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880511702 FD On-Demand Anodyne EPHX2 23 45 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880511702 FD On-Demand Anodyne L3MBTL3 52 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880511703 FD On-Demand Anodyne EPHX2 23 45 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880511703 FD On-Demand Anodyne L3MBTL3 52 34 CCOc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511723 EF On-Demand Anodyne ADRB2 28 40 CCOc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511723 EF On-Demand Anodyne ADRB1 35 40 CCOc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511724 EF On-Demand Anodyne ADRB2 28 40 CCOc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511724 EF On-Demand Anodyne ADRB1 35 40 CCOc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511725 EF On-Demand Anodyne ADRB2 28 40 CCOc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511725 EF On-Demand Anodyne ADRB1 35 40 CCOc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511726 EF On-Demand Anodyne ADRB2 28 40 CCOc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511726 EF On-Demand Anodyne ADRB1 35 40 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511770 EG On-Demand Anodyne ADRB2 29 52 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511770 EG On-Demand Anodyne ADRB1 25 52 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511770 EG On-Demand Anodyne ADRB3 15 52 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511771 EG On-Demand Anodyne ADRB2 29 52 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511771 EG On-Demand Anodyne ADRB1 25 52 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1cccc2ccccc12 ZINC000880511771 EG On-Demand Anodyne ADRB3 15 52 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511772 EG On-Demand Anodyne ADRB2 29 52 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511772 EG On-Demand Anodyne ADRB1 25 52 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511772 EG On-Demand Anodyne ADRB3 15 52 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511773 EG On-Demand Anodyne ADRB2 29 52 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511773 EG On-Demand Anodyne ADRB1 25 52 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880511773 EG On-Demand Anodyne ADRB3 15 52 COc1ccc(N2CCN(C(=O)CN[C@@H]3CCC[C@]34CCCO4)CC2)cc1 ZINC000880511815 FE On-Demand Clean MMP13 21 42 COc1ccc(N2CCN(C(=O)CN[C@@H]3CCC[C@]34CCCO4)CC2)cc1 ZINC000880511815 FE On-Demand Clean NPBWR1 44 31 COc1ccc(N2CCN(C(=O)CN[C@H]3CCC[C@]34CCCO4)CC2)cc1 ZINC000880511817 FE On-Demand Clean MMP13 21 42 COc1ccc(N2CCN(C(=O)CN[C@H]3CCC[C@]34CCCO4)CC2)cc1 ZINC000880511817 FE On-Demand Clean NPBWR1 44 31 COc1ccc(N2CCN(C(=O)CN[C@H]3CCC[C@@]34CCCO4)CC2)cc1 ZINC000880511819 FE On-Demand Clean MMP13 21 42 COc1ccc(N2CCN(C(=O)CN[C@H]3CCC[C@@]34CCCO4)CC2)cc1 ZINC000880511819 FE On-Demand Clean NPBWR1 44 31 COc1ccc(N2CCN(C(=O)CN[C@@H]3CCC[C@@]34CCCO4)CC2)cc1 ZINC000880511822 FE On-Demand Clean MMP13 21 42 COc1ccc(N2CCN(C(=O)CN[C@@H]3CCC[C@@]34CCCO4)CC2)cc1 ZINC000880511822 FE On-Demand Clean NPBWR1 44 31 O=C(CN[C@H]1CCC[C@]12CCCO2)N1CCc2ccccc2C1 ZINC000880511870 DE On-Demand Anodyne DPP8 21 46 O=C(CN[C@@H]1CCC[C@@]12CCCO2)N1CCc2ccccc2C1 ZINC000880511871 DE On-Demand Anodyne DPP8 21 46 O=C(CN[C@@H]1CCC[C@]12CCCO2)N1CCc2ccccc2C1 ZINC000880511872 DE On-Demand Anodyne DPP8 21 46 O=C(CN[C@H]1CCC[C@@]12CCCO2)N1CCc2ccccc2C1 ZINC000880511873 DE On-Demand Anodyne DPP8 21 46 CC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511893 EE On-Demand Anodyne ADRB2 28 42 CC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511893 EE On-Demand Anodyne ADRB1 40 41 CC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511894 EE On-Demand Anodyne ADRB2 28 42 CC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880511894 EE On-Demand Anodyne ADRB1 40 41 CC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511895 EE On-Demand Anodyne ADRB2 28 42 CC(=O)c1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880511895 EE On-Demand Anodyne ADRB1 40 41 CC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511896 EE On-Demand Anodyne ADRB2 28 42 CC(=O)c1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880511896 EE On-Demand Anodyne ADRB1 40 41 COc1cccc(C(=O)NCc2cc(O)nc(S)n2)c1OC(C)C ZINC000880511907 EE On-Demand Anodyne KCNK3 58 39 COc1cccc(C(=O)NCc2cc(O)nc(S)n2)c1OC(C)C ZINC000880511907 EE On-Demand Anodyne KCNK9 43 39 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N1c2ccccc2C[C@@H]1C ZINC000880511970 EG On-Demand Anodyne TPP2 53 34 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)N1c2ccccc2C[C@H]1C ZINC000880511971 EG On-Demand Anodyne TPP2 53 34 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N1c2ccccc2C[C@H]1C ZINC000880511972 EG On-Demand Anodyne TPP2 53 34 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N1c2ccccc2C[C@@H]1C ZINC000880511973 EG On-Demand Anodyne TPP2 53 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@H]1CCC[C@]12CCCO2 ZINC000880511978 EG On-Demand Anodyne HCN1 46 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@H]1CCC[C@]12CCCO2 ZINC000880511978 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@@H]1CCC[C@@]12CCCO2 ZINC000880511979 EG On-Demand Anodyne HCN1 46 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@@H]1CCC[C@@]12CCCO2 ZINC000880511979 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@H]1CCC[C@@]12CCCO2 ZINC000880511980 EG On-Demand Anodyne HCN1 46 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@H]1CCC[C@@]12CCCO2 ZINC000880511980 EG On-Demand Anodyne HCN4 44 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@@H]1CCC[C@]12CCCO2 ZINC000880511981 EG On-Demand Anodyne HCN1 46 34 CCOc1ccccc1NC(=O)[C@H](C)N[C@@H]1CCC[C@]12CCCO2 ZINC000880511981 EG On-Demand Anodyne HCN4 44 34 NS(=O)(=O)c1ccc(OCCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512020 ED On-Demand Anodyne CA7 22 41 NS(=O)(=O)c1ccc(OCCN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512020 ED On-Demand Anodyne CA12 15 42 NS(=O)(=O)c1ccc(OCCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880512022 ED On-Demand Anodyne CA7 22 41 NS(=O)(=O)c1ccc(OCCN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880512022 ED On-Demand Anodyne CA12 15 42 NS(=O)(=O)c1ccc(OCCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512024 ED On-Demand Anodyne CA7 22 41 NS(=O)(=O)c1ccc(OCCN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512024 ED On-Demand Anodyne CA12 15 42 NS(=O)(=O)c1ccc(OCCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512026 ED On-Demand Anodyne CA7 22 41 NS(=O)(=O)c1ccc(OCCN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512026 ED On-Demand Anodyne CA12 15 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCC[C@H]1Cc1ccccc1 ZINC000880512054 EF On-Demand Anodyne LNPEP 45 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCC[C@@H]1Cc1ccccc1 ZINC000880512056 EF On-Demand Anodyne LNPEP 45 35 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCC[C@@H]1Cc1ccccc1 ZINC000880512058 EF On-Demand Anodyne LNPEP 45 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCC[C@H]1Cc1ccccc1 ZINC000880512059 EF On-Demand Anodyne LNPEP 45 35 O=C(CCCc1cccnc1)NCc1cc(O)nc(S)n1 ZINC000880512067 DD On-Demand Anodyne TBXAS1 51 44 O=C(CCCc1cccnc1)NCc1cc(O)nc(S)n1 ZINC000880512067 DD On-Demand Anodyne PTAFR 40 48 O=C(CCCc1cccnc1)NCc1cc(O)nc(S)n1 ZINC000880512067 DD On-Demand Anodyne SUCNR1 62 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880512102 GE On-Demand Anodyne F2 34 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880512102 GE On-Demand Anodyne P2RX7 37 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880512103 GE On-Demand Anodyne F2 34 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880512103 GE On-Demand Anodyne P2RX7 37 42 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512108 GE On-Demand Anodyne NPY5R 33 43 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512108 GE On-Demand Anodyne EPHX2 19 48 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512108 GE On-Demand Anodyne TRPM8 21 48 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512109 GE On-Demand Anodyne NPY5R 33 43 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512109 GE On-Demand Anodyne EPHX2 19 48 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)nc1 ZINC000880512109 GE On-Demand Anodyne TRPM8 21 48 O=C(NCc1cc(O)nc(S)n1)[C@H]1Cc2ccccc2CO1 ZINC000880512220 DD On-Demand Anodyne PTPRF 41 32 O=C(NCc1cc(O)nc(S)n1)[C@@H]1Cc2ccccc2CO1 ZINC000880512221 DD On-Demand Anodyne PTPRF 41 32 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@](O)(C(F)F)C2)nc1 ZINC000880512327 EC On-Demand Anodyne NPY5R 25 42 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@](O)(C(F)F)C2)nc1 ZINC000880512327 EC On-Demand Anodyne S1PR2 25 42 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@](O)(C(F)F)C2)nc1 ZINC000880512328 EC On-Demand Anodyne NPY5R 25 42 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@](O)(C(F)F)C2)nc1 ZINC000880512328 EC On-Demand Anodyne S1PR2 25 42 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512455 CE On-Demand Anodyne ADRB2 42 47 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512455 CE On-Demand Anodyne ADRB1 56 41 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512455 CE On-Demand Anodyne ADRB3 38 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512456 CE On-Demand Anodyne ADRB2 42 47 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512456 CE On-Demand Anodyne ADRB1 56 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1 ZINC000880512456 CE On-Demand Anodyne ADRB3 38 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512457 CE On-Demand Anodyne ADRB2 42 47 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512457 CE On-Demand Anodyne ADRB1 56 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512457 CE On-Demand Anodyne ADRB3 38 41 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512458 CE On-Demand Anodyne ADRB2 42 47 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512458 CE On-Demand Anodyne ADRB1 56 41 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880512458 CE On-Demand Anodyne ADRB3 38 41 C[C@@H]1Cc2ccccc2N1C(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512507 DF On-Demand Anodyne DRD4 23 43 C[C@@H]1Cc2ccccc2N1C(=O)CN[C@H]1CCC[C@@]12CCCO2 ZINC000880512508 DF On-Demand Anodyne DRD4 23 43 C[C@@H]1Cc2ccccc2N1C(=O)CN[C@H]1CCC[C@]12CCCO2 ZINC000880512509 DF On-Demand Anodyne DRD4 23 43 C[C@@H]1Cc2ccccc2N1C(=O)CN[C@@H]1CCC[C@@]12CCCO2 ZINC000880512510 DF On-Demand Anodyne DRD4 23 43 O=C(c1cccc(CN[C@@H]2CCC[C@]23CCCO3)c1)N1CCCCC1 ZINC000880512585 EH On-Demand Anodyne L3MBTL3 45 40 O=C(c1cccc(CN[C@H]2CCC[C@]23CCCO3)c1)N1CCCCC1 ZINC000880512587 EH On-Demand Anodyne L3MBTL3 45 40 O=C(c1cccc(CN[C@H]2CCC[C@@]23CCCO3)c1)N1CCCCC1 ZINC000880512589 EH On-Demand Anodyne L3MBTL3 45 40 O=C(c1cccc(CN[C@@H]2CCC[C@@]23CCCO3)c1)N1CCCCC1 ZINC000880512592 EH On-Demand Anodyne L3MBTL3 45 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1C[C@H]1c1ccsc1 ZINC000880512605 DD On-Demand Anodyne NPBWR1 68 30 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccc2ccccc2c1 ZINC000880512672 EG On-Demand Anodyne ADRB2 28 52 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccc2ccccc2c1 ZINC000880512673 EG On-Demand Anodyne ADRB2 28 52 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccc2ccccc2c1 ZINC000880512675 EG On-Demand Anodyne ADRB2 28 52 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc2ccccc2c1 ZINC000880512676 EG On-Demand Anodyne ADRB2 28 52 O=C(CCCc1ccc(F)cc1)NCc1cc(O)nc(S)n1 ZINC000880512718 DE On-Demand Anodyne SUCNR1 59 38 Cc1cccc(NC(=O)[C@H](C)N[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880512730 DG On-Demand Anodyne KCNK3 42 34 CO[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880512751 DD On-Demand Anodyne MME 81 43 CO[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880512751 DD On-Demand Anodyne ACE2 41 34 CO[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880512751 DD On-Demand Anodyne AMP1_PLAFQ 45 38 CO[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880512751 DD On-Demand Anodyne GPR142 76 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne MME 60 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne TIMP3 81 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne CAPN1 45 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne ACE2 53 37 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne PSMB8 50 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880512760 ED On-Demand Anodyne BRCA1 50 30 N#Cc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512763 DD On-Demand Mild ADRB1 30 40 CC(C)c1cccc(CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880512768 DE On-Demand Anodyne ADRB2 44 38 Cc1cccc(NC(=O)[C@H](C)N[C@H]2CCC[C@@]23CCCO3)c1 ZINC000880512781 DG On-Demand Anodyne KCNK3 42 34 Cc1cccc(NC(=O)[C@H](C)N[C@@H]2CCC[C@@]23CCCO3)c1 ZINC000880512784 DG On-Demand Anodyne KCNK3 42 34 Cc1cccc(NC(=O)[C@H](C)N[C@H]2CCC[C@]23CCCO3)c1 ZINC000880512785 DG On-Demand Anodyne KCNK3 42 34 CC[C@@H](C)[C@H](NC(=O)CN[C@@H]1CCC[C@]12CCCO2)C(=O)OC ZINC000880512794 ED On-Demand Anodyne MAP2 41 33 CC[C@@H](C)[C@@H](NC(=O)CN[C@@H]1CCC[C@]12CCCO2)C(=O)OC ZINC000880512806 ED On-Demand Anodyne MAP2 41 33 O=C(CN[C@H]1CCC[C@]12CCCO2)Nc1ccc2c(c1)CCC2 ZINC000880512868 DF On-Demand Anodyne PTPRF 40 30 O=C(CN[C@@H]1CCC[C@@]12CCCO2)Nc1ccc2c(c1)CCC2 ZINC000880512869 DF On-Demand Anodyne PTPRF 40 30 O=C(CN[C@@H]1CCC[C@]12CCCO2)Nc1ccc2c(c1)CCC2 ZINC000880512870 DF On-Demand Anodyne PTPRF 40 30 O=C(CN[C@H]1CCC[C@@]12CCCO2)Nc1ccc2c(c1)CCC2 ZINC000880512871 DF On-Demand Anodyne PTPRF 40 30 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512876 EE On-Demand Anodyne ADRB2 40 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512876 EE On-Demand Anodyne ADRB1 73 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512876 EE On-Demand Anodyne ADRB3 48 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880512877 EE On-Demand Anodyne ADRB2 40 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880512877 EE On-Demand Anodyne ADRB1 73 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880512877 EE On-Demand Anodyne ADRB3 48 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512878 EE On-Demand Anodyne ADRB2 40 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512878 EE On-Demand Anodyne ADRB1 73 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880512878 EE On-Demand Anodyne ADRB3 48 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512879 EE On-Demand Anodyne ADRB2 40 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512879 EE On-Demand Anodyne ADRB1 73 56 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880512879 EE On-Demand Anodyne ADRB3 48 46 CC1(C)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC[S@]1=O ZINC000880512971 FD On-Demand Anodyne NPY5R 30 44 CC1(C)CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC[S@@]1=O ZINC000880512972 FD On-Demand Anodyne NPY5R 30 44 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCc1ccccc1 ZINC000880513018 DE On-Demand Anodyne PROC 55 34 C[C@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1 ZINC000880513066 CF On-Demand Anodyne TIMP3 61 32 C[C@H](N[C@@H]1CCC[C@@]12CCCO2)C(=O)Nc1ccccc1 ZINC000880513068 CF On-Demand Anodyne TIMP3 61 32 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880513125 EF On-Demand Anodyne ADRB2 24 41 O[C@H](CN[C@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880513125 EF On-Demand Anodyne ADRB1 19 41 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1Cl ZINC000880513126 EF On-Demand Anodyne ADRB2 24 41 O[C@H](CN[C@@H]1CCC[C@@]12CCCO2)COc1ccccc1Cl ZINC000880513126 EF On-Demand Anodyne ADRB1 19 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1Cl ZINC000880513127 EF On-Demand Anodyne ADRB2 24 41 O[C@H](CN[C@H]1CCC[C@@]12CCCO2)COc1ccccc1Cl ZINC000880513127 EF On-Demand Anodyne ADRB1 19 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880513128 EF On-Demand Anodyne ADRB2 24 41 O[C@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880513128 EF On-Demand Anodyne ADRB1 19 41 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880513180 FF On-Demand Anodyne ADRB2 40 42 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880513180 FF On-Demand Anodyne ADRB1 68 47 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880513180 FF On-Demand Anodyne ADRB3 48 40 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@]23CCCO3)cc1 ZINC000880513180 FF On-Demand Anodyne ABCB1 15 41 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513181 FF On-Demand Anodyne ADRB2 40 42 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513181 FF On-Demand Anodyne ADRB1 68 47 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513181 FF On-Demand Anodyne ADRB3 48 40 CC(=O)CCc1ccc(OC[C@H](O)CN[C@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513181 FF On-Demand Anodyne ABCB1 15 41 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513182 FF On-Demand Anodyne ADRB2 40 42 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513182 FF On-Demand Anodyne ADRB1 68 47 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513182 FF On-Demand Anodyne ADRB3 48 40 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@@]23CCCO3)cc1 ZINC000880513182 FF On-Demand Anodyne ABCB1 15 41 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513183 FF On-Demand Anodyne ADRB2 40 42 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513183 FF On-Demand Anodyne ADRB1 68 47 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513183 FF On-Demand Anodyne ADRB3 48 40 CC(=O)CCc1ccc(OC[C@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513183 FF On-Demand Anodyne ABCB1 15 41 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880513258 EE On-Demand Anodyne ADRB2 25 43 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880513258 EE On-Demand Anodyne ADRB3 19 40 CC(C)[C@H](CCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513267 EF On-Demand Anodyne MME 42 38 CC(C)[C@H](CCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513267 EF On-Demand Anodyne LAP3 40 32 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H](C)c1ccccc1 ZINC000880513271 DF On-Demand Anodyne BIRC8 44 33 C[C@H](NC(=O)[C@@H](C)N[C@@H]1CCC[C@]12CCCO2)c1ccccc1 ZINC000880513272 DF On-Demand Anodyne BIRC8 44 33 COC(=O)c1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513295 ED On-Demand Anodyne ADRB2 33 43 COC(=O)c1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513295 ED On-Demand Anodyne ADRB1 48 40 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OC1CC1 ZINC000880513296 DD On-Demand Anodyne HCN1 48 33 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OC1CC1 ZINC000880513296 DD On-Demand Anodyne HCN4 41 33 O=C(CCCc1c(F)cccc1F)NCc1cc(O)nc(S)n1 ZINC000880513299 EE On-Demand Anodyne SUCNR1 62 36 CCn1nc(C)c(CC(=O)NCc2cc(O)nc(S)n2)c1C ZINC000880513323 DD On-Demand Anodyne P2RX7 42 54 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCN(c2ccccc2)C1 ZINC000880513325 ED On-Demand Anodyne EPHX2 15 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCN(c2ccccc2)C1 ZINC000880513325 ED On-Demand Anodyne PDE8B 40 31 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCN(c2ccccc2)C1 ZINC000880513326 ED On-Demand Anodyne EPHX2 15 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCN(c2ccccc2)C1 ZINC000880513326 ED On-Demand Anodyne PDE8B 40 31 CCCc1ccc(CCCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880513330 EG On-Demand Anodyne MTNR1A 15 40 CCCc1ccc(CCCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880513330 EG On-Demand Anodyne SUCNR1 60 40 CS(=O)(=O)c1ccc(NC(=O)N[C@@H]2Cc3ccc(Cl)cc3C2)nc1 ZINC000880513344 FE On-Demand Anodyne CA7 21 48 CS(=O)(=O)c1ccc(NC(=O)N[C@H]2Cc3ccc(Cl)cc3C2)nc1 ZINC000880513346 FE On-Demand Anodyne CA7 21 48 C[C@@H](NC(=O)CN[C@@H]1CCC[C@]12CCCO2)c1ccc(Cl)cc1 ZINC000880513370 EG On-Demand Anodyne PRCP 15 41 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCCC2)c1 ZINC000880513372 FE On-Demand Anodyne ACHE 15 40 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCCC2)c1 ZINC000880513372 FE On-Demand Anodyne HRH2 36 42 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCCC2)c1 ZINC000880513372 FE On-Demand Anodyne CHRM3 20 46 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCCC2)c1 ZINC000880513372 FE On-Demand Anodyne BDKRB1 30 44 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCCC2)c1 ZINC000880513372 FE On-Demand Anodyne MCHR1 19 41 CSc1ccc(CCCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880513375 EF On-Demand Anodyne SUCNR1 60 38 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)C1CC1 ZINC000880513426 DC On-Demand Anodyne F2 47 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)C1CC1 ZINC000880513426 DC On-Demand Anodyne PREP 77 36 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)C1CC1 ZINC000880513426 DC On-Demand Anodyne TMPRSS11D 40 32 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880513427 DE On-Demand Anodyne ADRB2 26 41 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880513427 DE On-Demand Anodyne ADRB1 35 40 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc(F)cc1 ZINC000880513427 DE On-Demand Anodyne ADRB3 19 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880513433 DE On-Demand Anodyne ANPEP 15 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccccc1 ZINC000880513433 DE On-Demand Anodyne AMP1_PLAFQ 22 40 C[C@@H](OCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513437 ED On-Demand Anodyne AMP1_PLAFQ 40 34 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@H](c3ccccn3)C2)nc1 ZINC000880513446 ED On-Demand Anodyne RBP4 40 37 O=C(NCc1cc(O)nc(S)n1)c1ccccc1N1CCCCC1 ZINC000880513447 EE On-Demand Anodyne KCNQ2 66 36 O=C(NCc1cc(O)nc(S)n1)c1ccccc1N1CCCCC1 ZINC000880513447 EE On-Demand Anodyne SCN2A 18 41 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H](c3ccccn3)C2)nc1 ZINC000880513453 ED On-Demand Anodyne RBP4 40 37 C[C@H]1CCCCN1C(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880513484 CE On-Demand Anodyne DPP7 17 40 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513503 FD On-Demand Anodyne MTNR1A 17 47 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513503 FD On-Demand Anodyne MTNR1B 15 47 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513505 FD On-Demand Anodyne MTNR1A 17 47 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513505 FD On-Demand Anodyne MTNR1B 15 47 O=C(CCCc1cccc(C(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880513516 FG On-Demand Anodyne CSNK1D 26 40 O=C(CCCc1cccc(C(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880513516 FG On-Demand Anodyne SUCNR1 64 43 Cc1nc(CC2CC2)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880513523 EE On-Demand Anodyne SCD1 27 40 Cc1c(NC(=O)[C@@H](C)N[C@@H]2CCC[C@]23CCCO3)c(=O)n(-c2ccccc2)n1C ZINC000880513535 GF On-Demand Anodyne FPR2 39 41 CCCc1c(C(=O)NCc2cc(O)nc(S)n2)cnn1-c1ccc(C)cc1 ZINC000880513541 GF On-Demand Anodyne GPR142 56 37 O=C(NCc1cc(O)nc(S)n1)c1cc(F)c(N2CCOCC2)c(F)c1 ZINC000880513564 GD On-Demand Anodyne STAT6 43 32 Cc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513624 DE On-Demand Anodyne ADRB2 29 50 Cc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513624 DE On-Demand Anodyne ADRB1 35 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880513637 GE On-Demand Anodyne SIGMAR1 31 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880513637 GE On-Demand Anodyne NPFFR1 41 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880513640 GE On-Demand Anodyne SIGMAR1 31 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880513640 GE On-Demand Anodyne NPFFR1 41 35 O=C(NCc1cc(O)nc(S)n1)[C@@H]1C[C@H]1c1cccnc1 ZINC000880513658 DD On-Demand Anodyne NAMPT 27 48 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880513670 EF On-Demand Anodyne XIAP 30 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880513670 EF On-Demand Anodyne BIRC3 59 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCOc2ccccc21 ZINC000880513670 EF On-Demand Anodyne BIRC2 30 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880513672 EF On-Demand Anodyne XIAP 30 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880513672 EF On-Demand Anodyne BIRC3 59 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCOc2ccccc21 ZINC000880513672 EF On-Demand Anodyne BIRC2 30 40 O=C(CC12C[C@H]3C[C@@H](CC(F)(C3)C1)C2)NCc1cc(O)nc(S)n1 ZINC000880513674 FF On-Demand Anodyne BOTA 30 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880513694 FC On-Demand Anodyne F2 46 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880513695 FC On-Demand Anodyne F2 46 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1c1ccccc1 ZINC000880513704 ED On-Demand Anodyne PREP 40 33 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1c1ccccc1 ZINC000880513705 ED On-Demand Anodyne PREP 40 33 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880513725 DE On-Demand Anodyne ADRB2 24 43 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1F ZINC000880513725 DE On-Demand Anodyne ADRB1 24 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCN(c2ccccc2Cl)C1 ZINC000880513729 FE On-Demand Anodyne EPHX2 22 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880513730 FE On-Demand Anodyne EPHX2 22 40 CN1CCCC[C@@H]1CCC(=O)NCc1cc(O)nc(S)n1 ZINC000880513732 DD On-Demand Anodyne ACKR3 62 32 CN1CCCC[C@H]1CCC(=O)NCc1cc(O)nc(S)n1 ZINC000880513735 DD On-Demand Anodyne ACKR3 62 32 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne SSTR2 51 37 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne EDNRB 18 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne TACR1 21 44 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne CCKAR 34 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne BRS3 27 42 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne NMBR 86 36 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne GRPR 95 36 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne ECE1 46 36 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne CCKBR 38 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne MMP9 15 44 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1c[nH]c2ccccc12 ZINC000880513740 FF On-Demand Anodyne PSMB8 24 40 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513783 GF On-Demand Anodyne ACE 18 40 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513783 GF On-Demand Anodyne TRPV1 32 40 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513783 GF On-Demand Anodyne ACE2 58 36 CCOc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513793 EF On-Demand Anodyne ADRB2 28 40 CCOc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513793 EF On-Demand Anodyne ADRB1 35 40 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCC2)nc1 ZINC000880513807 DD On-Demand Anodyne HPGDS 21 42 CC(=O)c1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513832 EE On-Demand Anodyne ADRB2 28 42 CC(=O)c1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880513832 EE On-Demand Anodyne ADRB1 40 41 CN(C)[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1ccc(Cl)cc1 ZINC000880513849 FE On-Demand Anodyne UTS2 42 32 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCCC2)cc1 ZINC000880513881 FE On-Demand Anodyne ACHE 15 49 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCCC2)cc1 ZINC000880513881 FE On-Demand Anodyne HRH3 21 49 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCCC2)cc1 ZINC000880513881 FE On-Demand Anodyne MCHR1 23 41 CCCc1c(C(=O)NCc2cc(O)nc(S)n2)cnn1-c1cccc(C)c1 ZINC000880513890 GF On-Demand Anodyne GPR142 57 38 C[C@@H](Oc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513892 FF On-Demand Anodyne PPARA 15 41 C[C@@H](Oc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513892 FF On-Demand Anodyne PPARD 30 41 O=C(CCCCCc1ccc(F)cc1)NCc1cc(O)nc(S)n1 ZINC000880513896 EG On-Demand Anodyne FAAH 40 39 O=C(CCCCCc1ccc(F)cc1)NCc1cc(O)nc(S)n1 ZINC000880513896 EG On-Demand Anodyne CES1 45 35 O=C(CCCCCc1ccc(F)cc1)NCc1cc(O)nc(S)n1 ZINC000880513896 EG On-Demand Anodyne SUCNR1 55 36 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne ACE 67 42 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne MME 160 42 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne ANPEP 67 36 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne FCER2 76 36 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne CPA1 50 41 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne TIMP3 48 35 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne TPH1 46 33 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne CAPNS1 57 32 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne MMP3 21 42 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne GRIA1 42 37 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne CAPN1 57 40 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne CAPN2 68 39 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne ACE2 81 41 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne MMP1 26 40 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne FPR1 62 38 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne AMP1_PLAFQ 56 40 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne BLA1_STEMA 72 40 C[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880513915 DD On-Demand Anodyne GPR142 81 38 COc1cccc([C@H](C)CCCC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513932 FG On-Demand Anodyne MTNR1A 36 41 COc1cccc([C@H](C)CCCC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513932 FG On-Demand Anodyne MTNR1B 33 41 COc1cccc([C@@H](C)CCCC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513933 FG On-Demand Anodyne MTNR1A 36 41 COc1cccc([C@@H](C)CCCC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880513933 FG On-Demand Anodyne MTNR1B 33 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1C(F)(F)F ZINC000880513934 FH On-Demand Anodyne RBP4 51 34 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880513948 EG On-Demand Anodyne ADRB2 29 52 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880513948 EG On-Demand Anodyne ADRB1 25 52 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2ccccc12 ZINC000880513948 EG On-Demand Anodyne ADRB3 15 52 CC[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(OC)cc1 ZINC000880513949 EG On-Demand Anodyne TIMP3 70 43 COCCOc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880513951 ED On-Demand Anodyne CA9 18 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880513956 EG On-Demand Anodyne EPHX2 28 40 CCCOc1cc(OC)ccc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880513957 EE On-Demand Anodyne MTNR1A 23 42 CCCOc1cc(OC)ccc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880513957 EE On-Demand Anodyne MTNR1B 20 42 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N1c2ccccc2C[C@H]1C ZINC000880513983 EG On-Demand Anodyne TPP2 53 34 Cn1nc(C(F)(F)F)cc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880514009 ED On-Demand Anodyne CARM1 56 41 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880514044 CE On-Demand Anodyne ADRB2 42 47 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880514044 CE On-Demand Anodyne ADRB1 56 41 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1 ZINC000880514044 CE On-Demand Anodyne ADRB3 38 41 O=C(NCc1cc(O)nc(S)n1)c1ccc(NCC2CC2)nc1 ZINC000880514060 ED On-Demand Anodyne IKBKB 20 41 O=C(NCc1cc(O)nc(S)n1)c1ccc(NCC2CC2)nc1 ZINC000880514060 ED On-Demand Anodyne VCP 47 33 O=C(CCCc1ccccc1Cl)NCc1cc(O)nc(S)n1 ZINC000880514063 EF On-Demand Anodyne SUCNR1 64 41 CCCOc1cccnc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880514064 DD On-Demand Anodyne MAP1 27 40 O=C(CCCc1ccc(O)c(F)c1)NCc1cc(O)nc(S)n1 ZINC000880514077 ED On-Demand Anodyne SUCNR1 56 37 CN1CCOc2ccc(C(=O)NCc3cc(O)nc(S)n3)cc21 ZINC000880514078 ED On-Demand Anodyne CPT1A 17 43 CN1CCOc2ccc(C(=O)NCc3cc(O)nc(S)n3)cc21 ZINC000880514078 ED On-Demand Anodyne CPT1B 21 43 CCOc1ccccc1NC(=O)[C@@H](C)N[C@@H]1CCC[C@]12CCCO2 ZINC000880514095 EG On-Demand Anodyne HCN1 46 34 CCOc1ccccc1NC(=O)[C@@H](C)N[C@@H]1CCC[C@]12CCCO2 ZINC000880514095 EG On-Demand Anodyne HCN4 44 34 CCCc1c(C(=O)NCc2cc(O)nc(S)n2)cnn1-c1ccccc1C ZINC000880514129 GF On-Demand Anodyne GPR142 62 42 O=C(NCc1cc(O)nc(S)n1)c1cc(F)ccc1N1CCOCC1 ZINC000880514137 FD On-Demand Anodyne PIK3CD 15 41 O=C(NCc1cc(O)nc(S)n1)c1cc(F)ccc1N1CCOCC1 ZINC000880514137 FD On-Demand Anodyne PIK3CB 27 41 O=C(NCc1cc(O)nc(S)n1)c1cc(F)ccc1N1CCOCC1 ZINC000880514137 FD On-Demand Anodyne STAT6 55 36 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne F2 72 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne TRY1_BOVIN 72 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne DPP4 18 44 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne PREP 101 48 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne XIAP 34 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880514146 FD On-Demand Anodyne TMPRSS11D 71 39 CN1C[C@@H](C(=O)NCc2cc(O)nc(S)n2)c2ccccc2C1=O ZINC000880514187 EC On-Demand Anodyne P2RX7 49 36 CN1C[C@H](C(=O)NCc2cc(O)nc(S)n2)c2ccccc2C1=O ZINC000880514188 EC On-Demand Anodyne P2RX7 49 36 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne ACE 20 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne SSTR2 57 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne OPRM1 16 41 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MME 27 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne EDNRB 50 34 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne EDNRA 32 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne TACR1 35 47 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MC4R 48 37 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne TACR2 15 44 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne CCKAR 105 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne BRS3 27 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne NMBR 75 34 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MC3R 64 36 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MC5R 66 34 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MMP2 26 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MMP8 34 41 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne GRPR 103 37 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne ECE1 64 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MMP11 86 36 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne CCKBR 93 41 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne GHSR 66 44 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MMP9 25 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne MC1R 90 37 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne NPR 26 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne KISS1R 64 35 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne ERAP2 41 35 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514189 GE On-Demand Anodyne PSMB8 25 42 N#CCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514201 EE On-Demand Mild ADRB1 33 41 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccc2ccccc2c1 ZINC000880514212 EG On-Demand Anodyne ADRB2 28 52 Cc1cccc(NC(=O)[C@@H](C)N[C@@H]2CCC[C@]23CCCO3)c1 ZINC000880514215 DG On-Demand Anodyne KCNK3 42 34 O=C(CCc1cccc(C(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880514247 FF On-Demand Anodyne CSNK1D 26 41 O=C(CCc1cccc(C(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880514247 FF On-Demand Anodyne SUCNR1 43 39 O=C(CCc1cccc(C(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880514247 FF On-Demand Anodyne PDS 36 40 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCC2)cc1 ZINC000880514252 ED On-Demand Anodyne ACHE 16 47 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCC2)cc1 ZINC000880514252 ED On-Demand Anodyne HRH3 16 47 O=C(NCc1cc(O)nc(S)n1)c1ccc(CN2CCCC2)cc1 ZINC000880514252 ED On-Demand Anodyne MCHR1 25 41 O=C(NCc1cc(O)nc(S)n1)c1ccccc1N1CCOCC1 ZINC000880514300 ED On-Demand Anodyne SCN10A 15 43 O=C(NCc1cc(O)nc(S)n1)c1ccccc1N1CCOCC1 ZINC000880514300 ED On-Demand Anodyne PIK3CB 40 39 O=C(NCc1cc(O)nc(S)n1)c1ccccc1N1CCOCC1 ZINC000880514300 ED On-Demand Anodyne STAT6 53 34 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514309 EE On-Demand Anodyne ADRB2 40 56 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514309 EE On-Demand Anodyne ADRB1 73 56 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514309 EE On-Demand Anodyne ADRB3 48 46 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880514346 EF On-Demand Anodyne ADRB2 24 41 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1ccccc1Cl ZINC000880514346 EF On-Demand Anodyne ADRB1 19 41 O=C(NCc1cc(O)nc(S)n1)C1CCN(CC(F)(F)F)CC1 ZINC000880514359 FD On-Demand Anodyne HPGDS 34 40 CC(=O)CCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514371 FF On-Demand Anodyne ADRB2 40 42 CC(=O)CCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514371 FF On-Demand Anodyne ADRB1 68 47 CC(=O)CCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514371 FF On-Demand Anodyne ADRB3 48 40 CC(=O)CCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880514371 FF On-Demand Anodyne ABCB1 15 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCc1ccccc1 ZINC000880514410 DE On-Demand Anodyne PROC 55 34 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1 ZINC000880514433 CF On-Demand Anodyne TIMP3 61 32 O=C(NCc1cc(O)nc(S)n1)[C@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880514449 FD On-Demand Anodyne PDS 40 36 O=C(NCc1cc(O)nc(S)n1)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880514450 FD On-Demand Anodyne PDS 40 36 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1ccc(F)cc1 ZINC000880514471 DE On-Demand Anodyne KCNQ2 25 41 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1ccc(F)cc1 ZINC000880514472 DE On-Demand Anodyne KCNQ2 25 41 O=C(NCc1cc(O)nc(S)n1)C1Cc2ccccc2C1 ZINC000880514477 DD On-Demand Anodyne PDE8B 40 32 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCc2cccnc21 ZINC000880514484 DD On-Demand Anodyne CXCR4 68 39 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCc2cccnc21 ZINC000880514485 DD On-Demand Anodyne CXCR4 68 39 O=C1OCC[C@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880514532 BC On-Demand Anodyne LUXR 44 34 O=C1OCC[C@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880514532 BC On-Demand Anodyne TRAR 68 34 O=C1OCC[C@H]1N[C@@H]1CCC[C@]12CCCO2 ZINC000880514532 BC On-Demand Anodyne LASR 42 31 CCC(C)(C)c1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880514542 EG On-Demand Anodyne MT-ND1 15 46 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(c2ccc(Cl)c(F)c2)C1 ZINC000880514560 GD On-Demand Anodyne P2RX7 29 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(c2ccc(Cl)c(F)c2)C1 ZINC000880514561 GD On-Demand Anodyne P2RX7 29 42 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1ccc(OC)cc1 ZINC000880514588 EE On-Demand Anodyne KCNQ2 25 44 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1ccc(OC)cc1 ZINC000880514589 EE On-Demand Anodyne KCNQ2 25 44 C[C@@](O)(CN[C@@H]1CCC[C@]12CCCO2)c1ccccc1 ZINC000880514602 CF On-Demand Anodyne AMY2 44 30 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(CC(F)(F)F)C1 ZINC000880514613 FD On-Demand Anodyne SLC6A1 72 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(CC(F)(F)F)C1 ZINC000880514614 FD On-Demand Anodyne SLC6A1 72 34 CCCCSc1ccc(Cl)cc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880514663 GH On-Demand Anodyne UL54 43 32 CC1(C)C[C@@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880514678 CD On-Demand Anodyne DPEP1 46 34 CCOc1ccccc1C(F)(F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514721 FE On-Demand Anodyne KCNK3 19 40 CCOc1ccccc1C(F)(F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514721 FE On-Demand Anodyne KCNK9 18 40 COc1cccc(OC)c1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514735 FE On-Demand Anodyne ADRB2 21 43 COc1cccc(OC)c1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880514735 FE On-Demand Anodyne ADRB1 24 43 O=C(CCCc1cc(F)ccc1F)NCc1cc(O)nc(S)n1 ZINC000880514743 EE On-Demand Anodyne SUCNR1 56 35 O=C(CCCc1ccsc1)NCc1cc(O)nc(S)n1 ZINC000880514744 DE On-Demand Anodyne SUCNR1 42 38 C[C@@H](Cc1cccc(Cl)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514763 EF On-Demand Anodyne CTSL 19 44 C[C@@H](Cc1cccc(Cl)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514763 EF On-Demand Anodyne CTSV 39 44 Cc1ccc(C[C@@H](C)C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880514822 DE On-Demand Anodyne MME 74 38 Cc1ccc(C[C@@H](C)C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880514822 DE On-Demand Anodyne TPH1 53 34 Cc1ccc(C[C@@H](C)C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880514822 DE On-Demand Anodyne GRIA1 42 33 Cc1ccc(C[C@@H](C)C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880514822 DE On-Demand Anodyne ACE2 63 38 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne MME 50 40 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne MMP3 47 39 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne FAAH 43 34 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne FURIN 52 35 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne CES1 45 33 C[C@@H](CCCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514854 EF On-Demand Anodyne AMP1_PLAFQ 47 38 O=C(CCCCc1ccc(Cl)c(Cl)c1)NCc1cc(O)nc(S)n1 ZINC000880514860 GH On-Demand Anodyne SUCNR1 41 39 CCCOc1ccc(Cl)cc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880514960 FF On-Demand Anodyne PTGER1 26 45 CS(=O)(=O)c1ccc(NC(=O)NC23CCC(CC2)C3)nc1 ZINC000880514978 DD On-Demand Anodyne EPHX2 38 44 C[C@H](CSCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514988 EF On-Demand Anodyne ACE 26 49 C[C@H](CSCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514988 EF On-Demand Anodyne MME 37 49 C[C@H](CSCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880514988 EF On-Demand Anodyne LTA4H 15 44 O=C(CCCc1ccccc1Br)NCc1cc(O)nc(S)n1 ZINC000880515001 GF On-Demand Anodyne SUCNR1 51 36 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccccc1[N+](=O)[O-] ZINC000880515007 EF On-Demand Bother COLA 45 35 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(N2CCOCC2)cc1 ZINC000880515009 FF On-Demand Anodyne MTOR 56 37 O=C(Cc1cccc(OCC(F)(F)F)c1)NCc1cc(O)nc(S)n1 ZINC000880515019 FE On-Demand Anodyne PDS 55 38 O=C(CCCc1cccc(Br)c1)NCc1cc(O)nc(S)n1 ZINC000880515031 GF On-Demand Anodyne SUCNR1 55 36 COc1cc2c(cc1OC)CN(CC(=O)NCc1cc(O)nc(S)n1)CC2 ZINC000880515034 GD On-Demand Anodyne ABCB1B 67 39 COc1cc2c(cc1OC)CN(CC(=O)NCc1cc(O)nc(S)n1)CC2 ZINC000880515034 GD On-Demand Anodyne ABCB1 25 44 COc1cccc([C@@H](C)CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515036 EE On-Demand Anodyne MTNR1A 43 41 COc1cccc([C@@H](C)CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515036 EE On-Demand Anodyne MTNR1B 42 41 COc1cccc([C@H](C)CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515037 EE On-Demand Anodyne MTNR1A 43 41 COc1cccc([C@H](C)CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515037 EE On-Demand Anodyne MTNR1B 42 41 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515086 FG On-Demand Anodyne KCNQ2 28 48 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515086 FG On-Demand Anodyne CCR2 32 40 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515086 FG On-Demand Anodyne PDS 41 37 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515087 FG On-Demand Anodyne KCNQ2 28 48 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515087 FG On-Demand Anodyne CCR2 32 40 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515087 FG On-Demand Anodyne PDS 41 37 O=C(CCCc1ccc(F)c(F)c1)NCc1cc(O)nc(S)n1 ZINC000880515097 EE On-Demand Anodyne SUCNR1 61 39 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880515102 EF On-Demand Anodyne ADRB2 16 68 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)COc1cccc2[nH]ccc12 ZINC000880515102 EF On-Demand Anodyne ADRB1 24 68 CCCOc1cccc(CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515163 EE On-Demand Anodyne MTNR1A 37 44 CCCOc1cccc(CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515163 EE On-Demand Anodyne ROCK2 15 47 CCCOc1cccc(CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515163 EE On-Demand Anodyne PLA2G4B 25 40 CCCOc1cccc(CC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515163 EE On-Demand Anodyne PDS 59 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1C[C@@H]1Cc1ccccc1 ZINC000880515206 DD On-Demand Anodyne LNPEP 40 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1C[C@H]1Cc1ccccc1 ZINC000880515207 DD On-Demand Anodyne LNPEP 40 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1C[C@@H]1Cc1ccccc1 ZINC000880515208 DD On-Demand Anodyne LNPEP 40 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1C[C@H]1Cc1ccccc1 ZINC000880515209 DD On-Demand Anodyne LNPEP 40 34 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)nc1 ZINC000880515217 GD On-Demand Anodyne NPY5R 24 40 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)nc1 ZINC000880515217 GD On-Demand Anodyne S1PR2 25 44 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)nc1 ZINC000880515218 GD On-Demand Anodyne NPY5R 24 40 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)nc1 ZINC000880515218 GD On-Demand Anodyne S1PR2 25 44 CC(C)(C(=O)NCc1cc(O)nc(S)n1)c1cccc(C(F)(F)F)c1 ZINC000880515222 FG On-Demand Anodyne PDS 42 34 COc1ccc(OCC(=O)NCc2cc(O)nc(S)n2)cc1C ZINC000880515223 ED On-Demand Anodyne PPARD 42 40 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880515225 CG On-Demand Anodyne ADRB3 39 46 O[C@@H](CN[C@@H]1CCC[C@]12CCCO2)c1cccc(Cl)c1 ZINC000880515225 CG On-Demand Anodyne CYP3A4 46 37 O=C(CCCn1cnc2ccccc21)NCc1cc(O)nc(S)n1 ZINC000880515237 ED On-Demand Anodyne PKM 16 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(c2ccc(Cl)cc2)C1 ZINC000880515243 GD On-Demand Anodyne P2RX7 29 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(c2ccc(Cl)cc2)C1 ZINC000880515244 GD On-Demand Anodyne P2RX7 29 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne DRD4 34 48 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne ACHE 21 42 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne SIGMAR1 35 43 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne CCR3 25 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne MCHR1 24 46 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880515246 FE On-Demand Anodyne BIRC2 69 49 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne DRD4 34 48 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne ACHE 21 42 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne SIGMAR1 35 43 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne CCR3 25 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne MCHR1 24 46 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880515247 FE On-Demand Anodyne BIRC2 69 49 O=C(CCCc1ccc(Cl)c(Cl)c1)NCc1cc(O)nc(S)n1 ZINC000880515248 FG On-Demand Anodyne SUCNR1 42 40 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)cc1 ZINC000880515249 ED On-Demand Anodyne PIK3CA 40 39 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)cc1 ZINC000880515249 ED On-Demand Anodyne MTOR 46 39 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)cc1 ZINC000880515249 ED On-Demand Anodyne STAT6 58 37 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)cc1 ZINC000880515249 ED On-Demand Anodyne HPGDS 23 40 COc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515260 DD On-Demand Anodyne TRPV1 70 40 COc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515260 DD On-Demand Anodyne ROCK1 25 40 COc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515260 DD On-Demand Anodyne MTNR1A 37 42 COc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515260 DD On-Demand Anodyne MTNR1B 35 42 COc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515260 DD On-Demand Anodyne ROCK2 24 40 COc1cccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515261 DD On-Demand Anodyne TRPV1 70 40 COc1cccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515261 DD On-Demand Anodyne ROCK1 25 40 COc1cccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515261 DD On-Demand Anodyne MTNR1A 37 42 COc1cccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515261 DD On-Demand Anodyne MTNR1B 35 42 COc1cccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515261 DD On-Demand Anodyne ROCK2 24 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515267 DE On-Demand Anodyne TRPV1 41 38 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515267 DE On-Demand Anodyne ACE2 41 35 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515267 DE On-Demand Anodyne PIN1 22 41 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515267 DE On-Demand Anodyne CARM1 41 33 CCc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515282 GE On-Demand Anodyne GPR119 26 44 O=C(CCCc1ccc(Cl)cc1)NCc1cc(O)nc(S)n1 ZINC000880515288 EF On-Demand Anodyne SUCNR1 66 41 CCOc1ccc(CCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880515294 EE On-Demand Anodyne FFAR4 42 32 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515305 GE On-Demand Anodyne SLC6A1 114 38 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515305 GE On-Demand Anodyne CCR3 48 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515305 GE On-Demand Anodyne PDE8B 46 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515305 GE On-Demand Anodyne CACNA1G 32 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515306 GE On-Demand Anodyne SLC6A1 114 38 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515306 GE On-Demand Anodyne CCR3 48 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515306 GE On-Demand Anodyne PDE8B 46 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880515306 GE On-Demand Anodyne CACNA1G 32 43 Cc1nc(C(C)C)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515321 DE On-Demand Anodyne SCD1 26 42 Cc1nc(C(C)C)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515321 DE On-Demand Anodyne SCD 24 40 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne CHRM2 15 41 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne DRD2 19 43 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne DRD4 49 45 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne ACHE 51 46 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne DRD3 18 43 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne LTA4H 16 42 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne SIGMAR1 57 67 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne CCR3 30 42 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne EPHX2 20 43 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne PDE8B 45 33 O=C(NCc1cc(O)nc(S)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880515325 FD On-Demand Anodyne CACNA1G 50 49 N#C[C@@H](c1cccs1)N1CCN(C(=O)CN[C@@H]2CCC[C@]23CCCO3)CC1 ZINC000880515335 GE On-Demand Mild PTAFR 35 41 CCCc1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880515349 DE On-Demand Anodyne ECR 23 40 CCCc1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880515349 DE On-Demand Anodyne E3UJZ5_SPOLI 20 40 O=C(CCCOc1ccccc1F)NCc1cc(O)nc(S)n1 ZINC000880515352 EE On-Demand Anodyne SUCNR1 54 34 O=C(CCCOc1cccc(F)c1)NCc1cc(O)nc(S)n1 ZINC000880515360 EE On-Demand Anodyne SUCNR1 51 34 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC1CCCC1 ZINC000880515370 GF On-Demand Anodyne PDE4A 44 55 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC1CCCC1 ZINC000880515370 GF On-Demand Anodyne PDE4B 23 55 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC1CCCC1 ZINC000880515370 GF On-Demand Anodyne PDE4D 31 55 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC1CCCC1 ZINC000880515370 GF On-Demand Anodyne PDE4C 21 55 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC1CCCC1 ZINC000880515370 GF On-Demand Anodyne SLC5A7 38 47 O=C(CCCOc1cccc(Cl)c1Cl)NCc1cc(O)nc(S)n1 ZINC000880515376 GG On-Demand Anodyne SUCNR1 45 37 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515380 GD On-Demand Anodyne F2 50 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515380 GD On-Demand Anodyne PREP 92 37 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515380 GD On-Demand Anodyne TMPRSS11D 55 31 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515381 GD On-Demand Anodyne F2 50 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515381 GD On-Demand Anodyne PREP 92 37 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880515381 GD On-Demand Anodyne TMPRSS11D 55 31 CCCN(CC)c1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880515392 EF On-Demand Anodyne NAMPT 21 44 O=C(CCCc1ccccn1)NCc1cc(O)nc(S)n1 ZINC000880515401 DD On-Demand Anodyne SUCNR1 74 44 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne HTR1A 108 50 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne DRD2 83 47 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne DRD4 50 46 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne ADRA1D 29 41 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne HTR2A 74 50 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne HTR2C 33 48 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne SLC6A4 17 46 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne ADRA1A 32 42 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne ADRA1B 21 42 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne DRD3 91 50 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne DRD5 15 41 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne HTR7 141 61 O=C(CCCN1CCN(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515403 GD On-Demand Anodyne CACNA1G 16 43 O=C(CCCCCc1ccc(O)cc1)NCc1cc(O)nc(S)n1 ZINC000880515415 EF On-Demand Anodyne GRIA1 44 36 O=C(CCCCCc1ccc(O)cc1)NCc1cc(O)nc(S)n1 ZINC000880515415 EF On-Demand Anodyne HDAC1 16 42 O=C(CCCCCc1ccc(O)cc1)NCc1cc(O)nc(S)n1 ZINC000880515415 EF On-Demand Anodyne FAAH 50 39 O=C(CCCCCc1ccc(O)cc1)NCc1cc(O)nc(S)n1 ZINC000880515415 EF On-Demand Anodyne CES1 53 35 O=C(CCCCCc1ccc(O)cc1)NCc1cc(O)nc(S)n1 ZINC000880515415 EF On-Demand Anodyne SUCNR1 42 38 CCCCCCCCNC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880515423 EF On-Demand Mild EPHX2 19 44 CCCCCCCCNC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880515423 EF On-Demand Mild ASAH1 76 34 CCCCCCCCNC(=O)Nc1ccc(S(C)(=O)=O)cn1 ZINC000880515423 EF On-Demand Mild NAMPT 15 40 Cc1nc(C(C)(C)C)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515424 EE On-Demand Anodyne SCD1 28 42 Cc1nc(C(C)(C)C)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515424 EE On-Demand Anodyne SCD 26 41 O=C(C[C@@H]1CCc2ccccc2C1)NCc1cc(O)nc(S)n1 ZINC000880515425 EE On-Demand Anodyne PREP 25 40 O=C(C[C@H]1CCc2ccccc2C1)NCc1cc(O)nc(S)n1 ZINC000880515428 EE On-Demand Anodyne PREP 25 40 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCCCC2)cc1 ZINC000880515446 EE On-Demand Anodyne PRNP 41 34 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515449 FF On-Demand Anodyne TACR1 19 43 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515449 FF On-Demand Anodyne TRPV1 55 35 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515449 FF On-Demand Anodyne CCR2 48 40 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515449 FF On-Demand Anodyne CARM1 61 35 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515449 FF On-Demand Anodyne PDS 42 40 O=C(CCCC1CCCC1)NCc1cc(O)nc(S)n1 ZINC000880515452 CE On-Demand Anodyne BMP1 44 35 O=C(CCCc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515457 DE On-Demand Anodyne HDAC8 15 43 O=C(CCCc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515457 DE On-Demand Anodyne HDAC1 20 49 O=C(CCCc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515457 DE On-Demand Anodyne FAAH 60 41 O=C(CCCc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515457 DE On-Demand Anodyne CES1 66 35 O=C(CCCc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515457 DE On-Demand Anodyne SUCNR1 60 42 O=C(NCc1cc(O)nc(S)n1)c1ccc(OCC2CC2)cc1 ZINC000880515459 EE On-Demand Anodyne GRIN2B 21 54 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne F2 51 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne OPRM1 20 47 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne SIGMAR1 17 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne P2RX7 18 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne TRY1_BOVIN 50 37 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne PREP 60 37 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880515467 ED On-Demand Anodyne TMPRSS11D 60 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne F2 51 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne OPRM1 20 47 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne SIGMAR1 17 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne P2RX7 18 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne TRY1_BOVIN 50 37 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne PREP 60 37 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccccc1 ZINC000880515468 ED On-Demand Anodyne TMPRSS11D 60 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880515470 FD On-Demand Anodyne SLC6A1 75 32 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880515470 FD On-Demand Anodyne CHRNA7 40 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccnc2)C1 ZINC000880515471 FD On-Demand Anodyne SLC6A1 75 32 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2cccnc2)C1 ZINC000880515471 FD On-Demand Anodyne CHRNA7 40 35 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000880515488 FC On-Demand Anodyne DRD4 34 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000880515488 FC On-Demand Anodyne SIGMAR1 20 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000880515488 FC On-Demand Anodyne PDE8B 47 31 O=C(NCc1cc(O)nc(S)n1)[C@H]1CN(Cc2ccccc2)CCO1 ZINC000880515489 FC On-Demand Anodyne DRD4 34 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CN(Cc2ccccc2)CCO1 ZINC000880515489 FC On-Demand Anodyne SIGMAR1 20 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CN(Cc2ccccc2)CCO1 ZINC000880515489 FC On-Demand Anodyne PDE8B 47 31 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880515507 GD On-Demand Anodyne L3MBTL3 40 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880515508 GD On-Demand Anodyne L3MBTL3 40 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880515525 FE On-Demand Anodyne F2 40 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880515525 FE On-Demand Anodyne SIGMAR1 16 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880515525 FE On-Demand Anodyne P2RX7 20 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880515525 FE On-Demand Anodyne PREP 40 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880515525 FE On-Demand Anodyne TMPRSS11D 50 32 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880515526 FE On-Demand Anodyne F2 40 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880515526 FE On-Demand Anodyne SIGMAR1 16 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880515526 FE On-Demand Anodyne P2RX7 20 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880515526 FE On-Demand Anodyne PREP 40 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880515526 FE On-Demand Anodyne TMPRSS11D 50 32 O=C(CCc1cccc(OC2CCCC2)c1)NCc1cc(O)nc(S)n1 ZINC000880515531 FG On-Demand Anodyne TNKS 50 38 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(S(C)(=O)=O)cn3)C2)cc1 ZINC000880515553 GF On-Demand Anodyne GPR119 21 42 C[C@@H](OCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515562 DD On-Demand Anodyne CAPN1 42 36 C[C@@H](OCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515562 DD On-Demand Anodyne CAPN2 70 35 C[C@@H](OCc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515562 DD On-Demand Anodyne NPR 68 33 CCOC(=O)[C@@H](N[C@@H]1CCC[C@]12CCCO2)c1ccccc1 ZINC000880515565 DF On-Demand Anodyne TIMP3 68 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne F2 72 48 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne ACE 40 39 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne FKBP1A 27 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne OPRM1 31 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne P2RX7 17 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne TRY1_BOVIN 75 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne DPP4 22 48 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne PREP 106 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne XIAP 38 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne BRCA1 57 30 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515567 FD On-Demand Anodyne TMPRSS11D 71 38 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne F2 72 48 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne ACE 40 39 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne FKBP1A 27 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne OPRM1 31 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne P2RX7 17 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne TRY1_BOVIN 75 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne DPP4 22 48 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne PREP 106 40 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne XIAP 38 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne BRCA1 57 30 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880515568 FD On-Demand Anodyne TMPRSS11D 71 38 O=C(CCCCc1ccc(Br)cc1)NCc1cc(O)nc(S)n1 ZINC000880515582 GG On-Demand Anodyne HDAC1 15 41 O=C(CCCCc1ccc(Br)cc1)NCc1cc(O)nc(S)n1 ZINC000880515582 GG On-Demand Anodyne SUCNR1 44 37 CS(=O)(=O)c1ccc(NC(=O)NC2CCC(N3CCCCC3)CC2)nc1 ZINC000880515617 GE On-Demand Anodyne EPHX2 38 40 CS(=O)(=O)c1ccc(NC(=O)NC2CCC(N3CCCCC3)CC2)nc1 ZINC000880515617 GE On-Demand Anodyne L3MBTL3 58 35 Cc1ccc(-n2nc(C(=O)NCc3cc(O)nc(S)n3)c3c2CCC3)c(C)c1 ZINC000880515618 GF On-Demand Anodyne CNR1 41 35 Cn1nc(C(C)(C)C)cc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515624 DD On-Demand Anodyne CTSV 45 35 Cc1nc(NC2CC2)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880515635 ED On-Demand Anodyne SCD1 27 43 CS(=O)(=O)c1ccc(NC(=O)N2CCc3c(F)cccc3C2)nc1 ZINC000880515705 EE On-Demand Anodyne NPY5R 21 40 Cc1ccc(N2CCC(C(=O)NCc3cc(O)nc(S)n3)CC2)nc1 ZINC000880515712 FD On-Demand Anodyne EPHX2 23 43 C[C@H](CC(=O)NCc1cc(O)nc(S)n1)c1cccnc1 ZINC000880515714 DD On-Demand Anodyne KCNA5 23 48 C[C@@H](CC(=O)NCc1cc(O)nc(S)n1)c1cccnc1 ZINC000880515715 DD On-Demand Anodyne KCNA5 23 48 COCCCOc1cccc(C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515717 ED On-Demand Anodyne DRD4 43 34 O=C(NCc1cc(O)nc(S)n1)c1cccc(OC2CCCC2)c1 ZINC000880515724 EF On-Demand Anodyne DRD4 40 32 O=C(NCc1cc(O)nc(S)n1)c1cccc(OC2CCCC2)c1 ZINC000880515724 EF On-Demand Anodyne TNKS 42 35 O=C(C[C@H]1CN(Cc2ccccc2)CCO1)NCc1cc(O)nc(S)n1 ZINC000880515725 FD On-Demand Anodyne DRD4 30 47 O=C(C[C@H]1CN(Cc2ccccc2)CCO1)NCc1cc(O)nc(S)n1 ZINC000880515725 FD On-Demand Anodyne PDE8B 19 41 O=C(C[C@@H]1CN(Cc2ccccc2)CCO1)NCc1cc(O)nc(S)n1 ZINC000880515726 FD On-Demand Anodyne DRD4 30 47 O=C(C[C@@H]1CN(Cc2ccccc2)CCO1)NCc1cc(O)nc(S)n1 ZINC000880515726 FD On-Demand Anodyne PDE8B 19 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(c2ccc(F)cc2F)C1 ZINC000880515736 GD On-Demand Anodyne P2RX7 15 43 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(c2ccc(F)cc2F)C1 ZINC000880515737 GD On-Demand Anodyne P2RX7 15 43 CCCCCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880515753 CE On-Demand Mild LASR 42 39 COc1ccc2c(c1)C[C@H](C(=O)NCc1cc(O)nc(S)n1)CO2 ZINC000880515781 ED On-Demand Anodyne MTNR1A 19 50 COc1ccc2c(c1)C[C@H](C(=O)NCc1cc(O)nc(S)n1)CO2 ZINC000880515781 ED On-Demand Anodyne ROCK2 38 51 COc1ccc2c(c1)C[C@@H](C(=O)NCc1cc(O)nc(S)n1)CO2 ZINC000880515782 ED On-Demand Anodyne MTNR1A 19 50 COc1ccc2c(c1)C[C@@H](C(=O)NCc1cc(O)nc(S)n1)CO2 ZINC000880515782 ED On-Demand Anodyne ROCK2 38 51 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)nc1 ZINC000880515800 GG On-Demand Anodyne SFRP1 40 33 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)nc1 ZINC000880515800 GG On-Demand Anodyne WNT3 44 33 CCCCCCCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880515807 DG On-Demand Mild LASR 42 39 O=C(CCc1ccc(OC(F)F)cc1)NCc1cc(O)nc(S)n1 ZINC000880515824 FE On-Demand Anodyne PLA2G4A 21 42 c1ccc(CN2CC[C@@H](N[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880515825 DF On-Demand Anodyne DRD4 35 42 c1ccc(CN2CC[C@@H](N[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880515825 DF On-Demand Anodyne SIGMAR1 54 41 CCCc1c(C(=O)NCc2cc(O)nc(S)n2)cnn1Cc1ccccc1 ZINC000880515848 GF On-Demand Anodyne GPR142 51 35 O=C(CCCCC(=O)c1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515851 EF On-Demand Anodyne HDAC8 40 42 O=C(CCCCC(=O)c1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880515851 EF On-Demand Anodyne HDAC1 18 49 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne ACE 23 42 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne MME 50 42 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne TRPV1 61 36 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne GRIA1 40 32 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne ACE2 53 37 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne AMP1_PLAFQ 19 41 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880515862 DE On-Demand Anodyne LEF 42 32 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OCC1CC1 ZINC000880515865 EE On-Demand Anodyne HCN1 60 35 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OCC1CC1 ZINC000880515865 EE On-Demand Anodyne HCN4 45 35 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne DRD4 32 44 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne ACHE 35 41 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne SLC6A1 150 37 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne SIGMAR1 33 50 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne CCR3 24 44 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880515866 FD On-Demand Anodyne PDE8B 58 35 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne DRD4 32 44 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne ACHE 35 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne SLC6A1 150 37 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne SIGMAR1 33 50 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne CCR3 24 44 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880515867 FD On-Demand Anodyne PDE8B 58 35 CS(=O)(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880515890 GF On-Demand Anodyne DRD3 49 36 CS(=O)(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880515890 GF On-Demand Anodyne FGFR1 22 40 CS(=O)(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880515890 GF On-Demand Anodyne CCR3 23 47 CS(=O)(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880515890 GF On-Demand Anodyne CHRNA7 21 48 CS(=O)(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880515890 GF On-Demand Anodyne HNMT 48 37 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCCC2)nc1 ZINC000880515899 ED On-Demand Anodyne HPGDS 21 44 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCCC2)nc1 ZINC000880515899 ED On-Demand Anodyne NAMPT 24 41 CCCOc1cccc(C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880515904 DE On-Demand Anodyne DRD4 41 32 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne DRD4 40 32 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne ACHE 16 41 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne HRH2 34 40 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne CHRM3 20 47 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne SIGMAR1 18 40 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne BDKRB1 24 42 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCCC2)c1 ZINC000880515912 ED On-Demand Anodyne MCHR1 20 42 CN1C(=O)CC[C@H](C(=O)NCc2cc(O)nc(S)n2)[C@@H]1c1ccccc1 ZINC000880515931 FD On-Demand Anodyne P2RX7 28 42 CN1C(=O)CC[C@@H](C(=O)NCc2cc(O)nc(S)n2)[C@@H]1c1ccccc1 ZINC000880515932 FD On-Demand Anodyne P2RX7 28 42 CN1C(=O)CC[C@@H](C(=O)NCc2cc(O)nc(S)n2)[C@H]1c1ccccc1 ZINC000880515933 FD On-Demand Anodyne P2RX7 28 42 CN1C(=O)CC[C@H](C(=O)NCc2cc(O)nc(S)n2)[C@H]1c1ccccc1 ZINC000880515934 FD On-Demand Anodyne P2RX7 28 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCCN1Cc1ccc(F)cc1 ZINC000880515935 GE On-Demand Anodyne P2RX7 27 45 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCCN1Cc1ccc(F)cc1 ZINC000880515936 GE On-Demand Anodyne P2RX7 27 45 O=C(CC1CCC(c2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880515944 FG On-Demand Anodyne DGAT1 46 39 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCCCCC2)nc1 ZINC000880515952 FE On-Demand Anodyne HPGDS 21 45 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCCCCC2)nc1 ZINC000880515952 FE On-Demand Anodyne NAMPT 24 41 O=C(CCCOc1cccnc1)NCc1cc(O)nc(S)n1 ZINC000880515954 DD On-Demand Anodyne SUCNR1 57 36 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)c(F)c1 ZINC000880515964 FD On-Demand Anodyne SCN10A 15 42 O=C(NCc1cc(O)nc(S)n1)c1ccc(N2CCOCC2)c(F)c1 ZINC000880515964 FD On-Demand Anodyne STAT6 44 32 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean PDGFRB 41 39 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean MMP13 60 45 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean MMP3 42 45 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean MMP9 44 39 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean MMP7 42 36 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean MMP1 47 38 COc1ccc(N2CCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880515987 GD On-Demand Clean GPR119 26 40 Cc1cccc([C@@H](C)C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880516015 DE On-Demand Anodyne TRPV1 81 33 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1cccnc1Cl ZINC000880516020 DF On-Demand Anodyne G2YM83_BOTF4 71 36 CC[C@@H](C(=O)NCc1cc(O)nc(S)n1)c1ccccc1 ZINC000880516045 DE On-Demand Anodyne KCNQ2 40 39 CC[C@H](C(=O)NCc1cc(O)nc(S)n1)c1ccccc1 ZINC000880516046 DE On-Demand Anodyne KCNQ2 40 39 CCCCCCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880516064 CF On-Demand Mild LASR 42 39 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880516070 FD On-Demand Anodyne INHA 25 49 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880516071 FD On-Demand Anodyne INHA 25 49 O=C(CCCC1CCCCC1)NCc1cc(O)nc(S)n1 ZINC000880516072 DF On-Demand Anodyne BMP1 65 36 CC(C)c1cccc(OCC(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880516075 EE On-Demand Anodyne PDS 39 44 c1ccc(CN2CCCO[C@@H](CN[C@@H]3CCC[C@]34CCCO4)C2)cc1 ZINC000880516086 EF On-Demand Anodyne DRD4 21 44 CS(=O)(=O)c1ccc(NC(=O)N2CCS(=O)CC2)nc1 ZINC000880516092 DC On-Demand Anodyne NPY5R 24 42 COCCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880516094 EE On-Demand Anodyne ADRB2 37 55 COCCc1ccc(OC[C@@H](O)CN[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880516094 EE On-Demand Anodyne ADRB1 58 55 CS(=O)(=O)c1ccc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)nc1 ZINC000880516102 GF On-Demand Anodyne GCK 29 42 CS(=O)(=O)c1ccc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)nc1 ZINC000880516103 GF On-Demand Anodyne GCK 29 42 CCCCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880516123 CE On-Demand Anodyne LASR 42 39 Cc1cc(OCCCC(=O)NCc2cc(O)nc(S)n2)ccc1Cl ZINC000880516132 FF On-Demand Anodyne MCL1 26 42 Cc1cc(OCCCC(=O)NCc2cc(O)nc(S)n2)ccc1Cl ZINC000880516132 FF On-Demand Anodyne SUCNR1 25 41 O=C(CCCc1ccc(Br)s1)NCc1cc(O)nc(S)n1 ZINC000880516152 GF On-Demand Anodyne SUCNR1 40 34 O=C(NCc1cc(O)nc(S)n1)[C@H]1COc2ccc(Cl)cc2C1 ZINC000880516163 FD On-Demand Anodyne ROCK2 25 47 O=C(NCc1cc(O)nc(S)n1)[C@@H]1COc2ccc(Cl)cc2C1 ZINC000880516164 FD On-Demand Anodyne ROCK2 25 47 CCc1nc2ccccc2n1CC(=O)NCc1cc(O)nc(S)n1 ZINC000880516170 ED On-Demand Anodyne IMDH_CRYPV 34 41 CC[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1ccc(C)cc1 ZINC000880516174 DG On-Demand Anodyne TIMP3 64 32 CC(C)(C)OC(=O)N1CC[C@@H](CCN[C@@H]2CCC[C@]23CCCO3)C1 ZINC000880516175 EG On-Demand Anodyne GPR119 21 41 N#Cc1ccccc1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880516180 DD On-Demand Mild ADRB2 18 54 N#Cc1ccccc1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880516180 DD On-Demand Mild ADRB1 60 43 N#Cc1ccccc1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880516180 DD On-Demand Mild CASR 42 43 N#Cc1ccccc1OC[C@@H](O)CN[C@@H]1CCC[C@]12CCCO2 ZINC000880516180 DD On-Demand Mild CYP2D6 17 44 O=C(CC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2)NCc1cc(O)nc(S)n1 ZINC000880516189 ED On-Demand Anodyne BOTA 31 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880516205 GD On-Demand Anodyne P2RX7 54 57 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880516207 GD On-Demand Anodyne P2RX7 54 57 O=C(CCCOc1ccccc1)NCc1cc(O)nc(S)n1 ZINC000880516209 DD On-Demand Anodyne SUCNR1 43 36 CS(=O)(=O)c1ccc(NC(=O)NC2(Cc3ccccc3)CCC2)nc1 ZINC000880516230 FF On-Demand Anodyne SLC12A5 28 40 COCCNC(=O)c1ccccc1NC(=O)/C=C\c1cccnc1 ZINC000880516232 EE On-Demand Anodyne MMP2 15 45 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)nc1 ZINC000880516248 FG On-Demand Anodyne NPY5R 26 42 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)nc1 ZINC000880516248 FG On-Demand Anodyne EPHX2 23 46 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)nc1 ZINC000880516248 FG On-Demand Anodyne SFRP1 63 31 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)nc1 ZINC000880516248 FG On-Demand Anodyne WNT3 56 31 CS(=O)(=O)c1ccc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)nc1 ZINC000880516248 FG On-Demand Anodyne MAP3K12 28 40 CC(=O)N1CCc2ccccc2[C@@H]1CC(=O)NCc1cc(O)nc(S)n1 ZINC000880516253 FD On-Demand Anodyne MTNR1B 15 48 CCCCCOc1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880516266 EF On-Demand Anodyne PLA2G4A 24 42 CCCCCOc1ccc(C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880516266 EF On-Demand Anodyne PLA2G4B 96 42 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OC1CCC1 ZINC000880516271 EE On-Demand Anodyne HCN1 51 33 O=C(NCc1cc(O)nc(S)n1)c1ccccc1OC1CCC1 ZINC000880516271 EE On-Demand Anodyne HCN4 49 33 Cc1ccc(-n2nc(C(=O)NCc3cc(O)nc(S)n3)c3c2CCC3)c(F)c1 ZINC000880516301 GF On-Demand Anodyne CNR1 41 36 Cc1nc(CC(C)C)sc1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516302 EE On-Demand Anodyne SCD1 25 41 C[C@@H](Oc1ccccc1C(F)(F)F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516306 FF On-Demand Anodyne CARM1 42 36 CC(C)(C)C(=O)N1CCC[C@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516334 ED On-Demand Anodyne F2 51 46 CC(C)(C)C(=O)N1CCC[C@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516334 ED On-Demand Anodyne TRY1_BOVIN 46 38 CC(C)(C)C(=O)N1CCC[C@@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516335 ED On-Demand Anodyne F2 51 46 CC(C)(C)C(=O)N1CCC[C@@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516335 ED On-Demand Anodyne TRY1_BOVIN 46 38 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516339 FC On-Demand Anodyne DRD4 50 43 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516339 FC On-Demand Anodyne ACHE 36 45 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516339 FC On-Demand Anodyne DRD3 15 42 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516339 FC On-Demand Anodyne SIGMAR1 45 42 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516339 FC On-Demand Anodyne NPFFR1 43 36 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000880516353 DC On-Demand Anodyne INHA 22 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(C2CC2)C1 ZINC000880516354 DC On-Demand Anodyne INHA 22 42 CCCCSCC(=O)NCc1cc(O)nc(S)n1 ZINC000880516376 CD On-Demand Anodyne EST1_PIG 40 34 Cc1ccc(C(=O)N2CCC[C@H](C(=O)NCc3cc(O)nc(S)n3)C2)cc1 ZINC000880516411 GD On-Demand Anodyne EPHX2 15 42 Cc1ccc(C(=O)N2CCC[C@H](C(=O)NCc3cc(O)nc(S)n3)C2)cc1 ZINC000880516411 GD On-Demand Anodyne L3MBTL3 40 34 Cc1ccc(C(=O)N2CCC[C@H](C(=O)NCc3cc(O)nc(S)n3)C2)cc1 ZINC000880516411 GD On-Demand Anodyne MAP3K12 32 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne F2 72 43 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne TRY1_BOVIN 72 41 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne DPP4 18 44 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne PREP 101 48 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne XIAP 34 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880516416 FD On-Demand Anodyne TMPRSS11D 71 39 CCOc1ccccc1OCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880516457 FE On-Demand Anodyne HTR7 15 40 CCOc1ccccc1OCCCC(=O)NCc1cc(O)nc(S)n1 ZINC000880516457 FE On-Demand Anodyne SUCNR1 45 34 C=CCN1CCC(NC(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880516462 ED On-Demand Mild TGM2 39 42 O[C@@]1(CN[C@@H]2CCC[C@]23CCCO3)CCN(Cc2ccccc2)C1 ZINC000880516463 EE On-Demand Anodyne SIGMAR1 42 39 O=C(CCCCc1nc2ccccc2s1)NCc1cc(O)nc(S)n1 ZINC000880516467 FG On-Demand Anodyne SUCNR1 40 35 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880516514 FD On-Demand Anodyne PDE8B 41 33 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880516516 FD On-Demand Anodyne PDE8B 41 33 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC ZINC000880516521 ED On-Demand Anodyne HCRTR1 15 41 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC ZINC000880516521 ED On-Demand Anodyne TRPV1 17 48 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC ZINC000880516521 ED On-Demand Anodyne MT-ND1 23 41 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC ZINC000880516521 ED On-Demand Anodyne ENPP1 67 32 COc1ccc(CC(=O)NCc2cc(O)nc(S)n2)cc1OC ZINC000880516521 ED On-Demand Anodyne DRTS_TRYCR 46 33 CCc1ccc([C@H](C)C(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880516526 DE On-Demand Anodyne TRPV1 93 37 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516538 FD On-Demand Anodyne SLC6A1 55 33 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516538 FD On-Demand Anodyne NMT1 18 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516538 FD On-Demand Anodyne PREP 32 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516538 FD On-Demand Anodyne L3MBTL3 40 33 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516538 FD On-Demand Anodyne MAP3K12 34 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516540 FD On-Demand Anodyne SLC6A1 55 33 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516540 FD On-Demand Anodyne NMT1 18 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516540 FD On-Demand Anodyne PREP 32 42 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516540 FD On-Demand Anodyne L3MBTL3 40 33 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880516540 FD On-Demand Anodyne MAP3K12 34 42 CCN1CCCC[C@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516546 CC On-Demand Anodyne P2RX7 19 48 CCN1CCCC[C@@H]1C(=O)NCc1cc(O)nc(S)n1 ZINC000880516548 CC On-Demand Anodyne P2RX7 19 48 COCCNC(=O)c1ccccc1NC(=O)CCC(=O)OC ZINC000880516553 DC On-Demand Anodyne HCAR2 33 40 COCCNC(=O)c1ccccc1NC(=O)CCC(=O)OC ZINC000880516553 DC On-Demand Anodyne FAS 27 40 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CCCN1Cc1ccc(F)cc1 ZINC000880516562 FD On-Demand Anodyne P2RX7 27 48 O=C(NCc1cc(O)nc(S)n1)[C@H]1CCCN1Cc1ccc(F)cc1 ZINC000880516563 FD On-Demand Anodyne P2RX7 27 48 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516571 FC On-Demand Anodyne HTR1A 23 45 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516571 FC On-Demand Anodyne DRD2 19 45 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516571 FC On-Demand Anodyne DRD4 36 42 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516571 FC On-Demand Anodyne HTR7 25 43 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc(O)nc(S)n1 ZINC000880516571 FC On-Demand Anodyne SLC27A1 65 52 C[C@H](Cc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516580 DE On-Demand Anodyne TRPV1 78 35 C[C@H](Cc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516580 DE On-Demand Anodyne CARM1 27 40 C[C@@H](Cc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516581 DE On-Demand Anodyne TRPV1 78 35 C[C@@H](Cc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516581 DE On-Demand Anodyne CARM1 27 40 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)Nc1nccs1 ZINC000880516584 CE On-Demand Anodyne MAP1 92 37 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)nc1 ZINC000880516591 FG On-Demand Anodyne F10 30 41 CS(=O)(=O)c1ccc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)nc1 ZINC000880516592 FG On-Demand Anodyne F10 30 41 O=C(NCc1cc(O)nc(S)n1)c1ccc(OC2CCC2)cc1 ZINC000880516604 EE On-Demand Anodyne TNKS 41 32 COC(=O)c1ccc(CNC(=O)[C@@H](C)N[C@@H]2CCC[C@]23CCCO3)cc1 ZINC000880516605 FE On-Demand Anodyne PROC 55 31 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne CHRM2 21 43 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne CHRM1 15 43 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne DRD2 16 46 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne DRD4 38 47 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne ACHE 35 47 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne CHRM3 25 43 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne SIGMAR1 54 49 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne SSTR5 51 38 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne CCR3 22 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne C3AR1 40 38 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne MCHR1 43 45 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne CACNA1G 15 46 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NC1CCN(Cc2ccccc2)CC1 ZINC000880516618 GF On-Demand Anodyne BIRC2 46 42 O=C(NCc1cc(O)nc(S)n1)[C@@H]1COc2ccccc2C1 ZINC000880516638 DD On-Demand Anodyne ROCK2 28 44 O=C(NCc1cc(O)nc(S)n1)[C@H]1COc2ccccc2C1 ZINC000880516639 DD On-Demand Anodyne ROCK2 28 44 COc1cc(C(=O)NCc2cc(O)nc(S)n2)ccc1OC(C)C ZINC000880516661 EE On-Demand Anodyne SLC5A7 33 40 CN(C)[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516695 ED On-Demand Anodyne MME 78 40 CN(C)[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516695 ED On-Demand Anodyne ANPEP 20 40 CN(C)[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516695 ED On-Demand Anodyne AMP1_PLAFQ 42 38 CN(C)[C@@H](Cc1ccccc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516695 ED On-Demand Anodyne GPR142 69 34 O=C(NCc1cc(O)nc(S)n1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880516698 EC On-Demand Anodyne INHA 25 47 O=C(NCc1cc(O)nc(S)n1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880516699 EC On-Demand Anodyne INHA 25 47 O=C(CCCCCc1cccs1)NCc1cc(O)nc(S)n1 ZINC000880516704 EF On-Demand Anodyne SUCNR1 50 35 O=C(CC12CC3CC(CC(C3)C1)C2)NCc1cc(O)nc(S)n1 ZINC000880516724 EF On-Demand Anodyne BOTA 32 44 O=C(NCc1cc(O)nc(S)n1)c1cccc(CN2CCOCC2)c1 ZINC000880516730 FD On-Demand Anodyne CHRM3 19 46 COc1ccc(OCCCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880516731 ED On-Demand Anodyne MTNR1A 63 37 COc1ccc(OCCCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880516731 ED On-Demand Anodyne MTNR1B 51 37 O=C(CCc1ccc2c(c1)OCCO2)NCc1cc(O)nc(S)n1 ZINC000880516739 ED On-Demand Anodyne NOS2 81 33 O=C(CCc1ccc2c(c1)OCCO2)NCc1cc(O)nc(S)n1 ZINC000880516739 ED On-Demand Anodyne LUXR 31 44 CC(=O)N1CCc2cc(C(=O)NCc3cc(O)nc(S)n3)ccc21 ZINC000880516741 ED On-Demand Anodyne HSD17B3 43 29 C[C@@H](CCc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516759 EE On-Demand Anodyne TRPV1 68 34 C[C@H](CCc1ccccc1F)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516760 EE On-Demand Anodyne TRPV1 68 34 O=C(NCc1cc(O)nc(S)n1)c1ccccc1CN1CCOCC1 ZINC000880516788 FD On-Demand Anodyne SLC6A5 48 41 C[C@@H](N[C@@H]1CCC[C@]12CCCO2)C(=O)NCCc1ccc2c(c1)OCCO2 ZINC000880516794 FE On-Demand Anodyne NOS2 60 40 CCNc1nc(C)c(C(=O)NCc2cc(O)nc(S)n2)s1 ZINC000880516803 ED On-Demand Anodyne SCD1 25 46 CCNc1nc(C)c(C(=O)NCc2cc(O)nc(S)n2)s1 ZINC000880516803 ED On-Demand Anodyne SCD 23 40 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516814 FF On-Demand Anodyne PPARA 19 42 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516814 FF On-Demand Anodyne TRPV1 74 38 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516814 FF On-Demand Anodyne PPARD 25 41 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NCc1cc(O)nc(S)n1 ZINC000880516814 FF On-Demand Anodyne ACE2 48 40 Cc1cccc2c1CCN(C(=O)Nc1ccc(S(C)(=O)=O)cn1)C2 ZINC000880516820 EE On-Demand Anodyne P2RY14 44 33 CCCN(CCC)C(=O)c1cccc(C(=O)NCc2cc(O)nc(S)n2)c1 ZINC000880516835 GF On-Demand Anodyne TSPO 15 41 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne HTR1A 52 40 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne DRD2 40 41 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne DRD4 22 45 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne DRD3 47 38 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne HRH3 24 45 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne SIGMAR1 25 43 COc1ccccc1-c1nc(CN(C)CCCCN2CCCCC2)co1 ZINC000880516863 FI On-Demand Anodyne CHRNA7 16 46 Cc1ccc(N2CCCN(C(=O)Nc3ccc(S(C)(=O)=O)cn3)CC2)cc1 ZINC000880516894 GF On-Demand Anodyne SLC6A9 22 41 CC(C)n1nccc1CN(C)CCCCN1CCCCC1 ZINC000880516896 CG On-Demand Anodyne SIGMAR1 19 42 CC(C)n1nccc1CN(C)CCCCN1CCCCC1 ZINC000880516896 CG On-Demand Anodyne HNMT 54 38 Cc1ccc(OC[C@@H](C)NC(=O)Nc2ccc(S(C)(=O)=O)cn2)cc1 ZINC000880516918 FE On-Demand Anodyne GCK 32 47 Cc1ccc(OC[C@H](C)NC(=O)Nc2ccc(S(C)(=O)=O)cn2)cc1 ZINC000880516919 FE On-Demand Anodyne GCK 32 47 Cc1cccc(C(=O)NNC(=O)CN(C)CCCCN2CCCCC2)c1 ZINC000880516920 FD On-Demand Reactive DRD4 42 34 Cc1cccc(C(=O)NNC(=O)CN(C)CCCCN2CCCCC2)c1 ZINC000880516920 FD On-Demand Reactive DRD3 17 40 Cc1cccc(C(=O)NNC(=O)CN(C)CCCCN2CCCCC2)c1 ZINC000880516920 FD On-Demand Reactive HRH3 18 40 Cc1cccc(C(=O)NNC(=O)CN(C)CCCCN2CCCCC2)c1 ZINC000880516920 FD On-Demand Reactive KCNK3 51 36 Cc1cccc(C(=O)NNC(=O)CN(C)CCCCN2CCCCC2)c1 ZINC000880516920 FD On-Demand Reactive KCNK9 41 36 O=C(CCCc1cccs1)NCc1cc(O)nc(S)n1 ZINC000880516921 DE On-Demand Anodyne SUCNR1 53 36 Cc1nn(C)c2ncc(CN(C)CCCCN3CCCCC3)cc12 ZINC000880516943 EF On-Demand Anodyne SIGMAR1 18 42 Cc1nn(C)c2ncc(CN(C)CCCCN3CCCCC3)cc12 ZINC000880516943 EF On-Demand Anodyne HNMT 47 34 Cc1conc1CN(C)CCCCN1CCCCC1 ZINC000880516957 CF On-Demand Anodyne SIGMAR1 17 41 Cc1cc(O)nc(CN(C)CCCCN2CCCCC2)n1 ZINC000880517001 CE On-Demand Anodyne SIGMAR1 20 46 CNc1nc(C(=O)N2CCC(Cc3nc(C(C)C)n[nH]3)CC2)cs1 ZINC000880517032 EF On-Demand Anodyne TRPC6 56 42 CNc1nc(C(=O)N2CCC(Cc3nc(C(C)C)n[nH]3)CC2)cs1 ZINC000880517032 EF On-Demand Anodyne TRPC3 49 42 N#Cc1ccnc(N2CCN(C(=O)c3cc(S(=O)(=O)NC4CC4)ccc3Br)CC2)c1 ZINC000880517041 JE On-Demand Mild SLC6A9 19 40 COC(=O)c1ccc2c(c1)CCN2C(=O)c1cnc2ccccc2c1C(F)(F)F ZINC000880517044 HI On-Demand Anodyne EIF2AK3 49 34 Cc1cnc(CN(C)CCCCN2CCCCC2)cn1 ZINC000880517051 CE On-Demand Anodyne HRH3 43 41 Cc1cnc(CN(C)CCCCN2CCCCC2)cn1 ZINC000880517051 CE On-Demand Anodyne SIGMAR1 18 44 Cc1cnc(CN(C)CCCCN2CCCCC2)cn1 ZINC000880517051 CE On-Demand Anodyne HNMT 60 38 CN(Cc1ccc(N(C)C)cc1)C(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517055 GF On-Demand Clean PLA2G7 44 38 O=C(/C=C/c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517067 DI On-Demand Mild HDAC8 24 46 O=C(/C=C/c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517067 DI On-Demand Mild MMP2 15 51 O=C(/C=C/c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517067 DI On-Demand Mild HDAC6 16 46 O=C(/C=C/c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517067 DI On-Demand Mild MMP9 15 51 O=C(/C=C\c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517068 DI On-Demand Mild HDAC8 24 46 O=C(/C=C\c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517068 DI On-Demand Mild MMP2 15 51 O=C(/C=C\c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517068 DI On-Demand Mild HDAC6 16 46 O=C(/C=C\c1cccnc1)Nc1cccc(C#Cc2ccccc2)c1 ZINC000880517068 DI On-Demand Mild MMP9 15 51 COC(=O)c1ccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880517082 EG On-Demand Anodyne SLC6A3 24 42 COC(=O)c1ccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880517082 EG On-Demand Anodyne PANC 45 43 Cc1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517088 CH On-Demand Anodyne KCNH2 21 45 C#CCOCCN(C)CCCCN1CCCCC1 ZINC000880517145 CD On-Demand Mild HRH3 21 41 CN1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880517161 CC On-Demand Anodyne NPY5R 27 43 CN1CCN(C(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880517161 CC On-Demand Anodyne TGM2 20 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(O)nc(S)n1)C2 ZINC000880517184 ED On-Demand Anodyne MTNR1A 36 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(O)nc(S)n1)C2 ZINC000880517184 ED On-Demand Anodyne MTNR1B 33 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(O)nc(S)n1)C2 ZINC000880517184 ED On-Demand Anodyne FAAH 15 42 COC(=O)[C@@H](c1ccc(C#N)cc1)N(C)CCCCN1CCCCC1 ZINC000880517188 EF On-Demand Mild HRH3 32 51 Cc1c(NC(=O)Cc2ccc3cccnc3c2)c(=O)n(C2CCCCC2)n1C ZINC000880517194 GH On-Demand Anodyne CDK5 16 42 CC(C)(C)N1CCC(NC(=O)Nc2ccc(S(C)(=O)=O)cn2)CC1 ZINC000880517212 FD On-Demand Anodyne EPHX2 41 42 CON(C)C(=O)CCN(C)CCCCN1CCCCC1 ZINC000880517227 CD On-Demand Anodyne HRH3 18 41 Cc1cnc(CN(C)CCCCN2CCCCC2)s1 ZINC000880517242 CG On-Demand Anodyne HRH3 44 44 Cc1cnc(CN(C)CCCCN2CCCCC2)s1 ZINC000880517242 CG On-Demand Anodyne SIGMAR1 20 41 Cc1cnc(CN(C)CCCCN2CCCCC2)s1 ZINC000880517242 CG On-Demand Anodyne HNMT 51 37 COC(=O)C1CCN(C(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)CC1 ZINC000880517278 FD On-Demand Anodyne PTR1 44 33 CN(CCF)CCCCN1CCCCC1 ZINC000880517356 BE On-Demand Anodyne HRH3 16 50 CCOc1ccc(OCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880517357 ED On-Demand Anodyne MTNR1A 21 40 CCN1CC[C@H](CNC(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880517368 EC On-Demand Anodyne CCR3 17 41 CCN1CC[C@H](CNC(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880517368 EC On-Demand Anodyne CACNA1I 41 32 CCN1CC[C@H](CNC(=O)Nc2ccc(S(C)(=O)=O)cn2)C1 ZINC000880517368 EC On-Demand Anodyne NAMPT 40 43 COc1ccc(OC)c([C@H](O)CN(C)CCCCN2CCCCC2)c1 ZINC000880517401 FF On-Demand Anodyne HRH3 45 45 COc1ccc(OC)c([C@H](O)CN(C)CCCCN2CCCCC2)c1 ZINC000880517401 FF On-Demand Anodyne SIGMAR1 26 47 COc1ccc(OC)c([C@H](O)CN(C)CCCCN2CCCCC2)c1 ZINC000880517401 FF On-Demand Anodyne EBP 53 47 C[C@H]1CCc2[nH]c3ccc(C(=O)NCc4cc(O)nc(S)n4)cc3c2C1 ZINC000880517403 FG On-Demand Anodyne TTK 44 32 Cc1c(CN(C)CCCCN2CCCCC2)cnn1C ZINC000880517429 CE On-Demand Anodyne SIGMAR1 16 42 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517437 GE On-Demand Anodyne OPRM1 47 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517437 GE On-Demand Anodyne OPRD1 40 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517437 GE On-Demand Anodyne CMA1 44 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517437 GE On-Demand Anodyne CTSL 15 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517438 GE On-Demand Anodyne OPRM1 47 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517438 GE On-Demand Anodyne OPRD1 40 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517438 GE On-Demand Anodyne CMA1 44 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517438 GE On-Demand Anodyne CTSL 15 41 CCCCCNC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517448 DE On-Demand Anodyne ASAH1 78 34 Cc1cc(OCC(=O)NCc2cc(O)nc(S)n2)ccc1C(C)C ZINC000880517457 EF On-Demand Anodyne THRA 48 40 Cc1cc(OCC(=O)NCc2cc(O)nc(S)n2)ccc1C(C)C ZINC000880517457 EF On-Demand Anodyne THRB 46 40 Cc1oc(-c2ccccc2)nc1CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517464 FI On-Demand Anodyne PPARG 43 35 Cc1oc(-c2ccccc2)nc1CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517464 FI On-Demand Anodyne PPARA 44 38 Cc1oc(-c2ccccc2)nc1CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517464 FI On-Demand Anodyne PDE8B 74 44 CS(=O)(=O)c1ccc(NC(=O)NCC2CCCCCCC2)nc1 ZINC000880517554 EF On-Demand Anodyne GCK 30 44 O=C(CC[C@H]1CCc2ccccc21)NCc1cc(O)nc(S)n1 ZINC000880517560 EF On-Demand Anodyne NQO2 17 40 O=C(CC[C@H]1CCc2ccccc21)NCc1cc(O)nc(S)n1 ZINC000880517560 EF On-Demand Anodyne MTNR1A 16 42 O=C(CC[C@@H]1CCc2ccccc21)NCc1cc(O)nc(S)n1 ZINC000880517561 EF On-Demand Anodyne NQO2 17 40 O=C(CC[C@@H]1CCc2ccccc21)NCc1cc(O)nc(S)n1 ZINC000880517561 EF On-Demand Anodyne MTNR1A 16 42 O=C(Cc1ccc2c(c1)OCCO2)NCc1cc(O)nc(S)n1 ZINC000880517564 ED On-Demand Anodyne NOS2 90 34 CC(=O)Nc1ccc2c(CN(C)CCCCN3CCCCC3)cc(=O)oc2c1 ZINC000880517593 GG On-Demand Anodyne CHRNA7 20 43 C[C@H](C(=O)Nc1cccnc1Cl)N(C)CCCCN1CCCCC1 ZINC000880517612 FG On-Demand Anodyne KCNQ2 42 34 C[C@H](C(=O)Nc1cccnc1Cl)N(C)CCCCN1CCCCC1 ZINC000880517612 FG On-Demand Anodyne CHRNA7 18 40 C[C@H](C(=O)Nc1cccnc1Cl)N(C)CCCCN1CCCCC1 ZINC000880517612 FG On-Demand Anodyne HNMT 81 37 C[C@H](C(=O)Nc1cccnc1Cl)N(C)CCCCN1CCCCC1 ZINC000880517612 FG On-Demand Anodyne G2YM83_BOTF4 60 34 CCCOc1ccc(OCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880517618 ED On-Demand Anodyne MTNR1A 29 42 CCCOc1ccc(OCC(=O)NCc2cc(O)nc(S)n2)cc1 ZINC000880517618 ED On-Demand Anodyne PLA2G4B 80 33 Cc1c(NC(=O)[C@@H](F)c2ccccc2)c(=O)n(C2CCCCC2)n1C ZINC000880517636 EH On-Demand Anodyne KCNQ2 19 44 Cc1c(NC(=O)[C@H](F)c2ccccc2)c(=O)n(C2CCCCC2)n1C ZINC000880517638 EH On-Demand Anodyne KCNQ2 19 44 CN(Cc1ccc(F)cc1)C(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517649 FF On-Demand Anodyne PLA2G7 87 47 CS(=O)(=O)c1ccc(NC(=O)NC2CCN(CC3CCCCC3)CC2)nc1 ZINC000880517756 GF On-Demand Anodyne SSTR5 40 37 CS(=O)(=O)c1ccc(NC(=O)NC2CCN(CC3CCCCC3)CC2)nc1 ZINC000880517756 GF On-Demand Anodyne EPHX2 43 42 CS(=O)(=O)c1ccc(NC(=O)NC2CCN(CC3CCCCC3)CC2)nc1 ZINC000880517756 GF On-Demand Anodyne CXCR3 15 41 CS(=O)(=O)c1ccc(NC(=O)NC2CCN(CC3CCCCC3)CC2)nc1 ZINC000880517756 GF On-Demand Anodyne GCK 21 41 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1c(C)n(C)n(C2CCCCC2)c1=O ZINC000880517768 GF On-Demand Anodyne CAPN1 35 40 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1c(C)n(C)n(C2CCCCC2)c1=O ZINC000880517768 GF On-Demand Anodyne CAPN2 42 34 CO[C@@H]1CC[C@@H](N(C)CCCCN2CCCCC2)C1 ZINC000880517851 CF On-Demand Anodyne HRH3 22 43 CS(=O)(=O)c1ccc(NC(=O)NC2CCCCCCC2)nc1 ZINC000880517878 EF On-Demand Anodyne EPHX2 47 47 CS(=O)(=O)c1ccc(NC(=O)NC2CCCCCCC2)nc1 ZINC000880517878 EF On-Demand Anodyne GCK 20 40 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne ACHE 19 45 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne LTA4H 39 40 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne HRH3 90 53 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne SIGMAR1 36 49 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne EBP 42 42 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne HNMT 81 37 COc1ccc(CN(C)CCCCN2CCCCC2)nc1 ZINC000880517881 CF On-Demand Anodyne PSMB1 40 36 COC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517905 EG On-Demand Anodyne SLC6A3 31 41 COC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517905 EG On-Demand Anodyne KCNH2 39 42 COC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517905 EG On-Demand Anodyne ACHP_LYMST 18 40 COC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517905 EG On-Demand Anodyne PANC 41 34 COC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517905 EG On-Demand Anodyne Q8WSF8_APLCA 32 40 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne ACHE 29 43 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne SLC6A1 33 40 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne HRH1 19 42 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne HTR4 20 44 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne HRH3 55 48 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne SIGMAR1 45 44 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne BCHE 35 42 Cc1nc(CN(C)CCCCN2CCCCC2)nc2ccccc12 ZINC000880517917 EH On-Demand Anodyne HNMT 104 48 CC(=O)c1cccc(OC[C@@H](O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517922 GF On-Demand Anodyne ABCB1 18 46 CC(=O)c1cccc(OC[C@H](O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880517923 GF On-Demand Anodyne ABCB1 18 46 C[C@H](NC(=O)[C@@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880517934 FG On-Demand Anodyne XIAP 42 35 C[C@H](NC(=O)[C@@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880517934 FG On-Demand Anodyne BIRC8 48 34 Cc1ccccc1CNC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880517980 FF On-Demand Anodyne P2RX7 24 43 CC(=O)c1ccccc1OCCN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518001 FG On-Demand Anodyne HCN1 43 34 COC(=O)c1sccc1NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518013 GF On-Demand Anodyne FAS 39 46 Cc1c(NC(=O)COc2cccnc2)c(=O)n(C2CCCCC2)n1C ZINC000880518074 EE On-Demand Anodyne VCP 50 34 O=C(/C=C/c1ccc2c(c1)OCO2)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880518202 FH On-Demand Mild DYRK2 47 38 O=C(/C=C\c1ccc2c(c1)OCO2)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880518206 FH On-Demand Mild DYRK2 47 38 COc1ccc(NC(=O)[C@H](C)N2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1OC ZINC000880518305 GG On-Demand Anodyne ENPP1 69 33 Cc1c(NC(=O)COc2cccc(C#N)c2)c(=O)n(C2CCCCC2)n1C ZINC000880518317 FF On-Demand Mild ADORA2A 16 43 Cc1c(NC(=O)COc2cccc(C#N)c2)c(=O)n(C2CCCCC2)n1C ZINC000880518317 FF On-Demand Mild CHRNA10 25 43 Cc1c(NC(=O)COc2cccc(C#N)c2)c(=O)n(C2CCCCC2)n1C ZINC000880518317 FF On-Demand Mild PFKFB3 53 31 COC(=O)[C@@H](c1cccnc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518460 EE On-Demand Anodyne GLRA1 19 40 C[C@@H](C(=O)N1CCC[C@H]1c1cccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518530 GH On-Demand Anodyne ADAM17 16 41 C[C@@H](C(=O)N1CCC[C@@H]1c1cccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518531 GH On-Demand Anodyne ADAM17 16 41 C[C@H](C(=O)N1CCC[C@H]1c1cccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518532 GH On-Demand Anodyne ADAM17 16 41 C[C@H](C(=O)N1CCC[C@@H]1c1cccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518533 GH On-Demand Anodyne ADAM17 16 41 Cc1ccccc1CC(=O)NNC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518619 GD On-Demand Reactive TK 17 40 COC(=O)N[C@H](CC(C)C)C(=O)Nc1c(C)n(C)n(C2CCCCC2)c1=O ZINC000880518659 GF On-Demand Anodyne CAPN1 35 40 COC(=O)N[C@H](CC(C)C)C(=O)Nc1c(C)n(C)n(C2CCCCC2)c1=O ZINC000880518659 GF On-Demand Anodyne CAPN2 42 34 COC(=O)[C@@H](c1ccccc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518665 EG On-Demand Anodyne SLC6A3 41 39 COC(=O)[C@@H](c1ccccc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518665 EG On-Demand Anodyne GLRA1 40 31 COC(=O)[C@@H](c1ccc(F)cc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518722 FG On-Demand Anodyne SLC6A3 38 40 COc1cccc(OCCN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880518756 EG On-Demand Anodyne CHRNA10 22 41 CCOc1ccccc1NC(=O)CCN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518853 GH On-Demand Anodyne HCN1 44 35 CCOc1ccccc1NC(=O)CCN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518853 GH On-Demand Anodyne HCN4 42 35 C[C@@H](C(=O)Nc1nccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518958 EF On-Demand Anodyne MAP1 72 34 C[C@H](C(=O)Nc1nccs1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880518960 EF On-Demand Anodyne MAP1 72 34 C[C@H](CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880519035 DH On-Demand Anodyne SLC6A3 15 52 C[C@H](CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880519035 DH On-Demand Anodyne SLC18A3 16 52 COC(=O)c1cccc(NC(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880519121 GF On-Demand Anodyne KCNH2 34 46 CCOc1ccccc1NC(=O)[C@@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519179 GH On-Demand Anodyne HCN1 50 34 CCOc1ccccc1NC(=O)[C@@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519179 GH On-Demand Anodyne HCN4 43 34 CCOc1ccccc1NC(=O)[C@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519184 GH On-Demand Anodyne HCN1 50 34 CCOc1ccccc1NC(=O)[C@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519184 GH On-Demand Anodyne HCN4 43 34 CCCCCNC(=O)[C@@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519223 EF On-Demand Anodyne ASAH1 74 34 CCCCCNC(=O)[C@H](C)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519225 EF On-Demand Anodyne ASAH1 74 34 CNC(=O)[C@@H](NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880519228 GD On-Demand Anodyne XIAP 45 33 CNC(=O)[C@@H](NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880519228 GD On-Demand Anodyne BIRC8 44 30 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519251 GG On-Demand Anodyne PLA2G7 49 36 COc1ccc(CN(C)C(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880519438 GF On-Demand Anodyne PLA2G7 44 38 C[C@H](C(=O)Nc1cccc(C#N)c1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519473 FG On-Demand Mild CCR3 17 41 C[C@H](C(=O)Nc1cccc(C#N)c1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519473 FG On-Demand Mild ITGA4 46 31 Cc1c(NC(=O)C(=O)NCCCc2ccccc2)c(=O)n(C2CCCCC2)n1C ZINC000880519491 GF On-Demand Anodyne FKBP1A 33 40 Cc1c(NC(=O)C(=O)NCCCc2ccccc2)c(=O)n(C2CCCCC2)n1C ZINC000880519491 GF On-Demand Anodyne PREP 41 34 C[C@H](C(=O)Nc1cccnc1Cl)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519591 FG On-Demand Anodyne G2YM83_BOTF4 57 33 CSc1ccc(CN(C)C(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880519594 GH On-Demand Anodyne PLA2G7 61 40 CC(=O)c1cccc(NC(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880519621 FF On-Demand Anodyne KCNH2 34 46 CC(=O)c1cccc(NC(=O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880519621 FF On-Demand Anodyne CCR3 19 45 C[C@H](C(=O)Nc1ccccc1[N+](=O)[O-])N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519664 GG On-Demand Bother COLA 42 32 C[C@@H](c1ccc(F)cc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519743 DI On-Demand Anodyne SLC6A3 27 42 C#CCN1CCC[C@H]1C(=O)Nc1c(C)n(C)n(C2CCCCC2)c1=O ZINC000880519810 EE On-Demand Mild HSD11B1 40 31 COc1ccc2c(CN3[C@H]4CC[C@H]3CC(c3cnn(C)c3)C4)cc(=O)oc2c1 ZINC000880519837 GG On-Demand Anodyne CYP11B1 17 42 C[C@H](c1nc(-c2cccs2)no1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519930 FI On-Demand Anodyne ETHR 24 40 C[C@H](C(=O)Nc1ccccc1Cl)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519960 FH On-Demand Anodyne EPHB3 56 37 COC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880519963 CD On-Demand Anodyne SLC6A3 23 42 CC(=O)Nc1ccc(OC[C@@H](O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880519964 GF On-Demand Anodyne ADRB1 25 44 CC(=O)Nc1ccc(OC[C@H](O)CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)cc1 ZINC000880519965 GF On-Demand Anodyne ADRB1 25 44 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Cl)c(S(=O)(=O)N2CCOCC2)c1 ZINC000880519995 JG On-Demand Mild CPT1A 46 36 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Cl)c(S(=O)(=O)N2CCOCC2)c1 ZINC000880519995 JG On-Demand Mild GRM4 52 38 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Cl)c(S(=O)(=O)N2CCOCC2)c1 ZINC000880519995 JG On-Demand Mild DDR1 40 37 CN(C)C(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880520044 FG On-Demand Anodyne KCNH2 34 41 C[C@H](C(=O)N(C)Cc1ccccc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880520064 FG On-Demand Anodyne TACR1 22 43 C[C@@H](C(=O)N(C)Cc1ccccc1)N1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880520065 FG On-Demand Anodyne TACR1 22 43 COC(=O)CCCCN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880520104 DE On-Demand Anodyne SLC6A3 22 42 CO[C@@H](Cc1ccccc1)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880520264 EG On-Demand Anodyne SLC6A3 15 44 CO[C@@H](Cc1ccccc1)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2 ZINC000880520264 EG On-Demand Anodyne SLC18A3 15 44 CO[C@@H](CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccc(F)cc1 ZINC000880520323 EH On-Demand Anodyne SLC6A3 35 42 C[C@@H](NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880520336 FG On-Demand Anodyne PRCP 17 48 C[C@@H](NC(=O)CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880520336 FG On-Demand Anodyne BIRC8 45 32 CC(=O)c1cccc(CN2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)c1 ZINC000880520357 DH On-Demand Anodyne KCNH2 38 42 CO[C@@H](CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880520465 EH On-Demand Anodyne SLC6A3 31 50 CO[C@@H](CN1[C@H]2CC[C@H]1CC(c1cnn(C)c1)C2)c1ccccc1 ZINC000880520465 EH On-Demand Anodyne SLC18A3 15 50 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)ccc1F ZINC000880520548 JH On-Demand Mild CPT1A 45 32 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)ccc1F ZINC000880520548 JH On-Demand Mild KCNK3 64 36 COc1ccc([C@@H](NC(=O)CN2C[C@@H](O)CC[C@H]2C)C(C)C)cc1 ZINC000880520775 EE On-Demand Anodyne EDNRB 27 47 COC(=O)c1ccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880520828 DD On-Demand Anodyne ADRB2 17 41 Cc1c(NC(=O)[C@H]2CC(=O)N(C3CCCC3)C2)c(=O)n(C2CCCCC2)n1C ZINC000880520855 GF On-Demand Anodyne INHA 24 53 Cc1c(NC(=O)[C@@H]2CC(=O)N(C3CCCC3)C2)c(=O)n(C2CCCCC2)n1C ZINC000880520856 GF On-Demand Anodyne INHA 24 53 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)c1 ZINC000880520861 DD On-Demand Anodyne ACOX1 55 32 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)c1 ZINC000880520861 DD On-Demand Anodyne ABCB1 33 53 C[C@@H](NC(=O)CN1C[C@@H](O)CC[C@H]1C)c1ccc(Cl)cc1 ZINC000880520872 DE On-Demand Anodyne PRCP 25 48 CC(=O)c1cccc(OCC(=O)Nc2c(C)n(C)n(C3CCCCC3)c2=O)c1 ZINC000880520922 GG On-Demand Anodyne ADORA2B 30 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne ACE 80 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne OPRM1 60 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne OPRD1 53 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne MME 102 37 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CMA1 74 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CTRA_BOVIN 56 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne FCER2 50 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne PAPA1_CARPA 44 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CYSP_TRYCR 56 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CTSL 42 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne NPFFR2 61 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne TIMP3 62 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CAPNS1 68 31 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne HLA-DRB1 53 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CAPN1 66 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne CTRC 46 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne ACE2 72 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne FPR1 57 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne BLA1_STEMA 55 37 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne QRFPR 45 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne BRCA1 50 30 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520924 DD On-Demand Anodyne NPFFR1 63 35 CCOC(=O)C1=C(CN2C[C@@H](O)CC[C@H]2C)NC(=O)N[C@@H]1c1ccccc1 ZINC000880520932 FD On-Demand Anodyne SLC27A4 75 35 CCOC(=O)C1=C(CN2C[C@@H](O)CC[C@H]2C)NC(=O)N[C@H]1c1ccccc1 ZINC000880520933 FD On-Demand Anodyne SLC27A4 75 35 Cc1cc(NC(=O)NC[C@H]2CC(C)(C)CO2)ncc1C#N ZINC000880520953 CE On-Demand Mild CSNK2A1 44 34 Cc1cc(NC(=O)NC[C@@H]2CC(C)(C)CO2)ncc1C#N ZINC000880520954 CE On-Demand Mild CSNK2A1 44 34 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880520961 DD On-Demand Anodyne ADRB1 45 50 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880520961 DD On-Demand Anodyne ADRB3 24 44 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880520961 DD On-Demand Anodyne ACOX1 49 34 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne ACE 21 45 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne SSTR2 78 45 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne OPRM1 18 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne GHRHR 27 41 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MME 29 45 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne EDNRB 44 35 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne EDNRA 45 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne TACR1 44 50 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MC4R 56 39 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne TACR2 17 44 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne CCKAR 137 44 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne CTSL 23 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne BRS3 28 47 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne NMBR 42 45 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MC3R 83 39 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MC5R 89 35 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MMP2 29 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MMP8 36 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne GRPR 81 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne ECE1 66 45 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MMP11 102 38 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne CCKBR 115 41 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne GHSR 75 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MMP9 27 43 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MC1R 107 39 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne MMP1 19 40 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne NPR 27 42 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne KISS1R 75 35 COC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)CN1C[C@@H](O)CC[C@H]1C ZINC000880520964 FD On-Demand Anodyne ERAP2 44 38 Cc1cc(NC(=O)NCCOC(F)(F)C(F)(F)F)ncc1C#N ZINC000880520980 EF On-Demand Mild ADRB1 45 34 CC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521000 CE On-Demand Mild CSNK2A1 56 36 CC(=O)[C@H]1CCCN(C(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521001 CE On-Demand Mild CSNK2A1 56 36 Cc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ncc1C#N ZINC000880521006 DE On-Demand Mild ADRB1 43 34 Cc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ncc1C#N ZINC000880521007 DE On-Demand Mild ADRB1 43 34 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880521019 CF On-Demand Mild CSNK2A1 50 39 Cc1cc(NC(=O)NC[C@H]2CCC(C)(C)CO2)ncc1C#N ZINC000880521058 DF On-Demand Mild CSNK2A1 44 35 Cc1cc(NC(=O)NC[C@@H]2CCC(C)(C)CO2)ncc1C#N ZINC000880521059 DF On-Demand Mild CSNK2A1 44 35 Cc1cc(NC(=O)NC[C@@H](O)C(F)(F)C(F)(F)F)ncc1C#N ZINC000880521060 ED On-Demand Mild ADRB1 44 33 Cc1cc(NC(=O)NC[C@H](O)C(F)(F)C(F)(F)F)ncc1C#N ZINC000880521061 ED On-Demand Mild ADRB1 44 33 Cc1cc(NC(=O)NCC2(OC(C)C)CCC2)ncc1C#N ZINC000880521089 DF On-Demand Mild ADRB1 42 32 CCn1ncc(NC(=O)Nc2cc(C)c(C#N)cn2)c1C ZINC000880521104 CE On-Demand Mild CSNK2A1 42 34 CCn1ncc(NC(=O)Nc2cc(C)c(C#N)cn2)c1C ZINC000880521104 CE On-Demand Mild CHEK1 16 42 CC(=O)C1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880521141 CE On-Demand Mild CSNK2A1 72 38 CC[C@@H](NC(=O)Nc1cc(C)c(C#N)cn1)[C@H](O)c1ccccc1 ZINC000880521160 DF On-Demand Mild ADRB1 43 34 CC[C@@H](NC(=O)Nc1cc(C)c(C#N)cn1)[C@@H](O)c1ccccc1 ZINC000880521162 DF On-Demand Mild ADRB1 43 34 CCC[C@@H](NC(=O)CN1C[C@@H](O)CC[C@H]1C)c1ccccc1 ZINC000880521222 DE On-Demand Anodyne EDNRB 26 44 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1cc(C)c(C#N)cn1)CC2 ZINC000880521223 EF On-Demand Mild CSNK2A1 83 39 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1cc(C)c(C#N)cn1)CC2 ZINC000880521223 EF On-Demand Mild P2RY14 41 38 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1cc(C)c(C#N)cn1)CC2 ZINC000880521223 EF On-Demand Mild HIPK2 40 35 COCC(C)(C)CCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880521257 CE On-Demand Mild ADRB1 42 33 O=C1CC[C@@H](c2ccc(C(=O)NCC3(c4ccccc4F)CCC3)cc2)N1 ZINC000880521268 FH On-Demand Anodyne PLD1 40 33 O=C1CC[C@@H](c2ccc(C(=O)NCC3(c4ccccc4F)CCC3)cc2)N1 ZINC000880521268 FH On-Demand Anodyne PLD2 51 33 O=C1CC[C@H](c2ccc(C(=O)NCC3(c4ccccc4F)CCC3)cc2)N1 ZINC000880521269 FH On-Demand Anodyne PLD1 40 33 O=C1CC[C@H](c2ccc(C(=O)NCC3(c4ccccc4F)CCC3)cc2)N1 ZINC000880521269 FH On-Demand Anodyne PLD2 51 33 CS[C@@H]1C[C@@H](NC(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521299 CE On-Demand Mild CSNK2A1 59 38 Cc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ncc1C#N ZINC000880521304 CF On-Demand Mild CSNK2A1 67 37 O=C(COC1CC1)NCC1(c2ccccc2F)CCC1 ZINC000880521312 CF On-Demand Anodyne TIMP3 51 33 CC[C@@H](NC(=O)Nc1cc(C)c(C#N)cn1)c1ccccc1OC ZINC000880521322 DH On-Demand Mild ADRB1 43 33 C[C@@H]1CC[C@H](O)CN1CC(=O)NCc1cccnc1 ZINC000880521333 CC On-Demand Anodyne CHRNA7 48 38 C[C@@H]1CC[C@H](O)CN1CC(=O)NCc1cccnc1 ZINC000880521333 CC On-Demand Anodyne NAMPT 76 44 CS(=O)(=O)C1CCC(C(=O)NCC2(c3ccccc3F)CCC2)CC1 ZINC000880521362 FF On-Demand Anodyne CACNA1G 15 45 CS(=O)(=O)C1CCC(C(=O)NCc2cccc3ccsc23)CC1 ZINC000880521381 FG On-Demand Anodyne NQO2 22 52 CS(=O)(=O)C1CCC(C(=O)NCc2cccc3ccsc23)CC1 ZINC000880521381 FG On-Demand Anodyne MTNR1A 29 43 CS(=O)(=O)C1CCC(C(=O)NCc2cccc3ccsc23)CC1 ZINC000880521381 FG On-Demand Anodyne MTNR1B 18 41 O=C(NCC1(c2ccccc2F)CCC1)[C@H]1CCc2nncn2CC1 ZINC000880521387 EF On-Demand Anodyne CACNA1G 26 48 O=C(NCC1(c2ccccc2F)CCC1)[C@@H]1CCc2nncn2CC1 ZINC000880521388 EF On-Demand Anodyne CACNA1G 26 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc2ccsc12 ZINC000880521417 GG On-Demand Anodyne PAPA1_CARPA 44 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc2ccsc12 ZINC000880521417 GG On-Demand Anodyne FPR1 42 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc2ccsc12 ZINC000880521418 GG On-Demand Anodyne PAPA1_CARPA 44 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc2ccsc12 ZINC000880521418 GG On-Demand Anodyne FPR1 42 35 Cc1cc(NC(=O)NC[C@H]2c3ccccc3CN2C)ncc1C#N ZINC000880521420 DF On-Demand Mild CSNK2A1 41 32 Cc1cc(NC(=O)NC[C@@H]2c3ccccc3CN2C)ncc1C#N ZINC000880521421 DF On-Demand Mild CSNK2A1 41 32 COCC1CC(NC(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521424 CD On-Demand Mild CSNK2A1 45 35 Cc1cc(NC(=O)NCCSCCC(F)(F)F)ncc1C#N ZINC000880521428 EG On-Demand Mild ADRB1 41 31 O=C(C[C@@H]1CCNC1=O)NCc1cccc(Oc2ccccc2F)c1 ZINC000880521436 EF On-Demand Anodyne BRS3 16 41 O=C(C[C@H]1CCNC1=O)NCc1cccc(Oc2ccccc2F)c1 ZINC000880521437 EF On-Demand Anodyne BRS3 16 41 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H](O)CC[C@H]1C ZINC000880521442 ED On-Demand Anodyne HTR1A 17 45 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H](O)CC[C@H]1C ZINC000880521442 ED On-Demand Anodyne SLC6A4 17 45 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521449 CE On-Demand Mild CSNK2A1 51 37 Cc1cc(NC(=O)N[C@H]2CCc3ccccc3OC2)ncc1C#N ZINC000880521457 DF On-Demand Mild CSNK2A1 45 33 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880521478 JJ On-Demand Mild KDR 43 37 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880521478 JJ On-Demand Mild GRM4 30 51 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880521478 JJ On-Demand Mild KCNK3 51 42 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880521478 JJ On-Demand Mild KCNK9 43 40 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(OC)c1 ZINC000880521508 GF On-Demand Mild HTR1B 15 42 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(OC)c1 ZINC000880521508 GF On-Demand Mild P2RY12 16 41 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(OC)c1 ZINC000880521508 GF On-Demand Mild PDGFRB 62 43 O=C(COC1CC1)NCc1cccc(Oc2ccccc2F)c1 ZINC000880521526 DG On-Demand Anodyne CCR8 23 42 O=C(COC1CC1)NCc1cccc(Oc2ccccc2F)c1 ZINC000880521526 DG On-Demand Anodyne CRTM 52 38 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cc(C)c(C#N)cn1)CC2 ZINC000880521529 EF On-Demand Mild CSNK2A1 84 37 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cc(C)c(C#N)cn1)CC2 ZINC000880521529 EF On-Demand Mild P2RY14 49 40 Cc1cc(NC(=O)NCC[S@@](=O)CC(F)(F)F)ncc1C#N ZINC000880521546 ED On-Demand Mild ADRB1 43 34 Cc1cc(NC(=O)NCC[S@](=O)CC(F)(F)F)ncc1C#N ZINC000880521547 ED On-Demand Mild ADRB1 43 34 CON(C)CCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880521555 CC On-Demand Mild ADRB1 44 34 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCC2(CCc3ccccc3C2)CC1 ZINC000880521614 GG On-Demand Anodyne PREP 47 40 COc1ccccc1N1CC[C@@H](N2C[C@@H](O)CC[C@H]2C)C1=O ZINC000880521615 DD On-Demand Anodyne HTR1A 42 40 COc1ccccc1N1CC[C@@H](N2C[C@@H](O)CC[C@H]2C)C1=O ZINC000880521615 DD On-Demand Anodyne DRD2 19 40 Cc1cc(NC(=O)NCC(Cl)Cl)ncc1C#N ZINC000880521616 CE On-Demand Reactive ADRB1 47 36 Cc1cc(NC(=O)NCC[S@@](C)=O)ncc1C#N ZINC000880521623 CC On-Demand Mild ADRB1 43 33 Cc1cc(NC(=O)NCC[S@](C)=O)ncc1C#N ZINC000880521624 CC On-Demand Mild ADRB1 43 33 O=C1CC[C@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5C4)CC3)cc2)N1 ZINC000880521625 GI On-Demand Anodyne L3MBTL3 42 38 O=C1CC[C@@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5C4)CC3)cc2)N1 ZINC000880521626 GI On-Demand Anodyne L3MBTL3 42 38 COc1ccc(N2CC[C@H](NC(=O)Nc3cc(C)c(C#N)cn3)C2)cc1 ZINC000880521635 FF On-Demand Mild CSNK2A1 42 34 Cc1cc(NC(=O)N[C@H]2C=CCC2)ncc1C#N ZINC000880521643 BE On-Demand Mild CSNK2A1 40 36 Cc1cc(NC(=O)NCCC[C@@H]2CC2(Cl)Cl)ncc1C#N ZINC000880521651 EG On-Demand Mild ADRB1 42 32 Cc1cc(NC(=O)NCCC[C@H]2CC2(Cl)Cl)ncc1C#N ZINC000880521652 EG On-Demand Mild ADRB1 42 32 Cc1cc(NC(=O)NCCC2SCCS2)ncc1C#N ZINC000880521671 DF On-Demand Mild ADRB1 45 35 Cc1cc(NC(=O)NCC[C@@]2(C)C[C@@]2(F)Cl)ncc1C#N ZINC000880521688 DG On-Demand Mild ADRB1 41 31 Cc1cc(NC(=O)NCC[C@]2(C)C[C@@]2(F)Cl)ncc1C#N ZINC000880521689 DG On-Demand Mild ADRB1 41 31 Cc1cc(NC(=O)NCC[C@@]2(C)C[C@]2(F)Cl)ncc1C#N ZINC000880521690 DG On-Demand Mild ADRB1 41 31 Cc1cc(NC(=O)NCC[C@]2(C)C[C@]2(F)Cl)ncc1C#N ZINC000880521691 DG On-Demand Mild ADRB1 41 31 C#CC[C@@H]1CCCN(C(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521705 CF On-Demand Mild CSNK2A1 42 35 C#CC[C@H]1CCCN(C(=O)Nc2cc(C)c(C#N)cn2)C1 ZINC000880521706 CF On-Demand Mild CSNK2A1 42 35 Cc1cnc(Cl)c(C(=O)N2CCn3c(Cc4cccc(F)c4)nnc3C2)c1 ZINC000880521789 GG On-Demand Anodyne P2RX7 54 51 C=CC(C)(C)CC(=O)N1CCn2c(Cc3cccc(F)c3)nnc2C1 ZINC000880521807 EF On-Demand Mild P2RX7 24 40 C#CCN(C(=O)Nc1cc(C)c(C#N)cn1)C1CC1 ZINC000880521886 CD On-Demand Mild CSNK2A1 58 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(c2cccc(F)c2)C1 ZINC000880521912 GG On-Demand Anodyne GHRHR 49 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(c2cccc(F)c2)C1 ZINC000880521912 GG On-Demand Anodyne PAPA1_CARPA 31 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(c2cccc(F)c2)C1 ZINC000880521913 GG On-Demand Anodyne GHRHR 49 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(c2cccc(F)c2)C1 ZINC000880521913 GG On-Demand Anodyne PAPA1_CARPA 31 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(c2cccc(F)c2)C1 ZINC000880521914 GG On-Demand Anodyne GHRHR 49 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(c2cccc(F)c2)C1 ZINC000880521914 GG On-Demand Anodyne PAPA1_CARPA 31 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(c2cccc(F)c2)C1 ZINC000880521915 GG On-Demand Anodyne GHRHR 49 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(c2cccc(F)c2)C1 ZINC000880521915 GG On-Demand Anodyne PAPA1_CARPA 31 42 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc3c(nc1O)CCCC3)C2 ZINC000880521937 FG On-Demand Anodyne ROCK2 17 40 O=C(Cc1ccccc1N1CCCC1=O)Nc1cc2c(nc1O)CCCC2 ZINC000880521976 FF On-Demand Anodyne KCNQ2 49 41 Cc1cc(NC(=O)N[C@H]2CCn3ccnc32)ncc1C#N ZINC000880521983 CD On-Demand Mild CSNK2A1 64 36 Cc1nnc([C@@H]2CCCN(C(=O)C(=O)c3c[nH]c4cc(F)ccc34)C2)o1 ZINC000880522003 FF On-Demand Anodyne HTR1F 41 33 Cc1nnc([C@@H]2CCCN(C(=O)c3ncccc3-c3ccccn3)C2)o1 ZINC000880522046 EF On-Demand Anodyne MAP3K12 32 43 C#C[C@@H]1COCCN1C(=O)Nc1cc(C)c(C#N)cn1 ZINC000880522098 CD On-Demand Mild CSNK2A1 51 36 C#C[C@H]1COCCN1C(=O)Nc1cc(C)c(C#N)cn1 ZINC000880522099 CD On-Demand Mild CSNK2A1 51 36 O=C(c1ncsc1C1CC1)N1CCn2c(Cc3cccc(F)c3)nnc2C1 ZINC000880522155 GF On-Demand Anodyne P2RX7 29 40 Cn1nnc(C(=O)N2CCn3c(Cc4cccc(F)c4)nnc3C2)n1 ZINC000880522157 EC On-Demand Anodyne P2RX7 36 43 Cc1nc(C(C)C)ncc1C(=O)N1CCn2c(Cc3cccc(F)c3)nnc2C1 ZINC000880522198 GF On-Demand Anodyne P2RX7 41 45 O=C(CC[C@@H]1CCc2ccccc21)N1CCC12CCCC2 ZINC000880522209 CI On-Demand Anodyne EBP 17 42 O=C(CC[C@H]1CCc2ccccc21)N1CCC12CCCC2 ZINC000880522210 CI On-Demand Anodyne EBP 17 42 CON(C)C(=O)C1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880522213 ED On-Demand Mild CSNK2A1 68 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(C2(O)CC2)CC1 ZINC000880522236 GG On-Demand Anodyne RBP4 41 39 O=C(c1cnc2cc[nH]c2c1)N1CCC(C2(O)CC2)CC1 ZINC000880522249 CD On-Demand Anodyne L3MBTL3 53 36 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(C4(O)CC4)CC3)cc2)N1 ZINC000880522250 EE On-Demand Anodyne L3MBTL3 63 39 O=C1CC[C@H](c2ccc(C(=O)N3CCC(C4(O)CC4)CC3)cc2)N1 ZINC000880522251 EE On-Demand Anodyne L3MBTL3 63 39 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(C2(O)CC2)CC1 ZINC000880522307 EG On-Demand Anodyne L3MBTL3 55 36 O=C(Nc1cccc(C#Cc2ccccn2)c1)C(O)(c1ccccc1)c1ccccc1 ZINC000880522381 HI On-Demand Mild GRM5 28 43 O=C(Nc1cccc(C#Cc2ccccn2)c1)C(O)(c1ccccc1)c1ccccc1 ZINC000880522381 HI On-Demand Mild KCNK3 29 40 C[C@H](CSc1ccccc1)N(C)C(=O)COC1CC1 ZINC000880522391 CF On-Demand Anodyne TIMP3 54 33 COCCc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880522402 DD On-Demand Anodyne ADRB1 19 49 COC(=O)/C=C\c1ccc(OCCN2C[C@@H](O)CC[C@H]2C)cc1 ZINC000880522411 DE On-Demand Anodyne HRH3 24 40 C[C@@H](CCN1C[C@@H](O)CC[C@H]1C)OCc1ccccc1 ZINC000880522415 CF On-Demand Anodyne GBA2 41 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(C2(O)CC2)CC1 ZINC000880522424 GE On-Demand Anodyne CELA1 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(C2(O)CC2)CC1 ZINC000880522424 GE On-Demand Anodyne GRIN2B 24 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(C2(O)CC2)CC1 ZINC000880522424 GE On-Demand Anodyne PREP 69 53 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(C2(O)CC2)CC1 ZINC000880522424 GE On-Demand Anodyne SLC12A5 67 38 C#CCC[C@@H](O)CNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880522438 CD On-Demand Mild ADRB1 45 35 C#CCC[C@H](O)CNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880522440 CD On-Demand Mild ADRB1 45 35 CO[C@@H](CN1C[C@@H](O)CC[C@H]1C)c1ccc(F)cc1 ZINC000880522448 CE On-Demand Anodyne SLC6A3 20 41 O=C(c1ccc(OC(F)F)c(Br)c1)N1CCC(C2(O)CC2)CC1 ZINC000880522479 GG On-Demand Anodyne L3MBTL3 56 41 Cc1cc(NC(=O)N[C@H]2CCC2(C)C)ncc1C#N ZINC000880522485 CF On-Demand Mild CSNK2A1 43 37 Cc1ccc(C(=O)N2CCN(c3cc(C#N)ccn3)CC2)cc1-n1cccc1 ZINC000880522495 FG On-Demand Mild FASN 36 40 CCC[C@H](NC(=O)Nc1cc(C)c(C#N)cn1)[C@H](O)c1ccccc1 ZINC000880522507 EG On-Demand Mild ADRB1 43 33 CCC[C@H](NC(=O)Nc1cc(C)c(C#N)cn1)[C@@H](O)c1ccccc1 ZINC000880522511 EG On-Demand Mild ADRB1 43 33 CC(C)(C(=O)N1CCC(C2(O)CC2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880522523 FH On-Demand Anodyne HSD11B1 18 40 CC(C)(C(=O)N1CCC(C2(O)CC2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880522523 FH On-Demand Anodyne EPHX2 22 41 CC(C)(C(=O)N1CCC(C2(O)CC2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880522523 FH On-Demand Anodyne MCHR1 15 40 O=C1NCC[C@H]2CCCN(Cc3ccc4ncccc4c3)[C@H]12 ZINC000880522584 CE On-Demand Anodyne HRH3 27 41 O=C1NCC[C@H]2CCCN(Cc3ccc4ncccc4c3)[C@@H]12 ZINC000880522585 CE On-Demand Anodyne HRH3 27 41 O=C1NCC[C@@H]2CCCN(Cc3ccc4ncccc4c3)[C@@H]12 ZINC000880522586 CE On-Demand Anodyne HRH3 27 41 O=C1NCC[C@@H]2CCCN(Cc3ccc4ncccc4c3)[C@H]12 ZINC000880522587 CE On-Demand Anodyne HRH3 27 41 Cc1nc(C(C)C)ncc1C(=O)NC[C@]1(CO)CCc2ccccc21 ZINC000880522700 EF On-Demand Anodyne HCN1 56 33 Cc1nc(C(C)C)ncc1C(=O)NC[C@@]1(CO)CCc2ccccc21 ZINC000880522702 EF On-Demand Anodyne HCN1 56 33 COCCc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880523082 FD On-Demand Anodyne ADRB1 18 44 COCCc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880523083 FD On-Demand Anodyne ADRB1 18 44 COCCc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880523084 FD On-Demand Anodyne ADRB1 18 44 COCCc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880523085 FD On-Demand Anodyne ADRB1 18 44 CC(=O)c1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523091 ED On-Demand Anodyne CCR3 24 42 CC(=O)c1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880523092 ED On-Demand Anodyne CCR3 24 42 CC(=O)c1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880523093 ED On-Demand Anodyne CCR3 24 42 CC(=O)c1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523094 ED On-Demand Anodyne CCR3 24 42 O=C(COC1CC1)NC[C@]1(CO)CCc2ccccc21 ZINC000880523257 CD On-Demand Anodyne TIMP3 50 32 O=C(COC1CC1)NC[C@@]1(CO)CCc2ccccc21 ZINC000880523258 CD On-Demand Anodyne TIMP3 50 32 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne HTR1A 69 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne DRD2 39 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne DRD4 28 44 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne HTR2A 42 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne DRD3 32 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne HTR7 72 49 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@@H]12 ZINC000880523317 FD On-Demand Anodyne SIGMAR1 17 46 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne HTR1A 69 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne DRD2 39 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne DRD4 28 44 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne HTR2A 42 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne DRD3 32 52 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne HTR7 72 49 O=C1NCC[C@@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523318 FD On-Demand Anodyne SIGMAR1 17 46 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne HTR1A 69 52 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne DRD2 39 52 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne DRD4 28 44 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne HTR2A 42 52 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne DRD3 32 52 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne HTR7 72 49 O=C1NCC[C@H]2CCCN(CCCN3CCN(c4ccccc4)CC3)[C@H]12 ZINC000880523319 FD On-Demand Anodyne SIGMAR1 17 46 CC(C)(C)OC(=O)N1CCC(CN2CCC[C@@H]3CCNC(=O)[C@H]32)CC1 ZINC000880523321 FE On-Demand Anodyne GPR119 28 41 CC(C)(C)OC(=O)N1CCC(CN2CCC[C@H]3CCNC(=O)[C@H]32)CC1 ZINC000880523322 FE On-Demand Anodyne GPR119 28 41 CC(C)(C)OC(=O)N1CCC(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)CC1 ZINC000880523323 FE On-Demand Anodyne GPR119 28 41 CC(C)(C)OC(=O)N1CCC(CN2CCC[C@H]3CCNC(=O)[C@@H]32)CC1 ZINC000880523324 FE On-Demand Anodyne GPR119 28 41 CN(C[C@@H](O)c1cccc(C#N)c1)C(=O)c1ccc(CN2CCOCC2)o1 ZINC000880523403 FD On-Demand Mild CASR 17 41 O=C1NCC[C@@H]2CCCN(CCCOCc3ccccc3)[C@@H]12 ZINC000880523514 DE On-Demand Anodyne GBA2 49 39 O=C1NCC[C@H]2CCCN(CCCOCc3ccccc3)[C@@H]12 ZINC000880523515 DE On-Demand Anodyne GBA2 49 39 O=C1NCC[C@@H]2CCCN(CCCOCc3ccccc3)[C@H]12 ZINC000880523516 DE On-Demand Anodyne GBA2 49 39 O=C1NCC[C@H]2CCCN(CCCOCc3ccccc3)[C@H]12 ZINC000880523517 DE On-Demand Anodyne GBA2 49 39 O=C1NCC[C@@H]2CCCN(CCC(=O)N3CCOc4ccccc43)[C@@H]12 ZINC000880523606 ED On-Demand Anodyne GHRL 50 33 O=C1NCC[C@H]2CCCN(CCC(=O)N3CCOc4ccccc43)[C@H]12 ZINC000880523607 ED On-Demand Anodyne GHRL 50 33 O=C1NCC[C@@H]2CCCN(CCC(=O)N3CCOc4ccccc43)[C@H]12 ZINC000880523608 ED On-Demand Anodyne GHRL 50 33 O=C1NCC[C@H]2CCCN(CCC(=O)N3CCOc4ccccc43)[C@@H]12 ZINC000880523609 ED On-Demand Anodyne GHRL 50 33 CCCOc1cccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523630 DF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523630 DF On-Demand Anodyne CHRNA10 45 33 CCCOc1cccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523631 DF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880523631 DF On-Demand Anodyne CHRNA10 45 33 CCCOc1cccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880523632 DF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880523632 DF On-Demand Anodyne CHRNA10 45 33 CCCOc1cccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880523633 DF On-Demand Anodyne HRH2 26 40 CCCOc1cccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880523633 DF On-Demand Anodyne CHRNA10 45 33 O=C1NCC[C@@H]2CCCN(Cc3ccc(F)cc3Cl)[C@H]12 ZINC000880523738 CF On-Demand Anodyne P2RX7 46 45 O=C1NCC[C@@H]2CCCN(Cc3ccc(F)cc3Cl)[C@@H]12 ZINC000880523739 CF On-Demand Anodyne P2RX7 46 45 O=C1NCC[C@H]2CCCN(Cc3ccc(F)cc3Cl)[C@@H]12 ZINC000880523740 CF On-Demand Anodyne P2RX7 46 45 O=C1NCC[C@H]2CCCN(Cc3ccc(F)cc3Cl)[C@H]12 ZINC000880523741 CF On-Demand Anodyne P2RX7 46 45 Cc1cnc(Cl)c(C(=O)NC[C@@]2(CO)CCc3ccccc32)c1 ZINC000880523764 EF On-Demand Anodyne HCN1 43 32 Cc1cnc(Cl)c(C(=O)NC[C@@]2(CO)CCc3ccccc32)c1 ZINC000880523764 EF On-Demand Anodyne G2YM83_BOTF4 52 33 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1cccnc1 ZINC000880523798 DD On-Demand Anodyne CHRNA7 42 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1cccnc1 ZINC000880523798 DD On-Demand Anodyne NAMPT 27 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1cccnc1 ZINC000880523799 DD On-Demand Anodyne CHRNA7 42 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1cccnc1 ZINC000880523799 DD On-Demand Anodyne NAMPT 27 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1cccnc1 ZINC000880523800 DD On-Demand Anodyne CHRNA7 42 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1cccnc1 ZINC000880523800 DD On-Demand Anodyne NAMPT 27 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1cccnc1 ZINC000880523801 DD On-Demand Anodyne CHRNA7 42 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1cccnc1 ZINC000880523801 DD On-Demand Anodyne NAMPT 27 40 O=C(NC[C@]1(CO)CCc2ccccc21)c1cccn2nccc12 ZINC000880523810 DD On-Demand Anodyne HCN1 72 34 O=C(NC[C@]1(CO)CCc2ccccc21)c1cccn2nccc12 ZINC000880523810 DD On-Demand Anodyne HCN4 49 32 O=C(NC[C@@]1(CO)CCc2ccccc21)c1cccn2nccc12 ZINC000880523811 DD On-Demand Anodyne HCN1 72 34 O=C(NC[C@@]1(CO)CCc2ccccc21)c1cccn2nccc12 ZINC000880523811 DD On-Demand Anodyne HCN4 49 32 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523861 CF On-Demand Anodyne SIGMAR1 28 42 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523861 CF On-Demand Anodyne PREP 46 42 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523861 CF On-Demand Anodyne GHRL 64 34 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523862 CF On-Demand Anodyne SIGMAR1 28 42 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523862 CF On-Demand Anodyne PREP 46 42 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@@H]12 ZINC000880523862 CF On-Demand Anodyne GHRL 64 34 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523863 CF On-Demand Anodyne SIGMAR1 28 42 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523863 CF On-Demand Anodyne PREP 46 42 O=C1NCC[C@@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523863 CF On-Demand Anodyne GHRL 64 34 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523864 CF On-Demand Anodyne SIGMAR1 28 42 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523864 CF On-Demand Anodyne PREP 46 42 O=C1NCC[C@H]2CCCN(CCCCc3ccccc3)[C@H]12 ZINC000880523864 CF On-Demand Anodyne GHRL 64 34 O=C1NCC[C@@H]2CCCN(C[C@@H]3CN(Cc4ccccc4)CCCO3)[C@@H]12 ZINC000880523963 FD On-Demand Anodyne DRD4 15 42 O=C1NCC[C@@H]2CCCN(C[C@@H]3CN(Cc4ccccc4)CCCO3)[C@H]12 ZINC000880523964 FD On-Demand Anodyne DRD4 15 42 O=C1NCC[C@@H]2CCCN(C[C@H]3CN(Cc4ccccc4)CCCO3)[C@@H]12 ZINC000880523965 FD On-Demand Anodyne DRD4 15 42 O=C1NCC[C@@H]2CCCN(C[C@H]3CN(Cc4ccccc4)CCCO3)[C@H]12 ZINC000880523966 FD On-Demand Anodyne DRD4 15 42 C#CCN(C(=O)Nc1cc(C)c(C#N)cn1)C1CCCC1 ZINC000880523983 CF On-Demand Mild CSNK2A1 53 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(CO)CCc2ccccc21 ZINC000880524085 GD On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(CO)CCc2ccccc21 ZINC000880524085 GD On-Demand Anodyne FPR1 47 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(CO)CCc2ccccc21 ZINC000880524086 GD On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(CO)CCc2ccccc21 ZINC000880524086 GD On-Demand Anodyne FPR1 47 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(CO)CCc2ccccc21 ZINC000880524087 GD On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(CO)CCc2ccccc21 ZINC000880524087 GD On-Demand Anodyne FPR1 47 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(CO)CCc2ccccc21 ZINC000880524088 GD On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(CO)CCc2ccccc21 ZINC000880524088 GD On-Demand Anodyne FPR1 47 38 O=C1NCC[C@@H]2CCCN(CCc3ccncc3)[C@H]12 ZINC000880524115 CD On-Demand Anodyne HRH3 24 41 O=C1NCC[C@H]2CCCN(CCc3ccncc3)[C@H]12 ZINC000880524116 CD On-Demand Anodyne HRH3 24 41 O=C1NCC[C@@H]2CCCN(CCc3ccncc3)[C@@H]12 ZINC000880524117 CD On-Demand Anodyne HRH3 24 41 O=C1NCC[C@H]2CCCN(CCc3ccncc3)[C@@H]12 ZINC000880524118 CD On-Demand Anodyne HRH3 24 41 Cn1c(=O)c(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc2ccccc21 ZINC000880524297 ED On-Demand Anodyne NPSR1 31 40 Cn1c(=O)c(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc2ccccc21 ZINC000880524298 ED On-Demand Anodyne NPSR1 31 40 Cn1c(=O)c(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc2ccccc21 ZINC000880524299 ED On-Demand Anodyne NPSR1 31 40 Cn1c(=O)c(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc2ccccc21 ZINC000880524300 ED On-Demand Anodyne NPSR1 31 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(F)cc3)[C@@H]12 ZINC000880524333 CD On-Demand Anodyne SLC18A3 15 42 O=C1NCC[C@@H]2CCCN(Cc3ccc(F)cc3)[C@H]12 ZINC000880524334 CD On-Demand Anodyne SLC18A3 15 42 O=C1NCC[C@H]2CCCN(Cc3ccc(F)cc3)[C@H]12 ZINC000880524335 CD On-Demand Anodyne SLC18A3 15 42 O=C1NCC[C@H]2CCCN(Cc3ccc(F)cc3)[C@@H]12 ZINC000880524336 CD On-Demand Anodyne SLC18A3 15 42 O=C1NCC[C@@H]2CCCN(C[C@@H]3CCN(C(=O)c4ccccc4)C3)[C@H]12 ZINC000880524383 ED On-Demand Anodyne L3MBTL3 54 36 O=C1NCC[C@@H]2CCCN(C[C@H]3CCN(C(=O)c4ccccc4)C3)[C@H]12 ZINC000880524384 ED On-Demand Anodyne L3MBTL3 54 36 O=C1NCC[C@@H]2CCCN(C[C@H]3CCN(C(=O)c4ccccc4)C3)[C@@H]12 ZINC000880524385 ED On-Demand Anodyne L3MBTL3 54 36 O=C1NCC[C@@H]2CCCN(C[C@@H]3CCN(C(=O)c4ccccc4)C3)[C@@H]12 ZINC000880524386 ED On-Demand Anodyne L3MBTL3 54 36 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2c(s1)CCC2 ZINC000880524447 ED On-Demand Anodyne SLC27A1 37 47 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2c(s1)CCC2 ZINC000880524452 ED On-Demand Anodyne SLC27A1 37 47 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2c(s1)CCC2 ZINC000880524454 ED On-Demand Anodyne SLC27A1 37 47 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2c(s1)CCC2 ZINC000880524456 ED On-Demand Anodyne SLC27A1 37 47 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880524547 CD On-Demand Anodyne CYP2J2 45 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC[C@H]1SC ZINC000880524549 FF On-Demand Anodyne PAPA1_CARPA 33 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC[C@H]1SC ZINC000880524550 FF On-Demand Anodyne PAPA1_CARPA 33 46 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2cccc(Cl)c2)n1 ZINC000880524559 DE On-Demand Anodyne SLC12A5 66 36 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2cccc(Cl)c2)n1 ZINC000880524560 DE On-Demand Anodyne SLC12A5 66 36 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@H]12 ZINC000880524561 FD On-Demand Anodyne SSTR1 16 40 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@@H]12 ZINC000880524562 FD On-Demand Anodyne SSTR1 16 40 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@@H]12 ZINC000880524563 FD On-Demand Anodyne SSTR1 16 40 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@H]12 ZINC000880524564 FD On-Demand Anodyne SSTR1 16 40 C#CCOCCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880524589 CD On-Demand Mild ADRB1 44 33 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880524600 CD On-Demand Anodyne CYP2J2 45 32 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880524602 CD On-Demand Anodyne CYP2J2 45 32 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880524604 CD On-Demand Anodyne CYP2J2 45 32 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2ccccc2s1 ZINC000880524605 ED On-Demand Anodyne CSNK1D 35 45 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2ccccc2s1 ZINC000880524605 ED On-Demand Anodyne SLC27A1 33 49 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2ccccc2s1 ZINC000880524607 ED On-Demand Anodyne CSNK1D 35 45 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2ccccc2s1 ZINC000880524607 ED On-Demand Anodyne SLC27A1 33 49 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2ccccc2s1 ZINC000880524609 ED On-Demand Anodyne CSNK1D 35 45 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2ccccc2s1 ZINC000880524609 ED On-Demand Anodyne SLC27A1 33 49 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2ccccc2s1 ZINC000880524611 ED On-Demand Anodyne CSNK1D 35 45 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2ccccc2s1 ZINC000880524611 ED On-Demand Anodyne SLC27A1 33 49 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524713 CD On-Demand Anodyne SLC18A2 40 36 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524713 CD On-Demand Anodyne HRH3 27 42 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524713 CD On-Demand Anodyne SIGMAR1 22 40 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524716 CD On-Demand Anodyne SLC18A2 40 36 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524716 CD On-Demand Anodyne HRH3 27 42 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@H]12 ZINC000880524716 CD On-Demand Anodyne SIGMAR1 22 40 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524718 CD On-Demand Anodyne SLC18A2 40 36 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524718 CD On-Demand Anodyne HRH3 27 42 O=C1NCC[C@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524718 CD On-Demand Anodyne SIGMAR1 22 40 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524720 CD On-Demand Anodyne SLC18A2 40 36 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524720 CD On-Demand Anodyne HRH3 27 42 O=C1NCC[C@@H]2CCCN(CCc3ccccc3)[C@@H]12 ZINC000880524720 CD On-Demand Anodyne SIGMAR1 22 40 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880524746 GF On-Demand Anodyne PPARG 48 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880524746 GF On-Demand Anodyne PPARA 44 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880524746 GF On-Demand Anodyne PDE8B 41 34 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880524750 GF On-Demand Anodyne PPARG 48 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880524750 GF On-Demand Anodyne PPARA 44 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880524750 GF On-Demand Anodyne PDE8B 41 34 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880524752 GF On-Demand Anodyne PPARG 48 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880524752 GF On-Demand Anodyne PPARA 44 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880524752 GF On-Demand Anodyne PDE8B 41 34 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880524754 GF On-Demand Anodyne PPARG 48 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880524754 GF On-Demand Anodyne PPARA 44 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880524754 GF On-Demand Anodyne PDE8B 41 34 O=C(NC[C@]1(CO)CCc2ccccc21)c1ccc(CN2CCOCC2)o1 ZINC000880524809 FD On-Demand Anodyne SIGMAR1 18 40 O=C(NC[C@@]1(CO)CCc2ccccc21)c1ccc(CN2CCOCC2)o1 ZINC000880524811 FD On-Demand Anodyne SIGMAR1 18 40 O=C1NCC[C@H]2CCCN(Cc3cnc(Cl)s3)[C@@H]12 ZINC000880524846 CD On-Demand Anodyne NACHRBETA2 15 41 O=C1NCC[C@H]2CCCN(Cc3cnc(Cl)s3)[C@H]12 ZINC000880524847 CD On-Demand Anodyne NACHRBETA2 15 41 O=C1NCC[C@@H]2CCCN(Cc3cnc(Cl)s3)[C@@H]12 ZINC000880524848 CD On-Demand Anodyne NACHRBETA2 15 41 O=C1NCC[C@@H]2CCCN(Cc3cnc(Cl)s3)[C@H]12 ZINC000880524849 CD On-Demand Anodyne NACHRBETA2 15 41 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524862 FE On-Demand Anodyne PIM1 17 45 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524862 FE On-Demand Anodyne CDC7 21 45 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524862 FE On-Demand Anodyne PIM3 20 45 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524863 FE On-Demand Anodyne PIM1 17 45 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524863 FE On-Demand Anodyne CDC7 21 45 O=C1NCC[C@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524863 FE On-Demand Anodyne PIM3 20 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524864 FE On-Demand Anodyne PIM1 17 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524864 FE On-Demand Anodyne CDC7 21 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@@H]12 ZINC000880524864 FE On-Demand Anodyne PIM3 20 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524865 FE On-Demand Anodyne PIM1 17 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524865 FE On-Demand Anodyne CDC7 21 45 O=C1NCC[C@@H]2CCCN(Cc3nc(O)c4oc5ccccc5c4n3)[C@H]12 ZINC000880524865 FE On-Demand Anodyne PIM3 20 45 N#Cc1ccccc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880524943 CD On-Demand Mild DPP4 15 43 N#Cc1ccccc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880524944 CD On-Demand Mild DPP4 15 43 N#Cc1ccccc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880524945 CD On-Demand Mild DPP4 15 43 N#Cc1ccccc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880524946 CD On-Demand Mild DPP4 15 43 Cc1cc(NC(=O)NCCSC(C)(C)C)ncc1C#N ZINC000880524983 CF On-Demand Mild ADRB1 41 32 O=C1NCC[C@@H]2CCCN(C[C@H](O)c3cccc(Cl)c3)[C@H]12 ZINC000880524997 DD On-Demand Anodyne CYP3A4 40 33 O=C1NCC[C@@H]2CCCN(C[C@@H](O)c3cccc(Cl)c3)[C@H]12 ZINC000880525000 DD On-Demand Anodyne CYP3A4 40 33 O=C1NCC[C@@H]2CCCN(C[C@@H](O)c3cccc(Cl)c3)[C@@H]12 ZINC000880525001 DD On-Demand Anodyne CYP3A4 40 33 O=C1NCC[C@@H]2CCCN(C[C@H](O)c3cccc(Cl)c3)[C@@H]12 ZINC000880525003 DD On-Demand Anodyne CYP3A4 40 33 COc1ccc2c(CN3CCC[C@H]4CCNC(=O)[C@@H]43)cc(=O)oc2c1 ZINC000880525014 ED On-Demand Anodyne CYP11B1 17 42 COc1ccc2c(CN3CCC[C@@H]4CCNC(=O)[C@@H]43)cc(=O)oc2c1 ZINC000880525015 ED On-Demand Anodyne CYP11B1 17 42 COc1ccc2c(CN3CCC[C@H]4CCNC(=O)[C@H]43)cc(=O)oc2c1 ZINC000880525016 ED On-Demand Anodyne CYP11B1 17 42 COc1ccc2c(CN3CCC[C@@H]4CCNC(=O)[C@H]43)cc(=O)oc2c1 ZINC000880525017 ED On-Demand Anodyne CYP11B1 17 42 N#Cc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880525034 DD On-Demand Mild CCR3 16 40 N#Cc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880525034 DD On-Demand Mild MCHR1 39 50 N#Cc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880525035 DD On-Demand Mild CCR3 16 40 N#Cc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880525035 DD On-Demand Mild MCHR1 39 50 N#Cc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880525036 DD On-Demand Mild CCR3 16 40 N#Cc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880525036 DD On-Demand Mild MCHR1 39 50 N#Cc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880525037 DD On-Demand Mild CCR3 16 40 N#Cc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880525037 DD On-Demand Mild MCHR1 39 50 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCCC(F)(F)C2)N1Cc1ccccc1 ZINC000880525061 FD On-Demand Anodyne PREP 61 40 Cc1cc(NC(=O)NCC[C@@](C)(O)c2ccccc2)ncc1C#N ZINC000880525139 DF On-Demand Mild ADRB1 46 36 Cc1cc(NC(=O)NCC[C@](C)(O)c2ccccc2)ncc1C#N ZINC000880525140 DF On-Demand Mild ADRB1 46 36 Cc1ccccc1CN1CCC(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)CC1 ZINC000880525165 GD On-Demand Anodyne SIGMAR1 15 44 Cc1ccccc1CN1CCC(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)CC1 ZINC000880525166 GD On-Demand Anodyne SIGMAR1 15 44 Cc1ccccc1CN1CCC(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)CC1 ZINC000880525167 GD On-Demand Anodyne SIGMAR1 15 44 Cc1ccccc1CN1CCC(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)CC1 ZINC000880525168 GD On-Demand Anodyne SIGMAR1 15 44 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525268 ED On-Demand Anodyne ADRB1 18 46 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525268 ED On-Demand Anodyne HTR1A 17 51 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525268 ED On-Demand Anodyne SLC6A4 21 47 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525269 ED On-Demand Anodyne ADRB1 18 46 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525269 ED On-Demand Anodyne HTR1A 17 51 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@H]12 ZINC000880525269 ED On-Demand Anodyne SLC6A4 21 47 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525270 ED On-Demand Anodyne ADRB1 18 46 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525270 ED On-Demand Anodyne HTR1A 17 51 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525270 ED On-Demand Anodyne SLC6A4 21 47 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525271 ED On-Demand Anodyne ADRB1 18 46 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525271 ED On-Demand Anodyne HTR1A 17 51 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4[nH]ccc34)[C@@H]12 ZINC000880525271 ED On-Demand Anodyne SLC6A4 21 47 CN(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Cc1ccccc1 ZINC000880525341 DD On-Demand Anodyne GHRL 101 35 CN(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Cc1ccccc1 ZINC000880525342 DD On-Demand Anodyne GHRL 101 35 CN(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Cc1ccccc1 ZINC000880525343 DD On-Demand Anodyne GHRL 101 35 CN(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Cc1ccccc1 ZINC000880525344 DD On-Demand Anodyne GHRL 101 35 Cc1cc(NC(=O)NC[C@H]2CCC=CO2)ncc1C#N ZINC000880525435 CE On-Demand Mild CSNK2A1 55 36 Cc1cc(NC(=O)NC[C@@H]2CCC=CO2)ncc1C#N ZINC000880525436 CE On-Demand Mild CSNK2A1 55 36 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525441 EE On-Demand Anodyne ENV 43 39 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525441 EE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525442 EE On-Demand Anodyne ENV 43 39 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525442 EE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525443 EE On-Demand Anodyne ENV 43 39 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525443 EE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525444 EE On-Demand Anodyne ENV 43 39 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc(Cl)c(F)c1 ZINC000880525444 EE On-Demand Anodyne MCHR1 16 41 O=C1NCC[C@@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880525445 ED On-Demand Bother HTR3A 17 40 O=C1NCC[C@@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880525445 ED On-Demand Bother HRH3 43 42 O=C1NCC[C@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880525446 ED On-Demand Bother HTR3A 17 40 O=C1NCC[C@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880525446 ED On-Demand Bother HRH3 43 42 O=C1NCC[C@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880525447 ED On-Demand Bother HTR3A 17 40 O=C1NCC[C@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880525447 ED On-Demand Bother HRH3 43 42 O=C1NCC[C@@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880525448 ED On-Demand Bother HTR3A 17 40 O=C1NCC[C@@H]2CCCN(CCCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880525448 ED On-Demand Bother HRH3 43 42 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880525517 GD On-Demand Anodyne EPHX2 68 37 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880525518 GD On-Demand Anodyne EPHX2 68 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880525519 GD On-Demand Anodyne EPHX2 68 37 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880525520 GD On-Demand Anodyne EPHX2 68 37 O=C1NCC[C@@H]2CCCN(CCc3cccnc3)[C@H]12 ZINC000880525575 CD On-Demand Anodyne HRH3 19 42 O=C1NCC[C@@H]2CCCN(CCc3cccnc3)[C@H]12 ZINC000880525575 CD On-Demand Anodyne CHRNA7 46 37 O=C1NCC[C@H]2CCCN(CCc3cccnc3)[C@H]12 ZINC000880525576 CD On-Demand Anodyne HRH3 19 42 O=C1NCC[C@H]2CCCN(CCc3cccnc3)[C@H]12 ZINC000880525576 CD On-Demand Anodyne CHRNA7 46 37 O=C1NCC[C@@H]2CCCN(CCc3cccnc3)[C@@H]12 ZINC000880525577 CD On-Demand Anodyne HRH3 19 42 O=C1NCC[C@@H]2CCCN(CCc3cccnc3)[C@@H]12 ZINC000880525577 CD On-Demand Anodyne CHRNA7 46 37 O=C1NCC[C@H]2CCCN(CCc3cccnc3)[C@@H]12 ZINC000880525578 CD On-Demand Anodyne HRH3 19 42 O=C1NCC[C@H]2CCCN(CCc3cccnc3)[C@@H]12 ZINC000880525578 CD On-Demand Anodyne CHRNA7 46 37 O=C1NCC[C@@H]2CCCN(Cc3ccc(-n4ccnc4)cc3)[C@@H]12 ZINC000880525626 DD On-Demand Anodyne CYP2C19 16 40 O=C1NCC[C@H]2CCCN(Cc3ccc(-n4ccnc4)cc3)[C@@H]12 ZINC000880525628 DD On-Demand Anodyne CYP2C19 16 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(-n4ccnc4)cc3)[C@H]12 ZINC000880525630 DD On-Demand Anodyne CYP2C19 16 40 O=C1NCC[C@H]2CCCN(Cc3ccc(-n4ccnc4)cc3)[C@H]12 ZINC000880525632 DD On-Demand Anodyne CYP2C19 16 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccccc1-c1ccccc1 ZINC000880525819 GG On-Demand Anodyne CHRM3 17 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccccc1-c1ccccc1 ZINC000880525820 GG On-Demand Anodyne CHRM3 17 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccccc1-c1ccccc1 ZINC000880525822 GG On-Demand Anodyne CHRM3 17 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccccc1-c1ccccc1 ZINC000880525823 GG On-Demand Anodyne CHRM3 17 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1cccnc1Cl ZINC000880525837 DD On-Demand Anodyne G2YM83_BOTF4 52 32 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1cccnc1Cl ZINC000880525838 DD On-Demand Anodyne G2YM83_BOTF4 52 32 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1cccnc1Cl ZINC000880525839 DD On-Demand Anodyne G2YM83_BOTF4 52 32 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1cccnc1Cl ZINC000880525840 DD On-Demand Anodyne G2YM83_BOTF4 52 32 N#Cc1c(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@H]32)sc2c1CCC2 ZINC000880525841 FE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@H]32)sc2c1CCC2 ZINC000880525845 FE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)sc2c1CCC2 ZINC000880525848 FE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@@H]32)sc2c1CCC2 ZINC000880525850 FE On-Demand Mild VIPR1 28 46 CC(C)(C)OC(=O)N1CC[C@H](CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)C1 ZINC000880525888 FE On-Demand Anodyne GPR119 24 41 CC(C)(C)OC(=O)N1CC[C@H](CCN2CCC[C@H]3CCNC(=O)[C@@H]32)C1 ZINC000880525889 FE On-Demand Anodyne GPR119 24 41 CC(C)(C)OC(=O)N1CC[C@H](CCN2CCC[C@H]3CCNC(=O)[C@H]32)C1 ZINC000880525890 FE On-Demand Anodyne GPR119 24 41 CC(C)(C)OC(=O)N1CC[C@H](CCN2CCC[C@@H]3CCNC(=O)[C@H]32)C1 ZINC000880525891 FE On-Demand Anodyne GPR119 24 41 O=C1NCC[C@@H]2CCCN(Cc3cc(=O)oc4cc(O)ccc34)[C@@H]12 ZINC000880525908 ED On-Demand Anodyne HSD17B3 33 45 O=C1NCC[C@H]2CCCN(Cc3cc(=O)oc4cc(O)ccc34)[C@H]12 ZINC000880525909 ED On-Demand Anodyne HSD17B3 33 45 O=C1NCC[C@@H]2CCCN(Cc3cc(=O)oc4cc(O)ccc34)[C@H]12 ZINC000880525910 ED On-Demand Anodyne HSD17B3 33 45 O=C1NCC[C@H]2CCCN(Cc3cc(=O)oc4cc(O)ccc34)[C@@H]12 ZINC000880525912 ED On-Demand Anodyne HSD17B3 33 45 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@H](c1ccccc1)c1cccs1 ZINC000880525949 GF On-Demand Anodyne PRCP 20 41 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@@H](c1ccccc1)c1cccs1 ZINC000880525951 GF On-Demand Anodyne PRCP 20 41 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@@H](c1ccccc1)c1cccs1 ZINC000880525954 GF On-Demand Anodyne PRCP 20 41 O=C1NCC[C@H]2CCCN(CCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880526040 DD On-Demand Bother HRH3 21 41 O=C1NCC[C@H]2CCCN(CCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880526041 DD On-Demand Bother HRH3 21 41 O=C1NCC[C@@H]2CCCN(CCOc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880526042 DD On-Demand Bother HRH3 21 41 O=C1NCC[C@@H]2CCCN(CCOc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880526043 DD On-Demand Bother HRH3 21 41 C#CCCCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880526077 BD On-Demand Mild ADRB1 42 33 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@H](c1ccccc1)c1cccs1 ZINC000880526092 GF On-Demand Anodyne PRCP 20 41 Cc1ncc(CCNC(=O)Nc2cc(C)c(C#N)cn2)s1 ZINC000880526095 DE On-Demand Mild ADRB1 43 33 O=C(CC[C@@H]1CCc2ccccc21)N1CCCC(F)(F)C1 ZINC000880526181 CH On-Demand Anodyne EBP 19 51 O=C(CC[C@H]1CCc2ccccc21)N1CCCC(F)(F)C1 ZINC000880526183 CH On-Demand Anodyne EBP 19 51 O=C1NCC[C@@H]2CCCN(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@H]12 ZINC000880526277 GD On-Demand Anodyne SSTR1 33 43 O=C1NCC[C@@H]2CCCN(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@@H]12 ZINC000880526278 GD On-Demand Anodyne SSTR1 33 43 O=C1NCC[C@H]2CCCN(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@@H]12 ZINC000880526279 GD On-Demand Anodyne SSTR1 33 43 O=C1NCC[C@H]2CCCN(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)[C@H]12 ZINC000880526280 GD On-Demand Anodyne SSTR1 33 43 O=C(c1ncccc1-c1ccccn1)N1CCn2c(CC3CC3)nnc2C1 ZINC000880526325 FE On-Demand Anodyne P2RX7 28 45 C[C@@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880526387 DD On-Demand Anodyne BIRC8 44 31 C[C@@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880526390 DD On-Demand Anodyne BIRC8 44 31 C[C@@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880526392 DD On-Demand Anodyne BIRC8 44 31 C[C@@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880526394 DD On-Demand Anodyne BIRC8 44 31 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1ccc(F)cc1C(F)(F)F ZINC000880526422 GE On-Demand Anodyne P2RX7 35 50 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1ccc(F)cc1C(F)(F)F ZINC000880526423 GE On-Demand Anodyne P2RX7 35 50 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1ccc(F)cc1C(F)(F)F ZINC000880526425 GE On-Demand Anodyne P2RX7 35 50 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1ccc(F)cc1C(F)(F)F ZINC000880526427 GE On-Demand Anodyne P2RX7 35 50 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne AVPR2 34 41 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne LTA4H 22 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne PRNP 52 36 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne RPS6KA3 42 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne NOD1 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne NOD2 45 38 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526439 FG On-Demand Anodyne NAMPT 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne AVPR2 34 41 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne LTA4H 22 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne PRNP 52 36 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne RPS6KA3 42 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne NOD1 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne NOD2 45 38 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526442 FG On-Demand Anodyne NAMPT 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne AVPR2 34 41 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne LTA4H 22 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne PRNP 52 36 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne RPS6KA3 42 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne NOD1 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne NOD2 45 38 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880526444 FG On-Demand Anodyne NAMPT 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne AVPR2 34 41 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne LTA4H 22 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne PRNP 52 36 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne RPS6KA3 42 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne NOD1 17 40 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne NOD2 45 38 O=C(Nc1ccccc1)c1ccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880526447 FG On-Demand Anodyne NAMPT 17 40 COc1ccccc1N1CC[C@H](N2CCC[C@H]3CCNC(=O)[C@@H]32)C1=O ZINC000880526621 ED On-Demand Anodyne HTR1A 18 42 COc1ccccc1N1CC[C@H](N2CCC[C@@H]3CCNC(=O)[C@H]32)C1=O ZINC000880526623 ED On-Demand Anodyne HTR1A 18 42 COc1ccccc1N1CC[C@H](N2CCC[C@H]3CCNC(=O)[C@H]32)C1=O ZINC000880526624 ED On-Demand Anodyne HTR1A 18 42 COc1ccccc1N1CC[C@H](N2CCC[C@@H]3CCNC(=O)[C@@H]32)C1=O ZINC000880526626 ED On-Demand Anodyne HTR1A 18 42 O=C1CC[C@H](c2ccc(C(=O)N3CCCC(F)(F)C3)cc2)N1 ZINC000880526714 DF On-Demand Anodyne L3MBTL3 48 35 O=C1CC[C@@H](c2ccc(C(=O)N3CCCC(F)(F)C3)cc2)N1 ZINC000880526716 DF On-Demand Anodyne L3MBTL3 48 35 Cc1cc(NC(=O)N[C@H]2CC[C@H](C)C2)ncc1C#N ZINC000880526791 CF On-Demand Mild CSNK2A1 43 38 Cc1cc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)ncc1C#N ZINC000880526865 FE On-Demand Mild CACNA1I 56 35 CCC[C@H](C)[C@H](CO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880526879 DF On-Demand Anodyne MTNR1B 34 40 CCC[C@H](C)[C@H](CO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880526881 DF On-Demand Anodyne MTNR1B 34 40 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526888 DD On-Demand Mild HTR3A 20 42 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526888 DD On-Demand Mild HRH3 44 45 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526888 DD On-Demand Mild CHRNA10 58 50 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526889 DD On-Demand Mild HTR3A 20 42 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526889 DD On-Demand Mild HRH3 44 45 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880526889 DD On-Demand Mild CHRNA10 58 50 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880526890 DD On-Demand Mild HTR3A 20 42 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880526890 DD On-Demand Mild HRH3 44 45 N#Cc1cccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880526890 DD On-Demand Mild CHRNA10 58 50 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880526891 DD On-Demand Mild HTR3A 20 42 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880526891 DD On-Demand Mild HRH3 44 45 N#Cc1cccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880526891 DD On-Demand Mild CHRNA10 58 50 Cc1cc(NC(=O)N[C@H]2CC[C@@H](C)C2)ncc1C#N ZINC000880526893 CF On-Demand Mild CSNK2A1 43 38 C=CC(C)(C)CC(=O)Nc1cnn(-c2ccc(F)cc2)c1C ZINC000880527033 DH On-Demand Mild NR3C1 23 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527079 GC On-Demand Anodyne EDNRB 39 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527079 GC On-Demand Anodyne EDNRA 38 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527079 GC On-Demand Anodyne NOS2 42 33 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527080 GC On-Demand Anodyne EDNRB 39 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527080 GC On-Demand Anodyne EDNRA 38 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527080 GC On-Demand Anodyne NOS2 42 33 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527081 GC On-Demand Anodyne EDNRB 39 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527081 GC On-Demand Anodyne EDNRA 38 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527081 GC On-Demand Anodyne NOS2 42 33 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527082 GC On-Demand Anodyne EDNRB 39 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527082 GC On-Demand Anodyne EDNRA 38 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCOc1ccc2c(c1)OCO2 ZINC000880527082 GC On-Demand Anodyne NOS2 42 33 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1ccc2c(c1)OCO2 ZINC000880527083 EC On-Demand Anodyne NOS2 105 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1ccc2c(c1)OCO2 ZINC000880527084 EC On-Demand Anodyne NOS2 105 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1ccc2c(c1)OCO2 ZINC000880527085 EC On-Demand Anodyne NOS2 105 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1ccc2c(c1)OCO2 ZINC000880527086 EC On-Demand Anodyne NOS2 105 43 O=C1NCC[C@@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@@H]12 ZINC000880527173 EF On-Demand Anodyne HCRTR1 15 44 O=C1NCC[C@@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@@H]12 ZINC000880527173 EF On-Demand Anodyne HCRTR2 15 44 O=C1NCC[C@@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@H]12 ZINC000880527174 EF On-Demand Anodyne HCRTR1 15 44 O=C1NCC[C@@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@H]12 ZINC000880527174 EF On-Demand Anodyne HCRTR2 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@H]12 ZINC000880527175 EF On-Demand Anodyne HCRTR1 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@H]12 ZINC000880527175 EF On-Demand Anodyne HCRTR2 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@@H]12 ZINC000880527176 EF On-Demand Anodyne HCRTR1 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)[C@@H]12 ZINC000880527176 EF On-Demand Anodyne HCRTR2 15 44 NC(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880527189 DC On-Demand Anodyne HRH3 25 44 NC(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880527190 DC On-Demand Anodyne HRH3 25 44 NC(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880527191 DC On-Demand Anodyne HRH3 25 44 NC(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880527192 DC On-Demand Anodyne HRH3 25 44 CCC[C@H](C)[C@H](CO)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880527209 EE On-Demand Anodyne KCNQ2 58 36 C#CCCCCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880527219 CE On-Demand Mild ADRB1 41 32 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1F ZINC000880527241 FF On-Demand Mild P2RY12 16 40 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1F ZINC000880527241 FF On-Demand Mild PDGFRB 39 41 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1F ZINC000880527241 FF On-Demand Mild IGF1R 26 44 CN(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Cc1ccc(F)cc1 ZINC000880527343 DD On-Demand Anodyne GHRL 61 37 CN(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Cc1ccc(F)cc1 ZINC000880527344 DD On-Demand Anodyne GHRL 61 37 CN(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Cc1ccc(F)cc1 ZINC000880527345 DD On-Demand Anodyne GHRL 61 37 CN(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Cc1ccc(F)cc1 ZINC000880527346 DD On-Demand Anodyne GHRL 61 37 O=C1NCC[C@@H]2CCCN(C[C@H]3COc4ccccc4O3)[C@@H]12 ZINC000880527347 DD On-Demand Anodyne ADRA2B 17 40 O=C1NCC[C@@H]2CCCN(C[C@@H]3COc4ccccc4O3)[C@@H]12 ZINC000880527348 DD On-Demand Anodyne ADRA2B 17 40 O=C1NCC[C@@H]2CCCN(C[C@H]3COc4ccccc4O3)[C@H]12 ZINC000880527349 DD On-Demand Anodyne ADRA2B 17 40 O=C1NCC[C@@H]2CCCN(C[C@@H]3COc4ccccc4O3)[C@H]12 ZINC000880527350 DD On-Demand Anodyne ADRA2B 17 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne PGC 50 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne KLK3 49 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne CCKAR 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne CTSK 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne CTSL 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne REN 56 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne CAPN1 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@@H](C)O ZINC000880527443 GE On-Demand Anodyne FPR1 54 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne PGC 50 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne KLK3 49 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne CCKAR 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne CTSK 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne CTSL 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne REN 56 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne CAPN1 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1F)[C@H](C)O ZINC000880527444 GE On-Demand Anodyne FPR1 54 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne PGC 50 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne KLK3 49 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne CCKAR 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne CTSK 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne CTSL 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne REN 56 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne CAPN1 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@@H](C)O ZINC000880527445 GE On-Demand Anodyne FPR1 54 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne PGC 50 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne KLK3 49 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne CCKAR 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne CTSK 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne CTSL 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne REN 56 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne CAPN1 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1F)[C@H](C)O ZINC000880527446 GE On-Demand Anodyne FPR1 54 44 O=C1NCC[C@@H]2CCCN(Cc3ccc(CN4CCCCC4)cc3)[C@H]12 ZINC000880527557 EF On-Demand Anodyne HRH3 26 50 O=C1NCC[C@H]2CCCN(Cc3ccc(CN4CCCCC4)cc3)[C@H]12 ZINC000880527558 EF On-Demand Anodyne HRH3 26 50 O=C1NCC[C@@H]2CCCN(Cc3ccc(CN4CCCCC4)cc3)[C@@H]12 ZINC000880527559 EF On-Demand Anodyne HRH3 26 50 O=C1NCC[C@H]2CCCN(Cc3ccc(CN4CCCCC4)cc3)[C@@H]12 ZINC000880527560 EF On-Demand Anodyne HRH3 26 50 N#Cc1ccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1Cl ZINC000880527645 ED On-Demand Mild MCHR1 18 43 N#Cc1ccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1Cl ZINC000880527646 ED On-Demand Mild MCHR1 18 43 N#Cc1ccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1Cl ZINC000880527647 ED On-Demand Mild MCHR1 18 43 N#Cc1ccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1Cl ZINC000880527648 ED On-Demand Mild MCHR1 18 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880527677 GD On-Demand Anodyne CNR2 19 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880527678 GD On-Demand Anodyne CNR2 19 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880527679 GD On-Demand Anodyne CNR2 19 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(=O)NC1CCCC1 ZINC000880527680 GD On-Demand Anodyne CNR2 19 40 N#Cc1c(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)sc2c1CCCCC2 ZINC000880527694 GE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)sc2c1CCCCC2 ZINC000880527695 GE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)sc2c1CCCCC2 ZINC000880527696 GE On-Demand Mild VIPR1 28 46 N#Cc1c(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)sc2c1CCCCC2 ZINC000880527697 GE On-Demand Mild VIPR1 28 46 N#Cc1ccccc1OC[C@H](O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880527731 EC On-Demand Mild ADRB1 48 39 N#Cc1ccccc1OC[C@H](O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880527732 EC On-Demand Mild ADRB1 48 39 N#Cc1ccccc1OC[C@H](O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880527733 EC On-Demand Mild ADRB1 48 39 N#Cc1ccccc1OC[C@H](O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880527734 EC On-Demand Mild ADRB1 48 39 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)c1c[nH]c2ccc(F)cc12 ZINC000880527757 EE On-Demand Anodyne MPO 59 35 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)c1c[nH]c2ccc(F)cc12 ZINC000880527759 EE On-Demand Anodyne MPO 59 35 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)c1c[nH]c2ccc(F)cc12 ZINC000880527761 EE On-Demand Anodyne MPO 59 35 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1c[nH]c2ccc(F)cc12 ZINC000880527762 EE On-Demand Anodyne MPO 59 35 Cc1cc(NC(=O)NC[C@H](O)C(F)(F)F)ncc1C#N ZINC000880527798 CD On-Demand Mild ADRB1 46 36 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527832 CD On-Demand Anodyne CHRNA4 27 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527832 CD On-Demand Anodyne ACHP_LYMST 16 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527832 CD On-Demand Anodyne Q8WSF8_APLCA 49 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527832 CD On-Demand Anodyne NACHRBETA2 49 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527834 CD On-Demand Anodyne CHRNA4 27 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527834 CD On-Demand Anodyne ACHP_LYMST 16 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527834 CD On-Demand Anodyne Q8WSF8_APLCA 49 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527834 CD On-Demand Anodyne NACHRBETA2 49 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527836 CD On-Demand Anodyne CHRNA4 27 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527836 CD On-Demand Anodyne ACHP_LYMST 16 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527836 CD On-Demand Anodyne Q8WSF8_APLCA 49 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(Cl)nc3)[C@@H]12 ZINC000880527836 CD On-Demand Anodyne NACHRBETA2 49 43 CCC[C@H](C)[C@H](CO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880527849 FD On-Demand Anodyne KLK3 41 33 CCC[C@H](C)[C@H](CO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880527849 FD On-Demand Anodyne CAPN1 41 34 CCC[C@H](C)[C@H](CO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880527849 FD On-Demand Anodyne XIAP 67 35 CCC[C@H](C)[C@H](CO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880527849 FD On-Demand Anodyne BIRC8 45 36 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nccs1 ZINC000880527885 CC On-Demand Anodyne MAP1 113 45 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nccs1 ZINC000880527886 CC On-Demand Anodyne MAP1 113 45 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nccs1 ZINC000880527887 CC On-Demand Anodyne MAP1 113 45 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nccs1 ZINC000880527888 CC On-Demand Anodyne MAP1 113 45 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527898 CD On-Demand Anodyne CHRNA4 27 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527898 CD On-Demand Anodyne ACHP_LYMST 16 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527898 CD On-Demand Anodyne Q8WSF8_APLCA 49 43 O=C1NCC[C@H]2CCCN(Cc3ccc(Cl)nc3)[C@H]12 ZINC000880527898 CD On-Demand Anodyne NACHRBETA2 49 43 CCC[C@H](C)[C@H](CO)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880528073 DE On-Demand Anodyne MPO 50 35 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528131 FE On-Demand Anodyne EPHX2 55 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528131 FE On-Demand Anodyne MCHR1 17 41 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528132 FE On-Demand Anodyne EPHX2 55 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528132 FE On-Demand Anodyne MCHR1 17 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528133 FE On-Demand Anodyne EPHX2 55 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528133 FE On-Demand Anodyne MCHR1 17 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528134 FE On-Demand Anodyne EPHX2 55 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc(OC(F)(F)F)cc1 ZINC000880528134 FE On-Demand Anodyne MCHR1 17 41 Cc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccccc2)ncc1C#N ZINC000880528230 DF On-Demand Mild ADRB1 41 32 Cc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccccc2)ncc1C#N ZINC000880528231 DF On-Demand Mild ADRB1 41 32 O=C(CCCN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880528324 DE On-Demand Anodyne CYP2J2 52 37 O=C(CCCN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880528325 DE On-Demand Anodyne CYP2J2 52 37 O=C(CCCN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880528326 DE On-Demand Anodyne CYP2J2 52 37 O=C(CCCN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880528327 DE On-Demand Anodyne CYP2J2 52 37 O=C1NCC[C@@H]2CCCN(CCCON3C(=O)c4ccccc4C3=O)[C@H]12 ZINC000880528373 FD On-Demand Anodyne HRH3 17 40 O=C1NCC[C@H]2CCCN(CCCON3C(=O)c4ccccc4C3=O)[C@H]12 ZINC000880528374 FD On-Demand Anodyne HRH3 17 40 O=C1NCC[C@H]2CCCN(CCCON3C(=O)c4ccccc4C3=O)[C@@H]12 ZINC000880528375 FD On-Demand Anodyne HRH3 17 40 O=C1NCC[C@@H]2CCCN(CCCON3C(=O)c4ccccc4C3=O)[C@@H]12 ZINC000880528376 FD On-Demand Anodyne HRH3 17 40 O=C1NCC[C@@H]2CCCN(CCc3ccc(Cl)cc3)[C@@H]12 ZINC000880528393 CE On-Demand Anodyne HRH3 27 43 O=C1NCC[C@H]2CCCN(CCc3ccc(Cl)cc3)[C@H]12 ZINC000880528394 CE On-Demand Anodyne HRH3 27 43 O=C1NCC[C@H]2CCCN(CCc3ccc(Cl)cc3)[C@@H]12 ZINC000880528395 CE On-Demand Anodyne HRH3 27 43 O=C1NCC[C@@H]2CCCN(CCc3ccc(Cl)cc3)[C@H]12 ZINC000880528396 CE On-Demand Anodyne HRH3 27 43 O=C1NCC[C@@H]2CCCN(Cc3cccc(CN4CCCCC4)c3)[C@H]12 ZINC000880528433 EF On-Demand Anodyne HRH3 15 41 O=C1NCC[C@H]2CCCN(Cc3cccc(CN4CCCCC4)c3)[C@H]12 ZINC000880528434 EF On-Demand Anodyne HRH3 15 41 O=C1NCC[C@@H]2CCCN(Cc3cccc(CN4CCCCC4)c3)[C@@H]12 ZINC000880528435 EF On-Demand Anodyne HRH3 15 41 O=C1NCC[C@H]2CCCN(Cc3cccc(CN4CCCCC4)c3)[C@@H]12 ZINC000880528436 EF On-Demand Anodyne HRH3 15 41 N#Cc1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880528463 CD On-Demand Mild HRH3 32 45 N#Cc1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880528463 CD On-Demand Mild KCNJ1 17 45 N#Cc1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880528464 CD On-Demand Mild HRH3 32 45 N#Cc1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880528464 CD On-Demand Mild KCNJ1 17 45 N#Cc1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880528465 CD On-Demand Mild HRH3 32 45 N#Cc1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880528465 CD On-Demand Mild KCNJ1 17 45 N#Cc1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880528466 CD On-Demand Mild HRH3 32 45 N#Cc1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880528466 CD On-Demand Mild KCNJ1 17 45 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880528512 GD On-Demand Anodyne L3MBTL3 63 37 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880528514 GD On-Demand Anodyne L3MBTL3 63 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880528516 GD On-Demand Anodyne L3MBTL3 63 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880528518 GD On-Demand Anodyne L3MBTL3 63 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528522 FD On-Demand Anodyne CSNK1D 43 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528522 FD On-Demand Anodyne SLC27A1 34 44 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528524 FD On-Demand Anodyne CSNK1D 43 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528524 FD On-Demand Anodyne SLC27A1 34 44 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528526 FD On-Demand Anodyne CSNK1D 43 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528526 FD On-Demand Anodyne SLC27A1 34 44 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528528 FD On-Demand Anodyne CSNK1D 43 43 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2ccc(F)cc2s1 ZINC000880528528 FD On-Demand Anodyne SLC27A1 34 44 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1cccnc1 ZINC000880528552 DC On-Demand Anodyne CHRNA7 50 36 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1cccnc1 ZINC000880528552 DC On-Demand Anodyne NAMPT 64 42 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1cccnc1 ZINC000880528554 DC On-Demand Anodyne CHRNA7 50 36 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1cccnc1 ZINC000880528554 DC On-Demand Anodyne NAMPT 64 42 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1cccnc1 ZINC000880528556 DC On-Demand Anodyne CHRNA7 50 36 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1cccnc1 ZINC000880528556 DC On-Demand Anodyne NAMPT 64 42 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1cccnc1 ZINC000880528558 DC On-Demand Anodyne CHRNA7 50 36 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1cccnc1 ZINC000880528558 DC On-Demand Anodyne NAMPT 64 42 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCn2c(CC3CC3)nnc2C1 ZINC000880528580 FD On-Demand Anodyne P2RX7 39 42 O=C1NCC[C@@H]2CCCN(C[C@@H]3CC(c4ccc(Cl)cc4)=NO3)[C@@H]12 ZINC000880528637 EE On-Demand Anodyne LUCI_PHOPY 55 43 O=C1NCC[C@@H]2CCCN(C[C@H]3CC(c4ccc(Cl)cc4)=NO3)[C@H]12 ZINC000880528638 EE On-Demand Anodyne LUCI_PHOPY 55 43 O=C1NCC[C@@H]2CCCN(C[C@@H]3CC(c4ccc(Cl)cc4)=NO3)[C@H]12 ZINC000880528639 EE On-Demand Anodyne LUCI_PHOPY 55 43 O=C1NCC[C@@H]2CCCN(C[C@H]3CC(c4ccc(Cl)cc4)=NO3)[C@@H]12 ZINC000880528641 EE On-Demand Anodyne LUCI_PHOPY 55 43 O=C1NCC[C@@H]2CCCN(Cc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880528691 CD On-Demand Bother KCNJ1 22 40 O=C1NCC[C@@H]2CCCN(Cc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880528692 CD On-Demand Bother KCNJ1 22 40 O=C1NCC[C@H]2CCCN(Cc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880528693 CD On-Demand Bother KCNJ1 22 40 O=C1NCC[C@H]2CCCN(Cc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880528694 CD On-Demand Bother KCNJ1 22 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4ccncc4)cc3)[C@@H]12 ZINC000880528727 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4ccncc4)cc3)[C@H]12 ZINC000880528728 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4ccncc4)cc3)[C@H]12 ZINC000880528729 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4ccncc4)cc3)[C@@H]12 ZINC000880528730 FF On-Demand Anodyne HRH3 23 40 Cc1cc(NC(=O)NCCOC2CCC2)ncc1C#N ZINC000880528735 CD On-Demand Mild ADRB1 43 32 Cc1cc(NC(=O)NCCOC2CCC2)ncc1C#N ZINC000880528735 CD On-Demand Mild CSNK2A1 41 39 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCC1(c2ccccc2)CC1 ZINC000880528753 ED On-Demand Anodyne KCNA3 41 37 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCC1(c2ccccc2)CC1 ZINC000880528754 ED On-Demand Anodyne KCNA3 41 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCC1(c2ccccc2)CC1 ZINC000880528755 ED On-Demand Anodyne KCNA3 41 37 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCC1(c2ccccc2)CC1 ZINC000880528756 ED On-Demand Anodyne KCNA3 41 37 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528757 CE On-Demand Anodyne SIGMAR1 29 42 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528757 CE On-Demand Anodyne PREP 42 43 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528757 CE On-Demand Anodyne GHRL 53 33 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528758 CE On-Demand Anodyne SIGMAR1 29 42 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528758 CE On-Demand Anodyne PREP 42 43 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@H]12 ZINC000880528758 CE On-Demand Anodyne GHRL 53 33 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528759 CE On-Demand Anodyne SIGMAR1 29 42 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528759 CE On-Demand Anodyne PREP 42 43 O=C1NCC[C@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528759 CE On-Demand Anodyne GHRL 53 33 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528760 CE On-Demand Anodyne SIGMAR1 29 42 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528760 CE On-Demand Anodyne PREP 42 43 O=C1NCC[C@@H]2CCCN(CCCc3ccccc3)[C@@H]12 ZINC000880528760 CE On-Demand Anodyne GHRL 53 33 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccc(F)cc1 ZINC000880528770 DD On-Demand Anodyne HTR2A 17 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccc(F)cc1 ZINC000880528772 DD On-Demand Anodyne HTR2A 17 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccc(F)cc1 ZINC000880528773 DD On-Demand Anodyne HTR2A 17 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccc(F)cc1 ZINC000880528774 DD On-Demand Anodyne HTR2A 17 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc(F)c(Cl)c1 ZINC000880528802 EE On-Demand Anodyne MCHR1 30 42 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc(F)c(Cl)c1 ZINC000880528803 EE On-Demand Anodyne MCHR1 30 42 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc(F)c(Cl)c1 ZINC000880528804 EE On-Demand Anodyne MCHR1 30 42 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc(F)c(Cl)c1 ZINC000880528805 EE On-Demand Anodyne MCHR1 30 42 O=C(C(=O)N1CCn2c(CC3CC3)nnc2C1)c1c[nH]c2cc(F)ccc12 ZINC000880528897 FE On-Demand Anodyne GRIN2B 15 54 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880528943 DD On-Demand Anodyne PREP 40 38 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880528943 DD On-Demand Anodyne SLC12A5 64 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880528944 DD On-Demand Anodyne PREP 40 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880528944 DD On-Demand Anodyne SLC12A5 64 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880528945 DD On-Demand Anodyne PREP 40 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880528945 DD On-Demand Anodyne SLC12A5 64 38 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880528946 DD On-Demand Anodyne PREP 40 38 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880528946 DD On-Demand Anodyne SLC12A5 64 38 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880529037 EH On-Demand Anodyne CCR1 57 38 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@H]1CCCc2ccccc21 ZINC000880529040 FE On-Demand Anodyne HTR7 16 50 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@H]1CCCc2ccccc21 ZINC000880529040 FE On-Demand Anodyne BDKRB1 52 44 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@H]1CCCc2ccccc21 ZINC000880529041 FE On-Demand Anodyne HTR7 16 50 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@H]1CCCc2ccccc21 ZINC000880529041 FE On-Demand Anodyne BDKRB1 52 44 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880529042 FE On-Demand Anodyne HTR7 16 50 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880529042 FE On-Demand Anodyne BDKRB1 52 44 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880529043 FE On-Demand Anodyne HTR7 16 50 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880529043 FE On-Demand Anodyne BDKRB1 52 44 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880529059 EH On-Demand Anodyne CCR1 57 38 O=C(c1cccn2nccc12)N1CCn2c(CC3CC3)nnc2C1 ZINC000880529120 DD On-Demand Anodyne P2RX7 38 43 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529141 FE On-Demand Anodyne PREP 40 43 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529141 FE On-Demand Anodyne PARP1 18 46 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529141 FE On-Demand Anodyne L3MBTL3 67 41 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529142 FE On-Demand Anodyne PREP 40 43 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529142 FE On-Demand Anodyne PARP1 18 46 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529142 FE On-Demand Anodyne L3MBTL3 67 41 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529143 FE On-Demand Anodyne PREP 40 43 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529143 FE On-Demand Anodyne PARP1 18 46 O=C1NCC[C@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@H]12 ZINC000880529143 FE On-Demand Anodyne L3MBTL3 67 41 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529144 FE On-Demand Anodyne PREP 40 43 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529144 FE On-Demand Anodyne PARP1 18 46 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(=O)N4CCCCC4)c3)[C@@H]12 ZINC000880529144 FE On-Demand Anodyne L3MBTL3 67 41 O=C(c1cccc2nsnc12)N1CCn2c(CC3CC3)nnc2C1 ZINC000880529159 ED On-Demand Anodyne P2RX7 36 45 O=C1NCC[C@H]2CCCN(Cc3cccnc3)[C@@H]12 ZINC000880529168 BD On-Demand Anodyne CHRNA7 46 36 O=C1NCC[C@H]2CCCN(Cc3cccnc3)[C@@H]12 ZINC000880529168 BD On-Demand Anodyne ACHP_LYMST 25 40 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529193 EC On-Demand Anodyne CA2 24 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529193 EC On-Demand Anodyne CA1 23 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529193 EC On-Demand Anodyne CA7 16 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529193 EC On-Demand Anodyne HRH3 20 56 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529193 EC On-Demand Anodyne CA9 20 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529194 EC On-Demand Anodyne CA2 24 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529194 EC On-Demand Anodyne CA1 23 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529194 EC On-Demand Anodyne CA7 16 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529194 EC On-Demand Anodyne HRH3 20 56 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529194 EC On-Demand Anodyne CA9 20 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529195 EC On-Demand Anodyne CA2 24 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529195 EC On-Demand Anodyne CA1 23 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529195 EC On-Demand Anodyne CA7 16 41 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529195 EC On-Demand Anodyne HRH3 20 56 NS(=O)(=O)c1ccc(CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529195 EC On-Demand Anodyne CA9 20 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529196 EC On-Demand Anodyne CA2 24 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529196 EC On-Demand Anodyne CA1 23 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529196 EC On-Demand Anodyne CA7 16 41 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529196 EC On-Demand Anodyne HRH3 20 56 NS(=O)(=O)c1ccc(CCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529196 EC On-Demand Anodyne CA9 20 41 O=C1NCC[C@H]2CCCN(Cc3cccnc3)[C@H]12 ZINC000880529197 BD On-Demand Anodyne CHRNA7 46 36 O=C1NCC[C@H]2CCCN(Cc3cccnc3)[C@H]12 ZINC000880529197 BD On-Demand Anodyne ACHP_LYMST 25 40 O=C1NCC[C@@H]2CCCN(Cc3cccnc3)[C@@H]12 ZINC000880529199 BD On-Demand Anodyne CHRNA7 46 36 O=C1NCC[C@@H]2CCCN(Cc3cccnc3)[C@@H]12 ZINC000880529199 BD On-Demand Anodyne ACHP_LYMST 25 40 O=C1NCC[C@@H]2CCCN(Cc3cccnc3)[C@H]12 ZINC000880529201 BD On-Demand Anodyne CHRNA7 46 36 O=C1NCC[C@@H]2CCCN(Cc3cccnc3)[C@H]12 ZINC000880529201 BD On-Demand Anodyne ACHP_LYMST 25 40 COc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880529207 DD On-Demand Anodyne HRH3 25 47 COc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880529207 DD On-Demand Anodyne CHRNA10 58 47 COc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880529209 DD On-Demand Anodyne HRH3 25 47 COc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880529209 DD On-Demand Anodyne CHRNA10 58 47 COc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529211 DD On-Demand Anodyne HRH3 25 47 COc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529211 DD On-Demand Anodyne CHRNA10 58 47 COc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529213 DD On-Demand Anodyne HRH3 25 47 COc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529213 DD On-Demand Anodyne CHRNA10 58 47 O=C1NCC[C@H]2CCCN(CCCOCCc3ccccc3)[C@H]12 ZINC000880529224 DE On-Demand Anodyne HRH3 23 45 O=C1NCC[C@H]2CCCN(CCCOCCc3ccccc3)[C@@H]12 ZINC000880529226 DE On-Demand Anodyne HRH3 23 45 O=C1NCC[C@@H]2CCCN(CCCOCCc3ccccc3)[C@H]12 ZINC000880529229 DE On-Demand Anodyne HRH3 23 45 Cn1nnc(C(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)n1 ZINC000880529231 DC On-Demand Anodyne CCR1 65 37 Cn1nnc(C(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)n1 ZINC000880529232 DC On-Demand Anodyne CCR1 65 37 O=C1NCC[C@@H]2CCCN(CCCOCCc3ccccc3)[C@@H]12 ZINC000880529234 DE On-Demand Anodyne HRH3 23 45 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529285 FC On-Demand Anodyne ADRB1 31 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529285 FC On-Demand Anodyne ACOX1 46 34 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529287 FC On-Demand Anodyne ADRB1 31 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529287 FC On-Demand Anodyne ACOX1 46 34 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529289 FC On-Demand Anodyne ADRB1 31 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529289 FC On-Demand Anodyne ACOX1 46 34 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529291 FC On-Demand Anodyne ADRB1 31 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529291 FC On-Demand Anodyne ACOX1 46 34 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1ccccc1 ZINC000880529305 DC On-Demand Anodyne PREP 25 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1ccccc1 ZINC000880529309 DC On-Demand Anodyne PREP 25 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1ccccc1 ZINC000880529311 DC On-Demand Anodyne PREP 25 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1ccccc1 ZINC000880529315 DC On-Demand Anodyne PREP 25 40 CCOc1ccccc1NC(=O)CCN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529331 EE On-Demand Anodyne HCN4 40 31 CCOc1ccccc1NC(=O)CCN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529334 EE On-Demand Anodyne HCN4 40 31 CCOc1ccccc1NC(=O)CCN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529336 EE On-Demand Anodyne HCN4 40 31 O=C1NCC[C@@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880529337 DD On-Demand Bother HRH3 22 40 O=C1NCC[C@@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880529337 DD On-Demand Bother KCNJ1 31 47 CCOc1ccccc1NC(=O)CCN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529338 EE On-Demand Anodyne HCN4 40 31 O=C1NCC[C@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880529343 DD On-Demand Bother HRH3 22 40 O=C1NCC[C@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880529343 DD On-Demand Bother KCNJ1 31 47 O=C1NCC[C@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880529346 DD On-Demand Bother HRH3 22 40 O=C1NCC[C@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@@H]12 ZINC000880529346 DD On-Demand Bother KCNJ1 31 47 O=C1NCC[C@@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880529348 DD On-Demand Bother HRH3 22 40 O=C1NCC[C@@H]2CCCN(CCc3ccc([N+](=O)[O-])cc3)[C@H]12 ZINC000880529348 DD On-Demand Bother KCNJ1 31 47 O=C1NCC[C@@H]2CCCN(CCc3nc(-c4cccc(Cl)c4)no3)[C@@H]12 ZINC000880529370 FF On-Demand Anodyne GRM5 19 51 O=C1NCC[C@@H]2CCCN(CCc3nc(-c4cccc(Cl)c4)no3)[C@H]12 ZINC000880529372 FF On-Demand Anodyne GRM5 19 51 O=C1NCC[C@H]2CCCN(CCc3nc(-c4cccc(Cl)c4)no3)[C@@H]12 ZINC000880529374 FF On-Demand Anodyne GRM5 19 51 O=C1NCC[C@H]2CCCN(CCc3nc(-c4cccc(Cl)c4)no3)[C@H]12 ZINC000880529376 FF On-Demand Anodyne GRM5 19 51 O=C(c1coc(-c2ccccn2)n1)N1CCn2c(CC3CC3)nnc2C1 ZINC000880529378 FD On-Demand Anodyne P2RX7 21 42 Cc1nc(C(C)C)ncc1C(=O)N1CCn2c(Cc3ccccc3F)nnc2C1 ZINC000880529397 GF On-Demand Anodyne P2RX7 38 43 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1cccc(Cl)c1 ZINC000880529402 DD On-Demand Anodyne MCHR1 22 47 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1cccc(Cl)c1 ZINC000880529404 DD On-Demand Anodyne MCHR1 22 47 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1cccc(Cl)c1 ZINC000880529406 DD On-Demand Anodyne MCHR1 22 47 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1cccc(Cl)c1 ZINC000880529409 DD On-Demand Anodyne MCHR1 22 47 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCc1ccc(F)cc1 ZINC000880529446 ED On-Demand Anodyne GPBAR1 17 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCc1ccc(F)cc1 ZINC000880529447 ED On-Demand Anodyne GPBAR1 17 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCc1ccc(F)cc1 ZINC000880529448 ED On-Demand Anodyne GPBAR1 17 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCc1ccc(F)cc1 ZINC000880529449 ED On-Demand Anodyne GPBAR1 17 40 CS(=O)(=O)c1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529524 FD On-Demand Anodyne HTR3A 19 42 CS(=O)(=O)c1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529524 FD On-Demand Anodyne HRH3 60 44 CS(=O)(=O)c1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529526 FD On-Demand Anodyne HTR3A 19 42 CS(=O)(=O)c1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529526 FD On-Demand Anodyne HRH3 60 44 CS(=O)(=O)c1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529528 FD On-Demand Anodyne HTR3A 19 42 CS(=O)(=O)c1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529528 FD On-Demand Anodyne HRH3 60 44 CS(=O)(=O)c1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529531 FD On-Demand Anodyne HTR3A 19 42 CS(=O)(=O)c1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529531 FD On-Demand Anodyne HRH3 60 44 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529605 DD On-Demand Mild HTR3A 21 42 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529605 DD On-Demand Mild HRH3 61 57 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529605 DD On-Demand Mild MEN1 48 42 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529607 DD On-Demand Mild HTR3A 21 42 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529607 DD On-Demand Mild HRH3 61 57 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880529607 DD On-Demand Mild MEN1 48 42 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529609 DD On-Demand Mild HTR3A 21 42 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529609 DD On-Demand Mild HRH3 61 57 N#Cc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529609 DD On-Demand Mild MEN1 48 42 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529610 DD On-Demand Mild HTR3A 21 42 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529610 DD On-Demand Mild HRH3 61 57 N#Cc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880529610 DD On-Demand Mild MEN1 48 42 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880529626 GG On-Demand Anodyne HPGD 35 42 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880529628 GG On-Demand Anodyne HPGD 35 42 O=C1NCC[C@@H]1CC(=O)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880529639 ED On-Demand Anodyne CCR1 51 37 O=C1NCC[C@H]1CC(=O)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880529641 ED On-Demand Anodyne CCR1 51 37 O=C1NCC[C@@H]1CC(=O)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880529645 ED On-Demand Anodyne CCR1 51 37 O=C1NCC[C@H]1CC(=O)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880529648 ED On-Demand Anodyne CCR1 51 37 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529683 ED On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529683 ED On-Demand Anodyne TPP2 52 34 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529685 ED On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529685 ED On-Demand Anodyne TPP2 52 34 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529686 ED On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529686 ED On-Demand Anodyne TPP2 52 34 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529687 ED On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529687 ED On-Demand Anodyne TPP2 52 34 Cc1ccccc1CNC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529724 DD On-Demand Anodyne P2RX7 16 43 Cc1ccccc1CNC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529725 DD On-Demand Anodyne P2RX7 16 43 Cc1ccccc1CNC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529726 DD On-Demand Anodyne P2RX7 16 43 Cc1ccccc1CNC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529727 DD On-Demand Anodyne P2RX7 16 43 CCOc1ccccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529736 ED On-Demand Anodyne HCN1 40 32 CCOc1ccccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880529736 ED On-Demand Anodyne HCN4 41 32 CCOc1ccccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529737 ED On-Demand Anodyne HCN1 40 32 CCOc1ccccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880529737 ED On-Demand Anodyne HCN4 41 32 CCOc1ccccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529738 ED On-Demand Anodyne HCN1 40 32 CCOc1ccccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880529738 ED On-Demand Anodyne HCN4 41 32 CCOc1ccccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529739 ED On-Demand Anodyne HCN1 40 32 CCOc1ccccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880529739 ED On-Demand Anodyne HCN4 41 32 Cc1cc(NC(=O)NCCCCCCO)ncc1C#N ZINC000880529778 CD On-Demand Mild ADRB1 44 33 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529858 CE On-Demand Anodyne HTR3A 21 42 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529858 CE On-Demand Anodyne HRH3 66 44 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529858 CE On-Demand Anodyne CHRNA10 47 39 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529860 CE On-Demand Anodyne HTR3A 21 42 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529860 CE On-Demand Anodyne HRH3 66 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@@H]12 ZINC000880529860 CE On-Demand Anodyne CHRNA10 47 39 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529861 CE On-Demand Anodyne HTR3A 21 42 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529861 CE On-Demand Anodyne HRH3 66 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529861 CE On-Demand Anodyne CHRNA10 47 39 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529862 CE On-Demand Anodyne HTR3A 21 42 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529862 CE On-Demand Anodyne HRH3 66 44 O=C1NCC[C@H]2CCCN(CCCOc3ccccc3)[C@H]12 ZINC000880529862 CE On-Demand Anodyne CHRNA10 47 39 CC(=O)OC1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880529888 DD On-Demand Mild CSNK2A1 60 38 N#Cc1cccc(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880529903 ED On-Demand Mild CCR3 16 41 N#Cc1cccc(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880529903 ED On-Demand Mild MCHR1 40 41 N#Cc1cccc(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529905 ED On-Demand Mild CCR3 16 41 N#Cc1cccc(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529905 ED On-Demand Mild MCHR1 40 41 N#Cc1cccc(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529907 ED On-Demand Mild CCR3 16 41 N#Cc1cccc(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880529907 ED On-Demand Mild MCHR1 40 41 N#Cc1cccc(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880529909 ED On-Demand Mild CCR3 16 41 N#Cc1cccc(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880529909 ED On-Demand Mild MCHR1 40 41 O=C(c1c[nH]cc1C1CC1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880529921 EH On-Demand Anodyne CCR1 56 36 O=C(c1c[nH]cc1C1CC1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880529926 EH On-Demand Anodyne CCR1 56 36 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCOc1ccc(F)cc1 ZINC000880529934 EC On-Demand Anodyne HRH3 15 40 Cc1nn(CC(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)c(=O)o1 ZINC000880529935 FD On-Demand Anodyne CCR1 69 38 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCOc1ccc(F)cc1 ZINC000880529936 EC On-Demand Anodyne HRH3 15 40 Cc1nn(CC(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)c(=O)o1 ZINC000880529937 FD On-Demand Anodyne CCR1 69 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCOc1ccc(F)cc1 ZINC000880529938 EC On-Demand Anodyne HRH3 15 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCOc1ccc(F)cc1 ZINC000880529940 EC On-Demand Anodyne HRH3 15 40 C#CCCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880530012 BD On-Demand Mild ADRB1 44 34 O=C1NCC[C@H]2CCCN(CCOc3cccc(F)c3)[C@H]12 ZINC000880530024 CD On-Demand Anodyne CHRNA10 73 46 O=C1NCC[C@H]2CCCN(CCOc3cccc(F)c3)[C@@H]12 ZINC000880530025 CD On-Demand Anodyne CHRNA10 73 46 O=C1NCC[C@@H]2CCCN(CCOc3cccc(F)c3)[C@@H]12 ZINC000880530026 CD On-Demand Anodyne CHRNA10 73 46 O=C1NCC[C@@H]2CCCN(CCOc3cccc(F)c3)[C@H]12 ZINC000880530027 CD On-Demand Anodyne CHRNA10 73 46 O=C1NCC[C@@H]2CCCN(Cc3nc(-c4cccs4)no3)[C@H]12 ZINC000880530028 DD On-Demand Anodyne ETHR 31 41 O=C1NCC[C@@H]2CCCN(Cc3nc(-c4cccs4)no3)[C@@H]12 ZINC000880530029 DD On-Demand Anodyne ETHR 31 41 O=C1NCC[C@H]2CCCN(Cc3nc(-c4cccs4)no3)[C@H]12 ZINC000880530030 DD On-Demand Anodyne ETHR 31 41 O=C1NCC[C@H]2CCCN(Cc3nc(-c4cccs4)no3)[C@@H]12 ZINC000880530031 DD On-Demand Anodyne ETHR 31 41 COc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530032 DE On-Demand Anodyne HTR3A 22 45 COc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530032 DE On-Demand Anodyne HRH3 78 47 COc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880530033 DE On-Demand Anodyne HTR3A 22 45 COc1ccc(OCCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880530033 DE On-Demand Anodyne HRH3 78 47 COc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880530034 DE On-Demand Anodyne HTR3A 22 45 COc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880530034 DE On-Demand Anodyne HRH3 78 47 COc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530035 DE On-Demand Anodyne HTR3A 22 45 COc1ccc(OCCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530035 DE On-Demand Anodyne HRH3 78 47 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccc([N+](=O)[O-])cc1Cl ZINC000880530037 JK On-Demand Mild GRM4 61 43 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccc([N+](=O)[O-])cc1Cl ZINC000880530037 JK On-Demand Mild NR2E3 63 33 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccc([N+](=O)[O-])cc1Cl ZINC000880530037 JK On-Demand Mild G2YM83_BOTF4 45 32 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880530158 FF On-Demand Mild P2RY12 20 44 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880530158 FF On-Demand Mild PDGFRB 52 40 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880530158 FF On-Demand Mild IGF1R 19 43 COc1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880530158 FF On-Demand Mild CSNK2A1 59 33 N#Cc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880530223 CD On-Demand Mild CHRNA10 70 51 N#Cc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880530225 CD On-Demand Mild CHRNA10 70 51 N#Cc1cccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880530227 CD On-Demand Mild CHRNA10 70 51 N#Cc1cccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880530229 CD On-Demand Mild CHRNA10 70 51 O=C1NCC[C@H]2CCCN(CCc3ccc4c(c3)CCO4)[C@H]12 ZINC000880530256 DD On-Demand Anodyne GHRL 74 40 O=C1NCC[C@H]2CCCN(CCc3ccc4c(c3)CCO4)[C@@H]12 ZINC000880530260 DD On-Demand Anodyne GHRL 74 40 O=C1NCC[C@@H]2CCCN(CCc3ccc4c(c3)CCO4)[C@@H]12 ZINC000880530262 DD On-Demand Anodyne GHRL 74 40 O=C1NCC[C@@H]2CCCN(CCc3ccc4c(c3)CCO4)[C@H]12 ZINC000880530265 DD On-Demand Anodyne GHRL 74 40 Cc1cc(NC(=O)NCCC[S@](C)=O)ncc1C#N ZINC000880530300 CD On-Demand Mild ADRB1 44 34 Cc1cc(NC(=O)NCCC[S@@](C)=O)ncc1C#N ZINC000880530301 CD On-Demand Mild ADRB1 44 34 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880530327 EG On-Demand Anodyne ACACA 54 55 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880530327 EG On-Demand Anodyne ACACB 36 55 C[C@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccc(Cl)cc1 ZINC000880530341 EE On-Demand Anodyne PRCP 19 43 C[C@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccc(Cl)cc1 ZINC000880530342 EE On-Demand Anodyne PRCP 19 43 C[C@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccc(Cl)cc1 ZINC000880530343 EE On-Demand Anodyne PRCP 19 43 C[C@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccc(Cl)cc1 ZINC000880530344 EE On-Demand Anodyne PRCP 19 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530511 FF On-Demand Anodyne LTA4H 17 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530511 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530511 FF On-Demand Anodyne VCP 47 34 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530514 FF On-Demand Anodyne LTA4H 17 43 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530514 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530514 FF On-Demand Anodyne VCP 47 34 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530516 FF On-Demand Anodyne LTA4H 17 43 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530516 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@H]12 ZINC000880530516 FF On-Demand Anodyne VCP 47 34 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530517 FF On-Demand Anodyne LTA4H 17 43 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530517 FF On-Demand Anodyne HRH3 23 40 O=C1NCC[C@H]2CCCN(Cc3ccc(OCc4cccnc4)cc3)[C@@H]12 ZINC000880530517 FF On-Demand Anodyne VCP 47 34 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880530560 DD On-Demand Anodyne PREP 48 36 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880530560 DD On-Demand Anodyne SLC12A5 62 35 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880530561 DD On-Demand Anodyne PREP 48 36 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)OCc1ccccc1 ZINC000880530561 DD On-Demand Anodyne SLC12A5 62 35 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880530562 DD On-Demand Anodyne PREP 48 36 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880530562 DD On-Demand Anodyne SLC12A5 62 35 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880530563 DD On-Demand Anodyne PREP 48 36 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)OCc1ccccc1 ZINC000880530563 DD On-Demand Anodyne SLC12A5 62 35 CCN(CCNC(=O)Nc1cc(C)c(C#N)cn1)C(C)C ZINC000880530595 CE On-Demand Mild ADRB1 43 33 O=C(c1cc2ccccc2cc1F)N1CCn2c(CC3CC3)nnc2C1 ZINC000880530683 FG On-Demand Anodyne P2RX7 43 44 O=C1NCC[C@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@@H]12 ZINC000880530684 ED On-Demand Anodyne HTR3A 19 40 O=C1NCC[C@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@@H]12 ZINC000880530684 ED On-Demand Anodyne HRH3 33 44 O=C1NCC[C@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@H]12 ZINC000880530685 ED On-Demand Anodyne HTR3A 19 40 O=C1NCC[C@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@H]12 ZINC000880530685 ED On-Demand Anodyne HRH3 33 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@H]12 ZINC000880530686 ED On-Demand Anodyne HTR3A 19 40 O=C1NCC[C@@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@H]12 ZINC000880530686 ED On-Demand Anodyne HRH3 33 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@@H]12 ZINC000880530687 ED On-Demand Anodyne HTR3A 19 40 O=C1NCC[C@@H]2CCCN(CCCOc3ccc4c(c3)OCO4)[C@@H]12 ZINC000880530687 ED On-Demand Anodyne HRH3 33 44 O=C(COC1CC1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880530719 DE On-Demand Anodyne CCR1 68 38 O=C(COC1CC1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880530721 DE On-Demand Anodyne CCR1 68 38 N#CC1(CNC(=O)c2cc3ccccc3cc2F)CCCC1 ZINC000880530748 CH On-Demand Mild HCN1 50 31 N#CC1(CNC(=O)c2cc3ccccc3cc2F)CCCC1 ZINC000880530748 CH On-Demand Mild HCN4 48 31 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc(C(F)(F)F)c3)[C@H]12 ZINC000880530769 FE On-Demand Anodyne PDS 42 37 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc(C(F)(F)F)c3)[C@@H]12 ZINC000880530771 FE On-Demand Anodyne PDS 42 37 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc(C(F)(F)F)c3)[C@@H]12 ZINC000880530773 FE On-Demand Anodyne PDS 42 37 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc(C(F)(F)F)c3)[C@H]12 ZINC000880530774 FE On-Demand Anodyne PDS 42 37 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccc2nc(C(F)(F)F)[nH]c2c1 ZINC000880530786 GE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccc2nc(C(F)(F)F)[nH]c2c1 ZINC000880530788 GE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccc2nc(C(F)(F)F)[nH]c2c1 ZINC000880530791 GE On-Demand Anodyne MCHR1 16 41 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccc2nc(C(F)(F)F)[nH]c2c1 ZINC000880530793 GE On-Demand Anodyne MCHR1 16 41 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530866 GE On-Demand Anodyne CPT1A 44 34 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880530867 GE On-Demand Anodyne CPT1A 44 34 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880530868 GE On-Demand Anodyne CPT1A 44 34 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530886 DE On-Demand Anodyne LTA4H 30 43 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530886 DE On-Demand Anodyne EBP 17 44 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530886 DE On-Demand Anodyne CHRNA10 18 42 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530887 DE On-Demand Anodyne LTA4H 30 43 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530887 DE On-Demand Anodyne EBP 17 44 O=C1NCC[C@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530887 DE On-Demand Anodyne CHRNA10 18 42 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530888 DE On-Demand Anodyne LTA4H 30 43 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530888 DE On-Demand Anodyne EBP 17 44 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@@H]12 ZINC000880530888 DE On-Demand Anodyne CHRNA10 18 42 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530889 DE On-Demand Anodyne LTA4H 30 43 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530889 DE On-Demand Anodyne EBP 17 44 O=C1NCC[C@@H]2CCCN(CCOc3ccc(Cl)cc3)[C@H]12 ZINC000880530889 DE On-Demand Anodyne CHRNA10 18 42 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCCc1ccccc1 ZINC000880530928 ED On-Demand Anodyne FKBP1A 31 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)NCCCc1ccccc1 ZINC000880530928 ED On-Demand Anodyne PREP 48 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCCc1ccccc1 ZINC000880530929 ED On-Demand Anodyne FKBP1A 31 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)NCCCc1ccccc1 ZINC000880530929 ED On-Demand Anodyne PREP 48 38 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCCc1ccccc1 ZINC000880530930 ED On-Demand Anodyne FKBP1A 31 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCCCc1ccccc1 ZINC000880530930 ED On-Demand Anodyne PREP 48 38 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCCc1ccccc1 ZINC000880530931 ED On-Demand Anodyne FKBP1A 31 40 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)NCCCc1ccccc1 ZINC000880530931 ED On-Demand Anodyne PREP 48 38 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880531037 GE On-Demand Anodyne CPT1A 44 34 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1nc2c(s1)CCCC2 ZINC000880531056 ED On-Demand Anodyne SLC27A1 40 47 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1nc2c(s1)CCCC2 ZINC000880531058 ED On-Demand Anodyne SLC27A1 40 47 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1nc2c(s1)CCCC2 ZINC000880531060 ED On-Demand Anodyne SLC27A1 40 47 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1nc2c(s1)CCCC2 ZINC000880531062 ED On-Demand Anodyne SLC27A1 40 47 N#CC1(CNC(=O)c2cccn3nccc23)CCCC1 ZINC000880531073 CE On-Demand Mild HCN1 65 35 N#CC1(CNC(=O)c2cccn3nccc23)CCCC1 ZINC000880531073 CE On-Demand Mild HCN4 53 34 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(F)(F)F ZINC000880531108 FF On-Demand Anodyne RBP4 59 34 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(F)(F)F ZINC000880531109 FF On-Demand Anodyne RBP4 59 34 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(F)(F)F ZINC000880531110 FF On-Demand Anodyne RBP4 59 34 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(F)(F)F ZINC000880531111 FF On-Demand Anodyne RBP4 59 34 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCC2)c(O)n1 ZINC000880531112 FG On-Demand Mild KCNA3 46 40 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCC2)c(O)n1 ZINC000880531112 FG On-Demand Mild HCN1 72 41 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCC2)c(O)n1 ZINC000880531112 FG On-Demand Mild HCN4 55 41 CCOc1ccc(-c2nc(CN3CCC[C@H]4CCNC(=O)[C@@H]43)co2)cc1 ZINC000880531150 FF On-Demand Anodyne HRH3 16 46 CCOc1ccc(-c2nc(CN3CCC[C@@H]4CCNC(=O)[C@H]43)co2)cc1 ZINC000880531151 FF On-Demand Anodyne HRH3 16 46 CCOc1ccc(-c2nc(CN3CCC[C@H]4CCNC(=O)[C@H]43)co2)cc1 ZINC000880531152 FF On-Demand Anodyne HRH3 16 46 CCOc1ccc(-c2nc(CN3CCC[C@@H]4CCNC(=O)[C@@H]43)co2)cc1 ZINC000880531153 FF On-Demand Anodyne HRH3 16 46 Cc1cc(NC(=O)NCCc2ccnn2C)ncc1C#N ZINC000880531154 CD On-Demand Mild ADRB1 41 32 Cc1cc(NC(=O)NCCc2ccnn2C)ncc1C#N ZINC000880531154 CD On-Demand Mild CSNK2A1 40 33 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880531158 GF On-Demand Anodyne CCR1 60 39 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880531159 GF On-Demand Anodyne CCR1 60 39 Cc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)ncc1C#N ZINC000880531164 EF On-Demand Mild ADRB1 45 35 Cc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)ncc1C#N ZINC000880531165 EF On-Demand Mild ADRB1 45 35 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531188 FE On-Demand Anodyne ADRB2 18 47 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531188 FE On-Demand Anodyne ADRB1 17 42 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531188 FE On-Demand Anodyne SLC6A4 16 40 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531188 FE On-Demand Anodyne ABCB1 43 40 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531189 FE On-Demand Anodyne ADRB2 18 47 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531189 FE On-Demand Anodyne ADRB1 17 42 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531189 FE On-Demand Anodyne SLC6A4 16 40 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531189 FE On-Demand Anodyne ABCB1 43 40 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531190 FE On-Demand Anodyne ADRB2 18 47 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531190 FE On-Demand Anodyne ADRB1 17 42 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531190 FE On-Demand Anodyne SLC6A4 16 40 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3cccc4ccccc34)[C@@H]12 ZINC000880531190 FE On-Demand Anodyne ABCB1 43 40 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531191 FE On-Demand Anodyne ADRB2 18 47 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531191 FE On-Demand Anodyne ADRB1 17 42 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531191 FE On-Demand Anodyne SLC6A4 16 40 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3cccc4ccccc34)[C@H]12 ZINC000880531191 FE On-Demand Anodyne ABCB1 43 40 NC(=O)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531268 CC On-Demand Anodyne CHEK2 28 40 CSc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880531305 DE On-Demand Anodyne HRH3 27 41 CSc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880531306 DE On-Demand Anodyne HRH3 27 41 CSc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880531307 DE On-Demand Anodyne HRH3 27 41 CSc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880531308 DE On-Demand Anodyne HRH3 27 41 Cn1nnc(C(=O)N2CCN(c3cc(Cl)ccc3Cl)CC2)n1 ZINC000880531362 ED On-Demand Anodyne HRH4 25 40 O=C([C@@H]1CCc2nncn2CC1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880531386 FE On-Demand Anodyne CCR1 42 36 O=C([C@H]1CCc2nncn2CC1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880531389 FE On-Demand Anodyne CCR1 42 36 O=C([C@@H]1CCc2nncn2CC1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880531391 FE On-Demand Anodyne CCR1 42 36 O=C([C@H]1CCc2nncn2CC1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880531393 FE On-Demand Anodyne CCR1 42 36 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531423 FG On-Demand Anodyne RPS6KA3 46 41 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531423 FG On-Demand Anodyne KCNK3 72 38 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880531424 FG On-Demand Anodyne RPS6KA3 46 41 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880531424 FG On-Demand Anodyne KCNK3 72 38 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880531425 FG On-Demand Anodyne RPS6KA3 46 41 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880531425 FG On-Demand Anodyne KCNK3 72 38 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531426 FG On-Demand Anodyne RPS6KA3 46 41 O=C(Nc1ccccc1)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531426 FG On-Demand Anodyne KCNK3 72 38 O=C(CN1CCCCS1(=O)=O)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880531444 GD On-Demand Anodyne CCR1 57 36 O=C(CN1CCCCS1(=O)=O)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880531445 GD On-Demand Anodyne CCR1 57 36 NC(=O)c1cccc(CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880531469 CC On-Demand Anodyne CHEK2 28 40 NC(=O)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880531470 CC On-Demand Anodyne CHEK2 28 40 NC(=O)c1cccc(CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880531471 CC On-Demand Anodyne CHEK2 28 40 O=C1NCC[C@@H]2CCCN(CCCOc3ccc(F)cc3)[C@H]12 ZINC000880531501 DE On-Demand Anodyne HTR3A 21 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccc(F)cc3)[C@H]12 ZINC000880531501 DE On-Demand Anodyne HRH3 67 49 O=C1NCC[C@H]2CCCN(CCCOc3ccc(F)cc3)[C@H]12 ZINC000880531502 DE On-Demand Anodyne HTR3A 21 44 O=C1NCC[C@H]2CCCN(CCCOc3ccc(F)cc3)[C@H]12 ZINC000880531502 DE On-Demand Anodyne HRH3 67 49 O=C1NCC[C@H]2CCCN(CCCOc3ccc(F)cc3)[C@@H]12 ZINC000880531503 DE On-Demand Anodyne HTR3A 21 44 O=C1NCC[C@H]2CCCN(CCCOc3ccc(F)cc3)[C@@H]12 ZINC000880531503 DE On-Demand Anodyne HRH3 67 49 O=C1NCC[C@@H]2CCCN(CCCOc3ccc(F)cc3)[C@@H]12 ZINC000880531504 DE On-Demand Anodyne HTR3A 21 44 O=C1NCC[C@@H]2CCCN(CCCOc3ccc(F)cc3)[C@@H]12 ZINC000880531504 DE On-Demand Anodyne HRH3 67 49 C#CCSCCNC(=O)Nc1cc(C)c(C#N)cn1 ZINC000880531509 CD On-Demand Mild ADRB1 43 33 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1cc([N+](=O)[O-])ccc1N1CCCCC1 ZINC000880531581 IJ On-Demand Mild GRM5 18 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1cc([N+](=O)[O-])ccc1N1CCCCC1 ZINC000880531581 IJ On-Demand Mild TAAR1 28 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1cc([N+](=O)[O-])ccc1N1CCCCC1 ZINC000880531581 IJ On-Demand Mild WDR5 33 40 Cc1cnc(Cl)c(C(=O)N2CCn3c(CC4CC4)nnc3C2)c1 ZINC000880531593 EE On-Demand Anodyne P2RX7 39 43 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCn2c(CC3CC3)nnc2C1 ZINC000880531660 GG On-Demand Anodyne P2RX7 31 43 Cc1cnc(Cl)c(C(=O)N2CCN(CCN(C)C)C(=O)C2)c1 ZINC000880531704 DC On-Demand Anodyne P2RX7 21 41 Cc1cc(NC(=O)NC[C@]2(O)CCc3ccccc32)ncc1C#N ZINC000880531706 DE On-Demand Mild ADRB1 41 32 Cc1cc(NC(=O)NC[C@@]2(O)CCc3ccccc32)ncc1C#N ZINC000880531707 DE On-Demand Mild ADRB1 41 32 CS(=O)(=O)C1CCC(C(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)CC1 ZINC000880531742 GF On-Demand Anodyne CCR1 57 42 CS(=O)(=O)C1CCC(C(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)CC1 ZINC000880531743 GF On-Demand Anodyne CCR1 57 42 N#CC1(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CCCC1 ZINC000880531746 DF On-Demand Mild GABRA1 16 47 Cc1ncc(CC(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)o1 ZINC000880531784 EF On-Demand Anodyne CCR1 57 38 Cc1ncc(CC(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)o1 ZINC000880531788 EF On-Demand Anodyne CCR1 57 38 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880531813 FG On-Demand Anodyne SOAT1 46 39 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880531816 FG On-Demand Anodyne SOAT1 46 39 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880531818 FG On-Demand Anodyne SOAT1 46 39 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880531821 FG On-Demand Anodyne SOAT1 46 39 CC(C)(C(=O)N1CCn2c(CC3CC3)nnc2C1)c1ccc(C(F)(F)F)cc1 ZINC000880531850 GH On-Demand Anodyne P2RX7 19 43 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880531965 EF On-Demand Anodyne CCR1 33 40 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880531967 EF On-Demand Anodyne CCR1 33 40 N#CC1(CNC(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)CCCC1 ZINC000880531987 FD On-Demand Mild NPFFR1 43 37 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@@H]21)NCc1ccccc1Cl ZINC000880532105 ED On-Demand Anodyne P2RX7 36 40 O=C(CCN1CCC[C@@H]2CCNC(=O)[C@H]21)NCc1ccccc1Cl ZINC000880532106 ED On-Demand Anodyne P2RX7 36 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@H]21)NCc1ccccc1Cl ZINC000880532107 ED On-Demand Anodyne P2RX7 36 40 O=C(CCN1CCC[C@H]2CCNC(=O)[C@@H]21)NCc1ccccc1Cl ZINC000880532109 ED On-Demand Anodyne P2RX7 36 40 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@H]1CCCc2ccccc21 ZINC000880532139 ED On-Demand Anodyne BDKRB1 55 44 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@H]1CCCc2ccccc21 ZINC000880532140 ED On-Demand Anodyne BDKRB1 55 44 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880532141 ED On-Demand Anodyne BDKRB1 55 44 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)N[C@@H]1CCCc2ccccc21 ZINC000880532142 ED On-Demand Anodyne BDKRB1 55 44 O=C1NCC[C@@H]2CCCN(CCOc3ccccc3)[C@@H]12 ZINC000880532143 CD On-Demand Anodyne LTA4H 49 44 O=C1NCC[C@@H]2CCCN(CCOc3ccccc3)[C@@H]12 ZINC000880532143 CD On-Demand Anodyne CHRNA10 45 40 O=C1NCC[C@H]2CCCN(CCOc3ccccc3)[C@H]12 ZINC000880532144 CD On-Demand Anodyne LTA4H 49 44 O=C1NCC[C@H]2CCCN(CCOc3ccccc3)[C@H]12 ZINC000880532144 CD On-Demand Anodyne CHRNA10 45 40 O=C1NCC[C@H]2CCCN(CCOc3ccccc3)[C@@H]12 ZINC000880532145 CD On-Demand Anodyne LTA4H 49 44 O=C1NCC[C@H]2CCCN(CCOc3ccccc3)[C@@H]12 ZINC000880532145 CD On-Demand Anodyne CHRNA10 45 40 O=C1NCC[C@@H]2CCCN(CCOc3ccccc3)[C@H]12 ZINC000880532146 CD On-Demand Anodyne LTA4H 49 44 O=C1NCC[C@@H]2CCCN(CCOc3ccccc3)[C@H]12 ZINC000880532146 CD On-Demand Anodyne CHRNA10 45 40 Cc1cnc(Cl)c(C(=O)N2CCn3c(Cc4ccccc4F)nnc3C2)c1 ZINC000880532167 GG On-Demand Anodyne P2RX7 50 49 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880532193 ED On-Demand Anodyne ACOX1 44 32 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880532193 ED On-Demand Anodyne ABCB1 30 48 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880532194 ED On-Demand Anodyne ACOX1 44 32 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880532194 ED On-Demand Anodyne ABCB1 30 48 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880532195 ED On-Demand Anodyne ACOX1 44 32 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880532195 ED On-Demand Anodyne ABCB1 30 48 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880532196 ED On-Demand Anodyne ACOX1 44 32 CC(=O)c1cccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880532196 ED On-Demand Anodyne ABCB1 30 48 O=C(CN1CCC[C@@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(F)(F)F ZINC000880532234 FE On-Demand Anodyne RBP4 55 35 O=C(CN1CCC[C@@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(F)(F)F ZINC000880532235 FE On-Demand Anodyne RBP4 55 35 O=C(CN1CCC[C@H]2CCNC(=O)[C@H]21)Nc1ccccc1C(F)(F)F ZINC000880532236 FE On-Demand Anodyne RBP4 55 35 O=C(CN1CCC[C@H]2CCNC(=O)[C@@H]21)Nc1ccccc1C(F)(F)F ZINC000880532237 FE On-Demand Anodyne RBP4 55 35 N#Cc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532244 CD On-Demand Mild HRH3 36 50 N#Cc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532244 CD On-Demand Mild MEN1 41 38 N#Cc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532245 CD On-Demand Mild HRH3 36 50 N#Cc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532245 CD On-Demand Mild MEN1 41 38 N#Cc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532246 CD On-Demand Mild HRH3 36 50 N#Cc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532246 CD On-Demand Mild MEN1 41 38 N#Cc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532247 CD On-Demand Mild HRH3 36 50 N#Cc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532247 CD On-Demand Mild MEN1 41 38 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@@H]12 ZINC000880532270 FC On-Demand Anodyne ACHE 29 41 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@@H]12 ZINC000880532270 FC On-Demand Anodyne SIGMAR1 48 38 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@H]12 ZINC000880532271 FC On-Demand Anodyne ACHE 29 41 O=C1NCC[C@@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@H]12 ZINC000880532271 FC On-Demand Anodyne SIGMAR1 48 38 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@H]12 ZINC000880532272 FC On-Demand Anodyne ACHE 29 41 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@H]12 ZINC000880532272 FC On-Demand Anodyne SIGMAR1 48 38 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@@H]12 ZINC000880532273 FC On-Demand Anodyne ACHE 29 41 O=C1NCC[C@H]2CCCN(CC(=O)N3CCN(Cc4ccccc4)CC3)[C@@H]12 ZINC000880532273 FC On-Demand Anodyne SIGMAR1 48 38 COC(=O)c1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c(OC)c1 ZINC000880532311 GC On-Demand Anodyne ACKR3 51 32 COC(=O)c1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c(OC)c1 ZINC000880532312 GC On-Demand Anodyne ACKR3 51 32 COC(=O)c1ccc(OC[C@H](O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c(OC)c1 ZINC000880532313 GC On-Demand Anodyne ACKR3 51 32 COC(=O)c1ccc(OC[C@H](O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c(OC)c1 ZINC000880532314 GC On-Demand Anodyne ACKR3 51 32 COc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532319 DD On-Demand Anodyne LTA4H 30 43 COc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532319 DD On-Demand Anodyne HRH3 43 41 COc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532320 DD On-Demand Anodyne LTA4H 30 43 COc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532320 DD On-Demand Anodyne HRH3 43 41 COc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532321 DD On-Demand Anodyne LTA4H 30 43 COc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532321 DD On-Demand Anodyne HRH3 43 41 COc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532322 DD On-Demand Anodyne LTA4H 30 43 COc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532322 DD On-Demand Anodyne HRH3 43 41 CCC[C@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880532323 EE On-Demand Anodyne EDNRB 15 41 CCC[C@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880532324 EE On-Demand Anodyne EDNRB 15 41 CCC[C@H](NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21)c1ccccc1 ZINC000880532325 EE On-Demand Anodyne EDNRB 15 41 CCC[C@H](NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21)c1ccccc1 ZINC000880532326 EE On-Demand Anodyne EDNRB 15 41 CCCCCNC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532363 CC On-Demand Anodyne ASAH1 60 31 CCCCCNC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532364 CC On-Demand Anodyne ASAH1 60 31 CCCCCNC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532365 CC On-Demand Anodyne ASAH1 60 31 CCCCCNC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532366 CC On-Demand Anodyne ASAH1 60 31 Cn1nnc(C(=O)N2CCn3c(Cc4ccccc4F)nnc3C2)n1 ZINC000880532394 EC On-Demand Anodyne P2RX7 33 42 Cc1cc(NC(=O)NCC2Cc3ccccc3C2)ncc1C#N ZINC000880532395 DF On-Demand Mild ADRB1 42 33 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(F)(F)F)c3)[C@@H]12 ZINC000880532425 DF On-Demand Anodyne TACR1 15 44 O=C1NCC[C@@H]2CCCN(Cc3cccc(C(F)(F)F)c3)[C@H]12 ZINC000880532426 DF On-Demand Anodyne TACR1 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(C(F)(F)F)c3)[C@H]12 ZINC000880532427 DF On-Demand Anodyne TACR1 15 44 O=C1NCC[C@H]2CCCN(Cc3cccc(C(F)(F)F)c3)[C@@H]12 ZINC000880532428 DF On-Demand Anodyne TACR1 15 44 CCOc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532430 DE On-Demand Anodyne LTA4H 32 40 CCOc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532430 DE On-Demand Anodyne HRH3 39 41 CCOc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532431 DE On-Demand Anodyne LTA4H 32 40 CCOc1ccc(OCCN2CCC[C@@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532431 DE On-Demand Anodyne HRH3 39 41 CCOc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532432 DE On-Demand Anodyne LTA4H 32 40 CCOc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@@H]32)cc1 ZINC000880532432 DE On-Demand Anodyne HRH3 39 41 CCOc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532433 DE On-Demand Anodyne LTA4H 32 40 CCOc1ccc(OCCN2CCC[C@H]3CCNC(=O)[C@H]32)cc1 ZINC000880532433 DE On-Demand Anodyne HRH3 39 41 O=C1NCC[C@H]2CCCN(CCOc3ccc(F)cc3)[C@H]12 ZINC000880532480 CD On-Demand Anodyne LTA4H 29 44 O=C1NCC[C@H]2CCCN(CCOc3ccc(F)cc3)[C@H]12 ZINC000880532480 CD On-Demand Anodyne HRH3 38 43 O=C1NCC[C@H]2CCCN(CCOc3ccc(F)cc3)[C@@H]12 ZINC000880532481 CD On-Demand Anodyne LTA4H 29 44 O=C1NCC[C@H]2CCCN(CCOc3ccc(F)cc3)[C@@H]12 ZINC000880532481 CD On-Demand Anodyne HRH3 38 43 O=C1NCC[C@@H]2CCCN(CCOc3ccc(F)cc3)[C@@H]12 ZINC000880532482 CD On-Demand Anodyne LTA4H 29 44 O=C1NCC[C@@H]2CCCN(CCOc3ccc(F)cc3)[C@@H]12 ZINC000880532482 CD On-Demand Anodyne HRH3 38 43 O=C1NCC[C@@H]2CCCN(CCOc3ccc(F)cc3)[C@H]12 ZINC000880532483 CD On-Demand Anodyne LTA4H 29 44 O=C1NCC[C@@H]2CCCN(CCOc3ccc(F)cc3)[C@H]12 ZINC000880532483 CD On-Demand Anodyne HRH3 38 43 Cc1cc(NC(=O)NC[C@H](O)CC(C)C)ncc1C#N ZINC000880532484 CD On-Demand Mild ADRB1 47 37 Cc1cc(NC(=O)NC[C@@H](O)CC(C)C)ncc1C#N ZINC000880532485 CD On-Demand Mild ADRB1 47 37 O=C1NCC[C@H]2CCCN(CCOc3cccc(Cl)c3)[C@H]12 ZINC000880532536 DE On-Demand Anodyne HRH3 17 42 O=C1NCC[C@H]2CCCN(CCOc3cccc(Cl)c3)[C@H]12 ZINC000880532536 DE On-Demand Anodyne CHRNA10 53 46 O=C1NCC[C@H]2CCCN(CCOc3cccc(Cl)c3)[C@@H]12 ZINC000880532537 DE On-Demand Anodyne HRH3 17 42 O=C1NCC[C@H]2CCCN(CCOc3cccc(Cl)c3)[C@@H]12 ZINC000880532537 DE On-Demand Anodyne CHRNA10 53 46 O=C1NCC[C@@H]2CCCN(CCOc3cccc(Cl)c3)[C@@H]12 ZINC000880532538 DE On-Demand Anodyne HRH3 17 42 O=C1NCC[C@@H]2CCCN(CCOc3cccc(Cl)c3)[C@@H]12 ZINC000880532538 DE On-Demand Anodyne CHRNA10 53 46 O=C1NCC[C@@H]2CCCN(CCOc3cccc(Cl)c3)[C@H]12 ZINC000880532539 DE On-Demand Anodyne HRH3 17 42 O=C1NCC[C@@H]2CCCN(CCOc3cccc(Cl)c3)[C@H]12 ZINC000880532539 DE On-Demand Anodyne CHRNA10 53 46 COc1ccc([C@H](NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)C(C)C)cc1 ZINC000880532540 FE On-Demand Anodyne EDNRB 20 42 COc1ccc([C@H](NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)C(C)C)cc1 ZINC000880532541 FE On-Demand Anodyne EDNRB 20 42 COc1ccc([C@H](NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)C(C)C)cc1 ZINC000880532542 FE On-Demand Anodyne EDNRB 20 42 COc1ccc([C@H](NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)C(C)C)cc1 ZINC000880532543 FE On-Demand Anodyne EDNRB 20 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne ACE 43 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne OPRM1 47 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne CMA1 70 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne CTRA_BOVIN 55 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne CTRC 43 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne ACE2 46 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne C5AR1 44 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532552 FC On-Demand Anodyne BRCA1 60 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne ACE 43 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne OPRM1 47 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne CMA1 70 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne CTRA_BOVIN 55 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne CTRC 43 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne ACE2 46 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne C5AR1 44 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532553 FC On-Demand Anodyne BRCA1 60 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne ACE 43 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne OPRM1 47 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne CMA1 70 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne CTRA_BOVIN 55 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne CTRC 43 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne ACE2 46 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne C5AR1 44 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532554 FC On-Demand Anodyne BRCA1 60 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne ACE 43 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne OPRM1 47 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne CMA1 70 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne CTRA_BOVIN 55 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne CTRC 43 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne ACE2 46 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne C5AR1 44 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532555 FC On-Demand Anodyne BRCA1 60 32 N#Cc1c(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@H]32)sc2c1CCCC2 ZINC000880532635 GE On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN2CCC[C@@H]3CCNC(=O)[C@@H]32)sc2c1CCCC2 ZINC000880532636 GE On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@@H]32)sc2c1CCCC2 ZINC000880532637 GE On-Demand Mild VIPR1 30 48 N#Cc1c(NC(=O)CCN2CCC[C@H]3CCNC(=O)[C@H]32)sc2c1CCCC2 ZINC000880532638 GE On-Demand Mild VIPR1 30 48 COc1ccc(N2CCC(NC(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880532797 FG On-Demand Mild CSNK2A1 50 35 O=C1CC[C@H](c2ccc(C(=O)N3CCC4(CC3)C(F)(F)C4(F)F)cc2)N1 ZINC000880532854 FG On-Demand Anodyne L3MBTL3 55 37 O=C1CC[C@@H](c2ccc(C(=O)N3CCC4(CC3)C(F)(F)C4(F)F)cc2)N1 ZINC000880532855 FG On-Demand Anodyne L3MBTL3 55 37 COC(=O)c1sccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880532856 FD On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880532857 FD On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880532858 FD On-Demand Anodyne FAS 36 44 COC(=O)c1sccc1NC(=O)CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880532859 FD On-Demand Anodyne FAS 36 44 CCOC(=O)N(C)C1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880532956 EE On-Demand Mild P2RY12 20 42 Cc1nc(C(C)C)ncc1C(=O)NNc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880532957 FI On-Demand Reactive JUN 22 42 Cc1nc(C(C)C)ncc1C(=O)NNc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880532957 FI On-Demand Reactive ATF1 40 34 CC(=O)c1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(F)c1 ZINC000880532981 GF On-Demand Mild CSNK2A1 52 37 CC(=O)c1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(F)c1 ZINC000880532981 GF On-Demand Mild NPY2R 50 36 CC(=O)c1ccc(N2CCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)c(F)c1 ZINC000880532981 GF On-Demand Mild SLC6A9 23 45 Cc1cc(NC(=O)NCCSC(F)(F)F)ncc1C#N ZINC000880532996 DF On-Demand Mild ADRB1 42 32 O=C(/C=C/c1ccc(O)cc1)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880533026 EH On-Demand Mild MMP2 16 55 O=C(/C=C/c1ccc(O)cc1)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880533026 EH On-Demand Mild MMP9 16 55 O=C(/C=C\c1ccc(O)cc1)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880533027 EH On-Demand Mild MMP2 16 55 O=C(/C=C\c1ccc(O)cc1)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880533027 EH On-Demand Mild MMP9 16 55 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1C ZINC000880533170 FF On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1C ZINC000880533170 FF On-Demand Anodyne FPR1 47 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1C ZINC000880533172 FF On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1C ZINC000880533172 FF On-Demand Anodyne FPR1 47 36 CC(=O)Nc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@@H]32)c1 ZINC000880533177 ED On-Demand Anodyne MCHR1 18 40 CC(=O)Nc1cccc(NC(=O)CN2CCC[C@@H]3CCNC(=O)[C@H]32)c1 ZINC000880533179 ED On-Demand Anodyne MCHR1 18 40 CC(=O)Nc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@H]32)c1 ZINC000880533181 ED On-Demand Anodyne MCHR1 18 40 CC(=O)Nc1cccc(NC(=O)CN2CCC[C@H]3CCNC(=O)[C@@H]32)c1 ZINC000880533183 ED On-Demand Anodyne MCHR1 18 40 O[C@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533192 DG On-Demand Anodyne ADRB1 18 40 O[C@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533192 DG On-Demand Anodyne ADRB3 30 40 O[C@@H](CN[C@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533197 DG On-Demand Anodyne ADRB1 18 40 O[C@@H](CN[C@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533197 DG On-Demand Anodyne ADRB3 30 40 O[C@@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533199 DG On-Demand Anodyne ADRB1 18 40 O[C@@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533199 DG On-Demand Anodyne ADRB3 30 40 O[C@H](CN[C@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533201 DG On-Demand Anodyne ADRB1 18 40 O[C@H](CN[C@H](c1cccc(Cl)c1)C(F)F)C(F)(F)F ZINC000880533201 DG On-Demand Anodyne ADRB3 30 40 N#Cc1cc(NC(=O)NCCOC(F)(F)C(F)(F)F)ccn1 ZINC000880533214 DE On-Demand Mild ADRB1 43 34 N#Cc1cc(NC(=O)N2CCC(c3cccc(F)c3)CC2)ccn1 ZINC000880533266 DH On-Demand Mild CACNA1H 52 42 N#Cc1cc(NC(=O)N2CCC(c3cccc(F)c3)CC2)ccn1 ZINC000880533266 DH On-Demand Mild MCHR1 24 41 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880533284 DE On-Demand Mild EPHX2 33 40 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3ccc4ccccc4c3)[C@H]12 ZINC000880533416 FE On-Demand Anodyne ACOX1 50 36 O=C1NCC[C@@H]2CCCN(C[C@@H](O)COc3ccc4ccccc4c3)[C@@H]12 ZINC000880533417 FE On-Demand Anodyne ACOX1 50 36 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3ccc4ccccc4c3)[C@H]12 ZINC000880533418 FE On-Demand Anodyne ACOX1 50 36 O=C1NCC[C@@H]2CCCN(C[C@H](O)COc3ccc4ccccc4c3)[C@@H]12 ZINC000880533420 FE On-Demand Anodyne ACOX1 50 36 Cc1ccc(N2CCCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880533461 EG On-Demand Mild P2RY12 16 41 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880533490 FH On-Demand Mild PDGFRB 45 40 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880533490 FH On-Demand Mild RBP4 47 43 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880533492 FH On-Demand Mild PDGFRB 45 40 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880533492 FH On-Demand Mild RBP4 47 43 Cc1cc(NC(=O)NCc2ccc(N3CCCC3)cc2)ncc1C#N ZINC000880533503 EG On-Demand Mild CTSK 17 42 CC(=O)C1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880533526 CD On-Demand Mild TYK2 44 38 Cc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ncc1C#N ZINC000880533634 FF On-Demand Mild NAMPT 24 48 CS(=O)(=O)C1CCC(C(=O)NNc2ccc(Cl)c(C(F)(F)F)c2)CC1 ZINC000880533672 GG On-Demand Reactive EPHX2 33 53 CS(=O)(=O)C1CCC(C(=O)NNc2ccc(Cl)c(C(F)(F)F)c2)CC1 ZINC000880533672 GG On-Demand Reactive SFRP1 86 35 CS(=O)(=O)C1CCC(C(=O)NNc2ccc(Cl)c(C(F)(F)F)c2)CC1 ZINC000880533672 GG On-Demand Reactive WNT3 50 31 COCC(C)(C)CCNC(=O)Nc1ccnc(C#N)c1 ZINC000880533759 CE On-Demand Mild ADRB1 40 30 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880533791 CF On-Demand Mild EPHX2 32 40 CCOC(=O)N1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880533808 DD On-Demand Mild P2RY12 55 49 CCOC(=O)N1CCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880533808 DD On-Demand Mild CSNK2A1 44 34 N#Cc1cc(NC(=O)N2CCC(F)CC2)ccn1 ZINC000880533814 BD On-Demand Mild TYK2 46 37 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3ccnc(C#N)c3)C[C@]2(C)C1 ZINC000880533819 FF On-Demand Mild GPR119 19 45 CCOC(=O)N1CCCN(C(=O)Nc2cc(C)c(C#N)cn2)CC1 ZINC000880533873 ED On-Demand Mild P2RY12 46 47 CC(C)(C)C[C@@H]1C[C@H]1NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880533876 DG On-Demand Anodyne SSTR3 26 43 CC(C)(C)C[C@@H]1C[C@H]1NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880533878 DG On-Demand Anodyne SSTR3 26 43 N#Cc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccn1 ZINC000880533957 CE On-Demand Mild ADRB1 42 31 N#Cc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccn1 ZINC000880533957 CE On-Demand Mild PRMT3 27 42 N#Cc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccn1 ZINC000880533958 CE On-Demand Mild ADRB1 42 31 N#Cc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccn1 ZINC000880533958 CE On-Demand Mild PRMT3 27 42 O=C(COC1CC1)N1CCN(S(=O)(=O)NCc2ccccc2)CC1 ZINC000880533961 FC On-Demand Anodyne F13A1 45 36 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)C2(CCC2)CC1 ZINC000880533962 GG On-Demand Mild GPR119 24 46 Cc1cccc(CN2CCO[C@@H](CNC(=O)Nc3ccnc(C#N)c3)C2)c1 ZINC000880533969 FE On-Demand Mild DRD4 17 42 Cc1cccc(CN2CCO[C@@H](CNC(=O)Nc3ccnc(C#N)c3)C2)c1 ZINC000880533969 FE On-Demand Mild CCR3 24 44 Cc1cccc(CN2CCO[C@H](CNC(=O)Nc3ccnc(C#N)c3)C2)c1 ZINC000880533970 FE On-Demand Mild DRD4 17 42 Cc1cccc(CN2CCO[C@H](CNC(=O)Nc3ccnc(C#N)c3)C2)c1 ZINC000880533970 FE On-Demand Mild CCR3 24 44 Cc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ncc1C#N ZINC000880534037 CF On-Demand Mild CSNK2A1 41 33 Cc1nn(CC(=O)NNc2ccc(Cl)c(C(F)(F)F)c2)c(=O)o1 ZINC000880534069 FD On-Demand Reactive IMDH_CRYPV 19 44 O=C(NNc1ccc(Cl)c(C(F)(F)F)c1)[C@@H]1CCc2nncn2CC1 ZINC000880534070 FG On-Demand Reactive EPHX2 16 46 O=C(NNc1ccc(Cl)c(C(F)(F)F)c1)[C@H]1CCc2nncn2CC1 ZINC000880534071 FG On-Demand Reactive EPHX2 16 46 N#Cc1cc(NC(=O)NCCC[C@@H]2C=CCC2)ccn1 ZINC000880534125 CF On-Demand Mild CCR3 17 40 N#Cc1cc(NC(=O)NCCC[C@H]2C=CCC2)ccn1 ZINC000880534126 CF On-Demand Mild CCR3 17 40 Cc1ccc(CN2CCO[C@H](CNC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880534180 FE On-Demand Mild DRD4 15 41 Cc1ccc(CN2CCO[C@H](CNC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880534180 FE On-Demand Mild CCR3 22 47 CCCCCN(CCNC(=O)c1nnn(C)n1)Cc1ccccc1 ZINC000880534258 ED On-Demand Anodyne TSPO 30 41 CC[C@@H](NC(=O)Nc1ccnc(C#N)c1)c1cccc(OC)c1OC ZINC000880534277 EG On-Demand Mild KDR 44 40 CC[C@@H](NC(=O)Nc1ccnc(C#N)c1)c1cccc(OC)c1OC ZINC000880534277 EG On-Demand Mild PDGFRA 49 40 FC(F)[C@@H](NCCOC1CCOCC1)c1cccc(Cl)c1 ZINC000880534330 DG On-Demand Anodyne MAPK1 49 41 FC(F)[C@H](NCCOC1CCOCC1)c1cccc(Cl)c1 ZINC000880534332 DG On-Demand Anodyne MAPK1 49 41 N#Cc1cc(NC(=O)NCCC2CCC2)ccn1 ZINC000880534339 BE On-Demand Mild CCR3 25 43 N#Cc1cc(NC(=O)NCCC2CCC2)ccn1 ZINC000880534339 BE On-Demand Mild PRMT3 27 49 N#Cc1cc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)ccn1 ZINC000880534352 DH On-Demand Mild CACNA1H 41 39 N#Cc1cc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)ccn1 ZINC000880534352 DH On-Demand Mild FASN 41 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534363 DE On-Demand Anodyne PAPA1_CARPA 39 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534363 DE On-Demand Anodyne CTSK 18 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534363 DE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534363 DE On-Demand Anodyne FPR1 44 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534364 DE On-Demand Anodyne PAPA1_CARPA 39 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534364 DE On-Demand Anodyne CTSK 18 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534364 DE On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C(C)C ZINC000880534364 DE On-Demand Anodyne FPR1 44 38 C[C@]1(C(F)(F)F)CN(C(=O)Nc2ccnc(C#N)c2)CCO1 ZINC000880534370 DE On-Demand Mild EPHX2 30 42 O=C(CCN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880534377 DG On-Demand Anodyne DPP7 30 40 O=C(CCN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880534379 DG On-Demand Anodyne DPP7 30 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880534424 CD On-Demand Mild TYK2 44 36 CC(=O)[C@H]1CCCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880534425 CD On-Demand Mild TYK2 44 36 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880534432 CE On-Demand Mild TYK2 43 38 N#Cc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)ccn1 ZINC000880534440 DG On-Demand Mild NPY5R 37 44 N#Cc1cc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)ccn1 ZINC000880534441 DG On-Demand Mild NPY5R 37 44 O=C1NCC[C@@H]2CCCN(Cc3ccccc3)[C@H]12 ZINC000880534508 BD On-Demand Anodyne SIGMAR1 36 40 O=C1NCC[C@H]2CCCN(Cc3ccccc3)[C@H]12 ZINC000880534509 BD On-Demand Anodyne SIGMAR1 36 40 O=C1NCC[C@@H]2CCCN(Cc3ccccc3)[C@@H]12 ZINC000880534512 BD On-Demand Anodyne SIGMAR1 36 40 O=C1NCC[C@H]2CCCN(Cc3ccccc3)[C@@H]12 ZINC000880534514 BD On-Demand Anodyne SIGMAR1 36 40 COC[C@@H](O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880534520 CE On-Demand Anodyne ADRB2 15 40 COC[C@@H](O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880534521 CE On-Demand Anodyne ADRB2 15 40 N#Cc1cc(NC(=O)N2CCC(Oc3ccc(Cl)cn3)CC2)ccn1 ZINC000880534528 FG On-Demand Mild EPHX2 16 42 CN1CCN(C2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)CC1 ZINC000880534566 ED On-Demand Mild L3MBTL3 61 40 O=C1NCC[C@@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@@H]12 ZINC000880534606 EF On-Demand Anodyne HCRTR1 16 41 O=C1NCC[C@@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@@H]12 ZINC000880534606 EF On-Demand Anodyne HCRTR2 17 41 O=C1NCC[C@@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@H]12 ZINC000880534607 EF On-Demand Anodyne HCRTR1 16 41 O=C1NCC[C@@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@H]12 ZINC000880534607 EF On-Demand Anodyne HCRTR2 17 41 O=C1NCC[C@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@H]12 ZINC000880534608 EF On-Demand Anodyne HCRTR1 16 41 O=C1NCC[C@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@H]12 ZINC000880534608 EF On-Demand Anodyne HCRTR2 17 41 O=C1NCC[C@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@@H]12 ZINC000880534609 EF On-Demand Anodyne HCRTR1 16 41 O=C1NCC[C@H]2CCCN(Cc3ccc(OC(F)(F)F)cc3)[C@@H]12 ZINC000880534609 EF On-Demand Anodyne HCRTR2 17 41 O=C(CCN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880534646 EH On-Demand Anodyne DPP7 42 42 O=C(CCN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880534647 EH On-Demand Anodyne DPP7 42 42 C[C@H]1c2sccc2CCN1C(=O)Nc1ccnc(C#N)c1 ZINC000880534668 CG On-Demand Mild TRPM8 26 41 N#Cc1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccn1 ZINC000880534691 CD On-Demand Mild CACNA1H 40 45 C#CCC1(O)CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880534698 CD On-Demand Mild S1PR2 27 41 COc1ccc(N2CCCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880534773 FG On-Demand Mild P2RY12 18 42 COc1ccc(N2CCCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880534773 FG On-Demand Mild PDGFRB 48 38 COc1ccc(N2CCCN(C(=O)Nc3cc(C)c(C#N)cn3)CC2)cc1 ZINC000880534773 FG On-Demand Mild IGF1R 19 41 O=C(COC1CC1)NNc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880534798 DF On-Demand Reactive RAF1 25 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1CC(C)(C)C ZINC000880534807 EF On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1CC(C)(C)C ZINC000880534808 EF On-Demand Anodyne PAPA1_CARPA 35 42 O=C1NCC[C@H]2CCCN(Cc3nc(-c4cccc(Cl)c4)no3)[C@H]12 ZINC000880534908 EE On-Demand Anodyne GRM5 24 46 O=C1NCC[C@H]2CCCN(Cc3nc(-c4cccc(Cl)c4)no3)[C@@H]12 ZINC000880534910 EE On-Demand Anodyne GRM5 24 46 O=C1NCC[C@@H]2CCCN(Cc3nc(-c4cccc(Cl)c4)no3)[C@H]12 ZINC000880534913 EE On-Demand Anodyne GRM5 24 46 O=C1NCC[C@@H]2CCCN(Cc3nc(-c4cccc(Cl)c4)no3)[C@@H]12 ZINC000880534914 EE On-Demand Anodyne GRM5 24 46 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild HTR1A 16 49 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild HTR1B 17 49 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild PDGFRB 80 52 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild NPY2R 24 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild PDGFRA 48 44 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(OC)c1 ZINC000880534933 FE On-Demand Mild TNIK 49 41 N#Cc1cc(NC(=O)NC[C@@H](O)C(F)(F)C(F)(F)F)ccn1 ZINC000880534946 DD On-Demand Mild ADRB1 43 32 N#Cc1cc(NC(=O)NC[C@H](O)C(F)(F)C(F)(F)F)ccn1 ZINC000880534950 DD On-Demand Mild ADRB1 43 32 N#Cc1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccn1 ZINC000880534955 DF On-Demand Mild EPHX2 15 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880534973 EF On-Demand Anodyne PPARG 73 41 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880534973 EF On-Demand Anodyne PPARA 74 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@H]21 ZINC000880534973 EF On-Demand Anodyne PDE8B 65 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880534974 EF On-Demand Anodyne PPARG 73 41 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880534974 EF On-Demand Anodyne PPARA 74 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@@H]2CCNC(=O)[C@@H]21 ZINC000880534974 EF On-Demand Anodyne PDE8B 65 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880534975 EF On-Demand Anodyne PPARG 73 41 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880534975 EF On-Demand Anodyne PPARA 74 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@@H]21 ZINC000880534975 EF On-Demand Anodyne PDE8B 65 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880534976 EF On-Demand Anodyne PPARG 73 41 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880534976 EF On-Demand Anodyne PPARA 74 40 Cc1oc(-c2ccccc2)nc1CN1CCC[C@H]2CCNC(=O)[C@H]21 ZINC000880534976 EF On-Demand Anodyne PDE8B 65 40 COC(=O)CCCCN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880535050 DH On-Demand Anodyne ADRB1 19 41 COC(=O)CCCCN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880535051 DH On-Demand Anodyne ADRB1 19 41 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880535053 ED On-Demand Mild EPHX2 31 40 CC(C)(C)OC(=O)N1CCCC2(CN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880535062 FF On-Demand Mild GPR119 18 45 N#Cc1cc(NC(=O)N2CCC[C@](F)(c3ccccc3)C2)ccn1 ZINC000880535076 DG On-Demand Mild EPHX2 28 47 N#Cc1cc(NC(=O)N2CCC[C@@](F)(c3ccccc3)C2)ccn1 ZINC000880535077 DG On-Demand Mild EPHX2 28 47 N#Cc1cc(NC(=O)NCCCCC2CC2)ccn1 ZINC000880535106 CF On-Demand Mild CCR3 34 46 CN1CCN(C(=O)Nc2ccnc(C#N)c2)CCC1(C)C ZINC000880535107 CD On-Demand Mild PDGFRB 40 38 CC[C@H](C)NC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880535135 DG On-Demand Anodyne ADRB1 18 41 CC[C@H](C)NC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880535135 DG On-Demand Anodyne ADRB3 27 41 CC[C@H](C)NC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880535136 DG On-Demand Anodyne ADRB1 18 41 CC[C@H](C)NC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880535136 DG On-Demand Anodyne ADRB3 27 41 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)NCCCN1CCCC1=O ZINC000880535194 FE On-Demand Anodyne TYRO3 19 44 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)NCCCN1CCCC1=O ZINC000880535195 FE On-Demand Anodyne TYRO3 19 44 O=C(N[C@H](C1CCOCC1)C1CC1)c1coc(-c2ccccn2)n1 ZINC000880535236 EF On-Demand Anodyne MAPK1 45 33 O=C(N[C@@H](C1CCOCC1)C1CC1)c1coc(-c2ccccn2)n1 ZINC000880535237 EF On-Demand Anodyne MAPK1 45 33 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c1 ZINC000880535289 FF On-Demand Mild PDGFRB 48 38 FC(F)[C@H](NCCN1CCOCC1)c1cccc(Cl)c1 ZINC000880535291 DF On-Demand Anodyne CASR 41 36 FC(F)[C@@H](NCCN1CCOCC1)c1cccc(Cl)c1 ZINC000880535292 DF On-Demand Anodyne CASR 41 36 COC(=O)[C@@H](CCF)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880535295 ED On-Demand Anodyne KCNQ2 63 36 COC(=O)[C@@H](CCF)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880535295 ED On-Demand Anodyne FURIN 51 33 COC(=O)[C@@H](CCF)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880535295 ED On-Demand Anodyne POLG_WNV 47 35 Cn1c(=O)c(CN2C[C@@H]3CC[C@H]2c2ccccc23)cc2ccccc21 ZINC000880535367 EH On-Demand Anodyne NPSR1 32 41 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)c1ccc(OC(F)F)c(Cl)c1 ZINC000880535368 DF On-Demand Anodyne PDE4D 16 41 N#Cc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)ccn1 ZINC000880535374 EF On-Demand Mild EPHX2 31 40 N#Cc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)ccn1 ZINC000880535374 EF On-Demand Mild TRPM8 37 51 N#Cc1cc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)ccn1 ZINC000880535381 EF On-Demand Mild EPHX2 31 40 N#Cc1cc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)ccn1 ZINC000880535381 EF On-Demand Mild TRPM8 37 51 N#Cc1cc(NC(=O)NN2CCCC2)ccn1 ZINC000880535383 BD On-Demand Mild TYK2 41 36 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880535385 EE On-Demand Anodyne DRD4 46 37 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880535385 EE On-Demand Anodyne PLD1 40 37 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880535385 EE On-Demand Anodyne PLD2 57 37 NC(=O)[C@H]1C[C@@H](NC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880535397 DC On-Demand Anodyne KCNQ2 44 39 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1cccnc1 ZINC000880535418 DG On-Demand Anodyne CHRNA7 26 41 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1cccnc1 ZINC000880535418 DG On-Demand Anodyne NAMPT 28 42 CC(C)(C)OC(=O)N1CC[C@H](C2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880535446 GG On-Demand Mild GPR119 49 58 CC(C)(C)OC(=O)N1CC[C@@H](C2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880535449 GG On-Demand Mild GPR119 49 58 N#Cc1cc(NC(=O)N2CCCCCCCC2)ccn1 ZINC000880535462 CG On-Demand Mild TYK2 46 37 CC(C)(C)OC(=O)NCc1nc(CN2C[C@@H]3CC[C@H]2c2ccccc23)no1 ZINC000880535473 FH On-Demand Anodyne PANC 50 33 O=C(N[C@H](C1CCOCC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535520 EF On-Demand Anodyne GABRA1 15 41 O=C(N[C@H](C1CCOCC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535520 EF On-Demand Anodyne GABRA2 15 41 O=C(N[C@@H](C1CCOCC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535521 EF On-Demand Anodyne GABRA1 15 41 O=C(N[C@@H](C1CCOCC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535521 EF On-Demand Anodyne GABRA2 15 41 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)C[C@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535522 FD On-Demand Anodyne CTSK 15 42 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)C[C@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535522 FD On-Demand Anodyne CTSL 24 42 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)C[C@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535523 FD On-Demand Anodyne CTSK 15 42 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)C[C@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535523 FD On-Demand Anodyne CTSL 24 42 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)C[C@@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535524 FD On-Demand Anodyne CTSK 15 42 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)C[C@@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535524 FD On-Demand Anodyne CTSL 24 42 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)C[C@@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535525 FD On-Demand Anodyne CTSK 15 42 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)C[C@@H]1CCNC1=O)C2)OCc1ccccc1 ZINC000880535525 FD On-Demand Anodyne CTSL 24 42 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne ACE 16 44 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne CTSB 22 47 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne CTSK 24 47 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne CTSL 33 47 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne CAPN2 50 33 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne NAAA 46 41 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535540 ED On-Demand Anodyne Q9NAW4_PLAFA 37 41 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne ACE 16 44 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne CTSB 22 47 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne CTSK 24 47 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne CTSL 33 47 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne CAPN2 50 33 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne NAAA 46 41 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)COC1CC1)C2)OCc1ccccc1 ZINC000880535541 ED On-Demand Anodyne Q9NAW4_PLAFA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@]1(C)C[C@]1(F)Cl ZINC000880535542 FF On-Demand Anodyne PAPA1_CARPA 38 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@]1(C)C[C@]1(F)Cl ZINC000880535543 FF On-Demand Anodyne PAPA1_CARPA 38 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@]1(C)C[C@@]1(F)Cl ZINC000880535544 FF On-Demand Anodyne PAPA1_CARPA 38 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@]1(C)C[C@@]1(F)Cl ZINC000880535545 FF On-Demand Anodyne PAPA1_CARPA 38 45 CON(C)CCNC(=O)Nc1ccnc(C#N)c1 ZINC000880535566 BC On-Demand Mild ADRB1 42 31 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)c1c[nH]cc1C1CC1)C2)OCc1ccccc1 ZINC000880535577 FG On-Demand Anodyne CTSK 15 41 O=C(N[C@H]1[C@H]2C[C@H]1N(C(=O)c1c[nH]cc1C1CC1)C2)OCc1ccccc1 ZINC000880535577 FG On-Demand Anodyne CTSL 19 41 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)c1c[nH]cc1C1CC1)C2)OCc1ccccc1 ZINC000880535578 FG On-Demand Anodyne CTSK 15 41 O=C(N[C@@H]1[C@H]2C[C@H]1N(C(=O)c1c[nH]cc1C1CC1)C2)OCc1ccccc1 ZINC000880535578 FG On-Demand Anodyne CTSL 19 41 COC(=O)[C@@H](CCF)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535581 DD On-Demand Anodyne GABRA1 15 44 COC(=O)[C@@H](CCF)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880535581 DD On-Demand Anodyne MPO 64 37 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535601 FE On-Demand Mild EPHX2 23 40 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535601 FE On-Demand Mild TRPM8 31 42 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535602 FE On-Demand Mild EPHX2 23 40 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535602 FE On-Demand Mild TRPM8 31 42 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535603 FE On-Demand Mild EPHX2 23 40 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535603 FE On-Demand Mild TRPM8 31 42 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535604 FE On-Demand Mild EPHX2 23 40 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)ccn1 ZINC000880535604 FE On-Demand Mild TRPM8 31 42 COC(=O)[C@@H](CNC(=O)[C@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535645 EF On-Demand Anodyne MTNR1A 41 45 COC(=O)[C@@H](CNC(=O)[C@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535645 EF On-Demand Anodyne MTNR1B 37 45 COC(=O)[C@@H](CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535647 EF On-Demand Anodyne MTNR1A 41 45 COC(=O)[C@@H](CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535647 EF On-Demand Anodyne MTNR1B 37 45 COC(=O)[C@H](CNC(=O)[C@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535649 EF On-Demand Anodyne MTNR1A 41 45 COC(=O)[C@H](CNC(=O)[C@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535649 EF On-Demand Anodyne MTNR1B 37 45 COC(=O)[C@H](CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535651 EF On-Demand Anodyne MTNR1A 41 45 COC(=O)[C@H](CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)CC1CC1 ZINC000880535651 EF On-Demand Anodyne MTNR1B 37 45 N#Cc1cc(NC(=O)NCCCCCCO)ccn1 ZINC000880535653 CD On-Demand Mild ADRB1 42 32 CC(C)(C)OC(=O)N1C[C@@H]2CCN(C(=O)Nc3ccnc(C#N)c3)[C@@H]2C1 ZINC000880535666 FE On-Demand Mild GPR119 29 51 N#Cc1cc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)ccn1 ZINC000880535695 FF On-Demand Mild CACNA1H 45 42 N#Cc1cc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)ccn1 ZINC000880535695 FF On-Demand Mild S1PR2 29 42 N#Cc1cc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)ccn1 ZINC000880535695 FF On-Demand Mild KISS1R 54 33 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880535696 GG On-Demand Mild EPHX2 27 43 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880535696 GG On-Demand Mild GPR119 18 46 CC(C)(C)OC(=O)N1C[C@H]2CC[C@H]1CN2C(=O)Nc1ccnc(C#N)c1 ZINC000880535699 FF On-Demand Mild GPR119 19 41 CC(C)(C)OC(=O)N1CC[C@H]([C@@H]2CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880535700 GG On-Demand Mild GPR119 41 54 CC(C)(C)OC(=O)N1CC[C@H]([C@H]2CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880535701 GG On-Demand Mild GPR119 41 54 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H]2CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880535702 GG On-Demand Mild GPR119 41 54 CC(C)(C)OC(=O)N1CC[C@@H]([C@H]2CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880535703 GG On-Demand Mild GPR119 41 54 CC[C@H]1CN(C(=O)CCCCc2ccc(OC)c(OC)c2)[C@@H](C)CO1 ZINC000880535719 EG On-Demand Anodyne FKBP1A 45 40 CC[C@H]1CN(C(=O)CCCCc2ccc(OC)c(OC)c2)[C@H](C)CO1 ZINC000880535721 EG On-Demand Anodyne FKBP1A 45 40 O=C(NCCN1CCCC1=O)c1coc(-c2ccccn2)n1 ZINC000880535725 DD On-Demand Anodyne TYRO3 19 40 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535815 DC On-Demand Anodyne DRD4 40 31 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535815 DC On-Demand Anodyne PLD1 69 39 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535815 DC On-Demand Anodyne PLD2 89 39 O=C1CC[C@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535818 DC On-Demand Anodyne DRD4 40 31 O=C1CC[C@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535818 DC On-Demand Anodyne PLD1 69 39 O=C1CC[C@H](c2ccc(C(=O)NCCN3CCCC3=O)cc2)N1 ZINC000880535818 DC On-Demand Anodyne PLD2 89 39 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCn1ccnc1 ZINC000880535820 CF On-Demand Anodyne CYP19A1 15 47 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCn1ccnc1 ZINC000880535820 CF On-Demand Anodyne CYP11B1 26 40 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCn1ccnc1 ZINC000880535820 CF On-Demand Anodyne TBXAS1 27 43 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCn1ccnc1 ZINC000880535820 CF On-Demand Anodyne CYP11B2 16 40 O=C(NCCN1CCCC1=O)c1cc2ccccc2cc1F ZINC000880535831 DE On-Demand Anodyne DRD4 41 32 O=C(NCCN1CCCC1=O)c1cc2ccccc2cc1F ZINC000880535831 DE On-Demand Anodyne PLD1 66 37 O=C(NCCN1CCCC1=O)c1cc2ccccc2cc1F ZINC000880535831 DE On-Demand Anodyne PLD2 93 41 O=C(NCCN1CCCC1=O)c1cc2ccccc2cc1F ZINC000880535831 DE On-Demand Anodyne TYRO3 22 47 O=C(NCCN1CCCC1=O)c1cc2ccccc2cc1F ZINC000880535831 DE On-Demand Anodyne POLR1A 62 42 N#Cc1cc(NC(=O)N[C@@H]2CC[C@H]2O)ccn1 ZINC000880535838 BC On-Demand Mild TYK2 40 38 O=C(NCCN1CCCC1=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880535854 FE On-Demand Anodyne P2RX7 40 38 O=C(NCCN1CCCC1=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880535854 FE On-Demand Anodyne TYRO3 20 40 COc1cc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc(OC)c1OC ZINC000880535868 GE On-Demand Mild PDGFRB 68 50 COc1cc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc(OC)c1OC ZINC000880535868 GE On-Demand Mild PDGFRA 31 43 O=C(Cc1ccccc1N1CCCC1=O)NCCN1CCCC1=O ZINC000880535874 ED On-Demand Anodyne TYRO3 19 41 COc1ccccc1-c1ccc(C(=O)NCC[C@]2(C)C[C@@]2(F)Cl)c(O)n1 ZINC000880535897 GH On-Demand Anodyne HCN1 47 35 COc1ccccc1-c1ccc(C(=O)NCC[C@@]2(C)C[C@@]2(F)Cl)c(O)n1 ZINC000880535898 GH On-Demand Anodyne HCN1 47 35 COc1ccccc1-c1ccc(C(=O)NCC[C@@]2(C)C[C@]2(F)Cl)c(O)n1 ZINC000880535899 GH On-Demand Anodyne HCN1 47 35 COc1ccccc1-c1ccc(C(=O)NCC[C@]2(C)C[C@]2(F)Cl)c(O)n1 ZINC000880535901 GH On-Demand Anodyne HCN1 47 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535951 GG On-Demand Anodyne GHRHR 53 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535951 GG On-Demand Anodyne P2RY12 114 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535951 GG On-Demand Anodyne PGC 52 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535951 GG On-Demand Anodyne REN 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535951 GG On-Demand Anodyne FPR1 47 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535954 GG On-Demand Anodyne GHRHR 53 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535954 GG On-Demand Anodyne P2RY12 114 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535954 GG On-Demand Anodyne PGC 52 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535954 GG On-Demand Anodyne REN 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@@H](c2ccccc2)C1 ZINC000880535954 GG On-Demand Anodyne FPR1 47 36 CC(C)(C)N1CC[C@H](CNC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880535955 DE On-Demand Mild CACNA1I 41 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535956 GG On-Demand Anodyne GHRHR 53 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535956 GG On-Demand Anodyne P2RY12 114 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535956 GG On-Demand Anodyne PGC 52 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535956 GG On-Demand Anodyne REN 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535956 GG On-Demand Anodyne FPR1 47 36 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880535957 DE On-Demand Mild CACNA1I 41 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535958 GG On-Demand Anodyne GHRHR 53 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535958 GG On-Demand Anodyne P2RY12 114 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535958 GG On-Demand Anodyne PGC 52 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535958 GG On-Demand Anodyne REN 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCS[C@H](c2ccccc2)C1 ZINC000880535958 GG On-Demand Anodyne FPR1 47 36 C[C@@H]1C[C@H]1c1noc(CC2CCN(C(=O)CC[C@@H]3CC(C)(C)CO3)CC2)n1 ZINC000880535969 GH On-Demand Anodyne ETHR 41 35 N#Cc1cc(NC(=O)NCC[C@H]2CCSC2)ccn1 ZINC000880535970 CE On-Demand Mild PRMT3 24 41 N#Cc1cc(NC(=O)NCC[C@@H]2CCSC2)ccn1 ZINC000880535971 CE On-Demand Mild PRMT3 24 41 C[C@@H]1C[C@H]1c1noc(CC2CCN(C(=O)CC[C@H]3CC(C)(C)CO3)CC2)n1 ZINC000880535972 GH On-Demand Anodyne ETHR 41 35 CC(C)(C)OC(=O)N1C[C@@H](C(=O)N2CCC(Cn3cnnc3)CC2)C(C)(C)C1 ZINC000880535976 GE On-Demand Anodyne GPR119 32 41 CC(C)(C)OC(=O)N1C[C@H](C(=O)N2CCC(Cn3cnnc3)CC2)C(C)(C)C1 ZINC000880535978 GE On-Demand Anodyne GPR119 32 41 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)NCc1cccnc1 ZINC000880536032 EF On-Demand Anodyne NAMPT 53 41 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)NCc1cccnc1 ZINC000880536033 EF On-Demand Anodyne NAMPT 53 41 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA2 51 46 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA1 50 46 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA7 36 42 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA4 30 40 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA12 38 46 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA9 48 46 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CAH_METTE 19 41 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne NCE103 18 41 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne CA15 15 41 NS(=O)(=O)c1ccc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880536036 EF On-Demand Anodyne A6YCJ1_9METZ 22 41 Cc1cc(-c2nc(C)c(C(=O)N[C@@H]3C[C@H](C(N)=O)C3)s2)ccc1F ZINC000880536043 EF On-Demand Anodyne MAPK13 42 30 CC[C@H]1CN(C(=O)c2cccn3nccc23)[C@H](C)CO1 ZINC000880536052 CD On-Demand Anodyne HCRTR1 25 43 CC[C@H]1CN(C(=O)c2cccn3nccc23)[C@H](C)CO1 ZINC000880536052 CD On-Demand Anodyne HCRTR2 35 43 CC[C@@H]1CN(C(=O)c2cccn3nccc23)[C@@H](C)CO1 ZINC000880536054 CD On-Demand Anodyne HCRTR1 25 43 CC[C@@H]1CN(C(=O)c2cccn3nccc23)[C@@H](C)CO1 ZINC000880536054 CD On-Demand Anodyne HCRTR2 35 43 CC[C@H]1CN(C(=O)c2cccn3nccc23)[C@@H](C)CO1 ZINC000880536055 CD On-Demand Anodyne HCRTR1 25 43 CC[C@H]1CN(C(=O)c2cccn3nccc23)[C@@H](C)CO1 ZINC000880536055 CD On-Demand Anodyne HCRTR2 35 43 CC[C@@H]1CN(C(=O)c2cccn3nccc23)[C@H](C)CO1 ZINC000880536056 CD On-Demand Anodyne HCRTR1 25 43 CC[C@@H]1CN(C(=O)c2cccn3nccc23)[C@H](C)CO1 ZINC000880536056 CD On-Demand Anodyne HCRTR2 35 43 CC[C@H](NC(=O)COC1CC1)c1ccccc1F ZINC000880536061 CF On-Demand Anodyne TIMP3 73 34 CC(C)(C)OC(=O)N1CC[C@H]2CC[C@@H](C1)N2C(=O)Nc1ccnc(C#N)c1 ZINC000880536097 FF On-Demand Mild GPR119 51 51 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCCC1 ZINC000880536098 CG On-Demand Anodyne L3MBTL3 40 37 O=C(NCCN1CCCC1=O)c1cncc2[nH]ccc12 ZINC000880536106 CC On-Demand Anodyne TYRO3 21 42 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880536151 DD On-Demand Anodyne GABRA1 16 42 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880536151 DD On-Demand Anodyne GABRA2 16 42 NC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880536155 BD On-Demand Anodyne ADRB1 15 40 NC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880536157 BD On-Demand Anodyne ADRB1 15 40 O=C(NCCN1CCCC1=O)c1ncccc1-c1ccccn1 ZINC000880536160 DD On-Demand Anodyne TYRO3 19 41 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne HTR1A 39 41 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne DRD2 40 45 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne DRD4 40 32 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne ADRA1A 26 43 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne DRD3 53 45 COc1ccccc1-c1ccc(C(=O)NCCN2CCCC2=O)c(O)n1 ZINC000880536169 FD On-Demand Anodyne TYRO3 26 49 O=C(NCCN1CCCC1=O)c1cccc2nsnc12 ZINC000880536171 CD On-Demand Anodyne TYRO3 20 42 O=C(NCCN1CCCC1=O)c1cnc2cc[nH]c2c1 ZINC000880536174 CC On-Demand Anodyne DRD4 41 32 O=C(NCCN1CCCC1=O)c1cnc2cc[nH]c2c1 ZINC000880536174 CC On-Demand Anodyne PLD1 64 44 O=C(NCCN1CCCC1=O)c1cnc2cc[nH]c2c1 ZINC000880536174 CC On-Demand Anodyne PLD2 95 44 O=C(NCCN1CCCC1=O)c1cnc2cc[nH]c2c1 ZINC000880536174 CC On-Demand Anodyne TYRO3 20 43 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccn1 ZINC000880536175 DE On-Demand Mild CACNA1H 37 40 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)C[C@@](C)(F)C1 ZINC000880536177 GF On-Demand Mild GPR119 29 48 CC(C)(C(=O)NCCN1CCCC1=O)c1ccc(C(F)(F)F)cc1 ZINC000880536179 EF On-Demand Anodyne EPHX2 18 46 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)C[C@](C)(F)C1 ZINC000880536183 GF On-Demand Mild GPR119 29 48 COCCCCN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880536184 BG On-Demand Anodyne UGCG 44 34 COCCCCN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880536184 BG On-Demand Anodyne GBA2 51 34 COC(=O)C1CCN(C(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536185 FF On-Demand Anodyne SLC6A3 16 48 COC(=O)C1CCN(C(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536185 FF On-Demand Anodyne FDFT1 28 42 COC(=O)C1CCN(C(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536185 FF On-Demand Anodyne PTR1 44 31 COC(=O)C1CCN(C(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536187 FF On-Demand Anodyne SLC6A3 16 48 COC(=O)C1CCN(C(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536187 FF On-Demand Anodyne FDFT1 28 42 COC(=O)C1CCN(C(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880536187 FF On-Demand Anodyne PTR1 44 31 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCC1 ZINC000880536202 CF On-Demand Anodyne PREP 43 35 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCC1 ZINC000880536202 CF On-Demand Anodyne L3MBTL3 46 38 CN(CC1CCN(C[C@H](O)c2ccccc2)CC1)C(=O)Nc1ccnc(C#N)c1 ZINC000880536231 GF On-Demand Mild OPRK1 26 40 CN(CC1CCN(C[C@H](O)c2ccccc2)CC1)C(=O)Nc1ccnc(C#N)c1 ZINC000880536231 GF On-Demand Mild CCR3 23 43 CN(CC1CCN(C[C@@H](O)c2ccccc2)CC1)C(=O)Nc1ccnc(C#N)c1 ZINC000880536232 GF On-Demand Mild OPRK1 26 40 CN(CC1CCN(C[C@@H](O)c2ccccc2)CC1)C(=O)Nc1ccnc(C#N)c1 ZINC000880536232 GF On-Demand Mild CCR3 23 43 NC(=O)c1ccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1Cl ZINC000880536252 GH On-Demand Anodyne AVPR2 41 34 Oc1nc(CCN2C[C@@H]3CC[C@H]2c2ccccc23)nc2ccccc12 ZINC000880536269 EH On-Demand Anodyne TNKS 15 40 N#Cc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)ccn1 ZINC000880536282 EF On-Demand Mild EPHX2 24 55 N#Cc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)ccn1 ZINC000880536283 EF On-Demand Mild EPHX2 24 55 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CC1)CC2(F)F ZINC000880536294 CF On-Demand Anodyne ACACA 43 53 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CC1)CC2(F)F ZINC000880536294 CF On-Demand Anodyne ACACB 29 53 CNC(=O)[C@@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)c1ccccc1 ZINC000880536296 FF On-Demand Anodyne BIRC8 44 30 COc1ccc(N2CC[C@H](NC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880536313 EE On-Demand Mild EPHX2 40 37 COc1ccc(N2CC[C@H](NC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880536313 EE On-Demand Mild PDGFRA 34 41 COc1ccc(N2CC[C@H](NC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880536313 EE On-Demand Mild MCHR1 15 41 CC(C)(C)OC(=O)N1[C@H]2CC[C@H]1CN(C(=O)Nc1ccnc(C#N)c1)CC2 ZINC000880536343 FF On-Demand Mild GPR119 38 49 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@]1(F)Cl)C2 ZINC000880536355 EH On-Demand Anodyne NQO2 32 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@]1(F)Cl)C2 ZINC000880536355 EH On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@]1(F)Cl)C2 ZINC000880536355 EH On-Demand Anodyne MTNR1B 35 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@]1(F)Cl)C2 ZINC000880536357 EH On-Demand Anodyne NQO2 32 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@]1(F)Cl)C2 ZINC000880536357 EH On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@]1(F)Cl)C2 ZINC000880536357 EH On-Demand Anodyne MTNR1B 35 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536358 EH On-Demand Anodyne NQO2 32 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536358 EH On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536358 EH On-Demand Anodyne MTNR1B 35 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536359 EH On-Demand Anodyne NQO2 32 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536359 EH On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)C[C@@]1(F)Cl)C2 ZINC000880536359 EH On-Demand Anodyne MTNR1B 35 41 COC(=O)[C@@H](CCF)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880536394 EF On-Demand Anodyne PDE4D 18 41 Cc1coc(C(=O)N2C[C@H]3C[C@H]2[C@@H]3NC(=O)OCc2ccccc2)c1 ZINC000880536409 EF On-Demand Anodyne NAAA 58 37 Cc1coc(C(=O)N2C[C@H]3C[C@H]2[C@H]3NC(=O)OCc2ccccc2)c1 ZINC000880536410 EF On-Demand Anodyne NAAA 58 37 CC(C)(C)OC(=O)N1CC[C@]2(CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536419 GG On-Demand Mild EPHX2 30 41 CC(C)(C)OC(=O)N1CC[C@@]2(CCCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536420 GG On-Demand Mild EPHX2 30 41 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild F2 15 41 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild P2RY12 137 38 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild MC4R 69 46 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTRA_BOVIN 45 34 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild KLK3 65 34 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTSB 69 46 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild TRY2_BOVIN 60 34 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild PAPA1_CARPA 57 48 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CYSP_TRYCR 75 41 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTSK 37 48 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTSL 58 48 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CAPNS1 67 38 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CELA2A 52 34 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTSS 30 48 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CAPN1 80 40 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CAPN2 118 44 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild TGM2 29 53 N#Cc1ccnc(N2CCN(C(=O)[C@@H](Cc3ccccc3)NC(=O)OCc3ccccc3)CC2)c1 ZINC000880536502 JG On-Demand Mild CTRB_BOVIN 47 33 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880536526 DG On-Demand Anodyne KCNQ2 32 41 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880536526 DG On-Demand Anodyne DPP7 40 42 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880536528 DG On-Demand Anodyne KCNQ2 32 41 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCCC1 ZINC000880536528 DG On-Demand Anodyne DPP7 40 42 COC(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)n1 ZINC000880536536 FF On-Demand Anodyne HTR1F 43 33 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CCCC1=O ZINC000880536540 DE On-Demand Anodyne NQO2 20 40 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CCCC1=O ZINC000880536540 DE On-Demand Anodyne TYRO3 18 42 O=C(CC[C@H]1CCc2ccccc21)NCCN1CCCC1=O ZINC000880536541 DE On-Demand Anodyne NQO2 20 40 O=C(CC[C@H]1CCc2ccccc21)NCCN1CCCC1=O ZINC000880536541 DE On-Demand Anodyne TYRO3 18 42 O=C(NCCN1CCCC1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880536542 DD On-Demand Anodyne PLD1 81 46 O=C(NCCN1CCCC1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880536542 DD On-Demand Anodyne PLD2 103 46 O=C(NCCN1CCCC1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880536542 DD On-Demand Anodyne TYRO3 20 40 CN1CC[C@@H](CNC(=O)Nc2ccnc(C#N)c2)[C@@H]1c1cccnc1 ZINC000880536557 EE On-Demand Mild NAMPT 45 37 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)CC1 ZINC000880536608 GG On-Demand Mild EPHX2 33 45 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)CC1 ZINC000880536608 GG On-Demand Mild GPR119 25 48 CS(=O)(=O)N1CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880536638 FC On-Demand Anodyne GABRA1 16 41 CS(=O)(=O)N1CC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880536641 FC On-Demand Anodyne GABRA1 16 41 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cccc3nsnc23)C1 ZINC000880536650 EC On-Demand Anodyne HTR4 15 45 CS(=O)(=O)N1CC[C@H](NC(=O)c2cccc3nsnc23)C1 ZINC000880536651 EC On-Demand Anodyne HTR4 15 45 CC[C@H]1CN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)[C@@H](C)CO1 ZINC000880536716 EH On-Demand Anodyne HCRTR1 18 45 CC[C@H]1CN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)[C@@H](C)CO1 ZINC000880536716 EH On-Demand Anodyne HCRTR2 22 45 CC[C@H]1CN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)[C@H](C)CO1 ZINC000880536717 EH On-Demand Anodyne HCRTR1 18 45 CC[C@H]1CN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)[C@H](C)CO1 ZINC000880536717 EH On-Demand Anodyne HCRTR2 22 45 COC(=O)[C@@H](CCF)NC(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1 ZINC000880536730 FF On-Demand Anodyne CTSL 32 40 COC(=O)[C@@H](CCF)NC(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1 ZINC000880536730 FF On-Demand Anodyne CTSS 26 40 COC(=O)[C@@H](CCF)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880536759 DD On-Demand Anodyne FPGS 48 31 COC(=O)[C@@H](CCF)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880536761 DD On-Demand Anodyne FPGS 48 31 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536789 FG On-Demand Anodyne PAPA1_CARPA 40 48 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536789 FG On-Demand Anodyne CTSK 22 41 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536789 FG On-Demand Anodyne TACR3 16 40 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536789 FG On-Demand Anodyne FPR1 50 41 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536790 FG On-Demand Anodyne PAPA1_CARPA 40 48 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536790 FG On-Demand Anodyne CTSK 22 41 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536790 FG On-Demand Anodyne TACR3 16 40 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880536790 FG On-Demand Anodyne FPR1 50 41 O=C(c1ccccc1)N1CC[C@H](CN2C[C@@H]3CC[C@H]2c2ccccc23)C1 ZINC000880536803 EI On-Demand Anodyne L3MBTL3 83 41 O=C(c1ccccc1)N1CC[C@@H](CN2C[C@@H]3CC[C@H]2c2ccccc23)C1 ZINC000880536815 EI On-Demand Anodyne L3MBTL3 83 41 O=C(CCN[C@@H](c1cccc(Cl)c1)C(F)F)NC1CCCC1 ZINC000880536837 EH On-Demand Anodyne CNR1 15 42 O=C(CCN[C@H](c1cccc(Cl)c1)C(F)F)NC1CCCC1 ZINC000880536839 EH On-Demand Anodyne CNR1 15 42 N#Cc1cc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)ccn1 ZINC000880536840 FD On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)ccn1 ZINC000880536842 FD On-Demand Mild RBP4 47 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN1CCCC1=O ZINC000880536843 EC On-Demand Anodyne PAPA1_CARPA 40 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN1CCCC1=O ZINC000880536844 EC On-Demand Anodyne PAPA1_CARPA 40 47 N#Cc1cc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)ccn1 ZINC000880536845 FD On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)ccn1 ZINC000880536847 FD On-Demand Mild RBP4 47 35 NC(=O)[C@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880536849 DD On-Demand Anodyne PDE4D 18 44 NC(=O)[C@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880536849 DD On-Demand Anodyne EZH2 42 40 O=C(NCCN1CCCC1=O)c1cnc(CC2CC2)s1 ZINC000880536851 CD On-Demand Anodyne SIRT3 46 35 O=C(NCCN1CCCC1=O)c1cnc(CC2CC2)s1 ZINC000880536851 CD On-Demand Anodyne SIRT2 47 35 O=C(NCCN1CCCC1=O)c1cnc(CC2CC2)s1 ZINC000880536851 CD On-Demand Anodyne SIRT1 42 34 O=C(NCCN1CCCC1=O)c1cnc(CC2CC2)s1 ZINC000880536851 CD On-Demand Anodyne TYRO3 20 41 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne CELA1 20 41 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne PREP 29 42 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne LGMN 62 38 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne GHSR 24 40 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne KLK5 42 41 O=C(NCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880536904 GD On-Demand Anodyne Q9NAW4_PLAFA 37 42 C[C@@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccnc(C#N)c1 ZINC000880536917 EE On-Demand Mild GPR119 38 48 O=C1CCCN1CCCN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880536932 DG On-Demand Anodyne TYRO3 17 41 O=C1CCCN1CCCN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880536933 DG On-Demand Anodyne TYRO3 17 41 N#Cc1cc(NC(=O)NC23CCC(CC2)C3)ccn1 ZINC000880536934 CE On-Demand Mild EPHX2 48 50 C#CCOCCNC(=O)Nc1ccnc(C#N)c1 ZINC000880536951 BC On-Demand Mild ADRB1 42 32 O=C(NCCN1CCCC1=O)c1cccn2nccc12 ZINC000880536980 CC On-Demand Anodyne TYRO3 21 43 Cn1nnc(C(=O)N2CCO[C@H]3CCN(Cc4ccccc4)C[C@H]32)n1 ZINC000880536981 EC On-Demand Anodyne CYP2J2 42 30 Cn1nnc(C(=O)N2CCO[C@H]3CCN(Cc4ccccc4)C[C@@H]32)n1 ZINC000880536982 EC On-Demand Anodyne CYP2J2 42 30 Cn1nnc(C(=O)N2CCO[C@@H]3CCN(Cc4ccccc4)C[C@H]32)n1 ZINC000880536983 EC On-Demand Anodyne CYP2J2 42 30 Cn1nnc(C(=O)N2CCO[C@@H]3CCN(Cc4ccccc4)C[C@@H]32)n1 ZINC000880536984 EC On-Demand Anodyne CYP2J2 42 30 CC(C)(C)OC(=O)N1CC[C@]2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536985 FF On-Demand Mild EPHX2 32 43 CC(C)(C)OC(=O)N1CC[C@]2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536985 FF On-Demand Mild GPR119 18 46 CC(C)(C)OC(=O)N1CC[C@@]2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536987 FF On-Demand Mild EPHX2 32 43 CC(C)(C)OC(=O)N1CC[C@@]2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880536987 FF On-Demand Mild GPR119 18 46 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536991 ED On-Demand Anodyne DRD4 43 41 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536991 ED On-Demand Anodyne SIGMAR1 47 45 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536991 ED On-Demand Anodyne SLC18A3 28 40 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536994 ED On-Demand Anodyne DRD4 43 41 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536994 ED On-Demand Anodyne SIGMAR1 47 45 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880536994 ED On-Demand Anodyne SLC18A3 28 40 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536996 ED On-Demand Anodyne DRD4 43 41 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536996 ED On-Demand Anodyne SIGMAR1 47 45 O=C(COC1CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536996 ED On-Demand Anodyne SLC18A3 28 40 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536997 ED On-Demand Anodyne DRD4 43 41 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536997 ED On-Demand Anodyne SIGMAR1 47 45 O=C(COC1CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880536997 ED On-Demand Anodyne SLC18A3 28 40 C#CCCCNC(=O)Nc1ccnc(C#N)c1 ZINC000880537051 BD On-Demand Mild ADRB1 40 30 N#Cc1cc(NC(=O)N2CCCC[C@H]2c2ccccc2)ccn1 ZINC000880537064 DH On-Demand Mild CPT1A 77 37 N#Cc1cc(NC(=O)N2CCCC[C@@H]2c2ccccc2)ccn1 ZINC000880537065 DH On-Demand Mild CPT1A 77 37 O=C(NCC[C@]1(O)CCOC1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880537077 DC On-Demand Anodyne PLD2 57 39 O=C(NCC[C@@]1(O)CCOC1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880537078 DC On-Demand Anodyne PLD2 57 39 FC(F)[C@@H](NCCCN1CCOCC1)c1cccc(Cl)c1 ZINC000880537087 DF On-Demand Anodyne HRP1_PLAFA 47 31 FC(F)[C@H](NCCCN1CCOCC1)c1cccc(Cl)c1 ZINC000880537088 DF On-Demand Anodyne HRP1_PLAFA 47 31 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880537089 DF On-Demand Anodyne KCNQ2 35 42 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880537089 DF On-Demand Anodyne DPP7 33 41 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880537090 DF On-Demand Anodyne KCNQ2 35 42 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)N1CCCC1 ZINC000880537090 DF On-Demand Anodyne DPP7 33 41 O[C@@H](CN[C@H](c1cccc(Cl)c1)C(F)F)COC1CCOCC1 ZINC000880537117 EF On-Demand Anodyne MAPK1 44 39 O[C@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)COC1CCOCC1 ZINC000880537118 EF On-Demand Anodyne MAPK1 44 39 O[C@H](CN[C@H](c1cccc(Cl)c1)C(F)F)COC1CCOCC1 ZINC000880537119 EF On-Demand Anodyne MAPK1 44 39 O[C@@H](CN[C@@H](c1cccc(Cl)c1)C(F)F)COC1CCOCC1 ZINC000880537120 EF On-Demand Anodyne MAPK1 44 39 N#Cc1cc(NC(=O)NCC[C@H]2CCCS2)ccn1 ZINC000880537128 CE On-Demand Mild PRMT3 25 41 N#Cc1cc(NC(=O)NCC[C@@H]2CCCS2)ccn1 ZINC000880537129 CE On-Demand Mild PRMT3 25 41 CS(=O)(=O)N1CC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537149 DC On-Demand Anodyne HTR4 15 40 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537150 DC On-Demand Anodyne HTR4 15 40 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild CTSB 21 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild CTSK 25 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild CTSL 33 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild CAPN2 43 33 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild TGM2 37 41 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild NPR 42 33 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild F13A1 31 41 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880537159 EG On-Demand Mild NAAA 57 43 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild CTSB 21 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild CTSK 25 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild CTSL 33 42 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild CAPN2 43 33 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild TGM2 37 41 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild NPR 42 33 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild F13A1 31 41 C=CC(C)(C)CC(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880537160 EG On-Demand Mild NAAA 57 43 CC(C)(C)OC(=O)N1CC[C@H]2CN(C(=O)Nc3ccnc(C#N)c3)CC[C@@H]21 ZINC000880537183 FF On-Demand Mild GPR119 31 51 CC(C)(C)OC(=O)N1CC[C@@H]2CN(C(=O)Nc3ccnc(C#N)c3)CC[C@@H]21 ZINC000880537184 FF On-Demand Mild GPR119 31 51 CC(C)(C)OC(=O)N1CC[C@@H]2CN(C(=O)Nc3ccnc(C#N)c3)CC[C@H]21 ZINC000880537185 FF On-Demand Mild GPR119 31 51 CC(C)(C)OC(=O)N1CC[C@H]2CN(C(=O)Nc3ccnc(C#N)c3)CC[C@H]21 ZINC000880537186 FF On-Demand Mild GPR119 31 51 NC(=O)[C@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537203 CC On-Demand Anodyne JAK3 18 44 NC(=O)[C@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537203 CC On-Demand Anodyne JAK1 15 44 NC(=O)[C@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537203 CC On-Demand Anodyne TYK2 22 44 NC(=O)[C@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880537203 CC On-Demand Anodyne EPHB3 37 41 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)c1cccc2nsnc12 ZINC000880537204 CD On-Demand Anodyne HTR3A 26 41 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880537216 FE On-Demand Anodyne GRIN2B 18 40 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880537216 FE On-Demand Anodyne PREP 27 40 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880537216 FE On-Demand Anodyne LGMN 52 38 O=C(N[C@@H]1C[C@H]2CC[C@@H]1O2)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880537216 FE On-Demand Anodyne Q9NAW4_PLAFA 39 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](C(N)=O)C1)C2 ZINC000880537226 DD On-Demand Anodyne NQO2 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](C(N)=O)C1)C2 ZINC000880537226 DD On-Demand Anodyne MTNR1A 33 42 CC[C@H](NC(=O)CN1CCCCS1(=O)=O)c1ccccc1F ZINC000880537240 ED On-Demand Anodyne KCNQ2 29 41 O=C(NCCN1CCCC1=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880537243 DD On-Demand Anodyne GABRA1 16 46 O=C(NCCN1CCCC1=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880537243 DD On-Demand Anodyne MPO 40 35 O=C(NCCN1CCCC1=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880537243 DD On-Demand Anodyne PLD2 43 33 Cc1cnc(Cl)c(C(=O)NCCN2CCCC2=O)c1 ZINC000880537289 CD On-Demand Anodyne DRD4 41 31 Cc1cnc(Cl)c(C(=O)NCCN2CCCC2=O)c1 ZINC000880537289 CD On-Demand Anodyne TYRO3 25 43 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccnc(C#N)c2)C1 ZINC000880537314 ED On-Demand Mild EPHX2 34 43 O=C(NCCN1CCCC1=O)c1ncsc1C1CC1 ZINC000880537362 CD On-Demand Anodyne TYRO3 19 40 CC(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880537363 EH On-Demand Anodyne CCR3 22 42 CC(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880537363 EH On-Demand Anodyne CCKBR 42 38 CC(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880537363 EH On-Demand Anodyne KCNK3 55 36 N#Cc1cc(NC(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)ccn1 ZINC000880537420 FG On-Demand Mild EPHX2 17 46 N#Cc1cc(NC(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)ccn1 ZINC000880537424 FG On-Demand Mild EPHX2 17 46 N#Cc1cc(NC(=O)N2C[C@@H]3[C@H](C2)C3(F)F)ccn1 ZINC000880537426 CD On-Demand Mild TYK2 42 36 N#Cc1cc(NC(=O)N2C[C@@H]3[C@@H](C2)C3(F)F)ccn1 ZINC000880537427 CD On-Demand Mild TYK2 42 36 N#Cc1cc(NC(=O)N2C[C@H]3[C@H](C2)C3(F)F)ccn1 ZINC000880537428 CD On-Demand Mild TYK2 42 36 N#Cc1cc(NC(=O)N2CCN(c3nc(F)c(F)cc3F)CC2)ccn1 ZINC000880537451 FE On-Demand Mild PDGFRB 53 42 O=C([C@@H]1CCc2nncn2CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880537471 GD On-Demand Anodyne SIGMAR1 24 45 O=C([C@@H]1CCc2nncn2CC1)N1CCO[C@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880537472 GD On-Demand Anodyne SIGMAR1 24 45 O=C([C@@H]1CCc2nncn2CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@@H]21 ZINC000880537473 GD On-Demand Anodyne SIGMAR1 24 45 O=C([C@@H]1CCc2nncn2CC1)N1CCO[C@@H]2CCN(Cc3ccccc3)C[C@H]21 ZINC000880537474 GD On-Demand Anodyne SIGMAR1 24 45 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880537488 FC On-Demand Anodyne CCR3 32 49 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880537490 FC On-Demand Anodyne CCR3 32 49 Cc1ncc(CC(=O)N2C[C@H]3C[C@H]2[C@H]3NC(=O)OCc2ccccc2)o1 ZINC000880537506 FE On-Demand Anodyne NAAA 48 39 Cc1ncc(CC(=O)N2C[C@H]3C[C@H]2[C@@H]3NC(=O)OCc2ccccc2)o1 ZINC000880537508 FE On-Demand Anodyne NAAA 48 39 CC(C)(C)OC(=O)N1[C@H]2CC[C@H]1CN(C(=O)Nc1ccnc(C#N)c1)C2 ZINC000880537517 FF On-Demand Mild GPR119 31 48 CS(=O)(=O)N1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537521 FD On-Demand Anodyne HTR4 26 41 CS(=O)(=O)N1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537521 FD On-Demand Anodyne UTS2R 29 50 CS(=O)(=O)N1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537521 FD On-Demand Anodyne SLC6A5 28 41 CS(=O)(=O)N1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537521 FD On-Demand Anodyne EZH2 41 38 CS(=O)(=O)N1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537522 FD On-Demand Anodyne HTR4 26 41 CS(=O)(=O)N1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537522 FD On-Demand Anodyne UTS2R 29 50 CS(=O)(=O)N1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537522 FD On-Demand Anodyne SLC6A5 28 41 CS(=O)(=O)N1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880537522 FD On-Demand Anodyne EZH2 41 38 N#Cc1cc(NC(=O)NCC[S@](=O)CC(F)(F)F)ccn1 ZINC000880537524 DD On-Demand Mild ADRB1 40 30 N#Cc1cc(NC(=O)NCC[S@@](=O)CC(F)(F)F)ccn1 ZINC000880537528 DD On-Demand Mild ADRB1 40 30 Oc1nc(CN2C[C@@H]3CC[C@H]2c2ccccc23)nc2c1COCC2 ZINC000880537532 DF On-Demand Anodyne WNT3A 52 33 CS(=O)(=O)N1CC[C@H](NC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880537548 ED On-Demand Anodyne EPHX2 18 41 CS(=O)(=O)N1CC[C@@H](NC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880537549 ED On-Demand Anodyne EPHX2 18 41 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccnc(C#N)c3)CC2)CC1 ZINC000880537607 GH On-Demand Mild GPR119 32 50 CS(=O)(=O)c1ccc([C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537633 GG On-Demand Anodyne ADRB1 32 41 CS(=O)(=O)c1ccc([C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537633 GG On-Demand Anodyne ADRB3 56 44 CS(=O)(=O)c1ccc([C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537634 GG On-Demand Anodyne ADRB1 32 41 CS(=O)(=O)c1ccc([C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537634 GG On-Demand Anodyne ADRB3 56 44 CS(=O)(=O)c1ccc([C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537635 GG On-Demand Anodyne ADRB1 32 41 CS(=O)(=O)c1ccc([C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537635 GG On-Demand Anodyne ADRB3 56 44 CS(=O)(=O)c1ccc([C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537636 GG On-Demand Anodyne ADRB1 32 41 CS(=O)(=O)c1ccc([C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880537636 GG On-Demand Anodyne ADRB3 56 44 CCN1CCC(NC(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537637 FF On-Demand Anodyne SIGMAR1 15 48 CCN1CCC(NC(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537637 FF On-Demand Anodyne CCR2 22 40 CCN1CCC(NC(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537637 FF On-Demand Anodyne MCHR1 19 41 CCN1CCC(NC(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537638 FF On-Demand Anodyne SIGMAR1 15 48 CCN1CCC(NC(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537638 FF On-Demand Anodyne CCR2 22 40 CCN1CCC(NC(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880537638 FF On-Demand Anodyne MCHR1 19 41 N#CCNC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880537645 CD On-Demand Mild CTSL 24 42 N#CCNC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880537645 CD On-Demand Mild CTSS 17 42 N#CCNC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880537645 CD On-Demand Mild CTSV 36 42 N#CCNC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880537649 CD On-Demand Mild CTSL 24 42 N#CCNC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880537649 CD On-Demand Mild CTSS 17 42 N#CCNC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880537649 CD On-Demand Mild CTSV 36 42 COC(=O)[C@H](CNC(=O)c1ccc(-c2ccccc2OC)nc1O)CC1CC1 ZINC000880537672 GF On-Demand Anodyne KCNA3 40 37 COC(=O)[C@@H](CNC(=O)c1ccc(-c2ccccc2OC)nc1O)CC1CC1 ZINC000880537674 GF On-Demand Anodyne KCNA3 40 37 CC[C@H](NC(=O)c1cc(C)co1)c1ccccc1F ZINC000880537710 CH On-Demand Anodyne CTSA 70 37 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Br)c1 ZINC000880537723 GE On-Demand Anodyne DRD4 41 32 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Br)c1 ZINC000880537723 GE On-Demand Anodyne PLD1 40 34 O=C(NCCN1CCCC1=O)c1ccc(OC(F)F)c(Br)c1 ZINC000880537723 GE On-Demand Anodyne PLD2 57 34 Cc1nc(C(C)C)ncc1C(=O)NCCN1CCCC1=O ZINC000880537726 CD On-Demand Anodyne TYRO3 23 44 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CCCC2=O)N1Cc1ccccc1 ZINC000880537733 FC On-Demand Anodyne ACHE 21 48 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CCCC2=O)N1Cc1ccccc1 ZINC000880537733 FC On-Demand Anodyne SIGMAR1 15 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CCCC2=O)N1Cc1ccccc1 ZINC000880537733 FC On-Demand Anodyne P2RX7 25 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CCCC2=O)N1Cc1ccccc1 ZINC000880537733 FC On-Demand Anodyne TYRO3 18 40 O=C(NCCN1CCCC1=O)c1cc(Br)ccc1C1CC1 ZINC000880537752 FF On-Demand Anodyne TYRO3 22 43 O=C1CCc2cc(OC[C@@H](O)CN3C[C@@H]4CC[C@H]3c3ccccc34)ccc2N1 ZINC000880537834 GG On-Demand Anodyne ACOX1 45 39 O=C1CCc2cc(OC[C@H](O)CN3C[C@@H]4CC[C@H]3c3ccccc34)ccc2N1 ZINC000880537835 GG On-Demand Anodyne ACOX1 45 39 COC(=O)[C@@H](CCF)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880537843 DD On-Demand Anodyne NQO2 26 40 COC(=O)[C@@H](CCF)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880537843 DD On-Demand Anodyne MTNR1A 36 40 COC(=O)[C@@H](CCF)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880537847 DD On-Demand Anodyne NQO2 26 40 COC(=O)[C@@H](CCF)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880537847 DD On-Demand Anodyne MTNR1A 36 40 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne DRD2 22 41 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne ACHE 16 44 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne LTA4H 41 40 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne HRH3 94 50 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne SIGMAR1 15 40 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne BCHE 15 44 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne KDR 23 48 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne MET 26 45 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne EPHX2 33 53 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne FLT3 30 40 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne AURKA 21 45 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne NOD2 40 38 Cc1coc(C(=O)Nc2ccc(OCCCN3CCN(C)CC3)cc2)c1 ZINC000880537882 FF On-Demand Anodyne MEN1 41 32 COC(=O)c1ccc(CN[C@H](c2cccc(Cl)c2)C(F)F)s1 ZINC000880537896 EI On-Demand Anodyne ADRB1 18 40 COC(=O)c1ccc(CN[C@H](c2cccc(Cl)c2)C(F)F)s1 ZINC000880537896 EI On-Demand Anodyne ADRB3 25 40 COC(=O)c1ccc(CN[C@@H](c2cccc(Cl)c2)C(F)F)s1 ZINC000880537899 EI On-Demand Anodyne ADRB1 18 40 COC(=O)c1ccc(CN[C@@H](c2cccc(Cl)c2)C(F)F)s1 ZINC000880537899 EI On-Demand Anodyne ADRB3 25 40 N#Cc1cc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)ccn1 ZINC000880537928 DE On-Demand Mild EPHX2 22 46 C[C@@]1(CNC(=O)Nc2ccnc(C#N)c2)CCN(Cc2ccccc2)C1 ZINC000880537929 EF On-Demand Mild CCR3 26 41 C[C@@]1(CNC(=O)Nc2ccnc(C#N)c2)CCN(Cc2ccccc2)C1 ZINC000880537929 EF On-Demand Mild NPFFR1 46 38 N#Cc1cc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)ccn1 ZINC000880537930 DE On-Demand Mild EPHX2 22 46 CC[C@H]1CN(C(=O)c2cc(C)cnc2Cl)[C@H](C)CO1 ZINC000880537935 CF On-Demand Anodyne HCRTR2 17 46 CC[C@H]1CN(C(=O)c2cc(C)cnc2Cl)[C@@H](C)CO1 ZINC000880537937 CF On-Demand Anodyne HCRTR2 17 46 N#Cc1ccccc1OC[C@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880537994 EG On-Demand Mild ADRB1 49 40 N#Cc1ccccc1OC[C@@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880537995 EG On-Demand Mild ADRB1 49 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880538069 EE On-Demand Mild HTR1B 15 46 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880538069 EE On-Demand Mild PDGFRB 60 46 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880538069 EE On-Demand Mild FAAH 18 46 O=C(c1cc2ccccc2cc1F)N1CCC(Cn2cnnc2)CC1 ZINC000880538071 EG On-Demand Anodyne GRIN2B 40 36 O=C(c1cc2ccccc2cc1F)N1CCC(Cn2cnnc2)CC1 ZINC000880538071 EG On-Demand Anodyne PARP1 26 40 CC(=O)N1CCN(C(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880538102 FD On-Demand Anodyne KCNQ2 19 40 CC(=O)N1CCN(C(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880538103 FD On-Demand Anodyne KCNQ2 19 40 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc(Br)ccc2C2CC2)C1 ZINC000880538119 GE On-Demand Anodyne HTR4 21 40 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc(Br)ccc2C2CC2)C1 ZINC000880538121 GE On-Demand Anodyne HTR4 21 40 COC(=O)[C@@H](CCF)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880538126 EF On-Demand Anodyne CTSL 16 40 COC(=O)[C@@H](CCF)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880538126 EF On-Demand Anodyne LIPE 18 40 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880538174 FF On-Demand Mild EPHX2 26 41 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)Nc3ccnc(C#N)c3)CC2)C1 ZINC000880538174 FF On-Demand Mild GPR119 18 46 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538177 DC On-Demand Anodyne HTR4 16 41 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538177 DC On-Demand Anodyne JAK3 15 46 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538177 DC On-Demand Anodyne JAK1 27 40 CS(=O)(=O)N1CC[C@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538179 DC On-Demand Anodyne HTR4 16 41 CS(=O)(=O)N1CC[C@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538179 DC On-Demand Anodyne JAK3 15 46 CS(=O)(=O)N1CC[C@H](NC(=O)c2cncc3[nH]ccc23)C1 ZINC000880538179 DC On-Demand Anodyne JAK1 27 40 CC(C)(C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880538190 GE On-Demand Anodyne EPHX2 33 61 CC(C)(C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880538190 GE On-Demand Anodyne SFRP1 44 35 CC(C)(C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880538192 GE On-Demand Anodyne EPHX2 33 61 CC(C)(C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880538192 GE On-Demand Anodyne SFRP1 44 35 CN(Cc1cnn(C)c1)C(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880538207 FF On-Demand Anodyne PLA2G7 36 42 CN(Cc1cnn(C)c1)C(=O)CN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880538209 FF On-Demand Anodyne PLA2G7 36 42 N#Cc1cc(NC(=O)N2CCC3(CC2)OCCO3)ccn1 ZINC000880538216 CD On-Demand Mild PDGFRB 22 42 C[C@H]1CC[C@H](NC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880538236 BE On-Demand Mild TYK2 40 35 C[C@H]1CC[C@@H](NC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880538237 BE On-Demand Mild TYK2 40 35 C[C@@H]1CC[C@H](NC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880538239 BE On-Demand Mild TYK2 40 35 COC(=O)CCCN[C@H](c1cccc(Cl)c1)C(F)F ZINC000880538247 CG On-Demand Anodyne ADRB1 19 41 COC(=O)CCCN[C@@H](c1cccc(Cl)c1)C(F)F ZINC000880538248 CG On-Demand Anodyne ADRB1 19 41 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1ccc2nc(O)[nH]c2c1 ZINC000880538250 EG On-Demand Anodyne NR2E3 52 33 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538261 GH On-Demand Anodyne ADRB2 46 57 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538261 GH On-Demand Anodyne ADRB1 95 57 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538261 GH On-Demand Anodyne GRIN1 30 47 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538261 GH On-Demand Anodyne ADRB3 76 46 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538263 GH On-Demand Anodyne ADRB2 46 57 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538263 GH On-Demand Anodyne ADRB1 95 57 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538263 GH On-Demand Anodyne GRIN1 30 47 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538263 GH On-Demand Anodyne ADRB3 76 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538265 GH On-Demand Anodyne ADRB2 46 57 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538265 GH On-Demand Anodyne ADRB1 95 57 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538265 GH On-Demand Anodyne GRIN1 30 47 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538265 GH On-Demand Anodyne ADRB3 76 46 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538266 GH On-Demand Anodyne ADRB2 46 57 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538266 GH On-Demand Anodyne ADRB1 95 57 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538266 GH On-Demand Anodyne GRIN1 30 47 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](c2cccc(Cl)c2)C(F)F)cc1 ZINC000880538266 GH On-Demand Anodyne ADRB3 76 46 Cc1nc(C(C)C)ncc1C(=O)N1C[C@H]2C[C@H]1[C@H]2NC(=O)OCc1ccccc1 ZINC000880538284 GG On-Demand Anodyne CAPN2 43 32 Cc1nc(C(C)C)ncc1C(=O)N1C[C@H]2C[C@H]1[C@@H]2NC(=O)OCc1ccccc1 ZINC000880538289 GG On-Demand Anodyne CAPN2 43 32 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3ccnc(C#N)c3)C[C@@H]2C1 ZINC000880538349 FE On-Demand Mild GPR119 28 52 N#Cc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccn1 ZINC000880538375 EE On-Demand Mild PDGFRB 47 42 N#Cc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccn1 ZINC000880538375 EE On-Demand Mild TRPV1 17 48 C=CC(C)(C)CC(=O)Nc1ccc(OCCCN2CCN(C)CC2)cc1 ZINC000880538381 FG On-Demand Mild LTA4H 44 39 C=CC(C)(C)CC(=O)Nc1ccc(OCCCN2CCN(C)CC2)cc1 ZINC000880538381 FG On-Demand Mild HRH3 72 48 C=CC(C)(C)CC(=O)Nc1ccc(OCCCN2CCN(C)CC2)cc1 ZINC000880538381 FG On-Demand Mild EPHX2 33 54 C=CC(C)(C)CC(=O)Nc1ccc(OCCCN2CCN(C)CC2)cc1 ZINC000880538381 FG On-Demand Mild MEN1 40 31 O=C(NCC[C@@]1(O)CCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880538383 GD On-Demand Anodyne CTRA_BOVIN 52 30 O=C(NCC[C@@]1(O)CCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880538383 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 O=C(NCC[C@]1(O)CCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880538385 GD On-Demand Anodyne CTRA_BOVIN 52 30 O=C(NCC[C@]1(O)CCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880538385 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 C#CCC[C@@H](O)CNC(=O)Nc1ccnc(C#N)c1 ZINC000880538401 CC On-Demand Mild ADRB1 43 32 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880538405 FF On-Demand Mild PDGFRB 46 36 C#CCC[C@H](O)CNC(=O)Nc1ccnc(C#N)c1 ZINC000880538408 CC On-Demand Mild ADRB1 43 32 C[C@H](NC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F)C(=O)N1CCCCC1 ZINC000880538418 GF On-Demand Anodyne DPP7 43 41 C[C@H](NC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F)C(=O)N1CCCCC1 ZINC000880538419 GF On-Demand Anodyne DPP7 43 41 C[C@@H](NC(=O)CN[C@H](c1cccc(Cl)c1)C(F)F)C(=O)N1CCCCC1 ZINC000880538420 GF On-Demand Anodyne DPP7 43 41 C[C@@H](NC(=O)CN[C@@H](c1cccc(Cl)c1)C(F)F)C(=O)N1CCCCC1 ZINC000880538421 GF On-Demand Anodyne DPP7 43 41 CCOC(=O)C1CCN(C(=O)CN[C@@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880538422 GG On-Demand Anodyne FDFT1 30 49 CCOC(=O)C1CCN(C(=O)CN[C@H](c2cccc(Cl)c2)C(F)F)CC1 ZINC000880538423 GG On-Demand Anodyne FDFT1 30 49 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA2 29 50 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA1 23 44 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA5B 42 35 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA4 31 50 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA5A 49 35 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA12 15 45 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne ST14 44 39 NS(=O)(=O)c1cccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880538444 GF On-Demand Anodyne CA9 18 45 N#Cc1cc(NC(=O)N2CCC(F)(F)CC2)ccn1 ZINC000880538456 CE On-Demand Mild CACNA1H 44 39 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1F ZINC000880538481 FE On-Demand Mild PDGFRB 62 46 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1F ZINC000880538481 FE On-Demand Mild MET 54 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1F ZINC000880538481 FE On-Demand Mild RBP4 18 41 COCCCCCN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880538489 CH On-Demand Anodyne UGCG 58 36 COCCCCCN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880538489 CH On-Demand Anodyne GBA2 72 36 COC(=O)[C@@H](CCF)NC(=O)c1cc2ccccc2cc1F ZINC000880538495 DF On-Demand Anodyne PIN1 47 36 COC(=O)[C@@H](CCF)NC(=O)c1cc2ccccc2cc1F ZINC000880538495 DF On-Demand Anodyne UTS2 45 33 CN(CCC1CCN(C(=O)Nc2ccnc(C#N)c2)CC1)C(=O)OC(C)(C)C ZINC000880538501 GG On-Demand Mild GPR119 20 43 CC[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)[C@@H](C)CO1 ZINC000880538511 FH On-Demand Anodyne HCRTR2 15 43 CC[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)[C@H](C)CO1 ZINC000880538512 FH On-Demand Anodyne HCRTR2 15 43 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA2 100 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA1 89 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA7 59 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA5B 69 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA4 84 48 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA5A 75 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA14 43 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA12 64 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne CA9 67 50 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne F13A1 45 35 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne NCE103 16 40 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne MTCA1 51 45 NS(=O)(=O)c1ccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538518 FE On-Demand Anodyne P96878_MYCTU 63 45 NC(=O)c1ccc(NC(=O)CCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880538531 EG On-Demand Anodyne PLAU 16 40 COC(=O)[C@@H](CCF)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880538557 DF On-Demand Anodyne NQO2 23 44 COC(=O)[C@@H](CCF)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880538561 DF On-Demand Anodyne NQO2 23 44 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(Cn2cnnc2)CC1 ZINC000880538595 FD On-Demand Anodyne GRIN2B 40 42 O=C(N[C@H](C1CCOCC1)C1CC1)c1cc2ccccc2cc1F ZINC000880538608 EH On-Demand Anodyne PYGL 21 45 O=C(N[C@@H](C1CCOCC1)C1CC1)c1cc2ccccc2cc1F ZINC000880538609 EH On-Demand Anodyne PYGL 21 45 FC(F)[C@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538610 CH On-Demand Anodyne CYP19A1 17 40 FC(F)[C@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538610 CH On-Demand Anodyne CYP11B1 21 45 FC(F)[C@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538610 CH On-Demand Anodyne TBXAS1 36 43 FC(F)[C@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538610 CH On-Demand Anodyne HMOX2 55 40 FC(F)[C@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538610 CH On-Demand Anodyne CYP24A1 26 40 FC(F)[C@@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538611 CH On-Demand Anodyne CYP19A1 17 40 FC(F)[C@@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538611 CH On-Demand Anodyne CYP11B1 21 45 FC(F)[C@@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538611 CH On-Demand Anodyne TBXAS1 36 43 FC(F)[C@@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538611 CH On-Demand Anodyne HMOX2 55 40 FC(F)[C@@H](NCCCn1ccnc1)c1cccc(Cl)c1 ZINC000880538611 CH On-Demand Anodyne CYP24A1 26 40 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(O)CCOC1)C2 ZINC000880538639 DD On-Demand Anodyne MTNR1A 39 40 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(O)CCOC1)C2 ZINC000880538643 DD On-Demand Anodyne MTNR1A 39 40 COC(=O)[C@@H](CNC(=O)c1ncsc1C1CC1)CC1CC1 ZINC000880538644 DE On-Demand Anodyne MAP1 52 37 COC(=O)[C@H](CNC(=O)c1ncsc1C1CC1)CC1CC1 ZINC000880538645 DE On-Demand Anodyne MAP1 52 37 COc1cc(NC(=O)c2ncsc2C2CC2)cc(Cl)c1OC ZINC000880538656 EH On-Demand Anodyne MAP1 54 35 COc1cc(NC(=O)c2ncsc2C2CC2)cc(Cl)c1OC ZINC000880538656 EH On-Demand Anodyne GRM4 23 40 Cc1cnc(Cl)c(C(=O)N2CCO[C@H]3CCN(Cc4ccccc4)C[C@H]32)c1 ZINC000880538703 GG On-Demand Anodyne DRD4 50 39 Cc1cnc(Cl)c(C(=O)N2CCO[C@H]3CCN(Cc4ccccc4)C[C@@H]32)c1 ZINC000880538704 GG On-Demand Anodyne DRD4 50 39 Cc1cnc(Cl)c(C(=O)N2CCO[C@@H]3CCN(Cc4ccccc4)C[C@@H]32)c1 ZINC000880538705 GG On-Demand Anodyne DRD4 50 39 Cc1cnc(Cl)c(C(=O)N2CCO[C@@H]3CCN(Cc4ccccc4)C[C@H]32)c1 ZINC000880538706 GG On-Demand Anodyne DRD4 50 39 N#Cc1cc(NC(=O)NC[C@H](O)C(F)(F)F)ccn1 ZINC000880538724 CC On-Demand Mild ADRB1 44 33 N#Cc1cc(NC(=O)NC[C@H](O)C(F)(F)F)ccn1 ZINC000880538724 CC On-Demand Mild PRMT3 45 35 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538746 ED On-Demand Anodyne DRD4 23 40 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538746 ED On-Demand Anodyne HTR4 41 42 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538746 ED On-Demand Anodyne CCR3 25 47 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538746 ED On-Demand Anodyne EPHX2 23 40 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538747 ED On-Demand Anodyne DRD4 23 40 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538747 ED On-Demand Anodyne HTR4 41 42 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538747 ED On-Demand Anodyne CCR3 25 47 CS(=O)(=O)N1CC[C@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880538747 ED On-Demand Anodyne EPHX2 23 40 CC(C)(C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)c1ccc(F)cc1F ZINC000880538757 ED On-Demand Anodyne EPHX2 16 41 CC(C)(C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)c1ccc(F)cc1F ZINC000880538757 ED On-Demand Anodyne SFRP1 56 33 CC(C)(C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)c1ccc(F)cc1F ZINC000880538758 ED On-Demand Anodyne EPHX2 16 41 CC(C)(C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)c1ccc(F)cc1F ZINC000880538758 ED On-Demand Anodyne SFRP1 56 33 O=C(CN[C@H](c1cccc(Cl)c1)C(F)F)NCC1CC1 ZINC000880538835 DF On-Demand Anodyne CACNA1I 47 39 O=C(CN[C@@H](c1cccc(Cl)c1)C(F)F)NCC1CC1 ZINC000880538837 DF On-Demand Anodyne CACNA1I 47 39 O=C(N[C@H](C1CCOCC1)C1CC1)c1cnc2cc[nH]c2c1 ZINC000880538838 CE On-Demand Anodyne MAPK1 43 31 O=C(N[C@@H](C1CCOCC1)C1CC1)c1cnc2cc[nH]c2c1 ZINC000880538840 CE On-Demand Anodyne MAPK1 43 31 N#Cc1cc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)ccn1 ZINC000880538865 EE On-Demand Mild FAAH 29 51 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880538895 GG On-Demand Anodyne DRD4 18 41 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880538895 GG On-Demand Anodyne MAPK14 15 40 NS(=O)(=O)c1ccc2c(c1)CCN2C(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880538900 GE On-Demand Anodyne CA7 32 51 NS(=O)(=O)c1ccc2c(c1)CCN2C(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880538900 GE On-Demand Anodyne EIF2AK3 49 34 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1nccs1 ZINC000880538918 CG On-Demand Anodyne MAP1 134 46 C[C@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccnc(C#N)c1 ZINC000880538925 EE On-Demand Mild GPR119 38 48 O=C(COC1CC1)NNc1ccccc1Cc1ccccc1 ZINC000880538928 CF On-Demand Reactive TIMP3 73 36 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)ccn1 ZINC000880538936 FG On-Demand Mild CACNA1H 40 42 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)ccn1 ZINC000880538936 FG On-Demand Mild NPY5R 35 42 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)ccn1 ZINC000880538936 FG On-Demand Mild TYK2 55 36 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)ccn1 ZINC000880538936 FG On-Demand Mild TRPM8 17 42 C#CC(C)(C)NC(=O)Nc1ccnc(C#N)c1 ZINC000880538937 BD On-Demand Mild TYK2 55 36 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)ccn1 ZINC000880538964 GG On-Demand Mild TRPV1 15 44 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)ccn1 ZINC000880538964 GG On-Demand Mild NPY5R 30 43 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)ccn1 ZINC000880538964 GG On-Demand Mild RBP4 57 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC[C@H]1OC ZINC000880538988 ED On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC[C@H]1OC ZINC000880538989 ED On-Demand Anodyne PAPA1_CARPA 33 41 N#Cc1cc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)ccn1 ZINC000880538991 FF On-Demand Mild CACNA1H 46 42 N#Cc1cc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)ccn1 ZINC000880538991 FF On-Demand Mild TRPM8 33 40 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)cc(Cl)c1OC ZINC000880539008 EH On-Demand Anodyne JUN 21 47 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)cc(Cl)c1OC ZINC000880539008 EH On-Demand Anodyne ATF1 58 39 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)cc(Cl)c1OC ZINC000880539008 EH On-Demand Anodyne NFKB1 54 39 N#Cc1cc(NC(=O)N2CCCC3(CCCC3)C2)ccn1 ZINC000880539018 CG On-Demand Mild EPHX2 29 41 CON=Cc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880539033 FH On-Demand Mild KCNK3 96 42 CON=Cc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880539033 FH On-Demand Mild KCNK9 58 34 CC(C)(C)OC(=O)NCC1(CCNC(=O)c2cccn3nccc23)CC1 ZINC000880539039 FF On-Demand Anodyne HCN1 58 33 CC(C)(C)OC(=O)NCC1(CCNC(=O)c2cccn3nccc23)CC1 ZINC000880539039 FF On-Demand Anodyne HCN4 50 32 COc1cc(NC(=O)c2nnn(C)n2)cc(Cl)c1OC ZINC000880539041 CD On-Demand Anodyne ENPP1 62 33 COc1ccccc1NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880539051 DH On-Demand Anodyne DRD4 15 45 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA2 82 57 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA1 73 55 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA7 49 55 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA5B 56 55 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA4 52 52 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA5A 57 55 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA14 37 46 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA12 52 51 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CA9 61 57 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne CYNT 19 42 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne NCE103 23 45 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne P96878_MYCTU 23 45 NS(=O)(=O)c1ccc(CCNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880539052 GD On-Demand Anodyne A6YCJ1_9METZ 23 46 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NC(=O)NC1CCCC1 ZINC000880539063 EF On-Demand Anodyne EPHX2 27 41 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCc1cccnc1 ZINC000880539067 DF On-Demand Anodyne CHRNA7 47 36 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCc1cccnc1 ZINC000880539067 DF On-Demand Anodyne NAMPT 76 43 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1ccnc(C#N)c1 ZINC000880539075 FF On-Demand Mild GPR119 42 49 C[S@@](=O)CCNC(=O)Nc1ccnc(C#N)c1 ZINC000880539101 CC On-Demand Mild ADRB1 40 30 N#Cc1cc(NC(=O)NCCC2SCCS2)ccn1 ZINC000880539133 CE On-Demand Mild ADRB1 43 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C1CCOCC1)C1CC1 ZINC000880539134 FE On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C1CCOCC1)C1CC1 ZINC000880539135 FE On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C1CCOCC1)C1CC1 ZINC000880539136 FE On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C1CCOCC1)C1CC1 ZINC000880539137 FE On-Demand Anodyne PAPA1_CARPA 34 41 CS(=O)(=O)N1CC[C@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880539158 DC On-Demand Anodyne JAK3 20 52 CS(=O)(=O)N1CC[C@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880539158 DC On-Demand Anodyne JAK1 28 52 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880539159 DC On-Demand Anodyne JAK3 20 52 CS(=O)(=O)N1CC[C@@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880539159 DC On-Demand Anodyne JAK1 28 52 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP13 28 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP3 41 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP8 20 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP9 27 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne EPHX2 24 48 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP7 33 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539169 FC On-Demand Anodyne MMP1 34 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP13 28 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP3 41 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP8 20 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP9 27 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne EPHX2 24 48 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP7 33 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(S(C)(=O)=O)C1)C2 ZINC000880539171 FC On-Demand Anodyne MMP1 34 43 FC(F)[C@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539191 CG On-Demand Anodyne CYP19A1 19 44 FC(F)[C@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539191 CG On-Demand Anodyne CYP11B1 25 47 FC(F)[C@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539191 CG On-Demand Anodyne TBXAS1 29 40 FC(F)[C@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539191 CG On-Demand Anodyne HMOX2 50 37 FC(F)[C@@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539192 CG On-Demand Anodyne CYP19A1 19 44 FC(F)[C@@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539192 CG On-Demand Anodyne CYP11B1 25 47 FC(F)[C@@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539192 CG On-Demand Anodyne TBXAS1 29 40 FC(F)[C@@H](NCCn1ccnc1)c1cccc(Cl)c1 ZINC000880539192 CG On-Demand Anodyne HMOX2 50 37 N#Cc1cc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)ccn1 ZINC000880539217 FD On-Demand Mild EPHX2 39 44 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1cccnc1Cl ZINC000880539227 EH On-Demand Anodyne G2YM83_BOTF4 67 35 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1ccc(N2CCOCC2)cc1 ZINC000880539237 GG On-Demand Anodyne MTOR 61 37 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)Nc1ccc(N2CCOCC2)cc1 ZINC000880539237 GG On-Demand Anodyne STAT6 49 34 O=C1CC[C@@H](c2ccc(C(=O)N3CCC4(CC3)CC4(F)F)cc2)N1 ZINC000880539290 EF On-Demand Anodyne L3MBTL3 47 36 O=C1CC[C@H](c2ccc(C(=O)N3CCC4(CC3)CC4(F)F)cc2)N1 ZINC000880539291 EF On-Demand Anodyne L3MBTL3 47 36 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Br)c([N+](=O)[O-])c1 ZINC000880539326 HI On-Demand Mild TAAR1 46 56 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Br)c([N+](=O)[O-])c1 ZINC000880539326 HI On-Demand Mild DDR1 36 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(Br)c([N+](=O)[O-])c1 ZINC000880539326 HI On-Demand Mild KCNK3 68 40 CC(C)(C)OC(=O)N1CCC[C@@]2(CCN(C(=O)Nc3ccnc(C#N)c3)C2)C1 ZINC000880539356 GG On-Demand Mild EPHX2 30 41 C[C@@H]1CN(C(=O)Nc2ccnc(C#N)c2)CCN1C(=O)OC(C)(C)C ZINC000880539378 EE On-Demand Mild GPR119 31 46 C[C@H]1CN(C(=O)Nc2ccnc(C#N)c2)CCN1C(=O)OC(C)(C)C ZINC000880539379 EE On-Demand Mild GPR119 31 46 COc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cc(Cl)c1OC ZINC000880539391 FH On-Demand Anodyne CPT1A 46 35 COc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cc(Cl)c1OC ZINC000880539391 FH On-Demand Anodyne CPT2 40 33 COc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cc(Cl)c1OC ZINC000880539392 FH On-Demand Anodyne CPT1A 46 35 COc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cc(Cl)c1OC ZINC000880539392 FH On-Demand Anodyne CPT2 40 33 N#Cc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccn1 ZINC000880539440 CE On-Demand Mild CACNA1H 33 42 N#Cc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccn1 ZINC000880539441 CE On-Demand Mild CACNA1H 33 42 COC(=O)[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)CC1CC1 ZINC000880539456 EE On-Demand Anodyne GABRA1 18 44 COC(=O)[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)CC1CC1 ZINC000880539456 EE On-Demand Anodyne GABRA2 15 44 Cc1cccc(C(=O)NNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880539499 EF On-Demand Reactive KCNK3 56 38 Cc1cccc(C(=O)NNC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880539499 EF On-Demand Reactive KCNK9 44 38 C[C@H]1C[C@H]1c1noc(CC2CCN(C(=O)CC(C)(C)CC(F)(F)F)CC2)n1 ZINC000880539501 GI On-Demand Anodyne ETHR 42 37 C[C@@H]1C[C@H]1c1noc(CC2CCN(C(=O)CC(C)(C)CC(F)(F)F)CC2)n1 ZINC000880539504 GI On-Demand Anodyne ETHR 42 37 O=c1cc(CN2C[C@@H]3CC[C@H]2c2ccccc23)occ1O ZINC000880539509 CF On-Demand Anodyne DAO 21 43 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCC1 ZINC000880539511 CF On-Demand Anodyne PREP 52 36 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCC1 ZINC000880539511 CF On-Demand Anodyne L3MBTL3 51 38 N#Cc1cc(NC(=O)NC2CCC(N3CCCCC3)CC2)ccn1 ZINC000880539520 EF On-Demand Mild EPHX2 45 43 N#Cc1cc(NC(=O)NC2CCC(N3CCCCC3)CC2)ccn1 ZINC000880539520 EF On-Demand Mild L3MBTL3 52 34 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCCn1ccnc1 ZINC000880539526 CG On-Demand Anodyne TBXAS1 37 41 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCCn1ccnc1 ZINC000880539526 CG On-Demand Anodyne HMOX2 47 36 c1ccc2c(c1)[C@@H]1CC[C@H]2CN1CCCn1ccnc1 ZINC000880539526 CG On-Demand Anodyne QPCT 34 41 N#Cc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccn1 ZINC000880539530 EE On-Demand Mild MTOR 41 39 N#Cc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccn1 ZINC000880539530 EE On-Demand Mild SCN10A 18 45 CC(C)(C(=O)N1CCC(Cn2cnnc2)CC1)c1ccc(F)cc1F ZINC000880539531 EF On-Demand Anodyne PRCP 45 35 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539548 EE On-Demand Mild F10 21 40 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539548 EE On-Demand Mild NPY1R 28 41 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539548 EE On-Demand Mild CCKBR 42 37 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539549 EE On-Demand Mild F10 21 40 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539549 EE On-Demand Mild NPY1R 28 41 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccn1 ZINC000880539549 EE On-Demand Mild CCKBR 42 37 CN(C(=O)Nc1ccnc(C#N)c1)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880539573 EE On-Demand Mild GPR119 42 52 CN(C(=O)Nc1ccnc(C#N)c1)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880539574 EE On-Demand Mild GPR119 42 52 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(Cn2cnnc2)CC1 ZINC000880539575 GD On-Demand Anodyne P2RY12 67 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(Cn2cnnc2)CC1 ZINC000880539576 GD On-Demand Anodyne P2RY12 67 36 O=C(C(=O)N1CCC(Cn2cnnc2)CC1)c1c[nH]c2cc(F)ccc12 ZINC000880539577 FE On-Demand Anodyne GRIN2B 21 62 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(Cn2cnnc2)CC1 ZINC000880539582 FG On-Demand Anodyne PDE4D 26 40 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(Cn2cnnc2)CC1 ZINC000880539582 FG On-Demand Anodyne L3MBTL3 42 34 O=C(c1ncccc1-c1ccccn1)N1CCC(Cn2cnnc2)CC1 ZINC000880539583 EE On-Demand Anodyne MLNR 15 41 N#Cc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)ccn1 ZINC000880539590 DF On-Demand Mild ADRB1 42 33 N#Cc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)ccn1 ZINC000880539591 DF On-Demand Mild ADRB1 42 33 COC(=O)C1CCN(C(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880539605 EE On-Demand Anodyne PTR1 44 32 CCN1CCC(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880539609 EF On-Demand Anodyne DRD4 24 40 CCN1CCC(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880539609 EF On-Demand Anodyne SIGMAR1 18 44 Cn1nc2c(c1C(=O)N1CCCC[C@H]1Cc1ccccc1F)CSCC2 ZINC000880539616 FH On-Demand Anodyne HCRTR1 20 40 Cn1nc2c(c1C(=O)N1CCCC[C@@H]1Cc1ccccc1F)CSCC2 ZINC000880539617 FH On-Demand Anodyne HCRTR1 20 40 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne CELA1 20 42 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne GRIN2B 31 40 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne CTRA_BOVIN 46 30 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne DPP4 15 42 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne PREP 68 51 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne LGMN 64 37 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne SLC12A5 65 35 C[C@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539618 GF On-Demand Anodyne Q9NAW4_PLAFA 36 41 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne CELA1 20 42 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne GRIN2B 31 40 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne CTRA_BOVIN 46 30 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne DPP4 15 42 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne PREP 68 51 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne LGMN 64 37 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne SLC12A5 65 35 C[C@@H](CO)C1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1 ZINC000880539619 GF On-Demand Anodyne Q9NAW4_PLAFA 36 41 C[S@@](=O)CCCNC(=O)Nc1ccnc(C#N)c1 ZINC000880539628 CC On-Demand Mild ADRB1 42 31 Cn1nnc(C(=O)N2CCCC[C@@H]2Cc2ccccc2F)n1 ZINC000880539636 DD On-Demand Anodyne HCRTR1 21 42 Cn1nnc(C(=O)N2CCCC[C@H]2Cc2ccccc2F)n1 ZINC000880539637 DD On-Demand Anodyne HCRTR1 21 42 N#Cc1cc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)ccn1 ZINC000880539661 FE On-Demand Mild FAAH 31 48 N#Cc1cc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)ccn1 ZINC000880539661 FE On-Demand Mild Q8WSF8_APLCA 40 36 N#Cc1cc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)ccn1 ZINC000880539661 FE On-Demand Mild NACHRBETA2 42 36 N#Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539662 ED On-Demand Mild CCR1 47 39 N#Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539663 ED On-Demand Mild CCR1 47 39 O[C@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539668 ED On-Demand Anodyne ACOX1 47 36 O[C@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539668 ED On-Demand Anodyne CCR1 50 46 O[C@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539668 ED On-Demand Anodyne ABCB1 57 47 O[C@@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539669 ED On-Demand Anodyne ACOX1 47 36 O[C@@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539669 ED On-Demand Anodyne CCR1 50 46 O[C@@H](COc1ccc(F)cc1)CN1CCC2(CC1)COCCO2 ZINC000880539669 ED On-Demand Anodyne ABCB1 57 47 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCC(=O)N1CCCC1 ZINC000880539676 ED On-Demand Anodyne PREP 40 44 CCOC(=O)N1CCC(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880539679 FF On-Demand Anodyne P2RY12 47 37 CCOC(=O)N1CCC(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880539679 FF On-Demand Anodyne CCR8 54 47 C[C@H](CO)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1 ZINC000880539685 EE On-Demand Anodyne HRH4 15 48 C[C@@H](CO)C1CCN(C(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1 ZINC000880539686 EE On-Demand Anodyne HRH4 15 48 CCc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880539687 EF On-Demand Mild P2RY12 17 44 CCc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880539687 EF On-Demand Mild PDGFRB 50 39 CCc1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880539687 EF On-Demand Mild P2RY14 41 38 C[C@@H](CO)C1CCN(C(=O)[C@H]2CN(C(=O)OC(C)(C)C)CC2(C)C)CC1 ZINC000880539700 FF On-Demand Anodyne GPR119 15 40 C[C@@H](CO)C1CCN(C(=O)[C@@H]2CN(C(=O)OC(C)(C)C)CC2(C)C)CC1 ZINC000880539701 FF On-Demand Anodyne GPR119 15 40 C[C@H]1CCc2ccccc2N1C(=O)CN1CCC2(CC1)COCCO2 ZINC000880539710 EE On-Demand Anodyne DRD4 27 45 C[C@@H](CO)C1CCN(C(=O)C(=O)c2c[nH]c3cc(F)ccc23)CC1 ZINC000880539728 EE On-Demand Anodyne GRIN2B 15 58 C[C@@H](CO)C1CCN(C(=O)C(=O)c2c[nH]c3cc(F)ccc23)CC1 ZINC000880539728 EE On-Demand Anodyne MPO 52 33 COC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539750 FD On-Demand Anodyne ACOX1 66 34 COC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539750 FD On-Demand Anodyne CCR1 51 44 COC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539750 FD On-Demand Anodyne ABCB1 60 43 COC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539751 FD On-Demand Anodyne ACOX1 66 34 COC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539751 FD On-Demand Anodyne CCR1 51 44 COC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880539751 FD On-Demand Anodyne ABCB1 60 43 O=C(COC1CC1)Nc1ccc(SCCN2CCCC2)cc1 ZINC000880539758 DF On-Demand Anodyne CHRNA7 15 40 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NC[C@H]1CCCO1 ZINC000880539762 DE On-Demand Anodyne PDE8B 17 40 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NC[C@@H]1CCCO1 ZINC000880539763 DE On-Demand Anodyne PDE8B 17 40 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NC1CCCC1 ZINC000880539771 CF On-Demand Anodyne EPHX2 19 43 C[C@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539772 FE On-Demand Anodyne DPP7 64 37 C[C@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539772 FE On-Demand Anodyne BIRC3 41 32 C[C@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539772 FE On-Demand Anodyne BIRC2 46 35 C[C@@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539773 FE On-Demand Anodyne DPP7 64 37 C[C@@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539773 FE On-Demand Anodyne BIRC3 41 32 C[C@@H](NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12)C(=O)N1CCCCC1 ZINC000880539773 FE On-Demand Anodyne BIRC2 46 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539776 FF On-Demand Clean PAPA1_CARPA 43 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539776 FF On-Demand Clean CTSL 17 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539776 FF On-Demand Clean FPR1 40 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539777 FF On-Demand Clean PAPA1_CARPA 43 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539777 FF On-Demand Clean CTSL 17 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(Cl)ccc1O ZINC000880539777 FF On-Demand Clean FPR1 40 39 COc1ccccc1[C@H](C)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539780 ED On-Demand Anodyne PSMB8 39 40 COc1ccccc1[C@H](C)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539780 ED On-Demand Anodyne HCN1 40 36 CN(C)S(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880539817 GD On-Demand Anodyne ESR1 17 43 CN(C)S(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880539817 GD On-Demand Anodyne HRH3 15 43 CN(C)S(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880539817 GD On-Demand Anodyne MMP13 19 41 C[C@@H](CO)C1CCN(C(=O)c2ncccc2-c2ccccn2)CC1 ZINC000880539836 EF On-Demand Anodyne MLNR 19 41 C[C@H](CO)C1CCN(C(=O)c2ncccc2-c2ccccn2)CC1 ZINC000880539837 EF On-Demand Anodyne MLNR 19 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc(Cl)ccc2O)N1Cc1ccccc1 ZINC000880539838 GE On-Demand Clean F2 36 47 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc(Cl)ccc2O)N1Cc1ccccc1 ZINC000880539838 GE On-Demand Clean SIGMAR1 15 43 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc(Cl)ccc2O)N1Cc1ccccc1 ZINC000880539838 GE On-Demand Clean P2RX7 77 49 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc(Cl)ccc2O)N1Cc1ccccc1 ZINC000880539838 GE On-Demand Clean TMPRSS11D 40 32 O=C(COC1CC1)N1CCCC[C@H]1Cc1ccccc1F ZINC000880539841 CF On-Demand Anodyne CPT1A 98 40 O=C(COC1CC1)N1CCCC[C@H]1Cc1ccccc1F ZINC000880539841 CF On-Demand Anodyne CPT2 44 35 O=C(COC1CC1)N1CCCC[C@H]1Cc1ccccc1F ZINC000880539841 CF On-Demand Anodyne DPP4 17 42 O=C(COC1CC1)N1CCCC[C@@H]1Cc1ccccc1F ZINC000880539842 CF On-Demand Anodyne CPT1A 98 40 O=C(COC1CC1)N1CCCC[C@@H]1Cc1ccccc1F ZINC000880539842 CF On-Demand Anodyne CPT2 44 35 O=C(COC1CC1)N1CCCC[C@@H]1Cc1ccccc1F ZINC000880539842 CF On-Demand Anodyne DPP4 17 42 C[C@@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)CC1 ZINC000880539898 EG On-Demand Anodyne PDE4D 19 42 C[C@@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)CC1 ZINC000880539898 EG On-Demand Anodyne L3MBTL3 60 35 C[C@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)CC1 ZINC000880539899 EG On-Demand Anodyne PDE4D 19 42 C[C@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)CC1 ZINC000880539899 EG On-Demand Anodyne L3MBTL3 60 35 CCN(CCNC(=O)Nc1ccnc(C#N)c1)C(C)C ZINC000880539903 CD On-Demand Mild ADRB1 41 32 CCN(CCNC(=O)Nc1ccnc(C#N)c1)C(C)C ZINC000880539903 CD On-Demand Mild DOT1L 42 33 CCOc1ccccc1NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880539908 EH On-Demand Anodyne HCN1 43 33 CCOc1ccccc1NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880539908 EH On-Demand Anodyne HCN4 42 33 O=C(CCN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCN(c2ncccn2)CC1 ZINC000880539911 GE On-Demand Anodyne SSTR1 47 39 C[C@@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Br)c2)CC1 ZINC000880539919 GH On-Demand Anodyne L3MBTL3 61 40 C[C@H](CO)C1CCN(C(=O)c2ccc(OC(F)F)c(Br)c2)CC1 ZINC000880539920 GH On-Demand Anodyne L3MBTL3 61 40 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild DRD2 17 40 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild HRH2 28 42 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild DRD3 32 40 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild HRH3 21 42 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild CCR3 44 48 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild CHRNA7 26 53 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild HNMT 74 39 N#Cc1cc(NC(=O)NCCCCCCCN2CCCC2)ccn1 ZINC000880539932 EG On-Demand Mild MCHR1 17 40 COc1ccc(C)cc1NC(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880539949 EH On-Demand Anodyne DRD4 15 48 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCCC1 ZINC000880539954 CF On-Demand Anodyne PREP 47 35 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCCCC1 ZINC000880539954 CF On-Demand Anodyne L3MBTL3 43 37 c1ccc2cc(OCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880539961 EG On-Demand Anodyne LTA4H 51 43 c1ccc2cc(OCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880539961 EG On-Demand Anodyne HRH3 22 42 c1ccc2cc(OCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880539961 EG On-Demand Anodyne SIGMAR1 15 44 c1ccc2cc(OCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880539961 EG On-Demand Anodyne PSMB1 41 36 CC(=O)Nc1cccc(CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880539962 DI On-Demand Anodyne MCHR1 24 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne OPRM1 33 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne OPRD1 23 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne MME 61 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne FCER2 52 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne TIMP3 47 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne ACE2 60 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne QRFPR 18 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne PSMB8 76 50 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539969 FD On-Demand Anodyne NPFFR1 46 31 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne OPRM1 33 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne OPRD1 23 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne MME 61 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne FCER2 52 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne TIMP3 47 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne ACE2 60 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne QRFPR 18 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne PSMB8 76 50 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880539970 FD On-Demand Anodyne NPFFR1 46 31 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCN(C(=O)c2ccco2)CC1 ZINC000880539971 GE On-Demand Anodyne L3MBTL3 41 36 N#Cc1cc(NC(=O)N2CCC3(CCCC3)C2)ccn1 ZINC000880540002 CF On-Demand Mild EPHX2 33 42 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)NCCCN1CCCC1=O ZINC000880540011 EE On-Demand Anodyne TYRO3 20 43 COc1ccc([C@@H](NC(=O)CN2CCC3(CC2)COCCO3)C(C)C)cc1 ZINC000880540013 GE On-Demand Anodyne PSMB8 38 43 COc1ccc([C@H](NC(=O)CN2CCC3(CC2)COCCO3)C(C)C)cc1 ZINC000880540014 GE On-Demand Anodyne PSMB8 38 43 C[C@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc2ccccc2c1 ZINC000880540028 FF On-Demand Anodyne ACOX1 19 47 C[C@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc2ccccc2c1 ZINC000880540028 FF On-Demand Anodyne PSMB8 38 43 C[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc2ccccc2c1 ZINC000880540029 FF On-Demand Anodyne ACOX1 19 47 C[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc2ccccc2c1 ZINC000880540029 FF On-Demand Anodyne PSMB8 38 43 O=C(CN1CCCCS1(=O)=O)NCc1cc(Cl)ccc1O ZINC000880540033 ED On-Demand Clean P2RX7 21 41 O=C(COC1CC1)NCc1cc(Cl)ccc1O ZINC000880540046 CD On-Demand Clean P2RX7 40 39 CCOc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540056 FD On-Demand Anodyne ACOX1 67 31 CCOc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540056 FD On-Demand Anodyne CCR1 48 40 CCOc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540056 FD On-Demand Anodyne ABCB1 55 43 CCOc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540057 FD On-Demand Anodyne ACOX1 67 31 CCOc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540057 FD On-Demand Anodyne CCR1 48 40 CCOc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540057 FD On-Demand Anodyne ABCB1 55 43 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880540073 EE On-Demand Mild F13A1 16 40 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880540073 EE On-Demand Mild GPR119 38 52 O=[N+]([O-])c1cccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540075 FD On-Demand Bother CCR1 45 39 O=[N+]([O-])c1cccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540075 FD On-Demand Bother ABCB1 48 41 O=[N+]([O-])c1cccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540076 FD On-Demand Bother CCR1 45 39 O=[N+]([O-])c1cccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540076 FD On-Demand Bother ABCB1 48 41 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccnc(C#N)c3)C2)cc1 ZINC000880540083 EG On-Demand Mild EPHX2 22 40 CC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540084 ED On-Demand Anodyne ACOX1 74 33 CC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540084 ED On-Demand Anodyne CCR1 51 42 CC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540084 ED On-Demand Anodyne ABCB1 68 45 CC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540085 ED On-Demand Anodyne ACOX1 74 33 CC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540085 ED On-Demand Anodyne CCR1 51 42 CC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540085 ED On-Demand Anodyne ABCB1 68 45 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540090 FG On-Demand Anodyne ADRB2 22 47 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540090 FG On-Demand Anodyne ADRB1 55 47 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540090 FG On-Demand Anodyne ADRB3 31 42 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540090 FG On-Demand Anodyne ACOX1 56 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540091 FG On-Demand Anodyne ADRB2 22 47 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540091 FG On-Demand Anodyne ADRB1 55 47 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540091 FG On-Demand Anodyne ADRB3 31 42 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540091 FG On-Demand Anodyne ACOX1 56 40 CCOC(=O)C1CCN(C(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)CC1 ZINC000880540099 FF On-Demand Anodyne FDFT1 21 42 O=C(Cc1ccccc1N1CCCC1=O)NCc1cc(Cl)ccc1O ZINC000880540105 FG On-Demand Clean KCNQ2 34 40 O=C(Cc1ccccc1N1CCCC1=O)NCc1cc(Cl)ccc1O ZINC000880540105 FG On-Demand Clean P2RX7 56 39 O=C(CN1CCC2(CC1)COCCO2)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880540116 GD On-Demand Anodyne HTR1A 15 44 O=C(CN1CCC2(CC1)COCCO2)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880540116 GD On-Demand Anodyne MAPK1 19 47 O=C(c1cncc2[nH]ccc12)N1CCCC[C@H]1Cc1ccccc1F ZINC000880540120 EH On-Demand Anodyne HCRTR1 20 40 O=C(c1cncc2[nH]ccc12)N1CCCC[C@@H]1Cc1ccccc1F ZINC000880540121 EH On-Demand Anodyne HCRTR1 20 40 NS(=O)(=O)c1ccc(OCCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540122 FF On-Demand Anodyne LTA4H 33 41 NS(=O)(=O)c1ccc(OCCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540122 FF On-Demand Anodyne CA1 15 47 NS(=O)(=O)c1ccc(OCCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540122 FF On-Demand Anodyne CA7 28 46 NS(=O)(=O)c1ccc(OCCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540122 FF On-Demand Anodyne CA12 17 47 NS(=O)(=O)c1ccc(OCCN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540122 FF On-Demand Anodyne CA9 19 47 O[C@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540124 DD On-Demand Anodyne ACOX1 48 34 O[C@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540124 DD On-Demand Anodyne CCR1 47 43 O[C@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540124 DD On-Demand Anodyne ABCB1 75 47 O[C@@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540125 DD On-Demand Anodyne ACOX1 48 34 O[C@@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540125 DD On-Demand Anodyne CCR1 47 43 O[C@@H](COc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540125 DD On-Demand Anodyne ABCB1 75 47 N#Cc1cc(NC(=O)N[C@H](CCO)C2CC2)ccn1 ZINC000880540126 CD On-Demand Mild TYK2 50 36 N#Cc1cc(NC(=O)N[C@@H](CCO)C2CC2)ccn1 ZINC000880540127 CD On-Demand Mild TYK2 50 36 Cc1oc(-c2ccccc2)nc1CN1CCC2(CC1)COCCO2 ZINC000880540133 EG On-Demand Anodyne PPARG 52 44 Cc1oc(-c2ccccc2)nc1CN1CCC2(CC1)COCCO2 ZINC000880540133 EG On-Demand Anodyne PPARA 55 40 Cc1oc(-c2ccccc2)nc1CN1CCC2(CC1)COCCO2 ZINC000880540133 EG On-Demand Anodyne PDE8B 70 43 C[C@H](CO)C1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880540155 DF On-Demand Anodyne PTR1 43 29 C[C@@H](CO)C1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880540156 DF On-Demand Anodyne PTR1 43 29 NC(=O)c1ccc(CN2C[C@@H]3CC[C@H]2c2ccccc23)cc1 ZINC000880540161 CG On-Demand Anodyne MBTPS1 40 32 C[C@H](CO)C1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC1 ZINC000880540192 EE On-Demand Anodyne L3MBTL3 67 39 C[C@H](CO)C1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC1 ZINC000880540193 EE On-Demand Anodyne L3MBTL3 67 39 C[C@@H](CO)C1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC1 ZINC000880540194 EE On-Demand Anodyne L3MBTL3 67 39 C[C@@H](CO)C1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC1 ZINC000880540195 EE On-Demand Anodyne L3MBTL3 67 39 C[C@H]1CCCCN1C(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540197 CG On-Demand Anodyne CPT1A 57 34 C[C@@H]1CCCCN1C(=O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540198 CG On-Demand Anodyne CPT1A 57 34 C[C@H](CO)C1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880540199 CE On-Demand Anodyne L3MBTL3 53 35 C[C@@H](CO)C1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880540200 CE On-Demand Anodyne L3MBTL3 53 35 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880540215 GE On-Demand Anodyne F11 48 40 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880540216 GE On-Demand Anodyne F11 48 40 O=C(CN1CCC2(CC1)COCCO2)N1CCC(Cc2ccccc2)CC1 ZINC000880540221 FE On-Demand Anodyne GRIN2B 75 47 O=C(CN1CCC2(CC1)COCCO2)N1CCC(Cc2ccccc2)CC1 ZINC000880540221 FE On-Demand Anodyne SIGMAR1 21 41 O=C(CN1CCC2(CC1)COCCO2)N1CCC(Cc2ccccc2)CC1 ZINC000880540221 FE On-Demand Anodyne CCR3 26 40 COc1ccc(N2CCCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880540240 FF On-Demand Mild PDGFRB 57 43 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880540254 GF On-Demand Anodyne PREP 64 37 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880540254 GF On-Demand Anodyne L3MBTL3 42 36 CCCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540266 EF On-Demand Anodyne LTA4H 51 47 CCCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540266 EF On-Demand Anodyne HRH3 26 44 CCCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540266 EF On-Demand Anodyne PSMB2 43 42 CCCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540266 EF On-Demand Anodyne PSMB1 46 40 N#CCc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540272 ED On-Demand Mild CCR1 42 36 N#CCc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540273 ED On-Demand Mild CCR1 42 36 C=CCc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540275 GE On-Demand Mild CCR1 49 41 C=CCc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540275 GE On-Demand Mild ABCB1 48 36 C=CCc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540277 GE On-Demand Mild CCR1 49 41 C=CCc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540277 GE On-Demand Mild ABCB1 48 36 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880540291 GE On-Demand Anodyne KLKB1 24 40 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880540291 GE On-Demand Anodyne F11 53 44 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880540292 GE On-Demand Anodyne KLKB1 24 40 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880540292 GE On-Demand Anodyne F11 53 44 N#Cc1cc(NC(=O)NCCOC2CCC2)ccn1 ZINC000880540302 CD On-Demand Mild ADRB1 41 32 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCC1 ZINC000880540308 CE On-Demand Anodyne PREP 45 35 O=C(CN1C[C@@H]2CC[C@H]1c1ccccc12)N1CCC1 ZINC000880540308 CE On-Demand Anodyne L3MBTL3 43 37 CCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540312 DE On-Demand Anodyne ESR1 41 37 CCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540312 DE On-Demand Anodyne LTA4H 53 44 CCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540312 DE On-Demand Anodyne HRH3 28 44 CCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540312 DE On-Demand Anodyne PSMB2 43 42 CCOc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540312 DE On-Demand Anodyne PSMB1 46 40 O=[N+]([O-])c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540319 CD On-Demand Bother SIGMAR1 23 49 O=[N+]([O-])c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540319 CD On-Demand Bother KCNJ1 31 67 CCOc1ccccc1CN1CCC2(CC1)COCCO2 ZINC000880540321 CE On-Demand Anodyne HCN1 49 35 CCOc1ccccc1CN1CCC2(CC1)COCCO2 ZINC000880540321 CE On-Demand Anodyne HCN4 40 33 c1ccc2c(c1)oc1ccc(CN3CCC4(CC3)COCCO4)cc12 ZINC000880540326 EH On-Demand Anodyne MCHR2 76 36 N#Cc1cc(NC(=O)NC2CCN(c3ccc(OC(F)F)cc3)CC2)ccn1 ZINC000880540329 GG On-Demand Mild EPHX2 44 40 O[C@H](COc1ccc(Br)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540335 GE On-Demand Anodyne CCR1 47 38 O[C@H](COc1ccc(Br)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540335 GE On-Demand Anodyne ABCB1 42 38 O[C@@H](COc1ccc(Br)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540337 GE On-Demand Anodyne CCR1 47 38 O[C@@H](COc1ccc(Br)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540337 GE On-Demand Anodyne ABCB1 42 38 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA2 40 53 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA1 34 46 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA5B 48 37 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA4 42 53 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA5A 55 37 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA12 22 48 NS(=O)(=O)c1cccc(NC(=O)CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540359 FE On-Demand Anodyne CA9 25 48 Cc1nn(CC(=O)NCc2cc(Cl)ccc2O)c(=O)o1 ZINC000880540364 CC On-Demand Clean P2RX7 59 40 O=C(CN1CCC2(CC1)COCCO2)N1CCc2ccccc21 ZINC000880540367 DD On-Demand Anodyne DRD4 15 53 C/C=C\c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540373 GE On-Demand Anodyne CCR1 48 40 C/C=C\c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540373 GE On-Demand Anodyne ABCB1 47 39 C/C=C\c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540376 GE On-Demand Anodyne CCR1 48 40 C/C=C\c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540376 GE On-Demand Anodyne ABCB1 47 39 C/C=C/c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540378 GE On-Demand Anodyne CCR1 48 40 C/C=C/c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540378 GE On-Demand Anodyne ABCB1 47 39 C/C=C/c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540380 GE On-Demand Anodyne CCR1 48 40 C/C=C/c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540380 GE On-Demand Anodyne ABCB1 47 39 O=S(=O)(CCN1CCC2(CC1)COCCO2)c1ccc(Cl)cc1 ZINC000880540381 FD On-Demand Anodyne CCR1 25 41 NC(=O)c1cccc(CN2C[C@@H]3CC[C@H]2c2ccccc23)c1 ZINC000880540392 CG On-Demand Anodyne KCNH2 42 42 CS(=O)(=O)C1CCC(C(=O)NCc2cc(Cl)ccc2O)CC1 ZINC000880540400 EE On-Demand Clean F2 18 40 CS(=O)(=O)C1CCC(C(=O)NCc2cc(Cl)ccc2O)CC1 ZINC000880540400 EE On-Demand Clean P2RX7 53 43 CS(=O)(=O)C1CCC(C(=O)NCc2cc(Cl)ccc2O)CC1 ZINC000880540400 EE On-Demand Clean EPHX2 22 50 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540406 FG On-Demand Anodyne HTR1A 15 40 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540406 FG On-Demand Anodyne SLC6A4 15 40 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540406 FG On-Demand Anodyne ADRA1A 16 41 COc1cccc(OC)c1OC[C@@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540406 FG On-Demand Anodyne ABCB1 31 40 COc1cccc(OC)c1OC[C@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540407 FG On-Demand Anodyne HTR1A 15 40 COc1cccc(OC)c1OC[C@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540407 FG On-Demand Anodyne SLC6A4 15 40 COc1cccc(OC)c1OC[C@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540407 FG On-Demand Anodyne ADRA1A 16 41 COc1cccc(OC)c1OC[C@H](O)CN1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880540407 FG On-Demand Anodyne ABCB1 31 40 O=C(C[C@H]1CCNC1=O)NCc1cc(Cl)ccc1O ZINC000880540410 CD On-Demand Clean P2RX7 40 37 O=C(C[C@@H]1CCNC1=O)NCc1cc(Cl)ccc1O ZINC000880540411 CD On-Demand Clean P2RX7 40 37 O=C1NCC[C@@H]1CC(=O)N1CCCC[C@H]1Cc1ccccc1F ZINC000880540422 DE On-Demand Anodyne DPP4 16 45 O=C1NCC[C@H]1CC(=O)N1CCCC[C@H]1Cc1ccccc1F ZINC000880540423 DE On-Demand Anodyne DPP4 16 45 O=C1NCC[C@H]1CC(=O)N1CCCC[C@@H]1Cc1ccccc1F ZINC000880540425 DE On-Demand Anodyne DPP4 16 45 CN(C[C@@H]1CCN(C(=O)Nc2ccnc(C#N)c2)C1)C(=O)OC(C)(C)C ZINC000880540450 FF On-Demand Mild GPR119 20 44 O=C(CN1CCC2(CC1)COCCO2)N[C@H](Cc1ccccc1)c1ccccc1 ZINC000880540451 GF On-Demand Anodyne PSMB8 42 42 O=C(CN1CCC2(CC1)COCCO2)N[C@@H](Cc1ccccc1)c1ccccc1 ZINC000880540452 GF On-Demand Anodyne PSMB8 42 42 O[C@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540457 FE On-Demand Anodyne ACOX1 81 40 O[C@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540457 FE On-Demand Anodyne CCR1 48 42 O[C@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540457 FE On-Demand Anodyne ABCB1 67 44 O[C@@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540458 FE On-Demand Anodyne ACOX1 81 40 O[C@@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540458 FE On-Demand Anodyne CCR1 48 42 O[C@@H](COc1ccc2ccccc2c1)CN1CCC2(CC1)COCCO2 ZINC000880540458 FE On-Demand Anodyne ABCB1 67 44 CN(Cc1ccc(Cl)c(Cl)c1)C(=O)CN1CCC2(CC1)COCCO2 ZINC000880540463 GF On-Demand Anodyne OPRK1 23 45 CN(Cc1ccc(Cl)c(Cl)c1)C(=O)CN1CCC2(CC1)COCCO2 ZINC000880540463 GF On-Demand Anodyne TACR3 38 42 O[C@@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540468 FE On-Demand Anodyne ADRB2 17 54 O[C@@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540468 FE On-Demand Anodyne ADRB1 16 48 O[C@@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540468 FE On-Demand Anodyne CCR1 50 46 O[C@@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540468 FE On-Demand Anodyne ABCB1 78 52 O[C@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540469 FE On-Demand Anodyne ADRB2 17 54 O[C@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540469 FE On-Demand Anodyne ADRB1 16 48 O[C@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540469 FE On-Demand Anodyne CCR1 50 46 O[C@H](COc1cccc2ccccc12)CN1CCC2(CC1)COCCO2 ZINC000880540469 FE On-Demand Anodyne ABCB1 78 52 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne DRD4 15 41 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne ACHE 15 43 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne SIGMAR1 47 39 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne PRNP 49 38 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne HDAC1 23 44 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne MCHR1 19 40 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne NPFFR1 48 41 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne NOD1 20 47 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne NOD2 52 44 O=C(Nc1ccccc1)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540472 FG On-Demand Anodyne KCNK3 43 34 c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540495 BE On-Demand Anodyne DRD4 27 44 c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540495 BE On-Demand Anodyne ACHE 17 43 c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540495 BE On-Demand Anodyne SIGMAR1 91 55 Fc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540507 CE On-Demand Anodyne SIGMAR1 40 50 NC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540519 CD On-Demand Anodyne CHRM3 17 44 NC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540519 CD On-Demand Anodyne MCHR2 40 34 NC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540519 CD On-Demand Anodyne NPFFR1 46 36 Fc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540543 CE On-Demand Anodyne SIGMAR1 37 47 NS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540549 FC On-Demand Anodyne LTA4H 44 39 NS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540549 FC On-Demand Anodyne CA7 19 43 NS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540549 FC On-Demand Anodyne HRH3 15 60 NS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540549 FC On-Demand Anodyne MMP13 17 40 NS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540549 FC On-Demand Anodyne PSMB1 40 36 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(F)c1 ZINC000880540552 DD On-Demand Anodyne EPHX2 17 40 Cc1nc(C(C)C)ncc1C(=O)Nc1cc(F)cc(N(C)C)c1 ZINC000880540554 DG On-Demand Anodyne JUN 21 44 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)COC1CC1 ZINC000880540555 CD On-Demand Anodyne TIMP3 85 39 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)COC1CC1 ZINC000880540555 CD On-Demand Anodyne F11 42 36 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)COC1CC1 ZINC000880540556 CD On-Demand Anodyne TIMP3 85 39 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)COC1CC1 ZINC000880540556 CD On-Demand Anodyne F11 42 36 O[C@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540560 ED On-Demand Anodyne ACOX1 43 35 O[C@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540560 ED On-Demand Anodyne CCR1 54 46 O[C@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540560 ED On-Demand Anodyne ABCB1 45 38 O[C@@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540561 ED On-Demand Anodyne ACOX1 43 35 O[C@@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540561 ED On-Demand Anodyne CCR1 54 46 O[C@@H](COc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540561 ED On-Demand Anodyne ABCB1 45 38 O=C(CN1CCC2(CC1)COCCO2)NCCc1ccc(Cl)cc1 ZINC000880540572 FD On-Demand Anodyne CCR1 26 40 COc1ccc(N2CCC(NC(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880540574 FF On-Demand Mild EPHX2 48 40 COc1ccc(N2CCC(NC(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880540574 FF On-Demand Mild PDGFRA 28 42 COC(=O)[C@@H](CC(C)C)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880540577 EC On-Demand Anodyne PSMB8 45 41 O[C@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540585 GE On-Demand Anodyne ACOX1 57 33 O[C@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540585 GE On-Demand Anodyne CCR1 46 39 O[C@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540585 GE On-Demand Anodyne ABCB1 53 42 O[C@@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540586 GE On-Demand Anodyne ACOX1 57 33 O[C@@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540586 GE On-Demand Anodyne CCR1 46 39 O[C@@H](COc1cccc(Br)c1)CN1CCC2(CC1)COCCO2 ZINC000880540586 GE On-Demand Anodyne ABCB1 53 42 O[C@H](COc1ccc(Cl)cc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540587 GF On-Demand Anodyne CCR1 59 51 O[C@H](COc1ccc(Cl)cc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540587 GF On-Demand Anodyne ABCB1 49 40 O[C@@H](COc1ccc(Cl)cc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540588 GF On-Demand Anodyne CCR1 59 51 O[C@@H](COc1ccc(Cl)cc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540588 GF On-Demand Anodyne ABCB1 49 40 COC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540589 DD On-Demand Anodyne CHRM3 22 48 COC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540589 DD On-Demand Anodyne MCHR2 52 36 O[C@@H](COc1c(Cl)cccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540591 GF On-Demand Anodyne CCR1 47 42 O[C@@H](COc1c(Cl)cccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540591 GF On-Demand Anodyne ABCB1 57 40 O[C@H](COc1c(Cl)cccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540592 GF On-Demand Anodyne CCR1 47 42 O[C@H](COc1c(Cl)cccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540592 GF On-Demand Anodyne ABCB1 57 40 COc1ccc(OC)c([C@H](C)NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540603 GD On-Demand Anodyne PSMB8 38 40 CN(Cc1ccc(F)cc1)C(=O)CN1CCC2(CC1)COCCO2 ZINC000880540614 ED On-Demand Anodyne TACR3 23 40 O[C@H](COCc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540616 FE On-Demand Anodyne CCR1 45 40 O[C@@H](COCc1ccc(Cl)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540617 FE On-Demand Anodyne CCR1 45 40 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540618 GF On-Demand Anodyne ACOX1 72 39 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540618 GF On-Demand Anodyne CCR1 49 42 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540618 GF On-Demand Anodyne ABCB1 70 44 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540619 GF On-Demand Anodyne ACOX1 72 39 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540619 GF On-Demand Anodyne CCR1 49 42 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540619 GF On-Demand Anodyne ABCB1 70 44 O=C(CCN1CCC2(CC1)COCCO2)NC(=O)Nc1ccccc1 ZINC000880540637 ED On-Demand Anodyne EPHX2 28 45 O[C@@H](COC(c1ccccc1)c1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540640 GG On-Demand Anodyne SLC6A3 26 45 O[C@@H](COC(c1ccccc1)c1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540640 GG On-Demand Anodyne ABCB1 53 41 O[C@H](COC(c1ccccc1)c1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540641 GG On-Demand Anodyne SLC6A3 26 45 O[C@H](COC(c1ccccc1)c1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540641 GG On-Demand Anodyne ABCB1 53 41 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880540653 EE On-Demand Mild P2RY12 18 42 c1ccc(C(OCCN2CCC3(CC2)COCCO3)c2ccccc2)cc1 ZINC000880540660 FH On-Demand Anodyne SLC6A4 25 52 c1ccc(C(OCCN2CCC3(CC2)COCCO3)c2ccccc2)cc1 ZINC000880540660 FH On-Demand Anodyne SLC6A3 67 63 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880540675 GF On-Demand Anodyne TACR2 47 33 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880540675 GF On-Demand Anodyne PSMB8 41 36 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880540676 GF On-Demand Anodyne TACR2 47 33 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880540676 GF On-Demand Anodyne PSMB8 41 36 COC(=O)c1sccc1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880540678 FD On-Demand Anodyne FAS 44 47 Brc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540680 EF On-Demand Anodyne SIGMAR1 27 43 O[C@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540681 GG On-Demand Anodyne ACOX1 50 39 O[C@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540681 GG On-Demand Anodyne CCR1 44 41 O[C@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540681 GG On-Demand Anodyne ABCB1 70 44 O[C@@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540682 GG On-Demand Anodyne ACOX1 50 39 O[C@@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540682 GG On-Demand Anodyne CCR1 44 41 O[C@@H](COc1ccc(Oc2ccccc2)cc1)CN1CCC2(CC1)COCCO2 ZINC000880540682 GG On-Demand Anodyne ABCB1 70 44 O=[N+]([O-])c1ccccc1CN1CCC2(CC1)COCCO2 ZINC000880540690 CD On-Demand Bother COLA 60 32 N#Cc1cc(NC(=O)N2CCC([C@H](O)c3ccc(Cl)cc3)CC2)ccn1 ZINC000880540691 FH On-Demand Mild TYK2 53 37 N#Cc1cc(NC(=O)N2CCC([C@@H](O)c3ccc(Cl)cc3)CC2)ccn1 ZINC000880540692 FH On-Demand Mild TYK2 53 37 O=C(CN1CCC2(CC1)COCCO2)NCCCc1ccccc1 ZINC000880540698 ED On-Demand Anodyne CRTM 33 42 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne CASR 25 47 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne KCNQ2 31 40 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne NPY2R 51 40 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne MTNR1A 15 40 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne MTNR1B 21 42 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne TAAR1 32 40 COc1cccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540702 GG On-Demand Anodyne AKR1C3 17 40 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne CASR 25 47 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne KCNQ2 31 40 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne NPY2R 51 40 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne MTNR1A 15 40 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne MTNR1B 21 42 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne TAAR1 32 40 COc1cccc(NC(=O)[C@@H](c2ccccc2)N2CCC3(CC2)COCCO3)c1 ZINC000880540703 GG On-Demand Anodyne AKR1C3 17 40 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880540719 EF On-Demand Anodyne F11 40 35 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880540720 EF On-Demand Anodyne F11 40 35 C[C@@H](OC[C@H](O)CN1CCC2(CC1)COCCO2)c1ccc(Cl)cc1 ZINC000880540723 FF On-Demand Anodyne CCR1 43 41 C[C@@H](OC[C@@H](O)CN1CCC2(CC1)COCCO2)c1ccc(Cl)cc1 ZINC000880540725 FF On-Demand Anodyne CCR1 43 41 COc1cc2c(cc1OC)CN(C(=O)CN1CCC3(CC1)COCCO3)CC2 ZINC000880540727 GD On-Demand Anodyne ABCB1 18 46 O[C@H](COCc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540729 FE On-Demand Anodyne CCR1 42 39 O[C@@H](COCc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540730 FE On-Demand Anodyne CCR1 42 39 Fc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880540748 CE On-Demand Anodyne LTA4H 31 42 Fc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880540748 CE On-Demand Anodyne CHRNA10 32 40 c1ccc(Cc2nc(CN3CCC4(CC3)COCCO4)cs2)cc1 ZINC000880540751 EG On-Demand Anodyne SIGMAR1 22 41 c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540755 CD On-Demand Anodyne LTA4H 63 51 c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540755 CD On-Demand Anodyne HRH3 26 50 c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540755 CD On-Demand Anodyne PSMB2 43 42 c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540755 CD On-Demand Anodyne PSMB1 46 43 C[C@H](C(=O)Nc1ccccc1C(F)(F)F)N1CCC2(CC1)COCCO2 ZINC000880540764 FF On-Demand Anodyne RBP4 50 33 O=C(CN1CCC2(CC1)COCCO2)N1CCN(Cc2ccccc2)CC1 ZINC000880540803 FD On-Demand Anodyne DRD4 30 40 O=C(CN1CCC2(CC1)COCCO2)N1CCN(Cc2ccccc2)CC1 ZINC000880540803 FD On-Demand Anodyne SIGMAR1 62 43 O=C(CN1CCC2(CC1)COCCO2)N1CCN(Cc2ccccc2)CC1 ZINC000880540803 FD On-Demand Anodyne FAAH 17 41 O=C(CN1CCC2(CC1)COCCO2)N1CCN(Cc2ccccc2)CC1 ZINC000880540803 FD On-Demand Anodyne NPFFR1 40 36 c1ccc(C(c2ccccc2)N2CCC3(CC2)COCCO3)cc1 ZINC000880540808 DH On-Demand Anodyne OPRL1 35 54 c1ccc(-c2ncc(CN3CCC4(CC3)COCCO4)s2)cc1 ZINC000880540812 EG On-Demand Anodyne MGEA5 31 41 O=C(CN1CCC2(CC1)COCCO2)NCC1(c2ccccc2)CCCC1 ZINC000880540813 FE On-Demand Anodyne NPFFR1 35 44 O=[N+]([O-])c1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880540818 DD On-Demand Bother LTA4H 15 56 NC(=O)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540823 CD On-Demand Anodyne NPFFR1 44 38 c1ccc(-n2cc(CN3CCC4(CC3)COCCO4)cn2)cc1 ZINC000880540831 DE On-Demand Anodyne DRD4 15 58 C[C@H](C(=O)Nc1ccccc1Cl)N1CCC2(CC1)COCCO2 ZINC000880540833 EF On-Demand Anodyne KCNQ2 45 35 C[C@H](C(=O)Nc1ccccc1Cl)N1CCC2(CC1)COCCO2 ZINC000880540833 EF On-Demand Anodyne EPHB3 42 34 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne DRD2 19 56 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne DRD4 15 56 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne HTR2A 20 56 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne LTA4H 31 46 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne HRH3 69 51 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne SIGMAR1 16 49 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne HTR5A 15 47 Fc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880540835 DE On-Demand Anodyne EPHX2 17 43 O=C(CCN1CCC2(CC1)COCCO2)N[C@H]1CCCc2ccccc21 ZINC000880540836 FE On-Demand Anodyne HTR7 17 55 O=C(CCN1CCC2(CC1)COCCO2)N[C@H]1CCCc2ccccc21 ZINC000880540836 FE On-Demand Anodyne BDKRB1 41 37 O=C(CCN1CCC2(CC1)COCCO2)N[C@@H]1CCCc2ccccc21 ZINC000880540837 FE On-Demand Anodyne HTR7 17 55 O=C(CCN1CCC2(CC1)COCCO2)N[C@@H]1CCCc2ccccc21 ZINC000880540837 FE On-Demand Anodyne BDKRB1 41 37 Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540854 DD On-Demand Anodyne ACOX1 78 35 Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540854 DD On-Demand Anodyne CCR1 48 40 Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540854 DD On-Demand Anodyne ABCB1 62 41 Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540855 DD On-Demand Anodyne ACOX1 78 35 Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540855 DD On-Demand Anodyne CCR1 48 40 Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880540855 DD On-Demand Anodyne ABCB1 62 41 N#Cc1c(NC(=O)CCN2CCC3(CC2)COCCO3)sc2c1CCCC2 ZINC000880540874 GF On-Demand Mild VIPR1 31 50 O=[N+]([O-])c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880540879 CD On-Demand Bother SIGMAR1 24 52 N#Cc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880540892 CD On-Demand Mild SIGMAR1 21 44 O[C@H](COc1cc(Cl)ccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540898 GF On-Demand Anodyne CCR1 59 51 O[C@H](COc1cc(Cl)ccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540898 GF On-Demand Anodyne ABCB1 48 40 O[C@@H](COc1cc(Cl)ccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540899 GF On-Demand Anodyne CCR1 59 51 O[C@@H](COc1cc(Cl)ccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880540899 GF On-Demand Anodyne ABCB1 48 40 O=C(CN1CCC2(CC1)COCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880540921 GD On-Demand Anodyne HCN1 53 33 O=C(CN1CCC2(CC1)COCCO2)NCC1(N2CCOCC2)CCCCC1 ZINC000880540921 GD On-Demand Anodyne HCN4 49 33 O[C@H](COCc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540923 DD On-Demand Anodyne ABCB1 57 42 O[C@@H](COCc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880540924 DD On-Demand Anodyne ABCB1 57 42 COc1ccccc1COC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880540926 FD On-Demand Anodyne CCR1 40 40 COc1ccccc1COC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880540926 FD On-Demand Anodyne ABCB1 48 41 COc1ccccc1COC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880540927 FD On-Demand Anodyne CCR1 40 40 COc1ccccc1COC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880540927 FD On-Demand Anodyne ABCB1 48 41 Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(C)c1 ZINC000880540934 ED On-Demand Anodyne CCR1 51 43 Cc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(C)c1 ZINC000880540934 ED On-Demand Anodyne ABCB1 63 48 Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(C)c1 ZINC000880540935 ED On-Demand Anodyne CCR1 51 43 Cc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(C)c1 ZINC000880540935 ED On-Demand Anodyne ABCB1 63 48 COC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540937 GD On-Demand Anodyne CCR1 54 46 COC(=O)c1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540937 GD On-Demand Anodyne ABCB1 64 43 COC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540938 GD On-Demand Anodyne CCR1 54 46 COC(=O)c1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880540938 GD On-Demand Anodyne ABCB1 64 43 O[C@H](COc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880540939 ED On-Demand Anodyne CCR1 54 51 O[C@H](COc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880540939 ED On-Demand Anodyne ABCB1 70 48 O[C@@H](COc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880540940 ED On-Demand Anodyne CCR1 54 51 O[C@@H](COc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880540940 ED On-Demand Anodyne ABCB1 70 48 CCOC(=O)N1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880540953 DD On-Demand Mild P2RY12 50 47 CCOC(=O)N1CCCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880540953 DD On-Demand Mild PDGFRB 45 38 c1cc2c(cc1CCN1CCC3(CC1)COCCO3)CCO2 ZINC000880540977 DE On-Demand Anodyne KCNJ1 45 41 CC(=O)c1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880540981 ED On-Demand Anodyne AKR1C3 18 40 N#CCCn1cc(C(=O)CN2CCC3(CC2)COCCO3)c2ccccc21 ZINC000880540993 FF On-Demand Mild CNR1 17 45 N#CCCn1cc(C(=O)CN2CCC3(CC2)COCCO3)c2ccccc21 ZINC000880540993 FF On-Demand Mild CNR2 20 45 N#CCCn1cc(C(=O)CN2CCC3(CC2)COCCO3)c2ccccc21 ZINC000880540993 FF On-Demand Mild ADCY5 15 41 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(F)c1 ZINC000880541003 DE On-Demand Anodyne EPHX2 24 43 Fc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541010 CE On-Demand Anodyne ESR2 22 42 Fc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541010 CE On-Demand Anodyne LTA4H 50 53 Fc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541010 CE On-Demand Anodyne HRH3 23 44 Fc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541010 CE On-Demand Anodyne PSMB2 41 42 Fc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541010 CE On-Demand Anodyne PSMB1 44 40 N#Cc1cc(NC(=O)NC2CCN(CC3CCCCC3)CC2)ccn1 ZINC000880541012 EG On-Demand Mild CCR3 42 43 N#Cc1cc(NC(=O)NC2CCN(CC3CCCCC3)CC2)ccn1 ZINC000880541012 EG On-Demand Mild EPHX2 46 43 N#Cc1cc(NC(=O)NC2CCN(CC3CCCCC3)CC2)ccn1 ZINC000880541012 EG On-Demand Mild CXCR3 18 45 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne SLC6A4 15 45 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne LTA4H 31 44 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne HRH3 77 51 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne SIGMAR1 23 52 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne HTR5A 17 40 COc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541013 DE On-Demand Anodyne EBP 32 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541020 FD On-Demand Anodyne ADRB1 27 47 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541020 FD On-Demand Anodyne ADRB3 16 42 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541020 FD On-Demand Anodyne ACOX1 79 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541020 FD On-Demand Anodyne CCR1 53 47 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541020 FD On-Demand Anodyne ABCB1 57 42 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541021 FD On-Demand Anodyne ADRB1 27 47 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541021 FD On-Demand Anodyne ADRB3 16 42 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541021 FD On-Demand Anodyne ACOX1 79 40 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541021 FD On-Demand Anodyne CCR1 53 47 CC(=O)Nc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541021 FD On-Demand Anodyne ABCB1 57 42 COc1ccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)cc1 ZINC000880541046 GG On-Demand Anodyne NPY2R 43 36 COc1ccc(NC(=O)[C@H](c2ccccc2)N2CCC3(CC2)COCCO3)cc1 ZINC000880541046 GG On-Demand Anodyne AKR1C2 29 40 COC(=O)c1ccc(CN2CCC3(CC2)COCCO3)cc1F ZINC000880541072 DD On-Demand Anodyne MCHR2 46 35 O[C@@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541073 GF On-Demand Anodyne ACOX1 82 41 O[C@@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541073 GF On-Demand Anodyne CCR1 51 42 O[C@@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541073 GF On-Demand Anodyne ABCB1 45 38 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541075 GF On-Demand Anodyne ACOX1 82 41 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541075 GF On-Demand Anodyne CCR1 51 42 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880541075 GF On-Demand Anodyne ABCB1 45 38 O[C@H](COc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880541088 ED On-Demand Anodyne CCR1 55 50 O[C@H](COc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880541088 ED On-Demand Anodyne ABCB1 70 48 O[C@@H](COc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880541090 ED On-Demand Anodyne CCR1 55 50 O[C@@H](COc1ccccc1Cl)CN1CCC2(CC1)COCCO2 ZINC000880541090 ED On-Demand Anodyne ABCB1 70 48 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCc2nncn2CC1 ZINC000880541094 FE On-Demand Anodyne CCR5 17 40 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCc2nncn2CC1 ZINC000880541094 FE On-Demand Anodyne F11 47 38 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880541095 FE On-Demand Anodyne CCR5 17 40 Cn1ccnc1[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880541095 FE On-Demand Anodyne F11 47 38 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@H]1CCc2nncn2CC1 ZINC000880541097 FE On-Demand Anodyne CCR5 17 40 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@H]1CCc2nncn2CC1 ZINC000880541097 FE On-Demand Anodyne F11 47 38 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880541098 FE On-Demand Anodyne CCR5 17 40 Cn1ccnc1[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880541098 FE On-Demand Anodyne F11 47 38 c1nc(CN2CCC3(CC2)COCCO3)cs1 ZINC000880541099 CD On-Demand Anodyne SCN5A 40 33 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Oc2ccccc2)c1 ZINC000880541107 GG On-Demand Anodyne LTA4H 25 45 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Oc2ccccc2)c1 ZINC000880541107 GG On-Demand Anodyne ACOX1 23 44 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Oc2ccccc2)c1 ZINC000880541107 GG On-Demand Anodyne FAAH 17 42 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Oc2ccccc2)c1 ZINC000880541107 GG On-Demand Anodyne EPHX2 23 42 CCON(C)C(=O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880541108 DE On-Demand Anodyne NQO2 21 44 CCON(C)C(=O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880541108 DE On-Demand Anodyne MTNR1B 29 46 CCON(C)C(=O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880541109 DE On-Demand Anodyne NQO2 21 44 CCON(C)C(=O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880541109 DE On-Demand Anodyne MTNR1B 29 46 C[C@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc(Cl)cc1 ZINC000880541112 FE On-Demand Anodyne CCR1 46 36 C[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccc(Cl)cc1 ZINC000880541115 FE On-Demand Anodyne CCR1 46 36 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880541122 FF On-Demand Anodyne CASR 15 46 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880541122 FF On-Demand Anodyne EPHX2 35 49 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC2(CC1)COCCO2 ZINC000880541131 ED On-Demand Anodyne DRD4 33 56 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCC2(CC1)COCCO2 ZINC000880541131 ED On-Demand Anodyne TPP2 54 32 CC(=O)c1cccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541149 ED On-Demand Anodyne ACOX1 78 37 CC(=O)c1cccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541149 ED On-Demand Anodyne CCR1 50 43 CC(=O)c1cccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541149 ED On-Demand Anodyne ABCB1 76 59 CC(=O)c1cccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541150 ED On-Demand Anodyne ACOX1 78 37 CC(=O)c1cccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541150 ED On-Demand Anodyne CCR1 50 43 CC(=O)c1cccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)c1 ZINC000880541150 ED On-Demand Anodyne ABCB1 76 59 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc2ccccc2c1 ZINC000880541157 EF On-Demand Anodyne IMDH_CRYPV 19 40 COC(=O)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880541171 DD On-Demand Anodyne SIGMAR1 32 45 COC(=O)c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880541171 DD On-Demand Anodyne NPFFR1 37 47 FC(F)(F)COc1ccccc1CN1CCC2(CC1)COCCO2 ZINC000880541189 EG On-Demand Anodyne CCR8 16 40 O=C(CN1CCC2(CC1)COCCO2)Nc1ccccc1Cl ZINC000880541195 DE On-Demand Anodyne EPHB3 49 35 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(-c2ccccc2)cc1 ZINC000880541203 FG On-Demand Anodyne SLC1A2 21 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H](Cc1ccccc1)c1nccn1C ZINC000880541217 FF On-Demand Anodyne F11 42 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H](Cc1ccccc1)c1nccn1C ZINC000880541218 FF On-Demand Anodyne F11 42 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](Cc1ccccc1)c1nccn1C ZINC000880541219 FF On-Demand Anodyne F11 42 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](Cc1ccccc1)c1nccn1C ZINC000880541220 FF On-Demand Anodyne F11 42 36 c1ccc2cc(CN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880541226 CG On-Demand Anodyne SIGMAR1 40 40 c1ccc2cc(CN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880541226 CG On-Demand Anodyne MCHR2 55 32 O=C(CN1CCC2(CC1)COCCO2)NCc1ccccc1 ZINC000880541254 DD On-Demand Anodyne NPFFR1 42 37 CCOc1ccccc1NC(=O)[C@H](C)N1CCC2(CC1)COCCO2 ZINC000880541293 EE On-Demand Anodyne HCN1 64 44 CCOc1ccccc1NC(=O)[C@H](C)N1CCC2(CC1)COCCO2 ZINC000880541293 EE On-Demand Anodyne HCN4 54 39 CCOc1ccccc1NC(=O)[C@@H](C)N1CCC2(CC1)COCCO2 ZINC000880541294 EE On-Demand Anodyne HCN1 64 44 CCOc1ccccc1NC(=O)[C@@H](C)N1CCC2(CC1)COCCO2 ZINC000880541294 EE On-Demand Anodyne HCN4 54 39 COc1ccc(NC(=O)[C@H](C)N2CCC3(CC2)COCCO3)c(OC)c1 ZINC000880541301 FD On-Demand Anodyne CCR1 34 40 O=C1c2ccccc2C(=O)N1CCCCN1CCC2(CC1)COCCO2 ZINC000880541315 FD On-Demand Anodyne HTR1A 17 52 c1ccc2c(c1)OC[C@H](CN1CCC3(CC1)COCCO3)O2 ZINC000880541339 DD On-Demand Anodyne ADRA2B 19 49 c1ccc2c(c1)OC[C@@H](CN1CCC3(CC1)COCCO3)O2 ZINC000880541340 DD On-Demand Anodyne ADRA2B 19 49 c1ccc(Cn2nnnc2CN2CCC3(CC2)COCCO3)cc1 ZINC000880541363 ED On-Demand Anodyne SIGMAR1 27 40 CC(=O)c1cccc(NC(=O)[C@H](C)N2CCC3(CC2)COCCO3)c1 ZINC000880541374 EE On-Demand Anodyne AKR1C3 19 40 CC(=O)c1cccc(NC(=O)[C@@H](C)N2CCC3(CC2)COCCO3)c1 ZINC000880541376 EE On-Demand Anodyne AKR1C3 19 40 C[C@H](NC(=O)CN1CCC2(CC1)COCCO2)c1cccc2ccccc12 ZINC000880541387 FF On-Demand Anodyne PSMB8 38 40 C[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1cccc2ccccc12 ZINC000880541390 FF On-Demand Anodyne PSMB8 38 40 CS(=O)(=O)C1CCC(C(=O)Nc2ccc3c(c2)CCCCC3)CC1 ZINC000880541404 EG On-Demand Anodyne EPHX2 15 40 Fc1ccc(CN2CCC3(CC2)COCCO3)c(Cl)c1 ZINC000880541407 CF On-Demand Anodyne P2RX7 36 42 O=C(c1ccc(CN2CCC3(CC2)COCCO3)cc1)N1CCCC1 ZINC000880541424 EE On-Demand Anodyne CCR8 23 40 O=C(c1ccc(CN2CCC3(CC2)COCCO3)cc1)N1CCCC1 ZINC000880541424 EE On-Demand Anodyne L3MBTL3 72 53 C=CCN1CCC(NC(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541428 CD On-Demand Mild EPHX2 40 40 N#Cc1cc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)ccn1 ZINC000880541437 DH On-Demand Mild EPHX2 27 41 N#Cc1cc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)ccn1 ZINC000880541437 DH On-Demand Mild MCHR1 15 49 N#Cc1cc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)ccn1 ZINC000880541437 DH On-Demand Mild MAP3K12 42 40 N#Cc1cc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)ccn1 ZINC000880541438 DH On-Demand Mild EPHX2 27 41 N#Cc1cc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)ccn1 ZINC000880541438 DH On-Demand Mild MCHR1 15 49 N#Cc1cc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)ccn1 ZINC000880541438 DH On-Demand Mild MAP3K12 42 40 COC(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)c(Cl)c1 ZINC000880541445 FE On-Demand Anodyne SLC9A1 46 34 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Oc2ccccc2)cc1 ZINC000880541461 GG On-Demand Anodyne LTA4H 51 52 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Oc2ccccc2)cc1 ZINC000880541461 GG On-Demand Anodyne ACOX1 27 42 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Oc2ccccc2)cc1 ZINC000880541461 GG On-Demand Anodyne EPHX2 21 42 CSc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541468 DF On-Demand Anodyne LTA4H 44 41 CSc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541468 DF On-Demand Anodyne HRH3 19 42 CSc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541468 DF On-Demand Anodyne PSMB2 40 40 CSc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541468 DF On-Demand Anodyne PSMB1 43 38 CNC(=O)[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880541478 FC On-Demand Anodyne PSMB8 40 41 O[C@H](COCc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880541481 ED On-Demand Anodyne CCR1 40 39 O[C@@H](COCc1ccccc1F)CN1CCC2(CC1)COCCO2 ZINC000880541484 ED On-Demand Anodyne CCR1 40 39 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880541487 FF On-Demand Anodyne EPHX2 40 48 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(C(F)(F)F)cc1 ZINC000880541487 FF On-Demand Anodyne TRPM8 43 43 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541492 EE On-Demand Mild PDGFRB 41 39 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541492 EE On-Demand Mild F13A1 17 40 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541492 EE On-Demand Mild GPR119 44 54 CC[C@@H](C)c1ccccc1NC(=O)[C@@H](C)N1CCC2(CC1)COCCO2 ZINC000880541494 FG On-Demand Anodyne KCNQ2 41 35 CC[C@@H](C)c1ccccc1NC(=O)[C@H](C)N1CCC2(CC1)COCCO2 ZINC000880541496 FG On-Demand Anodyne KCNQ2 41 35 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(Cl)cc1 ZINC000880541499 ED On-Demand Anodyne CCR1 23 40 Cc1cccc(C(C)C)c1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880541502 EF On-Demand Anodyne SOAT1 46 39 c1ccc(OCCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541511 DF On-Demand Anodyne LTA4H 46 43 c1ccc(OCCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541511 DF On-Demand Anodyne HRH3 48 61 c1ccc(OCCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541511 DF On-Demand Anodyne SIGMAR1 37 44 c1ccc(OCCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541511 DF On-Demand Anodyne EPHX2 19 45 N#Cc1cc(NC(=O)N2CCCN(C(=O)Oc3ccccc3)CC2)ccn1 ZINC000880541518 FF On-Demand Mild PDGFRB 37 43 CCCN(CCC)c1ccc(NC(=O)c2nnn(C)n2)cc1 ZINC000880541523 DE On-Demand Anodyne HRAS 48 32 Brc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541524 FF On-Demand Anodyne LTA4H 49 53 Brc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541524 FF On-Demand Anodyne HRH3 19 44 Brc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541524 FF On-Demand Anodyne PSMB2 41 42 Brc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541524 FF On-Demand Anodyne PSMB1 44 40 O=C(CN1CCC2(CC1)COCCO2)NC(=O)NCc1ccccc1 ZINC000880541547 EC On-Demand Anodyne NPFFR1 41 35 CC(=O)c1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880541553 DE On-Demand Anodyne ABCB1 24 44 CC(=O)c1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880541553 DE On-Demand Anodyne HCN1 69 37 CC(=O)c1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880541553 DE On-Demand Anodyne HCN4 50 33 Cc1cccc(NC(=O)[C@H](C)N2CCC3(CC2)COCCO3)c1 ZINC000880541570 DE On-Demand Anodyne KCNK3 45 35 Cc1cccc(NC(=O)[C@@H](C)N2CCC3(CC2)COCCO3)c1 ZINC000880541571 DE On-Demand Anodyne KCNK3 45 35 Fc1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880541576 CE On-Demand Anodyne LTA4H 19 41 O=C(CCN1CCC2(CC1)COCCO2)NC(=O)NCc1ccccc1 ZINC000880541587 FD On-Demand Anodyne NPFFR1 40 34 O=C(CN1CCC2(CC1)COCCO2)Nc1ccccc1C(F)(F)F ZINC000880541588 FF On-Demand Anodyne RBP4 42 33 c1ccc(-c2ccc(CN3CCC4(CC3)COCCO4)cc2)cc1 ZINC000880541593 DH On-Demand Anodyne SIGMAR1 65 50 COc1ccc([C@@H](NC(=O)CN2CCC3(CC2)COCCO3)C2CC2)cc1 ZINC000880541624 FE On-Demand Anodyne PSMB8 39 42 COc1ccc([C@H](NC(=O)CN2CCC3(CC2)COCCO3)C2CC2)cc1 ZINC000880541625 FE On-Demand Anodyne PSMB8 39 42 CC(C)(C)OC(=O)NCc1ccc(CNC(=O)COC2CC2)c(F)c1 ZINC000880541627 FF On-Demand Anodyne TRPV1 31 41 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(CN2CCOCC2)cc1 ZINC000880541634 GD On-Demand Anodyne EPHX2 20 42 Cc1ncc(CC(=O)NCc2ccc(CNC(=O)OC(C)(C)C)cc2F)o1 ZINC000880541636 GG On-Demand Anodyne TRPV1 24 42 Cc1ncc(CC(=O)NCc2ccc(CNC(=O)OC(C)(C)C)cc2F)o1 ZINC000880541636 GG On-Demand Anodyne P2RX7 31 42 CC[C@@H](C)c1ccc(NC(=O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880541644 EG On-Demand Anodyne SCN2A 15 40 N#Cc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541662 DD On-Demand Mild LTA4H 43 42 N#Cc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541662 DD On-Demand Mild HRH3 19 50 N#Cc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541662 DD On-Demand Mild PSMB2 39 40 N#Cc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541662 DD On-Demand Mild PSMB1 42 38 N#Cc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541662 DD On-Demand Mild MEN1 40 38 CC(C)(C)OC(=O)N1CCC[C@@H]1C1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541667 GH On-Demand Mild GPR119 28 51 CC(C)(C)OC(=O)N1CCC[C@H]1C1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880541668 GH On-Demand Mild GPR119 28 51 CCON(C)C(=O)CNC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880541682 EE On-Demand Anodyne LIPE 18 43 Fc1ccc(CCN2CCC3(CC2)COCCO3)cc1F ZINC000880541691 CE On-Demand Anodyne ABCC1 101 41 Fc1ccc(CCN2CCC3(CC2)COCCO3)cc1F ZINC000880541691 CE On-Demand Anodyne ABCB1A 52 34 N#Cc1c(NC(=O)CN2CCC3(CC2)COCCO3)sc2c1CCCCC2 ZINC000880541716 GF On-Demand Mild VIPR1 30 48 O=C(CN1CCC2(CC1)COCCO2)Nc1ccccc1-c1ccccc1 ZINC000880541722 FG On-Demand Anodyne PRKDC 23 45 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(F)c1 ZINC000880541736 FF On-Demand Mild PDGFRB 45 41 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(F)c1 ZINC000880541736 FF On-Demand Mild NPY2R 83 39 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(C#N)c3)CC2)c(F)c1 ZINC000880541736 FF On-Demand Mild SLC6A9 24 44 CCON(C)C(=O)CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880541751 EE On-Demand Anodyne PDE4D 15 40 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(F)c(F)c1 ZINC000880541771 ED On-Demand Anodyne EPHX2 15 40 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880541786 FF On-Demand Anodyne CCR2 27 40 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(C(F)(F)F)c1 ZINC000880541786 FF On-Demand Anodyne EPHX2 28 46 c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541788 CE On-Demand Anodyne LTA4H 45 44 c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541788 CE On-Demand Anodyne HRH3 67 56 c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541788 CE On-Demand Anodyne SIGMAR1 33 48 c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541788 CE On-Demand Anodyne EPHX2 17 46 c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541788 CE On-Demand Anodyne PSMB1 40 37 O=C(CCN1CCC2(CC1)COCCO2)NCc1ccccc1Cl ZINC000880541794 FE On-Demand Anodyne P2RX7 19 41 O[C@@H]1CCCC[C@H]1N1CCC2(CC1)COCCO2 ZINC000880541808 CD On-Demand Anodyne SLC18A3 37 48 Brc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880541848 FF On-Demand Anodyne LTA4H 31 42 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(Cl)c1 ZINC000880541865 EF On-Demand Anodyne EPHX2 25 42 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(Cl)c1 ZINC000880541865 EF On-Demand Anodyne MCHR1 19 42 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880541902 GF On-Demand Anodyne HCN1 52 38 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880541902 GF On-Demand Anodyne HCN4 43 35 CCOc1ccccc1[C@H](CC)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880541903 GF On-Demand Anodyne HCN1 52 38 CCOc1ccccc1[C@H](CC)NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880541903 GF On-Demand Anodyne HCN4 43 35 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OC(F)(F)F)cc1 ZINC000880541905 FE On-Demand Anodyne P2RY1 64 41 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OC(F)(F)F)cc1 ZINC000880541905 FE On-Demand Anodyne EPHX2 66 48 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OC(F)(F)F)cc1 ZINC000880541905 FE On-Demand Anodyne TRPM8 21 43 O=C(CN1CCC2(CC1)COCCO2)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880541922 GD On-Demand Anodyne EPHX2 71 44 O=C(Nc1cccc(C#Cc2ccccn2)c1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880541941 II On-Demand Mild TYK2 41 33 O=C(Nc1cccc(C#Cc2ccccn2)c1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880541942 II On-Demand Mild TYK2 41 33 Ic1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880541949 FF On-Demand Anodyne SIGMAR1 30 50 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880541959 GG On-Demand Anodyne RAF1 24 41 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880541959 GG On-Demand Anodyne EPHX2 25 42 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880541959 GG On-Demand Anodyne IMDH_CRYPV 17 40 CCON(C)C(=O)CNC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880541967 DD On-Demand Anodyne RAF1 19 41 c1ccc(CCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541994 CF On-Demand Anodyne SLC6A3 19 40 c1ccc(CCCN2CCC3(CC2)COCCO3)cc1 ZINC000880541994 CF On-Demand Anodyne SIGMAR1 67 58 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880542025 FF On-Demand Anodyne EPHX2 22 48 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880542027 FH On-Demand Anodyne SOAT1 61 42 c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880542063 CE On-Demand Anodyne SIGMAR1 62 52 COc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542080 DD On-Demand Anodyne LTA4H 53 51 COc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542080 DD On-Demand Anodyne HRH3 32 44 COc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542080 DD On-Demand Anodyne PSMB2 42 42 COc1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542080 DD On-Demand Anodyne PSMB1 45 40 CCCOc1cccc(CNC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880542105 FD On-Demand Anodyne HRH2 27 40 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc2c(c1)OCO2 ZINC000880542123 EC On-Demand Anodyne NOS2 100 39 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc2c(c1)OCO2 ZINC000880542123 EC On-Demand Anodyne MCHR1 18 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(C#N)c1 ZINC000880542126 FE On-Demand Mild JAK2 15 43 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(C#N)c1 ZINC000880542126 FE On-Demand Mild CSF1R 18 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(C#N)c1 ZINC000880542126 FE On-Demand Mild EPHB4 82 37 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(C#N)c1 ZINC000880542126 FE On-Demand Mild STAT6 46 32 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(F)cc1C(F)(F)F ZINC000880542142 GE On-Demand Anodyne P2RX7 24 45 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCCCC2)cc1 ZINC000880542154 FE On-Demand Anodyne STAT6 50 31 N#Cc1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880542160 DD On-Demand Mild CCR3 15 40 N#Cc1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880542160 DD On-Demand Mild MCHR1 44 44 N#Cc1cccc(OCCCN2CCC3(CC2)COCCO3)c1 ZINC000880542165 DE On-Demand Mild HRH3 45 43 N#Cc1cccc(OCCCN2CCC3(CC2)COCCO3)c1 ZINC000880542165 DE On-Demand Mild EPHX2 16 40 N#Cc1cccc(OCCCN2CCC3(CC2)COCCO3)c1 ZINC000880542165 DE On-Demand Mild MEN1 40 37 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880542176 EE On-Demand Anodyne ERBB4 51 39 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(F)c(Cl)c1 ZINC000880542176 EE On-Demand Anodyne MCHR1 31 43 O=C(Nc1ccc(F)cc1)[C@H](c1ccccc1)N1CCC2(CC1)COCCO2 ZINC000880542198 GG On-Demand Anodyne NPY2R 54 36 O=C(Nc1ccc(F)cc1)[C@@H](c1ccccc1)N1CCC2(CC1)COCCO2 ZINC000880542199 GG On-Demand Anodyne NPY2R 54 36 O=C(CN1CCC2(CC1)COCCO2)N[C@@H]1CCCc2ccccc21 ZINC000880542203 EE On-Demand Anodyne BDKRB1 50 39 O=C(CN1CCC2(CC1)COCCO2)N[C@H]1CCCc2ccccc21 ZINC000880542205 EE On-Demand Anodyne BDKRB1 50 39 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccccc1 ZINC000880542214 DD On-Demand Anodyne EPHX2 24 41 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Cl)c1 ZINC000880542224 DE On-Demand Anodyne EPHX2 18 42 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(Cl)c1 ZINC000880542224 DE On-Demand Anodyne MCHR1 24 42 O=C(CN1CCC2(CC1)COCCO2)Nc1cc(C(F)(F)F)ccc1Cl ZINC000880542236 GG On-Demand Anodyne TRPM8 15 40 CCOc1ccccc1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880542240 ED On-Demand Anodyne CCR1 36 41 CCOc1ccccc1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880542240 ED On-Demand Anodyne HCN1 55 39 CCOc1ccccc1NC(=O)CN1CCC2(CC1)COCCO2 ZINC000880542240 ED On-Demand Anodyne HCN4 46 37 CCOc1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880542277 DE On-Demand Anodyne HCN1 49 35 CCOc1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880542277 DE On-Demand Anodyne HCN4 40 33 CCON(C)C(=O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880542305 DD On-Demand Anodyne NQO2 38 43 CCON(C)C(=O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880542305 DD On-Demand Anodyne MTNR1A 73 44 CCON(C)C(=O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880542305 DD On-Demand Anodyne MTNR1B 67 39 CCON(C)C(=O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880542306 DD On-Demand Anodyne NQO2 38 43 CCON(C)C(=O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880542306 DD On-Demand Anodyne MTNR1A 73 44 CCON(C)C(=O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880542306 DD On-Demand Anodyne MTNR1B 67 39 c1ccc2oc(CN3CCC4(CC3)COCCO4)cc2c1 ZINC000880542308 CF On-Demand Anodyne SIGMAR1 21 45 O=C(CN1CCC2(CC1)COCCO2)NCCOc1cccc(Cl)c1 ZINC000880542315 FD On-Demand Anodyne HRH2 26 40 O=C(CN1CCC2(CC1)COCCO2)NCCOc1cccc(Cl)c1 ZINC000880542315 FD On-Demand Anodyne AVPR1B 38 40 CCON(C)C(=O)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880542321 DD On-Demand Anodyne MPO 52 38 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc2c(c1)OCO2 ZINC000880542336 ED On-Demand Anodyne DYRK2 40 35 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)cc1 ZINC000880542339 DE On-Demand Anodyne EPHX2 22 42 CCON(C)C(=O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880542340 GD On-Demand Anodyne LGMN 40 36 CCON(C)C(=O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880542340 GD On-Demand Anodyne Q9NAW4_PLAFA 39 46 CS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542359 FD On-Demand Anodyne ESR1 15 41 CS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542359 FD On-Demand Anodyne LTA4H 42 39 CS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542359 FD On-Demand Anodyne HRH3 19 45 CS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542359 FD On-Demand Anodyne MMP13 23 42 CS(=O)(=O)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542359 FD On-Demand Anodyne PSMB1 41 36 O[C@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542372 ED On-Demand Anodyne ADRB1 18 47 O[C@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542372 ED On-Demand Anodyne HTR1A 18 56 O[C@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542372 ED On-Demand Anodyne SLC6A4 19 45 O[C@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542372 ED On-Demand Anodyne CCR1 46 41 O[C@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542372 ED On-Demand Anodyne ABCB1 56 42 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542373 ED On-Demand Anodyne ADRB1 18 47 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542373 ED On-Demand Anodyne HTR1A 18 56 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542373 ED On-Demand Anodyne SLC6A4 19 45 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542373 ED On-Demand Anodyne CCR1 46 41 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC2(CC1)COCCO2 ZINC000880542373 ED On-Demand Anodyne ABCB1 56 42 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OCc2ccccc2)cc1 ZINC000880542381 GG On-Demand Anodyne TSHR 42 33 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OCc2ccccc2)cc1 ZINC000880542381 GG On-Demand Anodyne LTA4H 43 51 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OCc2ccccc2)cc1 ZINC000880542381 GG On-Demand Anodyne ADAM17 25 42 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(OCc2ccccc2)cc1 ZINC000880542381 GG On-Demand Anodyne EPHX2 21 48 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880542387 GD On-Demand Anodyne MTOR 64 37 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880542387 GD On-Demand Anodyne EPHX2 19 43 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880542387 GD On-Demand Anodyne STAT6 61 35 c1ccc(CCc2nc(CN3CCC4(CC3)COCCO4)cs2)cc1 ZINC000880542395 FG On-Demand Anodyne SIGMAR1 25 40 c1ccc2cc(CCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880542418 DG On-Demand Anodyne SIGMAR1 28 44 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc(F)cc1 ZINC000880542423 DE On-Demand Anodyne EPHX2 25 43 O=C(CN1CCC2(CC1)COCCO2)NCc1cccnc1 ZINC000880542424 DC On-Demand Anodyne SCD 18 42 O=C(CN1CCC2(CC1)COCCO2)NCc1cccnc1 ZINC000880542424 DC On-Demand Anodyne NAMPT 63 45 O=C(NCc1ccco1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542457 FF On-Demand Anodyne CHRM3 21 44 O=C(c1cccc(CN2CCC3(CC2)COCCO3)c1)N1CCCCC1 ZINC000880542474 FF On-Demand Anodyne CHRM3 15 48 O=C(c1cccc(CN2CCC3(CC2)COCCO3)c1)N1CCCCC1 ZINC000880542474 FF On-Demand Anodyne CCR8 29 42 CC(C)(C)OC(=O)[C@](C)(CNC(=O)[C@H]1CCc2nncn2CC1)c1ccccc1 ZINC000880542476 GF On-Demand Anodyne CACNA1G 35 41 CC(C)(C)OC(=O)[C@](C)(CNC(=O)[C@@H]1CCc2nncn2CC1)c1ccccc1 ZINC000880542477 GF On-Demand Anodyne CACNA1G 35 41 O=C(CN1CCC2(CC1)COCCO2)NCC1(c2ccccc2)CC1 ZINC000880542503 ED On-Demand Anodyne NPFFR1 38 46 FC(F)(F)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542504 EF On-Demand Anodyne LTA4H 44 56 FC(F)(F)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542504 EF On-Demand Anodyne HRH3 17 41 FC(F)(F)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542504 EF On-Demand Anodyne PSMB2 38 40 FC(F)(F)c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542504 EF On-Demand Anodyne PSMB1 42 43 c1ccc(CCOCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542509 DF On-Demand Anodyne SIGMAR1 46 45 C[C@H](NC(=O)Nc1ccnc(C#N)c1)c1ccc(N2CCOCC2)cc1 ZINC000880542513 FF On-Demand Mild JAK2 15 40 C[C@H](NC(=O)Nc1ccnc(C#N)c1)c1ccc(N2CCOCC2)cc1 ZINC000880542513 FF On-Demand Mild EPHB4 54 34 COc1cccc(OC)c1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880542526 FD On-Demand Anodyne CCR1 49 44 COc1cccc(OC)c1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880542526 FD On-Demand Anodyne ABCB1 71 45 COc1cccc(OC)c1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880542527 FD On-Demand Anodyne CCR1 49 44 COc1cccc(OC)c1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880542527 FD On-Demand Anodyne ABCB1 71 45 c1ccc(Cn2ccnc2CN2CCC3(CC2)COCCO3)cc1 ZINC000880542529 EE On-Demand Anodyne SIGMAR1 30 40 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542562 GE On-Demand Anodyne ACOX1 57 36 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542562 GE On-Demand Anodyne CCR1 44 40 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542562 GE On-Demand Anodyne ABCB1 45 40 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542562 GE On-Demand Anodyne PDS 41 35 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542563 GE On-Demand Anodyne ACOX1 57 36 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542563 GE On-Demand Anodyne CCR1 44 40 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542563 GE On-Demand Anodyne ABCB1 45 40 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCC2(CC1)COCCO2 ZINC000880542563 GE On-Demand Anodyne PDS 41 35 Cc1ccc(N2CCCN(C(=O)Nc3ccnc(C#N)c3)CC2)cc1 ZINC000880542570 EG On-Demand Mild PDGFRB 43 40 CC(C)(C)N1CCC(NC(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880542588 DE On-Demand Mild EPHX2 49 42 N#Cc1cc(NC(=O)NCCc2ccc(N3CCCCC3)cc2)ccn1 ZINC000880542592 EG On-Demand Mild CTSK 25 42 N#Cc1cc(NC(=O)NCCc2ccc(N3CCCCC3)cc2)ccn1 ZINC000880542592 EG On-Demand Mild CTSL 23 42 O=C(CN1CCC2(CC1)COCCO2)OCc1ccccc1 ZINC000880542606 DD On-Demand Anodyne SLC12A5 76 39 c1ccc2c(CCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542609 EH On-Demand Anodyne SIGMAR1 31 49 c1ccc2c(CCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542609 EH On-Demand Anodyne EBP 46 47 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542616 JI On-Demand Mild GRM4 33 42 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542616 JI On-Demand Mild TYK2 25 40 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542616 JI On-Demand Mild KCNK3 51 40 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542616 JI On-Demand Mild KCNK9 43 40 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542617 JI On-Demand Mild GRM4 33 42 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542617 JI On-Demand Mild TYK2 25 40 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542617 JI On-Demand Mild KCNK3 51 40 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542617 JI On-Demand Mild KCNK9 43 40 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542618 JI On-Demand Mild GRM4 33 42 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542618 JI On-Demand Mild TYK2 25 40 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542618 JI On-Demand Mild KCNK3 51 40 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542618 JI On-Demand Mild KCNK9 43 40 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542619 JI On-Demand Mild GRM4 33 42 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542619 JI On-Demand Mild TYK2 25 40 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542619 JI On-Demand Mild KCNK3 51 40 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880542619 JI On-Demand Mild KCNK9 43 40 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne HTR1D 16 43 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne CHRM3 19 47 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne FAAH 18 40 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne MCHR1 25 44 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne MCHR2 53 37 CC(=O)Nc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542623 DE On-Demand Anodyne NPFFR1 43 36 c1cncc(Oc2ccccc2CN2CCC3(CC2)COCCO3)c1 ZINC000880542629 EG On-Demand Anodyne CCR8 23 47 FC(F)(F)COc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880542644 EG On-Demand Anodyne SIGMAR1 24 40 CC(=O)Nc1ccc(S(=O)(=O)CCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542649 GD On-Demand Anodyne EPHX2 18 58 c1ccc(OCCOCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542655 DD On-Demand Anodyne LTA4H 46 44 c1ccc(OCCOCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542655 DD On-Demand Anodyne HRH3 28 49 c1ccc(OCCOCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542655 DD On-Demand Anodyne PSMB1 40 37 c1cc(CN2CCC3(CC2)COCCO3)ccn1 ZINC000880542670 BD On-Demand Anodyne SIGMAR1 23 40 c1ccc2c(OCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542671 EG On-Demand Anodyne HTR1B 16 40 c1ccc2c(OCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542671 EG On-Demand Anodyne ALB 22 41 c1ccc2c(OCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542671 EG On-Demand Anodyne MCL1 34 41 C[C@@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1CCC2(CC1)COCCO2 ZINC000880542672 GE On-Demand Mild MLYCD 18 42 C[C@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1CCC2(CC1)COCCO2 ZINC000880542673 GE On-Demand Mild MLYCD 18 42 COc1cccc(S(=O)(=O)CCN2CCC3(CC2)COCCO3)c1 ZINC000880542675 FD On-Demand Anodyne DRD4 40 30 O=[N+]([O-])c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880542687 DE On-Demand Bother SIGMAR1 15 52 O=[N+]([O-])c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880542687 DE On-Demand Bother KCNJ1 52 62 O=C(CCN1CCC2(CC1)COCCO2)N1CCN(c2ccccn2)CC1 ZINC000880542702 FD On-Demand Anodyne DRD4 30 47 N#Cc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542711 DE On-Demand Mild HRH3 58 49 N#Cc1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542711 DE On-Demand Mild MEN1 47 44 c1ccc2cc(OCCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880542728 EG On-Demand Anodyne DRD2 16 42 c1ccc2cc(OCCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880542728 EG On-Demand Anodyne HRH3 64 46 c1ccc2cc(OCCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880542728 EG On-Demand Anodyne SIGMAR1 27 43 c1ccc2cc(OCCCN3CCC4(CC3)COCCO4)ccc2c1 ZINC000880542728 EG On-Demand Anodyne EPHX2 16 40 N#Cc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ccn1 ZINC000880542774 EF On-Demand Mild NAMPT 56 54 FC(F)Oc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542837 DF On-Demand Anodyne SIGMAR1 17 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ncccc1SC ZINC000880542843 FF On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ncccc1SC ZINC000880542843 FF On-Demand Anodyne FPR1 43 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ncccc1SC ZINC000880542844 FF On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ncccc1SC ZINC000880542844 FF On-Demand Anodyne FPR1 43 39 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ncccc1SC)C2 ZINC000880542845 EH On-Demand Anodyne FAAH 15 41 c1cc2c(cc1OCCCN1CCC3(CC1)COCCO3)OCO2 ZINC000880542852 EE On-Demand Anodyne HRH3 45 53 c1ccc2c(CN3CCC4(CC3)COCCO4)csc2c1 ZINC000880542862 DG On-Demand Anodyne FFAR2 44 35 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc2c(c1)OCO2 ZINC000880542911 ED On-Demand Anodyne DYRK2 47 36 CN(C)C(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542919 DD On-Demand Anodyne CHRM3 20 42 CN(C)C(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542919 DD On-Demand Anodyne MCHR2 46 34 C[C@H](c1nc(-c2cccs2)no1)N1CCC2(CC1)COCCO2 ZINC000880542921 EF On-Demand Anodyne ETHR 24 40 N#Cc1cc(NC(=O)NCCSC(F)(F)F)ccn1 ZINC000880542944 CE On-Demand Mild ADRB1 41 31 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880542948 GD On-Demand Anodyne MCHR2 41 34 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(CN2CCCC2)cc1 ZINC000880542948 GD On-Demand Anodyne NPFFR1 40 37 c1cncc(CN2CCC3(CC2)COCCO3)c1 ZINC000880542954 BD On-Demand Anodyne SIGMAR1 23 40 O=[N+]([O-])c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542968 EE On-Demand Bother LTA4H 17 51 O=[N+]([O-])c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542968 EE On-Demand Bother HRH3 51 47 O=[N+]([O-])c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880542968 EE On-Demand Bother KCNJ1 22 41 O=C(CCN1CCC2(CC1)COCCO2)N1CCN(c2ccc(F)cc2)CC1 ZINC000880542982 GD On-Demand Anodyne DRD4 15 41 O=C(CCN1CCC2(CC1)COCCO2)N1CCN(c2ccc(F)cc2)CC1 ZINC000880542982 GD On-Demand Anodyne SSTR1 24 41 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild JAK2 15 43 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild MTOR 47 38 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild EPHX2 21 40 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild CSF1R 17 40 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild EPHB4 62 33 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild STAT6 56 37 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccn1 ZINC000880542984 EE On-Demand Mild NAMPT 53 43 c1ccc2c(OCCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542987 EG On-Demand Anodyne ALB 22 41 c1ccc2c(OCCCN3CCC4(CC3)COCCO4)cccc2c1 ZINC000880542987 EG On-Demand Anodyne MCL1 38 41 CC(C)(C)OC(=O)[C@](C)(CNC(=O)COC1CC1)c1ccccc1 ZINC000880542991 EF On-Demand Anodyne AMY2 55 31 O=C(CN1CCC2(CC1)COCCO2)NCC1(c2ccccc2)CCOCC1 ZINC000880542995 GD On-Demand Anodyne NPFFR1 32 44 c1cc2c(cc1CN1CCC3(CC1)COCCO3)CCC2 ZINC000880542999 CF On-Demand Anodyne SIGMAR1 22 40 CS(=O)(=O)c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880543013 FD On-Demand Anodyne HRH3 63 47 CS(=O)(=O)c1ccc(OCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880543013 FD On-Demand Anodyne MMP13 24 44 CCN1CC[C@H](CNC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880543022 CD On-Demand Mild CCR3 58 41 CCN1CC[C@H](CNC(=O)Nc2ccnc(C#N)c2)C1 ZINC000880543022 CD On-Demand Mild CACNA1I 52 34 FC(F)(F)c1ccccc1OCCN1CCC2(CC1)COCCO2 ZINC000880543040 EF On-Demand Anodyne LTA4H 15 50 CC(=O)NCCCN1CCC2(CC1)COCCO2 ZINC000880543041 CC On-Demand Anodyne PAOX 17 41 O=S(=O)(NCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880543047 EC On-Demand Anodyne HTR7 25 53 O=S(=O)(NCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880543047 EC On-Demand Anodyne SIGMAR1 18 44 O=S(=O)(NCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880543047 EC On-Demand Anodyne CCR1 19 51 O=[N+]([O-])c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880543067 DD On-Demand Bother LTA4H 42 58 O=[N+]([O-])c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880543067 DD On-Demand Bother PSMB1 40 36 O=[N+]([O-])c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880543067 DD On-Demand Bother KCNJ1 22 42 CCN1CC[C@@H](NC(=O)Nc2cncc(OC)c2)C1=O ZINC000880543073 CC On-Demand Anodyne EPHX2 17 42 CCN1CC[C@H](NC(=O)Nc2cncc(OC)c2)C1=O ZINC000880543074 CC On-Demand Anodyne EPHX2 17 42 COc1cncc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)c1 ZINC000880543102 EF On-Demand Anodyne EPHX2 33 55 COc1cncc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)c1 ZINC000880543103 EF On-Demand Anodyne EPHX2 33 55 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2ccsc2)c1 ZINC000880543118 CF On-Demand Anodyne NPBWR1 86 35 COc1cncc(NC(=O)N2CCc3c(O)cccc3C2)c1 ZINC000880543128 CE On-Demand Anodyne DRD4 40 30 COc1cncc(NC(=O)N2CCc3c(O)cccc3C2)c1 ZINC000880543128 CE On-Demand Anodyne P2RY14 48 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543144 GD On-Demand Anodyne CELA1 19 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543144 GD On-Demand Anodyne PREP 62 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543144 GD On-Demand Anodyne SLC12A5 65 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543144 GD On-Demand Anodyne Q9NAW4_PLAFA 26 42 COc1cncc(NC(=O)N2CCN(CCC#N)CC2)c1 ZINC000880543145 CD On-Demand Mild DRD4 41 31 COc1cncc(NC(=O)N2CCN(CCC#N)CC2)c1 ZINC000880543145 CD On-Demand Mild PDGFRB 43 39 COc1cncc(NC(=O)N2CC[C@@H](O)[C@H]2c2ccc(Br)cc2)c1 ZINC000880543177 GG On-Demand Anodyne CHRNA7 15 45 O=C(c1cnc2cc[nH]c2c1)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543178 CC On-Demand Anodyne L3MBTL3 45 39 COc1cncc(NC(=O)N2CCC(c3nccc(-c4cccnc4)n3)CC2)c1 ZINC000880543179 GG On-Demand Anodyne ABL1 15 50 COc1cncc(NC(=O)N2CCC(c3nccc(-c4cccnc4)n3)CC2)c1 ZINC000880543179 GG On-Demand Anodyne CHRNA7 23 42 COc1cncc(NC(=O)N2CCC(c3nccc(-c4cccnc4)n3)CC2)c1 ZINC000880543179 GG On-Demand Anodyne CALCRL 15 40 COc1cncc(NC(=O)N2CCC(c3nccc(-c4cccnc4)n3)CC2)c1 ZINC000880543179 GG On-Demand Anodyne P2RY14 25 40 COc1cncc(NC(=O)N[C@H](C)c2ccccc2OC)c1 ZINC000880543183 DF On-Demand Anodyne KCNK3 39 43 COc1cncc(NC(=O)N[C@H](C)c2ccccc2OC)c1 ZINC000880543183 DF On-Demand Anodyne KCNK9 35 43 COc1cncc(NC(=O)N[C@@H](C)c2ccccc2OC)c1 ZINC000880543184 DF On-Demand Anodyne KCNK3 39 43 COc1cncc(NC(=O)N[C@@H](C)c2ccccc2OC)c1 ZINC000880543184 DF On-Demand Anodyne KCNK9 35 43 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne DRD4 43 35 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne MAPK14 32 40 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne SSTR5 45 43 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne CTSL 19 41 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne EPHX2 24 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne MCHR1 17 44 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne HPGDS 34 40 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne KCNK3 62 44 COc1cncc(NC(=O)N2CCC(NC(=O)c3cccc(C)c3)CC2)c1 ZINC000880543205 FF On-Demand Anodyne KCNK9 45 39 COc1cncc(NC(=O)NCc2ccnc(N3CCSCC3)c2)c1 ZINC000880543208 FE On-Demand Anodyne ROCK2 22 45 COc1ccc(CN(C)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880543219 DF On-Demand Anodyne ROCK1 15 48 COc1ccc(CN(C)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880543219 DF On-Demand Anodyne ROCK2 24 48 COc1ccc(CN(C)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880543219 DF On-Demand Anodyne NPY5R 24 42 COc1cncc(NC(=O)N(C)C[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543222 FE On-Demand Anodyne NPFFR2 30 43 COc1cncc(NC(=O)N(C)C[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543222 FE On-Demand Anodyne FAAH 17 43 COc1cncc(NC(=O)N(C)C[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543222 FE On-Demand Anodyne NPFFR1 43 43 COc1cncc(NC(=O)N(C)C[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543223 FE On-Demand Anodyne NPFFR2 30 43 COc1cncc(NC(=O)N(C)C[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543223 FE On-Demand Anodyne FAAH 17 43 COc1cncc(NC(=O)N(C)C[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880543223 FE On-Demand Anodyne NPFFR1 43 43 COc1cncc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880543231 EE On-Demand Anodyne SIGMAR1 20 41 COc1cncc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880543231 EE On-Demand Anodyne NPFFR2 17 40 COc1cncc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880543231 EE On-Demand Anodyne FAAH 31 57 COc1cncc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880543231 EE On-Demand Anodyne NPFFR1 22 40 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3)CC2)c1 ZINC000880543232 EF On-Demand Anodyne CACNA1H 51 38 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3)CC2)c1 ZINC000880543232 EF On-Demand Anodyne HTR1B 15 52 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3)CC2)c1 ZINC000880543232 EF On-Demand Anodyne PDGFRB 52 43 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3)CC2)c1 ZINC000880543232 EF On-Demand Anodyne SSTR1 20 45 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3)CC2)c1 ZINC000880543232 EF On-Demand Anodyne FAAH 20 45 COc1cncc(NC(=O)N2CCc3c(CC(N)=O)cccc3C2)c1 ZINC000880543253 ED On-Demand Anodyne P2RY14 49 35 COc1cncc(NC(=O)NCC[C@@H](O)COCc2ccccc2)c1 ZINC000880543262 EE On-Demand Anodyne ADRB1 43 35 COc1cncc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)c1 ZINC000880543276 DG On-Demand Anodyne RBP4 40 34 O=C(c1cc2ccccc2cc1F)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880543286 DD On-Demand Anodyne L3MBTL3 41 37 COc1cncc(NC(=O)N(C)Cc2ccns2)c1 ZINC000880543289 CE On-Demand Anodyne ROCK2 15 42 COc1cncc(NC(=O)NCCCn2cncn2)c1 ZINC000880543290 CC On-Demand Anodyne QPCT 31 44 COc1cncc(NC(=O)NC2CC3(CSC3)C2)c1 ZINC000880543300 CE On-Demand Anodyne EPHX2 16 40 COc1cncc(NC(=O)N(C)[C@@H](CCc2ccccc2)C(F)F)c1 ZINC000880543303 EH On-Demand Anodyne MMP3 24 41 COc1cncc(NC(=O)N(C)[C@@H](CCc2ccccc2)C(F)F)c1 ZINC000880543303 EH On-Demand Anodyne NPY5R 34 42 COc1cncc(NC(=O)N(C)[C@H](CCc2ccccc2)C(F)F)c1 ZINC000880543304 EH On-Demand Anodyne MMP3 24 41 COc1cncc(NC(=O)N(C)[C@H](CCc2ccccc2)C(F)F)c1 ZINC000880543304 EH On-Demand Anodyne NPY5R 34 42 CC(C)(C(=O)N1CC(N2CC[C@@H](O)C2)C1)c1ccc(C(F)(F)F)cc1 ZINC000880543305 FE On-Demand Anodyne MCHR1 17 41 COc1cncc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)c1 ZINC000880543306 EG On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)c1 ZINC000880543306 EG On-Demand Anodyne CPT1A 71 36 COc1cncc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)c1 ZINC000880543307 EG On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)c1 ZINC000880543307 EG On-Demand Anodyne CPT1A 71 36 COc1cncc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)c1 ZINC000880543308 EG On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)c1 ZINC000880543308 EG On-Demand Anodyne CPT1A 71 36 COc1cncc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)c1 ZINC000880543309 EG On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)c1 ZINC000880543309 EG On-Demand Anodyne CPT1A 71 36 COc1cncc(NC(=O)NCCC2(O)CCN(c3ccccc3)CC2)c1 ZINC000880543310 FF On-Demand Anodyne SOAT1 18 46 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne PDGFRB 26 41 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne GRIN2B 34 43 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne SIGMAR1 18 44 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne CTSB 15 49 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne CTSK 23 49 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne CTSL 27 49 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne CCR3 30 42 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne C3AR1 39 41 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne FAAH 37 42 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne EPHX2 39 42 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne TGM2 40 47 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne MCHR1 17 43 COc1cncc(NC(=O)N2CCC(NC(=O)OCc3ccccc3)CC2)c1 ZINC000880543320 GG On-Demand Anodyne F13A1 33 47 COc1cncc(NC(=O)NCc2cccc3c2CCOC3)c1 ZINC000880543331 DE On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880543340 CC On-Demand Anodyne DRD4 43 34 COc1cncc(NC(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880543340 CC On-Demand Anodyne CCR3 53 45 COc1cncc(NC(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880543340 CC On-Demand Anodyne MCHR1 15 40 COc1cncc(NC(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880543341 CC On-Demand Anodyne DRD4 43 34 COc1cncc(NC(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880543341 CC On-Demand Anodyne CCR3 53 45 COc1cncc(NC(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880543341 CC On-Demand Anodyne MCHR1 15 40 COc1cncc(NC(=O)N[C@@H](C)CC2CCC2)c1 ZINC000880543355 CF On-Demand Anodyne CCR3 53 34 COc1cncc(NC(=O)N[C@H](C)CC2CCC2)c1 ZINC000880543356 CF On-Demand Anodyne CCR3 53 34 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880543360 FD On-Demand Anodyne DRD4 20 42 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880543360 FD On-Demand Anodyne CCR3 27 47 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880543361 FD On-Demand Anodyne DRD4 20 42 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880543361 FD On-Demand Anodyne CCR3 27 47 COc1cncc(NC(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543363 FG On-Demand Anodyne ACACA 45 41 COc1cncc(NC(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543363 FG On-Demand Anodyne NPY5R 18 40 COc1cncc(NC(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543363 FG On-Demand Anodyne EPHX2 32 42 COc1cncc(NC(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543363 FG On-Demand Anodyne TRPM8 17 40 COc1cncc(NC(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543364 FG On-Demand Anodyne ACACA 45 41 COc1cncc(NC(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543364 FG On-Demand Anodyne NPY5R 18 40 COc1cncc(NC(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543364 FG On-Demand Anodyne EPHX2 32 42 COc1cncc(NC(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880543364 FG On-Demand Anodyne TRPM8 17 40 COc1cncc(NC(=O)N2CCC(F)(F)CC2)c1 ZINC000880543381 CE On-Demand Anodyne S1PR2 28 41 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2ccc(F)cc2)c1 ZINC000880543389 DF On-Demand Anodyne EPHX2 18 42 COc1cncc(NC(=O)N[C@](C)(CO)Cc2ccc(Cl)cc2)c1 ZINC000880543394 EF On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N[C@@](C)(CO)Cc2ccc(Cl)cc2)c1 ZINC000880543395 EF On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N2CC[C@@H](c3ccc(OC)c(F)c3)C2)c1 ZINC000880543411 EG On-Demand Anodyne GRIN2B 15 40 COc1cncc(NC(=O)N2CC[C@H](c3ccc(OC)c(F)c3)C2)c1 ZINC000880543412 EG On-Demand Anodyne GRIN2B 15 40 COc1cncc(NC(=O)NCCC2CCN(C(C)C)CC2)c1 ZINC000880543414 DF On-Demand Anodyne CCR3 43 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543415 GG On-Demand Anodyne GHRHR 54 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543415 GG On-Demand Anodyne P2RY12 60 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543415 GG On-Demand Anodyne FPR1 42 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543416 GG On-Demand Anodyne GHRHR 54 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543416 GG On-Demand Anodyne P2RY12 60 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543416 GG On-Demand Anodyne FPR1 42 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543417 GG On-Demand Anodyne GHRHR 54 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543417 GG On-Demand Anodyne P2RY12 60 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@H](C)C1 ZINC000880543417 GG On-Demand Anodyne FPR1 42 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543418 GG On-Demand Anodyne GHRHR 54 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543418 GG On-Demand Anodyne P2RY12 60 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2ccccc2[C@@H](C)C1 ZINC000880543418 GG On-Demand Anodyne FPR1 42 33 COc1cncc(NC(=O)N2CC3(CCCO3)C2)c1 ZINC000880543430 CD On-Demand Anodyne EPHX2 17 40 COc1cncc(NC(=O)N2CCN(CCc3cnccn3)CC2)c1 ZINC000880543456 ED On-Demand Anodyne DRD4 41 32 COc1cncc(NC(=O)N2CCN(CCc3cnccn3)CC2)c1 ZINC000880543456 ED On-Demand Anodyne PDGFRB 51 36 COc1cncc(NC(=O)N2CCN(CCc3cnccn3)CC2)c1 ZINC000880543456 ED On-Demand Anodyne FAAH 15 41 COc1cncc(NC(=O)N2CCN(c3cccc4[nH]ccc34)CC2)c1 ZINC000880543477 FF On-Demand Anodyne HTR1A 20 45 COc1cncc(NC(=O)N2CCN(c3cccc4[nH]ccc34)CC2)c1 ZINC000880543477 FF On-Demand Anodyne HTR1B 33 45 COc1cncc(NC(=O)N2CCN(c3cccc4[nH]ccc34)CC2)c1 ZINC000880543477 FF On-Demand Anodyne PDGFRB 51 48 COc1cncc(NC(=O)N2CCN(c3cccc4[nH]ccc34)CC2)c1 ZINC000880543477 FF On-Demand Anodyne HPGDS 27 44 COc1cncc(NC(=O)N2CC[C@H](Oc3cccc(F)c3)C2)c1 ZINC000880543480 EF On-Demand Anodyne CCR3 34 48 COc1cncc(NC(=O)N2CC[C@H](Oc3cccc(F)c3)C2)c1 ZINC000880543480 EF On-Demand Anodyne MLNR 20 42 COc1cncc(NC(=O)N2CC[C@H](Oc3cccc(F)c3)C2)c1 ZINC000880543480 EF On-Demand Anodyne EPHX2 27 43 COc1cncc(NC(=O)N2CC[C@H](Oc3cccc(F)c3)C2)c1 ZINC000880543480 EF On-Demand Anodyne SCD1 27 44 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccc(F)c3)C2)c1 ZINC000880543481 EF On-Demand Anodyne CCR3 34 48 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccc(F)c3)C2)c1 ZINC000880543481 EF On-Demand Anodyne MLNR 20 42 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccc(F)c3)C2)c1 ZINC000880543481 EF On-Demand Anodyne EPHX2 27 43 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccc(F)c3)C2)c1 ZINC000880543481 EF On-Demand Anodyne SCD1 27 44 COc1cncc(NC(=O)N[C@H](c2ccccn2)C2CCC2)c1 ZINC000880543490 DG On-Demand Anodyne TTK 19 41 COc1cncc(NC(=O)N[C@@H](c2ccccn2)C2CCC2)c1 ZINC000880543491 DG On-Demand Anodyne TTK 19 41 COc1cncc(NC(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)c1 ZINC000880543503 FF On-Demand Anodyne P2RY1 15 42 COc1cncc(NC(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)c1 ZINC000880543504 FF On-Demand Anodyne P2RY1 15 42 COc1cncc(NC(=O)NCc2c(Br)cnn2C)c1 ZINC000880543505 ED On-Demand Anodyne HTR2A 25 44 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880543508 EF On-Demand Anodyne HTR1B 15 48 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880543508 EF On-Demand Anodyne PDGFRB 52 42 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880543508 EF On-Demand Anodyne NPY2R 83 39 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880543518 EE On-Demand Anodyne EPHX2 45 39 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880543518 EE On-Demand Anodyne GPR119 38 40 COc1ccc(CN(C(=O)Nc2cncc(OC)c2)[C@@H](C)CCCO)cc1 ZINC000880543532 FG On-Demand Anodyne NPY5R 23 41 COc1ccc(CN(C(=O)Nc2cncc(OC)c2)[C@H](C)CCCO)cc1 ZINC000880543533 FG On-Demand Anodyne NPY5R 23 41 COc1cncc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880543539 EG On-Demand Anodyne CACNA1H 49 35 COc1cncc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880543539 EG On-Demand Anodyne CCR3 39 46 COc1cncc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880543539 EG On-Demand Anodyne MLNR 20 45 COc1cncc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880543539 EG On-Demand Anodyne EPHX2 30 48 COc1cncc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880543539 EG On-Demand Anodyne SCD1 35 49 COc1cncc(NC(=O)N2CCc3cccc(NC(C)=O)c3C2)c1 ZINC000880543540 EF On-Demand Anodyne P2RY14 49 35 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild DRD2 24 46 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild ADRA1D 26 46 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild ADRA1A 19 46 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild ADRA1B 18 46 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild NPY1R 22 44 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild EPHX2 43 39 COc1cncc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c1 ZINC000880543543 FF On-Demand Mild CXCR3 15 42 COc1cncc(NC(=O)N(C)Cc2ncc[nH]2)c1 ZINC000880543552 CD On-Demand Anodyne ROCK2 17 40 COC[C@@H]1CCCN1NC(=O)Nc1cncc(OC)c1 ZINC000880543578 CD On-Demand Anodyne CASP7 44 35 COc1cncc(NC(=O)N[C@H]2CCOc3c(C)cccc32)c1 ZINC000880543604 DG On-Demand Anodyne TRPV1 15 43 COc1cncc(NC(=O)N[C@@H]2CCOc3c(C)cccc32)c1 ZINC000880543605 DG On-Demand Anodyne TRPV1 15 43 COc1cncc(NC(=O)N2CCc3c(CC#N)cccc3C2)c1 ZINC000880543609 DF On-Demand Mild DRD4 40 30 COc1cncc(NC(=O)N2CCc3c(CC#N)cccc3C2)c1 ZINC000880543609 DF On-Demand Mild P2RY14 51 39 COc1cncc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)c1 ZINC000880543627 DD On-Demand Anodyne CCR3 27 42 COc1cncc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)c1 ZINC000880543627 DD On-Demand Anodyne CXCR3 19 42 COc1cncc(NC(=O)N2CCC(CCF)CC2)c1 ZINC000880543636 CF On-Demand Anodyne PDGFRB 40 35 COc1cncc(NC(=O)N2CCC(OCc3ccc(F)cc3)CC2)c1 ZINC000880543661 FG On-Demand Anodyne GRIN2B 31 40 COc1cncc(NC(=O)N2CCC(OCc3ccc(F)cc3)CC2)c1 ZINC000880543661 FG On-Demand Anodyne CCR3 64 49 COc1cncc(NC(=O)N2CCC(OCc3ccc(F)cc3)CC2)c1 ZINC000880543661 FG On-Demand Anodyne SCD1 24 40 COc1cncc(NC(=O)NC2CCN(CC(=O)OC(C)(C)C)CC2)c1 ZINC000880543662 FE On-Demand Anodyne EPHX2 42 40 COc1cncc(NC(=O)NC2CCN(CC(=O)OC(C)(C)C)CC2)c1 ZINC000880543662 FE On-Demand Anodyne CXCR3 19 43 N#Cc1ccnc(N2CCN(C(=O)/C=C\c3ccccc3Cl)CC2)c1 ZINC000880543670 FF On-Demand Mild ITGAL 42 33 N#Cc1ccnc(N2CCN(C(=O)/C=C\c3ccccc3Cl)CC2)c1 ZINC000880543670 FF On-Demand Mild PDK1 24 43 COc1cncc(NC(=O)NC2CCC(OC(C)(C)C)CC2)c1 ZINC000880543785 DG On-Demand Anodyne EPHX2 53 40 COc1cncc(NC(=O)N2CCN(c3nccnn3)CC2)c1 ZINC000880543790 DC On-Demand Anodyne PDGFRB 51 40 COc1cncc(NC(=O)N2CCC(C)(F)CC2)c1 ZINC000880543796 CE On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)NC[C@H](OC)c2cccc(OC)c2)c1 ZINC000880543806 EF On-Demand Anodyne ROCK1 26 42 COc1cncc(NC(=O)NC[C@H](OC)c2cccc(OC)c2)c1 ZINC000880543806 EF On-Demand Anodyne MTNR1B 32 43 COc1cncc(NC(=O)NC[C@@H](OC)c2cccc(OC)c2)c1 ZINC000880543807 EF On-Demand Anodyne ROCK1 26 42 COc1cncc(NC(=O)NC[C@@H](OC)c2cccc(OC)c2)c1 ZINC000880543807 EF On-Demand Anodyne MTNR1B 32 43 COc1cncc(NC(=O)NC[C@@H](C)c2ccncc2)c1 ZINC000880543809 CE On-Demand Anodyne ROCK2 15 43 COc1cncc(NC(=O)NC[C@H](C)c2ccncc2)c1 ZINC000880543810 CE On-Demand Anodyne ROCK2 15 43 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)c1 ZINC000880543828 EE On-Demand Mild PDGFRB 56 52 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)c1 ZINC000880543828 EE On-Demand Mild SSTR1 20 42 COc1cncc(NC(=O)NCc2ccc(C3(C)OCCO3)cc2)c1 ZINC000880543839 EF On-Demand Anodyne ROCK2 17 42 COc1cncc(NC(=O)NC[C@H]2CCCN2C)c1 ZINC000880543842 CD On-Demand Anodyne CCR3 33 41 COc1cncc(NC(=O)NC[C@H]2CCCN2C)c1 ZINC000880543842 CD On-Demand Anodyne CHRNA10 56 40 COc1cncc(NC(=O)NC[C@H]2CCCN2C)c1 ZINC000880543842 CD On-Demand Anodyne ACKR3 65 33 COc1cncc(NC(=O)NC[C@@H]2CCCN2C)c1 ZINC000880543843 CD On-Demand Anodyne CCR3 33 41 COc1cncc(NC(=O)NC[C@@H]2CCCN2C)c1 ZINC000880543843 CD On-Demand Anodyne CHRNA10 56 40 COc1cncc(NC(=O)NC[C@@H]2CCCN2C)c1 ZINC000880543843 CD On-Demand Anodyne ACKR3 65 33 COc1cncc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)c1 ZINC000880543845 FD On-Demand Anodyne ROCK2 23 42 COc1cncc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)c1 ZINC000880543845 FD On-Demand Anodyne PROKR1 50 31 COc1cncc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)c1 ZINC000880543845 FD On-Demand Anodyne NAMPT 49 42 COc1cncc(NC(=O)N(CCN(C)C)CC(=O)N(C)C)c1 ZINC000880543863 DC On-Demand Anodyne ROCK2 16 43 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccccc1C(F)(F)F ZINC000880543872 FF On-Demand Anodyne RBP4 44 32 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1CCC2(CC1)COCCO2 ZINC000880543890 GH On-Demand Anodyne PRNP 52 37 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1CCC2(CC1)COCCO2 ZINC000880543890 GH On-Demand Anodyne KCNK3 108 41 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1CCC2(CC1)COCCO2 ZINC000880543890 GH On-Demand Anodyne KCNK9 64 40 COc1cncc(NC(=O)N[C@@H]2CCc3ccccc32)c1 ZINC000880543897 CF On-Demand Anodyne TRPV1 16 42 COc1cncc(NC(=O)N[C@@H]2CCc3ccccc32)c1 ZINC000880543897 CF On-Demand Anodyne NPY1R 25 41 COc1cncc(NC(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880543919 DE On-Demand Anodyne HTR4 28 41 COc1cncc(NC(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880543919 DE On-Demand Anodyne CCR3 61 46 COc1cncc(NC(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880543919 DE On-Demand Anodyne CACNA1I 61 37 COc1cncc(NC(=O)N[C@H]2CCC[C@H]2Cc2cnn(C)c2)c1 ZINC000880543922 EE On-Demand Anodyne CCR3 37 42 COc1cncc(NC(=O)N[C@H]2CCC[C@@H]2Cc2cnn(C)c2)c1 ZINC000880543923 EE On-Demand Anodyne CCR3 37 42 COc1cncc(NC(=O)N[C@@H]2CCC[C@@H]2Cc2cnn(C)c2)c1 ZINC000880543924 EE On-Demand Anodyne CCR3 37 42 COc1cncc(NC(=O)N[C@@H]2CCC[C@H]2Cc2cnn(C)c2)c1 ZINC000880543925 EE On-Demand Anodyne CCR3 37 42 c1ccc(-c2ncc(CN3CCC4(CC3)COCCO4)cn2)cc1 ZINC000880543938 EF On-Demand Anodyne SIGMAR1 31 40 CCn1ccc(NC(=O)Nc2cncc(OC)c2)n1 ZINC000880543941 CD On-Demand Anodyne PDGFRB 21 44 COc1cncc(NC(=O)NCc2ccc(N3CCCNC3=O)cc2)c1 ZINC000880543963 FE On-Demand Anodyne ROCK2 17 41 COc1cncc(NC(=O)NCc2ccc(N3CCCNC3=O)cc2)c1 ZINC000880543963 FE On-Demand Anodyne NAMPT 39 40 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean HTR1A 39 53 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean DRD2 32 40 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean DRD4 22 40 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean HTR1D 15 53 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean HTR1B 20 53 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean DRD3 44 37 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean PDGFRB 75 51 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean HTR7 31 45 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean PDGFRA 17 46 COc1cncc(NC(=O)N2CCN(c3ccc(OC)cc3OC)CC2)c1 ZINC000880543964 FE On-Demand Clean RBP4 17 43 COc1cncc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)c1 ZINC000880543976 EF On-Demand Anodyne EPHX2 32 47 COc1cncc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)c1 ZINC000880543977 EF On-Demand Anodyne EPHX2 32 47 CCC1(N(C)C)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880543978 DE On-Demand Anodyne S1PR2 28 41 COc1cncc(NC(=O)NC2CCC(OC(C)C)CC2)c1 ZINC000880543981 DF On-Demand Anodyne EPHX2 51 40 COc1cncc(NC(=O)N2CCO[C@@](C)(C(F)(F)F)C2)c1 ZINC000880543986 DE On-Demand Anodyne EPHX2 31 42 COc1cncc(NC(=O)N2CCO[C@](C)(C(F)(F)F)C2)c1 ZINC000880543987 DE On-Demand Anodyne EPHX2 31 42 CCCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880543991 EH On-Demand Anodyne INHA 42 35 CCCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880543991 EH On-Demand Anodyne BMP1 21 41 CCCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880543991 EH On-Demand Anodyne ROCK1 15 44 CCCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880543991 EH On-Demand Anodyne ROCK2 24 44 COc1cncc(NC(=O)N2CCN(C)C(C)(C)CC2)c1 ZINC000880543992 CE On-Demand Anodyne PDGFRB 43 36 COc1cncc(NC(=O)N[C@@H]2CCO[C@H]2c2cccnc2)c1 ZINC000880544000 DE On-Demand Anodyne CHRNA7 30 46 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880544042 GD On-Demand Anodyne EPHX2 23 42 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc(N2CCOCC2)cc1 ZINC000880544042 GD On-Demand Anodyne STAT6 67 36 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)c1 ZINC000880544050 FE On-Demand Mild P2RY12 17 47 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)c1 ZINC000880544050 FE On-Demand Mild PDGFRB 51 41 COc1cncc(NC(=O)NCCC2CCC2)c1 ZINC000880544051 BE On-Demand Anodyne CCR3 34 41 O=C(CN1CCC2(CC1)COCCO2)Nc1nc(-c2ccccc2)cs1 ZINC000880544058 FF On-Demand Anodyne CPT1A 18 41 O=C(CN1CCC2(CC1)COCCO2)Nc1nc(-c2ccccc2)cs1 ZINC000880544058 FF On-Demand Anodyne ROCK1 20 42 O=C(CN1CCC2(CC1)COCCO2)Nc1nc(-c2ccccc2)cs1 ZINC000880544058 FF On-Demand Anodyne HDAC9 15 46 COc1cncc(NC(=O)N2CCN(C)c3ncccc3C2)c1 ZINC000880544060 DD On-Demand Anodyne PDGFRB 52 40 O=C(CN1CCC2(CC1)COCCO2)Nc1nccs1 ZINC000880544062 CC On-Demand Anodyne MAP1 101 50 O=C(CN1CCC2(CC1)COCCO2)Nc1nccs1 ZINC000880544062 CC On-Demand Anodyne SLC27A1 29 40 O=C(CCN1CCC2(CC1)COCCO2)NC(c1ccccc1)c1ccccc1 ZINC000880544067 GG On-Demand Anodyne PRCP 28 48 C#CCC1(O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880544091 CD On-Demand Mild S1PR2 30 43 COC(=O)c1ccc(OC)c2c1CCN(C(=O)Nc1cncc(OC)c1)C2 ZINC000880544092 FE On-Demand Anodyne P2RY14 46 35 COc1cncc(NC(=O)NCc2cc(C3CC3)ccc2OC)c1 ZINC000880544101 EG On-Demand Anodyne TSHR 50 33 O=C(CN1CCC2(CC1)COCCO2)Nc1cccnc1Cl ZINC000880544105 ED On-Demand Anodyne G2YM83_BOTF4 68 35 N#Cc1c(NC(=O)CCN2CCC3(CC2)COCCO3)sc2c1CCC2 ZINC000880544119 GE On-Demand Mild VIPR1 30 48 COc1ccc(CN(CCO)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880544134 EE On-Demand Anodyne BMP1 36 43 COc1ccc(CN(CCO)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880544134 EE On-Demand Anodyne ROCK1 15 52 COc1ccc(CN(CCO)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880544134 EE On-Demand Anodyne ROCK2 25 52 C[C@H](C(=O)Nc1cccc(C#N)c1)N1CCC2(CC1)COCCO2 ZINC000880544148 ED On-Demand Mild MCHR1 26 40 Nc1nc(CN2CCC3(CC2)COCCO3)nc(Nc2ccc(F)cc2)n1 ZINC000880544156 FD On-Demand Anodyne STAT6 40 33 COc1cncc(NC(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)c1 ZINC000880544204 FH On-Demand Anodyne KCNH2 41 42 COc1cncc(NC(=O)N2CC[C@](C)(c3cccc(OC)c3)C2)c1 ZINC000880544218 EG On-Demand Anodyne NPY5R 23 41 COc1cncc(NC(=O)N2CC[C@](C)(c3cccc(OC)c3)C2)c1 ZINC000880544218 EG On-Demand Anodyne EPHX2 35 43 COc1cncc(NC(=O)N2CC[C@@](C)(c3cccc(OC)c3)C2)c1 ZINC000880544219 EG On-Demand Anodyne NPY5R 23 41 COc1cncc(NC(=O)N2CC[C@@](C)(c3cccc(OC)c3)C2)c1 ZINC000880544219 EG On-Demand Anodyne EPHX2 35 43 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2OC)c1 ZINC000880544229 DF On-Demand Anodyne PDGFRA 41 35 COc1cncc(NC(=O)N2CCN(C(=O)c3cccn3C)CC2)c1 ZINC000880544250 ED On-Demand Anodyne PDGFRB 41 38 CCNC(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880544255 CC On-Demand Anodyne MTNR1B 15 44 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne CHRM3 23 45 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne SIGMAR1 38 40 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne FAAH 15 50 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne NPFFR1 46 37 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne NOD2 41 34 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne KCNK3 86 39 O=C(Nc1ccccc1)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880544275 FG On-Demand Anodyne KCNK9 40 36 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc(Br)c1 ZINC000880544284 GF On-Demand Anodyne EGFR 22 52 COc1cncc(NC(=O)NCc2cccc(OC)c2C)c1 ZINC000880544290 DF On-Demand Anodyne PDGFRB 36 41 COc1cncc(NC(=O)NCc2cccc(OC)c2C)c1 ZINC000880544290 DF On-Demand Anodyne RAF1 15 40 COc1cncc(NC(=O)NCc2cccc(OC)c2C)c1 ZINC000880544290 DF On-Demand Anodyne MTNR1B 24 40 COc1cncc(NC(=O)NCc2cccc(OC)c2C)c1 ZINC000880544290 DF On-Demand Anodyne ROCK2 28 48 COc1cncc(NC(=O)NCc2cccc(OC)c2C)c1 ZINC000880544290 DF On-Demand Anodyne KCNK3 43 37 CCN(CC)C(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880544302 CD On-Demand Anodyne MTNR1B 15 41 CCC1(N2CCCCC2)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880544305 EG On-Demand Anodyne HCN1 49 32 CCC1(N2CCCCC2)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880544305 EG On-Demand Anodyne HCN4 47 32 N#Cc1cccc(NC(=O)CCN2CCC3(CC2)COCCO3)c1 ZINC000880544308 ED On-Demand Mild CCR3 15 42 N#Cc1cccc(NC(=O)CCN2CCC3(CC2)COCCO3)c1 ZINC000880544308 ED On-Demand Mild MCHR1 39 42 c1cn(-c2ccc(CN3CCC4(CC3)COCCO4)cc2)cn1 ZINC000880544309 DE On-Demand Anodyne CYP2C19 16 44 C[C@H](C(=O)Nc1cccnc1Cl)N1CCC2(CC1)COCCO2 ZINC000880544316 ED On-Demand Anodyne G2YM83_BOTF4 69 36 COc1cncc(NC(=O)N2CCc3cc(F)ccc3[C@H]2C)c1 ZINC000880544320 DG On-Demand Anodyne TRPM8 31 46 COc1cncc(NC(=O)N2CCc3cc(F)ccc3[C@@H]2C)c1 ZINC000880544321 DG On-Demand Anodyne TRPM8 31 46 O=C(CN1CCC2(CC1)COCCO2)Nc1cc(Cl)ccc1F ZINC000880544328 EE On-Demand Anodyne CCR1 50 37 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCCCC2)nc1 ZINC000880544329 FD On-Demand Anodyne SLC27A1 57 44 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3[C@H]2C)c1 ZINC000880544330 FG On-Demand Anodyne SLC18A2 46 33 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3[C@H]2C)c1 ZINC000880544330 FG On-Demand Anodyne MTNR1B 17 43 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3[C@@H]2C)c1 ZINC000880544331 FG On-Demand Anodyne SLC18A2 46 33 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3[C@@H]2C)c1 ZINC000880544331 FG On-Demand Anodyne MTNR1B 17 43 COc1cncc(NC(=O)N2CCC(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000880544333 GF On-Demand Anodyne MMP13 22 40 COc1cncc(NC(=O)N2CCC(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000880544333 GF On-Demand Anodyne MMP3 21 40 COc1cncc(NC(=O)N2CCC(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000880544333 GF On-Demand Anodyne MMP9 15 40 COc1cncc(NC(=O)N2CCC(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000880544333 GF On-Demand Anodyne MMP1 18 40 COc1cncc(NC(=O)N2CCC(S(=O)(=O)c3ccc(C)cc3)CC2)c1 ZINC000880544333 GF On-Demand Anodyne NAMPT 17 40 C[C@H](C(=O)Nc1ccccc1[N+](=O)[O-])N1CCC2(CC1)COCCO2 ZINC000880544348 ED On-Demand Bother COLA 110 36 CN1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880544373 BC On-Demand Mild PDGFRB 46 41 COC(=O)c1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880544375 ED On-Demand Anodyne CASR 15 44 COC(=O)c1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880544375 ED On-Demand Anodyne EPHX2 19 41 COC(=O)c1cccc(NC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880544375 ED On-Demand Anodyne HIF1A 15 41 COc1cncc(NC(=O)N2CC[C@@](C)(NC(=O)C(F)(F)F)C2)c1 ZINC000880544389 ED On-Demand Anodyne EPHX2 33 41 COc1cncc(NC(=O)N2CC[C@](C)(NC(=O)C(F)(F)F)C2)c1 ZINC000880544390 ED On-Demand Anodyne EPHX2 33 41 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1cncc(OC)c1)C2 ZINC000880544391 EE On-Demand Anodyne P2RY14 42 33 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean HTR1A 16 41 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean DRD4 44 37 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean HTR1B 15 41 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean LCK 19 43 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean ROCK2 20 42 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean FLT3 23 44 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean AURKA 18 44 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880544393 FE On-Demand Clean NAMPT 48 39 COc1cncc(NC(=O)NC[C@@H](O)c2ccccc2OC)c1 ZINC000880544434 DD On-Demand Anodyne ADRB1 42 32 COc1cncc(NC(=O)NC[C@@H](O)c2ccccc2OC)c1 ZINC000880544434 DD On-Demand Anodyne MTNR1A 17 43 COc1cncc(NC(=O)NC[C@@H](O)c2ccccc2OC)c1 ZINC000880544434 DD On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)NC[C@@H](O)c2ccccc2OC)c1 ZINC000880544434 DD On-Demand Anodyne SOAT1 41 39 COc1cncc(NC(=O)N2CC(Cc3cccc(C)c3)C2)c1 ZINC000880544435 DG On-Demand Anodyne CCR3 21 49 COc1cncc(NC(=O)N2CCC(O)(CO)CC2)c1 ZINC000880544443 CC On-Demand Anodyne PDGFRB 44 38 COc1cncc(NC(=O)N2CCC(O)(CO)CC2)c1 ZINC000880544443 CC On-Demand Anodyne S1PR2 31 46 O=C1NC2(CCO1)CN(C(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C2 ZINC000880544445 GD On-Demand Anodyne PREP 24 41 COc1cncc(NC(=O)N2CC(Cc3ccccc3C)C2)c1 ZINC000880544446 DG On-Demand Anodyne PDGFRB 40 36 COc1cncc(NC(=O)N2CC(Cc3ccccc3C)C2)c1 ZINC000880544446 DG On-Demand Anodyne CCR3 18 45 COc1cncc(NC(=O)NCc2cccc(OC3CC3)c2F)c1 ZINC000880544455 EG On-Demand Anodyne PDE4A 15 40 COc1cncc(NC(=O)NCc2cccc(OC3CC3)c2F)c1 ZINC000880544455 EG On-Demand Anodyne P2RX7 19 40 COc1cncc(NC(=O)NCc2cccc(OC3CC3)c2F)c1 ZINC000880544455 EG On-Demand Anodyne CCR3 30 41 COc1cncc(NC(=O)N2CC(C)(c3ccccc3)C2)c1 ZINC000880544465 CF On-Demand Anodyne EPHX2 21 46 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544473 EF On-Demand Anodyne ROCK1 28 52 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544473 EF On-Demand Anodyne MTNR1A 26 40 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544473 EF On-Demand Anodyne MTNR1B 28 40 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544474 EF On-Demand Anodyne ROCK1 28 52 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544474 EF On-Demand Anodyne MTNR1A 26 40 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1cccc(OC)c1 ZINC000880544474 EF On-Demand Anodyne MTNR1B 28 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3OC)CC2)c1 ZINC000880544475 FE On-Demand Anodyne PDGFRB 54 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3OC)CC2)c1 ZINC000880544475 FE On-Demand Anodyne KCNK3 35 42 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3OC)CC2)c1 ZINC000880544475 FE On-Demand Anodyne KCNK9 27 42 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880544481 FE On-Demand Anodyne CSNK1D 45 40 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880544481 FE On-Demand Anodyne PIK3CA 18 44 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccc(F)cc2s1 ZINC000880544481 FE On-Demand Anodyne SLC27A1 45 51 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCCC2)cc1 ZINC000880544500 FE On-Demand Anodyne STAT6 55 31 C[C@H](C(=O)Nc1sc2c(c1C#N)CCC2)N1CCC2(CC1)COCCO2 ZINC000880544507 GE On-Demand Mild VIPR1 25 40 C[C@@H](C(=O)Nc1sc2c(c1C#N)CCC2)N1CCC2(CC1)COCCO2 ZINC000880544508 GE On-Demand Mild VIPR1 25 40 COc1cncc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880544510 EH On-Demand Anodyne CACNA1H 48 42 COc1cncc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880544510 EH On-Demand Anodyne GRIN2B 18 41 COc1cncc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880544510 EH On-Demand Anodyne CCR1 24 41 COc1cncc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880544510 EH On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880544510 EH On-Demand Anodyne EPHX2 20 40 COc1cncc(NC(=O)N2CC[C@@]3(CN(Cc4ccccc4)C(=O)CO3)C2)c1 ZINC000880544525 GE On-Demand Anodyne FAAH 15 41 COc1cncc(NC(=O)N2CC[C@@]3(CN(Cc4ccccc4)C(=O)CO3)C2)c1 ZINC000880544525 GE On-Demand Anodyne EPHX2 28 41 COc1cncc(NC(=O)N2CC[C@]3(CN(Cc4ccccc4)C(=O)CO3)C2)c1 ZINC000880544526 GE On-Demand Anodyne FAAH 15 41 COc1cncc(NC(=O)N2CC[C@]3(CN(Cc4ccccc4)C(=O)CO3)C2)c1 ZINC000880544526 GE On-Demand Anodyne EPHX2 28 41 COc1cncc(NC(=O)N2CCC3(CCCCO3)CC2)c1 ZINC000880544535 DF On-Demand Anodyne EPHX2 18 41 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccccc1-c1ccccc1 ZINC000880544536 GH On-Demand Anodyne CHRM3 19 42 COc1cncc(NC(=O)N2CCC[C@@H](CF)C2)c1 ZINC000880544537 CE On-Demand Anodyne CCR3 25 50 COc1cncc(NC(=O)N2CCC[C@H](CF)C2)c1 ZINC000880544538 CE On-Demand Anodyne CCR3 25 50 COc1cncc(NC(=O)NC[C@H](CO)c2ccc(Cl)cc2)c1 ZINC000880544557 EF On-Demand Anodyne SCN10A 31 41 COc1cncc(NC(=O)NC[C@@H](CO)c2ccc(Cl)cc2)c1 ZINC000880544558 EF On-Demand Anodyne SCN10A 31 41 C[C@H](C(=O)Nc1nccs1)N1CCC2(CC1)COCCO2 ZINC000880544567 DD On-Demand Anodyne MAP1 88 35 C[C@@H](C(=O)Nc1nccs1)N1CCC2(CC1)COCCO2 ZINC000880544568 DD On-Demand Anodyne MAP1 88 35 COc1cncc(NC(=O)Nc2cc3n(n2)CCN(Cc2ccccc2)C3)c1 ZINC000880544578 GF On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)Nc2cc3n(n2)CCN(Cc2ccccc2)C3)c1 ZINC000880544578 GF On-Demand Anodyne FAAH 15 41 COc1ccc2c(CN3CCC4(CC3)COCCO4)cc(=O)oc2c1 ZINC000880544584 EE On-Demand Anodyne CYP11B1 17 43 COc1cncc(NC(=O)N[C@@H]2CC[C@H](O)CC2)c1 ZINC000880544592 CD On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)NC[C@H](O)c2cccc(C(F)(F)F)c2)c1 ZINC000880544593 FF On-Demand Anodyne PDS 40 35 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(C(F)(F)F)c2)c1 ZINC000880544594 FF On-Demand Anodyne PDS 40 35 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne INHA 82 39 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne TRPV1 15 47 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne RAF1 37 44 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne MTNR1A 35 43 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne MTNR1B 29 43 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne QPCT 17 41 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne NCE103 17 43 COc1cncc(NC(=O)NCCc2ccc(OC)c(O)c2)c1 ZINC000880544596 DE On-Demand Anodyne P96878_MYCTU 17 43 O=C(CN1CCC2(CC1)COCCO2)Nc1nc(-c2ccc(F)cc2)cs1 ZINC000880544598 GF On-Demand Anodyne ROCK1 18 44 O=C(CN1CCC2(CC1)COCCO2)Nc1nc(-c2ccc(F)cc2)cs1 ZINC000880544598 GF On-Demand Anodyne SLC27A1 42 42 COc1cncc(NC(=O)NN2CCc3ccccc3C2)c1 ZINC000880544609 CE On-Demand Anodyne NOD1 15 42 COc1cncc(NC(=O)NN2CCc3ccccc3C2)c1 ZINC000880544609 CE On-Demand Anodyne NOD2 42 42 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccccc2s1 ZINC000880544611 EE On-Demand Anodyne CASR 17 44 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccccc2s1 ZINC000880544611 EE On-Demand Anodyne CSNK1D 39 48 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccccc2s1 ZINC000880544611 EE On-Demand Anodyne ACOX1 45 34 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2ccccc2s1 ZINC000880544611 EE On-Demand Anodyne SLC27A1 38 56 COc1cncc(NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)c1 ZINC000880544641 DE On-Demand Anodyne CCR3 101 43 COc1cncc(NC(=O)NC[C@H]2CCCN(CC3CC3)C2)c1 ZINC000880544642 DE On-Demand Anodyne CCR3 101 43 COc1cncc(NC(=O)NCCc2cncc(C)n2)c1 ZINC000880544657 CD On-Demand Anodyne PIK3CG 15 42 COc1cncc(NC(=O)NC2CCC3(CC2)CC3(F)F)c1 ZINC000880544658 DG On-Demand Anodyne EPHX2 43 35 CCC(CC)C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880544659 EE On-Demand Anodyne PDGFRB 45 36 CCC(CC)C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880544659 EE On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCC3(COC3)C2)c1 ZINC000880544661 CD On-Demand Anodyne EPHX2 32 44 O=c1ccc([N+](=O)[O-])cn1CCN1CCC2(CC1)COCCO2 ZINC000880544664 DC On-Demand Bother KCNJ1 21 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880544690 EE On-Demand Anodyne EPHX2 45 39 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880544690 EE On-Demand Anodyne GPR119 38 40 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne DRD2 36 45 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne SIGMAR1 25 46 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne CCR3 57 44 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne CHRNA7 23 41 COc1cncc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880544695 EE On-Demand Anodyne MCHR1 18 41 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne DRD2 36 45 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne SIGMAR1 25 46 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne CCR3 57 44 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne CHRNA7 23 41 COc1cncc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880544696 EE On-Demand Anodyne MCHR1 18 41 COC(=O)[C@@H](c1ccccc1)N1CCC2(CC1)COCCO2 ZINC000880544698 DD On-Demand Anodyne NPY2R 23 44 COc1cncc(NC(=O)N[C@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544716 EG On-Demand Anodyne PTAFR 22 42 COc1cncc(NC(=O)N[C@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544716 EG On-Demand Anodyne PDE4A 21 42 COc1cncc(NC(=O)N[C@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544716 EG On-Demand Anodyne CHRNA7 41 46 COc1cncc(NC(=O)N[C@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544716 EG On-Demand Anodyne C3AR1 36 43 COc1cncc(NC(=O)N[C@@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544717 EG On-Demand Anodyne PTAFR 22 42 COc1cncc(NC(=O)N[C@@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544717 EG On-Demand Anodyne PDE4A 21 42 COc1cncc(NC(=O)N[C@@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544717 EG On-Demand Anodyne CHRNA7 41 46 COc1cncc(NC(=O)N[C@@H](Cc2cccnc2)C2CCCC2)c1 ZINC000880544717 EG On-Demand Anodyne C3AR1 36 43 COC(=O)c1cnc(CC2CCN(C(=O)Nc3cncc(OC)c3)CC2)s1 ZINC000880544772 GF On-Demand Anodyne CCR3 15 43 COc1cncc(NC(=O)N2CCc3ccsc3[C@@H]2C)c1 ZINC000880544779 DG On-Demand Anodyne TRPM8 23 43 COc1cncc(NC(=O)N2CCc3ccsc3[C@H]2C)c1 ZINC000880544780 DG On-Demand Anodyne TRPM8 23 43 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(N2CCCCCC2)cc1 ZINC000880544785 GF On-Demand Anodyne STAT6 50 31 COCc1csc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880544812 DF On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880544816 DF On-Demand Anodyne CCR3 31 44 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880544816 DF On-Demand Anodyne CHRNA7 17 40 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880544816 DF On-Demand Anodyne PDE3B 41 39 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880544816 DF On-Demand Anodyne EPHX2 35 48 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880544816 DF On-Demand Anodyne SCD1 22 52 COc1cncc(NC(=O)N[C@@H](C)COc2c(F)cccc2F)c1 ZINC000880544837 EF On-Demand Anodyne MTNR1B 16 44 COc1cncc(NC(=O)N[C@H](C)COc2c(F)cccc2F)c1 ZINC000880544838 EF On-Demand Anodyne MTNR1B 16 44 c1cncc(CCN2CCC3(CC2)COCCO3)c1 ZINC000880544848 CD On-Demand Anodyne SIGMAR1 15 45 COc1cncc(NC(=O)N2CCc3nccnc3C2)c1 ZINC000880544849 CD On-Demand Anodyne P2RY14 45 34 COc1cncc(NC(=O)N2CCC(c3ccon3)CC2)c1 ZINC000880544851 DE On-Demand Anodyne SMO 21 47 CCOc1ccccc1NC(=O)CCN1CCC2(CC1)COCCO2 ZINC000880544855 EE On-Demand Anodyne CCR1 35 40 CCOc1ccccc1NC(=O)CCN1CCC2(CC1)COCCO2 ZINC000880544855 EE On-Demand Anodyne HCN1 55 38 CCOc1ccccc1NC(=O)CCN1CCC2(CC1)COCCO2 ZINC000880544855 EE On-Demand Anodyne HCN4 45 36 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne DRD4 23 46 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne ACHE 35 44 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne HRH2 20 43 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne SIGMAR1 28 44 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne SSTR5 50 36 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne CCR3 90 52 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne PDK1 34 41 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne CXCR3 26 43 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne MCHR1 42 43 COc1cncc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880544876 FF On-Demand Anodyne CACNA1I 70 42 Oc1nc(CN2CCC3(CC2)COCCO3)nc2c1oc1ccccc12 ZINC000880544914 FE On-Demand Anodyne CDC7 15 49 Oc1nc(CN2CCC3(CC2)COCCO3)nc2c1oc1ccccc12 ZINC000880544914 FE On-Demand Anodyne PIM3 22 49 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](C)CO)c1 ZINC000880544956 DF On-Demand Anodyne ROCK2 26 47 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](C)CO)c1 ZINC000880544956 DF On-Demand Anodyne NPY5R 35 43 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](C)CO)c1 ZINC000880544957 DF On-Demand Anodyne ROCK2 26 47 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](C)CO)c1 ZINC000880544957 DF On-Demand Anodyne NPY5R 35 43 COc1cncc(NC(=O)Nc2ccc(O)c(C(C)C)c2)c1 ZINC000880544958 DH On-Demand Anodyne THRA 72 39 COc1cncc(NC(=O)Nc2ccc(O)c(C(C)C)c2)c1 ZINC000880544958 DH On-Demand Anodyne THRB 74 44 COc1cncc(NC(=O)N2CC[C@@]3(CN(Cc4ccccc4)C[C@H](C)O3)C2)c1 ZINC000880544962 GF On-Demand Anodyne FAAH 21 45 COc1cncc(NC(=O)N2CC[C@]3(CN(Cc4ccccc4)C[C@H](C)O3)C2)c1 ZINC000880544963 GF On-Demand Anodyne FAAH 21 45 COc1cncc(NC(=O)N2CC[C@@]3(CN(Cc4ccccc4)C[C@@H](C)O3)C2)c1 ZINC000880544964 GF On-Demand Anodyne FAAH 21 45 COc1cncc(NC(=O)N2CC[C@]3(CN(Cc4ccccc4)C[C@@H](C)O3)C2)c1 ZINC000880544965 GF On-Demand Anodyne FAAH 21 45 COc1cncc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)c1 ZINC000880544966 EE On-Demand Anodyne ADRB1 40 32 COc1cncc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)c1 ZINC000880544966 EE On-Demand Anodyne CTSL 17 42 COc1cncc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)c1 ZINC000880544967 EE On-Demand Anodyne ADRB1 40 32 COc1cncc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)c1 ZINC000880544967 EE On-Demand Anodyne CTSL 17 42 COc1cncc(NC(=O)N2CCC(c3nc(C4CCC4)no3)CC2)c1 ZINC000880544968 FG On-Demand Anodyne SMO 36 51 COc1cncc(NC(=O)N2CCC(c3nc(C4CCC4)no3)CC2)c1 ZINC000880544968 FG On-Demand Anodyne ETHR 58 43 O=C(CN1CCC2(CC1)COCCO2)NC(=O)Nc1ccccc1 ZINC000880544983 ED On-Demand Anodyne EPHX2 20 42 COc1cncc(NC(=O)N2CCc3ncncc3C2)c1 ZINC000880544984 CD On-Demand Anodyne P2RY14 47 37 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccc2ccccc12 ZINC000880544988 FG On-Demand Anodyne PRKDC 52 38 O=c1cc(CN2CCC3(CC2)COCCO3)c2ccc(O)cc2o1 ZINC000880544993 ED On-Demand Anodyne HSD17B3 35 50 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc(Cl)cc1 ZINC000880545004 EF On-Demand Anodyne CCR1 39 40 O=C(CCN1CCC2(CC1)COCCO2)Nc1ccc(Cl)cc1 ZINC000880545004 EF On-Demand Anodyne EPHX2 27 45 COc1cncc(NC(=O)N2CCC(=O)N(C)CC2)c1 ZINC000880545005 CC On-Demand Anodyne PDGFRB 49 40 COc1cncc(NC(=O)N(CCN2CCOCC2)CC2CC2)c1 ZINC000880545006 ED On-Demand Anodyne CASR 61 53 Cc1cccc(C(=O)NNC(=O)CN2CCC3(CC2)COCCO3)c1 ZINC000880545008 EC On-Demand Reactive KCNK3 48 36 COc1cncc(NC(=O)N2Cc3ccccc3[C@H]2C)c1 ZINC000880545022 CG On-Demand Anodyne CFTR 42 35 COc1cncc(NC(=O)N2Cc3ccccc3[C@@H]2C)c1 ZINC000880545023 CG On-Demand Anodyne CFTR 42 35 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2c(s1)CCC2 ZINC000880545036 ED On-Demand Anodyne SLC27A1 60 54 COc1cncc(NC(=O)NCc2cccc(COC[C@H]3CCCO3)c2)c1 ZINC000880545043 FG On-Demand Anodyne ROCK2 33 44 COc1cncc(NC(=O)NCc2cccc(COC[C@@H]3CCCO3)c2)c1 ZINC000880545044 FG On-Demand Anodyne ROCK2 33 44 COc1cncc(NC(=O)N2CCC(c3nccc(N4CCOCC4)n3)CC2)c1 ZINC000880545053 GE On-Demand Anodyne EPHB4 36 41 COc1cncc(NC(=O)N2CCC[C@H](CCF)C2)c1 ZINC000880545061 CF On-Demand Anodyne CCR3 21 53 COc1cncc(NC(=O)N2CCC[C@@H](CCF)C2)c1 ZINC000880545062 CF On-Demand Anodyne CCR3 21 53 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCC2(CC1)COCCO2 ZINC000880545079 GF On-Demand Anodyne PDE8B 54 36 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)[C@H](CO)C2)c1 ZINC000880545087 EF On-Demand Anodyne EPHX2 22 41 COc1cncc(NC(=O)NC2CC(Nc3ccccc3)C2)c1 ZINC000880545100 DF On-Demand Anodyne EPHX2 32 41 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(OC(F)(F)F)cc1 ZINC000880545109 GE On-Demand Anodyne MMP2 22 40 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(OC(F)(F)F)cc1 ZINC000880545109 GE On-Demand Anodyne MMP14 19 40 O=C(CN1CCC2(CC1)COCCO2)NCc1ccc(OC(F)(F)F)cc1 ZINC000880545109 GE On-Demand Anodyne MMP9 21 40 COc1cncc(NC(=O)N2CC(O)(c3ccc(F)cc3)C2)c1 ZINC000880545113 DD On-Demand Anodyne S1PR2 29 43 COc1cncc(NC(=O)NCCn2ccc(C(F)(F)F)n2)c1 ZINC000880545114 EE On-Demand Anodyne QPCT 15 42 COc1cncc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545119 FD On-Demand Anodyne CCR3 69 41 COc1cncc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545119 FD On-Demand Anodyne CHRNA7 16 41 COc1cncc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545119 FD On-Demand Anodyne EPHX2 40 51 COc1cncc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545120 FD On-Demand Anodyne CCR3 69 41 COc1cncc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545120 FD On-Demand Anodyne CHRNA7 16 41 COc1cncc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)c1 ZINC000880545120 FD On-Demand Anodyne EPHX2 40 51 COc1cncc(NC(=O)N2CC[C@@](C)(C(F)(F)F)C2)c1 ZINC000880545135 DF On-Demand Anodyne EPHX2 34 42 COc1cncc(NC(=O)N2CC[C@](C)(C(F)(F)F)C2)c1 ZINC000880545136 DF On-Demand Anodyne EPHX2 34 42 COc1cncc(NC(=O)N2CC(Cc3ccc(C)cc3)C2)c1 ZINC000880545150 DG On-Demand Anodyne CCR3 34 49 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)c1 ZINC000880545151 ED On-Demand Mild PDGFRB 56 43 COc1cncc(NC(=O)NC2CCN([C@H]3CCOC3)CC2)c1 ZINC000880545152 DD On-Demand Anodyne CXCR3 17 40 COc1cncc(NC(=O)NC2CCN([C@@H]3CCOC3)CC2)c1 ZINC000880545154 DD On-Demand Anodyne CXCR3 17 40 COc1ccc(NC(=O)[C@H](C)N2CCC3(CC2)COCCO3)cc1OC ZINC000880545157 FD On-Demand Anodyne ENPP1 67 32 COc1cncc(NC(=O)N[C@H](C)CN2CCC(C)CC2)c1 ZINC000880545181 DE On-Demand Anodyne CCR3 47 33 COc1cncc(NC(=O)N[C@@H](C)CN2CCC(C)CC2)c1 ZINC000880545182 DE On-Demand Anodyne CCR3 47 33 COc1cncc(NC(=O)N2CCC(Oc3ccc(Cl)cn3)CC2)c1 ZINC000880545192 FG On-Demand Anodyne EPHX2 21 43 COc1cncc(NC(=O)N2CCC(Oc3ccc(Cl)cn3)CC2)c1 ZINC000880545192 FG On-Demand Anodyne SCD1 15 42 COc1cncc(NC(=O)N2CCC(CO)(CO)CC2)c1 ZINC000880545199 CC On-Demand Anodyne S1PR2 27 40 N#Cc1ccccc1-c1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880545200 EH On-Demand Mild SIGMAR1 29 43 COc1cncc(NC(=O)N[C@@H]2CCN(C(C)=O)C2)c1 ZINC000880545210 CC On-Demand Anodyne EPHX2 48 49 COc1cncc(NC(=O)N2CC[C@](OC)(C(F)(F)F)C2)c1 ZINC000880545218 DE On-Demand Anodyne EPHX2 33 41 COc1cncc(NC(=O)N2CC[C@@](OC)(C(F)(F)F)C2)c1 ZINC000880545219 DE On-Demand Anodyne EPHX2 33 41 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880545224 GF On-Demand Anodyne CPT1A 64 34 COc1cncc(NC(=O)N2CCOC[C@@H]2Cc2ccccc2)c1 ZINC000880545262 EF On-Demand Anodyne CHRNA7 23 44 COc1cncc(NC(=O)N2CCOC[C@H]2Cc2ccccc2)c1 ZINC000880545264 EF On-Demand Anodyne CHRNA7 23 44 NC(=O)c1ccc(NC(=O)CCN2CCC3(CC2)COCCO3)cc1Cl ZINC000880545284 GD On-Demand Anodyne STAT6 47 33 COc1cncc(NC(=O)NC[C@@H](O)[C@@H](C)c2ccccc2)c1 ZINC000880545297 DE On-Demand Anodyne SOAT1 43 40 COc1cncc(NC(=O)NC[C@H](O)[C@@H](C)c2ccccc2)c1 ZINC000880545298 DE On-Demand Anodyne SOAT1 43 40 COc1cncc(NC(=O)NC[C@@H](O)[C@H](C)c2ccccc2)c1 ZINC000880545299 DE On-Demand Anodyne SOAT1 43 40 COc1cncc(NC(=O)NC[C@H](O)[C@H](C)c2ccccc2)c1 ZINC000880545300 DE On-Demand Anodyne SOAT1 43 40 COc1cncc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)c1 ZINC000880545304 FE On-Demand Clean ROCK2 16 41 COc1cncc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)c1 ZINC000880545304 FE On-Demand Clean NAMPT 45 39 O=C(CN1CCC2(CC1)COCCO2)Nc1nc2c(s1)CCCC2 ZINC000880545311 FD On-Demand Anodyne SLC27A1 62 56 c1cc2c(cc1CN1CCC3(CC1)COCCO3)OCCO2 ZINC000880545312 DD On-Demand Anodyne SIGMAR1 18 46 Brc1ccccc1CCCN1CCC2(CC1)COCCO2 ZINC000880545324 FG On-Demand Anodyne SIGMAR1 22 46 COc1ccc(N2CC[C@H](NC(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880545346 EE On-Demand Clean HRH4 41 37 COc1ccc(N2CC[C@H](NC(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880545346 EE On-Demand Clean EPHX2 44 38 COc1ccc(N2CC[C@H](NC(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880545346 EE On-Demand Clean MCHR1 18 44 O=C(CN1CCC2(CC1)COCCO2)NOCc1ccccc1 ZINC000880545350 DD On-Demand Anodyne SLC12A5 64 39 COc1cncc(NC(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880545357 EE On-Demand Anodyne CCR3 30 40 COc1cncc(NC(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880545357 EE On-Demand Anodyne CACNA1I 51 32 COc1cncc(NC(=O)N(C)c2ccc(OC)c(OC)c2)c1 ZINC000880545363 DF On-Demand Anodyne ENPP1 61 33 COc1cncc(NC(=O)N2CCN(Cc3n[nH]c(C)n3)CC2)c1 ZINC000880545364 EC On-Demand Anodyne FAAH 15 48 COc1cncc(NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)c1 ZINC000880545379 CD On-Demand Anodyne PLM1_PLAFA 41 39 COc1cncc(NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)c1 ZINC000880545379 CD On-Demand Anodyne PLM2_PLAFA 83 39 COCC1(NC(=O)Nc2cncc(OC)c2)CCCC1 ZINC000880545400 CE On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)N2CCN(C(=O)N(C)C)CC2)c1 ZINC000880545415 DC On-Demand Anodyne PDGFRB 43 39 COc1cncc(NC(=O)N2CCN(CCCOC(C)(C)C)CC2)c1 ZINC000880545420 FE On-Demand Anodyne PDGFRB 51 40 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne CACNA1H 58 37 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne GRIN2B 22 43 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne CCR3 19 45 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne CCR5 43 34 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne MCHR1 26 44 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880545424 EH On-Demand Anodyne SCD1 21 42 COc1cncc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880545431 EF On-Demand Anodyne CCR3 31 46 COc1cncc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880545431 EF On-Demand Anodyne EPHX2 45 38 COc1cncc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880545431 EF On-Demand Anodyne SCD1 22 42 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne ACHE 22 42 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne HRH2 37 47 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne SIGMAR1 45 39 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne CCR3 29 45 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne NPFFR2 37 47 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne UTS2R 17 42 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne FAAH 20 43 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne MCHR1 23 42 COc1cncc(NC(=O)NCCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880545437 GF On-Demand Anodyne NPFFR1 49 47 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)cn1 ZINC000880545449 ED On-Demand Anodyne F10 40 43 COc1cncc(NC(=O)N[C@@]2(c3ccccc3)C[C@@H](O)C2)c1 ZINC000880545450 DE On-Demand Anodyne EPHX2 20 44 COc1cncc(NC(=O)N(C)CCCCN2CCCCC2)c1 ZINC000880545453 DF On-Demand Anodyne CHRNA7 21 42 COc1cncc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)c1 ZINC000880545469 EG On-Demand Anodyne PDGFRB 45 41 COc1cncc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)c1 ZINC000880545469 EG On-Demand Anodyne FAAH 15 45 COc1cncc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)c1 ZINC000880545470 EG On-Demand Anodyne PDGFRB 45 41 COc1cncc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)c1 ZINC000880545470 EG On-Demand Anodyne FAAH 15 45 COc1cncc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)c1 ZINC000880545495 ED On-Demand Anodyne L3MBTL3 55 39 COc1cncc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)c1 ZINC000880545496 DG On-Demand Anodyne NPY5R 37 45 COc1cncc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)c1 ZINC000880545497 DG On-Demand Anodyne NPY5R 37 45 O=C(CN1CCC2(CC1)COCCO2)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880545500 FD On-Demand Anodyne DRD4 22 40 Cc1c(NC(=O)[C@H](C)N2CCC3(CC2)COCCO3)cccc1[N+](=O)[O-] ZINC000880545501 FE On-Demand Bother COLA 78 38 Cc1c(NC(=O)[C@@H](C)N2CCC3(CC2)COCCO3)cccc1[N+](=O)[O-] ZINC000880545502 FE On-Demand Bother COLA 78 38 COc1cncc(NC(=O)N2Cc3cccc(OC)c3C2)c1 ZINC000880545517 CF On-Demand Anodyne SSTR1 51 35 COc1cncc(NC(=O)N(C)CCNC(C)=O)c1 ZINC000880545520 CC On-Demand Anodyne MTNR1A 53 40 COc1cncc(NC(=O)N(C)CCNC(C)=O)c1 ZINC000880545520 CC On-Demand Anodyne MTNR1B 52 40 OCc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880545531 CD On-Demand Anodyne SIGMAR1 27 40 O=[N+]([O-])c1ccc([C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880545540 DD On-Demand Bother KCNJ1 19 42 O=[N+]([O-])c1ccc([C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880545541 DD On-Demand Bother KCNJ1 19 42 FC(F)(F)Oc1cccc(CCN2CCC3(CC2)COCCO3)c1 ZINC000880545546 EG On-Demand Anodyne SIGMAR1 17 50 COc1cncc(NC(=O)NC[C@H]2CCN(C(C)(C)C)C2)c1 ZINC000880545559 DE On-Demand Anodyne CACNA1I 48 34 COc1cncc(NC(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c1 ZINC000880545562 DE On-Demand Anodyne CACNA1I 48 34 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880545570 FD On-Demand Anodyne HRH2 19 40 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880545570 FD On-Demand Anodyne CCR3 78 41 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880545570 FD On-Demand Anodyne CXCR3 30 40 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880545570 FD On-Demand Anodyne MCHR1 41 46 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880545570 FD On-Demand Anodyne NAMPT 42 37 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880545573 FD On-Demand Anodyne HRH2 19 40 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880545573 FD On-Demand Anodyne CCR3 78 41 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880545573 FD On-Demand Anodyne CXCR3 30 40 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880545573 FD On-Demand Anodyne MCHR1 41 46 COc1cncc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880545573 FD On-Demand Anodyne NAMPT 42 37 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cncc(OC)c1 ZINC000880545582 DD On-Demand Anodyne SLC6A4 16 45 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cncc(OC)c1 ZINC000880545583 DD On-Demand Anodyne SLC6A4 16 45 COc1cncc(NC(=O)N2CCC[C@H](N3CCOCC3)CC2)c1 ZINC000880545610 ED On-Demand Anodyne L3MBTL3 56 36 COc1cncc(NC(=O)N2CCC[C@@H](N3CCOCC3)CC2)c1 ZINC000880545613 ED On-Demand Anodyne L3MBTL3 56 36 CCOC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880545618 DD On-Demand Mild P2RY12 61 49 CCOC(=O)N1CCN(C(=O)Nc2ccnc(C#N)c2)CC1 ZINC000880545618 DD On-Demand Mild PDGFRB 51 40 COc1cncc(NC(=O)N(C)[C@H](C)CCO)c1 ZINC000880545646 CD On-Demand Anodyne NPY5R 33 42 COc1cncc(NC(=O)N(C)[C@@H](C)CCO)c1 ZINC000880545647 CD On-Demand Anodyne NPY5R 33 42 c1ccc(Cn2cncc2CN2CCC3(CC2)COCCO3)cc1 ZINC000880545669 EE On-Demand Anodyne SIGMAR1 27 40 COc1cncc(NC(=O)NC2CCN(C(=O)C(C)(C)C)CC2)c1 ZINC000880545689 EE On-Demand Anodyne EPHX2 55 47 COc1cncc(NC(=O)NC2CCN(C(=O)C(C)(C)C)CC2)c1 ZINC000880545689 EE On-Demand Anodyne CXCR3 17 50 N#CC(CCN1CCC2(CC1)COCCO2)(c1ccccc1)c1ccccc1 ZINC000880545698 GH On-Demand Mild CCR1 25 57 c1cc(CCCN2CCC3(CC2)COCCO3)ccn1 ZINC000880545703 CD On-Demand Anodyne SIGMAR1 25 41 COc1cncc(NC(=O)N2C[C@H]3C(=O)N(Cc4ccccc4)C(=O)[C@H]3C2)c1 ZINC000880545705 GD On-Demand Anodyne TSHR 47 31 COc1cncc(NC(=O)N2C[C@H]3C(=O)N(Cc4ccccc4)C(=O)[C@H]3C2)c1 ZINC000880545705 GD On-Demand Anodyne FAAH 17 44 O=C(c1ccccc1)N1CC[C@@H](CN2CCC3(CC2)COCCO3)C1 ZINC000880545728 EE On-Demand Anodyne L3MBTL3 48 34 O=C(c1ccccc1)N1CC[C@H](CN2CCC3(CC2)COCCO3)C1 ZINC000880545729 EE On-Demand Anodyne L3MBTL3 48 34 COc1cncc(NC(=O)N2CCN(C(=O)CC(C)(C)C)CC2)c1 ZINC000880545804 EE On-Demand Anodyne PDGFRB 41 37 COc1cncc(NC(=O)N2CC[C@@]3(CCCOC3)C2)c1 ZINC000880545816 CE On-Demand Anodyne EPHX2 32 41 COc1cncc(NC(=O)N2CC[C@]3(CCCOC3)C2)c1 ZINC000880545818 CE On-Demand Anodyne EPHX2 32 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne HTR1A 31 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne DRD2 42 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne DRD4 68 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne ACHE 40 43 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne HRH2 26 40 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne HTR1B 20 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne DRD3 40 39 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne PDGFRB 60 43 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne SIGMAR1 63 49 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne MMP13 16 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne CCR3 32 45 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne NPFFR2 26 43 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne FAAH 51 69 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne MCHR1 34 46 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne CCR8 32 40 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne NPFFR1 36 43 COc1cncc(NC(=O)N2CCN(Cc3ccccc3)CC2)c1 ZINC000880545824 EE On-Demand Anodyne NOD2 40 39 COc1cncc(NC(=O)N[C@H](C(=O)N2CCCC2)C(C)C)c1 ZINC000880545840 DD On-Demand Anodyne CCR1 31 42 c1cc2c(cc1CN1CCC3(CC1)COCCO3)COC2 ZINC000880545890 CE On-Demand Anodyne MCHR2 53 32 O=[N+]([O-])c1ccc(S(=O)(=O)CCN2CCC3(CC2)COCCO3)cc1 ZINC000880545902 FD On-Demand Bother KCNJ1 27 42 COc1cncc(NC(=O)N(C)CCN2CCCCC2)c1 ZINC000880545907 CE On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N(C)CCN2CCCCC2)c1 ZINC000880545907 CE On-Demand Anodyne ROCK2 22 41 COc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880545911 DD On-Demand Anodyne DRD4 40 30 COc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880545911 DD On-Demand Anodyne LTA4H 32 46 COc1cccc(OCCN2CCC3(CC2)COCCO3)c1 ZINC000880545911 DD On-Demand Anodyne HRH3 20 54 CCOc1cc(CN2CCC3(CC2)COCCO3)ccc1[N+](=O)[O-] ZINC000880545912 EE On-Demand Bother SSTR5 57 40 COc1cncc(NC(=O)N2CCN(Cc3nc[nH]n3)CC2)c1 ZINC000880545923 DC On-Demand Anodyne PDGFRB 44 35 COc1cncc(NC(=O)N2CCN(Cc3nc[nH]n3)CC2)c1 ZINC000880545923 DC On-Demand Anodyne FAAH 16 47 O=C(CCN1CCC2(CC1)COCCO2)c1ccc(F)cc1 ZINC000880545925 DE On-Demand Anodyne DRD2 31 50 O=C(CCN1CCC2(CC1)COCCO2)c1ccc(F)cc1 ZINC000880545925 DE On-Demand Anodyne HTR2A 20 50 O=C(CCN1CCC2(CC1)COCCO2)c1ccc(F)cc1 ZINC000880545925 DE On-Demand Anodyne ERG2 23 50 O=C(CCN1CCC2(CC1)COCCO2)c1ccc(F)cc1 ZINC000880545925 DE On-Demand Anodyne CYP2J2 43 31 O=C(OCc1ccccc1)N1CCC(CN2CCC3(CC2)COCCO3)CC1 ZINC000880545931 GF On-Demand Anodyne GRIN2B 42 49 O=C(OCc1ccccc1)N1CCC(CN2CCC3(CC2)COCCO3)CC1 ZINC000880545931 GF On-Demand Anodyne TACR2 23 43 O=C(OCc1ccccc1)N1CCC(CN2CCC3(CC2)COCCO3)CC1 ZINC000880545931 GF On-Demand Anodyne TGM2 25 41 O=C(OCc1ccccc1)N1CCC(CN2CCC3(CC2)COCCO3)CC1 ZINC000880545931 GF On-Demand Anodyne F13A1 34 41 O=C(OCc1ccccc1)N1CCC(CN2CCC3(CC2)COCCO3)CC1 ZINC000880545931 GF On-Demand Anodyne SLC12A5 64 38 COc1cncc(NC(=O)N2CC[C@@](C)(c3cccc(F)c3)C2)c1 ZINC000880545933 EG On-Demand Anodyne CACNA1H 50 39 COc1cncc(NC(=O)N2CC[C@@](C)(c3cccc(F)c3)C2)c1 ZINC000880545933 EG On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CC[C@@](C)(c3cccc(F)c3)C2)c1 ZINC000880545933 EG On-Demand Anodyne EPHX2 35 41 COc1cncc(NC(=O)N2CC[C@](C)(c3cccc(F)c3)C2)c1 ZINC000880545934 EG On-Demand Anodyne CACNA1H 50 39 COc1cncc(NC(=O)N2CC[C@](C)(c3cccc(F)c3)C2)c1 ZINC000880545934 EG On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CC[C@](C)(c3cccc(F)c3)C2)c1 ZINC000880545934 EG On-Demand Anodyne EPHX2 35 41 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne GRIN2B 39 41 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne MMP13 29 44 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne CCR3 26 47 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne EPHX2 36 46 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne MMP7 18 44 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne MMP1 15 44 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne CACNA1G 42 37 COc1cncc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545940 FE On-Demand Anodyne NAMPT 52 36 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne GRIN2B 39 41 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne MMP13 29 44 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne CCR3 26 47 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne EPHX2 36 46 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne MMP7 18 44 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne MMP1 15 44 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne CACNA1G 42 37 COc1cncc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c1 ZINC000880545941 FE On-Demand Anodyne NAMPT 52 36 c1ccc(Cn2cc(CN3CCC4(CC3)COCCO4)nn2)cc1 ZINC000880545942 ED On-Demand Anodyne SIGMAR1 42 43 COc1cncc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880545946 CC On-Demand Anodyne LUXR 72 40 COc1cncc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880545946 CC On-Demand Anodyne TRAR 88 39 COc1cncc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880545946 CC On-Demand Anodyne LASR 61 38 COc1ccc(N2CC[C@H](CNC(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880545954 FF On-Demand Clean CCR3 35 42 COc1cncc(NC(=O)N2CCC3(CC2)CC3(F)F)c1 ZINC000880545968 CF On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCO[C@@]3(CCS(=O)(=O)C3)C2)c1 ZINC000880545979 EC On-Demand Anodyne EPHX2 19 42 COC(=O)[C@@H]1CN(C(=O)Nc2cncc(OC)c2)C[C@H]1c1ccccc1 ZINC000880545980 FF On-Demand Anodyne SLC6A3 15 45 COc1cncc(NC(=O)N2CCO[C@]3(CCS(=O)(=O)C3)C2)c1 ZINC000880545981 EC On-Demand Anodyne EPHX2 19 42 COc1cncc(NC(=O)N2CC[C@@H](O)[C@H]2c2ccc(Cl)cc2)c1 ZINC000880545982 EG On-Demand Anodyne CCR1 26 40 COc1cncc(NC(=O)N2CC[C@@H](O)[C@H]2c2ccc(Cl)cc2)c1 ZINC000880545982 EG On-Demand Anodyne SCN10A 22 40 COc1cncc(NC(=O)NCCN2CCCC2=O)c1 ZINC000880545984 CC On-Demand Anodyne DRD4 41 31 COc1cncc(NC(=O)N2CCO[C@@](C)(c3ccccc3)C2)c1 ZINC000880545993 EF On-Demand Anodyne EPHX2 30 44 COc1cncc(NC(=O)N2CCO[C@](C)(c3ccccc3)C2)c1 ZINC000880545994 EF On-Demand Anodyne EPHX2 30 44 COc1cncc(NC(=O)N2CCC3(CC2)CN(C(=O)OC(C)(C)C)C3)c1 ZINC000880546002 GF On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)N2CCC3(CC2)CN(C(=O)OC(C)(C)C)C3)c1 ZINC000880546002 GF On-Demand Anodyne GPR119 16 44 COc1cncc(NC(=O)NC[C@@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880546003 FE On-Demand Anodyne CCR3 41 39 COc1cncc(NC(=O)NC[C@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880546004 FE On-Demand Anodyne CCR3 41 39 O=C(c1cc2ccccc2cc1F)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880546010 EE On-Demand Anodyne PARP1 50 41 O=C(CCN1CCC2(CC1)COCCO2)NCC(=O)c1ccccc1 ZINC000880546021 ED On-Demand Anodyne CYP2J2 43 30 O[C@H](COc1ccccc1C(F)(F)F)CN1CCC2(CC1)COCCO2 ZINC000880546024 GE On-Demand Anodyne CCR1 50 47 O[C@H](COc1ccccc1C(F)(F)F)CN1CCC2(CC1)COCCO2 ZINC000880546024 GE On-Demand Anodyne ABCB1 69 49 O[C@@H](COc1ccccc1C(F)(F)F)CN1CCC2(CC1)COCCO2 ZINC000880546026 GE On-Demand Anodyne CCR1 50 47 O[C@@H](COc1ccccc1C(F)(F)F)CN1CCC2(CC1)COCCO2 ZINC000880546026 GE On-Demand Anodyne ABCB1 69 49 c1ccc2c(c1)CC[C@H](CN1CCC3(CC1)COCCO3)C2 ZINC000880546047 DF On-Demand Anodyne SIGMAR1 19 54 c1ccc2c(c1)CC[C@@H](CN1CCC3(CC1)COCCO3)C2 ZINC000880546049 DF On-Demand Anodyne SIGMAR1 19 54 O=C(CCN1CCC2(CC1)COCCO2)OCc1ccccc1 ZINC000880546061 DE On-Demand Anodyne NPR 56 33 O=C(CCN1CCC2(CC1)COCCO2)OCc1ccccc1 ZINC000880546061 DE On-Demand Anodyne SLC12A5 74 38 O=C(CCN1CCC2(CC1)COCCO2)N1CCc2ccccc2C1 ZINC000880546064 ED On-Demand Anodyne HTR7 15 46 COc1cncc(NC(=O)N2CCN(C)C[C@@H]2Cc2ccccc2)c1 ZINC000880546076 EE On-Demand Anodyne CCR3 30 45 COc1cncc(NC(=O)N2CCN(C)C[C@@H]2Cc2ccccc2)c1 ZINC000880546076 EE On-Demand Anodyne CHRNA7 25 47 COc1cncc(NC(=O)N2CCN(C)C[C@H]2Cc2ccccc2)c1 ZINC000880546078 EE On-Demand Anodyne CCR3 30 45 COc1cncc(NC(=O)N2CCN(C)C[C@H]2Cc2ccccc2)c1 ZINC000880546078 EE On-Demand Anodyne CHRNA7 25 47 O=C(Cc1ccccc1)OCCN1CCC2(CC1)COCCO2 ZINC000880546092 DD On-Demand Anodyne SIGMAR1 25 45 O=C(Cc1ccccc1)OCCN1CCC2(CC1)COCCO2 ZINC000880546092 DD On-Demand Anodyne SLC12A5 54 33 Fc1ccc(CN2CCC3(CC2)COCCO3)cc1Cl ZINC000880546108 CF On-Demand Anodyne SIGMAR1 26 40 COc1cncc(NC(=O)NCc2cccc(C)c2OC)c1 ZINC000880546136 DF On-Demand Anodyne ROCK2 25 50 COc1cncc(NC(=O)NCc2cccc(C)c2OC)c1 ZINC000880546136 DF On-Demand Anodyne NAMPT 19 41 COc1cncc(NC(=O)N[C@@H](CO)c2cccc(OC)c2)c1 ZINC000880546194 DD On-Demand Anodyne ROCK1 28 55 COc1cncc(NC(=O)N[C@@H](CO)c2cccc(OC)c2)c1 ZINC000880546194 DD On-Demand Anodyne MTNR1A 28 41 COc1cncc(NC(=O)N[C@@H](CO)c2cccc(OC)c2)c1 ZINC000880546194 DD On-Demand Anodyne MTNR1B 29 41 COc1cncc(NC(=O)N[C@@H](CO)c2cccc(OC)c2)c1 ZINC000880546194 DD On-Demand Anodyne ROCK2 32 55 COc1cncc(NC(=O)N[C@H](CO)c2cccc(OC)c2)c1 ZINC000880546196 DD On-Demand Anodyne ROCK1 28 55 COc1cncc(NC(=O)N[C@H](CO)c2cccc(OC)c2)c1 ZINC000880546196 DD On-Demand Anodyne MTNR1A 28 41 COc1cncc(NC(=O)N[C@H](CO)c2cccc(OC)c2)c1 ZINC000880546196 DD On-Demand Anodyne MTNR1B 29 41 COc1cncc(NC(=O)N[C@H](CO)c2cccc(OC)c2)c1 ZINC000880546196 DD On-Demand Anodyne ROCK2 32 55 COc1cncc(NC(=O)N(C)[C@H](CO)Cc2ccccc2)c1 ZINC000880546198 DE On-Demand Anodyne NPY5R 39 55 COc1cncc(NC(=O)N(C)[C@@H](CO)Cc2ccccc2)c1 ZINC000880546200 DE On-Demand Anodyne NPY5R 39 55 c1cc(OC[C@@H]2CCCO2)ccc1CN1CCC2(CC1)COCCO2 ZINC000880546212 EF On-Demand Anodyne HRH3 15 51 c1cc(OC[C@H]2CCCO2)ccc1CN1CCC2(CC1)COCCO2 ZINC000880546213 EF On-Demand Anodyne HRH3 15 51 CN(C)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)c1 ZINC000880546220 HG On-Demand Mild GRM4 40 39 CN(C)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)c1 ZINC000880546220 HG On-Demand Mild KCNK3 46 34 COc1cncc(NC(=O)N(C)Cc2ccc(OC)nc2)c1 ZINC000880546223 DE On-Demand Anodyne ROCK2 21 45 COc1cncc(NC(=O)N2CCN(c3nncn3C)CC2)c1 ZINC000880546235 DC On-Demand Anodyne PDGFRB 49 40 COc1cncc(NC(=O)N2CCN(c3c(F)cccc3F)CC2)c1 ZINC000880546236 EF On-Demand Anodyne DRD4 41 32 COc1cncc(NC(=O)N2CCN(c3c(F)cccc3F)CC2)c1 ZINC000880546236 EF On-Demand Anodyne PDGFRB 55 42 COc1cncc(NC(=O)N2CCN(c3c(F)cccc3F)CC2)c1 ZINC000880546236 EF On-Demand Anodyne FAAH 26 46 Cc1ccc(C(=O)CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546257 DE On-Demand Anodyne CYP2J2 48 42 COc1cncc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)c1 ZINC000880546281 FF On-Demand Anodyne TRPM8 30 44 COc1cncc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)c1 ZINC000880546286 FF On-Demand Anodyne TRPM8 30 44 COc1cncc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)c1 ZINC000880546290 FF On-Demand Anodyne TRPM8 30 44 COc1cncc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)c1 ZINC000880546294 FF On-Demand Anodyne TRPM8 30 44 FCc1ccc(CN2CCC3(CC2)COCCO3)cc1 ZINC000880546317 CF On-Demand Anodyne SIGMAR1 28 40 COc1cncc(NC(=O)N(C)Cc2cnc[nH]2)c1 ZINC000880546328 CD On-Demand Anodyne ROCK2 15 44 COc1cncc(NC(=O)N(C)Cc2cnc[nH]2)c1 ZINC000880546328 CD On-Demand Anodyne TAAR1 22 41 COc1cncc(NC(=O)N[C@@H]2CCO[C@H]2c2ccnn2CC2CC2)c1 ZINC000880546329 FE On-Demand Anodyne CCR3 19 40 C(#Cc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880546334 CD On-Demand Mild GRIN2C 16 40 COc1cncc(NC(=O)N[C@@H]2CCO[C@@H](c3cccnc3)C2)c1 ZINC000880546341 EF On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)NC2CCN(OC)CC2)c1 ZINC000880546349 CD On-Demand Anodyne EPHX2 49 40 COc1cncc(NC(=O)NC2CCN(OC)CC2)c1 ZINC000880546349 CD On-Demand Anodyne CXCR3 17 43 COC(=O)/C=C\c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880546368 FE On-Demand Anodyne MMP13 16 41 COC(=O)/C=C\c1ccc(OCCN2CCC3(CC2)COCCO3)cc1 ZINC000880546368 FE On-Demand Anodyne PSMB1 40 33 COc1cncc(NC(=O)N2CC[C@@H](c3cccnc3)C2)c1 ZINC000880546385 CF On-Demand Anodyne CHRNA7 35 46 COc1cncc(NC(=O)N2CC[C@@H](c3cccnc3)C2)c1 ZINC000880546385 CF On-Demand Anodyne EPHX2 16 41 COc1cncc(NC(=O)N2CC[C@H](c3cccnc3)C2)c1 ZINC000880546386 CF On-Demand Anodyne CHRNA7 35 46 COc1cncc(NC(=O)N2CC[C@H](c3cccnc3)C2)c1 ZINC000880546386 CF On-Demand Anodyne EPHX2 16 41 COCC[C@@H](c1ccccc1)N1CCC2(CC1)COCCO2 ZINC000880546403 DF On-Demand Anodyne OPRL1 15 50 COCC[C@H](c1ccccc1)N1CCC2(CC1)COCCO2 ZINC000880546404 DF On-Demand Anodyne OPRL1 15 50 COc1cncc(NC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880546405 GG On-Demand Anodyne SIRT3 26 42 COc1cncc(NC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880546405 GG On-Demand Anodyne SIRT2 25 42 COc1cncc(NC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880546405 GG On-Demand Anodyne SIRT1 24 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880546423 JI On-Demand Mild EPHX2 20 40 COc1cncc(NC(=O)N2CCc3c(cccc3NC(C)=O)C2)c1 ZINC000880546435 EF On-Demand Anodyne P2RY14 46 33 Fc1cccc(CCCN2CCC3(CC2)COCCO3)c1 ZINC000880546455 CF On-Demand Anodyne SIGMAR1 36 52 COc1cncc(NC(=O)N2CCC(c3ccc4cccnc4n3)CC2)c1 ZINC000880546462 FG On-Demand Anodyne SMO 19 46 COc1cncc(NC(=O)NCCc2cnccc2C)c1 ZINC000880546465 CE On-Demand Anodyne RAF1 18 41 COc1cncc(NC(=O)NCCc2cnccc2C)c1 ZINC000880546465 CE On-Demand Anodyne MTNR1A 41 38 O=[N+]([O-])c1ccccc1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880546469 FD On-Demand Bother CCR1 50 47 O=[N+]([O-])c1ccccc1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880546469 FD On-Demand Bother ABCB1 67 47 O=[N+]([O-])c1ccccc1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880546470 FD On-Demand Bother CCR1 50 47 O=[N+]([O-])c1ccccc1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880546470 FD On-Demand Bother ABCB1 67 47 COc1cncc(NC(=O)N2CCO[C@@]3(CCSC3)C2)c1 ZINC000880546498 DD On-Demand Anodyne EPHX2 18 42 COc1cncc(NC(=O)N2CCO[C@]3(CCSC3)C2)c1 ZINC000880546499 DD On-Demand Anodyne EPHX2 18 42 Fc1cc(OCCN2CCC3(CC2)COCCO3)ccc1Cl ZINC000880546503 EF On-Demand Anodyne LTA4H 28 40 COc1cncc(NC(=O)Nc2ccc(COCCO)cc2)c1 ZINC000880546539 DE On-Demand Anodyne RAF1 19 43 COc1cncc(NC(=O)NCCCc2ncn(C)n2)c1 ZINC000880546541 CC On-Demand Anodyne QPCT 37 44 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3)C2)c1 ZINC000880546555 DF On-Demand Anodyne CCR3 31 44 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3)C2)c1 ZINC000880546555 DF On-Demand Anodyne CHRNA7 17 40 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3)C2)c1 ZINC000880546555 DF On-Demand Anodyne PDE3B 41 39 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3)C2)c1 ZINC000880546555 DF On-Demand Anodyne EPHX2 35 48 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3)C2)c1 ZINC000880546555 DF On-Demand Anodyne SCD1 22 52 O=C(CCN1CCC2(CC1)COCCO2)Nc1cccnc1 ZINC000880546566 DD On-Demand Anodyne CHRNA7 20 49 COc1cncc(NC(=O)N2CCN(Cc3cnn(C(C)(C)C)c3)CC2)c1 ZINC000880546584 FE On-Demand Anodyne PDGFRB 42 35 COc1cncc(NC(=O)N2CCN(Cc3cnn(C(C)(C)C)c3)CC2)c1 ZINC000880546584 FE On-Demand Anodyne FAAH 20 48 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne TRPV1 20 42 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne SCN2A 20 49 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne ROCK2 21 42 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne SCN10A 40 49 COc1cncc(NC(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880546604 EE On-Demand Anodyne NAMPT 48 42 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA2 37 44 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA1 39 44 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA7 22 43 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA4 22 40 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA12 25 44 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA9 32 43 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CAH_METTE 18 40 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne NCE103 19 40 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne CA15 15 40 NS(=O)(=O)c1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880546611 EC On-Demand Anodyne A6YCJ1_9METZ 21 40 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild DRD4 32 49 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild ACHE 15 42 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild HRH2 38 41 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild CHRM3 18 46 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild SIGMAR1 26 51 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild SSTR5 65 41 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild CCR3 69 51 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild CHRNA7 15 43 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild MLNR 20 40 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild FAAH 19 40 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild EPHX2 37 41 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild PDK1 48 37 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild CXCR3 29 48 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild MCHR1 72 53 COc1cncc(NC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880546622 FF On-Demand Mild CCR8 21 47 O=C(CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880546623 CE On-Demand Anodyne SIGMAR1 16 41 O=C(CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880546623 CE On-Demand Anodyne CYP2J2 51 36 COc1cncc(NC(=O)N2CCN(c3ccsc3C#N)CC2)c1 ZINC000880546636 EE On-Demand Mild PDGFRB 49 41 COc1cncc(NC(=O)NCCCC2CC2)c1 ZINC000880546692 BE On-Demand Anodyne CCR3 41 45 c1ccc(Cn2cc(CN3CCC4(CC3)COCCO4)cn2)cc1 ZINC000880546743 EE On-Demand Anodyne SIGMAR1 48 44 COc1cncc(NC(=O)NCc2c(OC)cccc2OC)c1 ZINC000880546761 DE On-Demand Anodyne PDGFRB 27 44 COc1cncc(NC(=O)NCc2c(OC)cccc2OC)c1 ZINC000880546761 DE On-Demand Anodyne RAF1 18 43 COc1cncc(NC(=O)NCc2c(OC)cccc2OC)c1 ZINC000880546761 DE On-Demand Anodyne MTNR1B 38 43 COc1cncc(NC(=O)NCc2c(OC)cccc2OC)c1 ZINC000880546761 DE On-Demand Anodyne ROCK2 39 58 COc1cncc(NC(=O)NCc2c(OC)cccc2OC)c1 ZINC000880546761 DE On-Demand Anodyne FLT4 23 44 c1csc(-c2ccc(CN3CCC4(CC3)COCCO4)cc2)c1 ZINC000880546822 EH On-Demand Anodyne SIGMAR1 26 44 c1ccc(COCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880546827 DE On-Demand Anodyne SIGMAR1 38 40 c1ccc(CCCCN2CCC3(CC2)COCCO3)cc1 ZINC000880546841 CF On-Demand Anodyne SIGMAR1 71 55 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3F)CC2)c1 ZINC000880546851 EH On-Demand Anodyne RBP4 50 43 COc1cncc(NC(=O)N2CCC(c3cccc(F)c3F)CC2)c1 ZINC000880546851 EH On-Demand Anodyne CALCRL 42 41 CN(C)S(=O)(=O)c1cc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)ccc1Br ZINC000880546862 JH On-Demand Mild KCNK3 82 39 CN(C)S(=O)(=O)c1cc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)ccc1Br ZINC000880546862 JH On-Demand Mild KCNK9 43 33 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880546879 ED On-Demand Anodyne EPHX2 32 41 COc1cncc(NC(=O)N2CCC3(CC2)C(F)(F)C3(F)F)c1 ZINC000880546914 EF On-Demand Anodyne S1PR2 27 41 Fc1cc(CN2CCC3(CC2)COCCO3)ccc1Cl ZINC000880546916 CF On-Demand Anodyne SIGMAR1 25 43 COc1cncc(NC(=O)NCCNC(=O)CCCc2ccccc2)c1 ZINC000880546935 FE On-Demand Anodyne HDAC8 18 41 COc1cncc(NC(=O)NCCNC(=O)CCCc2ccccc2)c1 ZINC000880546935 FE On-Demand Anodyne MTNR1A 50 42 COc1cncc(NC(=O)NCCNC(=O)CCCc2ccccc2)c1 ZINC000880546935 FE On-Demand Anodyne MTNR1B 47 42 COc1cncc(NC(=O)NCCNC(=O)CCCc2ccccc2)c1 ZINC000880546935 FE On-Demand Anodyne HDAC2 15 42 COc1cncc(NC(=O)NCCNC(=O)CCCc2ccccc2)c1 ZINC000880546935 FE On-Demand Anodyne FAAH 41 39 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C)COCC1CC1)C2 ZINC000880546937 DF On-Demand Anodyne NQO2 25 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C)COCC1CC1)C2 ZINC000880546937 DF On-Demand Anodyne MTNR1A 28 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C)COCC1CC1)C2 ZINC000880546938 DF On-Demand Anodyne NQO2 25 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C)COCC1CC1)C2 ZINC000880546938 DF On-Demand Anodyne MTNR1A 28 40 c1ccc(-c2nnc(CN3CCC4(CC3)COCCO4)s2)cc1 ZINC000880546954 EF On-Demand Anodyne SIGMAR1 16 40 CNC(=O)[C@@H](CNC(=O)Nc1cncc(OC)c1)Cc1ccc(F)cc1C ZINC000880546963 FE On-Demand Anodyne P2RX7 21 45 COc1cncc(NC(=O)N2CCOC3(CCN(C)CC3)C2)c1 ZINC000880546984 DD On-Demand Anodyne EPHX2 23 47 c1ccc(CN2CC[C@@H](N3CCC4(CC3)COCCO4)C2)cc1 ZINC000880547002 DE On-Demand Anodyne SIGMAR1 58 39 c1ccc(CN2CC[C@H](N3CCC4(CC3)COCCO4)C2)cc1 ZINC000880547003 DE On-Demand Anodyne SIGMAR1 58 39 O[C@@H](CCc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880547011 DD On-Demand Anodyne ABCB1 42 42 O[C@H](CCc1ccccc1)CN1CCC2(CC1)COCCO2 ZINC000880547012 DD On-Demand Anodyne ABCB1 42 42 COC(=O)c1ccc(CN2CCC3(CC2)COCCO3)cc1Cl ZINC000880547043 EF On-Demand Anodyne MCHR2 46 35 CC(C)(C(=O)N1CCC(CCO)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880547069 EH On-Demand Anodyne EPHX2 21 43 CC(C)(C(=O)N1CCC(CCO)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880547069 EH On-Demand Anodyne MCHR1 21 40 CC(C)(C(=O)N1CCC(CCO)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880547069 EH On-Demand Anodyne AKR1C3 15 40 CC(C)(C(=O)N1CCC(CCO)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880547069 EH On-Demand Anodyne LIPG 24 40 COc1cncc(NC(=O)NCc2cnccc2C(C)(C)C)c1 ZINC000880547094 DG On-Demand Anodyne RAF1 15 41 COc1cncc(NC(=O)NCc2cnccc2C(C)(C)C)c1 ZINC000880547094 DG On-Demand Anodyne ROCK2 21 46 COc1cncc(NC(=O)NCc2cnccc2C(C)(C)C)c1 ZINC000880547094 DG On-Demand Anodyne NAMPT 21 41 CCC1(c2ccccc2)CN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880547100 DG On-Demand Anodyne KCNA3 40 35 CCC1(c2ccccc2)CN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880547100 DG On-Demand Anodyne FAAH 16 45 CCC1(c2ccccc2)CN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880547100 DG On-Demand Anodyne EPHX2 19 45 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(Cl)c2)c1 ZINC000880547104 EG On-Demand Anodyne ROCK2 21 45 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(Cl)c2)c1 ZINC000880547104 EG On-Demand Anodyne PDE6A 45 34 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCN(C)CC2)c1 ZINC000880547106 FD On-Demand Anodyne HCN1 69 41 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCN(C)CC2)c1 ZINC000880547106 FD On-Demand Anodyne HCN4 48 34 COCC1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880547107 CE On-Demand Anodyne EPHX2 42 35 COCC(COC)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880547113 EC On-Demand Anodyne PDGFRB 46 37 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne HTR1A 54 55 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne DRD2 29 55 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne DRD4 29 48 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne HTR2A 33 55 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne DRD3 29 48 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne HTR7 57 43 c1ccc(N2CCN(CCCN3CCC4(CC3)COCCO4)CC2)cc1 ZINC000880547124 FE On-Demand Anodyne SIGMAR1 28 42 COc1cncc(NC(=O)N(C)c2ccc(OC)cc2OC)c1 ZINC000880547132 DF On-Demand Anodyne LUCI_LUCLA 16 41 COc1cncc(NC(=O)CCCCc2ccc(OC)c(OC)c2)n1 ZINC000880547140 EF On-Demand Anodyne INHA 58 42 COc1cncc(NC(=O)CCCCc2ccc(OC)c(OC)c2)n1 ZINC000880547140 EF On-Demand Anodyne ENPP1 70 35 O[C@@H](CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547145 CD On-Demand Anodyne OPRL1 17 48 O[C@H](CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547146 CD On-Demand Anodyne OPRL1 17 48 O=C(C(=O)N1CCC(CCO)CC1)c1c[nH]c2cc(F)ccc12 ZINC000880547209 DE On-Demand Anodyne GRIN2B 26 68 O=C(C(=O)N1CCC(CCO)CC1)c1c[nH]c2cc(F)ccc12 ZINC000880547209 DE On-Demand Anodyne MPO 46 34 O=C(C(=O)N1CCC(CCO)CC1)c1c[nH]c2cc(F)ccc12 ZINC000880547209 DE On-Demand Anodyne AKR1C3 15 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(CCO)CC3)cc2)N1 ZINC000880547216 DD On-Demand Anodyne AKR1C3 17 47 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(CCO)CC3)cc2)N1 ZINC000880547216 DD On-Demand Anodyne L3MBTL3 71 39 O=C1CC[C@H](c2ccc(C(=O)N3CCC(CCO)CC3)cc2)N1 ZINC000880547217 DD On-Demand Anodyne AKR1C3 17 47 O=C1CC[C@H](c2ccc(C(=O)N3CCC(CCO)CC3)cc2)N1 ZINC000880547217 DD On-Demand Anodyne L3MBTL3 71 39 COc1cncc(NC(=O)N[C@@H]2CC[C@@H](O)CC2)c1 ZINC000880547278 CD On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)N2CC[C@](C(N)=O)(c3ccccc3)C2)c1 ZINC000880547289 ED On-Demand Anodyne TACR2 19 44 COc1cncc(NC(=O)N2CC[C@@](C(N)=O)(c3ccccc3)C2)c1 ZINC000880547290 ED On-Demand Anodyne TACR2 19 44 COc1cncc(NC(=O)NCC(C)(C)c2cccnc2)c1 ZINC000880547305 DF On-Demand Anodyne NAMPT 34 40 COc1cncc(NC(=O)N(C)[C@H](C)Cc2cccc(F)c2)c1 ZINC000880547328 DG On-Demand Anodyne NPY5R 36 53 COc1cncc(NC(=O)N(C)[C@@H](C)Cc2cccc(F)c2)c1 ZINC000880547329 DG On-Demand Anodyne NPY5R 36 53 COc1cncc(NC(=O)NC2CCC(N(C)C)CC2)c1 ZINC000880547330 CE On-Demand Anodyne EPHX2 44 38 COc1cncc(NC(=O)N[C@H](C)CCCc2cccnc2)c1 ZINC000880547388 DG On-Demand Anodyne TBXAS1 29 44 COc1cncc(NC(=O)N[C@H](C)CCCc2cccnc2)c1 ZINC000880547388 DG On-Demand Anodyne PTAFR 44 59 COc1cncc(NC(=O)N[C@H](C)CCCc2cccnc2)c1 ZINC000880547388 DG On-Demand Anodyne CHRNA7 36 46 COc1cncc(NC(=O)N[C@H](C)CCCc2cccnc2)c1 ZINC000880547388 DG On-Demand Anodyne NAMPT 36 40 COc1cncc(NC(=O)N[C@@H](C)CCCc2cccnc2)c1 ZINC000880547389 DG On-Demand Anodyne TBXAS1 29 44 COc1cncc(NC(=O)N[C@@H](C)CCCc2cccnc2)c1 ZINC000880547389 DG On-Demand Anodyne PTAFR 44 59 COc1cncc(NC(=O)N[C@@H](C)CCCc2cccnc2)c1 ZINC000880547389 DG On-Demand Anodyne CHRNA7 36 46 COc1cncc(NC(=O)N[C@@H](C)CCCc2cccnc2)c1 ZINC000880547389 DG On-Demand Anodyne NAMPT 36 40 COC(=O)[C@@H]1CN(C(=O)Nc2cncc(OC)c2)C[C@@H]1c1ccccc1 ZINC000880547401 FF On-Demand Anodyne SLC6A3 15 45 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCOCC2)c1 ZINC000880547406 FD On-Demand Anodyne HCN1 61 39 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCOCC2)c1 ZINC000880547406 FD On-Demand Anodyne HCN4 50 35 COCCc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880547443 FD On-Demand Anodyne CCR1 44 39 COCCc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880547443 FD On-Demand Anodyne ABCB1 57 40 COCCc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880547444 FD On-Demand Anodyne CCR1 44 39 COCCc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880547444 FD On-Demand Anodyne ABCB1 57 40 COc1cncc(NC(=O)NCc2cc(F)c(N3CCOCC3)c(F)c2)c1 ZINC000880547464 GF On-Demand Clean NAMPT 28 43 COc1cncc(NC(=O)NCc2ccc(C)c(C)n2)c1 ZINC000880547475 CE On-Demand Anodyne ROCK2 16 40 COc1cncc(NC(=O)N2CCc3cccc(Cl)c3C2)c1 ZINC000880547478 DG On-Demand Anodyne HTR2C 15 42 COc1cncc(NC(=O)N2CCc3cccc(Cl)c3C2)c1 ZINC000880547478 DG On-Demand Anodyne P2RY14 50 41 O=C(CCCN1CCC2(CC1)COCCO2)c1ccc(Br)cc1 ZINC000880547493 GG On-Demand Anodyne DRD2 29 46 O=C(CCCN1CCC2(CC1)COCCO2)c1ccc(Br)cc1 ZINC000880547493 GG On-Demand Anodyne ERG2 21 46 O=C(CCCN1CCC2(CC1)COCCO2)c1ccc(Br)cc1 ZINC000880547493 GG On-Demand Anodyne CYP2J2 54 38 Cn1c(=O)c(CN2CCC3(CC2)COCCO3)cc2ccccc21 ZINC000880547498 ED On-Demand Anodyne NPSR1 32 44 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne DRD2 16 42 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne DRD4 30 42 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne ACHE 29 41 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne HRH2 38 46 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne DRD3 17 42 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne SIGMAR1 53 43 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne CCR3 41 44 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne NPFFR2 44 54 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne ROCK2 21 40 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne FAAH 26 46 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne MCHR1 30 42 COc1cncc(NC(=O)NCC2(O)CCN(Cc3ccccc3)CC2)c1 ZINC000880547509 FE On-Demand Anodyne NPFFR1 55 54 COc1cncc(NC(=O)N2CCC(c3ccncn3)CC2)c1 ZINC000880547510 DE On-Demand Anodyne PDGFRB 46 36 COc1cncc(NC(=O)NC2CCC(OC)CC2)c1 ZINC000880547538 CE On-Demand Anodyne EPHX2 57 42 Cc1cc(-c2nc(C)c(C(=O)N3CCC(CCO)CC3)s2)ccc1F ZINC000880547539 FH On-Demand Anodyne AKR1C3 16 40 CCCOc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880547543 DF On-Demand Anodyne HRH2 33 44 CCCOc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880547543 DF On-Demand Anodyne SIGMAR1 22 42 CC[C@@H](Nc1cccnc1Cl)C(=O)Nc1cncc(OC)n1 ZINC000880547555 DE On-Demand Anodyne G2YM83_BOTF4 56 32 CC[C@H](Nc1cccnc1Cl)C(=O)Nc1cncc(OC)n1 ZINC000880547556 DE On-Demand Anodyne G2YM83_BOTF4 56 32 O=C(c1ncsc1C1CC1)N1CCC(CCO)CC1 ZINC000880547559 CE On-Demand Anodyne AKR1C3 15 42 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne CTSL 45 37 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne BRS3 26 41 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne MTNR1A 48 37 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne MTNR1B 48 37 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne MMP3 41 41 COc1cncc(NC(=O)N[C@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880547562 ED On-Demand Anodyne ROCK2 19 42 COc1cccc(OC)c1OCCCCN1CCC2(CC1)COCCO2 ZINC000880547572 FF On-Demand Anodyne SIGMAR1 21 44 COc1cccc(OC)c1OCCCCN1CCC2(CC1)COCCO2 ZINC000880547572 FF On-Demand Anodyne EBP 30 41 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(CCO)CC1 ZINC000880547576 EG On-Demand Anodyne PDE4D 19 40 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(CCO)CC1 ZINC000880547576 EG On-Demand Anodyne CACNA1I 46 34 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(CCO)CC1 ZINC000880547576 EG On-Demand Anodyne AKR1C3 16 44 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(CCO)CC1 ZINC000880547576 EG On-Demand Anodyne L3MBTL3 56 36 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne DRD2 32 46 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne DRD4 15 46 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne HTR2A 15 46 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne ERG2 21 45 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne SIGMAR1 29 45 O=C(CCCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880547584 DF On-Demand Anodyne CYP2J2 62 44 COc1cncc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547610 FF On-Demand Anodyne ACACA 59 44 COc1cncc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547610 FF On-Demand Anodyne ACACB 35 42 COc1cncc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547610 FF On-Demand Anodyne NPY5R 23 42 COc1cncc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547610 FF On-Demand Anodyne EPHX2 36 40 COc1cncc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547610 FF On-Demand Anodyne TRPM8 28 43 COc1cncc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547611 FF On-Demand Anodyne ACACA 59 44 COc1cncc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547611 FF On-Demand Anodyne ACACB 35 42 COc1cncc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547611 FF On-Demand Anodyne NPY5R 23 42 COc1cncc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547611 FF On-Demand Anodyne EPHX2 36 40 COc1cncc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880547611 FF On-Demand Anodyne TRPM8 28 43 CC(C)(C(=O)N1CCC(CCO)CC1)c1ccc(F)cc1F ZINC000880547612 DF On-Demand Anodyne AKR1C3 16 40 COc1cncc(NC(=O)NC2(CO)C3CC4CC(C3)CC2C4)c1 ZINC000880547613 EE On-Demand Anodyne EPHX2 33 46 O=C(c1cccc2nsnc12)N1CCC(CCO)CC1 ZINC000880547620 CD On-Demand Anodyne AKR1C3 15 44 COc1cncc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)c1 ZINC000880547629 EE On-Demand Anodyne CHRNA7 46 43 COc1cncc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)c1 ZINC000880547629 EE On-Demand Anodyne NAMPT 49 38 O=C(c1cncc2[nH]ccc12)N1CCC(CCO)CC1 ZINC000880547638 CD On-Demand Anodyne AKR1C3 18 49 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC(CCO)CC2)N1Cc1ccccc1 ZINC000880547670 FD On-Demand Anodyne ACHE 35 42 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC(CCO)CC2)N1Cc1ccccc1 ZINC000880547670 FD On-Demand Anodyne PREP 52 39 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccsc2)c1 ZINC000880547674 EF On-Demand Anodyne ROCK1 15 51 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccsc2)c1 ZINC000880547674 EF On-Demand Anodyne ROCK2 26 51 COc1cncc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)c1 ZINC000880547690 ED On-Demand Anodyne PDGFRB 53 41 COc1cncc(NC(=O)N2CCC[C@@H](CC(F)(F)F)C2)c1 ZINC000880547691 DG On-Demand Anodyne CCR3 16 49 COc1cncc(NC(=O)N2CCC[C@H](CC(F)(F)F)C2)c1 ZINC000880547692 DG On-Demand Anodyne CCR3 16 49 O=C(c1cnc2cc[nH]c2c1)N1CCC(CCO)CC1 ZINC000880547693 CD On-Demand Anodyne GRIN2B 52 39 O=C(c1cnc2cc[nH]c2c1)N1CCC(CCO)CC1 ZINC000880547693 CD On-Demand Anodyne AKR1C3 20 54 O=C(c1cnc2cc[nH]c2c1)N1CCC(CCO)CC1 ZINC000880547693 CD On-Demand Anodyne L3MBTL3 56 36 COc1cncc(NC(=O)N(Cc2cccc(O)c2)[C@@H]2CC[C@@H](O)CC2)c1 ZINC000880547696 FG On-Demand Anodyne ROCK1 15 40 COc1cncc(NC(=O)N(Cc2cccc(O)c2)[C@@H]2CC[C@@H](O)CC2)c1 ZINC000880547696 FG On-Demand Anodyne ROCK2 25 54 COc1cncc(NC(=O)N(Cc2cccc(O)c2)[C@@H]2CC[C@@H](O)CC2)c1 ZINC000880547696 FG On-Demand Anodyne HSD17B2 16 43 COc1cncc(NC(=O)N(C)Cc2cccc(C)n2)c1 ZINC000880547700 CE On-Demand Anodyne ROCK2 23 44 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne CELA1 20 44 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne GRIN2B 43 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne PREP 84 54 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne LGMN 46 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne KLK5 22 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne SLC12A5 46 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(CCO)CC1 ZINC000880547701 GE On-Demand Anodyne Q9NAW4_PLAFA 35 41 CC(C)(C)OC(=O)N1CCCCN1C(=O)c1ccc2c(O)ncnc2c1 ZINC000880547705 FF On-Demand Anodyne HPGD 35 40 COc1cncc(NC(=O)N2CC[C@@](O)(Cc3ccc(F)cc3)C2)c1 ZINC000880547709 EE On-Demand Anodyne S1PR2 33 49 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne DRD4 30 54 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne ACHE 15 42 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne KCNH2 15 49 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne HTR4 19 40 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne CHRM3 17 44 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne LTA4H 25 42 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne SIGMAR1 29 54 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne SSTR5 76 44 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne CCR3 78 47 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne UTS2R 19 41 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne EPHX2 49 45 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne PDK1 53 41 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne CXCR3 39 48 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne MCHR1 70 58 COc1cncc(NC(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)CC2)c1 ZINC000880547710 GF On-Demand Anodyne CCR8 15 42 COc1cncc(NC(=O)Nc2cc(OC)c(C)c(OC)c2)c1 ZINC000880547712 DG On-Demand Anodyne PDGFRA 40 38 COc1cncc(NC(=O)N2CC[C@](O)(Cc3ccc(F)cc3)C2)c1 ZINC000880547713 EE On-Demand Anodyne S1PR2 33 49 COc1cncc(NC(=O)N2CCCN(C=O)CC2)c1 ZINC000880547720 CC On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)NCCc2ccc(C)cn2)c1 ZINC000880547721 CE On-Demand Anodyne PIK3CG 15 43 COc1cncc(NC(=O)c2ncsc2C2CC2)n1 ZINC000880547727 CE On-Demand Anodyne MAP1 53 36 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3[nH]2)c1 ZINC000880547744 FH On-Demand Anodyne PRCP 53 38 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3[nH]2)c1 ZINC000880547744 FH On-Demand Anodyne CPT1A 75 38 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3[nH]2)c1 ZINC000880547745 FH On-Demand Anodyne PRCP 53 38 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3[nH]2)c1 ZINC000880547745 FH On-Demand Anodyne CPT1A 75 38 Cc1cnc(Cl)c(C(=O)N2CCC(CCO)CC2)c1 ZINC000880547757 CE On-Demand Anodyne CACNA1I 41 31 Cc1cnc(Cl)c(C(=O)N2CCC(CCO)CC2)c1 ZINC000880547757 CE On-Demand Anodyne AKR1C3 17 42 COc1cncc(NC(=O)N2CCCc3ccccc3CC2)c1 ZINC000880547759 DG On-Demand Anodyne DRD5 25 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCC(CCO)CC1 ZINC000880547761 DG On-Demand Anodyne ETHR 42 33 O=C(CC[C@H]1CCc2ccccc21)N1CCC(CCO)CC1 ZINC000880547765 DG On-Demand Anodyne ETHR 42 33 COc1cncc(NC(=O)N2CCN(c3cccc(F)n3)CC2)c1 ZINC000880547783 ED On-Demand Anodyne PDGFRB 50 42 COc1cncc(NC(=O)N2CCN(c3cccc(F)n3)CC2)c1 ZINC000880547783 ED On-Demand Anodyne FAAH 21 46 COc1cncc(NC(=O)N2CCN(c3cccc(F)n3)CC2)c1 ZINC000880547783 ED On-Demand Anodyne DGAT1 18 42 O=C(c1csc(-c2ncc[nH]2)n1)N1CCC(CCO)CC1 ZINC000880547784 DD On-Demand Anodyne AKR1C3 17 44 COc1cncc(NC(=O)N2CCC[C@H](c3ccccc3)C2)c1 ZINC000880547788 DH On-Demand Anodyne EPHX2 24 40 COc1cncc(NC(=O)N2CCC[C@H](c3ccccc3)C2)c1 ZINC000880547788 DH On-Demand Anodyne MAP3K12 29 41 COc1cncc(NC(=O)N2CCC[C@@H](c3ccccc3)C2)c1 ZINC000880547789 DH On-Demand Anodyne EPHX2 24 40 COc1cncc(NC(=O)N2CCC[C@@H](c3ccccc3)C2)c1 ZINC000880547789 DH On-Demand Anodyne MAP3K12 29 41 COc1cncc(NC(=O)N2CC[C@@H]3CN(C(=O)OC(C)(C)C)C[C@@H]32)c1 ZINC000880547793 FF On-Demand Anodyne GPR119 24 40 O=C1CCc2cc(OC[C@@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547808 GD On-Demand Anodyne ACOX1 70 33 O=C1CCc2cc(OC[C@@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547808 GD On-Demand Anodyne CCR1 47 38 O=C1CCc2cc(OC[C@@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547808 GD On-Demand Anodyne ABCB1 41 36 O=C1CCc2cc(OC[C@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547809 GD On-Demand Anodyne ACOX1 70 33 O=C1CCc2cc(OC[C@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547809 GD On-Demand Anodyne CCR1 47 38 O=C1CCc2cc(OC[C@H](O)CN3CCC4(CC3)COCCO4)ccc2N1 ZINC000880547809 GD On-Demand Anodyne ABCB1 41 36 O=C(c1cc2ccccc2cc1F)N1CCC(CCO)CC1 ZINC000880547830 DG On-Demand Anodyne GRIN2B 49 39 O=C(c1cc2ccccc2cc1F)N1CCC(CCO)CC1 ZINC000880547830 DG On-Demand Anodyne AKR1C3 20 58 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)nc1 ZINC000880547837 ED On-Demand Anodyne PDGFRB 67 45 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)nc1 ZINC000880547837 ED On-Demand Anodyne FAAH 23 44 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)nc1 ZINC000880547837 ED On-Demand Anodyne DGAT1 39 48 CC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880547855 CE On-Demand Anodyne CHRM3 23 46 CC(=O)c1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880547855 CE On-Demand Anodyne MCHR2 51 34 c1cc(CN2CCOCC2)cc(CN2CCC3(CC2)COCCO3)c1 ZINC000880547858 ED On-Demand Anodyne SIGMAR1 32 41 CC[C@H](C)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880547875 CE On-Demand Anodyne PDGFRB 46 39 c1ccc(COc2ccc(CN3CCC4(CC3)COCCO4)cn2)cc1 ZINC000880547877 FG On-Demand Anodyne SIGMAR1 33 46 COc1ccc([C@@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547878 ED On-Demand Anodyne RAF1 15 40 COc1ccc([C@@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547878 ED On-Demand Anodyne MTNR1A 15 42 COc1ccc([C@@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547878 ED On-Demand Anodyne ROCK2 15 41 COc1ccc([C@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547880 ED On-Demand Anodyne RAF1 15 40 COc1ccc([C@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547880 ED On-Demand Anodyne MTNR1A 15 42 COc1ccc([C@H](CO)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880547880 ED On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)NCCc2cn(C)cn2)c1 ZINC000880547884 CD On-Demand Anodyne PIK3CG 15 61 O=C(c1coc(-c2ccccn2)n1)N1CCC(CCO)CC1 ZINC000880547922 DD On-Demand Anodyne AKR1C3 17 45 COc1cncc(NC(=O)N2CCCCCCCC2)c1 ZINC000880547924 CG On-Demand Anodyne PDGFRB 42 38 COc1cncc(NC(=O)N2CCC[C@@H](CCO)CC2)c1 ZINC000880547927 CE On-Demand Anodyne PDGFRB 42 37 COc1cncc(NC(=O)N2CCC[C@H](CCO)CC2)c1 ZINC000880547929 CE On-Demand Anodyne PDGFRB 42 37 Cc1nc(C(C)C)ncc1C(=O)N1CCC(CCO)CC1 ZINC000880547945 CE On-Demand Anodyne AKR1C3 16 41 O[C@@H]1CCC[C@H]1N1CCC2(CC1)COCCO2 ZINC000880547959 BC On-Demand Anodyne SLC18A3 34 44 COc1cncc(NC(=O)NCc2cc(C)nc(C)c2)c1 ZINC000880547971 CE On-Demand Anodyne ROCK2 28 47 COc1cncc(NC(=O)NCc2cc(C)nc(C)c2)c1 ZINC000880547971 CE On-Demand Anodyne NAMPT 27 40 COc1cncc(NC(=O)c2cc(Br)ccc2C2CC2)n1 ZINC000880547992 EG On-Demand Anodyne SORT1 15 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cncc(OC)n1)C2 ZINC000880547994 DE On-Demand Anodyne MTNR1A 27 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cncc(OC)n1)C2 ZINC000880547994 DE On-Demand Anodyne MTNR1B 26 41 O=C(c1ncccc1-c1ccccn1)N1CCC(CCO)CC1 ZINC000880547997 DE On-Demand Anodyne MLNR 19 44 Cc1ccc(-c2nc(C)c(C(=O)N3CCC(CCO)CC3)s2)c(F)c1 ZINC000880548007 FH On-Demand Anodyne AKR1C3 17 40 COc1cncc(NC(=O)NCC[C@H]2CCCN(C)C2)c1 ZINC000880548014 CD On-Demand Anodyne CCR3 67 47 COc1cncc(NC(=O)NCC[C@@H]2CCCN(C)C2)c1 ZINC000880548015 CD On-Demand Anodyne CCR3 67 47 COc1cncc(NC(=O)NC[C@@H]2C[C@H]2c2cccc(OC)c2)c1 ZINC000880548022 EG On-Demand Anodyne MTNR1B 36 41 COc1cncc(NC(=O)NC[C@@H]2C[C@H]2c2cccc(OC)c2)c1 ZINC000880548022 EG On-Demand Anodyne ROCK2 36 44 COc1cncc(NC(=O)N(C)C[C@H]2CCCN2C)c1 ZINC000880548035 CD On-Demand Anodyne CHRNA10 58 39 COc1cncc(NC(=O)N(C)C[C@H]2CCCN2C)c1 ZINC000880548035 CD On-Demand Anodyne ACKR3 65 33 COc1cncc(NC(=O)N(C)C[C@@H]2CCCN2C)c1 ZINC000880548036 CD On-Demand Anodyne CHRNA10 58 39 COc1cncc(NC(=O)N(C)C[C@@H]2CCCN2C)c1 ZINC000880548036 CD On-Demand Anodyne ACKR3 65 33 O=C(c1ccc(OC(F)F)c(Br)c1)N1CCC(CCO)CC1 ZINC000880548037 GG On-Demand Anodyne AKR1C3 16 44 O=C(c1ccc(OC(F)F)c(Br)c1)N1CCC(CCO)CC1 ZINC000880548037 GG On-Demand Anodyne L3MBTL3 56 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H](c3cccc(OC)c3)C2)c1 ZINC000880548044 EG On-Demand Anodyne MTNR1A 22 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H](c3cccc(OC)c3)C2)c1 ZINC000880548044 EG On-Demand Anodyne MTNR1B 27 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H](c3cccc(OC)c3)C2)c1 ZINC000880548044 EG On-Demand Anodyne EPHX2 28 45 COc1cncc(NC(=O)N2CC3(CC3)c3ccccc32)c1 ZINC000880548062 CG On-Demand Anodyne NPY5R 26 44 COc1cncc(NC(=O)N2CC[C@](O)(C(F)F)C2)c1 ZINC000880548070 CD On-Demand Anodyne S1PR2 29 42 COc1cncc(NC(=O)N2CC[C@@](O)(C(F)F)C2)c1 ZINC000880548071 CD On-Demand Anodyne S1PR2 29 42 COc1cncc(NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)c1 ZINC000880548106 DD On-Demand Anodyne DRD4 40 30 COc1cncc(NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)c1 ZINC000880548106 DD On-Demand Anodyne CCR3 29 41 COc1cncc(NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)c1 ZINC000880548106 DD On-Demand Anodyne MTOR 40 35 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(F)cc2C)c1 ZINC000880548118 EH On-Demand Anodyne CCR3 21 42 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(F)cc2C)c1 ZINC000880548119 EH On-Demand Anodyne CCR3 21 42 N#Cc1ccc(CCN2CCC3(CC2)COCCO3)cc1 ZINC000880548122 CD On-Demand Mild KCNJ1 52 60 COc1cncc(NC(=O)N2CCC3(CC2)OCCc2ccccc23)c1 ZINC000880548190 FG On-Demand Anodyne NPY5R 35 44 COc1cncc(NC(=O)N[C@H]2CCO[C@H](c3cccnc3)C2)c1 ZINC000880548193 EF On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@@H]2CCO[C@H](c3cccnc3)C2)c1 ZINC000880548194 EF On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@H]2CCO[C@@H](c3cccnc3)C2)c1 ZINC000880548195 EF On-Demand Anodyne CHRNA7 17 42 c1cc(CN2CCCCC2)cc(CN2CCC3(CC2)COCCO3)c1 ZINC000880548209 EG On-Demand Anodyne SIGMAR1 33 40 COc1cncc(NC(=O)N2CCN(CCO)C[C@H]2C)c1 ZINC000880548227 CC On-Demand Anodyne LIMK2 24 40 COc1cncc(NC(=O)N2CCN(CCO)C[C@@H]2C)c1 ZINC000880548228 CC On-Demand Anodyne LIMK2 24 40 COc1cncc(NC(=O)NCCCc2ncccc2C)c1 ZINC000880548246 DF On-Demand Anodyne HRH2 16 41 COc1cncc(NC(=O)N[C@@H]2CC[C@@H](Nc3ccccn3)CC2)c1 ZINC000880548249 EG On-Demand Anodyne EPHX2 44 37 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2cccc(OC)c2)c1 ZINC000880548257 DF On-Demand Anodyne MTNR1A 16 41 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2cccc(OC)c2)c1 ZINC000880548257 DF On-Demand Anodyne MTNR1B 22 41 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2cccc(OC)c2)c1 ZINC000880548257 DF On-Demand Anodyne EPHX2 20 45 COc1cncc(NC(=O)N(CCN2CCOCC2)Cc2ccco2)c1 ZINC000880548266 FE On-Demand Anodyne CASR 62 53 COc1cncc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)c1 ZINC000880548270 FD On-Demand Anodyne RBP4 46 34 COc1cncc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)c1 ZINC000880548271 FD On-Demand Anodyne RBP4 46 34 COc1cncc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)c1 ZINC000880548272 FD On-Demand Anodyne RBP4 46 34 COc1cncc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)c1 ZINC000880548273 FD On-Demand Anodyne RBP4 46 34 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(CCO)CC1 ZINC000880548274 DD On-Demand Anodyne GRIN2B 44 42 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(CCO)CC1 ZINC000880548274 DD On-Demand Anodyne AKR1C3 21 54 c1ccc(COCCN2CCC3(CC2)COCCO3)cc1 ZINC000880548317 CE On-Demand Anodyne LTA4H 19 40 c1cc(CN2CCC3(CC2)COCCO3)ccc1CN1CCCCC1 ZINC000880548321 EG On-Demand Anodyne HRH3 22 54 c1cc(CN2CCC3(CC2)COCCO3)ccc1CN1CCCCC1 ZINC000880548321 EG On-Demand Anodyne SIGMAR1 33 40 c1cc(CN2CCC3(CC2)COCCO3)ccc1CN1CCCCC1 ZINC000880548321 EG On-Demand Anodyne CXCR4 19 40 FC(F)(F)c1cc(CN2CCC3(CC2)COCCO3)ccc1Cl ZINC000880548335 EH On-Demand Anodyne SIGMAR1 16 40 CC(C)(C)OC(=O)N1CCC(CCCN2CCC3(CC2)COCCO3)CC1 ZINC000880548336 GG On-Demand Anodyne GPR119 26 41 COc1cncc(NC(=O)N2CCc3cccc(OC)c3C2)c1 ZINC000880548339 DF On-Demand Anodyne HTR2C 15 41 COc1cncc(NC(=O)N2CCc3cccc(OC)c3C2)c1 ZINC000880548339 DF On-Demand Anodyne SSTR1 50 35 COc1cncc(NC(=O)N2CCc3cccc(OC)c3C2)c1 ZINC000880548339 DF On-Demand Anodyne P2RY14 51 37 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(F)cc2F)c1 ZINC000880548357 EH On-Demand Anodyne CCR3 17 42 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(F)cc2F)c1 ZINC000880548358 EH On-Demand Anodyne CCR3 17 42 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne CTSL 45 37 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne BRS3 26 41 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne MTNR1A 48 37 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne MTNR1B 48 37 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne MMP3 41 41 COc1cncc(NC(=O)N[C@@H](C)C(=O)NCCc2ccccc2)c1 ZINC000880548362 ED On-Demand Anodyne ROCK2 19 42 COc1cncc(NC(=O)N(C)C2CCN(CC(F)(F)F)CC2)c1 ZINC000880548363 EF On-Demand Anodyne HPGDS 34 42 CSc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548376 FE On-Demand Anodyne ACOX1 47 31 CSc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548376 FE On-Demand Anodyne CCR1 47 40 CSc1ccc(OC[C@@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548376 FE On-Demand Anodyne ABCB1 50 39 CSc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548377 FE On-Demand Anodyne ACOX1 47 31 CSc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548377 FE On-Demand Anodyne CCR1 47 40 CSc1ccc(OC[C@H](O)CN2CCC3(CC2)COCCO3)cc1 ZINC000880548377 FE On-Demand Anodyne ABCB1 50 39 COc1cncc(NC(=O)NC2CCC(OC(F)F)CC2)c1 ZINC000880548390 DF On-Demand Anodyne EPHX2 50 41 C=C(C)CONC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880548391 CG On-Demand Mild PDE4D 18 42 COc1cncc(NC(=O)N(C)[C@@H]2C[C@@H](c3cccc(OC)c3)C2)c1 ZINC000880548397 EH On-Demand Anodyne ROCK1 17 41 COc1cncc(NC(=O)N(C)[C@@H]2C[C@@H](c3cccc(OC)c3)C2)c1 ZINC000880548397 EH On-Demand Anodyne ROCK2 32 41 COc1cncc(NC(=O)N2CCc3cc(OC)ccc32)c1 ZINC000880548413 CF On-Demand Anodyne CYP11B1 21 57 COc1cncc(NC(=O)N2CCc3cc(OC)ccc32)c1 ZINC000880548413 CF On-Demand Anodyne HTR2C 20 49 COc1cncc(NC(=O)N2CCc3cc(OC)ccc32)c1 ZINC000880548413 CF On-Demand Anodyne CYP11B2 38 47 COc1cncc(NC(=O)NC2CCN(C3CCC3)CC2)c1 ZINC000880548443 DE On-Demand Anodyne HRH3 23 42 COc1cncc(NC(=O)NC2CCN(C3CCC3)CC2)c1 ZINC000880548443 DE On-Demand Anodyne EPHX2 48 39 COc1cncc(NC(=O)NC2CCN(C3CCC3)CC2)c1 ZINC000880548443 DE On-Demand Anodyne CXCR3 18 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(CCO)CC1 ZINC000880548483 FG On-Demand Anodyne RBP4 47 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(CCO)CC1 ZINC000880548483 FG On-Demand Anodyne AKR1C3 18 47 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(CCO)CC1 ZINC000880548483 FG On-Demand Anodyne SCD1 28 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(CCO)CC1 ZINC000880548483 FG On-Demand Anodyne SCD 28 40 COc1cncc(NC(=O)NC23CCC(CC2)CC3)c1 ZINC000880548485 CF On-Demand Anodyne EPHX2 38 49 COc1cncc(NC(=O)N2CC(c3cccc(Cl)c3)C2)c1 ZINC000880548488 DG On-Demand Anodyne GRM5 15 43 C=C(C)CONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880548489 CE On-Demand Mild NQO2 28 42 C=C(C)CONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880548489 CE On-Demand Mild MTNR1A 45 43 C=C(C)CONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880548490 CE On-Demand Mild NQO2 28 42 C=C(C)CONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880548490 CE On-Demand Mild MTNR1A 45 43 COc1cncc(NC(=O)NC2C[C@@H]3CC[C@H](C2)N3C)c1 ZINC000880548508 CD On-Demand Anodyne GLRA1 43 35 C=C(C)CONC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880548509 DG On-Demand Mild INHA 48 38 O=C(c1cc(Br)ccc1C1CC1)N1CCC(CCO)CC1 ZINC000880548511 FH On-Demand Anodyne AKR1C3 21 45 COc1cncc(NC(=O)N2CC[C@H](c3nc(C)no3)C2)c1 ZINC000880548514 DD On-Demand Anodyne SMO 34 48 COc1cncc(NC(=O)N2CC[C@@H](c3nc(C)no3)C2)c1 ZINC000880548515 DD On-Demand Anodyne SMO 34 48 COc1cncc(NC(=O)NC[C@H](O)c2ccc(OC(F)(F)F)cc2)c1 ZINC000880548535 FF On-Demand Anodyne P2RY1 51 36 COc1cncc(NC(=O)NC[C@@H](O)c2ccc(OC(F)(F)F)cc2)c1 ZINC000880548536 FF On-Demand Anodyne P2RY1 51 36 COc1cncc(NC(=O)NCCCCN(C)C2CC2)c1 ZINC000880548558 CE On-Demand Anodyne CCR3 27 41 COC[C@@H]1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880548561 CE On-Demand Anodyne PDGFRB 45 36 COc1cncc(NC(=O)NC2CCC2)c1 ZINC000880548566 BD On-Demand Anodyne EPHX2 54 43 COc1cncc(NC(=O)NC2CCC2)c1 ZINC000880548566 BD On-Demand Anodyne PDGFRA 16 45 COc1cncc(NC(=O)N2CCC[C@H](Oc3ccccc3)C2)c1 ZINC000880548567 EG On-Demand Anodyne CCR3 19 49 COc1cncc(NC(=O)N2CCC[C@H](Oc3ccccc3)C2)c1 ZINC000880548567 EG On-Demand Anodyne EPHX2 27 43 COc1cncc(NC(=O)N2CCC[C@@H](Oc3ccccc3)C2)c1 ZINC000880548568 EG On-Demand Anodyne CCR3 19 49 COc1cncc(NC(=O)N2CCC[C@@H](Oc3ccccc3)C2)c1 ZINC000880548568 EG On-Demand Anodyne EPHX2 27 43 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne CA2 22 44 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne CA1 48 44 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne RAF1 17 44 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne ROCK2 15 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne PTPRB 48 37 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne CA12 38 44 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne CA9 39 44 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne MTCA1 41 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880548572 EF On-Demand Anodyne P96878_MYCTU 51 42 CCN1C[C@H](NC(=O)Nc2cncc(OC)c2)CC1=O ZINC000880548578 CC On-Demand Anodyne EPHX2 18 40 FC(F)(F)Oc1cccc(CN2CCC3(CC2)COCCO3)c1 ZINC000880548594 EF On-Demand Anodyne SIGMAR1 19 40 O=C(c1c[nH]cc1C1CC1)N1CCC(CCO)CC1 ZINC000880548595 CE On-Demand Anodyne AKR1C3 17 46 COc1cncc(NC(=O)N2CCCc3cc(OC)ccc32)c1 ZINC000880548612 DG On-Demand Anodyne CYP11B1 22 51 COc1cncc(NC(=O)N2CCCc3cc(OC)ccc32)c1 ZINC000880548612 DG On-Demand Anodyne HTR2C 18 44 COc1cncc(NC(=O)N2CCCc3cc(OC)ccc32)c1 ZINC000880548612 DG On-Demand Anodyne CYP11B2 42 42 COc1cncc(NC(=O)N2CC(c3ccc(Cl)cc3)C2)c1 ZINC000880548613 DG On-Demand Anodyne CACNA1H 42 37 COc1cncc(NC(=O)N2CC(c3ccc(Cl)cc3)C2)c1 ZINC000880548613 DG On-Demand Anodyne SCN10A 27 43 c1cc(CN2CCC3(CC2)COCCO3)ccc1CN1CCOCC1 ZINC000880548624 ED On-Demand Anodyne SIGMAR1 29 41 O=C(c1cccc(CN2CCC3(CC2)COCCO3)c1)C(F)(F)F ZINC000880548630 EF On-Demand Anodyne CHRM3 17 42 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3F)C2)c1 ZINC000880548715 DG On-Demand Anodyne CCR3 16 43 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3F)C2)c1 ZINC000880548715 DG On-Demand Anodyne RBP4 69 42 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3F)C2)c1 ZINC000880548716 DG On-Demand Anodyne CCR3 16 43 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3F)C2)c1 ZINC000880548716 DG On-Demand Anodyne RBP4 69 42 COc1cncc(NC(=O)N(C)C[C@@H](O)Cc2ccccc2)c1 ZINC000880548723 DE On-Demand Anodyne ROCK1 15 41 COc1cncc(NC(=O)N(C)C[C@@H](O)Cc2ccccc2)c1 ZINC000880548723 DE On-Demand Anodyne ROCK2 22 41 COc1cncc(NC(=O)N(C)C[C@@H](O)Cc2ccccc2)c1 ZINC000880548723 DE On-Demand Anodyne NPY5R 35 45 COc1cncc(NC(=O)N(C)C[C@H](O)Cc2ccccc2)c1 ZINC000880548724 DE On-Demand Anodyne ROCK1 15 41 COc1cncc(NC(=O)N(C)C[C@H](O)Cc2ccccc2)c1 ZINC000880548724 DE On-Demand Anodyne ROCK2 22 41 COc1cncc(NC(=O)N(C)C[C@H](O)Cc2ccccc2)c1 ZINC000880548724 DE On-Demand Anodyne NPY5R 35 45 COc1cncc(NC(=O)N(Cc2cccc(C(N)=O)c2)C2CC2)c1 ZINC000880548725 EE On-Demand Anodyne ROCK1 16 41 COc1cncc(NC(=O)N(Cc2cccc(C(N)=O)c2)C2CC2)c1 ZINC000880548725 EE On-Demand Anodyne ROCK2 29 54 COc1cncc(NC(=O)N[C@@H]2CCCN(CCCO)C2)c1 ZINC000880548730 DD On-Demand Anodyne CCR3 61 45 COc1cncc(NC(=O)N[C@@H]2CCCN(CCCO)C2)c1 ZINC000880548730 DD On-Demand Anodyne EPHX2 30 42 COc1cncc(NC(=O)N[C@H]2CCCN(CCCO)C2)c1 ZINC000880548731 DD On-Demand Anodyne CCR3 61 45 COc1cncc(NC(=O)N[C@H]2CCCN(CCCO)C2)c1 ZINC000880548731 DD On-Demand Anodyne EPHX2 30 42 COc1cncc(NC(=O)NC[C@H](Cc2ccccc2)OC)c1 ZINC000880548732 DE On-Demand Anodyne ROCK2 25 41 COc1cncc(NC(=O)NC[C@H](Cc2ccccc2)OC)c1 ZINC000880548732 DE On-Demand Anodyne NAMPT 15 42 COc1cncc(NC(=O)NC[C@@H](Cc2ccccc2)OC)c1 ZINC000880548733 DE On-Demand Anodyne ROCK2 25 41 COc1cncc(NC(=O)NC[C@@H](Cc2ccccc2)OC)c1 ZINC000880548733 DE On-Demand Anodyne NAMPT 15 42 COc1cncc(NC(=O)N(C)[C@@H](CO)c2ccc(Cl)cc2)c1 ZINC000880548751 EF On-Demand Anodyne SCN10A 23 42 COc1cncc(NC(=O)N(C)[C@H](CO)c2ccc(Cl)cc2)c1 ZINC000880548752 EF On-Demand Anodyne SCN10A 23 42 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HTR1A 29 41 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne DRD2 30 41 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HRH2 30 49 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HTR2A 17 50 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HTR2C 15 40 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne DRD3 58 41 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HTR4 17 43 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne HRH3 15 40 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne NPY1R 15 43 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne CCR3 52 50 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne CHRNA7 28 56 COc1cncc(NC(=O)NCCCCCN2CCCC2)c1 ZINC000880548769 DE On-Demand Anodyne QPCT 15 41 O[C@H](COc1cc(Cl)cc(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880548771 GF On-Demand Anodyne CCR1 51 43 O[C@@H](COc1cc(Cl)cc(Cl)c1)CN1CCC2(CC1)COCCO2 ZINC000880548772 GF On-Demand Anodyne CCR1 51 43 COc1cncc(NC(=O)N(Cc2ccc(C(N)=O)cc2F)C2CC2)c1 ZINC000880548773 FF On-Demand Anodyne ROCK2 30 41 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne ROCK1 29 40 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne ROCK2 42 48 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne SOAT1 17 41 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne MTOR 55 37 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne STAT6 50 46 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)c2)c1 ZINC000880548786 EE On-Demand Anodyne NAMPT 47 44 O[C@]1(CN2CCC3(CC2)COCCO3)CCN(Cc2ccccc2)C1 ZINC000880548799 ED On-Demand Anodyne SIGMAR1 36 42 O[C@@]1(CN2CCC3(CC2)COCCO3)CCN(Cc2ccccc2)C1 ZINC000880548800 ED On-Demand Anodyne SIGMAR1 36 42 COc1cncc(NC(=O)N2CCN(C3CCC3)C[C@@H](C)C2)c1 ZINC000880548801 DE On-Demand Anodyne HRH3 19 41 COc1cncc(NC(=O)N2CCN(C3CCC3)C[C@H](C)C2)c1 ZINC000880548802 DE On-Demand Anodyne HRH3 19 41 CCOC(=O)c1cnn(C2CCN(C(=O)Nc3cncc(OC)c3)CC2)c1 ZINC000880548811 FE On-Demand Anodyne P2RY12 16 47 COc1cncc(NC(=O)N2CCC(CO)(c3ccccc3)CC2)c1 ZINC000880548864 EF On-Demand Anodyne KCNA3 41 41 COc1cncc(NC(=O)N2CCC(CO)(c3ccccc3)CC2)c1 ZINC000880548864 EF On-Demand Anodyne SOAT1 17 40 COc1cncc(NC(=O)N2CCC(CO)(c3ccccc3)CC2)c1 ZINC000880548864 EF On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CCC(CO)(c3ccccc3)CC2)c1 ZINC000880548864 EF On-Demand Anodyne EPHX2 26 43 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880548868 FE On-Demand Anodyne EPHX2 35 41 C=C[C@@H](C)ONC(=O)Cc1ccccc1N1CCCC1=O ZINC000880548876 CD On-Demand Mild KCNQ2 44 34 C=C[C@H](C)ONC(=O)Cc1ccccc1N1CCCC1=O ZINC000880548877 CD On-Demand Mild KCNQ2 44 34 COc1cncc(NC(=O)N2CCC[C@@H](CO)CC2)c1 ZINC000880548888 CD On-Demand Anodyne PDGFRB 45 36 COc1cncc(NC(=O)N2CCC[C@H](CO)CC2)c1 ZINC000880548889 CD On-Demand Anodyne PDGFRB 45 36 COc1cncc(NC(=O)N2CCC3(CC2)CCN(C(=O)OC(C)(C)C)C3)c1 ZINC000880548896 GG On-Demand Anodyne EPHX2 27 43 COc1cncc(NC(=O)N2CCC3(CC2)CCN(C(=O)OC(C)(C)C)C3)c1 ZINC000880548896 GG On-Demand Anodyne GPR119 15 44 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc[nH]n2)c1 ZINC000880548907 DD On-Demand Anodyne CPT1A 63 36 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc[nH]n2)c1 ZINC000880548908 DD On-Demand Anodyne CPT1A 63 36 COc1cncc(NC(=O)N2CC(C)(C)[C@@H]2c2cccnc2)c1 ZINC000880548937 DG On-Demand Anodyne CHRNA7 17 49 COc1cncc(NC(=O)N2CC(C)(C)[C@H]2c2cccnc2)c1 ZINC000880548938 DG On-Demand Anodyne CHRNA7 17 49 COc1cncc(NC(=O)NCCCc2cnn(C)n2)c1 ZINC000880548950 CC On-Demand Anodyne QPCT 23 44 COc1cncc(NC(=O)NCCCS(=O)(=O)c2ccc(Cl)cc2)c1 ZINC000880548966 GF On-Demand Anodyne SCN10A 30 41 COc1cncc(NC(=O)NCCCS(=O)(=O)c2ccc(Cl)cc2)c1 ZINC000880548966 GF On-Demand Anodyne NAMPT 31 42 COC(=O)CCCCN1CCC2(CC1)COCCO2 ZINC000880548973 CD On-Demand Anodyne PAOX 19 40 COc1cncc(NC(=O)NCC(=O)NCCN2CCCCCC2)c1 ZINC000880548977 ED On-Demand Anodyne DRD4 46 36 COc1cncc(NC(=O)NCC(=O)NCCN2CCCCCC2)c1 ZINC000880548977 ED On-Demand Anodyne HRH2 37 43 COc1cncc(NC(=O)NCC(=O)NCCN2CCCCCC2)c1 ZINC000880548977 ED On-Demand Anodyne CCR3 26 41 COc1cncc(NC(=O)NCC(=O)NCCN2CCCCCC2)c1 ZINC000880548977 ED On-Demand Anodyne CHRNA7 17 46 C=C(C)CONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549004 DD On-Demand Mild PAPA1_CARPA 38 44 C=C(C)CONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549004 DD On-Demand Mild CTSK 17 51 C=C(C)CONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549005 DD On-Demand Mild PAPA1_CARPA 38 44 C=C(C)CONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549005 DD On-Demand Mild CTSK 17 51 COc1cncc(NC(=O)NC2CCC(CS(C)(=O)=O)CC2)c1 ZINC000880549024 ED On-Demand Anodyne EPHX2 40 36 C=C[C@@H](C)ONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880549037 CE On-Demand Mild MMP3 19 40 C=C[C@@H](C)ONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880549037 CE On-Demand Mild MMP8 17 40 C=C[C@H](C)ONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880549038 CE On-Demand Mild MMP3 19 40 C=C[C@H](C)ONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880549038 CE On-Demand Mild MMP8 17 40 C=C[C@@H](C)ONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880549039 CE On-Demand Mild MMP3 19 40 C=C[C@@H](C)ONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880549039 CE On-Demand Mild MMP8 17 40 C=C[C@H](C)ONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880549040 CE On-Demand Mild MMP3 19 40 C=C[C@H](C)ONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880549040 CE On-Demand Mild MMP8 17 40 C[C@@H](NC(=O)CN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880549041 DD On-Demand Anodyne PSMB8 39 40 COc1cncc(NC(=O)N[C@@H]2C[C@@H](c3ccc(F)cc3)C2)c1 ZINC000880549052 DG On-Demand Anodyne CCR3 16 41 COc1cncc(NC(=O)NCCc2cc(C(F)(F)F)ccn2)c1 ZINC000880549058 EF On-Demand Anodyne RAF1 45 42 COc1cncc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c1 ZINC000880549066 ED On-Demand Anodyne CHRNA4 28 45 COc1cncc(NC(=O)N[C@]2(C)C[C@H]2c2ccccc2)c1 ZINC000880549067 CG On-Demand Anodyne EPHX2 22 45 COc1cncc(NC(=O)NC[C@@H](O)Cc2cccc(F)c2)c1 ZINC000880549080 DD On-Demand Anodyne ADRB1 43 34 COc1cncc(NC(=O)NC[C@@H](O)Cc2cccc(F)c2)c1 ZINC000880549080 DD On-Demand Anodyne ROCK2 26 42 COc1cncc(NC(=O)NC[C@H](O)Cc2cccc(F)c2)c1 ZINC000880549081 DD On-Demand Anodyne ADRB1 43 34 COc1cncc(NC(=O)NC[C@H](O)Cc2cccc(F)c2)c1 ZINC000880549081 DD On-Demand Anodyne ROCK2 26 42 COc1cncc(NC(=O)N(C)[C@@H](CO)c2ccccc2)c1 ZINC000880549084 DE On-Demand Anodyne NPY5R 38 43 COc1cncc(NC(=O)N(C)[C@H](CO)c2ccccc2)c1 ZINC000880549085 DE On-Demand Anodyne NPY5R 38 43 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne CASP3 45 39 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne CHRNA7 30 56 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne CPT1A 104 37 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne CPT2 44 36 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne PREP 46 33 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne CHRNA10 81 45 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne MCHR1 16 41 COc1cncc(NC(=O)N2CCC[C@H]2COc2ccccc2)c1 ZINC000880549091 EG On-Demand Anodyne ACKR3 64 34 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild ELANE 20 40 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild PREP 26 41 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild CAPNS1 45 30 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild LGMN 69 38 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild CAPN1 45 43 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild CAPN2 44 34 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild TGM2 40 39 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild NPR 40 32 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild SLC12A5 54 35 C=C[C@@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549098 EE On-Demand Mild Q9NAW4_PLAFA 41 49 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild ELANE 20 40 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild PREP 26 41 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild CAPNS1 45 30 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild LGMN 69 38 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild CAPN1 45 43 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild CAPN2 44 34 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild TGM2 40 39 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild NPR 40 32 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild SLC12A5 54 35 C=C[C@H](C)ONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880549099 EE On-Demand Mild Q9NAW4_PLAFA 41 49 CC(=O)[C@@](C#N)(CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880549104 EE On-Demand Mild CCR1 23 46 CC(=O)[C@](C#N)(CCN1CCC2(CC1)COCCO2)c1ccccc1 ZINC000880549105 EE On-Demand Mild CCR1 23 46 COc1cncc(NC(=O)N2CCc3cc(OC)c(Cl)cc3C2)c1 ZINC000880549116 EG On-Demand Anodyne ABCB1 17 42 COc1cncc(NC(=O)N2CC[C@]3(CCN(C)C3)C2)c1 ZINC000880549124 CD On-Demand Anodyne EPHX2 29 42 COc1cncc(NC(=O)N2CC[C@@]3(CCN(C)C3)C2)c1 ZINC000880549125 CD On-Demand Anodyne EPHX2 29 42 COc1cncc(NC(=O)Nc2ccc([C@@H]3CCOC3)cc2)c1 ZINC000880549126 DG On-Demand Anodyne MTOR 45 39 COc1cncc(NC(=O)Nc2ccc([C@H]3CCOC3)cc2)c1 ZINC000880549127 DG On-Demand Anodyne MTOR 45 39 COc1cncc(NC(=O)NC[C@H]2CCCN2CCCO)c1 ZINC000880549137 DD On-Demand Anodyne DRD2 32 40 COc1cncc(NC(=O)NC[C@H]2CCCN2CCCO)c1 ZINC000880549137 DD On-Demand Anodyne CCR3 34 40 COc1cncc(NC(=O)NC[C@@H]2CCCN2CCCO)c1 ZINC000880549138 DD On-Demand Anodyne DRD2 32 40 COc1cncc(NC(=O)NC[C@@H]2CCCN2CCCO)c1 ZINC000880549138 DD On-Demand Anodyne CCR3 34 40 COc1cncc(NC(=O)NC[C@H](CO)C2CCCCC2)c1 ZINC000880549155 DE On-Demand Anodyne PRMT3 24 40 COc1cncc(NC(=O)NC[C@@H](CO)C2CCCCC2)c1 ZINC000880549156 DE On-Demand Anodyne PRMT3 24 40 C=C[C@@H](C)ONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549228 DD On-Demand Mild PAPA1_CARPA 35 43 C=C[C@@H](C)ONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549228 DD On-Demand Mild CTSK 15 50 C=C[C@@H](C)ONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549229 DD On-Demand Mild PAPA1_CARPA 35 43 C=C[C@@H](C)ONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549229 DD On-Demand Mild CTSK 15 50 C=C[C@H](C)ONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549230 DD On-Demand Mild PAPA1_CARPA 35 43 C=C[C@H](C)ONC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549230 DD On-Demand Mild CTSK 15 50 C=C[C@H](C)ONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549231 DD On-Demand Mild PAPA1_CARPA 35 43 C=C[C@H](C)ONC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880549231 DD On-Demand Mild CTSK 15 50 COc1cncc(NC(=O)N[C@H]2CCc3c(O)cccc32)c1 ZINC000880549254 CF On-Demand Anodyne TRPV1 18 42 COc1cncc(NC(=O)N[C@@H]2CCc3c(O)cccc32)c1 ZINC000880549255 CF On-Demand Anodyne TRPV1 18 42 COc1cncc(NC(=O)N2CCN(c3cnccc3C#N)CC2)c1 ZINC000880549279 ED On-Demand Mild DRD4 40 32 COc1cncc(NC(=O)N2CCN(c3cnccc3C#N)CC2)c1 ZINC000880549279 ED On-Demand Mild PDGFRB 56 44 COc1cncc(NC(=O)N2CCN(c3cnccc3C#N)CC2)c1 ZINC000880549279 ED On-Demand Mild FAAH 16 45 CCOC(=O)C1([S@@](C)=O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880549280 FD On-Demand Anodyne S1PR2 28 40 CCOC(=O)C1([S@](C)=O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880549281 FD On-Demand Anodyne S1PR2 28 40 C=C(C)CONC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880549297 GE On-Demand Mild GPR119 36 44 CC(=O)Nc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880549305 GG On-Demand Anodyne DRD4 19 44 CC(=O)Nc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880549305 GG On-Demand Anodyne CCKBR 31 43 N#Cc1ccccc1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549314 ED On-Demand Mild ADRB1 52 36 N#Cc1ccccc1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549314 ED On-Demand Mild CCR1 49 45 N#Cc1ccccc1OC[C@@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549314 ED On-Demand Mild ABCB1 70 48 N#Cc1ccccc1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549315 ED On-Demand Mild ADRB1 52 36 N#Cc1ccccc1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549315 ED On-Demand Mild CCR1 49 45 N#Cc1ccccc1OC[C@H](O)CN1CCC2(CC1)COCCO2 ZINC000880549315 ED On-Demand Mild ABCB1 70 48 COc1cncc(NC(=O)NCc2cccc(C3(C)OCCO3)c2)c1 ZINC000880549317 EF On-Demand Anodyne ROCK1 26 41 COc1cncc(NC(=O)NCc2cccc(C3(C)OCCO3)c2)c1 ZINC000880549317 EF On-Demand Anodyne ROCK2 43 49 COc1cncc(NC(=O)NCCCC2CCOCC2)c1 ZINC000880549322 CE On-Demand Anodyne CCR3 28 41 O=C(CN1CCC2(CC1)COCCO2)Nc1ccc(Cl)c(F)c1 ZINC000880549348 EE On-Demand Anodyne ENV 44 38 COc1cncc(NC(=O)NCCc2cccc(C(F)(F)F)n2)c1 ZINC000880549363 EF On-Demand Anodyne RAF1 31 41 COc1cncc(NC(=O)NCCc2cccc(C(F)(F)F)n2)c1 ZINC000880549363 EF On-Demand Anodyne MTNR1A 40 39 COc1cncc(NC(=O)NC[C@@H](O)CN2CCc3ccccc3C2)c1 ZINC000880549369 FD On-Demand Anodyne NOD1 16 43 COc1cncc(NC(=O)NC[C@@H](O)CN2CCc3ccccc3C2)c1 ZINC000880549369 FD On-Demand Anodyne NOD2 45 43 COc1cncc(NC(=O)N2CC[C@]3(CCCN(C)C3)C2)c1 ZINC000880549399 DE On-Demand Anodyne EPHX2 29 40 COc1cncc(NC(=O)N2CC[C@@]3(CCCN(C)C3)C2)c1 ZINC000880549400 DE On-Demand Anodyne EPHX2 29 40 COc1cncc(NC(=O)N2CCCC[C@H]2c2cc[nH]n2)c1 ZINC000880549414 DF On-Demand Anodyne CPT1A 53 37 COc1cncc(NC(=O)N2CCCC[C@@H]2c2cc[nH]n2)c1 ZINC000880549415 DF On-Demand Anodyne CPT1A 53 37 COCCCONC(=O)Nc1cncc(OC)c1 ZINC000880549417 CD On-Demand Anodyne SCN10A 22 40 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549424 DF On-Demand Anodyne DRD4 33 42 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549424 DF On-Demand Anodyne SIGMAR1 26 40 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549424 DF On-Demand Anodyne NOD2 42 35 COc1cncc(NC(=O)NCCCn2cc(Br)cn2)c1 ZINC000880549440 FE On-Demand Anodyne QPCT 18 42 N#CCc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549443 GF On-Demand Mild ABCB1 46 38 N#CCc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549444 GF On-Demand Mild ABCB1 46 38 COc1cncc(NC(=O)NCc2c(F)cccc2N2CCCC2)c1 ZINC000880549449 EG On-Demand Anodyne DRD4 45 37 COc1cncc(NC(=O)NCc2c(F)cccc2N2CCCC2)c1 ZINC000880549449 EG On-Demand Anodyne DRD3 49 37 COc1cncc(NC(=O)NCc2c(F)cccc2N2CCCC2)c1 ZINC000880549449 EG On-Demand Anodyne KCNQ2 64 38 COc1cncc(NC(=O)NCc2c(F)cccc2N2CCCC2)c1 ZINC000880549449 EG On-Demand Anodyne TAAR1 35 40 c1ccc2c(c1)CN(Cc1nc3ccccc3[nH]1)C[C@H]1CCCN21 ZINC000880549460 DH On-Demand Anodyne KCNN3 29 40 COc1cncc(NC(=O)N(C)CCc2ccccc2[N+](=O)[O-])c1 ZINC000880549478 EF On-Demand Bother COLA 115 42 C=CC(C)(C)CC(=O)N1C[C@@H](C(=O)OC)[C@H](c2ccccc2)C1 ZINC000880549488 DG On-Demand Mild SLC6A3 35 49 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC[C@H]1CCCO1 ZINC000880549490 ED On-Demand Anodyne PDE8B 15 40 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC[C@@H]1CCCO1 ZINC000880549491 ED On-Demand Anodyne PDE8B 15 40 COc1cncc(NC(=O)N2C[C@@H](CO)[C@H](c3ccsc3)C2)c1 ZINC000880549496 EE On-Demand Anodyne NPBWR1 79 33 COc1cncc(NC(=O)N(C)Cc2cccc(C)c2C)c1 ZINC000880549497 CG On-Demand Anodyne ROCK2 21 44 COC(=O)[C@@H]1CN(C(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)C[C@H]1c1ccccc1 ZINC000880549500 EE On-Demand Anodyne SLC6A3 23 47 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc(C)no2)c1 ZINC000880549506 DF On-Demand Anodyne CPT1A 84 45 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc(C)no2)c1 ZINC000880549507 DF On-Demand Anodyne CPT1A 84 45 COC(=O)[C@@H]1CN(C(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)C[C@H]1c1ccccc1 ZINC000880549508 FE On-Demand Anodyne SLC6A3 17 45 COC(=O)[C@@H]1CN(C(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)C[C@H]1c1ccccc1 ZINC000880549509 FE On-Demand Anodyne SLC6A3 17 45 COC(=O)[C@@H]1CN(C(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)C[C@H]1c1ccccc1 ZINC000880549510 FE On-Demand Anodyne SLC6A3 17 45 COC(=O)[C@@H]1CN(C(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)C[C@H]1c1ccccc1 ZINC000880549511 FE On-Demand Anodyne SLC6A3 17 45 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3F)C2)c1 ZINC000880549514 EF On-Demand Anodyne CCR3 34 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3F)C2)c1 ZINC000880549515 EF On-Demand Anodyne CCR3 34 42 O=C(CN1CCC2(CC1)COCCO2)c1c[nH]c2ccc(F)cc12 ZINC000880549516 EE On-Demand Anodyne MPO 74 37 c1ccc2c(c1)CC[C@H]2CCN1CCC2(CC1)COCCO2 ZINC000880549517 DF On-Demand Anodyne SIGMAR1 22 47 c1ccc2c(c1)CC[C@H]2CCN1CCC2(CC1)COCCO2 ZINC000880549517 DF On-Demand Anodyne EBP 24 41 c1ccc2c(c1)CC[C@@H]2CCN1CCC2(CC1)COCCO2 ZINC000880549518 DF On-Demand Anodyne SIGMAR1 22 47 c1ccc2c(c1)CC[C@@H]2CCN1CCC2(CC1)COCCO2 ZINC000880549518 DF On-Demand Anodyne EBP 24 41 COc1cncc(NC(=O)NCc2snnc2C)c1 ZINC000880549521 CD On-Demand Anodyne PRMT3 60 34 C=C[C@H](C)ONC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880549529 GE On-Demand Mild GPR119 23 42 C=C[C@@H](C)ONC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880549530 GE On-Demand Mild GPR119 23 42 CO[C@@H](CN1CCC2(CC1)COCCO2)c1ccc(F)cc1 ZINC000880549567 DE On-Demand Anodyne LEF 15 40 COc1cncc(NC(=O)N2CC[C@H]3[C@@H](CCN3C(=O)OC(C)(C)C)C2)c1 ZINC000880549575 GF On-Demand Anodyne GPR119 20 40 COc1cncc(NC(=O)N2CC[C@H]3[C@H](CCN3C(=O)OC(C)(C)C)C2)c1 ZINC000880549576 GF On-Demand Anodyne GPR119 20 40 COc1cncc(NC(=O)N2CC[C@@H]3[C@H](CCN3C(=O)OC(C)(C)C)C2)c1 ZINC000880549577 GF On-Demand Anodyne GPR119 20 40 COc1cncc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C(=O)OC(C)(C)C)C2)c1 ZINC000880549578 GF On-Demand Anodyne GPR119 20 40 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1ccccc1 ZINC000880549605 EG On-Demand Anodyne AVPR2 47 35 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549608 FF On-Demand Anodyne CCR3 32 48 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549608 FF On-Demand Anodyne CHRNA7 18 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549608 FF On-Demand Anodyne EPHX2 63 49 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549608 FF On-Demand Anodyne MCHR1 15 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549609 FF On-Demand Anodyne CCR3 32 48 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549609 FF On-Demand Anodyne CHRNA7 18 42 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549609 FF On-Demand Anodyne EPHX2 63 49 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)c1 ZINC000880549609 FF On-Demand Anodyne MCHR1 15 40 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne PREP 24 43 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne DPP7 50 34 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne XIAP 50 35 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne BIRC3 45 35 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne BIRC2 95 36 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549621 GD On-Demand Anodyne BIRC8 46 33 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne PREP 24 43 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne DPP7 50 34 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne XIAP 50 35 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne BIRC3 45 35 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne BIRC2 95 36 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N1CCCCC1 ZINC000880549622 GD On-Demand Anodyne BIRC8 46 33 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCN(C(=O)C2CC2)CC1 ZINC000880549627 GD On-Demand Anodyne PREP 65 41 COC[C@@H](O)CNC(=O)Nc1cncc(OC)c1 ZINC000880549637 CC On-Demand Anodyne ADRB1 43 32 O=C(O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549661 CD On-Demand Anodyne HTR1A 19 42 O=C(O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549661 CD On-Demand Anodyne SLC6A1 78 36 O=C(O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549661 CD On-Demand Anodyne HTR7 28 45 CS(=O)(=O)NCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549662 DD On-Demand Anodyne HTR7 18 41 COc1cncc(NC(=O)N2CCN(c3nccnc3C)CC2)c1 ZINC000880549673 ED On-Demand Anodyne PDGFRB 62 44 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne CCR3 48 43 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne CPT1A 15 40 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne PREP 46 34 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne CCKBR 16 40 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne EPHX2 37 43 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne MCHR1 17 40 COc1cncc(NC(=O)N[C@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549676 FE On-Demand Anodyne BIRC2 21 47 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne CCR3 48 43 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne CPT1A 15 40 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne PREP 46 34 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne CCKBR 16 40 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne EPHX2 37 43 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne MCHR1 17 40 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)Cc3ccccc3)C2)c1 ZINC000880549677 FE On-Demand Anodyne BIRC2 21 47 COc1ccc([C@H](CN(C)C)NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880549678 EF On-Demand Anodyne UTS2 36 40 COc1ccc([C@@H](CN(C)C)NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880549679 EF On-Demand Anodyne UTS2 36 40 CNC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549680 CD On-Demand Anodyne OPRL1 22 45 CNC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549680 CD On-Demand Anodyne BIRC2 63 36 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549683 GF On-Demand Anodyne LTA4H 50 37 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549683 GF On-Demand Anodyne HRH3 42 41 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549683 GF On-Demand Anodyne PSMB1 40 34 COc1cncc(NC(=O)NC[C@@H](O)Cc2ccccc2)c1 ZINC000880549704 DD On-Demand Anodyne ADRB1 44 34 COc1cncc(NC(=O)NC[C@@H](O)Cc2ccccc2)c1 ZINC000880549704 DD On-Demand Anodyne ADRB3 23 44 COc1cncc(NC(=O)NC[C@@H](O)Cc2ccccc2)c1 ZINC000880549704 DD On-Demand Anodyne ROCK2 27 42 COc1cncc(NC(=O)NC[C@@H](O)Cc2ccccc2)c1 ZINC000880549704 DD On-Demand Anodyne NAMPT 17 40 COc1cncc(NC(=O)NC[C@H](O)Cc2ccccc2)c1 ZINC000880549705 DD On-Demand Anodyne ADRB1 44 34 COc1cncc(NC(=O)NC[C@H](O)Cc2ccccc2)c1 ZINC000880549705 DD On-Demand Anodyne ADRB3 23 44 COc1cncc(NC(=O)NC[C@H](O)Cc2ccccc2)c1 ZINC000880549705 DD On-Demand Anodyne ROCK2 27 42 COc1cncc(NC(=O)NC[C@H](O)Cc2ccccc2)c1 ZINC000880549705 DD On-Demand Anodyne NAMPT 17 40 CCN1CCC(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)CC1 ZINC000880549706 FE On-Demand Anodyne CHRM1 16 42 CCN1CCC(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)CC1 ZINC000880549706 FE On-Demand Anodyne SIGMAR1 17 40 NC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880549710 DF On-Demand Anodyne KCNH2 41 40 NC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880549710 DF On-Demand Anodyne F10 17 48 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCCCN1CCCC1=O ZINC000880549723 FD On-Demand Anodyne TYRO3 19 44 COc1cncc(NC(=O)NC2(c3cccc(OC)c3)CC2)c1 ZINC000880549746 DF On-Demand Anodyne MTNR1A 18 42 COc1cncc(NC(=O)NC2(c3cccc(OC)c3)CC2)c1 ZINC000880549746 DF On-Demand Anodyne MTNR1B 25 42 COc1cncc(NC(=O)NC2(c3cccc(OC)c3)CC2)c1 ZINC000880549746 DF On-Demand Anodyne EPHX2 15 49 COC(=O)[C@@H]1CN(C(=O)c2cnc3cc[nH]c3c2)C[C@H]1c1ccccc1 ZINC000880549755 EF On-Demand Anodyne SLC6A3 18 47 CC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000880549757 EG On-Demand Anodyne PDE4A 25 42 CC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccc(OC)c(OC)c1 ZINC000880549757 EG On-Demand Anodyne ENPP1 71 36 COc1cncc(NC(=O)N2CC[C@@](CO)(c3ccccc3)C2)c1 ZINC000880549764 EE On-Demand Anodyne KCNA3 39 40 COc1cncc(NC(=O)N2CC[C@@](CO)(c3ccccc3)C2)c1 ZINC000880549764 EE On-Demand Anodyne EPHX2 35 48 COc1cncc(NC(=O)N2CC[C@](CO)(c3ccccc3)C2)c1 ZINC000880549765 EE On-Demand Anodyne KCNA3 39 40 COc1cncc(NC(=O)N2CC[C@](CO)(c3ccccc3)C2)c1 ZINC000880549765 EE On-Demand Anodyne EPHX2 35 48 CCN(CC(C)(C)C)C(=O)Nc1cncc(OC)c1 ZINC000880549768 CF On-Demand Anodyne ROCK2 16 41 COc1cncc(NC(=O)N2CCC(Oc3ccc(C#N)cc3F)CC2)c1 ZINC000880549775 FG On-Demand Mild PDGFRB 19 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(C#N)cc3F)CC2)c1 ZINC000880549775 FG On-Demand Mild EPHX2 17 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(C#N)cc3F)CC2)c1 ZINC000880549775 FG On-Demand Mild SCD1 23 49 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)CCC(F)(F)F)C2)c1 ZINC000880549780 FF On-Demand Anodyne EPHX2 40 38 COc1cncc(NC(=O)N[C@@H]2CCCN(C(=O)CCC(F)(F)F)C2)c1 ZINC000880549780 FF On-Demand Anodyne ETHR 47 36 COc1cncc(NC(=O)N(CCO)CC2CC2)c1 ZINC000880549790 CD On-Demand Anodyne ROCK2 15 41 O=C(COc1ccc2ccc(=O)oc2c1)NCc1cn(C2CCC2)nn1 ZINC000880549800 FD On-Demand Anodyne MAOA 52 40 COc1cncc(NC(=O)N2CCc3c(cccc3S(=O)(=O)N(C)C)C2)c1 ZINC000880549808 GD On-Demand Anodyne P2RY14 42 32 CCOC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549815 CE On-Demand Anodyne SLC6A1 43 32 CCOC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549815 CE On-Demand Anodyne CHRM4 17 42 O=C1CCCN1CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549816 DE On-Demand Anodyne HTR1A 19 44 O=C1CCCN1CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549816 DE On-Demand Anodyne HTR7 19 43 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549824 DG On-Demand Anodyne HTR1A 28 42 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549824 DG On-Demand Anodyne CHRM1 17 41 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549824 DG On-Demand Anodyne DRD2 15 40 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549824 DG On-Demand Anodyne CHRM4 17 41 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549824 DG On-Demand Anodyne HTR7 44 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne ELANE 29 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSD 23 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTRA_BOVIN 54 32 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CASP3 16 49 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne BMP1 26 54 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne KLK3 85 38 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSB 77 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne PAPA1_CARPA 86 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne TRY1_BOVIN 40 33 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CYSP_TRYCR 56 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne NTSR1 102 37 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne NTSR2 90 35 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSG 40 31 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSK 44 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSL 53 44 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne PGA 32 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne HLA-A 52 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne PREP 25 46 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CAPNS1 69 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne HLA-DRB1 46 33 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CELA2A 40 31 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne REN 66 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne SORT1 49 35 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CTSS 31 44 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CAPN1 104 49 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CASP1 26 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CAPN2 160 46 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CASP9 38 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne POLG_HCV1 17 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne NPR 73 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne GAG-PRO 54 36 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne XIAP 52 39 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne CASP10 38 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne PSMB5 56 47 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne F2RL1 64 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880549825 GF On-Demand Anodyne Q6PRC7_IXORI 23 40 OCCOCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549827 CD On-Demand Anodyne SLC6A1 33 41 COc1cncc(NC(=O)N2CCC[C@@H](CC(N)=O)CC2)c1 ZINC000880549830 DD On-Demand Anodyne PDGFRB 42 36 COc1cncc(NC(=O)N2CCC[C@H](CC(N)=O)CC2)c1 ZINC000880549831 DD On-Demand Anodyne PDGFRB 42 36 N#CCNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549833 CD On-Demand Mild CTSK 20 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880549851 FD On-Demand Anodyne CA14 23 52 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne BMP1 16 42 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne CA1 22 46 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne ROCK2 22 43 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne CA12 16 46 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne CA9 17 46 COc1cncc(NC(=O)NCCS(=O)(=O)CCc2ccccc2)c1 ZINC000880549868 FD On-Demand Anodyne NAMPT 40 40 COc1cncc(NC(=O)N2CCC(CNC(=O)C(F)(F)F)CC2)c1 ZINC000880549870 FE On-Demand Anodyne CACNA1I 48 33 COc1cncc(NC(=O)N2CCN(C[C@H](C)O)CC2)c1 ZINC000880549871 CC On-Demand Anodyne PDGFRB 45 37 COCCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549873 CG On-Demand Anodyne HTR1A 33 45 COCCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549873 CG On-Demand Anodyne DRD2 18 41 COCCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549873 CG On-Demand Anodyne DRD3 18 41 COc1cncc(NC(=O)N2CCc3cc(F)cc(C)c3C2)c1 ZINC000880549875 DG On-Demand Anodyne P2RY14 48 37 COc1cncc(NC(=O)N(C)CCc2cccc([N+](=O)[O-])c2)c1 ZINC000880549884 EF On-Demand Bother CACNA1C 41 36 COc1cncc(NC(=O)N(C)CCc2cccc([N+](=O)[O-])c2)c1 ZINC000880549884 EF On-Demand Bother CACNA1D 61 36 COc1cncc(NC(=O)N(C)CCc2cccc([N+](=O)[O-])c2)c1 ZINC000880549884 EF On-Demand Bother ROCK2 32 41 CN(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2cn(C3CCC3)nn2)c1 ZINC000880549889 GD On-Demand Anodyne CA14 15 42 COc1cncc(NC(=O)N2CCO[C@@]3(CCCOC3)C2)c1 ZINC000880549904 DD On-Demand Anodyne EPHX2 21 42 COc1cncc(NC(=O)N2CCO[C@]3(CCCOC3)C2)c1 ZINC000880549905 DD On-Demand Anodyne EPHX2 21 42 COC(=O)[C@@H]1CN(C(=O)c2cnc(CC3CC3)s2)C[C@H]1c1ccccc1 ZINC000880549906 FG On-Demand Anodyne SLC6A4 17 44 COC(=O)[C@@H]1CN(C(=O)c2cnc(CC3CC3)s2)C[C@H]1c1ccccc1 ZINC000880549906 FG On-Demand Anodyne SLC6A3 28 49 COC(=O)[C@@H]1CN(C(=O)c2cnc(CC3CC3)s2)C[C@H]1c1ccccc1 ZINC000880549906 FG On-Demand Anodyne PTR1 46 33 COc1cncc(NC(=O)N2CC(O)(c3ccccc3)C2)c1 ZINC000880549912 CD On-Demand Anodyne PDGFRB 28 40 CCOc1ccc([C@@H](O)C2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880549914 GG On-Demand Anodyne PDGFRB 43 37 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1cccc(Cl)c1 ZINC000880549916 EG On-Demand Anodyne ROCK1 15 46 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1cccc(Cl)c1 ZINC000880549917 EG On-Demand Anodyne ROCK1 15 46 CCCCNC(=O)NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549920 EE On-Demand Anodyne TPP2 41 39 COc1cncc(NC(=O)N[C@@H](CCO)c2ccc(Cl)cc2)c1 ZINC000880549923 EF On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N[C@@H](CCO)c2ccc(Cl)cc2)c1 ZINC000880549923 EF On-Demand Anodyne UTS2 54 42 COc1cncc(NC(=O)N[C@H](CCO)c2ccc(Cl)cc2)c1 ZINC000880549924 EF On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N[C@H](CCO)c2ccc(Cl)cc2)c1 ZINC000880549924 EF On-Demand Anodyne UTS2 54 42 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549933 GE On-Demand Anodyne LTA4H 51 39 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549933 GE On-Demand Anodyne CA7 21 41 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880549933 GE On-Demand Anodyne MEN1 17 44 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC1CCCC1 ZINC000880549956 DF On-Demand Anodyne SIGMAR1 17 40 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC1CCCC1 ZINC000880549956 DF On-Demand Anodyne BIRC2 45 36 COc1cncc(NC(=O)NC23C[C@H]4C[C@@H](CC(O)(C4)C2)C3)c1 ZINC000880549957 DE On-Demand Anodyne EPHX2 61 55 c1ccc2c(c1)CN(Cc1cscn1)C[C@H]1CCCN21 ZINC000880549969 CG On-Demand Anodyne SCN5A 43 36 COc1cncc(NC(=O)N2CCN(c3nccc4sccc34)CC2)c1 ZINC000880549974 FG On-Demand Anodyne PDGFRB 65 45 COC(=O)[C@@H]1CN(C(=O)c2cc(C)cnc2Cl)C[C@H]1c1ccccc1 ZINC000880549977 FG On-Demand Anodyne SLC6A3 20 45 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne HTR1A 30 46 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne DRD2 17 41 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne SLC6A1 101 42 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne CYSLTR2 42 31 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne HTR7 47 48 O=C(O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880549983 CE On-Demand Anodyne CYP2J2 47 33 CCCOc1ccc(OCC(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880550004 EE On-Demand Anodyne PLA2G4B 51 32 COc1cncc(NC(=O)N(C)CCCOCc2ccccc2)c1 ZINC000880550017 EG On-Demand Anodyne ROCK1 15 42 COc1cncc(NC(=O)N(C)CCCOCc2ccccc2)c1 ZINC000880550017 EG On-Demand Anodyne ROCK2 29 42 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne HTR1D 15 49 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne HTR1B 20 49 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne HTR2C 15 41 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne PDGFRB 53 44 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne FAAH 16 46 COc1cncc(NC(=O)N2CCN(c3cnccc3C)CC2)c1 ZINC000880550031 EE On-Demand Anodyne LIMK2 19 49 COc1cncc(NC(=O)N(CCNC(C)=O)Cc2ccsc2)c1 ZINC000880550040 EE On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880550047 DH On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880550047 DH On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880550047 DH On-Demand Anodyne CPT1A 113 38 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880550048 DH On-Demand Anodyne FKBP1A 48 35 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880550048 DH On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880550048 DH On-Demand Anodyne CPT1A 113 38 COc1cncc(NC(=O)N(C)Cc2ccc(C)o2)c1 ZINC000880550049 CF On-Demand Anodyne ROCK2 15 40 O=C(NCc1cn(C2CCC2)nn1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880550066 FG On-Demand Anodyne PDE4D 18 42 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1cccnc1 ZINC000880550077 EE On-Demand Anodyne CHRNA7 42 35 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1cccnc1 ZINC000880550077 EE On-Demand Anodyne PDE11A 43 38 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1cccnc1 ZINC000880550077 EE On-Demand Anodyne NAMPT 61 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1ccccc1 ZINC000880550080 EF On-Demand Anodyne SIGMAR1 24 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1ccccc1 ZINC000880550080 EF On-Demand Anodyne PDE11A 52 35 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCc1ccccc1 ZINC000880550080 EF On-Demand Anodyne TMPRSS11D 51 35 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1ccccc1 ZINC000880550082 DG On-Demand Anodyne DRD4 16 42 COc1cncc(NC(=O)N[C@H]2CC[C@@H](C(=O)N3CCCCC3)C2)c1 ZINC000880550088 EE On-Demand Anodyne EPHX2 44 44 COc1cncc(NC(=O)N[C@@H](CCO)Cc2ccccc2)c1 ZINC000880550089 DE On-Demand Anodyne ROCK1 15 43 COc1cncc(NC(=O)N[C@@H](CCO)Cc2ccccc2)c1 ZINC000880550089 DE On-Demand Anodyne FPR1 27 40 COc1cncc(NC(=O)N[C@H](CCO)Cc2ccccc2)c1 ZINC000880550090 DE On-Demand Anodyne ROCK1 15 43 COc1cncc(NC(=O)N[C@H](CCO)Cc2ccccc2)c1 ZINC000880550090 DE On-Demand Anodyne FPR1 27 40 COc1cncc(NC(=O)N2CC(OC)(c3ccccc3)C2)c1 ZINC000880550101 DE On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)N2CCC3(C2)Oc2ccccc2O3)c1 ZINC000880550109 EE On-Demand Anodyne NPY5R 31 40 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCCC1 ZINC000880550113 DE On-Demand Anodyne PREP 53 39 COc1cncc(NC(=O)NCc2cc(C)nc(N3CCCC3)c2)c1 ZINC000880550114 EF On-Demand Anodyne GALR2 41 33 CNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550124 CD On-Demand Anodyne OPRL1 21 52 CNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550124 CD On-Demand Anodyne BIRC2 80 35 COc1cncc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c1 ZINC000880550125 EE On-Demand Anodyne CCR3 31 41 COc1cncc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c1 ZINC000880550125 EE On-Demand Anodyne EPHX2 52 43 COc1cncc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c1 ZINC000880550125 EE On-Demand Anodyne CXCR3 23 45 COc1cncc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c1 ZINC000880550125 EE On-Demand Anodyne MCHR1 16 47 COc1cncc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c1 ZINC000880550125 EE On-Demand Anodyne HPGDS 41 51 COC(=O)[C@@H]1CN(C(=O)c2cc(C)co2)C[C@H]1c1ccccc1 ZINC000880550129 DF On-Demand Anodyne SLC6A4 17 43 COC(=O)[C@@H]1CN(C(=O)c2cc(C)co2)C[C@H]1c1ccccc1 ZINC000880550129 DF On-Demand Anodyne SLC6A3 34 40 CCCN(CCN1CCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550134 DE On-Demand Anodyne DRD4 41 32 CCCN(CCN1CCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550134 DE On-Demand Anodyne CASR 45 46 CCCN(CCN1CCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550134 DE On-Demand Anodyne ROCK2 21 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCC1 ZINC000880550136 CE On-Demand Anodyne PREP 60 40 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne HTR1A 30 57 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne HTR1B 18 57 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne PDGFRB 50 43 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne HTR7 25 44 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne KCNQ2 51 36 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne NPY2R 72 36 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne SSTR1 15 40 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne FAAH 18 43 COc1cncc(NC(=O)N2CCCN(c3ccccc3F)CC2)c1 ZINC000880550140 EF On-Demand Anodyne RBP4 20 44 COC(=O)[C@@H]1CN(C(=O)c2ncsc2C2CC2)C[C@H]1c1ccccc1 ZINC000880550167 FG On-Demand Anodyne SLC6A3 26 41 CCOC(=O)C1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880550179 DE On-Demand Anodyne EPHX2 41 38 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC1CC1 ZINC000880550185 CD On-Demand Anodyne DRD4 15 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NC1CC1 ZINC000880550185 CD On-Demand Anodyne SIGMAR1 16 40 COCCCNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550188 DD On-Demand Anodyne DRD4 23 44 COCCCNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550188 DD On-Demand Anodyne DRD3 43 46 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550194 DF On-Demand Anodyne HTR1A 27 44 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550194 DF On-Demand Anodyne DRD2 19 40 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550194 DF On-Demand Anodyne DRD3 22 45 COc1cncc(NC(=O)NC2CCN(c3nccs3)CC2)c1 ZINC000880550215 EE On-Demand Anodyne EPHX2 43 38 COc1cncc(NC(=O)N2C[C@@H](O)C[C@@H]2c2ccccc2C(F)(F)F)c1 ZINC000880550229 GG On-Demand Anodyne RBP4 84 39 COc1cncc(NC(=O)N2C[C@@H](O)C[C@H]2c2ccccc2C(F)(F)F)c1 ZINC000880550230 GG On-Demand Anodyne RBP4 84 39 COc1cncc(NC(=O)N2C[C@H](O)C[C@@H]2c2ccccc2C(F)(F)F)c1 ZINC000880550231 GG On-Demand Anodyne RBP4 84 39 COc1cncc(NC(=O)N2C[C@H](O)C[C@H]2c2ccccc2C(F)(F)F)c1 ZINC000880550232 GG On-Demand Anodyne RBP4 84 39 COc1cncc(NC(=O)N2CCc3cccc(F)c3C2)c1 ZINC000880550236 DF On-Demand Anodyne P2RY14 50 37 COc1cncc(NC(=O)N2CCC(N3CCc4ccccc43)CC2)c1 ZINC000880550237 FG On-Demand Anodyne AVPR1A 18 43 COc1cncc(NC(=O)N2CCC(N3CCc4ccccc43)CC2)c1 ZINC000880550237 FG On-Demand Anodyne SCD1 35 59 COc1cncc(NC(=O)N2CCN(c3ccc(F)c(OC)c3)CC2)c1 ZINC000880550247 FF On-Demand Anodyne PDGFRB 57 43 COc1cncc(NC(=O)N2CCN(c3ccc(F)c(OC)c3)CC2)c1 ZINC000880550247 FF On-Demand Anodyne SSTR1 27 40 COc1cncc(NC(=O)N2CCN(c3ccc(F)c(OC)c3)CC2)c1 ZINC000880550247 FF On-Demand Anodyne FAAH 15 40 COc1cncc(NC(=O)N2CCN(c3ccc(F)c(OC)c3)CC2)c1 ZINC000880550247 FF On-Demand Anodyne RBP4 18 41 O=C(NCc1cn(C2CCC2)nn1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880550250 ED On-Demand Anodyne PLD1 46 38 O=C(NCc1cn(C2CCC2)nn1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880550250 ED On-Demand Anodyne PLD2 45 38 COc1cncc(NC(=O)N2CCC(c3ccc(F)c(F)c3)CC2)c1 ZINC000880550252 EH On-Demand Anodyne CACNA1H 54 39 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550266 GF On-Demand Anodyne ADRB2 15 43 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550266 GF On-Demand Anodyne HTR1A 30 40 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550266 GF On-Demand Anodyne ABCB1 68 41 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550267 GF On-Demand Anodyne ADRB2 15 43 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550267 GF On-Demand Anodyne HTR1A 30 40 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550267 GF On-Demand Anodyne ABCB1 68 41 COc1cncc(NC(=O)N2CC[C@@H](c3ccccn3)C2)c1 ZINC000880550271 CF On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N2CC[C@@H](c3ccccn3)C2)c1 ZINC000880550271 CF On-Demand Anodyne SMO 15 43 COc1cncc(NC(=O)N2CC[C@H](c3ccccn3)C2)c1 ZINC000880550272 CF On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N2CC[C@H](c3ccccn3)C2)c1 ZINC000880550272 CF On-Demand Anodyne SMO 15 43 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCC(=O)N1CCCC1 ZINC000880550273 FD On-Demand Anodyne PREP 48 40 COc1cncc(NC(=O)N(C)[C@H](C)CO)c1 ZINC000880550277 BC On-Demand Anodyne NPY5R 34 44 COc1cncc(NC(=O)N(C)[C@@H](C)CO)c1 ZINC000880550278 BC On-Demand Anodyne NPY5R 34 44 COc1cncc(NC(=O)N2CCC[C@](CO)(Cc3ccccc3)C2)c1 ZINC000880550285 FF On-Demand Anodyne EPHX2 27 44 COc1cncc(NC(=O)N2CCC[C@](CO)(Cc3ccccc3)C2)c1 ZINC000880550285 FF On-Demand Anodyne SLC12A5 56 37 COc1cncc(NC(=O)N2CCC[C@@](CO)(Cc3ccccc3)C2)c1 ZINC000880550287 FF On-Demand Anodyne EPHX2 27 44 COc1cncc(NC(=O)N2CCC[C@@](CO)(Cc3ccccc3)C2)c1 ZINC000880550287 FF On-Demand Anodyne SLC12A5 56 37 COc1cncc(NC(=O)NCCN2CCN(C)C(C)(C)C2)c1 ZINC000880550291 DD On-Demand Anodyne DRD4 44 33 N#CCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550292 CG On-Demand Mild HTR7 16 41 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550296 DD On-Demand Anodyne HTR1A 22 42 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550296 DD On-Demand Anodyne SLC6A1 63 36 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550296 DD On-Demand Anodyne HTR7 45 42 COc1cncc(NC(=O)N2CC[C@](CO)(Cc3ccc(F)cc3)C2)c1 ZINC000880550298 FF On-Demand Anodyne S1PR2 28 42 COc1cncc(NC(=O)N2CC[C@@](CO)(Cc3ccc(F)cc3)C2)c1 ZINC000880550299 FF On-Demand Anodyne S1PR2 28 42 COC(=O)[C@@H]1CN(C(=O)c2cccn3nccc23)C[C@H]1c1ccccc1 ZINC000880550300 EE On-Demand Anodyne SLC6A3 15 46 COC(=O)[C@@H]1CN(C(=O)c2nccnc2SC)C[C@H]1c1ccccc1 ZINC000880550301 FE On-Demand Anodyne SLC6A3 18 46 COc1cncc(NC(=O)N2CC[C@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550306 FG On-Demand Anodyne SIGMAR1 27 40 COc1cncc(NC(=O)N2CC[C@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550306 FG On-Demand Anodyne NPFFR2 30 42 COc1cncc(NC(=O)N2CC[C@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550306 FG On-Demand Anodyne FAAH 29 60 COc1cncc(NC(=O)N2CC[C@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550306 FG On-Demand Anodyne CCR8 42 42 COc1cncc(NC(=O)N2CC[C@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550306 FG On-Demand Anodyne NPFFR1 40 42 COc1cncc(NC(=O)N2CC[C@@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550307 FG On-Demand Anodyne SIGMAR1 27 40 COc1cncc(NC(=O)N2CC[C@@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550307 FG On-Demand Anodyne NPFFR2 30 42 COc1cncc(NC(=O)N2CC[C@@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550307 FG On-Demand Anodyne FAAH 29 60 COc1cncc(NC(=O)N2CC[C@@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550307 FG On-Demand Anodyne CCR8 42 42 COc1cncc(NC(=O)N2CC[C@@]3(CCN(Cc4ccccc4)C3)C2)c1 ZINC000880550307 FG On-Demand Anodyne NPFFR1 40 42 c1ccc2c(c1)CN(CCc1ccncc1)C[C@H]1CCCN21 ZINC000880550320 CG On-Demand Anodyne SIGMAR1 17 42 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCCCC1 ZINC000880550327 EF On-Demand Anodyne PREP 53 39 COc1cncc(NC(=O)NC2CCN(C(=O)c3cc(Cl)c[nH]3)CC2)c1 ZINC000880550328 GE On-Demand Anodyne EPHX2 39 44 COc1cncc(NC(=O)N(C)Cc2ccccc2N(C)C)c1 ZINC000880550373 DF On-Demand Anodyne ROCK2 19 42 COc1cncc(NC(=O)NCc2ccc(C[S@@](C)=O)cc2)c1 ZINC000880550375 EE On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)NCc2ccc(C[S@@](C)=O)cc2)c1 ZINC000880550375 EE On-Demand Anodyne NAMPT 30 40 COc1cncc(NC(=O)NCc2ccc(C[S@](C)=O)cc2)c1 ZINC000880550376 EE On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)NCc2ccc(C[S@](C)=O)cc2)c1 ZINC000880550376 EE On-Demand Anodyne NAMPT 30 40 O[C@@H](CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccc(F)cc1 ZINC000880550385 EG On-Demand Anodyne SLC6A3 31 45 O[C@@H](CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccc(F)cc1 ZINC000880550385 EG On-Demand Anodyne SLC18A3 15 40 O[C@H](CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccc(F)cc1 ZINC000880550386 EG On-Demand Anodyne SLC6A3 31 45 O[C@H](CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccc(F)cc1 ZINC000880550386 EG On-Demand Anodyne SLC18A3 15 40 CCNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550387 CD On-Demand Anodyne DRD4 20 40 CCNC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550387 CD On-Demand Anodyne TPP2 41 37 CN(C)C(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550392 EG On-Demand Anodyne DRD2 15 45 CN(C)C(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550392 EG On-Demand Anodyne ACHE 15 41 COc1cncc(NC(=O)NC[C@@H]2CC(c3ccc(C)cc3)=NO2)c1 ZINC000880550397 EF On-Demand Anodyne LUCI_PHOPY 66 42 COc1cncc(NC(=O)NC[C@H]2CC(c3ccc(C)cc3)=NO2)c1 ZINC000880550398 EF On-Demand Anodyne LUCI_PHOPY 66 42 COc1cncc(NC(=O)N2CCC3(CCO3)CC2)c1 ZINC000880550406 CD On-Demand Anodyne EPHX2 21 41 c1ccc2c(c1)CN(CCN1CCCCC1)C[C@H]1CCCN21 ZINC000880550407 CF On-Demand Anodyne SIGMAR1 23 43 CCCCN(Cc1ccccc1O)C(=O)Nc1cncc(OC)c1 ZINC000880550414 EH On-Demand Clean INHA 73 37 COc1cncc(NC(=O)N2CC[C@@](F)(c3ccccc3)C2)c1 ZINC000880550417 DG On-Demand Anodyne EPHX2 36 41 COc1cncc(NC(=O)N2CC[C@](F)(c3ccccc3)C2)c1 ZINC000880550418 DG On-Demand Anodyne EPHX2 36 41 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCCC1 ZINC000880550439 EF On-Demand Anodyne SLC6A1 50 34 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCCC1 ZINC000880550439 EF On-Demand Anodyne PREP 48 37 COCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550443 CF On-Demand Anodyne HTR1A 31 46 COCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550443 CF On-Demand Anodyne DRD2 18 42 COCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550443 CF On-Demand Anodyne DRD3 19 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne CCR3 30 41 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne CHRNA7 25 43 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne CPT1A 109 45 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne CPT2 46 38 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne EPHX2 48 48 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550447 FD On-Demand Anodyne MCHR1 18 41 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne CCR3 30 41 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne CHRNA7 25 43 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne CPT1A 109 45 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne CPT2 46 38 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne EPHX2 48 48 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)COc3ccccc3)C2)c1 ZINC000880550448 FD On-Demand Anodyne MCHR1 18 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCCCN1CCCCCC1=O ZINC000880550453 GE On-Demand Anodyne TYRO3 18 41 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne HTR1A 20 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne DRD2 19 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne HTR1D 23 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne HTR1B 19 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne NPY1R 30 41 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne CCR3 54 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880550471 EH On-Demand Anodyne MCHR1 32 41 COc1cncc(NC(=O)N(C)CCCN2CCCC2)c1 ZINC000880550476 CE On-Demand Anodyne CHRNA7 17 40 COc1cncc(NC(=O)NCc2ccc(OC3CCN(C)CC3)cc2)c1 ZINC000880550484 FF On-Demand Anodyne CCR3 49 42 COc1cncc(NC(=O)NCc2ccc(OC3CCN(C)CC3)cc2)c1 ZINC000880550484 FF On-Demand Anodyne EPHX2 28 41 COc1cncc(NC(=O)NCc2ccc(OC3CCN(C)CC3)cc2)c1 ZINC000880550484 FF On-Demand Anodyne NAMPT 47 38 CC[C@H](C)NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550492 DE On-Demand Anodyne TPP2 40 33 CC[C@H](C)NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550492 DE On-Demand Anodyne BIRC2 68 34 COc1cncc(NC(=O)NCc2ncccc2N(C)C)c1 ZINC000880550505 DD On-Demand Anodyne ROCK2 24 44 COC(=O)[C@@H]1CN(C(=O)[C@@H]2CCc3nncn3CC2)C[C@H]1c1ccccc1 ZINC000880550507 FD On-Demand Anodyne SLC6A3 17 47 COC(=O)[C@@H]1CN(C(=O)[C@H]2CCc3nncn3CC2)C[C@H]1c1ccccc1 ZINC000880550508 FD On-Demand Anodyne SLC6A3 17 47 COC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550509 CD On-Demand Anodyne HTR1A 23 43 COC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550509 CD On-Demand Anodyne DRD2 15 40 COC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550509 CD On-Demand Anodyne OPRL1 17 45 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880550511 EE On-Demand Anodyne EPHX2 33 42 COc1cncc(NC(=O)NCc2ccncc2OCCCN(C)C)c1 ZINC000880550517 FE On-Demand Anodyne ROCK2 30 44 O[C@H](COc1ccccc1)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550520 EF On-Demand Anodyne ABCB1 65 42 O[C@@H](COc1ccccc1)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550521 EF On-Demand Anodyne ABCB1 65 42 COc1cncc(NC(=O)NCc2ccc(OC)nc2OC)c1 ZINC000880550526 DD On-Demand Anodyne ROCK2 15 44 COc1cncc(NC(=O)N(C)C2C[C@@H]3CC[C@H](C2)N3C)c1 ZINC000880550531 DE On-Demand Anodyne GLRA1 42 36 COC(=O)[C@@H]1CN(C(=O)c2nnn(C)n2)C[C@H]1c1ccccc1 ZINC000880550544 DC On-Demand Anodyne SLC6A3 39 52 COc1cncc(NC(=O)N[C@@H](CCSC)C(=O)N(C)C)c1 ZINC000880550547 ED On-Demand Anodyne FPR1 29 42 COc1cncc(NC(=O)NC2CCC(NC(C)=O)CC2)c1 ZINC000880550550 DD On-Demand Anodyne EPHX2 48 38 CCCN(CCN1CCCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550557 DF On-Demand Anodyne DRD4 41 32 CCCN(CCN1CCCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550557 DF On-Demand Anodyne CASR 42 46 CCCN(CCN1CCCCC1)C(=O)Nc1cncc(OC)c1 ZINC000880550557 DF On-Demand Anodyne ROCK2 21 40 COC(=O)[C@@H]1CN(C(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)C[C@H]1c1ccccc1 ZINC000880550572 GD On-Demand Anodyne SLC6A4 30 47 COC(=O)[C@@H]1CN(C(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)C[C@H]1c1ccccc1 ZINC000880550572 GD On-Demand Anodyne SLC6A3 53 54 COc1cncc(NC(=O)NC2CCN(C(=O)C(C)C)CC2)c1 ZINC000880550578 DD On-Demand Anodyne EPHX2 54 57 COc1cncc(NC(=O)NC2CCN(C(=O)C(C)C)CC2)c1 ZINC000880550578 DD On-Demand Anodyne CXCR3 15 40 COC(=O)[C@@H]1CN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C[C@H]1c1ccccc1 ZINC000880550584 GF On-Demand Anodyne SLC6A4 26 45 COC(=O)[C@@H]1CN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C[C@H]1c1ccccc1 ZINC000880550584 GF On-Demand Anodyne SLC6A3 44 42 COC(=O)[C@@H]1CN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C[C@H]1c1ccccc1 ZINC000880550585 GF On-Demand Anodyne SLC6A4 26 45 COC(=O)[C@@H]1CN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C[C@H]1c1ccccc1 ZINC000880550585 GF On-Demand Anodyne SLC6A3 44 42 COc1cncc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)c1 ZINC000880550588 EG On-Demand Anodyne EPHX2 40 41 COc1cncc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)c1 ZINC000880550588 EG On-Demand Anodyne TRPM8 33 51 COc1cncc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)c1 ZINC000880550589 EG On-Demand Anodyne EPHX2 40 41 COc1cncc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)c1 ZINC000880550589 EG On-Demand Anodyne TRPM8 33 51 COc1cncc(NC(=O)N[C@@H]2C[C@@H](c3cccc(F)c3)C2)c1 ZINC000880550594 DG On-Demand Anodyne CCR3 21 41 COc1cncc(NC(=O)N2CCC(C#N)(c3ccccn3)CC2)c1 ZINC000880550596 EF On-Demand Mild PDGFRB 42 38 COc1cncc(NC(=O)N(C)Cc2cnc(C(C)C)nc2)c1 ZINC000880550602 DF On-Demand Anodyne ROCK2 15 42 O=C1CCC(=O)N1CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550634 DD On-Demand Anodyne HTR1A 18 44 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550637 EF On-Demand Anodyne HTR1A 32 41 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550637 EF On-Demand Anodyne DRD2 27 53 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550637 EF On-Demand Anodyne DRD3 31 43 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCOCC3)C2)c1 ZINC000880550673 ED On-Demand Anodyne CCR3 17 56 COc1cncc(NC(=O)N2CCC[C@H](CN3CCOCC3)C2)c1 ZINC000880550674 ED On-Demand Anodyne CCR3 17 56 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550677 GF On-Demand Anodyne ADRB2 16 45 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550677 GF On-Demand Anodyne ADRB1 45 45 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550677 GF On-Demand Anodyne ACOX1 55 39 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550677 GF On-Demand Anodyne ABCB1 63 42 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550678 GF On-Demand Anodyne ADRB2 16 45 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550678 GF On-Demand Anodyne ADRB1 45 45 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550678 GF On-Demand Anodyne ACOX1 55 39 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550678 GF On-Demand Anodyne ABCB1 63 42 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne HTR1A 42 45 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne DRD2 38 43 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne DRD4 22 49 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne DRD3 60 50 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne HTR7 41 38 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550681 CD On-Demand Anodyne MTNR1A 16 42 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550682 DF On-Demand Anodyne HTR1A 27 42 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550682 DF On-Demand Anodyne CHRM1 16 41 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550682 DF On-Demand Anodyne SLC6A1 72 36 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550682 DF On-Demand Anodyne CHRM4 16 41 CC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550723 CE On-Demand Anodyne SLC6A1 48 33 CC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550723 CE On-Demand Anodyne HTR7 30 41 COc1cncc(NC(=O)NCc2ccc(C)n(C)c2=O)c1 ZINC000880550726 DD On-Demand Anodyne P2RX7 47 47 COCCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880550728 EF On-Demand Anodyne PDGFRB 16 44 COCCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880550728 EF On-Demand Anodyne ROCK2 28 44 CCS(=O)(=O)N1CCN(C(=O)Nc2cncc(OC)c2)[C@H](C)C1 ZINC000880550729 EC On-Demand Anodyne LIMK2 24 40 CCCC[C@@H](C)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880550730 CG On-Demand Anodyne NPY5R 31 41 CCCC[C@H](C)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880550731 CG On-Demand Anodyne NPY5R 31 41 COc1cncc(NC(=O)N(Cc2ccccc2OC)OC)c1 ZINC000880550732 DF On-Demand Anodyne TSPO 46 39 COc1cncc(NC(=O)N[C@@H]2CC(=O)N(C3CC3)[C@H]2c2cccnc2)c1 ZINC000880550749 FE On-Demand Anodyne CHRNA7 21 44 COc1cncc(NC(=O)N(CCO)Cc2cccnc2Cl)c1 ZINC000880550759 EE On-Demand Anodyne ROCK2 16 44 COc1cncc(NC(=O)N2CCC[C@@H]2c2nc(C)no2)c1 ZINC000880550763 DE On-Demand Anodyne CPT1A 55 41 COc1cncc(NC(=O)N2CCC[C@H]2c2nc(C)no2)c1 ZINC000880550766 DE On-Demand Anodyne CPT1A 55 41 COc1cncc(NC(=O)NCCN2CC=CCC2)c1 ZINC000880550773 CD On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NCCN2CC=CCC2)c1 ZINC000880550773 CD On-Demand Anodyne CCR3 21 40 COc1cncc(NC(=O)N2CCC[C@@H]2C(=O)OC(C)(C)C)c1 ZINC000880550775 DE On-Demand Anodyne FKBP1A 49 39 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3F)C2)c1 ZINC000880550776 EF On-Demand Anodyne NPY2R 43 34 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3F)C2)c1 ZINC000880550776 EF On-Demand Anodyne CCR3 69 41 COc1cncc(NC(=O)N(C[C@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550777 FF On-Demand Anodyne ADRB2 27 46 COc1cncc(NC(=O)N(C[C@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550777 FF On-Demand Anodyne ADRB1 36 42 COc1cncc(NC(=O)N(C[C@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550777 FF On-Demand Anodyne ADRB3 30 42 COc1cncc(NC(=O)N(C[C@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550777 FF On-Demand Anodyne ABCB1 17 43 COc1cncc(NC(=O)N(C[C@@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550778 FF On-Demand Anodyne ADRB2 27 46 COc1cncc(NC(=O)N(C[C@@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550778 FF On-Demand Anodyne ADRB1 36 42 COc1cncc(NC(=O)N(C[C@@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550778 FF On-Demand Anodyne ADRB3 30 42 COc1cncc(NC(=O)N(C[C@@H](O)COc2ccccc2)C(C)C)c1 ZINC000880550778 FF On-Demand Anodyne ABCB1 17 43 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3F)C2)c1 ZINC000880550779 EF On-Demand Anodyne NPY2R 43 34 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3F)C2)c1 ZINC000880550779 EF On-Demand Anodyne CCR3 69 41 C[C@H]1CCCCN1C(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550782 EF On-Demand Anodyne PREP 48 41 C[C@@H]1CCCCN1C(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550785 EF On-Demand Anodyne PREP 48 41 COc1cncc(NC(=O)N2CCC(COc3ccc(Cl)nc3)CC2)c1 ZINC000880550788 GG On-Demand Anodyne PDGFRB 49 37 COc1cncc(NC(=O)NCCCc2cccc(C)n2)c1 ZINC000880550792 DF On-Demand Anodyne MTNR1A 50 41 COc1cncc(NC(=O)NCCCc2cccc(C)n2)c1 ZINC000880550792 DF On-Demand Anodyne MTNR1B 48 41 COc1cncc(NC(=O)NCC2(c3ccccn3)CCC2)c1 ZINC000880550813 DF On-Demand Anodyne NMBR 69 43 COc1cncc(NC(=O)NCC2(c3ccccn3)CCC2)c1 ZINC000880550813 DF On-Demand Anodyne SLC6A9 15 40 COc1cncc(NC(=O)NCC2(c3ccccn3)CCC2)c1 ZINC000880550813 DF On-Demand Anodyne GRPR 38 43 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)C(F)(F)F)C2)c1 ZINC000880550822 FE On-Demand Anodyne CCR3 18 45 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)C(F)(F)F)C2)c1 ZINC000880550824 FE On-Demand Anodyne CCR3 18 45 COC(=O)[C@@H]1CN(C(=O)c2cnc(C(C)C)nc2C)C[C@H]1c1ccccc1 ZINC000880550834 FF On-Demand Anodyne SLC6A3 17 43 COc1cncc(NC(=O)N2CCC(F)(c3ccccc3)CC2)c1 ZINC000880550842 EH On-Demand Anodyne CACNA1H 40 35 COc1cncc(NC(=O)N2CCC(F)(c3ccccc3)CC2)c1 ZINC000880550842 EH On-Demand Anodyne S1PR2 28 41 COc1cncc(NC(=O)N[C@H]2c3ccccc3C[C@H]2O)c1 ZINC000880550843 CD On-Demand Anodyne PLM1_PLAFA 41 39 COc1cncc(NC(=O)N[C@H]2c3ccccc3C[C@H]2O)c1 ZINC000880550843 CD On-Demand Anodyne PLM2_PLAFA 83 39 COc1cncc(NC(=O)N[C@@H]2c3ccccc3C[C@H]2O)c1 ZINC000880550845 CD On-Demand Anodyne PLM1_PLAFA 41 39 COc1cncc(NC(=O)N[C@@H]2c3ccccc3C[C@H]2O)c1 ZINC000880550845 CD On-Demand Anodyne PLM2_PLAFA 83 39 COc1cncc(NC(=O)N[C@@H]2c3ccccc3C[C@@H]2O)c1 ZINC000880550846 CD On-Demand Anodyne PLM1_PLAFA 41 39 COc1cncc(NC(=O)N[C@@H]2c3ccccc3C[C@@H]2O)c1 ZINC000880550846 CD On-Demand Anodyne PLM2_PLAFA 83 39 C#CCn1ccc(CN(CC)C(=O)Nc2cncc(OC)c2)n1 ZINC000880550857 DD On-Demand Mild ROCK2 19 43 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne RAF1 25 52 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne TAAR1 29 40 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne RIPK1 20 40 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne IMDH_CRYPV 55 40 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne KCNK3 49 37 COc1cncc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880550860 DF On-Demand Anodyne KCNK9 41 37 COc1cncc(NC(=O)NC[C@]2(CO)C[C@@H]2c2ccccc2)c1 ZINC000880550861 EE On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N2CCC[C@](C)(O)CC2)c1 ZINC000880550862 CD On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CCC[C@@](C)(O)CC2)c1 ZINC000880550863 CD On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)NC[C@@]2(CO)C[C@H]2c2ccccc2)c1 ZINC000880550864 EE On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)NC[C@@]2(CO)C[C@@H]2c2ccccc2)c1 ZINC000880550868 EE On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)NC[C@]2(CO)C[C@H]2c2ccccc2)c1 ZINC000880550873 EE On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N2CC(O)(c3ccc(Cl)cc3)C2)c1 ZINC000880550892 EE On-Demand Anodyne PDGFRB 25 41 COc1cncc(NC(=O)N2CC(O)(c3ccc(Cl)cc3)C2)c1 ZINC000880550892 EE On-Demand Anodyne FAAH 15 43 COc1cncc(NC(=O)N2CC(O)(c3ccc(Cl)cc3)C2)c1 ZINC000880550892 EE On-Demand Anodyne SCN10A 23 43 COc1cncc(NC(=O)NCc2noc3c2CCCC3)c1 ZINC000880550902 DE On-Demand Anodyne PANC 41 32 N#Cc1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880550903 DH On-Demand Mild SIGMAR1 17 40 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne PDGFRB 15 40 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne KCNA3 45 38 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne NMBR 43 34 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne MTNR1A 37 42 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne MTNR1B 38 43 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne ROCK2 30 46 COc1cncc(NC(=O)NCC2(c3cccc(OC)c3)CC2)c1 ZINC000880550904 EF On-Demand Anodyne SOAT1 22 52 COc1cncc(NC(=O)N2CCC(c3noc4cc(F)ccc34)CC2)c1 ZINC000880550905 FH On-Demand Anodyne DRD2 16 53 COc1cncc(NC(=O)N2CCC(c3noc4cc(F)ccc34)CC2)c1 ZINC000880550905 FH On-Demand Anodyne HTR2A 27 49 COc1cncc(NC(=O)N2CCC(c3noc4cc(F)ccc34)CC2)c1 ZINC000880550905 FH On-Demand Anodyne HTR7 26 43 COc1cncc(NC(=O)N2CCCC[C@H]2c2n[nH]c(C(C)C)n2)c1 ZINC000880550906 EG On-Demand Anodyne CPT1A 44 35 COc1cncc(NC(=O)N2CCCC[C@@H]2c2n[nH]c(C(C)C)n2)c1 ZINC000880550907 EG On-Demand Anodyne CPT1A 44 35 CCOC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550913 CE On-Demand Anodyne ACE 15 40 CCOC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880550913 CE On-Demand Anodyne TPP2 51 37 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550918 ED On-Demand Anodyne OPRL1 17 42 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550918 ED On-Demand Anodyne XIAP 41 33 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550918 ED On-Demand Anodyne BIRC3 44 32 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550918 ED On-Demand Anodyne BIRC2 90 38 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550919 ED On-Demand Anodyne OPRL1 17 42 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550919 ED On-Demand Anodyne XIAP 41 33 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550919 ED On-Demand Anodyne BIRC3 44 32 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)C(=O)N(C)C ZINC000880550919 ED On-Demand Anodyne BIRC2 90 38 COc1cncc(NC(=O)NCCCn2ccnc2C)c1 ZINC000880550938 CD On-Demand Anodyne CCR3 16 40 COc1cncc(NC(=O)NCCCn2ccnc2C)c1 ZINC000880550938 CD On-Demand Anodyne QPCT 71 48 COc1cncc(NC(=O)NCc2ccncc2OCC(F)(F)F)c1 ZINC000880550945 FF On-Demand Anodyne ROCK2 19 43 COc1cncc(NC(=O)NC[C@@H]2CC(c3ccc(OC)c(F)c3)=NO2)c1 ZINC000880550946 FF On-Demand Anodyne MIF 17 41 COc1cncc(NC(=O)NC[C@@H]2CC(c3ccc(OC)c(F)c3)=NO2)c1 ZINC000880550946 FF On-Demand Anodyne LUCI_PHOPY 48 41 COc1cncc(NC(=O)NC[C@H]2CC(c3ccc(OC)c(F)c3)=NO2)c1 ZINC000880550947 FF On-Demand Anodyne MIF 17 41 COc1cncc(NC(=O)NC[C@H]2CC(c3ccc(OC)c(F)c3)=NO2)c1 ZINC000880550947 FF On-Demand Anodyne LUCI_PHOPY 48 41 COc1cncc(NC(=O)N2CCN(C)[C@@H](Cc3ccccc3)C2)c1 ZINC000880550949 EE On-Demand Anodyne PDGFRB 43 38 COc1cncc(NC(=O)N2CCN(C)[C@@H](Cc3ccccc3)C2)c1 ZINC000880550949 EE On-Demand Anodyne CCR3 24 48 COc1cncc(NC(=O)N2CCN(C)[C@@H](Cc3ccccc3)C2)c1 ZINC000880550949 EE On-Demand Anodyne FAAH 18 44 COc1cncc(NC(=O)N2CCN(C)[C@H](Cc3ccccc3)C2)c1 ZINC000880550950 EE On-Demand Anodyne PDGFRB 43 38 COc1cncc(NC(=O)N2CCN(C)[C@H](Cc3ccccc3)C2)c1 ZINC000880550950 EE On-Demand Anodyne CCR3 24 48 COc1cncc(NC(=O)N2CCN(C)[C@H](Cc3ccccc3)C2)c1 ZINC000880550950 EE On-Demand Anodyne FAAH 18 44 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne HTR1A 45 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne DRD2 35 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne DRD4 33 42 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne ADRA1A 18 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne DRD3 40 39 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551045 FG On-Demand Anodyne KCNQ2 40 34 CC[C@@](C)(O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880551048 EG On-Demand Anodyne ROCK2 22 45 COc1cncc(NC(=O)N2CCC(n3c(C)nc4ccccc43)CC2)c1 ZINC000880551049 FH On-Demand Anodyne CCR5 18 44 COc1cncc(NC(=O)N2CCC(n3c(C)nc4ccccc43)CC2)c1 ZINC000880551049 FH On-Demand Anodyne CALCRL 23 41 COc1cncc(NC(=O)N2CCC(n3c(C)nc4ccccc43)CC2)c1 ZINC000880551049 FH On-Demand Anodyne FPR2 23 44 COc1cncc(NC(=O)N2CCC(n3c(C)nc4ccccc43)CC2)c1 ZINC000880551049 FH On-Demand Anodyne SCD1 15 43 COc1cncc(NC(=O)N2CCC(n3c(C)nc4ccccc43)CC2)c1 ZINC000880551049 FH On-Demand Anodyne SMO 20 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccc(F)cc3)C2=O)c1 ZINC000880551051 FE On-Demand Anodyne CCR3 126 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccc(F)cc3)C2=O)c1 ZINC000880551052 FE On-Demand Anodyne CCR3 126 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccc(C)cc3)C2=O)c1 ZINC000880551053 FE On-Demand Anodyne CCKAR 17 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccc(C)cc3)C2=O)c1 ZINC000880551053 FE On-Demand Anodyne CCKBR 20 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccc(C)cc3)C2=O)c1 ZINC000880551054 FE On-Demand Anodyne CCKAR 17 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccc(C)cc3)C2=O)c1 ZINC000880551054 FE On-Demand Anodyne CCKBR 20 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1c(F)cccc1F ZINC000880551062 FG On-Demand Anodyne DRD4 17 42 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1cccnc1Cl ZINC000880551063 FG On-Demand Anodyne G2YM83_BOTF4 53 35 COc1cncc(NC(=O)N2CC[C@@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551069 EG On-Demand Anodyne CACNA1H 33 41 COc1cncc(NC(=O)N2CC[C@@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551069 EG On-Demand Anodyne S1PR2 29 43 COc1cncc(NC(=O)N2CC[C@@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551069 EG On-Demand Anodyne EPHX2 36 41 COc1cncc(NC(=O)N2CC[C@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551070 EG On-Demand Anodyne CACNA1H 33 41 COc1cncc(NC(=O)N2CC[C@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551070 EG On-Demand Anodyne S1PR2 29 43 COc1cncc(NC(=O)N2CC[C@](C)(c3ccc(F)cc3)C2)c1 ZINC000880551070 EG On-Demand Anodyne EPHX2 36 41 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c1 ZINC000880551072 FG On-Demand Anodyne FAAH 17 41 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c1 ZINC000880551072 FG On-Demand Anodyne NPY5R 37 42 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c1 ZINC000880551072 FG On-Demand Anodyne S1PR2 27 40 O=C(COc1ccc(Cl)cc1Cl)NCc1cn(C2CCC2)nn1 ZINC000880551086 FG On-Demand Anodyne P2RX7 26 42 O=C(COc1ccc(Cl)cc1Cl)NCc1cn(C2CCC2)nn1 ZINC000880551086 FG On-Demand Anodyne MCHR2 20 40 O=C(COc1ccc(Cl)cc1Cl)NCc1cn(C2CCC2)nn1 ZINC000880551086 FG On-Demand Anodyne MAP3K8 33 41 COc1cncc(NC(=O)N2CCN(Cc3ccccn3)CC2)c1 ZINC000880551108 ED On-Demand Anodyne HTR2C 15 40 COc1cncc(NC(=O)N2CCN(Cc3ccccn3)CC2)c1 ZINC000880551108 ED On-Demand Anodyne PDGFRB 55 42 COc1cncc(NC(=O)N2CCN(Cc3ccccn3)CC2)c1 ZINC000880551108 ED On-Demand Anodyne FAAH 31 53 C#CCN(C)C(=O)Nc1cncc(OC)c1 ZINC000880551121 BD On-Demand Mild ROCK2 15 40 O=C(NCc1cn(C2CCC2)nn1)C(O)(c1ccccc1)c1ccccc1 ZINC000880551127 FF On-Demand Anodyne CHRM3 15 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)c1 ZINC000880551128 EF On-Demand Anodyne EPHX2 30 42 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)c1 ZINC000880551128 EF On-Demand Anodyne SCD1 19 43 COc1cncc(NC(=O)NCCc2cn3c(n2)SCC3)c1 ZINC000880551154 DD On-Demand Anodyne PIK3CG 15 42 COc1cncc(NC(=O)N2CCCc3ccccc3C2)c1 ZINC000880551171 CG On-Demand Anodyne P2RY14 46 34 COc1cncc(NC(=O)N2CCCc3ccccc3C2)c1 ZINC000880551171 CG On-Demand Anodyne NOD2 40 39 O=C(Cc1cccs1)NCc1cn(C2CCC2)nn1 ZINC000880551177 CD On-Demand Anodyne CA5B 33 46 O=C(Cc1cccs1)NCc1cn(C2CCC2)nn1 ZINC000880551177 CD On-Demand Anodyne CA5A 32 46 COc1cncc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880551180 EE On-Demand Anodyne PDGFRB 63 44 COc1cncc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880551180 EE On-Demand Anodyne TRPV1 16 47 COc1cncc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880551180 EE On-Demand Anodyne FAAH 21 41 COc1cncc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880551180 EE On-Demand Anodyne S1PR2 24 40 COc1cncc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880551180 EE On-Demand Anodyne RBP4 18 51 COc1cncc(NC(=O)Nc2cc(C3CC3)[nH]n2)c1 ZINC000880551195 CE On-Demand Anodyne CDK2 15 58 COc1cncc(NC(=O)Nc2cc(C3CC3)[nH]n2)c1 ZINC000880551195 CE On-Demand Anodyne PKNB 55 34 CCCN(CCCN(C)C)C(=O)Nc1cncc(OC)c1 ZINC000880551196 CE On-Demand Anodyne ROCK2 18 41 COC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880551203 DD On-Demand Anodyne MTOR 20 41 COC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880551203 DD On-Demand Anodyne EPHX2 56 53 COC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880551203 DD On-Demand Anodyne CXCR3 17 42 COc1cncc(NC(=O)N(C)CCCNC(=O)C2CCC2)c1 ZINC000880551208 DD On-Demand Anodyne MTNR1A 17 41 COc1cncc(NC(=O)N(C)CCCNC(=O)C2CCC2)c1 ZINC000880551208 DD On-Demand Anodyne IKBKE 44 38 COc1cncc(NC(=O)N(C)CCCNC(=O)C2CCC2)c1 ZINC000880551208 DD On-Demand Anodyne TBK1 83 38 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne PDGFRB 40 38 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne SIGMAR1 28 42 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne CCR3 28 45 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne CHRNA7 26 41 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne FAAH 32 53 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne RBP4 41 35 COc1cncc(NC(=O)N2C[C@@H]3CN(Cc4ccccc4)C[C@@H]3C2)c1 ZINC000880551217 FF On-Demand Anodyne MCHR1 17 42 COc1cncc(NC(=O)N(CCO)Cc2ccc(C)o2)c1 ZINC000880551222 DE On-Demand Anodyne ROCK2 15 44 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccccc1 ZINC000880551224 GE On-Demand Anodyne XIAP 57 38 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccccc1 ZINC000880551224 GE On-Demand Anodyne BIRC3 46 34 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccccc1 ZINC000880551224 GE On-Demand Anodyne BIRC2 88 37 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccccc1 ZINC000880551224 GE On-Demand Anodyne BIRC8 57 34 COc1cncc(NC(=O)N2CCCC3(CCOCC3)C2)c1 ZINC000880551225 DF On-Demand Anodyne EPHX2 32 40 COc1cncc(NC(=O)NCCC#N)c1 ZINC000880551231 BD On-Demand Mild ADRB1 41 31 c1ccc2c(c1)CN(CCCc1ccncc1)C[C@H]1CCCN21 ZINC000880551237 DG On-Demand Anodyne SIGMAR1 28 43 COc1cncc(NC(=O)N2CCC(O)(Cc3ccc(F)cc3)CC2)c1 ZINC000880551254 FF On-Demand Anodyne CACNA1H 39 40 COc1cncc(NC(=O)N2CCC(O)(Cc3ccc(F)cc3)CC2)c1 ZINC000880551254 FF On-Demand Anodyne CCR3 17 43 COc1cncc(NC(=O)N2CCC(O)(Cc3ccc(F)cc3)CC2)c1 ZINC000880551254 FF On-Demand Anodyne S1PR2 35 51 COc1cncc(NC(=O)NCc2ccc(CCN(C)C)cc2)c1 ZINC000880551259 EF On-Demand Anodyne ROCK2 33 44 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NCC(=O)c1cccs1 ZINC000880551295 FF On-Demand Anodyne NOS1 25 42 COc1cncc(NC(=O)N2CC[C@H](CN3CCOCC3)C2)c1 ZINC000880551315 DD On-Demand Anodyne CCR3 15 54 COc1cncc(NC(=O)N2CC[C@@H](CN3CCOCC3)C2)c1 ZINC000880551316 DD On-Demand Anodyne CCR3 15 54 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3o2)c1 ZINC000880551332 FH On-Demand Anodyne CPT1A 90 39 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3o2)c1 ZINC000880551333 FH On-Demand Anodyne CPT1A 90 39 COc1cncc(NC(=O)N2CCN(c3nnc(C(F)(F)F)s3)CC2)c1 ZINC000880551334 GE On-Demand Anodyne NPBWR1 18 44 O=C(COc1cccc(C(F)(F)F)c1)NCc1cn(C2CCC2)nn1 ZINC000880551335 FF On-Demand Anodyne CCR2 74 39 O=C(COc1cccc(C(F)(F)F)c1)NCc1cn(C2CCC2)nn1 ZINC000880551335 FF On-Demand Anodyne PDS 44 41 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)C1CC1 ZINC000880551336 CF On-Demand Anodyne HTR1A 15 41 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)C1CC1 ZINC000880551336 CF On-Demand Anodyne SLC6A1 58 37 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)C1CC1 ZINC000880551336 CF On-Demand Anodyne HTR7 22 41 COc1cncc(NC(=O)N(CCO)Cc2ccc(Br)s2)c1 ZINC000880551347 GF On-Demand Anodyne ROCK2 15 43 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne PDGFRB 33 42 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne GRIN2B 60 49 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne CCR3 24 45 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne FAAH 19 42 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne CAPN2 48 37 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne TGM2 39 48 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne NPR 49 32 COc1cncc(NC(=O)N2CCC(CNC(=O)OCc3ccccc3)CC2)c1 ZINC000880551349 GG On-Demand Anodyne F13A1 34 48 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccncc3)C2)c1 ZINC000880551351 DE On-Demand Anodyne PDE3A 27 42 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccncc3)C2)c1 ZINC000880551351 DE On-Demand Anodyne PDE3B 33 42 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccncc3)C2)c1 ZINC000880551351 DE On-Demand Anodyne EPHX2 26 44 COc1cncc(NC(=O)N2CCOC3(CCCCC3)C2)c1 ZINC000880551355 DF On-Demand Anodyne EPHX2 26 49 COc1cncc(NC(=O)NCCc2cccc(C)n2)c1 ZINC000880551363 CE On-Demand Anodyne MTNR1A 63 42 COc1cncc(NC(=O)NCCc2cccc(C)n2)c1 ZINC000880551363 CE On-Demand Anodyne MTNR1B 56 38 COc1cncc(NC(=O)NCCc2cccc(C)n2)c1 ZINC000880551363 CE On-Demand Anodyne PIK3CG 15 42 COc1cncc(NC(=O)N[C@H]2C[C@@H]2c2cccc(F)c2)c1 ZINC000880551368 DF On-Demand Anodyne EPHX2 17 41 COc1cncc(NC(=O)N[C@H]2C[C@H]2c2cccc(F)c2)c1 ZINC000880551369 DF On-Demand Anodyne EPHX2 17 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H]2c2cccc(F)c2)c1 ZINC000880551370 DF On-Demand Anodyne EPHX2 17 41 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2cccc(F)c2)c1 ZINC000880551371 DF On-Demand Anodyne EPHX2 17 41 COc1cncc(NC(=O)N(C)Cc2cnccc2C)c1 ZINC000880551374 CE On-Demand Anodyne ROCK2 16 42 COc1cncc(NC(=O)N(C)Cc2nc[nH]n2)c1 ZINC000880551375 CC On-Demand Anodyne ROCK2 18 44 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne TSHR 42 31 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne PTGER1 44 34 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne PDE4A 18 42 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne CPT1A 44 31 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne PREP 22 42 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne CA14 16 40 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne SLC6A5 15 41 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne SLC5A7 35 41 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne ABCG2 17 40 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OCc1ccccc1 ZINC000880551378 GH On-Demand Anodyne ACKR3 42 36 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne DRD2 24 54 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne TSHR 41 30 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne DRD4 53 55 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne ACHE 53 49 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne HRH2 26 41 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne DRD3 22 54 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne HTR4 52 44 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne SIGMAR1 48 46 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne MMP13 16 41 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne BCHE 17 44 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne CCR3 121 51 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne CHRNA7 18 40 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne NPFFR2 19 40 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne SLC18A3 18 41 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne FAAH 19 40 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne MCHR1 40 45 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne CACNA1I 65 39 COc1cncc(NC(=O)NC[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551389 EF On-Demand Anodyne NPFFR1 26 40 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne DRD2 24 54 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne TSHR 41 30 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne DRD4 53 55 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne ACHE 53 49 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne HRH2 26 41 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne DRD3 22 54 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne HTR4 52 44 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne SIGMAR1 48 46 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne MMP13 16 41 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne BCHE 17 44 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne CCR3 121 51 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne CHRNA7 18 40 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne NPFFR2 19 40 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne SLC18A3 18 41 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne FAAH 19 40 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne MCHR1 40 45 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne CACNA1I 65 39 COc1cncc(NC(=O)NC[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880551390 EF On-Demand Anodyne NPFFR1 26 40 COCCONC(=O)Nc1cncc(OC)c1 ZINC000880551395 BC On-Demand Anodyne SCN10A 31 43 COc1cncc(NC(=O)N2CCC3(CCC3)C2)c1 ZINC000880551401 CE On-Demand Anodyne EPHX2 34 45 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NNC(=O)c1cccs1 ZINC000880551405 FD On-Demand Reactive NOS1 27 43 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1ccc(Cl)cc1 ZINC000880551407 EG On-Demand Anodyne SCN10A 23 42 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1ccc(Cl)cc1 ZINC000880551407 EG On-Demand Anodyne UTS2 42 38 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccc(Cl)cc1 ZINC000880551408 EG On-Demand Anodyne SCN10A 23 42 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccc(Cl)cc1 ZINC000880551408 EG On-Demand Anodyne UTS2 42 38 O=C(NCc1cn(C2CCC2)nn1)c1ccc(C2SCCS2)cc1 ZINC000880551410 FG On-Demand Anodyne CA14 16 48 COc1cncc(NC(=O)N2CCC(Oc3ccc(C#N)cc3)CC2)c1 ZINC000880551411 FG On-Demand Mild PDGFRB 31 43 COc1cncc(NC(=O)N2CCC(Oc3ccc(C#N)cc3)CC2)c1 ZINC000880551411 FG On-Demand Mild EPHX2 27 50 CCOC(=O)N1CC[C@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880551415 DD On-Demand Anodyne EPHX2 44 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880551416 DD On-Demand Anodyne EPHX2 44 42 COc1cncc(NC(=O)N2CCC[C@@H](CC(N)=O)C2)c1 ZINC000880551418 CD On-Demand Anodyne CCR3 15 49 COc1cncc(NC(=O)N2CCC[C@H](CC(N)=O)C2)c1 ZINC000880551419 CD On-Demand Anodyne CCR3 15 49 COc1cncc(NC(=O)N2CCS(=O)(=O)c3ccccc3C2)c1 ZINC000880551420 ED On-Demand Anodyne P2RY14 42 33 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551425 EF On-Demand Anodyne ROCK1 21 40 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551425 EF On-Demand Anodyne ROCK2 34 40 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551425 EF On-Demand Anodyne NPY5R 37 54 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551426 EF On-Demand Anodyne ROCK1 21 40 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551426 EF On-Demand Anodyne ROCK2 34 40 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551426 EF On-Demand Anodyne NPY5R 37 54 COCCC[C@@H](Cc1ccccc1)NC(=O)Nc1cncc(OC)c1 ZINC000880551445 EG On-Demand Anodyne ANPEP 40 31 COCCC[C@@H](Cc1ccccc1)NC(=O)Nc1cncc(OC)c1 ZINC000880551445 EG On-Demand Anodyne FPR1 27 40 COCCC[C@H](Cc1ccccc1)NC(=O)Nc1cncc(OC)c1 ZINC000880551447 EG On-Demand Anodyne ANPEP 40 31 COCCC[C@H](Cc1ccccc1)NC(=O)Nc1cncc(OC)c1 ZINC000880551447 EG On-Demand Anodyne FPR1 27 40 O=C(NCc1cn(C2CCC2)nn1)c1ccc(C2SCCCS2)cc1 ZINC000880551448 FH On-Demand Anodyne CA14 15 47 C=CCN(C)C(=O)Nc1cncc(OC)c1 ZINC000880551454 BD On-Demand Mild ROCK2 15 42 COc1cncc(NC(=O)N2CCN(c3nccc(C(C)C)n3)CC2)c1 ZINC000880551458 FE On-Demand Anodyne PDGFRB 52 42 COc1cncc(NC(=O)N2CCC(Oc3ccncc3C)CC2)c1 ZINC000880551459 EF On-Demand Anodyne PDE4A 17 45 COc1cncc(NC(=O)N2CCC(Oc3ccncc3C)CC2)c1 ZINC000880551459 EF On-Demand Anodyne EPHX2 19 41 COc1cncc(NC(=O)N2CCC(Oc3ccncc3C)CC2)c1 ZINC000880551459 EF On-Demand Anodyne SCD1 23 52 COc1cncc(NC(=O)N2CC[C@](O)(C(F)(F)F)C2)c1 ZINC000880551468 DD On-Demand Anodyne EPHX2 33 41 COc1cncc(NC(=O)N2CC[C@@](O)(C(F)(F)F)C2)c1 ZINC000880551470 DD On-Demand Anodyne EPHX2 33 41 COc1cncc(NC(=O)NC2CCC(O)(c3cccnc3)CC2)c1 ZINC000880551478 EE On-Demand Anodyne CHRNA7 21 46 COc1cncc(NC(=O)N2CCC(NC(=O)C3CC3)CC2)c1 ZINC000880551493 DD On-Demand Anodyne EPHX2 36 43 COc1cncc(NC(=O)N2CCN(c3ccc(CN(C)C)cn3)CC2)c1 ZINC000880551496 FD On-Demand Anodyne PDGFRB 53 39 COc1cncc(NC(=O)N2CCN(c3ccc(CN(C)C)cn3)CC2)c1 ZINC000880551496 FD On-Demand Anodyne DGAT1 27 42 COc1cncc(NC(=O)NC[C@@H]2CCN(C)C2)c1 ZINC000880551498 CD On-Demand Anodyne CCR3 47 43 COc1cncc(NC(=O)NC[C@@H]2CCN(C)C2)c1 ZINC000880551498 CD On-Demand Anodyne CACNA1I 57 34 COc1cncc(NC(=O)NC[C@H]2CCN(C)C2)c1 ZINC000880551499 CD On-Demand Anodyne CCR3 47 43 COc1cncc(NC(=O)NC[C@H]2CCN(C)C2)c1 ZINC000880551499 CD On-Demand Anodyne CACNA1I 57 34 COc1cncc(NC(=O)N2CC[C@H](Oc3cccnc3N(C)C)C2)c1 ZINC000880551508 FE On-Demand Anodyne SCD1 15 42 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccnc3N(C)C)C2)c1 ZINC000880551509 FE On-Demand Anodyne SCD1 15 42 COc1cncc(NC(=O)N2CCc3ncsc3C2)c1 ZINC000880551513 CE On-Demand Anodyne P2RY14 47 34 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551519 DE On-Demand Anodyne HTR1A 23 40 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551519 DE On-Demand Anodyne SLC6A1 50 39 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551519 DE On-Demand Anodyne HTR7 36 40 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551519 DE On-Demand Anodyne CYP2J2 44 31 COc1cncc(NC(=O)N2CC[C@@H](CN(C)Cc3cccnc3)C2)c1 ZINC000880551532 FE On-Demand Anodyne GRIN2B 18 41 COc1cncc(NC(=O)N2CC[C@@H](CN(C)Cc3cccnc3)C2)c1 ZINC000880551532 FE On-Demand Anodyne CHRNA7 50 43 COc1cncc(NC(=O)N2CC[C@H](CN(C)Cc3cccnc3)C2)c1 ZINC000880551533 FE On-Demand Anodyne GRIN2B 18 41 COc1cncc(NC(=O)N2CC[C@H](CN(C)Cc3cccnc3)C2)c1 ZINC000880551533 FE On-Demand Anodyne CHRNA7 50 43 CCCN(CCc1cccs1)C(=O)Nc1cncc(OC)c1 ZINC000880551534 DH On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)N2CC(Cc3ccc(F)c(F)c3)C2)c1 ZINC000880551539 EG On-Demand Anodyne CCR3 34 49 COc1cncc(NC(=O)NCc2ccc(C(C)(C)O)cc2)c1 ZINC000880551543 DF On-Demand Anodyne TRPV1 33 43 COc1cncc(NC(=O)NCc2ccc(C(C)(C)O)cc2)c1 ZINC000880551543 DF On-Demand Anodyne ROCK2 23 47 COc1cncc(NC(=O)NC[C@@H]2CCCN(c3ccccc3)C2)c1 ZINC000880551597 EG On-Demand Anodyne CCR3 61 46 COc1cncc(NC(=O)NC[C@H]2CCCN(c3ccccc3)C2)c1 ZINC000880551598 EG On-Demand Anodyne CCR3 61 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880551601 GE On-Demand Anodyne P2RX7 48 55 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880551605 GE On-Demand Anodyne P2RX7 48 55 COC[C@@H](c1ccc(Cl)cc1)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880551651 EH On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N2CCc3ccnc(O)c3C2)c1 ZINC000880551658 DD On-Demand Anodyne P2RY14 41 33 COc1cncc(NC(=O)NCCCN2CCCO[C@H](C)C2)c1 ZINC000880551677 DD On-Demand Anodyne HRH2 22 41 COc1cncc(NC(=O)NCCCN2CCCO[C@H](C)C2)c1 ZINC000880551677 DD On-Demand Anodyne CCR3 48 49 COc1cncc(NC(=O)N2CCC(Cn3cncn3)CC2)c1 ZINC000880551679 DD On-Demand Anodyne PDGFRB 40 35 COc1cncc(NC(=O)NCCCN2CCCO[C@@H](C)C2)c1 ZINC000880551681 DD On-Demand Anodyne HRH2 22 41 COc1cncc(NC(=O)NCCCN2CCCO[C@@H](C)C2)c1 ZINC000880551681 DD On-Demand Anodyne CCR3 48 49 COc1cncc(NC(=O)N[C@H]2CCC[C@H]2CCO)c1 ZINC000880551703 CD On-Demand Anodyne CCR3 24 41 COc1cncc(NC(=O)N[C@@H]2CCC[C@H]2CCO)c1 ZINC000880551704 CD On-Demand Anodyne CCR3 24 41 COc1cncc(NC(=O)N[C@H]2CCC[C@@H]2CCO)c1 ZINC000880551706 CD On-Demand Anodyne CCR3 24 41 COc1cncc(NC(=O)N[C@@H]2CCC[C@@H]2CCO)c1 ZINC000880551707 CD On-Demand Anodyne CCR3 24 41 O=C(NCCCN1Cc2ccccc2N2CCC[C@@H]2C1)C(F)(F)F ZINC000880551715 EF On-Demand Anodyne DRD2 21 41 O=C(NCCCN1Cc2ccccc2N2CCC[C@@H]2C1)C(F)(F)F ZINC000880551715 EF On-Demand Anodyne DRD3 33 48 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne NQO2 17 43 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne CCR3 22 40 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne MTNR1A 25 42 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne IKBKE 47 43 COc1cncc(NC(=O)NCCCNC(=O)C2CCC2)c1 ZINC000880551716 DD On-Demand Anodyne TBK1 92 43 COc1cncc(NC(=O)N(CCCO)Cc2ccccn2)c1 ZINC000880551717 DD On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)N2CCN(C3CCOCC3)C[C@H]2C)c1 ZINC000880551721 ED On-Demand Anodyne LIMK2 24 41 COc1cncc(NC(=O)N2CCN(C3CCOCC3)C[C@@H]2C)c1 ZINC000880551723 ED On-Demand Anodyne LIMK2 24 41 COc1cncc(NC(=O)NCc2cc(C)c(O)c(C)c2)c1 ZINC000880551743 DF On-Demand Anodyne ROCK2 19 47 COc1cncc(NC(=O)NCc2cc(C)c(O)c(C)c2)c1 ZINC000880551743 DF On-Demand Anodyne NAMPT 33 42 COc1cncc(NC(=O)NC(C)(C)C(F)F)c1 ZINC000880551748 CE On-Demand Anodyne IMDH_CRYPV 19 40 COc1cncc(NC(=O)NCC2CCN(C3CC3)CC2)c1 ZINC000880551750 DE On-Demand Anodyne CCR3 38 41 COc1cncc(NC(=O)NCC2CCN(C3CC3)CC2)c1 ZINC000880551750 DE On-Demand Anodyne CACNA1I 55 32 CCOC(=O)Nc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880551753 EF On-Demand Anodyne CA14 21 46 COc1cncc(NC(=O)N[C@H](CO)c2ccccc2OC(F)(F)F)c1 ZINC000880551757 FF On-Demand Anodyne KCNK3 37 40 COc1cncc(NC(=O)N[C@H](CO)c2ccccc2OC(F)(F)F)c1 ZINC000880551757 FF On-Demand Anodyne KCNK9 38 40 COc1cncc(NC(=O)N[C@@H](CO)c2ccccc2OC(F)(F)F)c1 ZINC000880551759 FF On-Demand Anodyne KCNK3 37 40 COc1cncc(NC(=O)N[C@@H](CO)c2ccccc2OC(F)(F)F)c1 ZINC000880551759 FF On-Demand Anodyne KCNK9 38 40 Oc1nc(CN2Cc3ccccc3N3CCC[C@@H]3C2)nc2c1oc1ccccc12 ZINC000880551763 GI On-Demand Anodyne PIM1 17 48 Oc1nc(CN2Cc3ccccc3N3CCC[C@@H]3C2)nc2c1oc1ccccc12 ZINC000880551763 GI On-Demand Anodyne CDC7 20 48 Oc1nc(CN2Cc3ccccc3N3CCC[C@@H]3C2)nc2c1oc1ccccc12 ZINC000880551763 GI On-Demand Anodyne PIM3 20 48 CCn1cccc(CNC(=O)Nc2cncc(OC)c2)c1=O ZINC000880551775 DD On-Demand Anodyne ROCK2 17 42 COc1cncc(NC(=O)NCCc2ccccc2OC(F)F)c1 ZINC000880551869 EG On-Demand Anodyne ADRB1 43 32 COc1cncc(NC(=O)NCCc2ccccc2OC(F)F)c1 ZINC000880551869 EG On-Demand Anodyne MTNR1A 52 40 COc1cncc(NC(=O)NCCc2ccccc2OC(F)F)c1 ZINC000880551869 EG On-Demand Anodyne MTNR1B 40 37 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne HTR1A 23 52 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne DRD4 43 35 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne HTR1D 17 52 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne HTR1B 22 48 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne PDGFRB 51 42 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne NPY2R 49 37 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne FAAH 22 44 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3F)CC2)c1 ZINC000880551873 EF On-Demand Anodyne RBP4 19 43 COc1cncc(NC(=O)NC2CCN(c3cccnn3)CC2)c1 ZINC000880551885 ED On-Demand Anodyne EPHX2 44 38 Cn1nc(C(=O)NCc2cn(C3CCC3)nn2)c2ccccc2c1=O ZINC000880551889 ED On-Demand Anodyne HTR3A 16 43 COCCCC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccccc1 ZINC000880551895 EH On-Demand Anodyne UTS2 41 33 COCCCC[C@H](NC(=O)Nc1cncc(OC)c1)c1ccccc1 ZINC000880551897 EH On-Demand Anodyne UTS2 41 33 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne CACNA1H 56 37 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne PDGFRB 46 39 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne FAAH 19 42 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne S1PR2 30 45 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne EPHX2 32 41 COc1cncc(NC(=O)N2CCC(O)(c3c(F)cccc3F)CC2)c1 ZINC000880551899 FF On-Demand Anodyne TRPM8 31 42 COc1cncc(NC(=O)N2CCC(CO)(Cc3ccccc3)CC2)c1 ZINC000880551915 FF On-Demand Anodyne FAAH 20 45 COc1cncc(NC(=O)N2CCC(CO)(Cc3ccccc3)CC2)c1 ZINC000880551915 FF On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne DRD4 39 44 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne HRH2 30 42 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne CCR3 50 45 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne NPFFR2 17 40 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne MCHR1 27 40 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551925 FF On-Demand Anodyne NPFFR1 20 40 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne DRD4 39 44 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne HRH2 30 42 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne CCR3 50 45 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne NPFFR2 17 40 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne MCHR1 27 40 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCCO2)c1 ZINC000880551926 FF On-Demand Anodyne NPFFR1 20 40 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000880551939 FE On-Demand Anodyne PDGFRB 52 43 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000880551939 FE On-Demand Anodyne CHRNA7 17 40 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000880551939 FE On-Demand Anodyne FAAH 28 51 COc1cncc(NC(=O)N2CCC(Oc3ncccc3F)CC2)c1 ZINC000880551941 EF On-Demand Anodyne EPHX2 23 40 COc1cncc(NC(=O)N2CCC(Oc3ncccc3F)CC2)c1 ZINC000880551941 EF On-Demand Anodyne SCD1 23 46 CCC(=O)CCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880551946 CF On-Demand Anodyne SLC6A1 42 32 COc1cncc(NC(=O)NCC2(N3CCOCC3)CC2)c1 ZINC000880551947 DD On-Demand Anodyne HCN1 61 37 COc1cncc(NC(=O)NCC2(N3CCOCC3)CC2)c1 ZINC000880551947 DD On-Demand Anodyne HCN4 51 36 COc1cncc(NC(=O)N2CCC(CCCN3CCOCC3)CC2)c1 ZINC000880551949 FE On-Demand Anodyne PDGFRB 32 42 COc1cncc(NC(=O)N2CCC(CCCN3CCOCC3)CC2)c1 ZINC000880551949 FE On-Demand Anodyne CCR3 15 41 COc1cncc(NC(=O)N2CCC(CCCN3CCOCC3)CC2)c1 ZINC000880551949 FE On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCC(CCCN3CCOCC3)CC2)c1 ZINC000880551949 FE On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne DRD2 35 41 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne AVPR2 20 42 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne DRD3 48 38 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne KCNQ2 76 43 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne SCN2A 21 48 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne ROCK2 16 42 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne SOAT1 17 40 COc1cncc(NC(=O)NCc2ccccc2N2CCCC2)c1 ZINC000880551954 EG On-Demand Anodyne SCN10A 38 48 COc1cncc(NC(=O)N2CCO[C@H](COc3ccccc3)C2)c1 ZINC000880551955 EE On-Demand Anodyne CHRNA7 18 44 COc1cncc(NC(=O)N2CCO[C@@H](COc3ccccc3)C2)c1 ZINC000880551957 EE On-Demand Anodyne CHRNA7 18 44 COc1cncc(NC(=O)N2CCC(c3ccsc3)CC2)c1 ZINC000880551967 DH On-Demand Anodyne NPBWR1 91 37 O=C(NCc1cn(C2CCC2)nn1)c1ccc(SC(F)(F)F)cc1 ZINC000880551968 FH On-Demand Anodyne CA14 15 45 COc1cncc(NC(=O)N2CCN(c3ncc(F)cn3)CC2)c1 ZINC000880551971 ED On-Demand Anodyne PDGFRB 53 41 O=C(CCc1ccc2ccccc2n1)NCc1cn(C2CCC2)nn1 ZINC000880551983 EF On-Demand Anodyne SUCNR1 47 35 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne CA2 31 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne CA1 29 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne CA7 20 40 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne CA12 19 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne CA9 27 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880551996 FE On-Demand Anodyne A6YCJ1_9METZ 15 40 NC(=O)NC(=O)OCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552010 ED On-Demand Anodyne SLC6A1 47 37 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccccc1Br ZINC000880552020 JK On-Demand Mild GRM4 58 41 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccccc1Br ZINC000880552020 JK On-Demand Mild NR2E3 43 31 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccccc1Br ZINC000880552020 JK On-Demand Mild KCNK3 59 38 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccccc1Br ZINC000880552020 JK On-Demand Mild KCNK9 50 37 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccccc1Br ZINC000880552020 JK On-Demand Mild G2YM83_BOTF4 45 33 COc1cncc(NC(=O)Nc2cc(OC)n(C)n2)c1 ZINC000880552027 CD On-Demand Anodyne HTR2A 21 41 COc1cncc(NC(=O)N[C@H]2CCOc3c(F)cccc32)c1 ZINC000880552028 DF On-Demand Anodyne TRPV1 19 44 COc1cncc(NC(=O)N2CCc3ccccc3[C@H]2C)c1 ZINC000880552039 CG On-Demand Anodyne TRPM8 39 45 COc1cncc(NC(=O)N2CCc3ccccc3[C@@H]2C)c1 ZINC000880552040 CG On-Demand Anodyne TRPM8 39 45 COc1cncc(NC(=O)N2CCN(CC(C)(C)O)C[C@H]2C)c1 ZINC000880552041 DD On-Demand Anodyne LIMK2 24 41 COc1cncc(NC(=O)N2CCN(CC(C)(C)O)C[C@@H]2C)c1 ZINC000880552042 DD On-Demand Anodyne LIMK2 24 41 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccc(C)o2)c1 ZINC000880552052 DH On-Demand Anodyne CPT1A 44 36 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccc(C)o2)c1 ZINC000880552053 DH On-Demand Anodyne CPT1A 44 36 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne F2 23 40 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne PDGFRB 26 40 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne GRIN2B 24 42 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne CCR3 31 53 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne PREP 33 41 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne TGM2 39 44 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552064 GG On-Demand Anodyne F13A1 28 44 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne F2 23 40 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne PDGFRB 26 40 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne GRIN2B 24 42 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne CCR3 31 53 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne PREP 33 41 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne TGM2 39 44 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OCc3ccccc3)C2)c1 ZINC000880552065 GG On-Demand Anodyne F13A1 28 44 COc1cncc(NC(=O)NCc2ccc3c(n2)CCCC3)c1 ZINC000880552066 DF On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C2CCOCC2)c1 ZINC000880552071 FG On-Demand Anodyne ROCK2 15 46 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne CYP11B1 17 42 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne PDGFRB 43 40 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne DRD5 18 43 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne CYP11B2 29 40 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne MTNR1A 16 41 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3CC2)c1 ZINC000880552073 EF On-Demand Anodyne MTNR1B 24 41 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1nccs1 ZINC000880552074 EF On-Demand Anodyne MAP1 108 45 COc1cncc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000880552078 CF On-Demand Anodyne EPHX2 29 52 COc1cncc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000880552079 CF On-Demand Anodyne EPHX2 29 52 COc1cncc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000880552080 CF On-Demand Anodyne EPHX2 29 52 COc1cncc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000880552081 CF On-Demand Anodyne EPHX2 29 52 COc1cncc(NC(=O)N(C)Cc2ccc(C)cn2)c1 ZINC000880552086 CE On-Demand Anodyne ROCK2 16 40 COc1cncc(NC(=O)NC[C@@](C)(Cc2ccccc2)[C@@H](C)O)c1 ZINC000880552090 EF On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)NC[C@@](C)(Cc2ccccc2)[C@H](C)O)c1 ZINC000880552092 EF On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)NC[C@](C)(Cc2ccccc2)[C@@H](C)O)c1 ZINC000880552094 EF On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)NC[C@](C)(Cc2ccccc2)[C@H](C)O)c1 ZINC000880552096 EF On-Demand Anodyne ROCK2 17 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880552097 ED On-Demand Anodyne INHA 21 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880552099 ED On-Demand Anodyne INHA 21 46 COc1cncc(NC(=O)N2CCc3c(C)cc(C)cc3C2)c1 ZINC000880552111 DG On-Demand Anodyne P2RY14 43 33 COc1cncc(NC(=O)N[C@H](CO)Cc2ccc(F)cc2)c1 ZINC000880552113 DD On-Demand Anodyne CCR3 49 30 COc1cncc(NC(=O)N[C@@H](CO)Cc2ccc(F)cc2)c1 ZINC000880552114 DD On-Demand Anodyne CCR3 49 30 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(C)c3)CC2)c1 ZINC000880552115 FG On-Demand Anodyne FAAH 19 41 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(C)c3)CC2)c1 ZINC000880552115 FG On-Demand Anodyne S1PR2 30 44 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)c1 ZINC000880552120 GH On-Demand Anodyne NPY5R 33 41 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)c1 ZINC000880552120 GH On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3C(F)(F)F)CC2)c1 ZINC000880552120 GH On-Demand Anodyne RBP4 60 39 COc1cncc(NC(=O)N(C)Cc2ccccc2SC)c1 ZINC000880552124 DG On-Demand Anodyne ROCK2 17 41 c1ccc2c(c1)CN(CC1CC1)C[C@H]1CCCN21 ZINC000880552130 BF On-Demand Anodyne SIGMAR1 15 41 NC(=O)c1ccc(NC(=O)CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552131 GF On-Demand Anodyne AVPR2 59 39 NC(=O)c1ccc(NC(=O)CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552131 GF On-Demand Anodyne NOD2 40 34 COc1cncc(NC(=O)NC2CC(N3CCC(C(F)(F)F)CC3)C2)c1 ZINC000880552134 FG On-Demand Anodyne EPHX2 44 38 COc1cncc(NC(=O)N[C@H](CO)Cc2cccc(C)c2)c1 ZINC000880552138 DE On-Demand Anodyne CTSL 22 40 COc1cncc(NC(=O)N[C@H](CO)Cc2cccc(C)c2)c1 ZINC000880552138 DE On-Demand Anodyne PIN1 21 40 COc1cncc(NC(=O)N[C@@H](CO)Cc2cccc(C)c2)c1 ZINC000880552140 DE On-Demand Anodyne CTSL 22 40 COc1cncc(NC(=O)N[C@@H](CO)Cc2cccc(C)c2)c1 ZINC000880552140 DE On-Demand Anodyne PIN1 21 40 COc1cncc(NC(=O)N2CC[C@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552145 GF On-Demand Anodyne PDE3A 40 41 COc1cncc(NC(=O)N2CC[C@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552145 GF On-Demand Anodyne PDGFRB 48 38 COc1cncc(NC(=O)N2CC[C@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552145 GF On-Demand Anodyne PDE3B 46 41 COc1cncc(NC(=O)N2CC[C@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552145 GF On-Demand Anodyne SCD1 22 42 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552148 GF On-Demand Anodyne PDE3A 40 41 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552148 GF On-Demand Anodyne PDGFRB 48 38 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552148 GF On-Demand Anodyne PDE3B 46 41 COc1cncc(NC(=O)N2CC[C@@H](Oc3cccnc3N3CCCC3)C2)c1 ZINC000880552148 GF On-Demand Anodyne SCD1 22 42 COc1cncc(NC(=O)N2CCN(c3c(C#N)c(C)nn3C)CC2)c1 ZINC000880552161 FD On-Demand Mild PDGFRB 50 41 COc1cncc(NC(=O)N2CCc3cc(Cl)ccc3C2)c1 ZINC000880552164 DG On-Demand Anodyne HTR2C 15 41 COc1cncc(NC(=O)NC[C@H]2CCCN(C(C)=O)C2)c1 ZINC000880552166 DD On-Demand Anodyne CCR3 53 42 COc1cncc(NC(=O)NC[C@@H]2CCCN(C(C)=O)C2)c1 ZINC000880552169 DD On-Demand Anodyne CCR3 53 42 N#Cc1ccc(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552170 EF On-Demand Mild MCHR1 21 40 CC[C@H]1c2ccccc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880552174 DH On-Demand Anodyne MTNR1B 27 43 CC[C@H]1c2ccccc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880552174 DH On-Demand Anodyne TRPM8 35 43 COC(=O)/C(C)=C\CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552176 DF On-Demand Anodyne SLC6A1 61 33 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880552177 DH On-Demand Anodyne MTNR1B 27 43 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880552177 DH On-Demand Anodyne TRPM8 35 43 COC(=O)/C(C)=C/CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552178 DF On-Demand Anodyne SLC6A1 61 33 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880552182 FG On-Demand Anodyne CCR3 15 44 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880552182 FG On-Demand Anodyne SLC18A3 47 50 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880552182 FG On-Demand Anodyne WNT3A 53 34 COc1cncc(NC(=O)N(C)[C@H](C)C[S@@](C)=O)c1 ZINC000880552183 CD On-Demand Anodyne NPY5R 32 43 COc1cncc(NC(=O)N(C)[C@H](C)C[S@](C)=O)c1 ZINC000880552184 CD On-Demand Anodyne NPY5R 32 43 COc1cncc(NC(=O)N(C)[C@@H](C)C[S@](C)=O)c1 ZINC000880552185 CD On-Demand Anodyne NPY5R 32 43 COc1cncc(NC(=O)N(C)[C@@H](C)C[S@@](C)=O)c1 ZINC000880552186 CD On-Demand Anodyne NPY5R 32 43 O=C(NCc1cn(C2CCC2)nn1)c1cc(Cl)nc2ccccc12 ZINC000880552197 EG On-Demand Anodyne TACR3 17 42 COc1cncc(NC(=O)NCc2ccccc2CN2CCC[C@@H]2CO)c1 ZINC000880552207 FE On-Demand Anodyne CCR3 28 40 COc1cncc(NC(=O)NCc2ccccc2CN2CCC[C@H]2CO)c1 ZINC000880552208 FE On-Demand Anodyne CCR3 28 40 O=C(NCc1cn(C2CCC2)nn1)c1cc(=O)c2ccccc2o1 ZINC000880552212 DE On-Demand Anodyne BCHE 29 42 CCOc1ccccc1OCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880552215 EE On-Demand Anodyne HCN1 46 38 CCOc1ccccc1OCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880552215 EE On-Demand Anodyne HCN4 46 38 COc1cncc(NC(=O)N2CCC(O)(C(F)F)CC2)c1 ZINC000880552220 DD On-Demand Anodyne S1PR2 30 44 COc1cncc(NC(=O)N2CCN(C(=O)NC(C)(C)C)CC2)c1 ZINC000880552229 ED On-Demand Anodyne PDGFRB 40 38 COc1cncc(NC(=O)N2CCC(c3nc4cccc(C)c4o3)CC2)c1 ZINC000880552230 FH On-Demand Anodyne SMO 33 50 COc1cncc(NC(=O)N2CCN(c3nc(F)c(F)cc3F)CC2)c1 ZINC000880552236 FE On-Demand Anodyne PDGFRB 55 41 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(F)c3)C2)c1 ZINC000880552238 DG On-Demand Anodyne GRIN2B 20 42 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(F)c3)C2)c1 ZINC000880552238 DG On-Demand Anodyne CCR3 27 46 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(F)c3)C2)c1 ZINC000880552238 DG On-Demand Anodyne CCR5 82 35 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(F)c3)C2)c1 ZINC000880552238 DG On-Demand Anodyne MCHR1 21 42 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(F)c3)C2)c1 ZINC000880552238 DG On-Demand Anodyne SCD1 18 40 COc1cncc(NC(=O)N2CC[C@H](c3cccc(F)c3)C2)c1 ZINC000880552239 DG On-Demand Anodyne GRIN2B 20 42 COc1cncc(NC(=O)N2CC[C@H](c3cccc(F)c3)C2)c1 ZINC000880552239 DG On-Demand Anodyne CCR3 27 46 COc1cncc(NC(=O)N2CC[C@H](c3cccc(F)c3)C2)c1 ZINC000880552239 DG On-Demand Anodyne CCR5 82 35 COc1cncc(NC(=O)N2CC[C@H](c3cccc(F)c3)C2)c1 ZINC000880552239 DG On-Demand Anodyne MCHR1 21 42 COc1cncc(NC(=O)N2CC[C@H](c3cccc(F)c3)C2)c1 ZINC000880552239 DG On-Demand Anodyne SCD1 18 40 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@@H]2c2ccccc2)c1 ZINC000880552243 EF On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@@H]2c2ccccc2)c1 ZINC000880552243 EF On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@@H]2c2ccccc2)c1 ZINC000880552244 EF On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@@H]2c2ccccc2)c1 ZINC000880552244 EF On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@H]2c2ccccc2)c1 ZINC000880552245 EF On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@H]2c2ccccc2)c1 ZINC000880552245 EF On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@H]2c2ccccc2)c1 ZINC000880552246 EF On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@H]2c2ccccc2)c1 ZINC000880552246 EF On-Demand Anodyne CHRNA7 15 42 N#Cc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880552254 EF On-Demand Mild CCR3 19 45 N#Cc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880552254 EF On-Demand Mild MCHR1 45 42 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)NNC(=O)c1ccccc1Cl ZINC000880552259 GF On-Demand Reactive AVPR2 43 36 COc1cncc(NC(=O)N2CCc3cccc(C)c3C2)c1 ZINC000880552266 CF On-Demand Anodyne HTR2C 15 41 COc1cncc(NC(=O)N2CCc3cccc(C)c3C2)c1 ZINC000880552266 CF On-Demand Anodyne P2RY14 57 42 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne HTR1A 38 54 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne ADRA1D 31 40 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne HTR1D 17 54 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne HTR1B 23 54 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne HTR2C 16 45 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne ADRA1A 26 40 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne ADRA1B 22 40 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne PDGFRB 72 53 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne HTR7 30 47 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne FAAH 18 46 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne PDGFRA 17 45 COc1cncc(NC(=O)N2CCN(c3ccncc3OC)CC2)c1 ZINC000880552271 ED On-Demand Anodyne RBP4 15 42 COc1cncc(NC(=O)NC2CCN(C3CCN(C)CC3)CC2)c1 ZINC000880552339 ED On-Demand Anodyne SLC6A5 19 41 COc1cncc(NC(=O)NC2CCN(C3CCN(C)CC3)CC2)c1 ZINC000880552339 ED On-Demand Anodyne EPHX2 43 38 COc1cncc(NC(=O)NC2CCN(C3CCN(C)CC3)CC2)c1 ZINC000880552339 ED On-Demand Anodyne CXCR3 17 40 COc1cncc(NC(=O)N[C@H](CO)Cc2ccccc2)c1 ZINC000880552347 DD On-Demand Anodyne MME 50 39 COc1cncc(NC(=O)N[C@H](CO)Cc2ccccc2)c1 ZINC000880552347 DD On-Demand Anodyne ANPEP 61 33 COc1cncc(NC(=O)N[C@H](CO)Cc2ccccc2)c1 ZINC000880552347 DD On-Demand Anodyne TIMP3 41 33 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne DRD4 45 35 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne HRH2 16 40 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne HTR2A 17 40 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne CCR3 28 41 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne CHRNA7 17 46 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne MTOR 21 43 COc1cncc(NC(=O)NCCN2CCCOCC2)c1 ZINC000880552360 CC On-Demand Anodyne EPHX2 25 44 COc1cncc(NC(=O)N2CCN(c3ncnc4sc(C)cc34)CC2)c1 ZINC000880552375 GF On-Demand Anodyne PDGFRB 83 50 COc1cncc(NC(=O)N2CCN(c3ncnc4sc(C)cc34)CC2)c1 ZINC000880552375 GF On-Demand Anodyne LIMK2 20 49 COc1cncc(NC(=O)N(C)CC2(c3ccccc3)CC2)c1 ZINC000880552396 DG On-Demand Anodyne KCNA3 42 44 COc1cncc(NC(=O)N2CCn3ncnc3C2)c1 ZINC000880552409 CC On-Demand Anodyne PDGFRB 45 38 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne PIK3CA 47 40 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne PIK3CD 24 46 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne MTOR 65 39 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne PIK3CB 40 46 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne DGAT1 21 43 COc1cncc(NC(=O)NCc2cccc(N3CCOCC3)n2)c1 ZINC000880552410 ED On-Demand Anodyne NAMPT 22 40 CC(C)(C)OC(=O)N1CCC(C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880552413 FE On-Demand Anodyne PREP 15 47 CC(C)(C)OC(=O)N1CCC(C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880552413 FE On-Demand Anodyne EPHX2 18 40 CC(C)(C)OC(=O)N1CCC(C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880552413 FE On-Demand Anodyne GPR119 45 39 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccco2)c1 ZINC000880552419 DG On-Demand Anodyne CPT1A 54 34 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccco2)c1 ZINC000880552420 DG On-Demand Anodyne CPT1A 54 34 COc1cncc(NC(=O)N2CCCN(C(=O)C3CC3)CC2)c1 ZINC000880552432 DD On-Demand Anodyne PDGFRB 46 38 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880552497 FE On-Demand Anodyne PREP 18 49 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880552498 FE On-Demand Anodyne PREP 18 49 COc1cncc(NC(=O)N(CCN(C)C)CCN(C)C)c1 ZINC000880552504 DD On-Demand Anodyne ROCK2 21 48 COc1cncc(NC(=O)N2CC[C@@H](CN3CCCCC3)C2)c1 ZINC000880552515 DE On-Demand Anodyne CCR3 22 55 COc1cncc(NC(=O)N2CC[C@H](CN3CCCCC3)C2)c1 ZINC000880552516 DE On-Demand Anodyne CCR3 22 55 O=C(NCc1cn(C2CCC2)nn1)c1ccc(-c2ccccc2)cc1 ZINC000880552517 EH On-Demand Anodyne CA14 16 48 COc1cncc(NC(=O)N2CCC3(CC2)CNC(=O)O3)c1 ZINC000880552521 DD On-Demand Anodyne S1PR2 26 40 COc1cncc(NC(=O)N2CCC(c3cccc(OC)c3)CC2)c1 ZINC000880552524 EH On-Demand Anodyne MTNR1A 17 40 COc1cncc(NC(=O)N2CCC(c3cccc(OC)c3)CC2)c1 ZINC000880552524 EH On-Demand Anodyne MTNR1B 27 40 COc1cncc(NC(=O)N2CCC(c3cccc(OC)c3)CC2)c1 ZINC000880552524 EH On-Demand Anodyne EPHX2 24 44 COc1cncc(NC(=O)N2CCC(c3cccc(OC)c3)CC2)c1 ZINC000880552524 EH On-Demand Anodyne MCHR1 29 46 COc1cncc(NC(=O)N[C@@](C)(CO)c2ccccc2)c1 ZINC000880552525 DE On-Demand Anodyne IMDH_CRYPV 43 40 COc1cncc(NC(=O)N[C@](C)(CO)c2ccccc2)c1 ZINC000880552526 DE On-Demand Anodyne IMDH_CRYPV 43 40 COC[C@@H](C)n1ccc(NC(=O)Nc2cncc(OC)c2)n1 ZINC000880552543 DE On-Demand Anodyne GCK 23 41 COc1cncc(NC(=O)N2CCCC3(CCCC3)C2)c1 ZINC000880552550 CG On-Demand Anodyne EPHX2 32 42 CC(C)(C)OC(=O)NCc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880552555 GF On-Demand Anodyne CA14 17 43 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)Nc1cccnc1 ZINC000880552556 EF On-Demand Anodyne CHRNA7 25 41 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne DRD4 42 34 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne HCRTR1 21 49 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne CHRNA7 17 43 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne CPT1A 72 36 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne PREP 29 42 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne MCHR1 17 45 COc1cncc(NC(=O)N2CCCC[C@H]2CNC(=O)c2ccccc2)c1 ZINC000880552557 FF On-Demand Anodyne ACKR3 63 34 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne DRD4 42 34 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne HCRTR1 21 49 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne CHRNA7 17 43 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne CPT1A 72 36 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne PREP 29 42 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne MCHR1 17 45 COc1cncc(NC(=O)N2CCCC[C@@H]2CNC(=O)c2ccccc2)c1 ZINC000880552558 FF On-Demand Anodyne ACKR3 63 34 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552575 EH On-Demand Anodyne DRD4 34 41 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552575 EH On-Demand Anodyne SIGMAR1 34 40 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552575 EH On-Demand Anodyne NOD2 41 37 COc1cncc(NC(=O)NCC2CCN(CC(F)(F)F)CC2)c1 ZINC000880552577 EE On-Demand Anodyne CCR3 52 43 COc1cncc(NC(=O)NCC2CCN(CC(F)(F)F)CC2)c1 ZINC000880552577 EE On-Demand Anodyne CACNA1I 73 39 COc1cncc(NC(=O)NCC2CCN(CC(F)(F)F)CC2)c1 ZINC000880552577 EE On-Demand Anodyne HPGDS 33 42 COc1ccc(-c2nnc(S)n2CC(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880552583 GD On-Demand Anodyne AVPR1B 56 36 COc1cncc(NC(=O)N2CCN(c3ccnc(C)n3)CC2)c1 ZINC000880552705 ED On-Demand Anodyne PDGFRB 55 43 COc1cncc(NC(=O)N2CCN(c3ccnc(C)n3)CC2)c1 ZINC000880552705 ED On-Demand Anodyne FAAH 20 44 COc1cncc(NC(=O)N2CCN(c3ccnc(C)n3)CC2)c1 ZINC000880552705 ED On-Demand Anodyne DGAT1 19 40 COc1cncc(NC(=O)N[C@@H](C)CCC2CC2)c1 ZINC000880552710 CF On-Demand Anodyne CCR3 49 33 COc1cncc(NC(=O)N[C@H](C)CCC2CC2)c1 ZINC000880552711 CF On-Demand Anodyne CCR3 49 33 NC(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@@H]3C2)cc1 ZINC000880552725 EF On-Demand Anodyne OPRM1 16 44 COc1cncc(NC(=O)N2CCN(c3nc(C)cc(C)n3)CC2)c1 ZINC000880552744 ED On-Demand Anodyne PDGFRB 49 39 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)c1 ZINC000880552748 FF On-Demand Anodyne CACNA1H 62 36 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)c1 ZINC000880552748 FF On-Demand Anodyne CCR3 21 41 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)c1 ZINC000880552748 FF On-Demand Anodyne FAAH 18 44 COc1cncc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)c1 ZINC000880552748 FF On-Demand Anodyne S1PR2 33 49 CCOC(=O)c1csc(CN2Cc3ccccc3N3CCC[C@@H]3C2)n1 ZINC000880552879 FG On-Demand Anodyne TPP2 40 32 COc1ccc2c(C)c(CCC(=O)NCc3cn(C4CCC4)nn3)c(=O)oc2c1 ZINC000880552904 GF On-Demand Anodyne MAOB 24 40 COc1cncc(NC(=O)N2CCOC3(CCOCC3)CC2)c1 ZINC000880552922 DD On-Demand Anodyne EPHX2 15 42 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne HTR1A 50 43 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne DRD2 35 42 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne DRD4 17 45 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne ADRA1A 15 43 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne DRD3 37 45 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552930 DF On-Demand Anodyne HTR7 65 41 COc1cncc(NC(=O)NC[C@@H](O)CCc2ccccc2)c1 ZINC000880552939 DE On-Demand Anodyne ADRB1 41 31 COc1cncc(NC(=O)NC[C@@H](O)CCc2ccccc2)c1 ZINC000880552939 DE On-Demand Anodyne MMP3 25 40 COc1cncc(NC(=O)NC[C@@H](O)CCc2ccccc2)c1 ZINC000880552939 DE On-Demand Anodyne ROCK2 21 41 COc1cncc(NC(=O)NC[C@H](O)CCc2ccccc2)c1 ZINC000880552940 DE On-Demand Anodyne ADRB1 41 31 COc1cncc(NC(=O)NC[C@H](O)CCc2ccccc2)c1 ZINC000880552940 DE On-Demand Anodyne MMP3 25 40 COc1cncc(NC(=O)NC[C@H](O)CCc2ccccc2)c1 ZINC000880552940 DE On-Demand Anodyne ROCK2 21 41 COc1cncc(NC(=O)N2CCN([C@H](C)c3ccsc3)CC2)c1 ZINC000880552943 EG On-Demand Anodyne NPBWR1 40 35 COc1cncc(NC(=O)N2CCN([C@@H](C)c3ccsc3)CC2)c1 ZINC000880552944 EG On-Demand Anodyne NPBWR1 40 35 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552947 CG On-Demand Anodyne HTR1A 25 41 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552947 CG On-Demand Anodyne SLC6A1 63 38 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552947 CG On-Demand Anodyne HTR7 36 41 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552947 CG On-Demand Anodyne CYP2J2 46 32 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c1 ZINC000880552964 EF On-Demand Anodyne OPRL1 16 45 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c1 ZINC000880552964 EF On-Demand Anodyne PDGFRB 40 42 COc1cncc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c1 ZINC000880552964 EF On-Demand Anodyne S1PR2 28 42 COc1cncc(NC(=O)N[C@H](C)CCN2CCN(C)CC2)c1 ZINC000880552971 DD On-Demand Anodyne CCR3 61 38 COc1cncc(NC(=O)N[C@@H](C)CCN2CCN(C)CC2)c1 ZINC000880552972 DD On-Demand Anodyne CCR3 61 38 CC(=O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880552981 BE On-Demand Anodyne OPRL1 16 40 COc1cncc(NC(=O)NCCCC#N)c1 ZINC000880552982 BD On-Demand Mild ADRB1 41 32 O=C1CCC(CN2Cc3ccccc3N3CCC[C@@H]3C2)CC1 ZINC000880552998 CG On-Demand Anodyne OPRL1 15 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne ACE 45 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne OPRM1 41 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CELA1 26 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne ELANE 30 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSD 24 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTRA_BOVIN 58 31 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CASP3 16 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne KLK3 91 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSB 78 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne PAPA1_CARPA 83 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne TRY1_BOVIN 43 31 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CYSP_TRYCR 59 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSG 41 31 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSK 45 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSL 50 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne PREP 36 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CAPNS1 79 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne HLA-DRB1 81 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CELA2A 47 31 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne REN 76 39 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne REN1 42 35 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne LGMN 20 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne MMP11 47 33 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CTSS 32 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CAPN1 108 46 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CASP1 28 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne CAPN2 160 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne PLAU 23 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne TPSAB1 33 50 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne PROC 40 34 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne NPR 79 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne XIAP 51 38 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne PSMB5 60 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne BIRC3 40 33 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880553006 FD On-Demand Anodyne Q6PRC7_IXORI 45 39 COc1cncc(NC(=O)N2CCC(Oc3cc(C)ccn3)CC2)c1 ZINC000880553017 EF On-Demand Anodyne EPHX2 17 40 COc1cncc(NC(=O)NCCCNc2cccc(F)c2)c1 ZINC000880553024 DF On-Demand Anodyne CCR3 42 49 COc1cncc(NC(=O)NCCCNc2cccc(F)c2)c1 ZINC000880553024 DF On-Demand Anodyne MTNR1B 33 40 COc1cncc(NC(=O)NCCCNc2cccc(F)c2)c1 ZINC000880553024 DF On-Demand Anodyne TBK1 33 42 COc1cncc(NC(=O)N2CCOc3cc(N(C)C)ccc32)c1 ZINC000880553029 EF On-Demand Clean KDR 18 45 CCC(=O)NNC(=O)Nc1cncc(OC)c1 ZINC000880553037 BC On-Demand Reactive MTNR1A 20 42 CCC(=O)NNC(=O)Nc1cncc(OC)c1 ZINC000880553037 BC On-Demand Reactive MTNR1B 22 42 COc1cncc(NC(=O)N2CCCCC[C@H]2c2noc(C)n2)c1 ZINC000880553048 EF On-Demand Anodyne CPT1A 64 42 COc1cncc(NC(=O)N2CCCCC[C@@H]2c2noc(C)n2)c1 ZINC000880553049 EF On-Demand Anodyne CPT1A 64 42 COc1cncc(NC(=O)N2CC[C@]3(C2)OCc2ccccc23)c1 ZINC000880553051 EF On-Demand Anodyne NPY5R 37 43 COc1cncc(NC(=O)N2CC[C@@]3(C2)OCc2ccccc23)c1 ZINC000880553052 EF On-Demand Anodyne NPY5R 37 43 COc1cncc(NC(=O)NNC(=O)C23CC4CC(CC(C4)C2)C3)c1 ZINC000880553064 EE On-Demand Reactive EPHX2 35 46 O=C(CN1Cc2ccccc2N2CCC[C@@H]2C1)c1ccccc1F ZINC000880553066 DG On-Demand Anodyne SLC6A1 51 40 COc1cncc(NC(=O)N(C)CC(C)(C)CN2CCOCC2)c1 ZINC000880553071 ED On-Demand Anodyne CASR 21 40 COc1cncc(NC(=O)N2CCN(C(=O)[C@H](C)O)CC2)c1 ZINC000880553072 DC On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)N2CCN(C(=O)[C@@H](C)O)CC2)c1 ZINC000880553073 DC On-Demand Anodyne PDGFRB 41 38 CCC1(CO)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880553075 CE On-Demand Anodyne S1PR2 28 41 c1ccc2c(c1)CN(CCCc1ccncc1)C[C@@H]1CCCN21 ZINC000880553076 DG On-Demand Anodyne SIGMAR1 28 43 COc1cncc(NC(=O)N2CC[C@H]2c2cccc(F)c2)c1 ZINC000880553083 DG On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)N2CC[C@@H]2c2cccc(F)c2)c1 ZINC000880553084 DG On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)N(C)Cc2cccc(OC(C)C)c2)c1 ZINC000880553088 EH On-Demand Anodyne ROCK1 34 56 COc1cncc(NC(=O)N(C)Cc2cccc(OC(C)C)c2)c1 ZINC000880553088 EH On-Demand Anodyne ROCK2 45 56 COc1cncc(NC(=O)N(C)Cc2cccc(OC(C)C)c2)c1 ZINC000880553088 EH On-Demand Anodyne HSD17B2 19 43 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne DRD4 16 40 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne F10 25 43 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne SIGMAR1 15 43 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne NPY1R 31 43 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne CCKAR 39 46 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne CCR3 31 42 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne CHRNA7 19 43 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne CCKBR 54 46 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553090 FE On-Demand Anodyne MCHR1 15 40 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne DRD4 16 40 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne F10 25 43 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne SIGMAR1 15 43 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne NPY1R 31 43 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne CCKAR 39 46 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne CCR3 31 42 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne CHRNA7 19 43 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne CCKBR 54 46 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880553091 FE On-Demand Anodyne MCHR1 15 40 COc1cncc(NC(=O)N2CCC(O)(C(F)(F)F)CC2)c1 ZINC000880553098 DE On-Demand Anodyne S1PR2 28 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553110 EE On-Demand Anodyne CCR3 25 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553110 EE On-Demand Anodyne EPHX2 19 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553113 EE On-Demand Anodyne CCR3 25 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553113 EE On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)NC(C)(C)[C@@H](C)O)c1 ZINC000880553122 CD On-Demand Anodyne IMDH_CRYPV 17 40 COc1cncc(NC(=O)NC(C)(C)[C@H](C)O)c1 ZINC000880553123 CD On-Demand Anodyne IMDH_CRYPV 17 40 O=C(NCc1cn(C2CCC2)nn1)c1ccc2c(c1)CCO2 ZINC000880553128 CD On-Demand Anodyne CA14 15 44 COc1cncc(NC(=O)N(CCO)CCO)c1 ZINC000880553134 CB On-Demand Anodyne ROCK2 16 46 COc1cncc(NC(=O)N2CCC[C@@H](C)[C@H]2C)c1 ZINC000880553139 CF On-Demand Anodyne TRPC6 49 36 COc1cncc(NC(=O)N2CCC[C@@H](C)[C@@H]2C)c1 ZINC000880553140 CF On-Demand Anodyne TRPC6 49 36 COc1cncc(NC(=O)N2CCC[C@H](C)[C@@H]2C)c1 ZINC000880553141 CF On-Demand Anodyne TRPC6 49 36 COc1cncc(NC(=O)N2CCC[C@H](C)[C@H]2C)c1 ZINC000880553142 CF On-Demand Anodyne TRPC6 49 36 COc1cncc(NC(=O)NCc2cccnc2OCC(F)F)c1 ZINC000880553147 EE On-Demand Anodyne ROCK2 17 42 COc1cncc(NC(=O)NCc2cccnc2OCC(F)F)c1 ZINC000880553147 EE On-Demand Anodyne SCN10A 22 40 COc1cncc(NC(=O)NC[C@@H]2CC(=O)N(Cc3ccccc3)C2)c1 ZINC000880553153 FE On-Demand Anodyne TSHR 41 30 COc1cncc(NC(=O)NC[C@@H]2CC(=O)N(Cc3ccccc3)C2)c1 ZINC000880553153 FE On-Demand Anodyne CCR3 38 43 COc1cncc(NC(=O)NC[C@H]2CC(=O)N(Cc3ccccc3)C2)c1 ZINC000880553154 FE On-Demand Anodyne TSHR 41 30 COc1cncc(NC(=O)NC[C@H]2CC(=O)N(Cc3ccccc3)C2)c1 ZINC000880553154 FE On-Demand Anodyne CCR3 38 43 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)C1CC1 ZINC000880553163 CF On-Demand Anodyne HTR1A 15 41 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)C1CC1 ZINC000880553163 CF On-Demand Anodyne SLC6A1 58 37 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)C1CC1 ZINC000880553163 CF On-Demand Anodyne HTR7 22 41 COc1cncc(NC(=O)NCC2(CO)CCOCC2)c1 ZINC000880553164 CD On-Demand Anodyne NAMPT 22 40 COc1cncc(NC(=O)N2CC[C@@H](c3c(F)cccc3F)C2)c1 ZINC000880553180 EG On-Demand Anodyne CCR3 17 46 COc1cncc(NC(=O)N2CC[C@@H](c3c(F)cccc3F)C2)c1 ZINC000880553180 EG On-Demand Anodyne EPHX2 18 41 COc1cncc(NC(=O)N2CC[C@H](c3c(F)cccc3F)C2)c1 ZINC000880553181 EG On-Demand Anodyne CCR3 17 46 COc1cncc(NC(=O)N2CC[C@H](c3c(F)cccc3F)C2)c1 ZINC000880553181 EG On-Demand Anodyne EPHX2 18 41 FCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553194 CG On-Demand Anodyne HTR1A 19 41 FCCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553194 CG On-Demand Anodyne HTR7 26 41 COc1cncc(NC(=O)NC(C)(C)c2ccc(C)nc2)c1 ZINC000880553205 DF On-Demand Anodyne IMDH_CRYPV 60 43 O=C(c1ccccc1)N1CC[C@H](CN2Cc3ccccc3N3CCC[C@@H]3C2)C1 ZINC000880553210 GH On-Demand Anodyne L3MBTL3 70 38 O=C(c1ccccc1)N1CC[C@@H](CN2Cc3ccccc3N3CCC[C@@H]3C2)C1 ZINC000880553211 GH On-Demand Anodyne L3MBTL3 70 38 COc1cncc(NC(=O)N[C@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553217 EF On-Demand Anodyne CTSK 25 41 COc1cncc(NC(=O)N[C@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553217 EF On-Demand Anodyne CAPNS1 52 32 COc1cncc(NC(=O)N[C@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553217 EF On-Demand Anodyne CAPN1 48 36 COc1cncc(NC(=O)N[C@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553217 EF On-Demand Anodyne CAPN2 69 38 COc1cncc(NC(=O)N[C@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553217 EF On-Demand Anodyne NPR 57 32 COc1cncc(NC(=O)N[C@@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553218 EF On-Demand Anodyne CTSK 25 41 COc1cncc(NC(=O)N[C@@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553218 EF On-Demand Anodyne CAPNS1 52 32 COc1cncc(NC(=O)N[C@@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553218 EF On-Demand Anodyne CAPN1 48 36 COc1cncc(NC(=O)N[C@@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553218 EF On-Demand Anodyne CAPN2 69 38 COc1cncc(NC(=O)N[C@@H](C)CC(=O)OCc2ccccc2)c1 ZINC000880553218 EF On-Demand Anodyne NPR 57 32 COc1cncc(NC(=O)N2CCN(c3cc(OC)ncn3)CC2)c1 ZINC000880553221 ED On-Demand Anodyne PDGFRB 62 46 CCOC(=O)COCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553227 DE On-Demand Anodyne SLC6A1 56 37 COc1cncc(NC(=O)NC(C)(C)CCN2CCN(C)CC2)c1 ZINC000880553232 ED On-Demand Anodyne FGFR1 24 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(N2CCOCC2)nc1 ZINC000880553234 ED On-Demand Anodyne HPGDS 22 49 O=C(NCc1cn(C2CCC2)nn1)c1ccc(N2CCOCC2)nc1 ZINC000880553234 ED On-Demand Anodyne NAMPT 16 47 COc1cncc(NC(=O)NCc2ccccc2CN2CC[C@H](O)C2)c1 ZINC000880553235 FD On-Demand Anodyne CCR3 58 45 COc1cncc(NC(=O)NCc2ccccc2CN2CC[C@H](O)C2)c1 ZINC000880553235 FD On-Demand Anodyne MCHR1 30 42 COc1cncc(NC(=O)NCc2ccccc2CN2CC[C@@H](O)C2)c1 ZINC000880553236 FD On-Demand Anodyne CCR3 58 45 COc1cncc(NC(=O)NCc2ccccc2CN2CC[C@@H](O)C2)c1 ZINC000880553236 FD On-Demand Anodyne MCHR1 30 42 COc1cncc(NC(=O)NCCc2ccnn2C)c1 ZINC000880553247 CD On-Demand Anodyne HTR2A 28 41 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCC1 ZINC000880553253 DE On-Demand Anodyne SLC6A1 53 34 O=C(CCN1Cc2ccccc2N2CCC[C@@H]2C1)N1CCCC1 ZINC000880553253 DE On-Demand Anodyne PREP 53 38 O=C1c2ccccc2C(=O)N1OCCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553254 GG On-Demand Anodyne HTR1A 18 40 COc1cncc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880553268 FE On-Demand Anodyne CACNA1I 55 36 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553275 GF On-Demand Anodyne LTA4H 50 37 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553275 GF On-Demand Anodyne HRH3 42 41 CS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553275 GF On-Demand Anodyne PSMB1 40 34 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne INHA 42 34 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne ROCK1 17 42 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne MTNR1A 21 40 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne MTNR1B 26 40 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne ROCK2 31 42 COc1cncc(NC(=O)N(C)CCCc2ccccc2)c1 ZINC000880553279 CG On-Demand Anodyne CRTM 37 42 COc1cncc(NC(=O)N[C@@H](CC(C)C)C(=O)NCCN(C)C)c1 ZINC000880553285 FD On-Demand Anodyne ANPEP 26 53 COc1cncc(NC(=O)N[C@@H](CC(C)C)C(=O)NCCN(C)C)c1 ZINC000880553285 FD On-Demand Anodyne CTSK 26 44 COc1cncc(NC(=O)N[C@@H](CC(C)C)C(=O)NCCN(C)C)c1 ZINC000880553285 FD On-Demand Anodyne CTSL 25 41 COc1cncc(NC(=O)N[C@@H](CC(C)C)C(=O)NCCN(C)C)c1 ZINC000880553285 FD On-Demand Anodyne CTSS 15 42 COc1cncc(NC(=O)N2CCC(Cn3ccnn3)CC2)c1 ZINC000880553310 DD On-Demand Anodyne PDGFRB 31 40 COc1cncc(NC(=O)NCCCNC(=O)C(C)C)c1 ZINC000880553320 CD On-Demand Anodyne MTNR1A 23 40 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553326 CG On-Demand Anodyne HTR1A 25 41 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553326 CG On-Demand Anodyne SLC6A1 63 38 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553326 CG On-Demand Anodyne HTR7 36 41 CCC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553326 CG On-Demand Anodyne CYP2J2 46 32 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553329 DE On-Demand Anodyne HTR1A 23 40 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553329 DE On-Demand Anodyne SLC6A1 50 39 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553329 DE On-Demand Anodyne HTR7 36 40 CN(C)C(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553329 DE On-Demand Anodyne CYP2J2 44 31 COc1cncc(NC(=O)NC2CCN(CC3CCCC3)CC2)c1 ZINC000880553331 EF On-Demand Anodyne SSTR5 40 36 COc1cncc(NC(=O)NC2CCN(CC3CCCC3)CC2)c1 ZINC000880553331 EF On-Demand Anodyne CCR3 60 51 COc1cncc(NC(=O)NC2CCN(CC3CCCC3)CC2)c1 ZINC000880553331 EF On-Demand Anodyne EPHX2 50 39 COc1cncc(NC(=O)NC2CCN(CC3CCCC3)CC2)c1 ZINC000880553331 EF On-Demand Anodyne CXCR3 23 48 COc1cncc(NC(=O)NC2CCN(CC3CCCC3)CC2)c1 ZINC000880553331 EF On-Demand Anodyne MCHR1 17 47 COc1cncc(NC(=O)NCc2cccc(N(C)C)n2)c1 ZINC000880553355 DD On-Demand Anodyne ROCK2 31 43 COc1cncc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880553449 FE On-Demand Anodyne CACNA1I 55 36 COc1cncc(NC(=O)NCCc2ccn(C)n2)c1 ZINC000880553469 CD On-Demand Anodyne QPCT 16 42 COc1cncc(NC(=O)N2CCN(c3cccc(C#N)n3)CC2)c1 ZINC000880553475 ED On-Demand Mild PDGFRB 53 41 COc1cncc(NC(=O)N2CCN(c3cccc(C#N)n3)CC2)c1 ZINC000880553475 ED On-Demand Mild FAAH 21 44 COc1cncc(NC(=O)N2CCN(c3cccc(C#N)n3)CC2)c1 ZINC000880553475 ED On-Demand Mild GALR2 41 34 COc1cncc(NC(=O)N2CC[C@H](c3cccc(C)c3)C2)c1 ZINC000880553498 DG On-Demand Anodyne MCHR1 19 42 COc1cncc(NC(=O)N2CC[C@H](c3cccc(C)c3)C2)c1 ZINC000880553498 DG On-Demand Anodyne MGEA5 23 41 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(C)c3)C2)c1 ZINC000880553499 DG On-Demand Anodyne MCHR1 19 42 COc1cncc(NC(=O)N2CC[C@@H](c3cccc(C)c3)C2)c1 ZINC000880553499 DG On-Demand Anodyne MGEA5 23 41 COc1cncc(NC(=O)NCc2cccc(C(=O)N3CCOCC3)c2)c1 ZINC000880553507 FD On-Demand Anodyne ROCK2 43 46 COc1cncc(NC(=O)NCc2cccc(C(=O)N3CCOCC3)c2)c1 ZINC000880553507 FD On-Demand Anodyne MTOR 44 37 COc1cncc(NC(=O)NCc2cccc(C(=O)N3CCOCC3)c2)c1 ZINC000880553507 FD On-Demand Anodyne EPHX2 28 45 COc1cncc(NC(=O)NCc2cccc(C(=O)N3CCOCC3)c2)c1 ZINC000880553507 FD On-Demand Anodyne NAMPT 42 45 COc1cncc(NC(=O)N2CCN(c3ccc(C)cc3)CC2)c1 ZINC000880553536 EF On-Demand Anodyne DRD4 25 42 COc1cncc(NC(=O)N2CCN(c3ccc(C)cc3)CC2)c1 ZINC000880553536 EF On-Demand Anodyne HTR1B 15 48 COc1cncc(NC(=O)N2CCN(c3ccc(C)cc3)CC2)c1 ZINC000880553536 EF On-Demand Anodyne PDGFRB 53 47 COc1cncc(NC(=O)N2CCN(c3ccc(C)cc3)CC2)c1 ZINC000880553536 EF On-Demand Anodyne CCKAR 27 42 Oc1nc(CN2Cc3ccccc3N3CCC[C@@H]3C2)nc2c1COCC2 ZINC000880553540 FE On-Demand Anodyne WNT3A 44 31 COc1cncc(NC(=O)N[C@H]2CCCN(Cc3ccccn3)C2=O)c1 ZINC000880553547 FD On-Demand Anodyne CCKAR 18 43 COc1cncc(NC(=O)N[C@@H]2CCCN(Cc3ccccn3)C2=O)c1 ZINC000880553548 FD On-Demand Anodyne CCKAR 18 43 COc1cncc(NC(=O)N2CCC(OCc3ccccc3F)CC2)c1 ZINC000880553550 FG On-Demand Anodyne CCR3 19 43 COc1cncc(NC(=O)N2CCC(OCc3ccccc3F)CC2)c1 ZINC000880553550 FG On-Demand Anodyne SCD1 21 44 COc1cncc(NC(=O)N(C)C[C@H]2CCN(C(C)=O)C2)c1 ZINC000880553561 DD On-Demand Anodyne CCR3 15 41 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(C(C)=O)C2)c1 ZINC000880553562 DD On-Demand Anodyne CCR3 15 41 COc1cncc(NC(=O)N2CCC(CCCN3CCCC3)CC2)c1 ZINC000880553565 EG On-Demand Anodyne PDGFRB 41 40 COc1cncc(NC(=O)N2CCC(CCCN3CCCC3)CC2)c1 ZINC000880553565 EG On-Demand Anodyne NPY1R 40 33 COc1cncc(NC(=O)N2CCC(CCCN3CCCC3)CC2)c1 ZINC000880553565 EG On-Demand Anodyne CCR3 28 45 COc1cncc(NC(=O)N2CCC(CCCN3CCCC3)CC2)c1 ZINC000880553565 EG On-Demand Anodyne CHRNA7 19 40 COc1cncc(NC(=O)N[C@H]2CCN(C(C)=O)c3ccccc32)c1 ZINC000880553580 EF On-Demand Anodyne CCKAR 18 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(C)=O)c3ccccc32)c1 ZINC000880553581 EF On-Demand Anodyne CCKAR 18 40 COc1cncc(NC(=O)NCc2cccc(OC(C)(C)C)n2)c1 ZINC000880553596 EF On-Demand Anodyne ROCK2 20 42 COc1cncc(NC(=O)NC[C@@H](C)COc2ccccc2OC)c1 ZINC000880553598 EF On-Demand Anodyne ADRB1 45 35 COc1cncc(NC(=O)NC[C@@H](C)COc2ccccc2OC)c1 ZINC000880553598 EF On-Demand Anodyne ROCK2 15 42 COc1cncc(NC(=O)NC[C@H](C)COc2ccccc2OC)c1 ZINC000880553599 EF On-Demand Anodyne ADRB1 45 35 COc1cncc(NC(=O)NC[C@H](C)COc2ccccc2OC)c1 ZINC000880553599 EF On-Demand Anodyne ROCK2 15 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(S(=O)(=O)C(F)(F)F)cc1 ZINC000880553604 GE On-Demand Anodyne CA14 25 53 O=C1CCC(CN2Cc3ccccc3N3CCC[C@H]3C2)CC1 ZINC000880553606 CG On-Demand Anodyne OPRL1 15 44 O=C(NCCCN1Cc2ccccc2N2CCC[C@H]2C1)C(F)(F)F ZINC000880553635 EF On-Demand Anodyne DRD2 21 41 O=C(NCCCN1Cc2ccccc2N2CCC[C@H]2C1)C(F)(F)F ZINC000880553635 EF On-Demand Anodyne DRD3 33 48 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880553636 EE On-Demand Clean HTR1B 16 50 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880553636 EE On-Demand Clean PDGFRB 58 45 COc1ccc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880553636 EE On-Demand Clean FAAH 23 48 COc1cncc(NC(=O)N(Cc2ccccc2[N+](=O)[O-])C2CC2)c1 ZINC000880553637 EG On-Demand Bother COLA 125 45 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP13 31 45 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP3 35 45 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP8 18 40 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne S1PR2 28 42 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP9 22 45 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne PKM 29 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne TGM2 84 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP7 36 40 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne MMP1 31 45 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne F13A1 96 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)c1 ZINC000880553646 GD On-Demand Anodyne NAMPT 41 43 COc1cncc(NC(=O)N(CCO)Cc2ccc(C)cc2)c1 ZINC000880553655 DE On-Demand Anodyne ROCK1 15 52 COc1cncc(NC(=O)N(CCO)Cc2ccc(C)cc2)c1 ZINC000880553655 DE On-Demand Anodyne ROCK2 28 52 COc1cncc(NC(=O)N2CCNC(=O)[C@@H]2c2ccccc2C(F)(F)F)c1 ZINC000880553658 GF On-Demand Anodyne RBP4 82 38 COc1cncc(NC(=O)N2CCNC(=O)[C@@H]2c2ccccc2C(F)(F)F)c1 ZINC000880553658 GF On-Demand Anodyne TRPM8 45 44 COc1cncc(NC(=O)N2CCNC(=O)[C@H]2c2ccccc2C(F)(F)F)c1 ZINC000880553659 GF On-Demand Anodyne RBP4 82 38 COc1cncc(NC(=O)N2CCNC(=O)[C@H]2c2ccccc2C(F)(F)F)c1 ZINC000880553659 GF On-Demand Anodyne TRPM8 45 44 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive HTR1A 95 53 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive DRD2 62 53 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive DRD4 55 53 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive ADRA1D 33 41 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive HTR2A 40 43 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive HTR2C 18 41 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive DRD3 77 46 COc1cncc(NC(=O)NNC(=O)CCN2CCN(c3ccccc3)CC2)c1 ZINC000880553670 GD On-Demand Reactive HTR7 96 41 COc1cncc(NC(=O)N2[C@H]3CC[C@H]2CN(C(=O)OC(C)(C)C)CC3)c1 ZINC000880553676 GG On-Demand Anodyne GPR119 43 39 COc1cncc(NC(=O)N[C@@H](CO)Cc2ccccc2)c1 ZINC000880553682 DD On-Demand Anodyne MME 50 39 COc1cncc(NC(=O)N[C@@H](CO)Cc2ccccc2)c1 ZINC000880553682 DD On-Demand Anodyne ANPEP 61 33 COc1cncc(NC(=O)N[C@@H](CO)Cc2ccccc2)c1 ZINC000880553682 DD On-Demand Anodyne TIMP3 41 33 COc1cncc(NC(=O)N2C[C@@H](C)C[C@@H]2c2cccnc2)c1 ZINC000880553691 DG On-Demand Anodyne CHRNA7 20 47 COc1cncc(NC(=O)N2C[C@@H](C)C[C@H]2c2cccnc2)c1 ZINC000880553692 DG On-Demand Anodyne CHRNA7 20 47 COc1cncc(NC(=O)N2C[C@H](C)C[C@@H]2c2cccnc2)c1 ZINC000880553693 DG On-Demand Anodyne CHRNA7 20 47 COc1cncc(NC(=O)N2C[C@H](C)C[C@H]2c2cccnc2)c1 ZINC000880553694 DG On-Demand Anodyne CHRNA7 20 47 COc1cncc(NC(=O)N(CCCOc2ccccc2)C2CCOCC2)c1 ZINC000880553695 GH On-Demand Anodyne CASR 23 40 COc1cncc(NC(=O)N(CCCOc2ccccc2)C2CCOCC2)c1 ZINC000880553695 GH On-Demand Anodyne ROCK2 21 41 COc1cncc(NC(=O)N2CC[C@@]3(CC[C@H](C)C3)C2)c1 ZINC000880553705 CG On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)N2CC[C@]3(CC[C@H](C)C3)C2)c1 ZINC000880553706 CG On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)N2CC[C@@]3(CC[C@@H](C)C3)C2)c1 ZINC000880553707 CG On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)N2CC[C@]3(CC[C@@H](C)C3)C2)c1 ZINC000880553708 CG On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne P2RY12 68 37 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne MC4R 47 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne TACR2 24 54 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne TRY2_BOVIN 86 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne CYSP_TRYCR 27 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne TIMP3 42 33 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne CCKBR 18 44 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne ACE2 44 34 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne MC1R 15 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne ST14 40 34 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne FPR1 29 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553721 GD On-Demand Anodyne PSMB8 59 39 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne P2RY12 68 37 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne MC4R 47 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne TACR2 24 54 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne TRY2_BOVIN 86 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne CYSP_TRYCR 27 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne TIMP3 42 33 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne CCKBR 18 44 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne ACE2 44 34 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne MC1R 15 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne ST14 40 34 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne FPR1 29 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCOCC2)c1 ZINC000880553722 GD On-Demand Anodyne PSMB8 59 39 COc1cncc(NC(=O)N2CCO[C@@]3(CCOC3)C2)c1 ZINC000880553732 CD On-Demand Anodyne EPHX2 22 43 COc1cncc(NC(=O)N2CCO[C@]3(CCOC3)C2)c1 ZINC000880553733 CD On-Demand Anodyne EPHX2 22 43 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne HTR1A 30 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne DRD2 16 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne HTR2A 15 40 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne SLC6A1 87 37 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne OPRL1 19 44 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne HTR7 55 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne CYP2J2 44 31 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553740 CD On-Demand Anodyne BIRC2 49 33 COc1cncc(NC(=O)N2CCCC3(CC3)C2)c1 ZINC000880553741 CE On-Demand Anodyne EPHX2 31 41 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne PDGFRB 66 46 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne TRPV1 19 50 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne FAAH 26 42 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne S1PR2 26 42 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne RBP4 20 48 COc1cncc(NC(=O)N2CCN(c3ncccc3F)CC2)c1 ZINC000880553749 ED On-Demand Anodyne LIMK2 19 49 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553785 DD On-Demand Anodyne CCR3 46 38 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553785 DD On-Demand Anodyne EPHX2 23 43 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553786 DD On-Demand Anodyne CCR3 46 38 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553786 DD On-Demand Anodyne EPHX2 23 43 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553787 DD On-Demand Anodyne CCR3 46 38 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553787 DD On-Demand Anodyne EPHX2 23 43 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553788 DD On-Demand Anodyne CCR3 46 38 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880553788 DD On-Demand Anodyne EPHX2 23 43 COc1cncc(NC(=O)N2CCc3c(cccc3[N+](=O)[O-])C2)c1 ZINC000880553790 EF On-Demand Bother TAAR1 31 43 COc1cncc(NC(=O)N2CCc3c(cccc3[N+](=O)[O-])C2)c1 ZINC000880553790 EF On-Demand Bother P2RY14 40 32 COCC1(O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880553802 CD On-Demand Anodyne PDGFRB 43 36 COCC1(O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880553802 CD On-Demand Anodyne S1PR2 31 46 FCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553804 CG On-Demand Anodyne HTR1A 19 41 FCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553804 CG On-Demand Anodyne HTR7 26 41 CCC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553805 CF On-Demand Anodyne SLC6A1 42 32 COc1cncc(NC(=O)N(CCCO)Cc2cccc(Cl)c2)c1 ZINC000880553808 EG On-Demand Anodyne ROCK1 20 50 COc1cncc(NC(=O)N(CCCO)Cc2cccc(Cl)c2)c1 ZINC000880553808 EG On-Demand Anodyne ROCK2 33 50 O=C(c1ccccc1)N1CC[C@H](CN2Cc3ccccc3N3CCC[C@H]3C2)C1 ZINC000880553809 GH On-Demand Anodyne L3MBTL3 70 38 O=C(c1ccccc1)N1CC[C@@H](CN2Cc3ccccc3N3CCC[C@H]3C2)C1 ZINC000880553810 GH On-Demand Anodyne L3MBTL3 70 38 CCOC(=O)COCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553815 DE On-Demand Anodyne SLC6A1 56 37 COc1cncc(NC(=O)N[C@H]2CCN(C(C)=O)C[C@@H]2C)c1 ZINC000880553821 DD On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(C)=O)C[C@@H]2C)c1 ZINC000880553822 DD On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(C)=O)C[C@H]2C)c1 ZINC000880553823 DD On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@H]2CCN(C(C)=O)C[C@H]2C)c1 ZINC000880553824 DD On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N2C[C@H](O)C[C@@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000880553831 GG On-Demand Anodyne TRPM8 44 40 COc1cncc(NC(=O)N2C[C@@H](O)C[C@@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000880553832 GG On-Demand Anodyne TRPM8 44 40 COc1cncc(NC(=O)N2C[C@@H](O)C[C@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000880553833 GG On-Demand Anodyne TRPM8 44 40 COc1cncc(NC(=O)N2C[C@H](O)C[C@H]2c2ccc(C(F)(F)F)cc2)c1 ZINC000880553834 GG On-Demand Anodyne TRPM8 44 40 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne CA2 31 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne CA1 29 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne CA7 20 40 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne CA12 19 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne CA9 27 42 NS(=O)(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880553845 FE On-Demand Anodyne A6YCJ1_9METZ 15 40 COc1cncc(NC(=O)N2CC[C@]3(CCN(C(=O)OC(C)(C)C)C3)C2)c1 ZINC000880553866 GF On-Demand Anodyne EPHX2 32 43 COc1cncc(NC(=O)N2CC[C@]3(CCN(C(=O)OC(C)(C)C)C3)C2)c1 ZINC000880553866 GF On-Demand Anodyne GPR119 15 42 COc1cncc(NC(=O)N2CC[C@@]3(CCN(C(=O)OC(C)(C)C)C3)C2)c1 ZINC000880553867 GF On-Demand Anodyne EPHX2 32 43 COc1cncc(NC(=O)N2CC[C@@]3(CCN(C(=O)OC(C)(C)C)C3)C2)c1 ZINC000880553867 GF On-Demand Anodyne GPR119 15 42 COc1cncc(NC(=O)N2CCC(CCCn3ccnc3)CC2)c1 ZINC000880553877 EG On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)N2CCC(CCCn3ccnc3)CC2)c1 ZINC000880553877 EG On-Demand Anodyne QPCT 38 45 CC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880553882 DH On-Demand Anodyne HTR1A 16 46 CC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@@H]3C2)c1 ZINC000880553882 DH On-Demand Anodyne DRD2 18 42 O=C(NCc1cn(C2CCC2)nn1)c1cc(-c2ccccc2)on1 ZINC000880553886 DF On-Demand Anodyne HDAC10 15 45 COc1cncc(NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)c1 ZINC000880553897 DD On-Demand Anodyne EPHX2 44 46 COc1cncc(NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)c1 ZINC000880553898 DD On-Demand Anodyne EPHX2 44 46 COc1cncc(NC(=O)N2C[C@H](C)C[C@H]2c2cccc(OC)c2)c1 ZINC000880553910 EH On-Demand Anodyne TAAR1 22 40 COc1cncc(NC(=O)N2C[C@H](C)C[C@@H]2c2cccc(OC)c2)c1 ZINC000880553911 EH On-Demand Anodyne TAAR1 22 40 COc1cncc(NC(=O)N2C[C@@H](C)C[C@@H]2c2cccc(OC)c2)c1 ZINC000880553912 EH On-Demand Anodyne TAAR1 22 40 COc1cncc(NC(=O)N2C[C@@H](C)C[C@H]2c2cccc(OC)c2)c1 ZINC000880553913 EH On-Demand Anodyne TAAR1 22 40 COc1cncc(NC(=O)NCC[C@@H](C)N2CCCCC2)c1 ZINC000880553914 DE On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NCC[C@@H](C)N2CCCCC2)c1 ZINC000880553914 DE On-Demand Anodyne CCR5 15 41 COc1cncc(NC(=O)NCC[C@H](C)N2CCCCC2)c1 ZINC000880553915 DE On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NCC[C@H](C)N2CCCCC2)c1 ZINC000880553915 DE On-Demand Anodyne CCR5 15 41 CCOP(=O)(OCC)[C@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553922 FG On-Demand Anodyne ADAM9 50 33 CCOP(=O)(OCC)[C@@H](O)CN1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880553923 FG On-Demand Anodyne ADAM9 50 33 COc1cncc(NC(=O)NCCCNc2ccccc2F)c1 ZINC000880553928 DF On-Demand Anodyne CCR3 22 42 COc1cncc(NC(=O)NC23CCC(CC2)C3)c1 ZINC000880553930 CF On-Demand Anodyne EPHX2 53 53 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCc1cn(C2CCC2)nn1 ZINC000880553936 FD On-Demand Anodyne APP 45 34 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCc1cn(C2CCC2)nn1 ZINC000880553936 FD On-Demand Anodyne CA14 17 43 COc1cncc(NC(=O)N2CCC(C)(CO)CC2)c1 ZINC000880553937 CD On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCO[C@@H](CCc3ccccc3)C2)c1 ZINC000880553965 EF On-Demand Anodyne DRD4 15 50 COc1cncc(NC(=O)N2CCO[C@@H](CCc3ccccc3)C2)c1 ZINC000880553965 EF On-Demand Anodyne FAAH 18 40 COc1cncc(NC(=O)N2CCO[C@H](CCc3ccccc3)C2)c1 ZINC000880553966 EF On-Demand Anodyne DRD4 15 50 COc1cncc(NC(=O)N2CCO[C@H](CCc3ccccc3)C2)c1 ZINC000880553966 EF On-Demand Anodyne FAAH 18 40 COc1cncc(NC(=O)N[C@@H](C)[C@H](O)Cc2ccccc2)c1 ZINC000880553969 DE On-Demand Anodyne FPR1 30 40 COc1cncc(NC(=O)N[C@@H](C)[C@@H](O)Cc2ccccc2)c1 ZINC000880553970 DE On-Demand Anodyne FPR1 30 40 COc1cncc(NC(=O)N[C@H](C)[C@H](O)Cc2ccccc2)c1 ZINC000880553971 DE On-Demand Anodyne FPR1 30 40 COc1cncc(NC(=O)N[C@H](C)[C@@H](O)Cc2ccccc2)c1 ZINC000880553972 DE On-Demand Anodyne FPR1 30 40 NC(=O)NC(=O)OCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880553979 ED On-Demand Anodyne SLC6A1 47 37 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3Cl)C2)c1 ZINC000880553988 EG On-Demand Anodyne PDE3A 33 45 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3Cl)C2)c1 ZINC000880553988 EG On-Demand Anodyne PDE3B 37 45 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3Cl)C2)c1 ZINC000880553988 EG On-Demand Anodyne EPHX2 26 45 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3Cl)C2)c1 ZINC000880553988 EG On-Demand Anodyne SCD1 37 56 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccc3Cl)C2)c1 ZINC000880553988 EG On-Demand Anodyne SCD 22 44 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3Cl)C2)c1 ZINC000880553989 EG On-Demand Anodyne PDE3A 33 45 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3Cl)C2)c1 ZINC000880553989 EG On-Demand Anodyne PDE3B 37 45 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3Cl)C2)c1 ZINC000880553989 EG On-Demand Anodyne EPHX2 26 45 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3Cl)C2)c1 ZINC000880553989 EG On-Demand Anodyne SCD1 37 56 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccc3Cl)C2)c1 ZINC000880553989 EG On-Demand Anodyne SCD 22 44 COc1cncc(NC(=O)N2CCN(C(=O)CO)CC2)c1 ZINC000880553999 CB On-Demand Anodyne PDGFRB 47 37 COc1cncc(NC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)c1 ZINC000880554000 EE On-Demand Anodyne CACNA1I 45 32 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne CA2 21 42 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne BMP1 15 42 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne CA1 45 42 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne RAF1 17 43 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne CA12 36 42 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne CA9 37 42 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne MTCA1 40 41 COc1cncc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)c1 ZINC000880554001 EE On-Demand Anodyne P96878_MYCTU 47 42 c1ccc2c(c1)CN(CCN1CCCCC1)C[C@@H]1CCCN21 ZINC000880554011 CF On-Demand Anodyne SIGMAR1 23 43 COc1cncc(NC(=O)N2CCN(S(C)(=O)=O)c3ccccc3C2)c1 ZINC000880554012 GD On-Demand Anodyne NPY5R 24 43 COc1cncc(NC(=O)NC2CCC(CN(C)C)CC2)c1 ZINC000880554013 DE On-Demand Anodyne EPHX2 43 36 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne ACE 22 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne MME 71 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne ANPEP 47 31 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne FCER2 64 36 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne TACR2 16 48 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CTSB 36 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne PAPA1_CARPA 68 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CTSK 20 44 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CTSL 64 45 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne TIMP3 78 37 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CAPNS1 51 31 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne MMP3 29 45 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne GRIA1 46 38 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne HLA-DRB1 48 33 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne PTPRA 63 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne PTPN1 18 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CTSS 29 45 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CAPN1 36 42 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CAPN2 35 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne ACE2 49 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne CTSV 54 38 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne FPR1 57 44 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne BLA1_STEMA 56 37 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne PSMB8 51 33 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)NCCN(C)C)c1 ZINC000880554026 GD On-Demand Anodyne GPR142 50 39 COc1cncc(NC(=O)N2CCN(C3=NCC(C)(C)S3)CC2)c1 ZINC000880554030 EE On-Demand Anodyne PDGFRB 44 37 COc1cncc(NC(=O)N2CCCN(CC(F)F)CC2)c1 ZINC000880554034 DD On-Demand Anodyne PDGFRB 41 35 c1ccc2c(c1)CN(CCc1ccncc1)C[C@@H]1CCCN21 ZINC000880554036 CG On-Demand Anodyne SIGMAR1 17 42 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCCC1 ZINC000880554049 EF On-Demand Anodyne SLC6A1 50 34 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCCC1 ZINC000880554049 EF On-Demand Anodyne PREP 48 37 COCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554058 CF On-Demand Anodyne HTR1A 31 46 COCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554058 CF On-Demand Anodyne DRD2 18 42 COCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554058 CF On-Demand Anodyne DRD3 19 42 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3OC)CC2)c1 ZINC000880554071 GD On-Demand Anodyne HTR1A 22 42 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3OC)CC2)c1 ZINC000880554071 GD On-Demand Anodyne DRD4 28 45 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3OC)CC2)c1 ZINC000880554071 GD On-Demand Anodyne PDGFRB 58 40 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3OC)CC2)c1 ZINC000880554071 GD On-Demand Anodyne FAAH 18 47 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3OC)CC2)c1 ZINC000880554071 GD On-Demand Anodyne RBP4 19 40 COc1cncc(NC(=O)N2CCO[C@@]3(CCc4ccccc43)C2)c1 ZINC000880554079 EF On-Demand Anodyne EPHX2 23 40 COc1cncc(NC(=O)N2CCO[C@]3(CCc4ccccc43)C2)c1 ZINC000880554080 EF On-Demand Anodyne EPHX2 23 40 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C2CC2)c1 ZINC000880554085 EG On-Demand Bother MMP2 18 41 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C2CC2)c1 ZINC000880554085 EG On-Demand Bother MMP8 35 41 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C2CC2)c1 ZINC000880554085 EG On-Demand Bother MMP9 18 41 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C2CC2)c1 ZINC000880554085 EG On-Demand Bother MMP1 25 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccn3)C2)c1 ZINC000880554123 DD On-Demand Anodyne DRD4 19 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccn3)C2)c1 ZINC000880554123 DD On-Demand Anodyne EPHX2 37 40 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccn3)C2)c1 ZINC000880554124 DD On-Demand Anodyne DRD4 19 41 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccn3)C2)c1 ZINC000880554124 DD On-Demand Anodyne EPHX2 37 40 COc1cncc(NC(=O)N2CCC(c3cccnc3)CC2)c1 ZINC000880554137 DF On-Demand Anodyne CHRNA7 35 44 COc1cncc(NC(=O)N2CCC(c3cccnc3)CC2)c1 ZINC000880554137 DF On-Demand Anodyne EPHX2 22 44 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880554146 EE On-Demand Anodyne CCR3 33 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cncc(OC)c1 ZINC000880554147 EE On-Demand Anodyne CCR3 33 40 COc1cncc(NC(=O)NC2CCC(F)(F)CC2)c1 ZINC000880554151 CF On-Demand Anodyne EPHX2 49 37 COc1cncc(NC(=O)N[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000880554158 EE On-Demand Anodyne ROCK2 23 40 COc1cncc(NC(=O)N[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000880554159 EE On-Demand Anodyne ROCK2 23 40 O=C1CCC(=O)N1CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554161 DD On-Demand Anodyne HTR1A 18 44 COc1cncc(NC(=O)NCc2ccnc(OC(C)C)c2)c1 ZINC000880554166 DF On-Demand Anodyne ROCK2 28 46 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554168 EF On-Demand Anodyne HTR1A 32 41 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554168 EF On-Demand Anodyne DRD2 27 53 CC(C)(C)OC(=O)NCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554168 EF On-Demand Anodyne DRD3 31 43 COc1cncc(NC(=O)N2CCc3ccc(F)cc3C2)c1 ZINC000880554171 DF On-Demand Anodyne HDAC6 32 42 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne HRH2 32 49 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne ROCK1 40 46 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne MTNR1A 26 40 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne MTNR1B 32 40 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne ROCK2 63 56 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne NAMPT 41 42 COCCCOc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880554176 EF On-Demand Anodyne PDS 43 37 CC[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554194 EF On-Demand Anodyne ROCK1 16 42 CC[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554194 EF On-Demand Anodyne ROCK2 26 46 CC[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554194 EF On-Demand Anodyne NPY5R 33 42 CC[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554194 EF On-Demand Anodyne PTGES 23 40 CC[C@@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554195 EF On-Demand Anodyne ROCK1 16 42 CC[C@@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554195 EF On-Demand Anodyne ROCK2 26 46 CC[C@@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554195 EF On-Demand Anodyne NPY5R 33 42 CC[C@@H](O)CN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880554195 EF On-Demand Anodyne PTGES 23 40 COc1cncc(NC(=O)N[C@H](c2cccnc2)C2CC2)c1 ZINC000880554197 CF On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N[C@@H](c2cccnc2)C2CC2)c1 ZINC000880554198 CF On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N2CCC(CCCN(C)C)CC2)c1 ZINC000880554204 DF On-Demand Anodyne PDGFRB 39 40 COc1cncc(NC(=O)NC2CCN([C@@H](C)c3ccncc3)CC2)c1 ZINC000880554210 FF On-Demand Anodyne EPHX2 45 42 COc1cncc(NC(=O)NC2CCN([C@H](C)c3ccncc3)CC2)c1 ZINC000880554211 FF On-Demand Anodyne EPHX2 45 42 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554216 DF On-Demand Anodyne HTR1A 27 42 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554216 DF On-Demand Anodyne CHRM1 16 41 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554216 DF On-Demand Anodyne SLC6A1 72 36 CCOC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554216 DF On-Demand Anodyne CHRM4 16 41 COc1cncc(NC(=O)N2CCc3c(F)cccc3C2)c1 ZINC000880554220 DF On-Demand Anodyne DRD4 41 32 COc1cncc(NC(=O)N2CCc3c(F)cccc3C2)c1 ZINC000880554220 DF On-Demand Anodyne P2RY14 48 35 COc1cncc(NC(=O)N2CCN(c3nc(C)c(C)s3)CC2)c1 ZINC000880554238 EF On-Demand Anodyne PDGFRB 43 37 COc1cncc(NC(=O)N2CCC(c3ccccn3)CC2)c1 ZINC000880554246 DF On-Demand Anodyne PDGFRB 48 41 COc1cncc(NC(=O)N2CCC(c3ccccn3)CC2)c1 ZINC000880554246 DF On-Demand Anodyne EPHX2 21 41 COc1cncc(NC(=O)N2CCC(c3ccccn3)CC2)c1 ZINC000880554246 DF On-Demand Anodyne SMO 16 46 COC[C@@H](O)CCNC(=O)Nc1cncc(OC)c1 ZINC000880554253 CC On-Demand Anodyne ADRB1 42 32 COc1cncc(NC(=O)NCCC(=O)N2CCCCC2)c1 ZINC000880554256 DD On-Demand Anodyne HRH2 19 43 COc1cncc(NC(=O)N2CCC[C@H]2C(=O)NCc2ccco2)c1 ZINC000880554258 ED On-Demand Anodyne F2 38 44 COc1cncc(NC(=O)N2CCC[C@H]2C(=O)NCc2ccco2)c1 ZINC000880554258 ED On-Demand Anodyne ELANE 40 35 COc1cncc(NC(=O)N2CCC[C@@H]2C(=O)NCc2ccco2)c1 ZINC000880554259 ED On-Demand Anodyne F2 38 44 COc1cncc(NC(=O)N2CCC[C@@H]2C(=O)NCc2ccco2)c1 ZINC000880554259 ED On-Demand Anodyne ELANE 40 35 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3F)CC2)c1 ZINC000880554260 GE On-Demand Anodyne PDGFRB 40 36 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3F)CC2)c1 ZINC000880554260 GE On-Demand Anodyne FAAH 22 45 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3F)CC2)c1 ZINC000880554260 GE On-Demand Anodyne DGAT1 15 45 COc1cncc(NC(=O)NCCc2ccncc2C)c1 ZINC000880554269 CE On-Demand Anodyne RAF1 18 41 COc1cncc(NC(=O)NCCc2ccncc2C)c1 ZINC000880554269 CE On-Demand Anodyne MTNR1A 42 39 COc1cncc(NC(=O)NCCc2ccncc2C)c1 ZINC000880554269 CE On-Demand Anodyne ROCK2 15 44 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne HTR1A 18 40 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne DRD2 16 40 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne HRH2 25 41 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne PDGFRB 51 38 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne SIGMAR1 19 42 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne CCR3 55 44 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne MLNR 43 36 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne FAAH 41 57 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne MCHR1 29 42 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)CC2)c1 ZINC000880554272 EF On-Demand Anodyne CACNA1G 39 43 COc1cncc(NC(=O)N2CCN(C[C@H](O)COc3ccccc3)CC2)c1 ZINC000880554283 GD On-Demand Anodyne ADRB1 41 39 COc1cncc(NC(=O)N2CCN(C[C@H](O)COc3ccccc3)CC2)c1 ZINC000880554283 GD On-Demand Anodyne PDGFRB 56 42 COc1cncc(NC(=O)N2CCN(C[C@H](O)COc3ccccc3)CC2)c1 ZINC000880554283 GD On-Demand Anodyne ACOX1 85 44 COc1cncc(NC(=O)N2CCN(C[C@H](O)COc3ccccc3)CC2)c1 ZINC000880554283 GD On-Demand Anodyne FAAH 24 48 COc1cncc(NC(=O)N2CCN(C[C@H](O)COc3ccccc3)CC2)c1 ZINC000880554283 GD On-Demand Anodyne ABCB1 85 53 COc1cncc(NC(=O)N2CCN(C[C@@H](O)COc3ccccc3)CC2)c1 ZINC000880554284 GD On-Demand Anodyne ADRB1 41 39 COc1cncc(NC(=O)N2CCN(C[C@@H](O)COc3ccccc3)CC2)c1 ZINC000880554284 GD On-Demand Anodyne PDGFRB 56 42 COc1cncc(NC(=O)N2CCN(C[C@@H](O)COc3ccccc3)CC2)c1 ZINC000880554284 GD On-Demand Anodyne ACOX1 85 44 COc1cncc(NC(=O)N2CCN(C[C@@H](O)COc3ccccc3)CC2)c1 ZINC000880554284 GD On-Demand Anodyne FAAH 24 48 COc1cncc(NC(=O)N2CCN(C[C@@H](O)COc3ccccc3)CC2)c1 ZINC000880554284 GD On-Demand Anodyne ABCB1 85 53 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)Nc1ccccc1 ZINC000880554293 EG On-Demand Anodyne AVPR2 47 35 COc1cncc(NC(=O)N2CCOC3(CCC3)C2)c1 ZINC000880554298 CD On-Demand Anodyne EPHX2 26 46 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)Nc1cccnc1 ZINC000880554306 EF On-Demand Anodyne CHRNA7 25 41 COc1cncc(NC(=O)N2CC[C@@](O)(Cc3cccc(Cl)c3)C2)c1 ZINC000880554308 FF On-Demand Anodyne FAAH 20 47 COc1cncc(NC(=O)N2CC[C@@](O)(Cc3cccc(Cl)c3)C2)c1 ZINC000880554308 FF On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CC[C@](O)(Cc3cccc(Cl)c3)C2)c1 ZINC000880554310 FF On-Demand Anodyne FAAH 20 47 COc1cncc(NC(=O)N2CC[C@](O)(Cc3cccc(Cl)c3)C2)c1 ZINC000880554310 FF On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccccc2)c1 ZINC000880554311 EG On-Demand Anodyne Q8WSF8_APLCA 17 41 COc1cncc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880554313 EG On-Demand Anodyne Q8WSF8_APLCA 17 41 COc1cncc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880554315 EG On-Demand Anodyne Q8WSF8_APLCA 17 41 COc1cncc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccccc2)c1 ZINC000880554317 EG On-Demand Anodyne Q8WSF8_APLCA 17 41 C#CCN(CC)C(=O)Nc1cncc(OC)c1 ZINC000880554330 BD On-Demand Mild ROCK2 17 42 N#Cc1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880554341 DH On-Demand Mild SIGMAR1 17 40 COc1cncc(NC(=O)NCc2ccnc(OCCN(C)C)c2)c1 ZINC000880554343 ED On-Demand Anodyne ROCK2 32 45 CCOC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)C(C)C ZINC000880554345 DD On-Demand Anodyne HLA-DRB1 60 40 CCOC(=O)N[C@H](C(=O)NCc1cn(C2CCC2)nn1)C(C)C ZINC000880554347 DD On-Demand Anodyne HLA-DRB1 60 40 COc1cncc(NC(=O)N2CC[C@H]2Cc2ccccc2)c1 ZINC000880554351 CF On-Demand Anodyne CCR3 35 46 COc1cncc(NC(=O)N2CC[C@H]2Cc2ccccc2)c1 ZINC000880554351 CF On-Demand Anodyne CHRNA7 43 47 COc1cncc(NC(=O)N2CC[C@@H]2Cc2ccccc2)c1 ZINC000880554353 CF On-Demand Anodyne CCR3 35 46 COc1cncc(NC(=O)N2CC[C@@H]2Cc2ccccc2)c1 ZINC000880554353 CF On-Demand Anodyne CHRNA7 43 47 CCOC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554357 CE On-Demand Anodyne ACE 15 40 CCOC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554357 CE On-Demand Anodyne TPP2 51 37 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880554365 ED On-Demand Anodyne PDGFRB 41 38 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554367 DD On-Demand Anodyne CAPNS1 53 33 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554367 DD On-Demand Anodyne HLA-DRB1 43 32 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554367 DD On-Demand Anodyne CAPN1 79 41 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554367 DD On-Demand Anodyne CAPN2 114 36 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554367 DD On-Demand Anodyne FPR1 58 36 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554369 DD On-Demand Anodyne CAPNS1 53 33 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554369 DD On-Demand Anodyne HLA-DRB1 43 32 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554369 DD On-Demand Anodyne CAPN1 79 41 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554369 DD On-Demand Anodyne CAPN2 114 36 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554369 DD On-Demand Anodyne FPR1 58 36 COc1cncc(NC(=O)N2CCCN(C(=O)Cc3cccc(F)c3)CC2)c1 ZINC000880554378 GF On-Demand Anodyne CCR3 23 43 COc1cncc(NC(=O)N2CCCN(C(=O)Cc3cccc(F)c3)CC2)c1 ZINC000880554378 GF On-Demand Anodyne MLNR 19 40 COc1cncc(NC(=O)N2CCCN(C(=O)Cc3cccc(F)c3)CC2)c1 ZINC000880554378 GF On-Demand Anodyne FAAH 20 42 COc1cncc(NC(=O)N2CCCN(C(=O)Cc3cccc(F)c3)CC2)c1 ZINC000880554378 GF On-Demand Anodyne S1PR2 26 40 O=C(NCc1cn(C2CCC2)nn1)c1ccc2n[nH]cc2c1 ZINC000880554383 CD On-Demand Anodyne CA14 15 42 COc1cncc(NC(=O)N2CC[C@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554402 EF On-Demand Anodyne LTA4H 17 40 COc1cncc(NC(=O)N2CC[C@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554402 EF On-Demand Anodyne CCR3 18 46 COc1cncc(NC(=O)N2CC[C@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554402 EF On-Demand Anodyne MCHR1 18 47 COc1cncc(NC(=O)N2CC[C@@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554404 EF On-Demand Anodyne LTA4H 17 40 COc1cncc(NC(=O)N2CC[C@@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554404 EF On-Demand Anodyne CCR3 18 46 COc1cncc(NC(=O)N2CC[C@@H](N(C)Cc3ccccc3)C2)c1 ZINC000880554404 EF On-Demand Anodyne MCHR1 18 47 COc1cncc(NC(=O)NCc2ccccc2CN2CCC(O)CC2)c1 ZINC000880554406 FE On-Demand Anodyne SIGMAR1 20 41 COc1cncc(NC(=O)NCc2ccccc2CN2CCC(O)CC2)c1 ZINC000880554406 FE On-Demand Anodyne CCR3 52 49 COc1cncc(NC(=O)NCc2ccccc2CN2CCC(O)CC2)c1 ZINC000880554406 FE On-Demand Anodyne MCHR1 37 43 CCc1nc2ccccc2n1C1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880554415 GH On-Demand Anodyne CALCRL 24 41 CCc1nc2ccccc2n1C1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880554415 GH On-Demand Anodyne FPR2 31 58 CCc1nc2ccccc2n1C1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880554415 GH On-Demand Anodyne SMO 28 45 O=C(O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554419 CD On-Demand Anodyne HTR1A 19 42 O=C(O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554419 CD On-Demand Anodyne SLC6A1 78 36 O=C(O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554419 CD On-Demand Anodyne HTR7 28 45 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne HTR1A 45 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne DRD2 35 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne DRD4 33 42 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne ADRA1A 18 43 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne DRD3 40 39 COc1ccccc1NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554421 FG On-Demand Anodyne KCNQ2 40 34 CS(=O)(=O)NCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554422 DD On-Demand Anodyne HTR7 18 41 CNc1nc(CNC(=O)Nc2cncc(OC)c2)cs1 ZINC000880554431 CD On-Demand Anodyne ROCK2 18 42 CCc1nc([C@H]2CCCN2C(=O)Nc2cncc(OC)c2)no1 ZINC000880554437 DE On-Demand Anodyne CPT1A 44 39 COc1cncc(NC(=O)NCC(=O)N2CCOCC2)c1 ZINC000880554443 CC On-Demand Anodyne EPHX2 15 44 COc1cncc(NC(=O)NCC(=O)N2CCOCC2)c1 ZINC000880554443 CC On-Demand Anodyne PIK3CG 23 42 N#CCc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880554451 GF On-Demand Mild ABCB1 46 38 N#CCc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880554452 GF On-Demand Mild ABCB1 46 38 COc1cncc(NC(=O)N2CCC[C@H]2C(=O)OC(C)(C)C)c1 ZINC000880554453 DE On-Demand Anodyne FKBP1A 49 39 NC(=O)c1ccc(CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880554459 EF On-Demand Anodyne OPRM1 16 44 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne P2RY12 16 41 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne PDGFRB 53 42 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne GRIN2B 43 41 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne CCR3 36 51 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne CHRNA7 28 46 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne FAAH 19 44 COc1cncc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c1 ZINC000880554479 EG On-Demand Anodyne DGAT1 21 42 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne P2RY12 16 41 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne PDGFRB 53 42 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne GRIN2B 43 41 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne CCR3 36 51 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne CHRNA7 28 46 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne FAAH 19 44 COc1cncc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c1 ZINC000880554480 EG On-Demand Anodyne DGAT1 21 42 COc1cncc(NC(=O)Nc2cc(C)n(C)n2)c1 ZINC000880554497 CD On-Demand Anodyne HTR2A 21 41 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccncc3)C2)c1 ZINC000880554499 DF On-Demand Anodyne GRIN2B 44 38 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccncc3)C2)c1 ZINC000880554499 DF On-Demand Anodyne CCR3 93 52 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccncc3)C2)c1 ZINC000880554499 DF On-Demand Anodyne CHRNA7 20 41 COc1cncc(NC(=O)N2CC[C@H](Cc3ccncc3)C2)c1 ZINC000880554500 DF On-Demand Anodyne GRIN2B 44 38 COc1cncc(NC(=O)N2CC[C@H](Cc3ccncc3)C2)c1 ZINC000880554500 DF On-Demand Anodyne CCR3 93 52 COc1cncc(NC(=O)N2CC[C@H](Cc3ccncc3)C2)c1 ZINC000880554500 DF On-Demand Anodyne CHRNA7 20 41 CCOC(=O)c1csc(CN2Cc3ccccc3N3CCC[C@H]3C2)n1 ZINC000880554507 FG On-Demand Anodyne TPP2 40 32 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](CO)C2CC2)c1 ZINC000880554508 EF On-Demand Anodyne ROCK2 20 41 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](CO)C2CC2)c1 ZINC000880554509 EF On-Demand Anodyne ROCK2 20 41 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)Nc1c(F)cccc1F ZINC000880554513 FG On-Demand Anodyne DRD4 17 42 COc1cncc(NC(=O)N(C)Cc2nccs2)c1 ZINC000880554527 CE On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)NC2CCN(CCOC(C)C)CC2)c1 ZINC000880554540 EE On-Demand Anodyne SSTR5 40 35 COc1cncc(NC(=O)NC2CCN(CCOC(C)C)CC2)c1 ZINC000880554540 EE On-Demand Anodyne EPHX2 40 44 COc1cncc(NC(=O)NC2CCN(CCOC(C)C)CC2)c1 ZINC000880554540 EE On-Demand Anodyne CXCR3 20 45 COc1cncc(NC(=O)NC2CCN(CCOC(C)C)CC2)c1 ZINC000880554540 EE On-Demand Anodyne MCHR1 22 47 CCOC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554546 CE On-Demand Anodyne SLC6A1 43 32 CCOC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554546 CE On-Demand Anodyne CHRM4 17 42 O=C1CCCN1CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554547 DE On-Demand Anodyne HTR1A 19 44 O=C1CCCN1CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554547 DE On-Demand Anodyne HTR7 19 43 COc1cncc(NC(=O)N[C@H](C[S@](C)=O)c2ccccc2)c1 ZINC000880554548 EE On-Demand Anodyne SOAT1 21 41 COc1cncc(NC(=O)N[C@H](C[S@@](C)=O)c2ccccc2)c1 ZINC000880554549 EE On-Demand Anodyne SOAT1 21 41 COc1cncc(NC(=O)N[C@@H](C[S@@](C)=O)c2ccccc2)c1 ZINC000880554550 EE On-Demand Anodyne SOAT1 21 41 COc1cncc(NC(=O)N[C@@H](C[S@](C)=O)c2ccccc2)c1 ZINC000880554551 EE On-Demand Anodyne SOAT1 21 41 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554553 DG On-Demand Anodyne HTR1A 28 42 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554553 DG On-Demand Anodyne CHRM1 17 41 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554553 DG On-Demand Anodyne DRD2 15 40 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554553 DG On-Demand Anodyne CHRM4 17 41 CCOC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554553 DG On-Demand Anodyne HTR7 44 41 N#CCNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554559 CD On-Demand Mild CTSK 20 42 COc1cncc(NC(=O)N(C)CC(C)(C)O)c1 ZINC000880554569 CD On-Demand Anodyne ROCK2 19 42 COc1cncc(NC(=O)N2CCN(c3nccn(C)c3=O)CC2)c1 ZINC000880554587 EC On-Demand Anodyne PDGFRB 58 42 COc1cncc(NC(=O)NCC[C@H](O)c2ccccc2)c1 ZINC000880554605 DE On-Demand Anodyne ADRB1 42 32 COc1cncc(NC(=O)NCC[C@H](O)c2ccccc2)c1 ZINC000880554605 DE On-Demand Anodyne MTNR1A 19 40 COc1cncc(NC(=O)NCC[C@H](O)c2ccccc2)c1 ZINC000880554605 DE On-Demand Anodyne MTNR1B 20 40 COc1cncc(NC(=O)NCC[C@@H](O)c2ccccc2)c1 ZINC000880554606 DE On-Demand Anodyne ADRB1 42 32 COc1cncc(NC(=O)NCC[C@@H](O)c2ccccc2)c1 ZINC000880554606 DE On-Demand Anodyne MTNR1A 19 40 COc1cncc(NC(=O)NCC[C@@H](O)c2ccccc2)c1 ZINC000880554606 DE On-Demand Anodyne MTNR1B 20 40 CC[C@@H]1CCCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880554608 CF On-Demand Anodyne CCR3 19 50 CC[C@H]1CCCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880554609 CF On-Demand Anodyne CCR3 19 50 COCCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554698 CG On-Demand Anodyne HTR1A 33 45 COCCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554698 CG On-Demand Anodyne DRD2 18 41 COCCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554698 CG On-Demand Anodyne DRD3 18 41 COc1cncc(NC(=O)N2CC[C@H](CSc3ccccc3)C2)c1 ZINC000880554699 EH On-Demand Anodyne CCR3 19 47 COc1cncc(NC(=O)N2CC[C@@H](CSc3ccccc3)C2)c1 ZINC000880554700 EH On-Demand Anodyne CCR3 19 47 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccc(C)cc3)CC2)c1 ZINC000880554709 GF On-Demand Anodyne EPHX2 34 43 COc1cncc(NC(=O)N(C)CCN(C)C)c1 ZINC000880554710 CD On-Demand Anodyne ROCK2 17 41 COc1cncc(NC(=O)NCCN(C)Cc2ccc(F)cc2)c1 ZINC000880554722 EE On-Demand Anodyne CCR3 43 50 COc1cncc(NC(=O)NCCN(C)Cc2ccc(F)cc2)c1 ZINC000880554722 EE On-Demand Anodyne ROCK2 30 44 COc1cncc(NC(=O)N(CCN(C)C)CC(C)C)c1 ZINC000880554723 CE On-Demand Anodyne ROCK2 16 43 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne HTR1A 30 46 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne DRD2 17 41 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne SLC6A1 101 42 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne CYSLTR2 42 31 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne HTR7 47 48 O=C(O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554725 CE On-Demand Anodyne CYP2J2 47 33 COc1cncc(NC(=O)NCCOCc2ccccc2)c1 ZINC000880554729 DE On-Demand Anodyne HRH2 16 41 COc1cncc(NC(=O)NCCOCc2ccccc2)c1 ZINC000880554729 DE On-Demand Anodyne NAMPT 18 40 COc1ccc(O[C@H](C)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880554730 EF On-Demand Anodyne MTNR1A 23 48 COc1ccc(O[C@H](C)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880554730 EF On-Demand Anodyne MTNR1B 21 48 COc1ccc(O[C@@H](C)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880554731 EF On-Demand Anodyne MTNR1A 23 48 COc1ccc(O[C@@H](C)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880554731 EF On-Demand Anodyne MTNR1B 21 48 CCN(C)C(=O)Nc1cncc(OC)c1 ZINC000880554745 BD On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N(CCO)CCCO)c1 ZINC000880554770 CC On-Demand Anodyne ROCK2 15 43 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccccc1 ZINC000880554772 GE On-Demand Anodyne XIAP 57 38 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccccc1 ZINC000880554772 GE On-Demand Anodyne BIRC3 46 34 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccccc1 ZINC000880554772 GE On-Demand Anodyne BIRC2 88 37 CNC(=O)[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccccc1 ZINC000880554772 GE On-Demand Anodyne BIRC8 57 34 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1cccnc1 ZINC000880554777 EE On-Demand Anodyne CHRNA7 42 35 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1cccnc1 ZINC000880554777 EE On-Demand Anodyne PDE11A 43 38 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1cccnc1 ZINC000880554777 EE On-Demand Anodyne NAMPT 61 41 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554787 DF On-Demand Anodyne HTR1A 27 44 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554787 DF On-Demand Anodyne DRD2 19 40 CCCCNC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554787 DF On-Demand Anodyne DRD3 22 45 COc1cncc(NC(=O)NCCC2CC2)c1 ZINC000880554789 BE On-Demand Anodyne CCR3 28 42 COc1cncc(NC(=O)N[C@H](C)COCc2ccccc2)c1 ZINC000880554794 DF On-Demand Anodyne GHSR 18 40 COc1cncc(NC(=O)N[C@H](C)COCc2ccccc2)c1 ZINC000880554794 DF On-Demand Anodyne CAPN2 46 33 COc1cncc(NC(=O)N[C@@H](C)COCc2ccccc2)c1 ZINC000880554795 DF On-Demand Anodyne GHSR 18 40 COc1cncc(NC(=O)N[C@@H](C)COCc2ccccc2)c1 ZINC000880554795 DF On-Demand Anodyne CAPN2 46 33 COc1cncc(NC(=O)N2CCc3cnc(C(C)C)nc3C2)c1 ZINC000880554802 EF On-Demand Anodyne MAPK1 55 41 COc1cncc(NC(=O)N(C)C2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880554803 FF On-Demand Anodyne GPR119 45 43 COc1cncc(NC(=O)N2CC[C@H](CN3CCCC3)C2)c1 ZINC000880554804 DE On-Demand Anodyne CCR3 25 56 COc1cncc(NC(=O)N2CC[C@@H](CN3CCCC3)C2)c1 ZINC000880554805 DE On-Demand Anodyne CCR3 25 56 COc1cncc(NC(=O)N[C@H]2CCCC[C@H]2CO)c1 ZINC000880554821 CD On-Demand Anodyne CCR3 27 43 COc1cncc(NC(=O)N[C@@H]2CCCC[C@H]2CO)c1 ZINC000880554822 CD On-Demand Anodyne CCR3 27 43 COc1cncc(NC(=O)N[C@H]2CCCC[C@@H]2CO)c1 ZINC000880554823 CD On-Demand Anodyne CCR3 27 43 COc1cncc(NC(=O)N[C@@H]2CCCC[C@@H]2CO)c1 ZINC000880554824 CD On-Demand Anodyne CCR3 27 43 COc1cncc(NC(=O)N(C)Cc2ccc([S@@](C)=O)cc2)c1 ZINC000880554829 EE On-Demand Anodyne ROCK2 18 44 COc1cncc(NC(=O)N(C)Cc2ccc([S@](C)=O)cc2)c1 ZINC000880554830 EE On-Demand Anodyne ROCK2 18 44 COc1cncc(NC(=O)N2CCC3(CCOCC3)C2)c1 ZINC000880554834 CE On-Demand Anodyne EPHX2 35 46 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554835 GF On-Demand Anodyne ADRB2 15 43 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554835 GF On-Demand Anodyne HTR1A 30 40 COc1cccc(OC)c1OC[C@@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554835 GF On-Demand Anodyne ABCB1 68 41 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554836 GF On-Demand Anodyne ADRB2 15 43 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554836 GF On-Demand Anodyne HTR1A 30 40 COc1cccc(OC)c1OC[C@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554836 GF On-Demand Anodyne ABCB1 68 41 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCC(=O)N1CCCC1 ZINC000880554842 FD On-Demand Anodyne PREP 48 40 C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554847 DD On-Demand Anodyne PGC 45 34 C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554847 DD On-Demand Anodyne REN 57 37 C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554847 DD On-Demand Anodyne FPR1 50 38 COc1cncc(NC(=O)N2CC[C@H](Cc3cnn(C)c3)C2)c1 ZINC000880554857 DD On-Demand Anodyne CCR3 42 49 COc1cncc(NC(=O)N2CC[C@@H](Cc3cnn(C)c3)C2)c1 ZINC000880554858 DD On-Demand Anodyne CCR3 42 49 COc1cncc(NC(=O)N(C)CC[C@@H]2CCCCN2C)c1 ZINC000880554873 DE On-Demand Anodyne ACKR3 73 36 COc1cncc(NC(=O)N(C)CC[C@H]2CCCCN2C)c1 ZINC000880554874 DE On-Demand Anodyne ACKR3 73 36 N#CCCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554875 CG On-Demand Mild HTR7 16 41 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554884 DD On-Demand Anodyne HTR1A 22 42 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554884 DD On-Demand Anodyne SLC6A1 63 36 NC(=O)NC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880554884 DD On-Demand Anodyne HTR7 45 42 CN(C)C(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554887 EG On-Demand Anodyne DRD2 15 45 CN(C)C(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554887 EG On-Demand Anodyne ACHE 15 41 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880554889 DF On-Demand Anodyne CCR3 47 33 COc1cncc(NC(=O)NCC2(N3CCCCC3)CCN(C)CC2)c1 ZINC000880554918 FE On-Demand Anodyne HCN1 71 47 COc1cncc(NC(=O)NCC2(N3CCCCC3)CCN(C)CC2)c1 ZINC000880554918 FE On-Demand Anodyne HCN4 55 39 COc1cncc(NC(=O)NC2CCN(C3CCCC3)CC2)c1 ZINC000880554919 DF On-Demand Anodyne HRH3 15 40 COc1cncc(NC(=O)NC2CCN(C3CCCC3)CC2)c1 ZINC000880554919 DF On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)NC2CCN(C3CCCC3)CC2)c1 ZINC000880554919 DF On-Demand Anodyne EPHX2 49 40 COc1cncc(NC(=O)NC2CCN(C3CCCC3)CC2)c1 ZINC000880554919 DF On-Demand Anodyne CXCR3 17 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3cc(OC)cc(OC)c3)C2)c1 ZINC000880554931 FF On-Demand Anodyne EPHX2 42 37 COc1cncc(NC(=O)N[C@H]2CCN(c3cc(OC)cc(OC)c3)C2)c1 ZINC000880554932 FF On-Demand Anodyne EPHX2 42 37 COc1cncc(NC(=O)N2CCN(c3nc(C)ns3)CC2)c1 ZINC000880554933 ED On-Demand Anodyne PDGFRB 46 37 COc1cncc(NC(=O)N2CCN(c3nc(C)ns3)CC2)c1 ZINC000880554933 ED On-Demand Anodyne FAAH 15 56 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccc(F)cc2)c1 ZINC000880554942 EG On-Demand Anodyne CCR3 136 42 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccc(F)cc2)c1 ZINC000880554942 EG On-Demand Anodyne CHRNA7 22 45 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccc(F)cc2)c1 ZINC000880554943 EG On-Demand Anodyne CCR3 136 42 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccc(F)cc2)c1 ZINC000880554943 EG On-Demand Anodyne CHRNA7 22 45 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554944 FF On-Demand Anodyne DRD4 43 34 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554944 FF On-Demand Anodyne CCR3 39 51 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554944 FF On-Demand Anodyne PREP 24 40 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554944 FF On-Demand Anodyne CACNA1I 66 35 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554945 FF On-Demand Anodyne DRD4 43 34 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554945 FF On-Demand Anodyne CCR3 39 51 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554945 FF On-Demand Anodyne PREP 24 40 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)c3ccccc3)C2)c1 ZINC000880554945 FF On-Demand Anodyne CACNA1I 66 35 COc1cncc(NC(=O)NCc2csc(N(C)C)n2)c1 ZINC000880554950 DD On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)NC2CCN(C3CCCCC3)CC2)c1 ZINC000880554955 EG On-Demand Anodyne CCR3 17 42 COc1cncc(NC(=O)NC2CCN(C3CCCCC3)CC2)c1 ZINC000880554955 EG On-Demand Anodyne EPHX2 49 41 COc1cncc(NC(=O)NC2CCN(C3CCCCC3)CC2)c1 ZINC000880554955 EG On-Demand Anodyne CXCR3 18 40 COc1cncc(NC(=O)N[C@@H]2C[C@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554956 EE On-Demand Anodyne CCKAR 38 41 COc1cncc(NC(=O)N[C@@H]2C[C@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554956 EE On-Demand Anodyne CCKBR 49 41 COc1cncc(NC(=O)N[C@H]2C[C@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554957 EE On-Demand Anodyne CCKAR 38 41 COc1cncc(NC(=O)N[C@H]2C[C@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554957 EE On-Demand Anodyne CCKBR 49 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554958 EE On-Demand Anodyne CCKAR 38 41 COc1cncc(NC(=O)N[C@@H]2C[C@@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554958 EE On-Demand Anodyne CCKBR 49 41 COc1cncc(NC(=O)N[C@H]2C[C@@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554959 EE On-Demand Anodyne CCKAR 38 41 COc1cncc(NC(=O)N[C@H]2C[C@@H](C)N(c3ccccc3)C2=O)c1 ZINC000880554959 EE On-Demand Anodyne CCKBR 49 41 CCN(CC(C)(C)O)C(=O)Nc1cncc(OC)c1 ZINC000880554976 CD On-Demand Anodyne ROCK2 17 42 COc1cncc(NC(=O)N2CCC[C@@H](c3noc(C4CC4)n3)C2)c1 ZINC000880554977 EF On-Demand Anodyne SMO 23 45 COc1cncc(NC(=O)N2CCC[C@H](c3noc(C4CC4)n3)C2)c1 ZINC000880554978 EF On-Demand Anodyne SMO 23 45 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne HTR1A 20 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne DRD2 19 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne HTR1D 23 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne HTR1B 19 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne NPY1R 30 41 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne CCR3 54 40 CC(=O)Nc1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880554986 EH On-Demand Anodyne MCHR1 32 41 COc1cncc(NC(=O)NCCC2CCN(CC(F)(F)F)CC2)c1 ZINC000880555025 FF On-Demand Anodyne CCR3 54 46 COc1cncc(NC(=O)NCCC2CCN(CC(F)(F)F)CC2)c1 ZINC000880555025 FF On-Demand Anodyne HPGDS 34 43 COc1cncc(NC(=O)N2CCC(OCC3CCCCC3)CC2)c1 ZINC000880555028 EH On-Demand Anodyne PDGFRB 42 36 COc1cncc(NC(=O)NCc2c(C)nn(C)c2C)c1 ZINC000880555035 CD On-Demand Anodyne P2RX7 15 46 COc1cncc(NC(=O)NC2CCC(C)(O)CC2)c1 ZINC000880555038 CD On-Demand Anodyne EPHX2 44 35 COc1cncc(NC(=O)N2CCN(Cc3ncc(-c4ccccc4)o3)CC2)c1 ZINC000880555040 GG On-Demand Anodyne PDGFRB 50 40 COc1cncc(NC(=O)N2CCN(Cc3ncc(-c4ccccc4)o3)CC2)c1 ZINC000880555040 GG On-Demand Anodyne FAAH 47 50 COc1cccc(OC)c1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555045 DD On-Demand Anodyne DRD2 37 40 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ncc[nH]2)c1 ZINC000880555075 DF On-Demand Anodyne CPT1A 41 36 COc1cncc(NC(=O)N2CCCC[C@H]2c2ncc[nH]2)c1 ZINC000880555076 DF On-Demand Anodyne CPT1A 41 36 COc1cncc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c1 ZINC000880555086 EG On-Demand Anodyne PDGFRB 35 42 COc1cncc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c1 ZINC000880555086 EG On-Demand Anodyne GRIN2B 56 45 COc1cncc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c1 ZINC000880555086 EG On-Demand Anodyne CCR3 34 51 COc1cncc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c1 ZINC000880555086 EG On-Demand Anodyne CHRNA7 18 41 COc1cncc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c1 ZINC000880555086 EG On-Demand Anodyne FAAH 15 42 COc1cncc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c1 ZINC000880555087 EG On-Demand Anodyne PDGFRB 35 42 COc1cncc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c1 ZINC000880555087 EG On-Demand Anodyne GRIN2B 56 45 COc1cncc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c1 ZINC000880555087 EG On-Demand Anodyne CCR3 34 51 COc1cncc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c1 ZINC000880555087 EG On-Demand Anodyne CHRNA7 18 41 COc1cncc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c1 ZINC000880555087 EG On-Demand Anodyne FAAH 15 42 CCC1(O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555092 CD On-Demand Anodyne PDGFRB 42 36 CCC1(O)CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555092 CD On-Demand Anodyne S1PR2 33 48 COc1cncc(NC(=O)N(C)CCc2cccs2)c1 ZINC000880555105 CF On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2OC)c1 ZINC000880555116 EF On-Demand Anodyne ADRB1 40 30 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2OC)c1 ZINC000880555116 EF On-Demand Anodyne MTNR1A 20 44 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2OC)c1 ZINC000880555116 EF On-Demand Anodyne MTNR1B 23 44 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2OC)c1 ZINC000880555117 EF On-Demand Anodyne ADRB1 40 30 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2OC)c1 ZINC000880555117 EF On-Demand Anodyne MTNR1A 20 44 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2OC)c1 ZINC000880555117 EF On-Demand Anodyne MTNR1B 23 44 COc1cncc(NC(=O)NCCN2CCC(N(C)C)CC2)c1 ZINC000880555139 DD On-Demand Anodyne DRD4 44 34 COc1cncc(NC(=O)NCCN2CCC(N(C)C)CC2)c1 ZINC000880555139 DD On-Demand Anodyne CCR3 51 47 COc1cncc(NC(=O)NCCN2CCC(N(C)C)CC2)c1 ZINC000880555139 DD On-Demand Anodyne MCHR1 16 44 COc1cncc(NC(=O)N2CCN(CCOC(C)C)CC2)c1 ZINC000880555149 DD On-Demand Anodyne PDGFRB 46 41 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne DRD2 17 44 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne DRD4 40 45 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne ACHE 50 46 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne LTA4H 27 42 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne SIGMAR1 46 45 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne BCHE 18 40 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne CCR3 71 44 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne SLC18A3 18 42 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne MLNR 42 34 COc1cncc(NC(=O)N(C)C[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555152 FG On-Demand Anodyne MCHR1 40 46 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne DRD2 17 44 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne DRD4 40 45 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne ACHE 50 46 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne LTA4H 27 42 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne SIGMAR1 46 45 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne BCHE 18 40 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne CCR3 71 44 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne SLC18A3 18 42 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne MLNR 42 34 COc1cncc(NC(=O)N(C)C[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880555153 FG On-Demand Anodyne MCHR1 40 46 COc1cncc(NC(=O)N(Cc2ccccc2)C2CCN(C)CC2)c1 ZINC000880555155 FG On-Demand Anodyne ROCK2 27 49 CC[C@@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555165 DD On-Demand Anodyne PDGFRB 41 35 CC[C@@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555165 DD On-Demand Anodyne S1PR2 27 40 CC[C@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555166 DD On-Demand Anodyne PDGFRB 41 35 CC[C@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880555166 DD On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCN(c3cnn(C)c3)CC2)c1 ZINC000880555168 DD On-Demand Anodyne PDGFRB 52 39 COc1cncc(NC(=O)N(C)[C@H](C)Cc2ccccc2OC)c1 ZINC000880555176 EG On-Demand Anodyne NPY5R 37 51 COc1cncc(NC(=O)N(C)[C@@H](C)Cc2ccccc2OC)c1 ZINC000880555177 EG On-Demand Anodyne NPY5R 37 51 COc1cncc(NC(=O)N[C@@H](CO)c2ccccc2C)c1 ZINC000880555182 DE On-Demand Anodyne CTSA 55 36 COc1cncc(NC(=O)N[C@H](CO)c2ccccc2C)c1 ZINC000880555183 DE On-Demand Anodyne CTSA 55 36 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](CO)C(C)C)c1 ZINC000880555190 EG On-Demand Anodyne ROCK2 22 46 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](CO)C(C)C)c1 ZINC000880555190 EG On-Demand Anodyne NPY5R 33 40 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](CO)C(C)C)c1 ZINC000880555191 EG On-Demand Anodyne ROCK2 22 46 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](CO)C(C)C)c1 ZINC000880555191 EG On-Demand Anodyne NPY5R 33 40 c1ccc2c(c1)CN(CC1CC1)C[C@@H]1CCCN21 ZINC000880555193 BF On-Demand Anodyne SIGMAR1 15 41 N#CCOc1ccccc1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555202 DD On-Demand Mild HCN1 64 39 N#CCOc1ccccc1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555202 DD On-Demand Mild HCN4 54 39 CC(C)(C)OC(=O)N1CCC(CC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880555203 GF On-Demand Anodyne GPR119 46 39 COc1cncc(NC(=O)N2CCC3(CCCC3)C2)c1 ZINC000880555205 CF On-Demand Anodyne EPHX2 35 46 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne PREP 42 51 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne CAPNS1 47 32 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne CAPN1 52 36 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne CAPN2 85 36 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne TPSAB1 15 46 O=C(CNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880555206 ED On-Demand Anodyne NPR 59 33 COc1cncc(NC(=O)N2CCN(Cc3nccn3C(F)F)CC2)c1 ZINC000880555209 FE On-Demand Anodyne PDGFRB 43 34 N#Cc1ccc(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880555215 EF On-Demand Mild MCHR1 21 40 COC(=O)/C(C)=C/CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555221 DF On-Demand Anodyne SLC6A1 61 33 COC(=O)/C(C)=C\CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555222 DF On-Demand Anodyne SLC6A1 61 33 COc1cncc(NC(=O)Nc2cnn(CC3CC3)c2)c1 ZINC000880555228 CE On-Demand Anodyne PANC 51 33 COc1cncc(NC(=O)NC2CCS(=O)(=O)CC2)c1 ZINC000880555236 CC On-Demand Anodyne EPHX2 42 36 N#Cc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880555242 EF On-Demand Mild CCR3 19 45 N#Cc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880555242 EF On-Demand Mild MCHR1 45 42 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne FKBP1A 46 40 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne SIGMAR1 16 40 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne CCKAR 33 43 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne CCR3 31 42 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne CHRNA7 21 44 COc1cncc(NC(=O)N[C@@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555246 FE On-Demand Anodyne CCKBR 49 43 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne FKBP1A 46 40 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne SIGMAR1 16 40 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne CCKAR 33 43 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne CCR3 31 42 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne CHRNA7 21 44 COc1cncc(NC(=O)N[C@H]2CCN(CCCc3ccccc3)C2=O)c1 ZINC000880555247 FE On-Demand Anodyne CCKBR 49 43 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555274 EE On-Demand Anodyne F2 49 40 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555274 EE On-Demand Anodyne PREP 16 46 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555274 EE On-Demand Anodyne LGMN 56 33 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555274 EE On-Demand Anodyne TMPRSS11D 61 40 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555275 EE On-Demand Anodyne F2 49 40 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555275 EE On-Demand Anodyne PREP 16 46 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555275 EE On-Demand Anodyne LGMN 56 33 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555275 EE On-Demand Anodyne TMPRSS11D 61 40 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne HTR1A 50 43 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne DRD2 35 42 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne DRD4 17 45 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne ADRA1A 15 43 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne DRD3 37 45 COC(=O)CCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555306 DF On-Demand Anodyne HTR7 65 41 COc1cncc(NC(=O)N2CCC3(CCN(C(=O)OC(C)(C)C)CC3)C2)c1 ZINC000880555308 GG On-Demand Anodyne EPHX2 33 45 COc1cncc(NC(=O)N2CCC3(CCN(C(=O)OC(C)(C)C)CC3)C2)c1 ZINC000880555308 GG On-Demand Anodyne GPR119 19 44 OCCOCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555311 CD On-Demand Anodyne SLC6A1 33 41 COc1cncc(NC(=O)N[C@@H]2CC(=O)N(C3CCCCC3)C2)c1 ZINC000880555312 EE On-Demand Anodyne INHA 18 41 COc1cncc(NC(=O)N[C@H]2CC(=O)N(C3CCCCC3)C2)c1 ZINC000880555313 EE On-Demand Anodyne INHA 18 41 COc1cncc(NC(=O)NCc2ccnc(N(C)C)n2)c1 ZINC000880555319 DD On-Demand Anodyne ROCK2 19 42 COc1cncc(NC(=O)N2CCC(F)(F)C2)c1 ZINC000880555326 CD On-Demand Anodyne EPHX2 32 40 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)/C=C\c2ccccc2)CC1 ZINC000880555340 GF On-Demand Anodyne PREP 19 41 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)/C=C/c2ccccc2)CC1 ZINC000880555341 GF On-Demand Anodyne PREP 19 41 COc1cncc(NC(=O)NCc2ccc(OC(C)(C)C)nc2)c1 ZINC000880555342 EF On-Demand Anodyne ROCK2 18 42 COc1cncc(NC(=O)N[C@H]2CCCOc3cc(F)ccc32)c1 ZINC000880555377 EG On-Demand Anodyne TRPV1 18 42 COc1cncc(NC(=O)N[C@@H]2CCCOc3cc(F)ccc32)c1 ZINC000880555378 EG On-Demand Anodyne TRPV1 18 42 COc1cncc(NC(=O)N2CC(Cc3ccccc3)C2)c1 ZINC000880555387 CF On-Demand Anodyne GRIN2B 43 38 COc1cncc(NC(=O)N2CC(Cc3ccccc3)C2)c1 ZINC000880555387 CF On-Demand Anodyne CCR3 41 56 COc1cncc(NC(=O)N2CC(Cc3ccccc3)C2)c1 ZINC000880555387 CF On-Demand Anodyne FAAH 16 43 COc1cncc(NC(=O)N2CCC(OCc3ccccc3OC)CC2)c1 ZINC000880555388 FG On-Demand Anodyne TSHR 53 31 COc1cncc(NC(=O)N2CCC(OCc3ccccc3OC)CC2)c1 ZINC000880555388 FG On-Demand Anodyne PDGFRB 44 38 COc1cncc(NC(=O)N2CCC(OCc3ccccc3OC)CC2)c1 ZINC000880555388 FG On-Demand Anodyne EPHX2 21 41 COc1cncc(NC(=O)N2CCC(OCc3ccccc3OC)CC2)c1 ZINC000880555388 FG On-Demand Anodyne SCD1 19 46 CC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555389 BE On-Demand Anodyne OPRL1 16 40 COc1cncc(NC(=O)N2CCC(C)(C)CC2)c1 ZINC000880555390 CF On-Demand Anodyne S1PR2 27 40 COC(=O)c1ccc2c(c1)CN(C(=O)Nc1cncc(OC)c1)CC2 ZINC000880555391 EE On-Demand Anodyne HDAC6 36 42 COC(=O)c1ccc2c(c1)CN(C(=O)Nc1cncc(OC)c1)CC2 ZINC000880555391 EE On-Demand Anodyne P2RY14 42 33 CCCCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555393 CG On-Demand Mild GBA 15 40 CCCCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555393 CG On-Demand Mild LASR 42 38 COc1cncc(NC(=O)NCCCc2c(C)nn(C)c2C)c1 ZINC000880555448 DE On-Demand Anodyne QPCT 20 41 C=CCNC(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880555457 CC On-Demand Mild F7 21 40 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccccc1F ZINC000880555462 DG On-Demand Anodyne SLC6A1 51 40 COc1cncc(NC(=O)N2CCc3c(cccc3OC)C2)c1 ZINC000880555468 DF On-Demand Anodyne DRD4 40 30 COc1cncc(NC(=O)N2CCc3c(cccc3OC)C2)c1 ZINC000880555468 DF On-Demand Anodyne PDGFRB 45 38 COc1cncc(NC(=O)N2CCc3c(cccc3OC)C2)c1 ZINC000880555468 DF On-Demand Anodyne SSTR1 52 37 COc1cncc(NC(=O)N2CCc3c(cccc3OC)C2)c1 ZINC000880555468 DF On-Demand Anodyne P2RY14 48 36 CCCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555486 CF On-Demand Mild GBA 15 40 CCCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555486 CF On-Demand Mild LASR 42 38 Cc1ccc(N2C[C@@H](C(=O)NCc3cn(C4CCC4)nn3)CC2=O)cc1F ZINC000880555521 FE On-Demand Anodyne P2RX7 15 40 CNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555528 CD On-Demand Anodyne OPRL1 21 52 CNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555528 CD On-Demand Anodyne BIRC2 80 35 COc1cncc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)c1 ZINC000880555539 EE On-Demand Anodyne CACNA1H 31 40 COc1cncc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)c1 ZINC000880555539 EE On-Demand Anodyne S1PR2 30 44 COc1cncc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)c1 ZINC000880555540 EE On-Demand Anodyne CACNA1H 31 40 COc1cncc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)c1 ZINC000880555540 EE On-Demand Anodyne S1PR2 30 44 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCC1 ZINC000880555556 DE On-Demand Anodyne SLC6A1 53 34 O=C(CCN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCC1 ZINC000880555556 DE On-Demand Anodyne PREP 53 38 O=C1c2ccccc2C(=O)N1OCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555557 GG On-Demand Anodyne HTR1A 18 40 COc1cncc(NC(=O)NCCCc2cccs2)c1 ZINC000880555568 CF On-Demand Anodyne BMP1 21 43 COc1cncc(NC(=O)NC2CCC(C(=O)OC(C)(C)C)CC2)c1 ZINC000880555572 EG On-Demand Anodyne EPHX2 40 38 COc1cncc(NC(=O)NCCc2ccc(CO)cc2)c1 ZINC000880555573 DD On-Demand Anodyne MTNR1A 38 40 COc1cncc(NC(=O)NCCc2ccc(CO)cc2)c1 ZINC000880555573 DD On-Demand Anodyne MTNR1B 31 40 COc1cncc(NC(=O)NCCc2ccc(CO)cc2)c1 ZINC000880555573 DD On-Demand Anodyne CA9 15 40 COc1cncc(NC(=O)N2CCc3cc(OC)c(F)cc3C2)c1 ZINC000880555576 EF On-Demand Anodyne ABCB1 18 42 COc1cncc(NC(=O)N2CCO[C@@H](Cc3ccccc3)C2)c1 ZINC000880555577 EF On-Demand Anodyne CCR3 22 54 COc1cncc(NC(=O)N2CCO[C@@H](Cc3ccccc3)C2)c1 ZINC000880555577 EF On-Demand Anodyne FAAH 15 42 COc1cncc(NC(=O)N2CCO[C@H](Cc3ccccc3)C2)c1 ZINC000880555578 EF On-Demand Anodyne CCR3 22 54 COc1cncc(NC(=O)N2CCO[C@H](Cc3ccccc3)C2)c1 ZINC000880555578 EF On-Demand Anodyne FAAH 15 42 COc1cncc(NC(=O)N2CCC[C@@H]2c2noc(C)n2)c1 ZINC000880555613 DE On-Demand Anodyne CPT1A 41 39 COc1cncc(NC(=O)N2CCC[C@H]2c2noc(C)n2)c1 ZINC000880555614 DE On-Demand Anodyne CPT1A 41 39 COc1cncc(NC(=O)NCCN2CCNC(=O)C2)c1 ZINC000880555615 CB On-Demand Anodyne DRD4 41 31 O=C(NCc1cn(C2CCC2)nn1)c1cc(Cl)nc(Cl)c1 ZINC000880555631 EF On-Demand Anodyne CA14 18 44 O=C(NCc1cn(C2CCC2)nn1)c1cc(Cl)nc(Cl)c1 ZINC000880555631 EF On-Demand Anodyne CACNA1I 40 31 CCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555634 CF On-Demand Anodyne GBA 15 40 CCCCCCC(=O)NCc1cn(C2CCC2)nn1 ZINC000880555634 CF On-Demand Anodyne LASR 42 38 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne PDGFRB 44 37 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne GRIN2B 65 45 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne CCR3 53 53 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne CHRNA7 66 51 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne C3AR1 42 46 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne FAAH 22 47 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne ACHP_LYMST 25 43 COc1cncc(NC(=O)N2CCC(Cc3cccnc3)CC2)c1 ZINC000880555645 EF On-Demand Anodyne NAMPT 43 38 COC[C@H](NC(=O)Nc1cncc(OC)c1)c1ccccc1 ZINC000880555646 DF On-Demand Anodyne SOAT1 21 40 COC[C@@H](NC(=O)Nc1cncc(OC)c1)c1ccccc1 ZINC000880555647 DF On-Demand Anodyne SOAT1 21 40 Oc1nc(CN2Cc3ccccc3N3CCC[C@H]3C2)nc2c1COCC2 ZINC000880555743 FE On-Demand Anodyne WNT3A 44 31 COc1cncc(NC(=O)N(Cc2ccccc2)CC(C)(C)O)c1 ZINC000880555784 EF On-Demand Anodyne LTA4H 15 40 COc1cncc(NC(=O)N(Cc2ccccc2)CC(C)(C)O)c1 ZINC000880555784 EF On-Demand Anodyne ROCK1 21 44 COc1cncc(NC(=O)N(Cc2ccccc2)CC(C)(C)O)c1 ZINC000880555784 EF On-Demand Anodyne ROCK2 36 46 COc1cncc(NC(=O)N(Cc2ccccc2)CC(C)(C)O)c1 ZINC000880555784 EF On-Demand Anodyne LIMK2 15 40 COc1cncc(NC(=O)NCc2ccc(C)nc2N2CCCC2)c1 ZINC000880555787 EF On-Demand Anodyne TRPV1 17 47 COC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555791 CD On-Demand Anodyne HTR1A 23 43 COC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555791 CD On-Demand Anodyne DRD2 15 40 COC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555791 CD On-Demand Anodyne OPRL1 17 45 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne HTR1A 30 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne DRD2 16 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne HTR2A 15 40 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne SLC6A1 87 37 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne OPRL1 19 44 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne HTR7 55 41 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne CYP2J2 44 31 CNC(=O)CCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555880 CD On-Demand Anodyne BIRC2 49 33 COc1cncc(NC(=O)N2CCCN(C)CC2)c1 ZINC000880555896 CD On-Demand Anodyne PDGFRB 44 37 CC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880555911 DH On-Demand Anodyne HTR1A 16 46 CC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880555911 DH On-Demand Anodyne DRD2 18 42 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555915 GE On-Demand Anodyne PAPA1_CARPA 34 49 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555915 GE On-Demand Anodyne REN 52 37 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555915 GE On-Demand Anodyne FPR1 58 45 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555916 GE On-Demand Anodyne PAPA1_CARPA 34 49 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555916 GE On-Demand Anodyne REN 52 37 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880555916 GE On-Demand Anodyne FPR1 58 45 COc1cncc(NC(=O)N[C@H]2CCCOc3c(F)cccc32)c1 ZINC000880555925 EG On-Demand Anodyne TRPV1 17 40 COc1cncc(NC(=O)N[C@@H]2CCCOc3c(F)cccc32)c1 ZINC000880555926 EG On-Demand Anodyne TRPV1 17 40 COc1cncc(NC(=O)N2CCN(c3ccc(F)cn3)CC2)c1 ZINC000880555947 ED On-Demand Anodyne PDGFRB 56 42 COc1cncc(NC(=O)N2CCN(c3ccc(F)cn3)CC2)c1 ZINC000880555947 ED On-Demand Anodyne FAAH 17 41 COc1cncc(NC(=O)N2CCN(c3ccc(F)cn3)CC2)c1 ZINC000880555947 ED On-Demand Anodyne DGAT1 37 49 COc1cncc(NC(=O)N2CCN(c3ccc(F)cn3)CC2)c1 ZINC000880555947 ED On-Demand Anodyne SLC27A1 40 38 CCOP(=O)(OCC)[C@@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555963 FG On-Demand Anodyne ADAM9 50 33 CCOP(=O)(OCC)[C@H](O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880555964 FG On-Demand Anodyne ADAM9 50 33 COc1cncc(NC(=O)NCC2CCN(c3ccncc3)CC2)c1 ZINC000880555967 EF On-Demand Anodyne F10 16 54 COc1cncc(NC(=O)NCC2CCN(c3ccncc3)CC2)c1 ZINC000880555967 EF On-Demand Anodyne CCR3 48 42 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CSCN1C(=O)c1ccccc1 ZINC000880555980 FD On-Demand Anodyne TMPRSS11D 58 35 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CSCN1C(=O)c1ccccc1 ZINC000880555981 FD On-Demand Anodyne TMPRSS11D 58 35 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](C)CCO)c1 ZINC000880555992 EF On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)N(Cc2ccccc2)[C@@H](C)CCO)c1 ZINC000880555992 EF On-Demand Anodyne NPY5R 34 41 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](C)CCO)c1 ZINC000880555993 EF On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)N(Cc2ccccc2)[C@H](C)CCO)c1 ZINC000880555993 EF On-Demand Anodyne NPY5R 34 41 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2Br)c1 ZINC000880556014 GE On-Demand Anodyne ADRB2 31 41 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2Br)c1 ZINC000880556014 GE On-Demand Anodyne ADRB1 71 47 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2Br)c1 ZINC000880556014 GE On-Demand Anodyne ADRB3 25 41 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2Br)c1 ZINC000880556015 GE On-Demand Anodyne ADRB2 31 41 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2Br)c1 ZINC000880556015 GE On-Demand Anodyne ADRB1 71 47 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2Br)c1 ZINC000880556015 GE On-Demand Anodyne ADRB3 25 41 COc1cncc(NC(=O)N2CCC[C@H]2c2cccc(C)n2)c1 ZINC000880556017 DG On-Demand Anodyne CPT1A 77 36 COc1cncc(NC(=O)N2CCC[C@@H]2c2cccc(C)n2)c1 ZINC000880556018 DG On-Demand Anodyne CPT1A 77 36 CC[C@H](O)CCNC(=O)Nc1cncc(OC)c1 ZINC000880556032 CD On-Demand Anodyne ADRB1 41 30 CC[C@@H](O)CCNC(=O)Nc1cncc(OC)c1 ZINC000880556033 CD On-Demand Anodyne ADRB1 41 30 COc1cncc(NC(=O)N2CCOC3(CCOCC3)C2)c1 ZINC000880556043 DD On-Demand Anodyne EPHX2 25 45 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCC(=O)c1cccs1 ZINC000880556045 FF On-Demand Anodyne NOS1 25 42 COc1cncc(NC(=O)N2CC[C@]3(CCOC3)C2)c1 ZINC000880556048 CD On-Demand Anodyne EPHX2 33 42 COc1cncc(NC(=O)N2CC[C@@]3(CCOC3)C2)c1 ZINC000880556049 CD On-Demand Anodyne EPHX2 33 42 COc1cncc(NC(=O)N2CCC[C@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556051 GG On-Demand Anodyne CCR3 22 41 COc1cncc(NC(=O)N2CCC[C@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556051 GG On-Demand Anodyne CHRNA7 15 43 COc1cncc(NC(=O)N2CCC[C@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556051 GG On-Demand Anodyne MCHR1 22 40 COc1cncc(NC(=O)N2CCC[C@@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556052 GG On-Demand Anodyne CCR3 22 41 COc1cncc(NC(=O)N2CCC[C@@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556052 GG On-Demand Anodyne CHRNA7 15 43 COc1cncc(NC(=O)N2CCC[C@@H](NC(=O)c3cc4ccccc4o3)C2)c1 ZINC000880556052 GG On-Demand Anodyne MCHR1 22 40 COc1cncc(NC(=O)N2CCc3ccccc3[C@@H]2CO)c1 ZINC000880556058 DE On-Demand Anodyne MTNR1B 26 41 COc1cncc(NC(=O)N2CCc3ccccc3[C@@H]2CO)c1 ZINC000880556058 DE On-Demand Anodyne TRPM8 38 44 COc1cncc(NC(=O)N2CCc3ccccc3[C@H]2CO)c1 ZINC000880556059 DE On-Demand Anodyne MTNR1B 26 41 COc1cncc(NC(=O)N2CCc3ccccc3[C@H]2CO)c1 ZINC000880556059 DE On-Demand Anodyne TRPM8 38 44 COc1cncc(NC(=O)NC[C@@H]2CCCN(CC(C)C)C2)c1 ZINC000880556060 DF On-Demand Anodyne CCR3 84 36 COc1cncc(NC(=O)NC[C@H]2CCCN(CC(C)C)C2)c1 ZINC000880556061 DF On-Demand Anodyne CCR3 84 36 COc1cncc(NC(=O)NCC2CCN(CC(=O)NC(C)(C)C)CC2)c1 ZINC000880556076 GD On-Demand Anodyne CCR3 32 41 COc1cncc(NC(=O)NCC2CCN(CC(=O)NC(C)(C)C)CC2)c1 ZINC000880556076 GD On-Demand Anodyne CACNA1I 76 52 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cncc(OC)c1 ZINC000880556081 CC On-Demand Anodyne UL80 40 39 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556084 FE On-Demand Anodyne NPY1R 30 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556084 FE On-Demand Anodyne CCKAR 41 48 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556084 FE On-Demand Anodyne CCKBR 61 46 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556085 FE On-Demand Anodyne NPY1R 30 42 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556085 FE On-Demand Anodyne CCKAR 41 48 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2=O)c1 ZINC000880556085 FE On-Demand Anodyne CCKBR 61 46 COc1cncc(NC(=O)N(CCN(C)C)Cc2cccs2)c1 ZINC000880556090 EF On-Demand Anodyne ROCK2 27 49 COc1cncc(NC(=O)NCCCc2ccc3c(c2)OCCO3)c1 ZINC000880556091 EF On-Demand Anodyne BMP1 50 37 COc1cncc(NC(=O)NCCCc2ccc3c(c2)OCCO3)c1 ZINC000880556091 EF On-Demand Anodyne QPCT 25 41 COc1cncc(NC(=O)NC2(c3ccc4c(c3)OCO4)CC2)c1 ZINC000880556093 EF On-Demand Anodyne EDNRA 41 39 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)Nc1cccnc1Cl ZINC000880556095 FG On-Demand Anodyne G2YM83_BOTF4 53 35 COCCNc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880556102 EE On-Demand Anodyne ROCK2 17 42 COc1ccc([C@H](CO)N(C)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880556108 EE On-Demand Anodyne NPY5R 32 40 COc1ccc([C@@H](CO)N(C)C(=O)Nc2cncc(OC)c2)cc1 ZINC000880556109 EE On-Demand Anodyne NPY5R 32 40 COc1cncc(NC(=O)N2CCN(CCO)CC2)c1 ZINC000880556111 CC On-Demand Anodyne DRD4 41 31 COc1cncc(NC(=O)N2CCN(CCO)CC2)c1 ZINC000880556111 CC On-Demand Anodyne PDGFRB 52 38 COc1cncc(NC(=O)N2CCN(CCO)CC2)c1 ZINC000880556111 CC On-Demand Anodyne FAAH 18 46 COc1cncc(NC(=O)NC2CCN([C@H]3CCCC[C@H]3O)CC2)c1 ZINC000880556113 ED On-Demand Anodyne EPHX2 49 38 COc1cncc(NC(=O)NC2CCN([C@H]3CCCC[C@H]3O)CC2)c1 ZINC000880556113 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@@H]3CCCC[C@H]3O)CC2)c1 ZINC000880556114 ED On-Demand Anodyne EPHX2 49 38 COc1cncc(NC(=O)NC2CCN([C@@H]3CCCC[C@H]3O)CC2)c1 ZINC000880556114 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@H]3CCCC[C@@H]3O)CC2)c1 ZINC000880556115 ED On-Demand Anodyne EPHX2 49 38 COc1cncc(NC(=O)NC2CCN([C@H]3CCCC[C@@H]3O)CC2)c1 ZINC000880556115 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@@H]3CCCC[C@@H]3O)CC2)c1 ZINC000880556116 ED On-Demand Anodyne EPHX2 49 38 COc1cncc(NC(=O)NC2CCN([C@@H]3CCCC[C@@H]3O)CC2)c1 ZINC000880556116 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)N(C)[C@H](C)CC#N)c1 ZINC000880556119 BD On-Demand Mild NPY5R 30 41 COc1cncc(NC(=O)N(C)[C@@H](C)CC#N)c1 ZINC000880556120 BD On-Demand Mild NPY5R 30 41 COc1cncc(NC(=O)NCc2ccccc2CS(C)(=O)=O)c1 ZINC000880556128 ED On-Demand Anodyne ROCK2 17 44 COc1cncc(NC(=O)NCc2ccccc2CS(C)(=O)=O)c1 ZINC000880556128 ED On-Demand Anodyne NAMPT 38 41 COc1cncc(NC(=O)NC2CCN([C@@H]3CCC[C@@H]3O)CC2)c1 ZINC000880556129 ED On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)NC2CCN([C@@H]3CCC[C@@H]3O)CC2)c1 ZINC000880556129 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@H]3CCC[C@@H]3O)CC2)c1 ZINC000880556130 ED On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)NC2CCN([C@H]3CCC[C@@H]3O)CC2)c1 ZINC000880556130 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@@H]3CCC[C@H]3O)CC2)c1 ZINC000880556131 ED On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)NC2CCN([C@@H]3CCC[C@H]3O)CC2)c1 ZINC000880556131 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NC2CCN([C@H]3CCC[C@H]3O)CC2)c1 ZINC000880556132 ED On-Demand Anodyne EPHX2 48 38 COc1cncc(NC(=O)NC2CCN([C@H]3CCC[C@H]3O)CC2)c1 ZINC000880556132 ED On-Demand Anodyne CXCR3 15 40 COc1cncc(NC(=O)NCCN2CCC(OC)CC2)c1 ZINC000880556133 DD On-Demand Anodyne DRD4 45 34 COc1cncc(NC(=O)NCCN2CCC(OC)CC2)c1 ZINC000880556133 DD On-Demand Anodyne CCR3 58 48 COc1cncc(NC(=O)N(C)CCOCc2ccccc2)c1 ZINC000880556139 DF On-Demand Anodyne ROCK2 26 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3ncccc3Cl)C2)c1 ZINC000880556157 EF On-Demand Anodyne TRPV1 15 44 COc1cncc(NC(=O)N[C@@H]2CCN(c3ncccc3Cl)C2)c1 ZINC000880556157 EF On-Demand Anodyne CHRNA7 16 41 COc1cncc(NC(=O)N[C@H]2CCN(c3ncccc3Cl)C2)c1 ZINC000880556158 EF On-Demand Anodyne TRPV1 15 44 COc1cncc(NC(=O)N[C@H]2CCN(c3ncccc3Cl)C2)c1 ZINC000880556158 EF On-Demand Anodyne CHRNA7 16 41 COc1cncc(NC(=O)N(CCO)CCN2CCOCC2)c1 ZINC000880556162 DC On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N(CCO)CCN2CCOCC2)c1 ZINC000880556162 DC On-Demand Anodyne CASR 66 58 COc1cncc(NC(=O)N[C@@H]2CC[C@H](CO)CC2)c1 ZINC000880556163 CD On-Demand Anodyne EPHX2 44 36 COc1cncc(NC(=O)N[C@@H]2CC[C@@H](CO)CC2)c1 ZINC000880556164 CD On-Demand Anodyne EPHX2 44 36 COc1cncc(NC(=O)NCc2ccc3c(c2)CCS3(=O)=O)c1 ZINC000880556165 ED On-Demand Anodyne ROCK2 21 43 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne DRD2 24 40 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne DRD4 40 33 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne PIK3CA 40 40 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne SCN2A 17 40 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne PIK3CD 22 41 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne SOAT1 17 40 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne MTOR 59 40 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne SCN10A 33 51 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne PIK3CB 30 41 COc1cncc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880556175 EE On-Demand Anodyne NAMPT 27 41 CCOc1ccnc(N2CCCN(C(=O)Nc3cncc(OC)c3)CC2)n1 ZINC000880556176 FE On-Demand Anodyne PDGFRB 50 38 COc1cncc(NC(=O)N[C@H](C)Cc2ccncc2)c1 ZINC000880556189 CE On-Demand Anodyne PDE4A 19 44 COc1cncc(NC(=O)N[C@H](C)Cc2ccncc2)c1 ZINC000880556189 CE On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)N[C@@H](C)Cc2ccncc2)c1 ZINC000880556190 CE On-Demand Anodyne PDE4A 19 44 COc1cncc(NC(=O)N[C@@H](C)Cc2ccncc2)c1 ZINC000880556190 CE On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)N2CCOC[C@H]2C[C@H](O)c2ccccc2)c1 ZINC000880556192 FE On-Demand Anodyne CASR 28 41 COc1cncc(NC(=O)N2CCOC[C@@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880556193 FE On-Demand Anodyne CASR 28 41 COc1cncc(NC(=O)N2CCOC[C@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880556194 FE On-Demand Anodyne CASR 28 41 COc1cncc(NC(=O)N2CCOC[C@@H]2C[C@H](O)c2ccccc2)c1 ZINC000880556195 FE On-Demand Anodyne CASR 28 41 CNC(=O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880556196 DB On-Demand Anodyne PDGFRB 45 36 COCC1(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556209 CD On-Demand Anodyne EPHX2 17 41 COc1cncc(NC(=O)N2C[C@@H](C)O[C@H](c3ccsc3)C2)c1 ZINC000880556217 EG On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2C[C@H](c3ccsc3)O[C@H](C)C2)c1 ZINC000880556218 EG On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2C[C@H](C)O[C@H](c3ccsc3)C2)c1 ZINC000880556219 EG On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2C[C@H](C)O[C@@H](c3ccsc3)C2)c1 ZINC000880556220 EG On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2CCN(c3cc(C)ccn3)CC2)c1 ZINC000880556226 EE On-Demand Anodyne PDGFRB 54 44 COc1cncc(NC(=O)N2CCN(c3cc(C)ccn3)CC2)c1 ZINC000880556226 EE On-Demand Anodyne FAAH 15 41 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne KLK3 44 33 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne PREP 41 50 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne GHSR 22 41 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne CAPN1 49 43 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne CAPN2 83 43 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne NPR 58 34 O=C(CCCNC(=O)OCc1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880556235 FE On-Demand Anodyne POLG_WNV 47 37 COc1cncc(NC(=O)N[C@@H]2CCCC[C@@H]2N2CCOCC2)c1 ZINC000880556240 ED On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)N[C@H]2CCCC[C@@H]2N2CCOCC2)c1 ZINC000880556241 ED On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)N[C@@H]2CCCC[C@H]2N2CCOCC2)c1 ZINC000880556242 ED On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)N[C@H]2CCCC[C@H]2N2CCOCC2)c1 ZINC000880556243 ED On-Demand Anodyne CCR3 15 40 COC(=O)c1cccc(NC2CCN(C(=O)Nc3cncc(OC)c3)CC2)c1 ZINC000880556244 GF On-Demand Anodyne EPHX2 21 43 COc1cncc(NC(=O)NC[C@@H]2CCN(c3cc(OC)cc(OC)c3)C2)c1 ZINC000880556249 GF On-Demand Anodyne CCR3 34 40 COc1cncc(NC(=O)NC[C@H]2CCN(c3cc(OC)cc(OC)c3)C2)c1 ZINC000880556250 GF On-Demand Anodyne CCR3 34 40 COc1cncc(NC(=O)N2CC[C@@H](C)C2)c1 ZINC000880556264 BD On-Demand Anodyne TRPC6 20 40 COc1cncc(NC(=O)N2CC[C@@H](C)C2)c1 ZINC000880556264 BD On-Demand Anodyne TRPC3 22 40 COc1cncc(NC(=O)N2CC[C@H](C)C2)c1 ZINC000880556265 BD On-Demand Anodyne TRPC6 20 40 COc1cncc(NC(=O)N2CC[C@H](C)C2)c1 ZINC000880556265 BD On-Demand Anodyne TRPC3 22 40 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccco2)c1 ZINC000880556269 DE On-Demand Anodyne ROCK2 25 47 COc1cncc(NC(=O)N2CCC(C)(O)CC2)c1 ZINC000880556272 CD On-Demand Anodyne PDGFRB 41 37 COc1cncc(NC(=O)N2CCC(C)(O)CC2)c1 ZINC000880556272 CD On-Demand Anodyne S1PR2 28 43 COc1cncc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880556280 DH On-Demand Anodyne CCR1 22 41 COc1cncc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880556280 DH On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880556281 DH On-Demand Anodyne CCR1 22 41 COc1cncc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880556281 DH On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N2CCC3(CC2)OCc2ccccc23)c1 ZINC000880556284 EG On-Demand Anodyne NPY5R 39 46 COc1cncc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)c1 ZINC000880556287 FE On-Demand Anodyne EPHX2 34 46 COc1cncc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)c1 ZINC000880556287 FE On-Demand Anodyne CACNA1I 49 35 COc1cncc(NC(=O)N[C@@H]2CCN(c3ncccc3F)C2)c1 ZINC000880556288 EE On-Demand Anodyne CCR3 26 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3ncccc3F)C2)c1 ZINC000880556288 EE On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N[C@H]2CCN(c3ncccc3F)C2)c1 ZINC000880556289 EE On-Demand Anodyne CCR3 26 41 COc1cncc(NC(=O)N[C@H]2CCN(c3ncccc3F)C2)c1 ZINC000880556289 EE On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCCN(c3cc(OC)cc(OC)c3)CC2)c1 ZINC000880556300 GF On-Demand Anodyne PDGFRB 52 41 COc1cncc(NC(=O)N2CCN(c3nc4ccccc4o3)CC2)c1 ZINC000880556346 FF On-Demand Anodyne PDGFRB 54 42 COc1cncc(NC(=O)N2CCN(c3nc4ccccc4o3)CC2)c1 ZINC000880556346 FF On-Demand Anodyne SSTR1 40 36 COc1cncc(NC(=O)N2CCN(c3nc4ccccc4o3)CC2)c1 ZINC000880556346 FF On-Demand Anodyne FAAH 25 44 COc1cncc(NC(=O)N2CCN(c3nc4ccccc4o3)CC2)c1 ZINC000880556346 FF On-Demand Anodyne DGAT1 18 40 COc1cncc(NC(=O)N2CCN(c3nc4ccccc4o3)CC2)c1 ZINC000880556346 FF On-Demand Anodyne NPBWR1 61 46 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556363 DF On-Demand Anodyne DRD4 33 42 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556363 DF On-Demand Anodyne SIGMAR1 26 40 NC(=O)c1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556363 DF On-Demand Anodyne NOD2 42 35 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne PREP 24 43 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne DPP7 50 34 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne XIAP 50 35 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne BIRC3 45 35 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne BIRC2 95 36 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556367 GD On-Demand Anodyne BIRC8 46 33 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne PREP 24 43 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne DPP7 50 34 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne XIAP 50 35 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne BIRC3 45 35 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne BIRC2 95 36 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N1CCCCC1 ZINC000880556368 GD On-Demand Anodyne BIRC8 46 33 COc1cncc(NC(=O)N[C@H](C)Cc2ccc(OC)c(OC)c2)c1 ZINC000880556376 EF On-Demand Anodyne ENPP1 56 32 COc1cncc(NC(=O)N[C@@H](C)Cc2ccc(OC)c(OC)c2)c1 ZINC000880556377 EF On-Demand Anodyne ENPP1 56 32 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)N1CCN(C(=O)C2CC2)CC1 ZINC000880556385 GD On-Demand Anodyne PREP 65 41 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556388 FE On-Demand Anodyne PAPA1_CARPA 35 47 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556388 FE On-Demand Anodyne REN 59 37 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556388 FE On-Demand Anodyne FPR1 44 37 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2N2CCCC2=O)C1 ZINC000880556390 FC On-Demand Anodyne KCNQ2 49 35 c1ccc2c(c1)CN(Cc1nc3ccccc3[nH]1)C[C@@H]1CCCN21 ZINC000880556393 DH On-Demand Anodyne KCNN3 29 40 COc1cncc(NC(=O)N[C@H]2CCOc3cc(OC)ccc32)c1 ZINC000880556398 EF On-Demand Anodyne TRPV1 16 49 COc1cncc(NC(=O)N[C@@H]2CCOc3cc(OC)ccc32)c1 ZINC000880556399 EF On-Demand Anodyne TRPV1 16 49 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne HRH2 24 43 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne SIGMAR1 30 40 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne CCR3 30 43 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne NPFFR2 43 52 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne UTS2R 15 40 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne FAAH 18 42 COc1cncc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556402 FD On-Demand Anodyne NPFFR1 54 52 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne HRH2 24 43 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne SIGMAR1 30 40 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne CCR3 30 43 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne NPFFR2 43 52 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne UTS2R 15 40 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne FAAH 18 42 COc1cncc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c1 ZINC000880556403 FD On-Demand Anodyne NPFFR1 54 52 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC1CCCCC1 ZINC000880556409 EF On-Demand Anodyne BIRC2 46 37 COc1cncc(NC(=O)NCC2(O)Cc3ccccc3C2)c1 ZINC000880556411 DD On-Demand Anodyne MTNR1B 27 40 COc1cncc(NC(=O)NCC2(O)Cc3ccccc3C2)c1 ZINC000880556411 DD On-Demand Anodyne ROCK2 24 45 COc1ccccc1/C(C)=C/C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556414 EF On-Demand Anodyne DRD2 21 40 COc1ccccc1/C(C)=C/C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556414 EF On-Demand Anodyne KCNA3 43 39 COc1ccccc1/C(C)=C\C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556415 EF On-Demand Anodyne DRD2 21 40 COc1ccccc1/C(C)=C\C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556415 EF On-Demand Anodyne KCNA3 43 39 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC[C@H]1CCCO1 ZINC000880556417 ED On-Demand Anodyne PDE8B 15 40 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC[C@@H]1CCCO1 ZINC000880556418 ED On-Demand Anodyne PDE8B 15 40 COc1cncc(NC(=O)NC[C@H](c2cccnc2)C(C)C)c1 ZINC000880556452 DG On-Demand Anodyne KCNA5 23 49 COc1cncc(NC(=O)NC[C@H](c2cccnc2)C(C)C)c1 ZINC000880556452 DG On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)NC[C@@H](c2cccnc2)C(C)C)c1 ZINC000880556453 DG On-Demand Anodyne KCNA5 23 49 COc1cncc(NC(=O)NC[C@@H](c2cccnc2)C(C)C)c1 ZINC000880556453 DG On-Demand Anodyne ROCK2 15 41 O=C(NCc1cn(C2CCC2)nn1)c1ccc(N2CCOC2=O)cc1 ZINC000880556454 ED On-Demand Anodyne CA14 17 48 COc1cncc(NC(=O)N[C@H](C)CNc2ccccc2)c1 ZINC000880556457 DF On-Demand Anodyne CTSK 16 47 COc1cncc(NC(=O)N[C@H](C)CNc2ccccc2)c1 ZINC000880556457 DF On-Demand Anodyne CTSL 18 40 COc1cncc(NC(=O)N[C@@H](C)CNc2ccccc2)c1 ZINC000880556458 DF On-Demand Anodyne CTSK 16 47 COc1cncc(NC(=O)N[C@@H](C)CNc2ccccc2)c1 ZINC000880556458 DF On-Demand Anodyne CTSL 18 40 COc1cncc(NC(=O)N(C)[C@H](C)Cc2ccc(O)cc2)c1 ZINC000880556459 DF On-Demand Anodyne NPY5R 36 56 COc1cncc(NC(=O)N(C)[C@@H](C)Cc2ccc(O)cc2)c1 ZINC000880556460 DF On-Demand Anodyne NPY5R 36 56 COc1cncc(NC(=O)N2CCC[C@H](Nc3ccccc3)C2)c1 ZINC000880556498 EG On-Demand Anodyne PDGFRB 44 40 COc1cncc(NC(=O)N2CCC[C@H](Nc3ccccc3)C2)c1 ZINC000880556498 EG On-Demand Anodyne CCR3 17 49 COc1cncc(NC(=O)N2CCC[C@H](Nc3ccccc3)C2)c1 ZINC000880556498 EG On-Demand Anodyne FAAH 17 46 COc1cncc(NC(=O)N2CCC[C@@H](Nc3ccccc3)C2)c1 ZINC000880556499 EG On-Demand Anodyne PDGFRB 44 40 COc1cncc(NC(=O)N2CCC[C@@H](Nc3ccccc3)C2)c1 ZINC000880556499 EG On-Demand Anodyne CCR3 17 49 COc1cncc(NC(=O)N2CCC[C@@H](Nc3ccccc3)C2)c1 ZINC000880556499 EG On-Demand Anodyne FAAH 17 46 COc1cncc(NC(=O)N2CCc3c(F)ccc(F)c3C2)c1 ZINC000880556506 DF On-Demand Anodyne P2RY14 48 35 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCC1 ZINC000880556513 CE On-Demand Anodyne PREP 60 40 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NNC(=O)c1cccs1 ZINC000880556516 FD On-Demand Reactive NOS1 27 43 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccn3)C2)c1 ZINC000880556523 DE On-Demand Anodyne PDE3A 38 45 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccn3)C2)c1 ZINC000880556523 DE On-Demand Anodyne PDE3B 44 45 COc1cncc(NC(=O)N2CC[C@@H](Oc3ccccn3)C2)c1 ZINC000880556523 DE On-Demand Anodyne EPHX2 18 46 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccn3)C2)c1 ZINC000880556524 DE On-Demand Anodyne PDE3A 38 45 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccn3)C2)c1 ZINC000880556524 DE On-Demand Anodyne PDE3B 44 45 COc1cncc(NC(=O)N2CC[C@H](Oc3ccccn3)C2)c1 ZINC000880556524 DE On-Demand Anodyne EPHX2 18 46 CCn1nc2c(cc1=O)CN(C(=O)Nc1cncc(OC)c1)CC2 ZINC000880556527 ED On-Demand Anodyne P2RY14 48 35 CNC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880556545 CD On-Demand Anodyne OPRL1 22 45 CNC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880556545 CD On-Demand Anodyne BIRC2 63 36 COc1cncc(NC(=O)N2CCC3(CCCCC3)C2)c1 ZINC000880556549 CG On-Demand Anodyne EPHX2 34 47 CCN1CCC(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)CC1 ZINC000880556570 FE On-Demand Anodyne CHRM1 16 42 CCN1CCC(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)CC1 ZINC000880556570 FE On-Demand Anodyne SIGMAR1 17 40 COc1cncc(NC(=O)NC2CCN(c3ccc(N(C)C)cc3)CC2)c1 ZINC000880556571 FF On-Demand Anodyne EPHX2 43 37 NC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880556576 DF On-Demand Anodyne KCNH2 41 40 NC(=O)c1cccc(CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880556576 DF On-Demand Anodyne F10 17 48 O=C1CCCc2cc(C(=O)NCc3cn(C4CCC4)nn3)ccc2N1 ZINC000880556578 EE On-Demand Anodyne HDAC9 19 42 COc1cncc(NC(=O)N2CCN(C[C@H]3CCOC3)CC2)c1 ZINC000880556586 DD On-Demand Anodyne PDGFRB 41 36 COc1cncc(NC(=O)N2CCN(C[C@@H]3CCOC3)CC2)c1 ZINC000880556587 DD On-Demand Anodyne PDGFRB 41 36 COc1cncc(NC(=O)N[C@H](C)CCc2cccn2C)c1 ZINC000880556595 DF On-Demand Anodyne CCR3 52 34 COc1cncc(NC(=O)N[C@@H](C)CCc2cccn2C)c1 ZINC000880556596 DF On-Demand Anodyne CCR3 52 34 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCCCN1CCCC1=O ZINC000880556597 FD On-Demand Anodyne TYRO3 19 44 COCCC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556601 ED On-Demand Anodyne C3AR1 37 41 COCCC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556601 ED On-Demand Anodyne EPHX2 52 55 COCCC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556601 ED On-Demand Anodyne CXCR3 15 42 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne HTR1A 68 50 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne DRD2 55 38 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne ADRA1D 48 40 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne HTR1D 17 50 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne HTR1B 21 50 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne HTR2A 16 40 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne ADRA1A 45 40 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne ADRA1B 33 40 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne DRD3 65 38 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne PDGFRB 70 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne HTR7 51 44 COc1cncc(NC(=O)N2CCN(c3ccccc3OCCN(C)C)CC2)c1 ZINC000880556602 GE On-Demand Anodyne RBP4 21 41 COc1cncc(NC(=O)N2CCn3c(Cc4ccccc4)nnc3C2)c1 ZINC000880556611 FE On-Demand Anodyne PDGFRB 28 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(C)cc3)CC2)c1 ZINC000880556623 EG On-Demand Anodyne PDGFRB 30 41 COc1cncc(NC(=O)N2CCC(Oc3ccc(C)cc3)CC2)c1 ZINC000880556623 EG On-Demand Anodyne PRSS2 54 30 COc1cncc(NC(=O)N2CCC(Oc3ccc(C)cc3)CC2)c1 ZINC000880556623 EG On-Demand Anodyne EPHX2 34 49 COc1cncc(NC(=O)N2CCC(Oc3ccc(C)cc3)CC2)c1 ZINC000880556623 EG On-Demand Anodyne SCD1 19 48 COc1cncc(NC(=O)Nc2cnn(C)c2C)c1 ZINC000880556626 CD On-Demand Anodyne HTR2A 23 41 COc1cncc(NC(=O)N[C@@H](C)c2cccc(N3CCCC3)c2)c1 ZINC000880556628 EH On-Demand Anodyne KCNQ2 41 40 COc1cncc(NC(=O)N[C@H](C)c2cccc(N3CCCC3)c2)c1 ZINC000880556630 EH On-Demand Anodyne KCNQ2 41 40 COc1cncc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880556644 EG On-Demand Anodyne EPHX2 47 39 COc1cncc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880556644 EG On-Demand Anodyne L3MBTL3 45 33 CC[C@@H](O)CCCNC(=O)Nc1cncc(OC)c1 ZINC000880556648 CD On-Demand Anodyne ADRB1 40 29 CC[C@H](O)CCCNC(=O)Nc1cncc(OC)c1 ZINC000880556649 CD On-Demand Anodyne ADRB1 40 29 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)[C@H]2C)c1 ZINC000880556656 DH On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)[C@H]2C)c1 ZINC000880556656 DH On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)[C@H]2C)c1 ZINC000880556661 DH On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)[C@H]2C)c1 ZINC000880556661 DH On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)[C@@H]2C)c1 ZINC000880556663 DH On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)[C@@H]2C)c1 ZINC000880556663 DH On-Demand Anodyne EPHX2 15 40 COCc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1F ZINC000880556664 DF On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)[C@@H]2C)c1 ZINC000880556665 DH On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)[C@@H]2C)c1 ZINC000880556665 DH On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)N2CCOC3(CCCC3)C2)c1 ZINC000880556671 CE On-Demand Anodyne EPHX2 28 47 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccccc2)C1 ZINC000880556672 DC On-Demand Anodyne MMP13 28 42 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccccc2)C1 ZINC000880556672 DC On-Demand Anodyne ADAM17 32 42 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccccc2)C1 ZINC000880556672 DC On-Demand Anodyne MMP9 18 42 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccccc2)C1 ZINC000880556672 DC On-Demand Anodyne SLC12A5 46 37 COc1cncc(NC(=O)N2CCC3(C2)OCCO3)c1 ZINC000880556674 CD On-Demand Anodyne EPHX2 32 40 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne DRD4 15 40 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne HTR4 52 45 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne SSTR5 40 36 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne CCR3 44 43 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne CHRNA7 17 41 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne EPHX2 54 48 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne CXCR3 20 45 CCCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880556680 DE On-Demand Anodyne MCHR1 20 47 COc1cncc(NC(=O)N[C@@H]2CCN(c3c(F)cccc3F)C2)c1 ZINC000880556686 EF On-Demand Anodyne CCR3 34 41 COc1cncc(NC(=O)N[C@@H]2CCN(c3c(F)cccc3F)C2)c1 ZINC000880556686 EF On-Demand Anodyne EPHX2 44 37 COc1cncc(NC(=O)N[C@H]2CCN(c3c(F)cccc3F)C2)c1 ZINC000880556687 EF On-Demand Anodyne CCR3 34 41 COc1cncc(NC(=O)N[C@H]2CCN(c3c(F)cccc3F)C2)c1 ZINC000880556687 EF On-Demand Anodyne EPHX2 44 37 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne F2 25 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PLG 22 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne KLKB1 15 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PRSS1 15 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne ACE 42 39 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne OPRM1 48 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne OPRD1 42 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CELA1 18 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne MME 54 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne TACR1 25 49 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSD 46 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PGC 84 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CMA1 36 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTRA_BOVIN 25 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne FCER2 72 38 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSB 63 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PAPA1_CARPA 88 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne TRY1_BOVIN 41 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CYSP_TRYCR 62 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CCKAR 73 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSK 35 53 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSL 67 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CACNA1B 57 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PGA 44 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne NPFFR2 57 32 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne TIMP3 80 39 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PREP 15 50 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne TACR3 27 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CAPNS1 74 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne MMP3 21 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne HLA-DRB1 65 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne REN 163 50 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne REN1 81 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CCKBR 28 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSS 35 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CAPN1 92 51 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CAPN2 109 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSE 36 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PGA5 31 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne SCN10A 24 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne CTSV 42 32 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne MMP1 25 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne FPR1 93 53 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne PSMB5 60 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne BRCA1 60 32 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556694 GF On-Demand Anodyne NPFFR1 52 32 O=C(NCCCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556696 ED On-Demand Anodyne FKBP1A 27 42 O=C(NCCCc1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880556696 ED On-Demand Anodyne PREP 49 48 COc1cncc(NC(=O)N2CCC[C@@H]2c2ncc(-c3ccc(F)cc3)[nH]2)c1 ZINC000880556706 GH On-Demand Anodyne PRCP 27 48 COc1cncc(NC(=O)N2CCC[C@H]2c2ncc(-c3ccc(F)cc3)[nH]2)c1 ZINC000880556708 GH On-Demand Anodyne PRCP 27 48 COc1cncc(NC(=O)NCc2ccc(C)cc2OC)c1 ZINC000880556729 DF On-Demand Anodyne ROCK2 15 53 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)C3CC3)C[C@H]2C)c1 ZINC000880556742 ED On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)C3CC3)C[C@H]2C)c1 ZINC000880556743 ED On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)C3CC3)C[C@@H]2C)c1 ZINC000880556744 ED On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)C3CC3)C[C@@H]2C)c1 ZINC000880556745 ED On-Demand Anodyne EPHX2 19 40 CCC(=O)N1CC[C@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880556746 CD On-Demand Anodyne EPHX2 46 62 CCC(=O)N1CC[C@@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880556747 CD On-Demand Anodyne EPHX2 46 62 COc1cncc(NC(=O)NCc2ccc3c(c2)COC3)c1 ZINC000880556752 CE On-Demand Anodyne ROCK2 34 45 COc1cncc(NC(=O)N[C@H](C)C[C@@H](O)c2ccc(F)cc2)c1 ZINC000880556754 EF On-Demand Anodyne CCR3 51 37 COc1cncc(NC(=O)N[C@H](C)C[C@H](O)c2ccc(F)cc2)c1 ZINC000880556755 EF On-Demand Anodyne CCR3 51 37 COc1cncc(NC(=O)N[C@@H](C)C[C@@H](O)c2ccc(F)cc2)c1 ZINC000880556756 EF On-Demand Anodyne CCR3 51 37 COc1cncc(NC(=O)N[C@@H](C)C[C@H](O)c2ccc(F)cc2)c1 ZINC000880556757 EF On-Demand Anodyne CCR3 51 37 COC(=O)C1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880556758 CD On-Demand Anodyne PTR1 46 34 COc1cncc(NC(=O)N2CCCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880556762 GF On-Demand Anodyne PDGFRB 40 40 COc1cncc(NC(=O)N2CCCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880556762 GF On-Demand Anodyne C3AR1 39 42 COc1cncc(NC(=O)N2CCCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880556762 GF On-Demand Anodyne FAAH 35 47 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880556769 GF On-Demand Anodyne F2 26 40 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880556769 GF On-Demand Anodyne GRIN2B 24 47 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880556769 GF On-Demand Anodyne PREP 50 54 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880556769 GF On-Demand Anodyne EPHX2 23 40 O=C(NCc1cn(C2CCC2)nn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880556769 GF On-Demand Anodyne TMPRSS11D 65 41 Oc1nc(CN2Cc3ccccc3N3CCC[C@H]3C2)nc2c1oc1ccccc12 ZINC000880556778 GI On-Demand Anodyne PIM1 17 48 Oc1nc(CN2Cc3ccccc3N3CCC[C@H]3C2)nc2c1oc1ccccc12 ZINC000880556778 GI On-Demand Anodyne CDC7 20 48 Oc1nc(CN2Cc3ccccc3N3CCC[C@H]3C2)nc2c1oc1ccccc12 ZINC000880556778 GI On-Demand Anodyne PIM3 20 48 CCN1CCC[C@@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880556782 CD On-Demand Anodyne CCR3 61 44 CCN1CCC[C@H](NC(=O)Nc2cncc(OC)c2)C1 ZINC000880556784 CD On-Demand Anodyne CCR3 61 44 COc1cncc(NC(=O)N(Cc2ccccc2)CC(F)F)c1 ZINC000880556793 DG On-Demand Anodyne ROCK1 18 42 COc1cncc(NC(=O)N(Cc2ccccc2)CC(F)F)c1 ZINC000880556793 DG On-Demand Anodyne ROCK2 28 44 COc1cncc(NC(=O)N(Cc2ccccc2)CC(F)F)c1 ZINC000880556793 DG On-Demand Anodyne PTGES 24 41 COc1cncc(NC(=O)NCCCN2C(=O)COc3ccccc32)c1 ZINC000880556794 FE On-Demand Anodyne DRD2 18 40 COc1cncc(NC(=O)NCCCN2C(=O)COc3ccccc32)c1 ZINC000880556794 FE On-Demand Anodyne CCR3 21 42 COc1cncc(NC(=O)N(C)CCCn2ccnc2)c1 ZINC000880556803 CD On-Demand Anodyne TBXAS1 41 39 COc1cncc(NC(=O)N(C)CCCn2ccnc2)c1 ZINC000880556803 CD On-Demand Anodyne QPCT 43 52 COc1cncc(NC(=O)N2CCN(c3cc(N4CCOCC4)ncn3)CC2)c1 ZINC000880556822 GD On-Demand Anodyne PDGFRB 61 43 COc1cncc(NC(=O)N2CCN(c3cc(N4CCOCC4)ncn3)CC2)c1 ZINC000880556822 GD On-Demand Anodyne DGAT1 21 42 COc1cncc(NC(=O)N2CCc3ncnc(N4CCOCC4)c3C2)c1 ZINC000880556827 FD On-Demand Anodyne PDGFRB 53 42 O=C(NCc1cn(C2CCC2)nn1)c1ccnc(-n2ccnc2)c1 ZINC000880556828 DD On-Demand Anodyne NOS2 60 33 COc1cncc(NC(=O)N(C)C[C@@H](O)CN2CCOCC2)c1 ZINC000880556829 DC On-Demand Anodyne CASR 26 42 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2cc(Cl)ccc2Cl)C1 ZINC000880556830 GD On-Demand Anodyne CCR1 18 47 COc1cncc(NC(=O)N(C)C[C@H](O)CN2CCOCC2)c1 ZINC000880556831 DC On-Demand Anodyne CASR 26 42 COc1cncc(NC(=O)N[C@H]2CCc3c(OC)cccc32)c1 ZINC000880556846 DF On-Demand Anodyne TRPV1 19 42 COc1cncc(NC(=O)N[C@@H]2CCc3c(OC)cccc32)c1 ZINC000880556848 DF On-Demand Anodyne TRPV1 19 42 COc1cncc(NC(=O)N[C@@H](CCSC)C(=O)N(C)OC)c1 ZINC000880556853 ED On-Demand Anodyne FPR1 28 41 COc1cncc(NC(=O)NCCCCN2CCC[C@H]2CO)c1 ZINC000880556865 DD On-Demand Anodyne CCR3 45 45 COc1cncc(NC(=O)NCCCCN2CCC[C@@H]2CO)c1 ZINC000880556867 DD On-Demand Anodyne CCR3 45 45 COc1cncc(NC(=O)Nc2cccc(CS(C)(=O)=O)c2C)c1 ZINC000880556880 EF On-Demand Anodyne LPL 42 34 COc1cncc(NC(=O)Nc2cccc(CS(C)(=O)=O)c2C)c1 ZINC000880556880 EF On-Demand Anodyne CA12 15 40 CCCCNC(=O)NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880556885 EE On-Demand Anodyne TPP2 41 39 COc1cncc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)c1 ZINC000880556897 EF On-Demand Anodyne PIK3CA 17 40 COc1cncc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)c1 ZINC000880556897 EF On-Demand Anodyne RAF1 22 42 COc1cncc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)c1 ZINC000880556897 EF On-Demand Anodyne MTOR 36 40 COc1cncc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)c1 ZINC000880556897 EF On-Demand Anodyne PIK3CG 16 40 COc1cncc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)c1 ZINC000880556897 EF On-Demand Anodyne PDGFRA 41 35 COc1cncc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)c1 ZINC000880556898 EF On-Demand Anodyne PIK3CA 17 40 COc1cncc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)c1 ZINC000880556898 EF On-Demand Anodyne RAF1 22 42 COc1cncc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)c1 ZINC000880556898 EF On-Demand Anodyne MTOR 36 40 COc1cncc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)c1 ZINC000880556898 EF On-Demand Anodyne PIK3CG 16 40 COc1cncc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)c1 ZINC000880556898 EF On-Demand Anodyne PDGFRA 41 35 COc1cncc(NC(=O)N[C@H](CCO)c2ccccc2)c1 ZINC000880556902 DE On-Demand Anodyne ROCK1 15 56 COc1cncc(NC(=O)N[C@H](CCO)c2ccccc2)c1 ZINC000880556902 DE On-Demand Anodyne TACR3 20 40 COc1cncc(NC(=O)N[C@H](CCO)c2ccccc2)c1 ZINC000880556902 DE On-Demand Anodyne ROCK2 15 56 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)c1 ZINC000880556903 EF On-Demand Anodyne F7 17 44 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)c1 ZINC000880556904 EF On-Demand Anodyne F7 17 44 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@@H](C)O)c1 ZINC000880556908 DF On-Demand Anodyne ROCK1 20 44 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@@H](C)O)c1 ZINC000880556908 DF On-Demand Anodyne ROCK2 30 44 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@@H](C)O)c1 ZINC000880556908 DF On-Demand Anodyne NPY5R 35 42 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@@H](C)O)c1 ZINC000880556908 DF On-Demand Anodyne PTGES 27 43 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@H](C)O)c1 ZINC000880556909 DF On-Demand Anodyne ROCK1 20 44 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@H](C)O)c1 ZINC000880556909 DF On-Demand Anodyne ROCK2 30 44 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@H](C)O)c1 ZINC000880556909 DF On-Demand Anodyne NPY5R 35 42 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@H](C)O)c1 ZINC000880556909 DF On-Demand Anodyne PTGES 27 43 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556910 GE On-Demand Anodyne LTA4H 51 39 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556910 GE On-Demand Anodyne CA7 21 41 NS(=O)(=O)c1ccc(OCCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880556910 GE On-Demand Anodyne MEN1 17 44 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@H](C)C2)c1 ZINC000880556911 CD On-Demand Anodyne EPHX2 40 38 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@H](C)C2)c1 ZINC000880556912 CD On-Demand Anodyne EPHX2 40 38 COc1cncc(NC(=O)N[C@H]2CCN(C)[C@@H](C)C2)c1 ZINC000880556913 CD On-Demand Anodyne EPHX2 40 38 COc1cncc(NC(=O)N[C@@H]2CCN(C)[C@@H](C)C2)c1 ZINC000880556914 CD On-Demand Anodyne EPHX2 40 38 COC(=O)[C@@]1(O)CCN(CC(=O)NCCC(c2ccccc2)c2ccccc2)C1 ZINC000880556920 GD On-Demand Anodyne ADRA1A 24 44 COC(=O)[C@@]1(O)CCN(CC(=O)NCCC(c2ccccc2)c2ccccc2)C1 ZINC000880556920 GD On-Demand Anodyne ADRA1B 16 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCCC(c2ccccc2)c2ccccc2)C1 ZINC000880556920 GD On-Demand Anodyne OPRL1 19 42 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne HTR1A 27 47 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne DRD2 22 44 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne DRD4 42 47 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne DRD3 25 42 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne P2RX3 26 42 COc1cncc(NC(=O)N[C@@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556929 FD On-Demand Anodyne EBP 19 40 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne HTR1A 27 47 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne DRD2 22 44 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne DRD4 42 47 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne DRD3 25 42 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne P2RX3 26 42 COc1cncc(NC(=O)N[C@H](C)CN2CCN(c3ccccn3)CC2)c1 ZINC000880556930 FD On-Demand Anodyne EBP 19 40 COc1cncc(NC(=O)NC2CCN(CC(=O)N(C)C)CC2)c1 ZINC000880556931 EC On-Demand Anodyne CCR3 25 41 COc1cncc(NC(=O)NC2CCN(CC(=O)N(C)C)CC2)c1 ZINC000880556931 EC On-Demand Anodyne EPHX2 44 39 COc1cncc(NC(=O)NC2CCN(CC(=O)N(C)C)CC2)c1 ZINC000880556931 EC On-Demand Anodyne CXCR3 19 44 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC1CCCC1 ZINC000880556934 DF On-Demand Anodyne SIGMAR1 17 40 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC1CCCC1 ZINC000880556934 DF On-Demand Anodyne BIRC2 45 36 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCOC3)CC2)c1 ZINC000880556940 ED On-Demand Anodyne CCR3 23 44 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCOC3)CC2)c1 ZINC000880556940 ED On-Demand Anodyne EPHX2 35 42 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCOC3)CC2)c1 ZINC000880556940 ED On-Demand Anodyne PDK1 46 36 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCOC3)CC2)c1 ZINC000880556940 ED On-Demand Anodyne CXCR3 19 44 COc1cncc(NC(=O)NC(C)(C)C)c1 ZINC000880556945 BE On-Demand Anodyne IMDH_CRYPV 20 41 COc1cncc(NC(=O)N2CCN(CC(=O)N(C)C)CC2)c1 ZINC000880556947 DC On-Demand Anodyne PDGFRB 41 37 COc1cncc(NC(=O)NC[C@H](CO)c2ccccc2)c1 ZINC000880556953 DD On-Demand Anodyne ROCK2 22 42 COc1cncc(NC(=O)NC[C@@H](CO)c2ccccc2)c1 ZINC000880556954 DD On-Demand Anodyne ROCK2 22 42 COc1cncc(NC(=O)N2CCOC3(CCCCCC3)C2)c1 ZINC000880556958 DG On-Demand Anodyne EPHX2 26 49 COc1cncc(NC(=O)N2CCc3ccc(F)c(F)c3C2)c1 ZINC000880556960 DF On-Demand Anodyne P2RY14 40 33 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)C3CCCC3)C2)c1 ZINC000880556961 EE On-Demand Anodyne EPHX2 43 45 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)C3CCCC3)C2)c1 ZINC000880556962 EE On-Demand Anodyne EPHX2 43 45 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(O)cc3)CC2)c1 ZINC000880556965 FD On-Demand Anodyne PDGFRB 49 39 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne DRD4 17 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne GRIN2B 23 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne SIGMAR1 15 44 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne CCR3 36 42 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne CHRNA7 23 44 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne C3AR1 46 47 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne EPHX2 42 47 COc1cncc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556967 FE On-Demand Anodyne MCHR1 17 48 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne DRD4 17 42 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne GRIN2B 23 42 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne SIGMAR1 15 44 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne CCR3 36 42 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne CHRNA7 23 44 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne C3AR1 46 47 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne EPHX2 42 47 COc1cncc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c1 ZINC000880556968 FE On-Demand Anodyne MCHR1 17 48 COc1cncc(NC(=O)N(CCCO)Cc2ccccc2)c1 ZINC000880556980 DF On-Demand Anodyne ROCK1 18 49 COc1cncc(NC(=O)N(CCCO)Cc2ccccc2)c1 ZINC000880556980 DF On-Demand Anodyne ROCK2 30 49 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne HTR1A 49 53 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne HTR1D 17 53 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne HTR1B 23 53 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne HTR2C 15 44 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne DRD3 49 36 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne PDGFRB 56 47 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne HTR7 40 48 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne FAAH 22 47 COc1cncc(NC(=O)N2CCN(c3ccccc3O)CC2)c1 ZINC000880556981 EE On-Demand Anodyne RBP4 17 46 COc1cncc(NC(=O)NCCc2csc(C)n2)c1 ZINC000880556996 CE On-Demand Anodyne PIK3CG 15 44 COc1cncc(NC(=O)NCCS(=O)(=O)CC2CC2)c1 ZINC000880556997 DD On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)N[C@@H]2CCC(F)(F)C2)c1 ZINC000880556998 CE On-Demand Anodyne EPHX2 40 33 COc1cncc(NC(=O)N[C@H]2CCC(F)(F)C2)c1 ZINC000880556999 CE On-Demand Anodyne EPHX2 40 33 COc1cncc(NC(=O)N2CCN(c3cccs3)CC2)c1 ZINC000880557000 DF On-Demand Anodyne PDGFRB 52 41 COc1cncc(NC(=O)N2CCN(c3cccs3)CC2)c1 ZINC000880557000 DF On-Demand Anodyne FAAH 19 46 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne HTR1A 42 45 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne DRD2 38 43 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne DRD4 22 49 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne DRD3 60 50 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne HTR7 41 38 CC(=O)NCCCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557004 CD On-Demand Anodyne MTNR1A 16 42 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)Nc1nccs1 ZINC000880557006 EF On-Demand Anodyne MAP1 108 45 COc1cncc(NC(=O)N2CCN(C3CCCCC3)CC2)c1 ZINC000880557009 DF On-Demand Anodyne HRH3 27 43 COc1cncc(NC(=O)N(Cc2cccc([N+](=O)[O-])c2)C2CC2)c1 ZINC000880557011 EG On-Demand Bother CACNA1C 54 38 COc1cncc(NC(=O)N(Cc2cccc([N+](=O)[O-])c2)C2CC2)c1 ZINC000880557011 EG On-Demand Bother CACNA1D 83 38 COc1cncc(NC(=O)N(Cc2cccc([N+](=O)[O-])c2)C2CC2)c1 ZINC000880557011 EG On-Demand Bother ROCK2 33 54 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCOC3)CC2)c1 ZINC000880557012 ED On-Demand Anodyne CCR3 23 44 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCOC3)CC2)c1 ZINC000880557012 ED On-Demand Anodyne EPHX2 35 42 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCOC3)CC2)c1 ZINC000880557012 ED On-Demand Anodyne PDK1 46 36 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCOC3)CC2)c1 ZINC000880557012 ED On-Demand Anodyne CXCR3 19 44 COc1cncc(NC(=O)N2CCN(c3ccc(OC)c(F)c3)CC2)c1 ZINC000880557013 FF On-Demand Clean HTR1B 15 54 COc1cncc(NC(=O)N2CCN(c3ccc(OC)c(F)c3)CC2)c1 ZINC000880557013 FF On-Demand Clean PDGFRB 57 41 COc1cncc(NC(=O)N2CCN(c3ccc(OC)c(F)c3)CC2)c1 ZINC000880557013 FF On-Demand Clean SSTR1 29 40 COc1cncc(NC(=O)N2CCN(c3ccc(OC)c(F)c3)CC2)c1 ZINC000880557013 FF On-Demand Clean RBP4 20 41 COc1cncc(NC(=O)N2CCCN(Cc3nccn3C)CC2)c1 ZINC000880557016 ED On-Demand Anodyne PDGFRB 45 35 COc1cncc(NC(=O)Nc2ccccc2CCC(F)(F)F)c1 ZINC000880557017 EI On-Demand Anodyne TRPV1 15 42 COc1cncc(NC(=O)Nc2ccccc2CCC(F)(F)F)c1 ZINC000880557017 EI On-Demand Anodyne P2RY1 87 41 COc1cncc(NC(=O)NC[C@H]2CCN(CC(C)C)C2)c1 ZINC000880557021 DE On-Demand Anodyne HTR4 31 40 COc1cncc(NC(=O)NC[C@H]2CCN(CC(C)C)C2)c1 ZINC000880557021 DE On-Demand Anodyne CCR3 50 41 COc1cncc(NC(=O)NC[C@H]2CCN(CC(C)C)C2)c1 ZINC000880557021 DE On-Demand Anodyne CACNA1I 59 36 COc1cncc(NC(=O)NC[C@@H]2CCN(CC(C)C)C2)c1 ZINC000880557023 DE On-Demand Anodyne HTR4 31 40 COc1cncc(NC(=O)NC[C@@H]2CCN(CC(C)C)C2)c1 ZINC000880557023 DE On-Demand Anodyne CCR3 50 41 COc1cncc(NC(=O)NC[C@@H]2CCN(CC(C)C)C2)c1 ZINC000880557023 DE On-Demand Anodyne CACNA1I 59 36 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne HTR1A 59 44 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne DRD2 53 47 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne DRD4 36 42 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne ADRA1D 53 47 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne ADRA1A 47 47 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne ADRA1B 41 47 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne DRD3 59 40 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne HTR7 41 37 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne MTNR1A 15 42 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne MTNR1B 15 42 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557030 EE On-Demand Anodyne EPHX2 36 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne HTR1A 59 44 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne DRD2 53 47 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne DRD4 36 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne ADRA1D 53 47 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne ADRA1A 47 47 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne ADRA1B 41 47 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne DRD3 59 40 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne HTR7 41 37 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne MTNR1A 15 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne MTNR1B 15 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880557031 EE On-Demand Anodyne EPHX2 36 42 COc1cncc(NC(=O)N2CCCCC[C@H]2c2ccco2)c1 ZINC000880557034 DH On-Demand Anodyne CPT1A 46 34 COc1cncc(NC(=O)N2CCCCC[C@@H]2c2ccco2)c1 ZINC000880557036 DH On-Demand Anodyne CPT1A 46 34 c1ccc2c(c1)CN(Cc1cscn1)C[C@@H]1CCCN21 ZINC000880557037 CG On-Demand Anodyne SCN5A 43 36 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne PDGFRB 31 40 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne MAPK14 15 40 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne SSTR5 43 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne FAAH 15 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne EPHX2 45 41 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne MCHR1 25 48 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne SCD1 15 46 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne SMO 19 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000880557045 FF On-Demand Anodyne HPGDS 36 40 COc1cncc(NC(=O)N2CCO[C@H](c3ccsc3)C2)c1 ZINC000880557048 DF On-Demand Anodyne NPBWR1 78 33 COc1cncc(NC(=O)N2CCO[C@@H](c3ccsc3)C2)c1 ZINC000880557051 DF On-Demand Anodyne NPBWR1 78 33 COc1cncc(NC(=O)NCCCc2nnc3n2CCCCC3)c1 ZINC000880557056 EE On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)N(Cc2ccccc2)C2CC2)c1 ZINC000880557061 CG On-Demand Anodyne ROCK2 29 56 COc1cncc(NC(=O)N2CCC(c3ccccc3F)CC2)c1 ZINC000880557070 EH On-Demand Anodyne RBP4 67 46 COc1cncc(NC(=O)N2CCC(c3ccccc3F)CC2)c1 ZINC000880557070 EH On-Demand Anodyne SCD1 16 43 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1ccccc1 ZINC000880557071 EF On-Demand Anodyne SIGMAR1 24 41 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1ccccc1 ZINC000880557071 EF On-Demand Anodyne PDE11A 52 35 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCc1ccccc1 ZINC000880557071 EF On-Demand Anodyne TMPRSS11D 51 35 Nc1cc(C(=O)NCc2cn(C3CCC3)nn2)cc(Cl)n1 ZINC000880557072 DD On-Demand Anodyne CA14 17 43 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)Nc1ccccc1 ZINC000880557079 DG On-Demand Anodyne DRD4 16 42 COc1cncc(NC(=O)N(C)[C@@H](C)CCSC)c1 ZINC000880557080 CF On-Demand Anodyne NPY5R 30 40 COc1cncc(NC(=O)N(C)[C@H](C)CCSC)c1 ZINC000880557081 CF On-Demand Anodyne NPY5R 30 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)C1 ZINC000880557090 GC On-Demand Anodyne MAPK1 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)C1 ZINC000880557090 GC On-Demand Anodyne EPHX2 21 40 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557091 GD On-Demand Anodyne F2 45 37 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557091 GD On-Demand Anodyne PREP 19 40 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557091 GD On-Demand Anodyne LGMN 71 37 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557091 GD On-Demand Anodyne TMPRSS11D 60 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557092 GD On-Demand Anodyne F2 45 37 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557092 GD On-Demand Anodyne PREP 19 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557092 GD On-Demand Anodyne LGMN 71 37 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880557092 GD On-Demand Anodyne TMPRSS11D 60 34 COc1cncc(NC(=O)N2CCc3cccc(F)c3[C@H]2C)c1 ZINC000880557093 DG On-Demand Anodyne TRPM8 36 46 COc1cncc(NC(=O)N2CCc3cccc(F)c3[C@@H]2C)c1 ZINC000880557094 DG On-Demand Anodyne TRPM8 36 46 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne PDGFRB 94 52 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne FLT3 15 49 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne SIRT3 62 31 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne SIRT2 63 31 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne SIRT1 53 31 COc1cncc(NC(=O)N2CCN(c3ncnc4ccsc34)CC2)c1 ZINC000880557101 FE On-Demand Anodyne LIMK2 20 49 COc1cncc(NC(=O)NC(C)(C)c2cccs2)c1 ZINC000880557108 CG On-Demand Anodyne IMDH_CRYPV 43 40 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCCC1 ZINC000880557112 DE On-Demand Anodyne PREP 53 39 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc(Cl)c(Cl)c2)C1 ZINC000880557114 GD On-Demand Anodyne TACR1 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc(Cl)c(Cl)c2)C1 ZINC000880557114 GD On-Demand Anodyne TACR2 53 35 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc(Cl)c(Cl)c2)C1 ZINC000880557116 GD On-Demand Anodyne TACR1 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc(Cl)c(Cl)c2)C1 ZINC000880557116 GD On-Demand Anodyne TACR2 53 35 COc1cncc(NC(=O)NCc2cc(F)ccc2N2CCOCC2)c1 ZINC000880557127 FE On-Demand Anodyne P2RX7 33 43 COc1cncc(NC(=O)NCc2cc(F)ccc2N2CCOCC2)c1 ZINC000880557127 FE On-Demand Anodyne PIK3CA 31 40 COc1cncc(NC(=O)NCc2cc(F)ccc2N2CCOCC2)c1 ZINC000880557127 FE On-Demand Anodyne MTOR 45 40 COc1cncc(NC(=O)NCc2cc(F)ccc2N2CCOCC2)c1 ZINC000880557127 FE On-Demand Anodyne PIK3CG 29 40 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne HRH2 43 57 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne CCR3 18 45 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne RAF1 15 45 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne MTNR1A 66 55 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne MTNR1B 66 55 COc1cncc(NC(=O)NCCCOc2cccc(OC)c2)c1 ZINC000880557128 EF On-Demand Anodyne ROCK2 36 45 COc1cncc(NC(=O)N(C)Cc2ccc(S(C)(=O)=O)cc2)c1 ZINC000880557129 EE On-Demand Anodyne BMP1 43 40 COc1cncc(NC(=O)N(C)Cc2ccc(S(C)(=O)=O)cc2)c1 ZINC000880557129 EE On-Demand Anodyne ROCK2 17 44 COc1cncc(NC(=O)N(C)Cc2ccc(S(C)(=O)=O)cc2)c1 ZINC000880557129 EE On-Demand Anodyne LIMK2 21 42 COc1cncc(NC(=O)NC[C@@H](C)Oc2cccc(OC)c2)c1 ZINC000880557130 EF On-Demand Anodyne MTNR1A 45 60 COc1cncc(NC(=O)NC[C@@H](C)Oc2cccc(OC)c2)c1 ZINC000880557130 EF On-Demand Anodyne MTNR1B 44 60 COc1cncc(NC(=O)NC[C@@H](C)Oc2cccc(OC)c2)c1 ZINC000880557130 EF On-Demand Anodyne SOAT1 20 40 COc1cncc(NC(=O)NC[C@H](C)Oc2cccc(OC)c2)c1 ZINC000880557131 EF On-Demand Anodyne MTNR1A 45 60 COc1cncc(NC(=O)NC[C@H](C)Oc2cccc(OC)c2)c1 ZINC000880557131 EF On-Demand Anodyne MTNR1B 44 60 COc1cncc(NC(=O)NC[C@H](C)Oc2cccc(OC)c2)c1 ZINC000880557131 EF On-Demand Anodyne SOAT1 20 40 COc1cncc(NC(=O)Nc2ccc(CN(C(C)=O)C3CC3)cc2)c1 ZINC000880557132 FG On-Demand Anodyne RAF1 18 41 COc1cncc(NC(=O)Nc2ccc(CN(C(C)=O)C3CC3)cc2)c1 ZINC000880557132 FG On-Demand Anodyne ROCK2 18 46 COc1cncc(NC(=O)NC[C@H](CCO)c2ccccc2)c1 ZINC000880557137 DE On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)NC[C@@H](CCO)c2ccccc2)c1 ZINC000880557138 DE On-Demand Anodyne ROCK2 15 41 NC(=O)c1ccc(NC(=O)CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557153 GF On-Demand Anodyne AVPR2 59 39 NC(=O)c1ccc(NC(=O)CCN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557153 GF On-Demand Anodyne NOD2 40 34 COc1cncc(NC(=O)NCCOc2cc(OC)cc(OC)c2)c1 ZINC000880557156 EE On-Demand Anodyne HRH2 16 42 CCN(Cc1ccccn1)C(=O)Nc1cncc(OC)c1 ZINC000880557161 CF On-Demand Anodyne ROCK2 21 45 COc1cncc(NC(=O)NCc2ccc(OC)cc2C)c1 ZINC000880557162 DF On-Demand Anodyne P2RX7 21 46 COc1cncc(NC(=O)NCc2ccc(OC)cc2C)c1 ZINC000880557162 DF On-Demand Anodyne MTNR1A 44 34 COc1cncc(NC(=O)NCc2ccc(OC)cc2C)c1 ZINC000880557162 DF On-Demand Anodyne MTNR1B 35 41 COc1cncc(NC(=O)NCc2ccc(OC)cc2C)c1 ZINC000880557162 DF On-Demand Anodyne ROCK2 20 50 COc1cncc(NC(=O)N2CCN(c3cc(F)ccc3F)CC2)c1 ZINC000880557174 EF On-Demand Anodyne HTR1B 17 48 COc1cncc(NC(=O)N2CCN(c3cc(F)ccc3F)CC2)c1 ZINC000880557174 EF On-Demand Anodyne PDGFRB 52 42 COc1cncc(NC(=O)N2CCN(c3cc(F)ccc3F)CC2)c1 ZINC000880557174 EF On-Demand Anodyne FAAH 19 41 COc1cncc(NC(=O)N2CCN(c3cc(F)ccc3F)CC2)c1 ZINC000880557174 EF On-Demand Anodyne RBP4 15 42 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne DRD2 20 43 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne DRD4 53 43 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne ACHE 43 44 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne DRD3 18 43 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne OPRK1 16 41 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne LTA4H 32 49 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne SIGMAR1 48 47 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne CCR3 49 42 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne CCR5 29 49 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne SLC18A3 22 42 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne MLNR 47 38 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne FAAH 22 42 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne ALOX15 15 43 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne MCHR1 55 46 COc1cncc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557182 EF On-Demand Anodyne CCR8 25 40 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne DRD2 20 43 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne DRD4 53 43 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne ACHE 43 44 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne DRD3 18 43 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne OPRK1 16 41 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne LTA4H 32 49 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne SIGMAR1 48 47 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne CCR3 49 42 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne CCR5 29 49 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne SLC18A3 22 42 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne MLNR 47 38 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne FAAH 22 42 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne ALOX15 15 43 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne MCHR1 55 46 COc1cncc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880557183 EF On-Demand Anodyne CCR8 25 40 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne DRD2 16 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne DRD4 42 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne ACHE 34 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne SIGMAR1 39 49 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne SSTR5 43 36 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne CCR3 87 49 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne SLC18A3 17 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne MCHR1 37 48 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557188 FE On-Demand Anodyne CCR8 18 40 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne DRD2 16 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne DRD4 42 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne ACHE 34 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne SIGMAR1 39 49 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne SSTR5 43 36 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne CCR3 87 49 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne SLC18A3 17 42 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne MCHR1 37 48 COc1cncc(NC(=O)N[C@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557189 FE On-Demand Anodyne CCR8 18 40 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne DRD2 16 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne DRD4 42 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne ACHE 34 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne SIGMAR1 39 49 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne SSTR5 43 36 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne CCR3 87 49 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne SLC18A3 17 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne MCHR1 37 48 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@H]2CO)c1 ZINC000880557190 FE On-Demand Anodyne CCR8 18 40 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne DRD2 16 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne DRD4 42 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne ACHE 34 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne DRD3 15 46 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne SIGMAR1 39 49 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne SSTR5 43 36 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne CCR3 87 49 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne CHRNA7 22 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne SLC18A3 17 42 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne MCHR1 37 48 COc1cncc(NC(=O)N[C@@H]2CN(Cc3ccccc3)CC[C@@H]2CO)c1 ZINC000880557191 FE On-Demand Anodyne CCR8 18 40 COc1cncc(NC(=O)N2CCN(C(C)=O)C[C@@H]2C)c1 ZINC000880557200 CD On-Demand Anodyne LIMK2 24 42 COc1cncc(NC(=O)N2CCN(C(C)=O)C[C@H]2C)c1 ZINC000880557201 CD On-Demand Anodyne LIMK2 24 42 COc1cncc(NC(=O)N(C)Cc2cccc(N(C)C)c2)c1 ZINC000880557202 DF On-Demand Anodyne ROCK1 21 53 COc1cncc(NC(=O)N(C)Cc2cccc(N(C)C)c2)c1 ZINC000880557202 DF On-Demand Anodyne ROCK2 37 53 COc1cncc(NC(=O)N(C)CC2CCN(C[C@H](O)c3ccccc3)CC2)c1 ZINC000880557215 GF On-Demand Anodyne OPRK1 31 43 COc1cncc(NC(=O)N(C)CC2CCN(C[C@H](O)c3ccccc3)CC2)c1 ZINC000880557215 GF On-Demand Anodyne CCR3 31 47 COc1cncc(NC(=O)N(C)CC2CCN(C[C@@H](O)c3ccccc3)CC2)c1 ZINC000880557216 GF On-Demand Anodyne OPRK1 31 43 COc1cncc(NC(=O)N(C)CC2CCN(C[C@@H](O)c3ccccc3)CC2)c1 ZINC000880557216 GF On-Demand Anodyne CCR3 31 47 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557226 EH On-Demand Anodyne DRD4 34 41 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557226 EH On-Demand Anodyne SIGMAR1 34 40 CC(=O)Oc1ccc(CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557226 EH On-Demand Anodyne NOD2 41 37 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NNC(=O)c1ccccc1Cl ZINC000880557230 GF On-Demand Reactive AVPR2 43 36 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne HRH2 24 46 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne KIT 20 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne RAF1 24 51 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne KDR 35 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne MTNR1A 27 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne MTNR1B 32 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne EPHX2 24 45 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne PDGFRA 32 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne CSF1R 20 41 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne TEK 21 42 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne LIMK1 19 41 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne BRAF 15 44 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne TAAR1 32 44 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne RIPK1 25 45 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne KCNK3 48 41 COCCCOc1cccc(NC(=O)Nc2cncc(OC)c2)c1 ZINC000880557236 EG On-Demand Anodyne KCNK9 46 38 COc1cncc(NC(=O)N2Cc3ccccc3C[C@H]2C)c1 ZINC000880557246 CG On-Demand Anodyne CFTR 66 41 COc1cncc(NC(=O)N2Cc3ccccc3C[C@@H]2C)c1 ZINC000880557247 CG On-Demand Anodyne CFTR 66 41 O=C(COc1cccnc1)NCc1cn(C2CCC2)nn1 ZINC000880557257 CD On-Demand Anodyne VCP 56 33 O=C(COc1cccnc1)NCc1cn(C2CCC2)nn1 ZINC000880557257 CD On-Demand Anodyne NAMPT 32 41 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne ADRB1 15 40 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne CCR3 23 40 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne MTNR1A 24 44 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne MTNR1B 24 44 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne GRIA1 48 33 COc1cncc(NC(=O)NCCCc2ccc(O)cc2)c1 ZINC000880557258 DF On-Demand Anodyne SLC6A5 18 44 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC1CC1 ZINC000880557290 CD On-Demand Anodyne DRD4 15 41 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NC1CC1 ZINC000880557290 CD On-Demand Anodyne SIGMAR1 16 40 COCCCNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557295 DD On-Demand Anodyne DRD4 23 44 COCCCNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557295 DD On-Demand Anodyne DRD3 43 46 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)C(=O)C2)c1 ZINC000880557302 FE On-Demand Anodyne CCR3 24 40 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)C(=O)C2)c1 ZINC000880557302 FE On-Demand Anodyne FAAH 21 44 COc1cncc(NC(=O)N2CCN(Cc3cccc(F)c3)C(=O)C2)c1 ZINC000880557302 FE On-Demand Anodyne P2RY14 47 37 CCN(Cc1ccccc1)C(=O)[C@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880557333 ED On-Demand Anodyne SLC12A5 59 37 CCN(Cc1ccccc1)C(=O)[C@@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880557334 ED On-Demand Anodyne SLC12A5 59 37 CCN(Cc1ccccc1)C(=O)[C@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880557335 ED On-Demand Anodyne SLC12A5 59 37 CCN(Cc1ccccc1)C(=O)[C@@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880557336 ED On-Demand Anodyne SLC12A5 59 37 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)N1CCCCCC1 ZINC000880557339 EF On-Demand Anodyne PREP 53 39 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne GRIN2B 58 39 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne CCR3 67 45 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne EPHX2 37 51 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne CACNA1I 55 35 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne L3MBTL3 49 33 COc1cncc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880557348 FF On-Demand Anodyne NAMPT 24 43 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCc3ccccc3C2)C1 ZINC000880557350 DC On-Demand Anodyne NOD2 41 36 COc1cncc(NC(=O)N2CCC(Nc3cccc(C)c3)CC2)c1 ZINC000880557351 EH On-Demand Anodyne PTPN2 61 35 COc1cncc(NC(=O)N2CCC(Nc3cccc(C)c3)CC2)c1 ZINC000880557351 EH On-Demand Anodyne PTPN1 50 35 COc1cncc(NC(=O)N2CCC(Nc3cccc(C)c3)CC2)c1 ZINC000880557351 EH On-Demand Anodyne EPHX2 18 44 COc1cncc(NC(=O)N2CCCN(C3CCCC3)CC2)c1 ZINC000880557357 DF On-Demand Anodyne L3MBTL3 46 33 CCOC[C@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880557385 EC On-Demand Anodyne ACOX1 49 33 CCOC[C@H](O)CN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880557385 EC On-Demand Anodyne ABCB1 28 42 O=C(CN1Cc2ccccc2N2CCC[C@H]2C1)NCCCN1CCCCCC1=O ZINC000880557387 GE On-Demand Anodyne TYRO3 18 41 COc1cncc(NC(=O)NCCc2cccc(C(=O)N(C)C)c2)c1 ZINC000880557393 EE On-Demand Anodyne ROCK2 34 44 O=C(CNc1cccc(C(F)(F)F)c1)NCc1cn(C2CCC2)nn1 ZINC000880557398 FF On-Demand Anodyne CCR2 99 39 COc1cncc(NC(=O)N[C@H](C)CCSC)c1 ZINC000880557399 CE On-Demand Anodyne FPR1 28 41 COc1cncc(NC(=O)N[C@@H](C)CCSC)c1 ZINC000880557400 CE On-Demand Anodyne FPR1 28 41 O[C@H](CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccc(F)cc1 ZINC000880557403 EG On-Demand Anodyne SLC6A3 31 45 O[C@H](CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccc(F)cc1 ZINC000880557403 EG On-Demand Anodyne SLC18A3 15 40 O[C@@H](CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccc(F)cc1 ZINC000880557404 EG On-Demand Anodyne SLC6A3 31 45 O[C@@H](CN1Cc2ccccc2N2CCC[C@H]2C1)c1ccc(F)cc1 ZINC000880557404 EG On-Demand Anodyne SLC18A3 15 40 CCNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557405 CD On-Demand Anodyne DRD4 20 40 CCNC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557405 CD On-Demand Anodyne TPP2 41 37 CC[C@H](C)NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557411 DE On-Demand Anodyne TPP2 40 33 CC[C@H](C)NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557411 DE On-Demand Anodyne BIRC2 68 34 CCC(CC)[C@@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557416 JH On-Demand Anodyne OPRD1 63 38 CCC(CC)[C@@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557416 JH On-Demand Anodyne CFTR 75 42 CCC(CC)[C@@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557416 JH On-Demand Anodyne ADAM9 56 36 CCC(CC)[C@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557417 JH On-Demand Anodyne OPRD1 63 38 CCC(CC)[C@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557417 JH On-Demand Anodyne CFTR 75 42 CCC(CC)[C@H](CNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1)N1CCOCC1 ZINC000880557417 JH On-Demand Anodyne ADAM9 56 36 COc1cncc(NC(=O)N2CCC(O)(c3cccc(C)c3C)CC2)c1 ZINC000880557418 FG On-Demand Anodyne NPY5R 30 40 COc1cncc(NC(=O)N(CCC#N)CCN2CCOCC2)c1 ZINC000880557430 ED On-Demand Mild DRD4 40 31 COc1cncc(NC(=O)N(CCC#N)CCN2CCOCC2)c1 ZINC000880557430 ED On-Demand Mild CASR 63 54 COc1cncc(NC(=O)N(CCC#N)CCN2CCOCC2)c1 ZINC000880557430 ED On-Demand Mild MAP2K1 18 41 O[C@H](COc1ccccc1)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557438 EF On-Demand Anodyne ABCB1 65 42 O[C@@H](COc1ccccc1)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557462 EF On-Demand Anodyne ABCB1 65 42 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557465 EG On-Demand Anodyne GRIN2B 62 41 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557465 EG On-Demand Anodyne CCR3 164 45 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557465 EG On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N2CC[C@@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557465 EG On-Demand Anodyne CYP2D6 28 40 COc1cncc(NC(=O)N2CC[C@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557466 EG On-Demand Anodyne GRIN2B 62 41 COc1cncc(NC(=O)N2CC[C@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557466 EG On-Demand Anodyne CCR3 164 45 COc1cncc(NC(=O)N2CC[C@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557466 EG On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)N2CC[C@H](Cc3ccc(F)cc3)C2)c1 ZINC000880557466 EG On-Demand Anodyne CYP2D6 28 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc3ccccc3c2)C1 ZINC000880557469 FD On-Demand Anodyne ACOX1 22 47 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc3ccccc3c2)C1 ZINC000880557470 FD On-Demand Anodyne ACOX1 22 47 COc1cncc(NC(=O)NCC2(N(C)C)Cc3ccccc3C2)c1 ZINC000880557473 EE On-Demand Anodyne ROCK2 28 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(-c2ncon2)cc1 ZINC000880557474 DD On-Demand Anodyne CA14 17 47 CC(=O)Nc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880557476 GG On-Demand Anodyne DRD4 19 44 CC(=O)Nc1cccc(NC(=O)CN2Cc3ccccc3N3CCC[C@H]3C2)c1 ZINC000880557476 GG On-Demand Anodyne CCKBR 31 43 COc1cncc(NC(=O)N2CCc3c(Cl)cccc3C2)c1 ZINC000880557478 DG On-Demand Anodyne DRD4 45 37 COc1cncc(NC(=O)N2CCc3c(Cl)cccc3C2)c1 ZINC000880557478 DG On-Demand Anodyne CPT2 15 42 COc1cncc(NC(=O)N2CCc3c(Cl)cccc3C2)c1 ZINC000880557478 DG On-Demand Anodyne TAAR1 28 42 COc1cncc(NC(=O)N2CCc3c(Cl)cccc3C2)c1 ZINC000880557478 DG On-Demand Anodyne P2RY14 49 40 COc1cncc(NC(=O)N2CCCC[C@H]2CN2CCOCC2)c1 ZINC000880557479 ED On-Demand Anodyne CASR 20 41 COc1cncc(NC(=O)N2CCCC[C@@H]2CN2CCOCC2)c1 ZINC000880557480 ED On-Demand Anodyne CASR 20 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne DRD4 36 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne ACHE 27 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne SIGMAR1 34 48 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne CCR3 80 51 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557484 FE On-Demand Anodyne MCHR1 30 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne DRD4 36 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne ACHE 27 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne SIGMAR1 34 48 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne CCR3 80 51 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557485 FE On-Demand Anodyne MCHR1 30 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne DRD4 36 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne ACHE 27 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne SIGMAR1 34 48 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne CCR3 80 51 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@H]2CO)c1 ZINC000880557486 FE On-Demand Anodyne MCHR1 30 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne DRD4 36 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne ACHE 27 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne SIGMAR1 34 48 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne CCR3 80 51 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C[C@@H]2CO)c1 ZINC000880557487 FE On-Demand Anodyne MCHR1 30 45 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne CTSD 27 45 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne PGA 21 45 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne ECE1 41 43 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne REN 47 42 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne CTSE 18 45 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne PGA5 25 40 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557517 FF On-Demand Anodyne FPR1 42 34 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne CTSD 27 45 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne PGA 21 45 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne ECE1 41 43 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne REN 47 42 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne CTSE 18 45 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne PGA5 25 40 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880557518 FF On-Demand Anodyne FPR1 42 34 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557524 GF On-Demand Anodyne ADRB2 16 45 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557524 GF On-Demand Anodyne ADRB1 45 45 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557524 GF On-Demand Anodyne ACOX1 55 39 CC(=O)Nc1ccc(OC[C@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557524 GF On-Demand Anodyne ABCB1 63 42 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557525 GF On-Demand Anodyne ADRB2 16 45 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557525 GF On-Demand Anodyne ADRB1 45 45 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557525 GF On-Demand Anodyne ACOX1 55 39 CC(=O)Nc1ccc(OC[C@@H](O)CN2Cc3ccccc3N3CCC[C@H]3C2)cc1 ZINC000880557525 GF On-Demand Anodyne ABCB1 63 42 CCCn1cc(CN2CCCN(C(=O)Nc3cncc(OC)c3)CC2)cn1 ZINC000880557531 FE On-Demand Anodyne FAAH 18 45 CC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557537 CE On-Demand Anodyne SLC6A1 48 33 CC(=O)CCN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557537 CE On-Demand Anodyne HTR7 30 41 COc1cncc(NC(=O)NCCCCn2ccnc2C)c1 ZINC000880557545 DE On-Demand Anodyne QPCT 53 45 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557546 ED On-Demand Anodyne OPRL1 17 42 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557546 ED On-Demand Anodyne XIAP 41 33 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557546 ED On-Demand Anodyne BIRC3 44 32 C[C@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557546 ED On-Demand Anodyne BIRC2 90 38 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557547 ED On-Demand Anodyne OPRL1 17 42 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557547 ED On-Demand Anodyne XIAP 41 33 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557547 ED On-Demand Anodyne BIRC3 44 32 C[C@@H](NC(=O)CN1Cc2ccccc2N2CCC[C@H]2C1)C(=O)N(C)C ZINC000880557547 ED On-Demand Anodyne BIRC2 90 38 COc1cncc(NC(=O)N2CCN(CC3CCOCC3)CC2)c1 ZINC000880557554 ED On-Demand Anodyne PDGFRB 46 36 C[C@@H]1CCCCN1C(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557566 EF On-Demand Anodyne PREP 48 41 C[C@H]1CCCCN1C(=O)CN1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880557567 EF On-Demand Anodyne PREP 48 41 COc1cncc(NC(=O)Nc2ccc(CN(C(C)=O)C(C)C)cc2)c1 ZINC000880557569 FG On-Demand Anodyne ROCK2 21 46 COc1cncc(NC(=O)N2CCC(CC(=O)N3CCN(C)CC3)CC2)c1 ZINC000880557571 GD On-Demand Anodyne PDGFRB 43 35 COC(=O)[C@@]1(O)CCN(Cc2ccccc2Cl)C1 ZINC000880557609 CD On-Demand Anodyne SIGMAR1 17 43 CCOc1ccc(-c2nc(CN3CC[C@@](O)(C(=O)OC)C3)cs2)cc1OC ZINC000880557617 GE On-Demand Anodyne PPARD 18 43 CCOc1ccc(-c2nc(CN3CC[C@](O)(C(=O)OC)C3)cs2)cc1OC ZINC000880557619 GE On-Demand Anodyne PPARD 18 43 COc1cncc(NC(=O)N(C)Cc2ccon2)c1 ZINC000880557621 CD On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3OC)C2)c1 ZINC000880557622 EG On-Demand Anodyne DRD4 15 42 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3OC)C2)c1 ZINC000880557622 EG On-Demand Anodyne CCR3 15 42 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3OC)C2)c1 ZINC000880557622 EG On-Demand Anodyne RBP4 64 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2F)C1 ZINC000880557623 DC On-Demand Anodyne BDKRB1 17 40 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3OC)C2)c1 ZINC000880557625 EG On-Demand Anodyne DRD4 15 42 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3OC)C2)c1 ZINC000880557625 EG On-Demand Anodyne CCR3 15 42 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3OC)C2)c1 ZINC000880557625 EG On-Demand Anodyne RBP4 64 43 COc1cncc(NC(=O)NCc2cc(C)[nH]n2)c1 ZINC000880557632 CD On-Demand Anodyne ROCK2 20 44 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2F)c1 ZINC000880557635 DF On-Demand Anodyne ADRB1 40 31 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2F)c1 ZINC000880557635 DF On-Demand Anodyne MTNR1B 17 42 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2F)c1 ZINC000880557637 DF On-Demand Anodyne ADRB1 40 31 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2F)c1 ZINC000880557637 DF On-Demand Anodyne MTNR1B 17 42 COc1cncc(NC(=O)N2CCC(OCCc3ccccc3)CC2)c1 ZINC000880557647 FG On-Demand Anodyne CCR3 19 43 COc1cncc(NC(=O)N2CCC(OCCc3ccccc3)CC2)c1 ZINC000880557647 FG On-Demand Anodyne CHRNA7 36 41 COc1cncc(NC(=O)N2CCC(OCCc3ccccc3)CC2)c1 ZINC000880557647 FG On-Demand Anodyne TIMP3 42 33 COc1cncc(NC(=O)N2CCC(OCCc3ccccc3)CC2)c1 ZINC000880557647 FG On-Demand Anodyne FAAH 20 44 COc1cncc(NC(=O)N2CCC(OCCc3ccccc3)CC2)c1 ZINC000880557647 FG On-Demand Anodyne SCD1 15 44 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccccc3)no2)C1 ZINC000880557658 DC On-Demand Anodyne NPPA 20 43 COc1cncc(NC(=O)N(CCCN2CCOCC2)Cc2ccncc2)c1 ZINC000880557668 GE On-Demand Anodyne CASR 56 50 COc1cncc(NC(=O)N(CCCN2CCOCC2)Cc2ccncc2)c1 ZINC000880557668 GE On-Demand Anodyne EPHX2 23 41 COc1cncc(NC(=O)NC2C[C@@H]3CCC[C@H](C2)N3C)c1 ZINC000880557671 DE On-Demand Anodyne HTR3A 34 45 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne CA2 16 47 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne RAF1 38 49 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne KDR 37 42 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne MTNR1B 19 41 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne EPHX2 17 50 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne CA12 27 47 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne PDGFRA 58 42 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne CA9 27 47 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne MTCA1 29 47 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)cc1 ZINC000880557689 DF On-Demand Anodyne P96878_MYCTU 38 47 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2)c1 ZINC000880557698 DF On-Demand Anodyne MTNR1A 32 51 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2)c1 ZINC000880557698 DF On-Demand Anodyne MTNR1B 34 51 COc1cncc(NC(=O)NC[C@@H](C)Oc2ccccc2)c1 ZINC000880557698 DF On-Demand Anodyne ROCK2 18 40 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2)c1 ZINC000880557699 DF On-Demand Anodyne MTNR1A 32 51 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2)c1 ZINC000880557699 DF On-Demand Anodyne MTNR1B 34 51 COc1cncc(NC(=O)NC[C@H](C)Oc2ccccc2)c1 ZINC000880557699 DF On-Demand Anodyne ROCK2 18 40 COC(=O)[C@@]1(O)CCN(Cc2c(Cl)cccc2Cl)C1 ZINC000880557705 DE On-Demand Anodyne OPRL1 17 40 CCOc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557713 EC On-Demand Anodyne ACOX1 55 33 CCOc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557713 EC On-Demand Anodyne CCR1 41 37 CCOc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557713 EC On-Demand Anodyne ABCB1 56 43 CCOc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557714 EC On-Demand Anodyne ACOX1 55 33 CCOc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557714 EC On-Demand Anodyne CCR1 41 37 CCOc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557714 EC On-Demand Anodyne ABCB1 56 43 CCOc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557715 EC On-Demand Anodyne ACOX1 55 33 CCOc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557715 EC On-Demand Anodyne CCR1 41 37 CCOc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880557715 EC On-Demand Anodyne ABCB1 56 43 CCOc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557716 EC On-Demand Anodyne ACOX1 55 33 CCOc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557716 EC On-Demand Anodyne CCR1 41 37 CCOc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880557716 EC On-Demand Anodyne ABCB1 56 43 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000880557721 FC On-Demand Anodyne ACOX1 66 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000880557721 FC On-Demand Anodyne CCR1 41 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Br)cc2)C1 ZINC000880557721 FC On-Demand Anodyne ABCB1 47 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Br)cc2)C1 ZINC000880557722 FC On-Demand Anodyne ACOX1 66 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Br)cc2)C1 ZINC000880557722 FC On-Demand Anodyne CCR1 41 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Br)cc2)C1 ZINC000880557722 FC On-Demand Anodyne ABCB1 47 40 COc1cncc(NC(=O)N(CCO)Cc2cnn(Cc3ccccc3)c2)c1 ZINC000880557727 GE On-Demand Anodyne ROCK2 22 47 COc1cncc(NC(=O)NCCN2CCSCC2)c1 ZINC000880557733 CD On-Demand Anodyne DRD4 47 36 COc1cncc(NC(=O)NCCN2CCSCC2)c1 ZINC000880557733 CD On-Demand Anodyne CCR3 30 43 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OC)C1 ZINC000880557749 CD On-Demand Anodyne DRD4 15 45 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OC)C1 ZINC000880557749 CD On-Demand Anodyne CPT1A 51 43 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OC)C1 ZINC000880557749 CD On-Demand Anodyne CPT1B 52 36 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OC)C1 ZINC000880557749 CD On-Demand Anodyne CCR8 19 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557753 EC On-Demand Anodyne ACOX1 54 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557753 EC On-Demand Anodyne CCR1 41 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557753 EC On-Demand Anodyne ABCB1 50 43 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557754 EC On-Demand Anodyne ACOX1 54 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557754 EC On-Demand Anodyne CCR1 41 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)=O)cc2)C1 ZINC000880557754 EC On-Demand Anodyne ABCB1 50 43 COc1cncc(NC(=O)NCc2cc(C(C)C)no2)c1 ZINC000880557757 CF On-Demand Anodyne SLC5A7 24 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3cccc(Cl)c3)CC2)C1 ZINC000880557771 GC On-Demand Anodyne HTR1A 23 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3cccc(Cl)c3)CC2)C1 ZINC000880557771 GC On-Demand Anodyne DRD4 41 35 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3cccc(Cl)c3)CC2)C1 ZINC000880557771 GC On-Demand Anodyne HTR2A 16 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3cccc(Cl)c3)CC2)C1 ZINC000880557771 GC On-Demand Anodyne MAPK1 21 49 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(Br)c2)C1 ZINC000880557774 ED On-Demand Anodyne MMP13 17 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(Br)c2)C1 ZINC000880557774 ED On-Demand Anodyne MCHR2 44 34 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccs3)no2)C1 ZINC000880557803 DC On-Demand Anodyne ETHR 32 43 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne DRD4 23 45 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne SIGMAR1 35 46 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne MMP13 20 56 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne CCR3 30 42 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne NPFFR2 29 45 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne ADAM17 21 56 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne FAAH 16 46 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne MMP9 17 56 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne MCHR1 19 56 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne MCHR2 74 38 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne NPFFR1 41 45 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3c2)C1 ZINC000880557810 CD On-Demand Anodyne SLC12A5 42 35 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)c(OC)c2)C1 ZINC000880557823 FB On-Demand Anodyne MT-ND1 18 40 COC(=O)[C@@]1(O)CCN(CC(=O)NC2C3CC4CC(C3)CC2C4)C1 ZINC000880557826 EC On-Demand Anodyne HSD11B1 44 37 COC(=O)[C@@]1(O)CCN(Cc2cccc3ccccc23)C1 ZINC000880557901 CD On-Demand Anodyne SIGMAR1 15 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2c(C)cccc2C(C)C)C1 ZINC000880557904 ED On-Demand Anodyne SOAT1 45 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)C(F)F)cc2)C1 ZINC000880557911 EC On-Demand Anodyne MMP13 27 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)C(F)F)cc2)C1 ZINC000880557911 EC On-Demand Anodyne ADAM17 26 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)C(F)F)cc2)C1 ZINC000880557911 EC On-Demand Anodyne MMP9 22 44 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc3cc(OC)ccc3c2)C1 ZINC000880557913 GD On-Demand Anodyne MMP13 15 40 COc1cncc(NC(=O)Nc2cc(OC)c(OC)cc2C)c1 ZINC000880557914 DG On-Demand Anodyne PDGFRA 45 40 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(C)=O)C1 ZINC000880557918 DC On-Demand Anodyne SLC12A5 46 34 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(C)=O)C1 ZINC000880557918 DC On-Demand Anodyne HCN1 76 36 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(C)=O)C1 ZINC000880557918 DC On-Demand Anodyne HCN4 52 35 COc1cncc(NC(=O)NCCCC(=O)N2Cc3ccccc3C2)c1 ZINC000880557923 FF On-Demand Anodyne HRH2 15 40 COc1cncc(NC(=O)NCCCC(=O)N2Cc3ccccc3C2)c1 ZINC000880557923 FF On-Demand Anodyne CCR3 18 42 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)c(C)c1 ZINC000880557924 EG On-Demand Anodyne KDR 23 43 COCCOc1ccc(NC(=O)Nc2cncc(OC)c2)c(C)c1 ZINC000880557924 EG On-Demand Anodyne PDGFRA 41 38 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2Cl)C1 ZINC000880557926 ED On-Demand Anodyne HTR4 24 41 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)[C@H](C)c2ccccc2)C1 ZINC000880557931 DC On-Demand Anodyne OPRK1 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)[C@@H](C)c2ccccc2)C1 ZINC000880557934 DC On-Demand Anodyne OPRK1 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCCc3ccccc32)C1 ZINC000880557945 DC On-Demand Anodyne DRD4 16 51 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCCc3ccccc32)C1 ZINC000880557945 DC On-Demand Anodyne AVPR2 40 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne DRD4 16 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne CHRM3 16 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne SIGMAR1 30 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne MCHR2 52 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne CACNA1G 28 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(F)c2)C1 ZINC000880557952 CC On-Demand Anodyne SLC12A5 56 36 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCCC[C@H]3C)C2)c1 ZINC000880557956 EG On-Demand Anodyne PDGFRB 17 40 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCCC[C@@H]3C)C2)c1 ZINC000880557957 EG On-Demand Anodyne PDGFRB 17 40 COc1cncc(NC(=O)N2CCC[C@H](CN3CCCC[C@H]3C)C2)c1 ZINC000880557958 EG On-Demand Anodyne PDGFRB 17 40 COc1cncc(NC(=O)N2CCC[C@H](CN3CCCC[C@@H]3C)C2)c1 ZINC000880557959 EG On-Demand Anodyne PDGFRB 17 40 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Cl)c2)C1 ZINC000880557962 CD On-Demand Anodyne DRD4 43 34 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Cl)c2)C1 ZINC000880557962 CD On-Demand Anodyne LTA4H 33 42 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Cl)c2)C1 ZINC000880557962 CD On-Demand Anodyne HRH3 19 47 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Cl)c2)C1 ZINC000880557962 CD On-Demand Anodyne MMP13 16 43 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)c1 ZINC000880557963 ED On-Demand Anodyne CCR3 25 42 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)c1 ZINC000880557963 ED On-Demand Anodyne PDK1 47 35 COc1cncc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)c1 ZINC000880557963 ED On-Demand Anodyne CXCR3 19 43 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)c1 ZINC000880557964 ED On-Demand Anodyne CCR3 25 42 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)c1 ZINC000880557964 ED On-Demand Anodyne PDK1 47 35 COc1cncc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)c1 ZINC000880557964 ED On-Demand Anodyne CXCR3 19 43 COc1cncc(NC(=O)N2CCC(C(N)=O)(c3ccccc3)CC2)c1 ZINC000880557974 FE On-Demand Anodyne TACR2 18 45 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557979 GD On-Demand Anodyne MMP13 16 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557979 GD On-Demand Anodyne P2RY1 67 48 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557979 GD On-Demand Anodyne MMP2 19 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557979 GD On-Demand Anodyne MMP9 17 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557979 GD On-Demand Anodyne EPHX2 65 46 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557980 GD On-Demand Anodyne MMP13 16 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557980 GD On-Demand Anodyne P2RY1 67 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557980 GD On-Demand Anodyne MMP2 19 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557980 GD On-Demand Anodyne MMP9 17 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880557980 GD On-Demand Anodyne EPHX2 65 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne ACHE 20 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne DRD3 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne LTA4H 23 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne SIGMAR1 40 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne ADAM17 15 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne CPT1A 46 32 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne PRNP 56 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne HDAC1 18 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne MCHR1 20 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne NPFFR1 45 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne NOD1 22 51 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne NOD2 58 51 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)Nc3ccccc3)cc2)C1 ZINC000880558002 FE On-Demand Anodyne KCNK3 60 36 COc1cncc(NC(=O)NCCCC(=O)N2CCc3ccccc32)c1 ZINC000880558003 FF On-Demand Anodyne DRD4 41 34 COc1cncc(NC(=O)NCCCC(=O)N2CCc3ccccc32)c1 ZINC000880558003 FF On-Demand Anodyne AVPR2 29 41 COc1cncc(NC(=O)NCCCC(=O)N2CCc3ccccc32)c1 ZINC000880558003 FF On-Demand Anodyne CCR3 16 41 CCOc1ccnc(N2CCN(C(=O)Nc3cncc(OC)c3)CC2)n1 ZINC000880558004 FD On-Demand Anodyne PDGFRB 54 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne DRD4 45 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne MMP13 27 45 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne ROCK1 37 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne MTNR1A 54 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne MTNR1B 53 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OC)c2)C1 ZINC000880558009 DB On-Demand Anodyne ROCK2 42 41 COc1cncc(NC(=O)N(CCO)Cc2ccc(OC)cc2OC)c1 ZINC000880558010 FE On-Demand Anodyne ROCK2 22 46 COc1cncc(NC(=O)N2CCN(C[C@@H](C)O)CC2)c1 ZINC000880558016 CC On-Demand Anodyne PDGFRB 45 37 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(C)C)cc2)C1 ZINC000880558018 CD On-Demand Anodyne MMP13 15 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(C#N)c2)C1 ZINC000880558043 CC On-Demand Mild SIGMAR1 17 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(C#N)c2)C1 ZINC000880558043 CC On-Demand Mild CCR3 15 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(C#N)c2)C1 ZINC000880558043 CC On-Demand Mild MCHR1 31 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C#N)c2)C1 ZINC000880558043 CC On-Demand Mild SLC12A5 44 47 COc1cncc(NC(=O)NCc2ccc(F)c(CN(C)C)c2)c1 ZINC000880558048 EF On-Demand Anodyne ROCK2 31 44 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3ccc(OC)cc3)CC2)C1 ZINC000880558050 GB On-Demand Clean MMP13 15 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne ESR1 42 38 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne PPARG 17 46 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne LTA4H 56 40 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne MMP13 21 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne ADAM17 28 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne MMP9 17 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc3ccccc3c2)C1 ZINC000880558057 DD On-Demand Anodyne PSMB1 42 37 COc1cncc(NC(=O)N2CCN([C@H](CO)c3ccc(Cl)cc3)CC2)c1 ZINC000880558059 GF On-Demand Anodyne FAAH 18 42 COc1cncc(NC(=O)N2CCN([C@@H](CO)c3ccc(Cl)cc3)CC2)c1 ZINC000880558060 GF On-Demand Anodyne FAAH 18 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(C)(C)C)cc2)C1 ZINC000880558062 CE On-Demand Anodyne MMP13 15 41 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Br)cc2)C1 ZINC000880558064 GC On-Demand Anodyne MMP13 35 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Br)cc2)C1 ZINC000880558064 GC On-Demand Anodyne ADAM17 38 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Br)cc2)C1 ZINC000880558064 GC On-Demand Anodyne MMP9 24 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Br)cc2)C1 ZINC000880558064 GC On-Demand Anodyne MMP1 15 44 COc1cncc(NC(=O)N[C@H]2CCCN(c3ccccc3)C2=O)c1 ZINC000880558065 EE On-Demand Anodyne CCKAR 36 44 COc1cncc(NC(=O)N[C@H]2CCCN(c3ccccc3)C2=O)c1 ZINC000880558065 EE On-Demand Anodyne CCKBR 45 40 COc1cncc(NC(=O)N[C@@H]2CCCN(c3ccccc3)C2=O)c1 ZINC000880558066 EE On-Demand Anodyne CCKAR 36 44 COc1cncc(NC(=O)N[C@@H]2CCCN(c3ccccc3)C2=O)c1 ZINC000880558066 EE On-Demand Anodyne CCKBR 45 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)c(F)c2)C1 ZINC000880558069 CD On-Demand Anodyne MCHR2 69 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc(Cl)cc2)C1 ZINC000880558081 ED On-Demand Anodyne CCR1 61 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc(Cl)cc2)C1 ZINC000880558083 ED On-Demand Anodyne CCR1 61 36 COc1cncc(NC(=O)N(C)[C@H](C)CS(C)(=O)=O)c1 ZINC000880558091 DC On-Demand Anodyne NPY5R 30 41 COc1cncc(NC(=O)N(C)[C@@H](C)CS(C)(=O)=O)c1 ZINC000880558092 DC On-Demand Anodyne NPY5R 30 41 COc1cncc(NC(=O)NC[C@H](O)c2ccccc2OC)c1 ZINC000880558103 DD On-Demand Anodyne ADRB1 42 32 COc1cncc(NC(=O)NC[C@H](O)c2ccccc2OC)c1 ZINC000880558103 DD On-Demand Anodyne MTNR1A 17 43 COc1cncc(NC(=O)NC[C@H](O)c2ccccc2OC)c1 ZINC000880558103 DD On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)NC[C@H](O)c2ccccc2OC)c1 ZINC000880558103 DD On-Demand Anodyne SOAT1 41 39 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cn2c3ccccc3c3ccccc32)C1 ZINC000880558105 FD On-Demand Anodyne MCHR2 40 34 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cn2c3ccccc3c3ccccc32)C1 ZINC000880558107 FD On-Demand Anodyne MCHR2 40 34 COc1cncc(NC(=O)N(CCO)CCc2ccccc2)c1 ZINC000880558108 DE On-Demand Anodyne BMP1 15 44 COc1cncc(NC(=O)N(CCO)CCc2ccccc2)c1 ZINC000880558108 DE On-Demand Anodyne ROCK2 26 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne TACR2 46 35 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne SIGMAR1 28 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne CCR3 20 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne NPFFR2 19 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne CXCR3 23 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne MCHR2 45 34 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558109 DE On-Demand Anodyne NPFFR1 28 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(Cc3ccccc3)CC2)C1 ZINC000880558138 FD On-Demand Anodyne GRIN2B 90 44 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(Cc3ccccc3)CC2)C1 ZINC000880558138 FD On-Demand Anodyne SIGMAR1 32 50 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(Cc3ccccc3)CC2)C1 ZINC000880558138 FD On-Demand Anodyne CCR3 45 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(Cc3ccccc3)CC2)C1 ZINC000880558138 FD On-Demand Anodyne SLC12A5 42 35 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCc3cc(OC)c(OC)cc3C2)C1 ZINC000880558140 GC On-Demand Anodyne ABCB1B 42 33 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCc3cc(OC)c(OC)cc3C2)C1 ZINC000880558140 GC On-Demand Anodyne ABCB1 19 48 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3C[C@H]2C)C1 ZINC000880558145 DC On-Demand Anodyne DRD4 34 56 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3C[C@H]2C)C1 ZINC000880558145 DC On-Demand Anodyne TPP2 55 32 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3C[C@@H]2C)C1 ZINC000880558146 DC On-Demand Anodyne DRD4 34 56 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3C[C@@H]2C)C1 ZINC000880558146 DC On-Demand Anodyne TPP2 55 32 COCC1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880558168 CD On-Demand Anodyne PDGFRB 44 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2OC)C1 ZINC000880558180 DB On-Demand Anodyne HTR7 19 43 COc1cncc(NC(=O)N(Cc2cccc(O)c2)CC2CC2)c1 ZINC000880558194 EG On-Demand Anodyne ROCK1 18 43 COc1cncc(NC(=O)N(Cc2cccc(O)c2)CC2CC2)c1 ZINC000880558194 EG On-Demand Anodyne ROCK2 29 45 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)cc2)C1 ZINC000880558208 DB On-Demand Anodyne MMP13 29 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)cc2)C1 ZINC000880558208 DB On-Demand Anodyne ADAM17 19 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)cc2)C1 ZINC000880558208 DB On-Demand Anodyne MMP9 23 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)cc2)C1 ZINC000880558208 DB On-Demand Anodyne CA9 18 45 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC)cc2)C1 ZINC000880558208 DB On-Demand Anodyne MMP1 17 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000880558209 ED On-Demand Anodyne HRH3 15 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000880558209 ED On-Demand Anodyne CCR8 27 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000880558209 ED On-Demand Anodyne L3MBTL3 58 46 COc1cncc(NC(=O)Nc2cccc(COC(C)C)c2)c1 ZINC000880558216 DH On-Demand Anodyne ROCK2 37 42 COc1cncc(NC(=O)Nc2cccc(COC(C)C)c2)c1 ZINC000880558216 DH On-Demand Anodyne TAAR1 30 40 COc1cncc(NC(=O)Nc2cccc(COC(C)C)c2)c1 ZINC000880558216 DH On-Demand Anodyne KCNK3 45 37 COc1cncc(NC(=O)NCC2Cc3ccccc3C2)c1 ZINC000880558219 CF On-Demand Anodyne MTNR1A 19 40 COc1cncc(NC(=O)NCC2Cc3ccccc3C2)c1 ZINC000880558219 CF On-Demand Anodyne MTNR1B 21 40 COc1cncc(NC(=O)NCCN(C)CC(F)(F)F)c1 ZINC000880558220 DD On-Demand Anodyne RAF1 16 40 COC(=O)[C@@]1(O)CCN(CCOC(c2ccccc2)c2ccccc2)C1 ZINC000880558226 FE On-Demand Anodyne SLC6A4 25 49 COC(=O)[C@@]1(O)CCN(CCOC(c2ccccc2)c2ccccc2)C1 ZINC000880558226 FE On-Demand Anodyne SLC6A3 69 55 COc1cncc(NC(=O)N2CCN(C3CCC3)CC2)c1 ZINC000880558231 CD On-Demand Anodyne HRH3 32 46 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne INHA 46 34 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne TRPV1 20 47 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne RAF1 28 41 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne MTNR1A 32 51 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne MTNR1B 24 51 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne NCE103 20 46 COc1cncc(NC(=O)NCCc2ccc(O)c(OC)c2)c1 ZINC000880558232 DE On-Demand Anodyne P96878_MYCTU 21 46 COC(=O)[C@@]1(O)CCN(Cc2ncc(-c3ccc(Cl)cc3)o2)C1 ZINC000880558240 EE On-Demand Anodyne NPPA 21 43 COC(=O)[C@@]1(O)CCN(Cc2ccc3oc4ccccc4c3c2)C1 ZINC000880558242 EF On-Demand Anodyne MCHR2 84 42 COc1cncc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c1 ZINC000880558247 ED On-Demand Anodyne MAP2K1 17 40 COc1cncc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c1 ZINC000880558247 ED On-Demand Anodyne EPHX2 27 45 CCCCC[C@@H](C)NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880558248 DC On-Demand Anodyne NOD1 45 32 CCCCC[C@@H](C)NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880558249 DC On-Demand Anodyne NOD1 45 32 O=C(NCc1cn(C2CCC2)nn1)C(=O)c1ccc(Br)cc1 ZINC000880558260 FE On-Demand Anodyne CA14 15 41 COc1cncc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c1 ZINC000880558263 FE On-Demand Anodyne PDGFRB 52 37 COc1cncc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c1 ZINC000880558263 FE On-Demand Anodyne FAAH 33 57 COc1cncc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c1 ZINC000880558263 FE On-Demand Anodyne MCHR1 19 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(C)c2)C1 ZINC000880558272 BD On-Demand Anodyne DRD4 21 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(C)c2)C1 ZINC000880558272 BD On-Demand Anodyne SIGMAR1 26 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C)c2)C1 ZINC000880558272 BD On-Demand Anodyne MCHR2 45 34 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne PDGFRB 34 44 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne SSTR5 40 38 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne ROCK2 31 52 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne FLT4 23 44 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne MT-ND1 23 40 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne ENPP1 40 31 CCOc1cc(CNC(=O)Nc2cncc(OC)c2)ccc1OC ZINC000880558273 EF On-Demand Anodyne DRTS_TRYCR 48 35 CC[C@@H]1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880558274 CG On-Demand Anodyne PDGFRB 46 36 CC[C@H]1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880558275 CG On-Demand Anodyne PDGFRB 46 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne ADRA1D 16 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne ADRA1A 30 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne ADRA1B 20 45 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne SIGMAR1 30 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne MTNR1A 19 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne MTNR1B 20 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne FAAH 15 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne CRTM 33 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCc2ccccc2)C1 ZINC000880558279 DC On-Demand Anodyne SLC12A5 49 38 CCOc1ccc(-c2noc(CN3CC[C@@](O)(C(=O)OC)C3)n2)cc1 ZINC000880558281 ED On-Demand Anodyne MMP13 15 45 CCOc1ccc(-c2noc(CN3CC[C@](O)(C(=O)OC)C3)n2)cc1 ZINC000880558282 ED On-Demand Anodyne MMP13 15 45 COc1cncc(NC(=O)N2CCCN(Cc3cnn(C)c3)CC2)c1 ZINC000880558285 ED On-Demand Anodyne FAAH 20 48 COc1cncc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880558291 FF On-Demand Anodyne F13A1 16 40 COc1cncc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880558291 FF On-Demand Anodyne GPR119 31 41 COc1cncc(NC(=O)N2CCN(c3nc(C)cc(OC)n3)CC2)c1 ZINC000880558310 FD On-Demand Anodyne PDGFRB 43 37 COC(=O)[C@@]1(O)CCN(Cc2ccccc2[N+](=O)[O-])C1 ZINC000880558311 CC On-Demand Bother COLA 111 35 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCSc2ccccc2)C1 ZINC000880558325 FC On-Demand Anodyne ADRA1A 24 41 COc1cncc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c1 ZINC000880558328 FG On-Demand Anodyne HTR1D 22 47 COc1cncc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c1 ZINC000880558328 FG On-Demand Anodyne HTR1B 19 47 COc1cncc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c1 ZINC000880558328 FG On-Demand Anodyne HTR1F 60 38 COc1cncc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c1 ZINC000880558328 FG On-Demand Anodyne CCR2 21 55 COc1cncc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c1 ZINC000880558328 FG On-Demand Anodyne LIMK2 23 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(-n3cccn3)cc2)C1 ZINC000880558331 DC On-Demand Anodyne AMP1_PLAFQ 52 37 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne HCRTR1 16 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne MMP13 27 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne P2RY1 47 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne ADAM17 16 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne MMP2 30 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne MMP14 28 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne MMP9 27 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne EPHX2 47 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne HCRTR2 16 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880558332 DD On-Demand Anodyne NOD2 33 44 CCC[C@H](NC(=O)[C@@H](C)N1CC[C@@](O)(C(=O)OC)C1)c1ccccc1 ZINC000880558334 ED On-Demand Anodyne OPRL1 17 42 CCC[C@H](NC(=O)[C@H](C)N1CC[C@@](O)(C(=O)OC)C1)c1ccccc1 ZINC000880558335 ED On-Demand Anodyne OPRL1 17 42 CCC[C@H](NC(=O)[C@@H](C)N1CC[C@](O)(C(=O)OC)C1)c1ccccc1 ZINC000880558336 ED On-Demand Anodyne OPRL1 17 42 CCC[C@H](NC(=O)[C@H](C)N1CC[C@](O)(C(=O)OC)C1)c1ccccc1 ZINC000880558337 ED On-Demand Anodyne OPRL1 17 42 O=C(Cc1ccc(Cl)cc1Br)NCc1cn(C2CCC2)nn1 ZINC000880558344 GG On-Demand Anodyne P2RX7 42 43 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne LTA4H 48 43 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne MMP13 29 48 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne ADAM17 15 48 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne PLA2G4B 51 33 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne MMP9 18 48 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne PSMB2 41 39 CCCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558347 DD On-Demand Anodyne PSMB1 43 39 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne LTA4H 48 43 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne MMP13 29 48 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne ADAM17 15 48 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne PLA2G4B 51 33 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne MMP9 18 48 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne PSMB2 41 39 CCCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558348 DD On-Demand Anodyne PSMB1 43 39 COCCN(CCO)C(=O)Nc1cncc(OC)c1 ZINC000880558349 CC On-Demand Anodyne ROCK2 15 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)cc2Cl)C1 ZINC000880558350 CD On-Demand Anodyne P2RX7 72 42 COc1cncc(NC(=O)NC[C@H](O)c2ccccc2C)c1 ZINC000880558358 DE On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)NC[C@@H](O)c2ccccc2C)c1 ZINC000880558359 DE On-Demand Anodyne ROCK2 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(C#N)cc2)C1 ZINC000880558361 CC On-Demand Mild MMP13 15 41 COc1cncc(NC(=O)Nc2ccc(OC[C@@H]3CCCO3)cc2)c1 ZINC000880558362 EG On-Demand Anodyne RAF1 25 40 COc1cncc(NC(=O)Nc2ccc(OC[C@@H]3CCCO3)cc2)c1 ZINC000880558362 EG On-Demand Anodyne PDGFRA 48 37 COc1cncc(NC(=O)Nc2ccc(OC[C@H]3CCCO3)cc2)c1 ZINC000880558363 EG On-Demand Anodyne RAF1 25 40 COc1cncc(NC(=O)Nc2ccc(OC[C@H]3CCCO3)cc2)c1 ZINC000880558363 EG On-Demand Anodyne PDGFRA 48 37 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558366 EG On-Demand Mild ROCK1 37 44 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558366 EG On-Demand Mild ROCK2 52 52 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558366 EG On-Demand Mild PDS 40 37 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558367 EG On-Demand Mild ROCK1 37 44 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558367 EG On-Demand Mild ROCK2 52 52 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880558367 EG On-Demand Mild PDS 40 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2)C1 ZINC000880558369 CC On-Demand Anodyne ADRB2 31 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2)C1 ZINC000880558369 CC On-Demand Anodyne ACOX1 54 39 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2)C1 ZINC000880558369 CC On-Demand Anodyne CCR1 40 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2)C1 ZINC000880558369 CC On-Demand Anodyne ABCB1 80 48 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2)C1 ZINC000880558370 CC On-Demand Anodyne ADRB2 31 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2)C1 ZINC000880558370 CC On-Demand Anodyne ACOX1 54 39 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2)C1 ZINC000880558370 CC On-Demand Anodyne CCR1 40 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2)C1 ZINC000880558370 CC On-Demand Anodyne ABCB1 80 48 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)c2ccccc2)C1 ZINC000880558378 GD On-Demand Anodyne SLC12A5 45 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)c2ccccc2)C1 ZINC000880558380 GD On-Demand Anodyne SLC12A5 45 37 COC(=O)[C@@]1(O)CCN(Cc2cccc(Br)c2)C1 ZINC000880558384 DD On-Demand Anodyne SIGMAR1 25 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(Br)c2)C1 ZINC000880558384 DD On-Demand Anodyne ADAM17 15 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(Br)c2)C1 ZINC000880558384 DD On-Demand Anodyne MCHR2 45 36 COC[C@@H]1CCCN(C(=O)Nc2cncc(OC)c2)C1 ZINC000880558389 CD On-Demand Anodyne PDGFRB 41 35 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(F)cc2)C1 ZINC000880558408 DC On-Demand Anodyne ACOX1 56 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(F)cc2)C1 ZINC000880558408 DC On-Demand Anodyne CCR1 46 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(F)cc2)C1 ZINC000880558408 DC On-Demand Anodyne ABCB1 63 48 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(F)cc2)C1 ZINC000880558409 DC On-Demand Anodyne ACOX1 56 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(F)cc2)C1 ZINC000880558409 DC On-Demand Anodyne CCR1 46 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(F)cc2)C1 ZINC000880558409 DC On-Demand Anodyne ABCB1 63 48 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne CYP11B1 15 43 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne HTR2C 18 41 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne PDGFRB 40 41 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne FAAH 15 45 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne NOD1 15 40 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne NOD2 40 40 COc1cncc(NC(=O)N2CCc3ccccc3CC2)c1 ZINC000880558419 CF On-Demand Anodyne TRPC6 15 43 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccccc3)oc2C)C1 ZINC000880558421 DD On-Demand Anodyne PPARG 90 43 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccccc3)oc2C)C1 ZINC000880558421 DD On-Demand Anodyne PPARA 97 43 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccccc3)oc2C)C1 ZINC000880558421 DD On-Demand Anodyne PDE8B 81 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne LTA4H 45 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne MMP13 28 47 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne ADAM17 22 47 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne MMP9 21 47 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne PSMB2 40 38 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Br)cc2)C1 ZINC000880558423 ED On-Demand Anodyne PSMB1 42 38 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)C(c2ccccc2)c2ccccc2)C1 ZINC000880558428 GD On-Demand Anodyne OPRK1 32 41 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558431 GD On-Demand Anodyne OPRK1 22 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558431 GD On-Demand Anodyne TACR2 51 37 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(Cl)c(Cl)c2)C1 ZINC000880558431 GD On-Demand Anodyne TACR3 40 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccc(OC)c(OC)c2)C1 ZINC000880558432 FB On-Demand Anodyne MTNR1B 15 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne DRD2 17 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne DRD4 34 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne DRD3 15 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne CHRM3 17 50 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne SIGMAR1 41 48 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne FAAH 22 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne MCHR2 45 36 COC(=O)[C@@]1(O)CCN(Cc2cccc(Cl)c2)C1 ZINC000880558435 CD On-Demand Anodyne CCR8 27 41 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)C(C)(C)C)C2)c1 ZINC000880558443 EE On-Demand Anodyne CCR3 18 46 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)C(C)(C)C)C2)c1 ZINC000880558444 EE On-Demand Anodyne CCR3 18 46 COc1cncc(NC(=O)NCCN2CCN(C(=O)C3CCCCC3)CC2)c1 ZINC000880558447 GD On-Demand Anodyne DRD4 46 35 COc1cncc(NC(=O)NCCN2CCN(C(=O)C3CCCCC3)CC2)c1 ZINC000880558447 GD On-Demand Anodyne HRH2 22 41 COc1cncc(NC(=O)NCCN2CCN(C(=O)C3CCCCC3)CC2)c1 ZINC000880558447 GD On-Demand Anodyne CCR3 40 42 COc1cncc(NC(=O)NCCN2CCN(C(=O)C3CCCCC3)CC2)c1 ZINC000880558447 GD On-Demand Anodyne CHRNA7 16 45 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne LTA4H 53 41 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne HRH3 27 40 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne MMP13 26 45 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne MMP9 17 45 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne PSMB2 41 39 CCOc1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558455 DD On-Demand Anodyne PSMB1 43 39 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne LTA4H 53 41 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne HRH3 27 40 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne MMP13 26 45 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne MMP9 17 45 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne PSMB2 41 39 CCOc1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558456 DD On-Demand Anodyne PSMB1 43 39 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne HTR1A 28 41 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne DRD2 28 41 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne DRD4 48 39 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne HRH2 15 41 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne DRD3 46 42 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne CCR3 28 45 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne NOD1 15 40 COc1cncc(NC(=O)NCCN2Cc3ccccc3C2)c1 ZINC000880558457 DE On-Demand Anodyne NOD2 40 40 COc1cncc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)c1 ZINC000880558458 FD On-Demand Anodyne PDGFRB 47 40 COc1cncc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)c1 ZINC000880558458 FD On-Demand Anodyne FAAH 21 50 COc1cncc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)c1 ZINC000880558458 FD On-Demand Anodyne ABCB1 23 42 COc1cncc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)c1 ZINC000880558459 FD On-Demand Anodyne PDGFRB 47 40 COc1cncc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)c1 ZINC000880558459 FD On-Demand Anodyne FAAH 21 50 COc1cncc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)c1 ZINC000880558459 FD On-Demand Anodyne ABCB1 23 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2ccc(F)cc2)C1 ZINC000880558465 CC On-Demand Anodyne SLC6A3 16 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2ccc(F)cc2)C1 ZINC000880558468 CC On-Demand Anodyne SLC6A3 16 42 COc1cncc(NC(=O)N(C)CCN2CCCC2)c1 ZINC000880558473 CD On-Demand Anodyne DRD4 41 31 COc1cncc(NC(=O)N(C)CCN2CCCC2)c1 ZINC000880558473 CD On-Demand Anodyne CASR 17 40 COc1cncc(NC(=O)N(C)CCN2CCCC2)c1 ZINC000880558473 CD On-Demand Anodyne ROCK2 23 42 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C(C)C)C1 ZINC000880558478 ED On-Demand Anodyne SLC12A5 48 36 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2ccc(OC)c(OC)c2)C1 ZINC000880558480 FC On-Demand Anodyne MT-ND1 22 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2ccc(OC)c(OC)c2)C1 ZINC000880558481 FC On-Demand Anodyne MT-ND1 22 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3CC[C@H]2C)C1 ZINC000880558486 EC On-Demand Anodyne DRD4 26 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2c3ccccc3CC[C@@H]2C)C1 ZINC000880558487 EC On-Demand Anodyne DRD4 26 45 O=C(CCCn1ccnc1)NCc1cn(C2CCC2)nn1 ZINC000880558491 CD On-Demand Anodyne TBXAS1 36 41 COc1cncc(NC(=O)N(C)Cc2cc[nH]n2)c1 ZINC000880558492 CD On-Demand Anodyne ROCK2 28 45 COc1cncc(NC(=O)N2CCC(C(=O)N3CCOCC3)CC2)c1 ZINC000880558493 ED On-Demand Anodyne EPHX2 15 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880558495 FB On-Demand Anodyne MMP13 69 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880558495 FB On-Demand Anodyne ADAM17 52 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880558495 FB On-Demand Anodyne MMP9 50 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880558495 FB On-Demand Anodyne MMP1 39 49 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2)C1 ZINC000880558507 DC On-Demand Anodyne ADRB2 16 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2)C1 ZINC000880558507 DC On-Demand Anodyne ACOX1 81 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2)C1 ZINC000880558507 DC On-Demand Anodyne CCR1 41 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2)C1 ZINC000880558507 DC On-Demand Anodyne ABCB1 58 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2)C1 ZINC000880558508 DC On-Demand Anodyne ADRB2 16 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2)C1 ZINC000880558508 DC On-Demand Anodyne ACOX1 81 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2)C1 ZINC000880558508 DC On-Demand Anodyne CCR1 41 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2)C1 ZINC000880558508 DC On-Demand Anodyne ABCB1 58 42 COc1cncc(NC(=O)NC2CCN(CC#N)CC2)c1 ZINC000880558513 CD On-Demand Mild EPHX2 43 38 COc1cncc(NC(=O)NC2CCN(CC#N)CC2)c1 ZINC000880558513 CD On-Demand Mild CXCR3 20 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558519 FD On-Demand Anodyne ACOX1 64 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558519 FD On-Demand Anodyne CCR1 40 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558519 FD On-Demand Anodyne ABCB1 45 39 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558520 FD On-Demand Anodyne ACOX1 64 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558520 FD On-Demand Anodyne CCR1 40 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C(C)(C)C)cc2)C1 ZINC000880558520 FD On-Demand Anodyne ABCB1 45 39 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)CC(F)(F)F)C1 ZINC000880558528 FD On-Demand Anodyne SLC12A5 56 36 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880558533 FE On-Demand Anodyne EDNRB 47 35 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880558533 FE On-Demand Anodyne EDNRA 47 39 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880558533 FE On-Demand Anodyne BMP1 70 40 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880558533 FE On-Demand Anodyne ROCK2 20 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3cccc(Cl)c3)CC2)C1 ZINC000880558540 GC On-Demand Anodyne DRD4 32 46 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3cccc(Cl)c3)CC2)C1 ZINC000880558540 GC On-Demand Anodyne SIGMAR1 25 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3cccc(Cl)c3)CC2)C1 ZINC000880558540 GC On-Demand Anodyne FAAH 30 49 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccc(F)cc3F)C2)c1 ZINC000880558542 EF On-Demand Anodyne CCR3 41 42 COc1cncc(NC(=O)N[C@H]2CCN(c3ccc(F)cc3F)C2)c1 ZINC000880558544 EF On-Demand Anodyne CCR3 41 42 COc1cncc(NC(=O)N[C@H]2CCCN(c3ccccc3)C2)c1 ZINC000880558545 EF On-Demand Anodyne CCR3 25 41 COc1cncc(NC(=O)N[C@@H]2CCCN(c3ccccc3)C2)c1 ZINC000880558546 EF On-Demand Anodyne CCR3 25 41 COc1cncc(NC(=O)N2CCN(Cc3nc(C)c(C)o3)CC2)c1 ZINC000880558547 EE On-Demand Anodyne FAAH 17 47 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccccc2OC)C1 ZINC000880558551 EB On-Demand Anodyne DRD2 22 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccccc2OC)C1 ZINC000880558551 EB On-Demand Anodyne DRD3 34 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccccc2OC)C1 ZINC000880558551 EB On-Demand Anodyne MBTPS1 50 34 COC(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558564 CC On-Demand Anodyne SIGMAR1 17 46 COC(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558564 CC On-Demand Anodyne MMP13 15 41 COC(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558564 CC On-Demand Anodyne NPFFR1 37 47 COC(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880558564 CC On-Demand Anodyne NOD2 41 36 COC(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558565 CC On-Demand Anodyne SIGMAR1 17 46 COC(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558565 CC On-Demand Anodyne MMP13 15 41 COC(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558565 CC On-Demand Anodyne NPFFR1 37 47 COC(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880558565 CC On-Demand Anodyne NOD2 41 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne OPRM1 34 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne OPRD1 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne MME 63 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne CMA1 41 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne PAPA1_CARPA 41 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne CYSP_TRYCR 45 33 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne TIMP3 73 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne CAPNS1 50 32 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne ACE2 64 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne PSMB8 67 41 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne NPFFR1 46 34 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558568 EB On-Demand Anodyne SLC12A5 63 37 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(=O)(=O)N(C)C)c2)C1 ZINC000880558569 EC On-Demand Anodyne MMP13 18 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(=O)(=O)N(C)C)c2)C1 ZINC000880558569 EC On-Demand Anodyne MMP9 15 44 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne OPRM1 34 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne OPRD1 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne MME 63 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne CMA1 41 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne PAPA1_CARPA 41 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne CYSP_TRYCR 45 33 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne TIMP3 73 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne CAPNS1 50 32 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne ACE2 64 36 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne PSMB8 67 41 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne NPFFR1 46 34 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](Cc2ccccc2)C(C)=O)C1 ZINC000880558571 EB On-Demand Anodyne SLC12A5 63 37 COc1cncc(NC(=O)NCCCNc2ccccc2)c1 ZINC000880558578 DF On-Demand Anodyne ADRB1 40 31 COc1cncc(NC(=O)NCCCNc2ccccc2)c1 ZINC000880558578 DF On-Demand Anodyne CCR3 34 48 COc1cncc(NC(=O)NCCCNc2ccccc2)c1 ZINC000880558578 DF On-Demand Anodyne RAF1 15 43 COc1cncc(NC(=O)NCCCNc2ccccc2)c1 ZINC000880558578 DF On-Demand Anodyne MTNR1A 48 38 COc1cncc(NC(=O)NCCCNc2ccccc2)c1 ZINC000880558578 DF On-Demand Anodyne MTNR1B 50 40 COc1cncc(NC(=O)N2CCN(CC(C)(C)O)CC2)c1 ZINC000880558592 DD On-Demand Anodyne PDGFRB 45 36 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558593 GH On-Demand Anodyne CPT1A 131 59 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558593 GH On-Demand Anodyne GRM5 26 62 COc1cncc(NC(=O)N2CCCC[C@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558593 GH On-Demand Anodyne SMO 38 45 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558595 GH On-Demand Anodyne CPT1A 131 59 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558595 GH On-Demand Anodyne GRM5 26 62 COc1cncc(NC(=O)N2CCCC[C@@H]2c2nc(-c3ccccc3)no2)c1 ZINC000880558595 GH On-Demand Anodyne SMO 38 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2ccccc2OC)C1 ZINC000880558647 EC On-Demand Anodyne ABCB1 51 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2ccccc2OC)C1 ZINC000880558649 EC On-Demand Anodyne ABCB1 51 41 COc1cncc(NC(=O)Nc2ccc(NC(=O)CC(C)C)cc2)c1 ZINC000880558653 EH On-Demand Anodyne RAF1 18 45 COc1cncc(NC(=O)Nc2ccc(NC(=O)CC(C)C)cc2)c1 ZINC000880558653 EH On-Demand Anodyne MTNR1A 15 42 COc1cncc(NC(=O)Nc2ccc(NC(=O)CC(C)C)cc2)c1 ZINC000880558653 EH On-Demand Anodyne MTNR1B 21 56 COc1cncc(NC(=O)Nc2ccc(NC(=O)CC(C)C)cc2)c1 ZINC000880558653 EH On-Demand Anodyne ENPP1 56 33 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(F)(F)F)cc2)C1 ZINC000880558678 DD On-Demand Anodyne MMP13 19 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(F)(F)F)cc2)C1 ZINC000880558678 DD On-Demand Anodyne SLC6A5 31 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(F)(F)F)cc2)C1 ZINC000880558678 DD On-Demand Anodyne MMP9 16 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(F)(F)F)cc2)C1 ZINC000880558678 DD On-Demand Anodyne SLC12A5 16 41 COc1cncc(NC(=O)NCc2ccnc(OC3CCOCC3)c2)c1 ZINC000880558686 FE On-Demand Anodyne ROCK2 16 41 COc1cncc(NC(=O)N2CCC([C@H](O)c3ccc(Cl)cc3)CC2)c1 ZINC000880558689 GH On-Demand Anodyne SCN10A 23 41 COc1cncc(NC(=O)N2CCC([C@@H](O)c3ccc(Cl)cc3)CC2)c1 ZINC000880558693 GH On-Demand Anodyne SCN10A 23 41 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccc(Cl)c3)no2)C1 ZINC000880558694 ED On-Demand Anodyne GRM5 21 46 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccc(OC)cc2)C2CC2)C1 ZINC000880558704 FC On-Demand Anodyne MMP13 29 41 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccc(OC)cc2)C2CC2)C1 ZINC000880558704 FC On-Demand Anodyne MMP9 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccc(OC)cc2)C2CC2)C1 ZINC000880558704 FC On-Demand Anodyne MMP1 23 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3cccc(C)c3)CC2)C1 ZINC000880558710 GC On-Demand Anodyne FAAH 25 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)Cc2ccco2)C1 ZINC000880558716 FD On-Demand Anodyne MRGPRX1 23 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(N3CCOCC3)CCCCC2)C1 ZINC000880558719 GB On-Demand Anodyne HCN1 55 35 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(N3CCOCC3)CCCCC2)C1 ZINC000880558719 GB On-Demand Anodyne HCN4 51 34 CCCCCN(CCO)C(=O)Nc1cncc(OC)c1 ZINC000880558743 CE On-Demand Anodyne INHA 42 34 COC(=O)[C@@]1(O)CCN(Cc2csc(Nc3ccccc3)n2)C1 ZINC000880558757 ED On-Demand Anodyne TRPC6 49 38 COC(=O)[C@@]1(O)CCN(Cc2csc(Nc3ccccc3)n2)C1 ZINC000880558757 ED On-Demand Anodyne TRPC3 47 36 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)cc2)C1 ZINC000880558764 BD On-Demand Anodyne SIGMAR1 21 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)cc2)C1 ZINC000880558764 BD On-Demand Anodyne MMP13 17 50 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000880558770 EC On-Demand Anodyne MMP13 29 43 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000880558770 EC On-Demand Anodyne CCR1 39 45 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000880558770 EC On-Demand Anodyne ADAM17 32 43 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(Cl)cc2)C1 ZINC000880558770 EC On-Demand Anodyne MMP9 22 43 COc1cncc(NC(=O)NCCCN2CCCCC2=O)c1 ZINC000880558773 DD On-Demand Anodyne HRH2 21 42 COc1cncc(NC(=O)NCCCN2CCCCC2=O)c1 ZINC000880558773 DD On-Demand Anodyne CCR3 31 43 COc1cncc(NC(=O)NCCCN2CCCCC2=O)c1 ZINC000880558773 DD On-Demand Anodyne QPCT 21 40 COc1cncc(NC(=O)NCCCN2CCCCC2=O)c1 ZINC000880558773 DD On-Demand Anodyne TYRO3 20 45 COc1cncc(NC(=O)N2CCN([C@@H](C)c3cccnc3)CC2)c1 ZINC000880558778 EE On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)N2CCN([C@@H](C)c3cccnc3)CC2)c1 ZINC000880558778 EE On-Demand Anodyne PTAFR 27 42 COc1cncc(NC(=O)N2CCN([C@@H](C)c3cccnc3)CC2)c1 ZINC000880558778 EE On-Demand Anodyne S1PR2 16 42 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne HTR1A 25 49 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne DRD2 18 49 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne ADRA1D 21 49 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne ADRA1A 31 49 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne ADRA1B 25 49 COC(=O)[C@@]1(O)CCN(CCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880558780 EC On-Demand Anodyne HTR7 20 49 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne MME 49 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne PAPA1_CARPA 55 38 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne CTSL 40 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne TIMP3 58 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne MMP3 22 42 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne NPY5R 20 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne CTSS 20 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne MMP9 19 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne ACE2 49 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne MMP1 27 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne FPR1 35 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne PSMB8 49 33 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558781 ED On-Demand Anodyne GPR142 46 39 COc1cncc(NC(=O)N2CCN([C@H](C)c3cccnc3)CC2)c1 ZINC000880558782 EE On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)N2CCN([C@H](C)c3cccnc3)CC2)c1 ZINC000880558782 EE On-Demand Anodyne PTAFR 27 42 COc1cncc(NC(=O)N2CCN([C@H](C)c3cccnc3)CC2)c1 ZINC000880558782 EE On-Demand Anodyne S1PR2 16 42 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne MME 49 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne PAPA1_CARPA 55 38 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne CTSL 40 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne TIMP3 58 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne MMP3 22 42 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne NPY5R 20 40 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne CTSS 20 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne MMP9 19 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne ACE2 49 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne MMP1 27 40 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne FPR1 35 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne PSMB8 49 33 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N(C)C)c1 ZINC000880558783 ED On-Demand Anodyne GPR142 46 39 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC)c2)c1 ZINC000880558786 DD On-Demand Anodyne ADRB3 45 39 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC)c2)c1 ZINC000880558786 DD On-Demand Anodyne ROCK1 35 43 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC)c2)c1 ZINC000880558786 DD On-Demand Anodyne MTNR1A 32 40 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC)c2)c1 ZINC000880558786 DD On-Demand Anodyne MTNR1B 35 44 COc1cncc(NC(=O)NC[C@H](O)c2cccc(OC)c2)c1 ZINC000880558786 DD On-Demand Anodyne ROCK2 43 47 COc1cncc(NC(=O)N(C)Cc2ccccc2N2CCOCC2)c1 ZINC000880558787 FF On-Demand Anodyne CASR 27 42 COc1cncc(NC(=O)N(C)Cc2ccccc2N2CCOCC2)c1 ZINC000880558787 FF On-Demand Anodyne PIK3CD 16 40 COc1cncc(NC(=O)N(C)Cc2ccccc2N2CCOCC2)c1 ZINC000880558787 FF On-Demand Anodyne PIK3CB 29 40 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)c1 ZINC000880558788 DD On-Demand Anodyne ADRB3 45 39 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)c1 ZINC000880558788 DD On-Demand Anodyne ROCK1 35 43 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)c1 ZINC000880558788 DD On-Demand Anodyne MTNR1A 32 40 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)c1 ZINC000880558788 DD On-Demand Anodyne MTNR1B 35 44 COc1cncc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)c1 ZINC000880558788 DD On-Demand Anodyne ROCK2 43 47 COc1cncc(NC(=O)N2CCC(c3n[nH]c(-c4ccccc4)n3)CC2)c1 ZINC000880558790 GG On-Demand Anodyne AKT2 41 39 COc1cncc(NC(=O)N2CCC(C(F)(F)F)(C(F)(F)F)C2)c1 ZINC000880558791 FG On-Demand Anodyne EPHX2 34 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(C)cccc2C)C1 ZINC000880558795 DC On-Demand Anodyne ACOX1 51 35 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(C)cccc2C)C1 ZINC000880558795 DC On-Demand Anodyne ABCB1 70 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(C)cccc2C)C1 ZINC000880558796 DC On-Demand Anodyne ACOX1 51 35 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(C)cccc2C)C1 ZINC000880558796 DC On-Demand Anodyne ABCB1 70 42 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccccc2)C1 ZINC000880558797 DC On-Demand Anodyne SLC12A5 61 37 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880558799 DD On-Demand Anodyne NPY5R 31 41 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1cncc(OC)c1 ZINC000880558800 DD On-Demand Anodyne NPY5R 31 41 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(OC)cc2)C1 ZINC000880558803 EC On-Demand Anodyne MMP13 24 42 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(OC)cc2)C1 ZINC000880558803 EC On-Demand Anodyne MMP9 24 42 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(OC)cc2)C1 ZINC000880558803 EC On-Demand Anodyne MMP1 19 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne DRD4 46 35 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne HRH2 29 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne SIGMAR1 37 53 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MMP13 28 56 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne NPFFR2 25 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne ADAM17 17 56 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MTNR1A 41 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MTNR1B 42 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne FAAH 26 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MMP9 15 56 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MCHR1 20 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne MCHR2 56 34 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne CACNA1G 15 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne CCR8 30 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2)C1 ZINC000880558821 CC On-Demand Anodyne NPFFR1 34 45 COC(=O)c1cccc(CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880558822 CC On-Demand Anodyne CHRM3 17 46 COC(=O)c1cccc(CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880558822 CC On-Demand Anodyne MCHR2 45 33 COC(=O)c1cccc(CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880558823 CC On-Demand Anodyne CHRM3 17 46 COC(=O)c1cccc(CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880558823 CC On-Demand Anodyne MCHR2 45 33 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCc3ccccc32)C1 ZINC000880558832 DC On-Demand Anodyne DRD4 18 49 CC(C)(C)OC(=O)NC[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880558833 GF On-Demand Anodyne REN 58 35 CC(C)(C)OC(=O)NC[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880558833 GF On-Demand Anodyne FPR1 44 35 CC(C)(C)OC(=O)NC[C@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880558835 GF On-Demand Anodyne REN 58 35 CC(C)(C)OC(=O)NC[C@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880558835 GF On-Demand Anodyne FPR1 44 35 COc1cncc(NC(=O)NCC2CCN(C(C)=O)CC2)c1 ZINC000880558836 DD On-Demand Anodyne CCR3 50 43 COc1cncc(NC(=O)NCC2CCN(C(C)=O)CC2)c1 ZINC000880558836 DD On-Demand Anodyne EPHX2 25 43 COc1cncc(NC(=O)NCC2CCN(C(C)=O)CC2)c1 ZINC000880558836 DD On-Demand Anodyne CACNA1I 56 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2cccc(OC)c2)C1 ZINC000880558840 EC On-Demand Anodyne DRD4 40 30 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2cccc(OC)c2)C1 ZINC000880558840 EC On-Demand Anodyne MTNR1A 17 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2cccc(OC)c2)C1 ZINC000880558840 EC On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2cccc(OC)c2)C1 ZINC000880558840 EC On-Demand Anodyne ABCB1 45 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2cccc(OC)c2)C1 ZINC000880558842 EC On-Demand Anodyne DRD4 40 30 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2cccc(OC)c2)C1 ZINC000880558842 EC On-Demand Anodyne MTNR1A 17 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2cccc(OC)c2)C1 ZINC000880558842 EC On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2cccc(OC)c2)C1 ZINC000880558842 EC On-Demand Anodyne ABCB1 45 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne HTR1A 23 46 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne DRD2 28 46 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne DRD4 24 46 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne ACHE 20 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne ADRA1D 21 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne ADRA1A 38 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne ADRA1B 26 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne DRD3 36 46 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne KCNH2 15 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne LTA4H 44 38 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne HTR7 19 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne HRH3 72 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne SIGMAR1 42 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne MMP13 23 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne HTR5A 19 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne ADAM17 20 53 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne MMP9 18 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne EPHX2 23 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2)C1 ZINC000880558864 CD On-Demand Anodyne SLC12A5 55 37 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C(C)(C)C)C1 ZINC000880558871 ED On-Demand Anodyne SLC12A5 51 35 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(Br)c2)C1 ZINC000880558889 FC On-Demand Anodyne ACOX1 69 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(Br)c2)C1 ZINC000880558889 FC On-Demand Anodyne ABCB1 55 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(Br)c2)C1 ZINC000880558890 FC On-Demand Anodyne ACOX1 69 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(Br)c2)C1 ZINC000880558890 FC On-Demand Anodyne ABCB1 55 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880558893 FF On-Demand Anodyne PDGFRB 46 37 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880558893 FF On-Demand Anodyne HRH3 24 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CHRM2 15 48 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne DRD2 27 44 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne DRD4 58 44 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne ACHE 55 47 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne DRD3 22 43 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne KCNH2 15 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CHRM3 18 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne LTA4H 34 46 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne SIGMAR1 62 49 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne SSTR5 52 37 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne BCHE 20 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CCR3 52 46 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CCR5 23 49 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne NPFFR2 19 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne FAAH 30 44 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne NPY5R 23 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CXCR3 17 40 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne MCHR1 67 49 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne CCR8 28 43 COc1cncc(NC(=O)N(C)C2CCN(Cc3ccccc3)CC2)c1 ZINC000880558904 FG On-Demand Anodyne NPFFR1 26 40 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccc(OC)cc3)no2)C1 ZINC000880558906 EC On-Demand Anodyne PDK1 40 34 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne DRD2 15 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne HRH2 18 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne DRD3 23 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne LTA4H 29 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne HRH3 81 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne SIGMAR1 23 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne MMP13 35 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne HTR5A 17 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne ADAM17 21 48 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne MMP9 26 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne EPHX2 20 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(OC)cc2)C1 ZINC000880558926 DD On-Demand Anodyne MMP1 24 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne LTA4H 49 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne HRH3 26 51 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne MMP13 25 44 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne CCR1 58 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne ADAM17 17 44 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne EBP 22 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne MMP9 19 44 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)cc2)C1 ZINC000880558936 CD On-Demand Anodyne PSMB1 42 36 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne LTA4H 54 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne SIGMAR1 15 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne MMP13 35 53 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne ADAM17 20 53 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne MMP9 27 53 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne MMP1 22 53 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne PSMB2 41 39 COC(=O)[C@@]1(O)CCN(CCOc2ccc(OC)cc2)C1 ZINC000880558944 CC On-Demand Anodyne PSMB1 44 37 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccccn2)c1 ZINC000880558945 EE On-Demand Anodyne ROCK2 30 47 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2C)C1 ZINC000880558971 DC On-Demand Anodyne CCR1 45 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(C)cc2C)C1 ZINC000880558971 DC On-Demand Anodyne ABCB1 65 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2C)C1 ZINC000880558972 DC On-Demand Anodyne CCR1 45 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(C)cc2C)C1 ZINC000880558972 DC On-Demand Anodyne ABCB1 65 46 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(C)c2)C1 ZINC000880558992 EC On-Demand Anodyne HRH2 35 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(C)c2)C1 ZINC000880558992 EC On-Demand Anodyne MTNR1A 18 41 COc1cncc(NC(=O)N(C)C2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880559004 FF On-Demand Anodyne L3MBTL3 46 35 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc([N+](=O)[O-])c2)C1 ZINC000880559006 CD On-Demand Bother CACNA1C 54 37 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc([N+](=O)[O-])c2)C1 ZINC000880559006 CD On-Demand Bother CACNA1D 81 37 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc([N+](=O)[O-])c2)C1 ZINC000880559007 CD On-Demand Bother CACNA1C 54 37 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc([N+](=O)[O-])c2)C1 ZINC000880559007 CD On-Demand Bother CACNA1D 81 37 COc1cncc(NC(=O)NCCNC(=O)C(C)C)c1 ZINC000880559012 CC On-Demand Anodyne MTNR1A 21 42 COc1cncc(NC(=O)NCCNC(=O)C(C)C)c1 ZINC000880559012 CC On-Demand Anodyne MTNR1B 19 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559016 EC On-Demand Anodyne DRD4 40 31 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559016 EC On-Demand Anodyne ACOX1 58 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559016 EC On-Demand Anodyne ABCB1 58 56 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559017 EC On-Demand Anodyne DRD4 40 31 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559017 EC On-Demand Anodyne ACOX1 58 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(C)=O)c2)C1 ZINC000880559017 EC On-Demand Anodyne ABCB1 58 56 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3=O)c2)c1 ZINC000880559019 FF On-Demand Anodyne HRH2 26 43 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3=O)c2)c1 ZINC000880559019 FF On-Demand Anodyne ROCK2 43 47 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3=O)c2)c1 ZINC000880559019 FF On-Demand Anodyne NAMPT 41 39 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2ccc(Cl)cc2)C1 ZINC000880559020 EC On-Demand Anodyne CCR1 71 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2ccc(Cl)cc2)C1 ZINC000880559021 EC On-Demand Anodyne CCR1 71 36 COC(=O)[C@@]1(O)CCN(Cc2cnc(-c3ccccc3)s2)C1 ZINC000880559025 DD On-Demand Anodyne MGEA5 36 47 COc1cncc(NC(=O)NC[C@@H](O)COCC2CC2)c1 ZINC000880559026 CC On-Demand Anodyne ADRB1 40 32 COc1cncc(NC(=O)NC[C@H](O)COCC2CC2)c1 ZINC000880559027 CC On-Demand Anodyne ADRB1 40 32 COC(=O)[C@@]1(O)CCN(Cc2csc(Nc3ccc(C)cc3)n2)C1 ZINC000880559058 EE On-Demand Anodyne TRPC6 49 42 COC(=O)[C@@]1(O)CCN(Cc2csc(Nc3ccc(C)cc3)n2)C1 ZINC000880559058 EE On-Demand Anodyne TRPC3 48 42 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne F2 34 40 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne ACE 34 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne P2RY12 106 38 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne MME 44 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne MC4R 76 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne CMA1 47 34 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne TACR2 16 46 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne TRY2_BOVIN 92 38 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne CTSL 49 39 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne CACNA1B 20 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne F2R 53 34 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne TIMP3 68 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne PREP 25 53 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne MMP3 17 55 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne CCKBR 27 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne ACE2 76 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne MC1R 27 43 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne DPP7 42 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne ST14 67 35 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne FPR1 31 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne PSMB8 43 34 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne Q9N6S8_PLAFA 15 41 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559059 FE On-Demand Anodyne BRCA1 50 30 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne F2 34 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne ACE 34 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne P2RY12 106 38 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne MME 44 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne MC4R 76 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne CMA1 47 34 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne TACR2 16 46 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne TRY2_BOVIN 92 38 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne CTSL 49 39 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne CACNA1B 20 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne F2R 53 34 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne TIMP3 68 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne PREP 25 53 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne MMP3 17 55 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne CCKBR 27 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne ACE2 76 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne MC1R 27 43 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne DPP7 42 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne ST14 67 35 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne FPR1 31 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne PSMB8 43 34 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne Q9N6S8_PLAFA 15 41 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c1 ZINC000880559060 FE On-Demand Anodyne BRCA1 50 30 COC(=O)[C@@]1(O)CCN(Cc2ncc(-c3ccccc3)o2)C1 ZINC000880559068 DD On-Demand Anodyne NPPA 35 42 COC(=O)[C@@]1(O)CCN(Cc2coc(-c3ccccc3)n2)C1 ZINC000880559071 DD On-Demand Anodyne PDE8B 56 33 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCC(C)CC3)C2)c1 ZINC000880559087 EG On-Demand Anodyne CCR3 20 59 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559088 GD On-Demand Anodyne OPRL1 15 45 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559088 GD On-Demand Anodyne NPY2R 42 38 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559088 GD On-Demand Anodyne MTNR1B 30 42 COc1cncc(NC(=O)N2CCC[C@H](CN3CCC(C)CC3)C2)c1 ZINC000880559089 EG On-Demand Anodyne CCR3 20 59 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCCCCC3)C2)c1 ZINC000880559090 EG On-Demand Anodyne PDGFRB 40 35 COc1cncc(NC(=O)N2CCC[C@@H](CN3CCCCCC3)C2)c1 ZINC000880559090 EG On-Demand Anodyne CCR3 46 37 COc1cncc(NC(=O)N2CCC[C@H](CN3CCCCCC3)C2)c1 ZINC000880559092 EG On-Demand Anodyne PDGFRB 40 35 COc1cncc(NC(=O)N2CCC[C@H](CN3CCCCCC3)C2)c1 ZINC000880559092 EG On-Demand Anodyne CCR3 46 37 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559095 GD On-Demand Anodyne OPRL1 15 45 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559095 GD On-Demand Anodyne NPY2R 42 38 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2cccc(OC)c2)c2ccccc2)C1 ZINC000880559095 GD On-Demand Anodyne MTNR1B 30 42 COc1cncc(NC(=O)NCCCNC2CCCCC2)c1 ZINC000880559097 DF On-Demand Anodyne HRH2 20 42 COc1cncc(NC(=O)NCCCNC2CCCCC2)c1 ZINC000880559097 DF On-Demand Anodyne EPHX2 15 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne DRD4 41 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne SIGMAR1 35 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne MMP13 20 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne CCR1 62 39 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne ADAM17 15 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne MMP9 15 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne CXCR3 26 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2)C1 ZINC000880559099 CD On-Demand Anodyne PA 27 43 COc1cncc(NC(=O)N2CCN(c3cc(OC)ccn3)CC2)c1 ZINC000880559102 ED On-Demand Anodyne PDGFRB 58 44 COc1cncc(NC(=O)N2CCN(c3cc(OC)ccn3)CC2)c1 ZINC000880559102 ED On-Demand Anodyne KARS 41 32 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne PDGFRB 37 40 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne CCR3 30 45 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne CHRNA7 18 42 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne FAAH 15 46 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne EPHX2 79 53 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne CXCR3 17 44 COc1cncc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c1 ZINC000880559106 FF On-Demand Anodyne MCHR1 16 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559117 EC On-Demand Anodyne ACOX1 70 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559117 EC On-Demand Anodyne CCR1 86 43 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559117 EC On-Demand Anodyne EBP 17 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559117 EC On-Demand Anodyne ABCB1 52 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559119 EC On-Demand Anodyne ACOX1 70 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559119 EC On-Demand Anodyne CCR1 86 43 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559119 EC On-Demand Anodyne EBP 17 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2)C1 ZINC000880559119 EC On-Demand Anodyne ABCB1 52 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880559123 EC On-Demand Anodyne PDGFRB 43 36 COC(=O)[C@@]1(O)CCN(CCOCCOc2ccccc2)C1 ZINC000880559124 DC On-Demand Anodyne HRH3 25 41 COC(=O)[C@@]1(O)CCN(CCOCCOc2ccccc2)C1 ZINC000880559124 DC On-Demand Anodyne SIGMAR1 16 42 COC(=O)[C@@]1(O)CCN(CCOCCOc2ccccc2)C1 ZINC000880559124 DC On-Demand Anodyne MMP13 17 48 COC(=O)[C@@]1(O)CCN(CCOCCOc2ccccc2)C1 ZINC000880559124 DC On-Demand Anodyne MMP9 15 48 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne HTR4 26 45 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne CCR3 37 42 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne SLC6A5 20 40 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne EPHX2 48 47 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne CXCR3 21 46 COc1cncc(NC(=O)NC2CCN(CCO)CC2)c1 ZINC000880559126 CC On-Demand Anodyne MCHR1 21 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC(c2ccccc2)c2ccccc2)C1 ZINC000880559138 GD On-Demand Anodyne OPRL1 22 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC(c2ccccc2)c2ccccc2)C1 ZINC000880559138 GD On-Demand Anodyne BIRC8 44 31 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC(c2ccccc2)c2ccccc2)C1 ZINC000880559140 GD On-Demand Anodyne OPRL1 22 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC(c2ccccc2)c2ccccc2)C1 ZINC000880559140 GD On-Demand Anodyne BIRC8 44 31 COc1cncc(NC(=O)N2CCCN(C(=O)Oc3ccccc3)CC2)c1 ZINC000880559141 FF On-Demand Anodyne PDGFRB 43 43 COc1cncc(NC(=O)N2CCCN(C(=O)Oc3ccccc3)CC2)c1 ZINC000880559141 FF On-Demand Anodyne FAAH 23 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne SIGMAR1 18 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne MMP13 19 52 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne NPFFR2 17 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne ADAM17 15 52 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne MMP9 16 52 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2)C1 ZINC000880559146 DD On-Demand Anodyne NPFFR1 28 40 COC(=O)[C@@]1(O)CCN([C@H](C(=O)N2CCCCC2)c2ccccc2)C1 ZINC000880559151 ED On-Demand Anodyne DPP7 45 36 COc1cncc(NC(=O)NCC2(N3CCC(OC)CC3)CCCC2)c1 ZINC000880559158 FF On-Demand Anodyne HCN1 61 40 COc1cncc(NC(=O)NCC2(N3CCC(OC)CC3)CCCC2)c1 ZINC000880559158 FF On-Demand Anodyne HCN4 57 38 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne DRD4 44 35 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne PDGFRB 16 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne MTNR1A 31 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne MTNR1B 37 46 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne EPHX2 19 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(OC)c2)C1 ZINC000880559162 DC On-Demand Anodyne TAAR1 36 40 COC(=O)[C@@]1(O)CCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000880559163 CC On-Demand Anodyne ADRA2B 22 50 COC(=O)[C@@]1(O)CCN(C[C@@H]2COc3ccccc3O2)C1 ZINC000880559163 CC On-Demand Anodyne ADRA2C 15 42 COC(=O)[C@@]1(O)CCN(C[C@H]2COc3ccccc3O2)C1 ZINC000880559167 CC On-Demand Anodyne ADRA2B 22 50 COC(=O)[C@@]1(O)CCN(C[C@H]2COc3ccccc3O2)C1 ZINC000880559167 CC On-Demand Anodyne ADRA2C 15 42 CCOc1ccccc1CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880559169 CD On-Demand Anodyne CCR8 30 41 CCOc1ccccc1CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880559169 CD On-Demand Anodyne HCN1 63 38 CCOc1ccccc1CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880559169 CD On-Demand Anodyne HCN4 54 38 CCOc1ccccc1CN1CC[C@](O)(C(=O)OC)C1 ZINC000880559171 CD On-Demand Anodyne CCR8 30 41 CCOc1ccccc1CN1CC[C@](O)(C(=O)OC)C1 ZINC000880559171 CD On-Demand Anodyne HCN1 63 38 CCOc1ccccc1CN1CC[C@](O)(C(=O)OC)C1 ZINC000880559171 CD On-Demand Anodyne HCN4 54 38 O=C(NCc1cn(C2CCC2)nn1)c1cc(OCc2ccccc2)ccn1 ZINC000880559172 FF On-Demand Anodyne PREP 28 41 O=C(NCc1cn(C2CCC2)nn1)c1cc(OCc2ccccc2)ccn1 ZINC000880559172 FF On-Demand Anodyne SCD1 21 40 O=C(NCc1cn(C2CCC2)nn1)c1cc(OCc2ccccc2)ccn1 ZINC000880559172 FF On-Demand Anodyne SCD 20 40 COc1cncc(NC(=O)NCCCc2cnn(C)c2)c1 ZINC000880559197 CD On-Demand Anodyne CCR3 24 42 COc1cncc(NC(=O)NCCCc2cnn(C)c2)c1 ZINC000880559197 CD On-Demand Anodyne QPCT 21 40 COc1cncc(NC(=O)N[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559205 EE On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559205 EE On-Demand Anodyne CCR3 24 42 COc1cncc(NC(=O)N[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559205 EE On-Demand Anodyne MTNR1A 24 59 COc1cncc(NC(=O)N[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559205 EE On-Demand Anodyne MTNR1B 29 59 COc1cncc(NC(=O)N[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559205 EE On-Demand Anodyne EPHX2 41 42 COc1cncc(NC(=O)N[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559206 EE On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559206 EE On-Demand Anodyne CCR3 24 42 COc1cncc(NC(=O)N[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559206 EE On-Demand Anodyne MTNR1A 24 59 COc1cncc(NC(=O)N[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559206 EE On-Demand Anodyne MTNR1B 29 59 COc1cncc(NC(=O)N[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559206 EE On-Demand Anodyne EPHX2 41 42 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(C)c2)c1 ZINC000880559209 DG On-Demand Anodyne ROCK2 20 46 COC(=O)[C@@]1(O)CCN(Cc2cnn(-c3ccccc3)c2)C1 ZINC000880559212 DC On-Demand Anodyne DRD4 16 52 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COC(c2ccccc2)c2ccccc2)C1 ZINC000880559222 GD On-Demand Anodyne SLC6A3 26 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COC(c2ccccc2)c2ccccc2)C1 ZINC000880559222 GD On-Demand Anodyne ABCB1 56 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COC(c2ccccc2)c2ccccc2)C1 ZINC000880559224 GD On-Demand Anodyne SLC6A3 26 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COC(c2ccccc2)c2ccccc2)C1 ZINC000880559224 GD On-Demand Anodyne ABCB1 56 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)cc2)C1 ZINC000880559228 CC On-Demand Anodyne SIGMAR1 36 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)cc2)C1 ZINC000880559228 CC On-Demand Anodyne MMP13 19 51 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)cc2)C1 ZINC000880559228 CC On-Demand Anodyne ADAM17 15 51 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)cc2)C1 ZINC000880559228 CC On-Demand Anodyne MLNR 45 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559232 FD On-Demand Anodyne HRH1 24 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559232 FD On-Demand Anodyne ACOX1 86 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559232 FD On-Demand Anodyne CCR1 45 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559232 FD On-Demand Anodyne CCR3 25 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559232 FD On-Demand Anodyne ABCB1 46 39 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559233 FD On-Demand Anodyne HRH1 24 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559233 FD On-Demand Anodyne ACOX1 86 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559233 FD On-Demand Anodyne CCR1 45 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559233 FD On-Demand Anodyne CCR3 25 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)c(Cl)c2)C1 ZINC000880559233 FD On-Demand Anodyne ABCB1 46 39 CCOCCN1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880559238 DD On-Demand Anodyne PDGFRB 48 39 COC(=O)[C@@]1(O)CCN(Cc2csc(-c3ccc(OC)c(OC)c3)n2)C1 ZINC000880559247 GD On-Demand Anodyne PPARD 15 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccn3)CC2)c1 ZINC000880559251 ED On-Demand Anodyne PDGFRB 54 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccn3)CC2)c1 ZINC000880559251 ED On-Demand Anodyne GRM4 51 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccn3)CC2)c1 ZINC000880559251 ED On-Demand Anodyne FAAH 18 43 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne DRD2 16 40 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne ADRA1B 15 40 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne OPRM1 28 56 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne OPRD1 22 56 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne OPRK1 20 56 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne OPRL1 15 50 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne SIGMAR1 67 46 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne MMP13 15 50 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne NPFFR2 23 42 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne EBP 15 42 COC(=O)[C@@]1(O)CCN(CCc2ccccc2)C1 ZINC000880559253 BC On-Demand Anodyne SLC12A5 78 44 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne MTNR1A 24 40 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne MTNR1B 21 40 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne ROCK2 21 50 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne HCN1 43 32 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne HCN4 40 31 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne KCNK3 38 41 CCOc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880559254 DF On-Demand Anodyne KCNK9 24 41 COc1cncc(NC(=O)N2CC[C@H](NC(=O)Nc3ccc(F)cc3)C2)c1 ZINC000880559255 FF On-Demand Anodyne CCR3 69 46 COc1cncc(NC(=O)N2CC[C@H](NC(=O)Nc3ccc(F)cc3)C2)c1 ZINC000880559255 FF On-Demand Anodyne EPHX2 67 45 COc1cncc(NC(=O)N2CC[C@@H](NC(=O)Nc3ccc(F)cc3)C2)c1 ZINC000880559256 FF On-Demand Anodyne CCR3 69 46 COc1cncc(NC(=O)N2CC[C@@H](NC(=O)Nc3ccc(F)cc3)C2)c1 ZINC000880559256 FF On-Demand Anodyne EPHX2 67 45 COCCN(CCN(C)C)C(=O)Nc1cncc(OC)c1 ZINC000880559258 CD On-Demand Anodyne ROCK2 20 44 CCNc1nc(C)c(C(=O)NCc2cn(C3CCC3)nn2)s1 ZINC000880559262 DE On-Demand Anodyne SCD1 25 44 CCNc1nc(C)c(C(=O)NCc2cn(C3CCC3)nn2)s1 ZINC000880559262 DE On-Demand Anodyne SCD 23 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2Cl)C1 ZINC000880559268 EC On-Demand Anodyne ADRB2 24 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2Cl)C1 ZINC000880559268 EC On-Demand Anodyne ADRB1 17 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2Cl)C1 ZINC000880559268 EC On-Demand Anodyne CCR1 51 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2Cl)C1 ZINC000880559268 EC On-Demand Anodyne ABCB1 80 49 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2Cl)C1 ZINC000880559270 EC On-Demand Anodyne ADRB2 24 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2Cl)C1 ZINC000880559270 EC On-Demand Anodyne ADRB1 17 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2Cl)C1 ZINC000880559270 EC On-Demand Anodyne CCR1 51 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2Cl)C1 ZINC000880559270 EC On-Demand Anodyne ABCB1 80 49 COC(=O)[C@@]1(O)CCN(Cc2ccc([N+](=O)[O-])cc2)C1 ZINC000880559271 CC On-Demand Bother MMP13 15 42 COC(=O)[C@@]1(O)CCN(Cc2ccc([N+](=O)[O-])cc2)C1 ZINC000880559271 CC On-Demand Bother MMP9 22 42 COC(=O)[C@@]1(O)CCN(Cc2ccc([N+](=O)[O-])cc2)C1 ZINC000880559271 CC On-Demand Bother KCNJ1 29 46 O=C(NCc1cn(C2CCC2)nn1)c1cc(N2CCNC2=O)ccc1Cl ZINC000880559282 FE On-Demand Anodyne P2RX7 18 42 C=C(C)CN(CC)C(=O)Nc1cncc(OC)c1 ZINC000880559285 BF On-Demand Mild ROCK2 15 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne ADRB2 26 55 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne ADRB1 22 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne HTR1A 15 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne ACOX1 43 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne CCR1 43 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3ccccc23)C1 ZINC000880559287 ED On-Demand Anodyne ABCB1 82 49 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne ADRB2 26 55 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne ADRB1 22 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne HTR1A 15 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne ACOX1 43 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne CCR1 43 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3ccccc23)C1 ZINC000880559288 ED On-Demand Anodyne ABCB1 82 49 COc1cncc(NC(=O)N(C)[C@H](C)CNC(=O)OC(C)(C)C)c1 ZINC000880559300 EE On-Demand Anodyne NPY5R 31 40 COc1cncc(NC(=O)N(C)[C@@H](C)CNC(=O)OC(C)(C)C)c1 ZINC000880559301 EE On-Demand Anodyne NPY5R 31 40 C=CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880559305 CD On-Demand Mild EPHX2 44 38 C=CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880559305 CD On-Demand Mild CXCR3 20 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(SC)cc2)C1 ZINC000880559307 CD On-Demand Anodyne SIGMAR1 16 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(SC)cc2)C1 ZINC000880559307 CD On-Demand Anodyne MMP13 15 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(SC)cc2)C1 ZINC000880559307 CD On-Demand Anodyne NOD2 24 41 COc1cncc(NC(=O)NCCCCNc2ccccn2)c1 ZINC000880559313 DE On-Demand Anodyne ADRB1 40 31 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Br)c2)C1 ZINC000880559315 ED On-Demand Anodyne MMP13 16 45 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Br)c2)C1 ZINC000880559315 ED On-Demand Anodyne ADAM17 17 45 COC(=O)[C@@]1(O)CCN(CCOc2cccc(Br)c2)C1 ZINC000880559315 ED On-Demand Anodyne MMP9 15 45 COc1cncc(NC(=O)NCC2CCN(C)CC2)c1 ZINC000880559317 CD On-Demand Anodyne CCR3 48 44 COc1cncc(NC(=O)NCC2CCN(C)CC2)c1 ZINC000880559317 CD On-Demand Anodyne CACNA1I 59 35 COc1cncc(NC(=O)NC[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559323 FF On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NC[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559323 FF On-Demand Anodyne CCR3 51 46 COc1cncc(NC(=O)NC[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559323 FF On-Demand Anodyne MTNR1A 19 47 COc1cncc(NC(=O)NC[C@@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559323 FF On-Demand Anodyne MTNR1B 24 47 COc1cncc(NC(=O)NC[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559324 FF On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NC[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559324 FF On-Demand Anodyne CCR3 51 46 COc1cncc(NC(=O)NC[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559324 FF On-Demand Anodyne MTNR1A 19 47 COc1cncc(NC(=O)NC[C@H]2CCN(c3cccc(OC)c3)C2)c1 ZINC000880559324 FF On-Demand Anodyne MTNR1B 24 47 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne CPT1A 43 43 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne GRM5 21 45 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne FAAH 15 46 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne EPHX2 15 51 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne SMO 52 61 COc1cncc(NC(=O)N2CCC(c3nc(-c4ccccc4)no3)CC2)c1 ZINC000880559330 GH On-Demand Anodyne ETHR 63 49 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)nc2)C1 ZINC000880559331 CC On-Demand Anodyne Q8WSF8_APLCA 42 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)nc2)C1 ZINC000880559331 CC On-Demand Anodyne NACHRBETA2 53 38 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)c2ccccc2)C1 ZINC000880559357 FD On-Demand Anodyne SLC12A5 46 37 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(C)c2)C1 ZINC000880559372 CC On-Demand Anodyne KCNK3 58 36 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(C)c2)C1 ZINC000880559372 CC On-Demand Anodyne KCNK9 50 36 CCN(Cc1ccc(C(=O)N(C)C)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880559382 FF On-Demand Anodyne ROCK1 16 41 CCN(Cc1ccc(C(=O)N(C)C)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880559382 FF On-Demand Anodyne ROCK2 23 47 COc1cncc(NC(=O)NC[C@@H](O)COCC(C)C)c1 ZINC000880559399 CD On-Demand Anodyne ADRB1 40 31 COc1cncc(NC(=O)NC[C@H](O)COCC(C)C)c1 ZINC000880559401 CD On-Demand Anodyne ADRB1 40 31 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(F)cc2)c2ccccc2)C1 ZINC000880559402 FE On-Demand Anodyne OPRL1 15 40 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(F)cc2)c2ccccc2)C1 ZINC000880559402 FE On-Demand Anodyne NPY2R 62 36 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(F)cc2)c2ccccc2)C1 ZINC000880559409 FE On-Demand Anodyne OPRL1 15 40 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(F)cc2)c2ccccc2)C1 ZINC000880559409 FE On-Demand Anodyne NPY2R 62 36 COc1cncc(NC(=O)N2CCN(Cc3nccn3C)CC2)c1 ZINC000880559411 ED On-Demand Anodyne PDGFRB 49 36 COc1cncc(NC(=O)N2CCN(Cc3nccn3C)CC2)c1 ZINC000880559411 ED On-Demand Anodyne FAAH 18 45 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne HTR1A 38 42 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne DRD2 40 42 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne DRD4 44 33 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne HRH2 20 43 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne HTR2A 21 49 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne HTR2C 16 42 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne ADRA1A 18 42 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne DRD3 72 42 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne FGFR1 27 45 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne CCR3 47 49 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne CHRNA7 18 49 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne EPHX2 19 41 COc1cncc(NC(=O)NCCCCN2CCN(C)CC2)c1 ZINC000880559416 DD On-Demand Anodyne QPCT 15 41 COc1cncc(NC(=O)N2CCc3c(C)cccc3C2)c1 ZINC000880559417 CF On-Demand Anodyne DRD4 40 32 COc1cncc(NC(=O)N2CCc3c(C)cccc3C2)c1 ZINC000880559417 CF On-Demand Anodyne P2RY14 54 39 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccccc2)C1 ZINC000880559421 CC On-Demand Anodyne TIMP3 42 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccccc2)C1 ZINC000880559425 CC On-Demand Anodyne TIMP3 42 33 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C(C)C)c1 ZINC000880559427 EG On-Demand Bother COLA 34 40 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C(C)C)c1 ZINC000880559427 EG On-Demand Bother MMP2 21 47 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C(C)C)c1 ZINC000880559427 EG On-Demand Bother MMP8 41 47 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C(C)C)c1 ZINC000880559427 EG On-Demand Bother MMP9 24 47 COc1cncc(NC(=O)N(Cc2ccc([N+](=O)[O-])cc2)C(C)C)c1 ZINC000880559427 EG On-Demand Bother MMP1 29 47 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2ccccc2)C1 ZINC000880559442 DC On-Demand Anodyne ABCB1 58 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2ccccc2)C1 ZINC000880559442 DC On-Demand Anodyne SLC12A5 70 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2ccccc2)C1 ZINC000880559443 DC On-Demand Anodyne ABCB1 58 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2ccccc2)C1 ZINC000880559443 DC On-Demand Anodyne SLC12A5 70 40 COc1cncc(NC(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000880559448 DE On-Demand Anodyne CHRNA7 15 46 COc1cncc(NC(=O)N2CCC[C@@H]2CN2CCCC2)c1 ZINC000880559449 DE On-Demand Anodyne CHRNA7 15 46 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)CCC(=O)N3)c1 ZINC000880559460 EF On-Demand Anodyne GRIN2B 17 45 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)CCC(=O)N3)c1 ZINC000880559461 EF On-Demand Anodyne GRIN2B 17 45 COc1cncc(NC(=O)N2CCC[C@@H](C)CC2)c1 ZINC000880559462 CF On-Demand Anodyne TRPC6 26 42 COc1cncc(NC(=O)N2CCC[C@@H](C)CC2)c1 ZINC000880559462 CF On-Demand Anodyne TRPC3 23 42 COc1cncc(NC(=O)N2CCC[C@H](C)CC2)c1 ZINC000880559463 CF On-Demand Anodyne TRPC6 26 42 COc1cncc(NC(=O)N2CCC[C@H](C)CC2)c1 ZINC000880559463 CF On-Demand Anodyne TRPC3 23 42 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccs3)oc2C)C1 ZINC000880559472 DD On-Demand Anodyne PPARG 23 42 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccs3)oc2C)C1 ZINC000880559472 DD On-Demand Anodyne PPARA 38 42 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccs3)oc2C)C1 ZINC000880559472 DD On-Demand Anodyne PDE8B 62 36 COc1cncc(NC(=O)NCCc2ccc(C)nc2)c1 ZINC000880559473 CE On-Demand Anodyne RAF1 27 40 COc1cncc(NC(=O)NCCc2ccc(C)nc2)c1 ZINC000880559473 CE On-Demand Anodyne PIK3CG 15 43 C=CCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559474 FC On-Demand Mild CCR1 43 36 C=CCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559474 FC On-Demand Mild ABCB1 50 38 C=CCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559475 FC On-Demand Mild CCR1 43 36 C=CCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559475 FC On-Demand Mild ABCB1 50 38 C=CCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559476 FC On-Demand Mild CCR1 43 36 C=CCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559476 FC On-Demand Mild ABCB1 50 38 C=CCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559477 FC On-Demand Mild CCR1 43 36 C=CCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880559477 FC On-Demand Mild ABCB1 50 38 COc1cncc(NC(=O)N2CCCC[C@H](N3CCCC3)C2)c1 ZINC000880559478 DF On-Demand Anodyne HRH3 18 40 COc1cncc(NC(=O)N2CCCC[C@H](N3CCCC3)C2)c1 ZINC000880559478 DF On-Demand Anodyne L3MBTL3 54 36 COc1cncc(NC(=O)N2CCCC[C@@H](N3CCCC3)C2)c1 ZINC000880559479 DF On-Demand Anodyne HRH3 18 40 COc1cncc(NC(=O)N2CCCC[C@@H](N3CCCC3)C2)c1 ZINC000880559479 DF On-Demand Anodyne L3MBTL3 54 36 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)[C@H]2CCCc3ccccc32)C1 ZINC000880559482 ED On-Demand Anodyne SIGMAR1 16 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)[C@@H]2CCCc3ccccc32)C1 ZINC000880559483 ED On-Demand Anodyne SIGMAR1 16 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C)c2)C1 ZINC000880559486 DC On-Demand Anodyne ADRB2 19 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C)c2)C1 ZINC000880559486 DC On-Demand Anodyne ADRB1 17 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C)c2)C1 ZINC000880559486 DC On-Demand Anodyne ACOX1 80 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C)c2)C1 ZINC000880559486 DC On-Demand Anodyne CCR1 43 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C)c2)C1 ZINC000880559486 DC On-Demand Anodyne ABCB1 66 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C)c2)C1 ZINC000880559487 DC On-Demand Anodyne ADRB2 19 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C)c2)C1 ZINC000880559487 DC On-Demand Anodyne ADRB1 17 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C)c2)C1 ZINC000880559487 DC On-Demand Anodyne ACOX1 80 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C)c2)C1 ZINC000880559487 DC On-Demand Anodyne CCR1 43 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C)c2)C1 ZINC000880559487 DC On-Demand Anodyne ABCB1 66 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2Cl)C1 ZINC000880559490 DE On-Demand Anodyne P2RX7 32 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2Cl)C1 ZINC000880559490 DE On-Demand Anodyne EPHX2 17 43 C#CCOc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880559497 DD On-Demand Mild CA14 17 46 COC(=O)[C@@]1(O)CCN(CCOc2cccc(C)c2)C1 ZINC000880559507 CC On-Demand Anodyne DRD4 40 33 CCc1nc(CNC(=O)Nc2cncc(OC)c2)cs1 ZINC000880559514 CE On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559515 FD On-Demand Anodyne ADRB2 24 42 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559515 FD On-Demand Anodyne ADRB1 54 41 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559515 FD On-Demand Anodyne ADRB3 24 40 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559516 FD On-Demand Anodyne ADRB2 24 42 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559516 FD On-Demand Anodyne ADRB1 54 41 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)c(F)c2)c1 ZINC000880559516 FD On-Demand Anodyne ADRB3 24 40 COC(=O)[C@@]1(O)CCN(CCOc2cccc(F)c2)C1 ZINC000880559524 CC On-Demand Anodyne CHRNA10 32 40 COC(=O)[C@@]1(O)CCN(CCC(=O)NCc2ccccc2Cl)C1 ZINC000880559526 EC On-Demand Anodyne HTR7 15 44 COc1cncc(NC(=O)NCCc2ccc(OC)c(F)c2)c1 ZINC000880559527 DF On-Demand Anodyne CCR3 16 41 COc1cncc(NC(=O)NCCc2ccc(OC)c(F)c2)c1 ZINC000880559527 DF On-Demand Anodyne RAF1 33 43 O=C(NCc1cn(C2CCC2)nn1)c1cnc(Cc2ccccc2)s1 ZINC000880559530 FF On-Demand Anodyne PREP 22 40 O=C(Nc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1)OCC(F)(F)F ZINC000880559541 GG On-Demand Anodyne CA14 20 46 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccc(C)cc3)CC2)c1 ZINC000880559542 FF On-Demand Anodyne EPHX2 60 52 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccc(C)cc3)CC2)c1 ZINC000880559542 FF On-Demand Anodyne L3MBTL3 52 33 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C)c(C)c2)C1 ZINC000880559555 DD On-Demand Anodyne DRD2 16 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C)c(C)c2)C1 ZINC000880559555 DD On-Demand Anodyne DRD3 19 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C)c(C)c2)C1 ZINC000880559555 DD On-Demand Anodyne HRH3 78 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C)c(C)c2)C1 ZINC000880559555 DD On-Demand Anodyne MMP13 19 43 COC(=O)[C@@]1(O)CCN(CCC(=O)N2CCN(c3ccc(F)cc3)CC2)C1 ZINC000880559558 GC On-Demand Anodyne SSTR1 32 42 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCCO3)c1 ZINC000880559559 EF On-Demand Anodyne BMP1 43 36 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCCO3)c1 ZINC000880559559 EF On-Demand Anodyne NOS2 57 33 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCCO3)c1 ZINC000880559559 EF On-Demand Anodyne ROCK2 23 44 CC(C)(C)OC(=O)N1CCN(CCC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880559564 GD On-Demand Anodyne GPR119 40 37 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne HTR1A 38 44 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne DRD2 36 42 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne DRD4 35 50 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne DRD3 42 42 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne PDGFRB 60 42 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne HTR7 30 40 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne CCR3 20 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne FAAH 31 54 COc1cncc(NC(=O)N2CCN(Cc3ccccc3OC)CC2)c1 ZINC000880559573 FE On-Demand Anodyne CCR8 30 43 CC[C@@H](NC(=O)CN1CC[C@@](O)(C(=O)OC)C1)c1ccc(Cl)cc1 ZINC000880559590 FD On-Demand Anodyne AKT3 23 41 CC[C@@H](NC(=O)CN1CC[C@](O)(C(=O)OC)C1)c1ccc(Cl)cc1 ZINC000880559591 FD On-Demand Anodyne AKT3 23 41 CC[C@H](NC(=O)CN1CC[C@](O)(C(=O)OC)C1)c1ccc(Cl)cc1 ZINC000880559592 FD On-Demand Anodyne AKT3 23 41 CC[C@H](NC(=O)CN1CC[C@@](O)(C(=O)OC)C1)c1ccc(Cl)cc1 ZINC000880559593 FD On-Demand Anodyne AKT3 23 41 COc1cncc(NC(=O)NC2CCOCC2)c1 ZINC000880559601 CD On-Demand Anodyne EPHX2 45 37 COCCN(Cc1cccnc1)C(=O)Nc1cncc(OC)c1 ZINC000880559633 DE On-Demand Anodyne PTAFR 26 40 COCCN(Cc1cccnc1)C(=O)Nc1cncc(OC)c1 ZINC000880559633 DE On-Demand Anodyne CHRNA7 34 41 COCCN(Cc1cccnc1)C(=O)Nc1cncc(OC)c1 ZINC000880559633 DE On-Demand Anodyne ROCK1 20 47 COCCN(Cc1cccnc1)C(=O)Nc1cncc(OC)c1 ZINC000880559633 DE On-Demand Anodyne ROCK2 35 47 CCN(Cc1ccc(CN(C)C)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880559635 EG On-Demand Anodyne ROCK1 15 45 CCN(Cc1ccc(CN(C)C)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880559635 EG On-Demand Anodyne ROCK2 25 49 COc1cncc(NC(=O)NCc2cnn(C)c2)c1 ZINC000880559645 CD On-Demand Anodyne ROCK2 17 44 COc1cncc(NC(=O)NCc2cnn(C)c2)c1 ZINC000880559645 CD On-Demand Anodyne NAMPT 36 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559652 ED On-Demand Anodyne ADRB2 21 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559652 ED On-Demand Anodyne ACOX1 85 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559652 ED On-Demand Anodyne CCR1 42 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559652 ED On-Demand Anodyne ABCB1 72 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559653 ED On-Demand Anodyne ADRB2 21 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559653 ED On-Demand Anodyne ACOX1 85 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559653 ED On-Demand Anodyne CCR1 42 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc3ccccc3c2)C1 ZINC000880559653 ED On-Demand Anodyne ABCB1 72 42 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne HTR1A 28 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne DRD2 21 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne ADRA1D 24 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne ADRA1A 35 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne ADRA1B 28 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne DRD3 16 50 COC(=O)[C@@]1(O)CCN(CCCCN2C(=O)c3ccccc3C2=O)C1 ZINC000880559654 EC On-Demand Anodyne HTR7 24 50 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(N)=O)c2)C1 ZINC000880559664 CB On-Demand Anodyne NPFFR2 35 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(N)=O)c2)C1 ZINC000880559664 CB On-Demand Anodyne MCHR2 44 36 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(N)=O)c2)C1 ZINC000880559664 CB On-Demand Anodyne NPFFR1 46 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(N)=O)c2)C1 ZINC000880559664 CB On-Demand Anodyne SLC12A5 45 35 COc1cncc(NC(=O)N2CCN3CCCC[C@@H]3C2)c1 ZINC000880559669 CD On-Demand Anodyne HRH3 22 42 COc1cncc(NC(=O)N2CCN3CCCC[C@@H]3C2)c1 ZINC000880559669 CD On-Demand Anodyne L3MBTL3 47 35 COc1cncc(NC(=O)N2CCN3CCCC[C@H]3C2)c1 ZINC000880559670 CD On-Demand Anodyne HRH3 22 42 COc1cncc(NC(=O)N2CCN3CCCC[C@H]3C2)c1 ZINC000880559670 CD On-Demand Anodyne L3MBTL3 47 35 COc1cncc(NC(=O)N2CC[C@@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559671 EH On-Demand Anodyne CACNA1H 43 38 COc1cncc(NC(=O)N2CC[C@@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559671 EH On-Demand Anodyne CCR1 42 41 COc1cncc(NC(=O)N2CC[C@@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559671 EH On-Demand Anodyne SCN10A 30 41 COc1cncc(NC(=O)N2CC[C@@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559671 EH On-Demand Anodyne MCHR1 20 47 COc1cncc(NC(=O)N2CC[C@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559672 EH On-Demand Anodyne CACNA1H 43 38 COc1cncc(NC(=O)N2CC[C@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559672 EH On-Demand Anodyne CCR1 42 41 COc1cncc(NC(=O)N2CC[C@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559672 EH On-Demand Anodyne SCN10A 30 41 COc1cncc(NC(=O)N2CC[C@H](c3ccc(Cl)cc3)C2)c1 ZINC000880559672 EH On-Demand Anodyne MCHR1 20 47 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother HRH2 19 42 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother CACNA1C 62 39 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother SIGMAR1 15 48 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother CACNA1D 93 38 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother FAAH 15 45 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2)C1 ZINC000880559677 CC On-Demand Bother SLC12A5 41 34 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccccc2OC)C1 ZINC000880559680 EC On-Demand Anodyne MBTPS1 49 33 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccccc2OC)c1 ZINC000880559689 EH On-Demand Anodyne FKBP1A 66 36 COc1cncc(NC(=O)N2CCCC[C@H]2c2ccccc2OC)c1 ZINC000880559689 EH On-Demand Anodyne CPT1A 80 36 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccccc2OC)c1 ZINC000880559690 EH On-Demand Anodyne FKBP1A 66 36 COc1cncc(NC(=O)N2CCCC[C@@H]2c2ccccc2OC)c1 ZINC000880559690 EH On-Demand Anodyne CPT1A 80 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559696 DC On-Demand Anodyne ACOX1 54 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559696 DC On-Demand Anodyne CCR1 43 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559696 DC On-Demand Anodyne ABCB1 45 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559697 DC On-Demand Anodyne ACOX1 54 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559697 DC On-Demand Anodyne CCR1 43 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)cc(C)c2)C1 ZINC000880559697 DC On-Demand Anodyne ABCB1 45 38 CCOCCN(CC)C(=O)Nc1cncc(OC)c1 ZINC000880559705 CD On-Demand Anodyne ROCK2 16 40 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccccc2Cl)C1 ZINC000880559711 CE On-Demand Anodyne OPRL1 38 42 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccccc2Cl)C1 ZINC000880559712 CE On-Demand Anodyne OPRL1 38 42 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne LTA4H 49 38 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne HRH3 29 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne MMP13 23 45 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne ADAM17 17 45 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne MMP9 17 45 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne PSMB2 40 38 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C)cc2)C1 ZINC000880559715 CC On-Demand Anodyne PSMB1 43 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C)C1 ZINC000880559718 DC On-Demand Anodyne ADRB2 26 46 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C)C1 ZINC000880559718 DC On-Demand Anodyne ADRB1 18 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C)C1 ZINC000880559718 DC On-Demand Anodyne ACOX1 41 32 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C)C1 ZINC000880559718 DC On-Demand Anodyne CCR1 46 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C)C1 ZINC000880559718 DC On-Demand Anodyne ABCB1 87 50 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C)C1 ZINC000880559719 DC On-Demand Anodyne ADRB2 26 46 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C)C1 ZINC000880559719 DC On-Demand Anodyne ADRB1 18 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C)C1 ZINC000880559719 DC On-Demand Anodyne ACOX1 41 32 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C)C1 ZINC000880559719 DC On-Demand Anodyne CCR1 46 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C)C1 ZINC000880559719 DC On-Demand Anodyne ABCB1 87 50 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccccc2C(F)(F)F)C1 ZINC000880559724 FD On-Demand Anodyne RBP4 49 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccccc2C(F)(F)F)C1 ZINC000880559725 FD On-Demand Anodyne RBP4 49 33 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccc2OC)c1 ZINC000880559736 EG On-Demand Anodyne FKBP1A 44 35 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccc2OC)c1 ZINC000880559736 EG On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccc2OC)c1 ZINC000880559737 EG On-Demand Anodyne FKBP1A 44 35 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccc2OC)c1 ZINC000880559737 EG On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)N2CCN(C(=O)C(C)C)CC2)c1 ZINC000880559752 DD On-Demand Anodyne PDGFRB 44 39 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccccc2)C1 ZINC000880559754 CC On-Demand Anodyne SLC12A5 51 38 COc1cncc(NC(=O)N(C)C[C@@H](C)c2ccccc2)c1 ZINC000880559755 CG On-Demand Anodyne NPY5R 36 41 COc1cncc(NC(=O)N(C)C[C@H](C)c2ccccc2)c1 ZINC000880559756 CG On-Demand Anodyne NPY5R 36 41 COc1cncc(NC(=O)N(CCc2ccccc2)C2CC2)c1 ZINC000880559757 DG On-Demand Anodyne ROCK2 24 47 COc1cncc(NC(=O)N(CCc2ccccc2)C2CC2)c1 ZINC000880559757 DG On-Demand Anodyne MBTPS1 40 36 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Cl)c2)C1 ZINC000880559763 DC On-Demand Anodyne MCHR1 37 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Cl)c2)C1 ZINC000880559763 DC On-Demand Anodyne CACNA1I 15 45 COc1cncc(NC(=O)NCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880559764 FD On-Demand Anodyne HTR1A 24 42 COc1cncc(NC(=O)NCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880559764 FD On-Demand Anodyne DRD2 17 41 COc1cncc(NC(=O)NCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880559764 FD On-Demand Anodyne DRD4 43 35 COc1cncc(NC(=O)NCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880559764 FD On-Demand Anodyne DRD3 26 42 COc1cncc(NC(=O)NCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880559764 FD On-Demand Anodyne SOAT1 27 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2ccccc2)C1 ZINC000880559779 CC On-Demand Anodyne OPRK1 21 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2ccccc2)C1 ZINC000880559782 CC On-Demand Anodyne OPRK1 21 41 COc1cncc(NC(=O)N(CCO)CC(C)(C)C)c1 ZINC000880559796 CD On-Demand Anodyne ROCK2 15 44 COc1cncc(NC(=O)N(CCO)Cc2cc(OC)ccc2OC)c1 ZINC000880559797 FE On-Demand Anodyne ROCK2 22 47 COC(=O)[C@@]1(O)CCN(Cc2nc3ccccc3[nH]2)C1 ZINC000880559813 CC On-Demand Anodyne PIN1 22 40 COC(=O)C1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880559816 DD On-Demand Anodyne EPHX2 41 38 COC(=O)[C@@]1(O)CCN(Cc2cc(-c3ccc(OC)cc3)no2)C1 ZINC000880559821 ED On-Demand Anodyne MMP13 19 41 COC(=O)[C@@]1(O)CCN(Cc2cc(-c3ccc(OC)cc3)no2)C1 ZINC000880559821 ED On-Demand Anodyne MMP9 15 41 COC(=O)[C@@]1(O)CCN(Cc2cc(-c3ccc(OC)cc3)no2)C1 ZINC000880559821 ED On-Demand Anodyne PDK1 49 35 CCN1CCC[C@@H]1CN(Cc1ccncc1)C(=O)Nc1cncc(OC)c1 ZINC000880559823 FG On-Demand Anodyne PDE4A 15 43 CCN1CCC[C@H]1CN(Cc1ccncc1)C(=O)Nc1cncc(OC)c1 ZINC000880559825 FG On-Demand Anodyne PDE4A 15 43 COc1cncc(NC(=O)NC2CCN(C(=O)CC(F)(F)F)CC2)c1 ZINC000880559831 FE On-Demand Anodyne EPHX2 58 59 COc1cncc(NC(=O)NC2CCN(C(=O)CC(F)(F)F)CC2)c1 ZINC000880559831 FE On-Demand Anodyne CXCR3 19 43 CCOc1ccccc1NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880559838 DC On-Demand Anodyne HCN1 52 36 CCOc1ccccc1NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880559838 DC On-Demand Anodyne HCN4 44 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)ccc2C)C1 ZINC000880559839 DC On-Demand Anodyne CCR1 45 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)ccc2C)C1 ZINC000880559839 DC On-Demand Anodyne ABCB1 65 46 CCOc1ccccc1NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880559840 DC On-Demand Anodyne HCN1 52 36 CCOc1ccccc1NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880559840 DC On-Demand Anodyne HCN4 44 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)ccc2C)C1 ZINC000880559841 DC On-Demand Anodyne CCR1 45 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)ccc2C)C1 ZINC000880559841 DC On-Demand Anodyne ABCB1 65 46 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HTR1A 26 41 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne DRD2 28 41 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne DRD4 42 32 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HRH2 38 51 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HTR2A 17 49 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne DRD3 56 41 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HTR4 18 45 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HRH3 24 42 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne NPY1R 15 44 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne CCR3 50 49 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne CHRNA7 28 58 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne HNMT 46 35 COc1cncc(NC(=O)NCCCCCN2CCCCC2)c1 ZINC000880559857 DF On-Demand Anodyne QPCT 15 40 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccccc2)C1 ZINC000880559859 BD On-Demand Anodyne OPRL1 29 52 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccccc2)C1 ZINC000880559863 BD On-Demand Anodyne OPRL1 29 52 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2cccc(OC)c2)C1 ZINC000880559865 EC On-Demand Anodyne DRD4 41 31 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2cccc(OC)c2)C1 ZINC000880559865 EC On-Demand Anodyne MMP13 15 43 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2cccc(OC)c2)C1 ZINC000880559865 EC On-Demand Anodyne ROCK1 27 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2cccc(OC)c2)C1 ZINC000880559865 EC On-Demand Anodyne TACR3 21 43 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2cccc(OC)c2)C1 ZINC000880559865 EC On-Demand Anodyne HSD17B2 17 46 Cc1nc(NC2CC2)sc1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880559872 EE On-Demand Anodyne SCD1 25 44 Cc1nc(NC2CC2)sc1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880559872 EE On-Demand Anodyne SCD 23 44 COc1cncc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)c1 ZINC000880559881 CD On-Demand Anodyne CCR3 53 45 COc1cncc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)c1 ZINC000880559881 CD On-Demand Anodyne EPHX2 40 36 COc1cncc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)c1 ZINC000880559881 CD On-Demand Anodyne CXCR3 19 44 COc1cncc(NC(=O)N[C@H]2CCN(CC3CC3)C2)c1 ZINC000880559882 CD On-Demand Anodyne CCR3 53 45 COc1cncc(NC(=O)N[C@H]2CCN(CC3CC3)C2)c1 ZINC000880559882 CD On-Demand Anodyne EPHX2 40 36 COc1cncc(NC(=O)N[C@H]2CCN(CC3CC3)C2)c1 ZINC000880559882 CD On-Demand Anodyne CXCR3 19 44 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCc1cn(C2CCC2)nn1 ZINC000880559883 GD On-Demand Anodyne CA14 15 42 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)Cc2ccc(F)cc2)C1 ZINC000880559890 DC On-Demand Anodyne TACR3 24 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559891 GD On-Demand Anodyne ACOX1 56 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559891 GD On-Demand Anodyne CCR1 40 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559891 GD On-Demand Anodyne ABCB1 77 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559893 GD On-Demand Anodyne ACOX1 56 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559893 GD On-Demand Anodyne CCR1 40 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Oc3ccccc3)cc2)C1 ZINC000880559893 GD On-Demand Anodyne ABCB1 77 45 COc1cncc(NC(=O)N2CCN3CCC[C@@H]3C2)c1 ZINC000880559919 CD On-Demand Anodyne HRH3 22 42 COc1cncc(NC(=O)N2CCN3CCC[C@H]3C2)c1 ZINC000880559920 CD On-Demand Anodyne HRH3 22 42 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3cccc(C)c3)no2)C1 ZINC000880559931 DD On-Demand Anodyne GRM5 20 46 COc1cncc(NC(=O)NCCc2ccc(OC)c(OC)c2OC)c1 ZINC000880559932 FE On-Demand Anodyne NQO2 40 38 COc1cncc(NC(=O)NCCc2ccc(OC)c(OC)c2OC)c1 ZINC000880559932 FE On-Demand Anodyne MTNR1A 67 42 COc1cncc(NC(=O)NCCc2ccc(OC)c(OC)c2OC)c1 ZINC000880559932 FE On-Demand Anodyne MTNR1B 48 41 COc1cncc(NC(=O)N2CCC[C@H]2c2nc3ccccc3[nH]2)c1 ZINC000880559943 EG On-Demand Anodyne PRCP 60 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2nc3ccccc3[nH]2)c1 ZINC000880559944 EG On-Demand Anodyne PRCP 60 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2C(F)(F)F)C1 ZINC000880559951 ED On-Demand Anodyne RBP4 46 33 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(C)cc2)c2ccccc2)C1 ZINC000880559952 FE On-Demand Anodyne OPRL1 15 40 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(C)cc2)c2ccccc2)C1 ZINC000880559952 FE On-Demand Anodyne NPY2R 35 42 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(C)cc2)c2ccccc2)C1 ZINC000880559955 FE On-Demand Anodyne OPRL1 15 40 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(C)cc2)c2ccccc2)C1 ZINC000880559955 FE On-Demand Anodyne NPY2R 35 42 COc1cncc(NC(=O)N2CCN(C(=O)c3c(F)cccc3F)CC2)c1 ZINC000880559956 GE On-Demand Anodyne FAAH 21 42 COc1cncc(NC(=O)N2CCN(C(=O)c3c(F)cccc3F)CC2)c1 ZINC000880559956 GE On-Demand Anodyne EPHX2 19 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1C[C@H]1Cc1ccccc1 ZINC000880559966 DE On-Demand Anodyne PREP 21 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1C[C@H]1Cc1ccccc1 ZINC000880559966 DE On-Demand Anodyne TMPRSS11D 56 35 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1C[C@H]1Cc1ccccc1 ZINC000880559967 DE On-Demand Anodyne PREP 21 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1C[C@H]1Cc1ccccc1 ZINC000880559967 DE On-Demand Anodyne TMPRSS11D 56 35 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1C[C@@H]1Cc1ccccc1 ZINC000880559968 DE On-Demand Anodyne PREP 21 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1C[C@@H]1Cc1ccccc1 ZINC000880559968 DE On-Demand Anodyne TMPRSS11D 56 35 O=C(NCc1cn(C2CCC2)nn1)[C@H]1C[C@@H]1Cc1ccccc1 ZINC000880559969 DE On-Demand Anodyne PREP 21 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1C[C@@H]1Cc1ccccc1 ZINC000880559969 DE On-Demand Anodyne TMPRSS11D 56 35 COc1cncc(NC(=O)N2CCN(CC(=O)NC3CCCCC3)CC2)c1 ZINC000880559974 GD On-Demand Anodyne FAAH 17 40 COc1cncc(NC(=O)N2CCN(CC(=O)NC3CCCCC3)CC2)c1 ZINC000880559974 GD On-Demand Anodyne EPHX2 17 40 COc1cncc(NC(=O)N2CCN(C(=O)CN3CCCC3)CC2)c1 ZINC000880559977 EC On-Demand Anodyne PDGFRB 45 36 COC(=O)[C@@]1(O)CCN(CCCc2nc(-c3cccs3)no2)C1 ZINC000880559983 ED On-Demand Anodyne ETHR 30 40 COc1cncc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880559987 FF On-Demand Anodyne MTOR 15 44 COc1cncc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880559987 FF On-Demand Anodyne EPHX2 54 43 COc1cncc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880559987 FF On-Demand Anodyne GPR119 47 44 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne DRD4 23 41 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne ACHE 19 40 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne SIGMAR1 28 42 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne SSTR5 46 36 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne CCR3 74 42 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne CXCR3 34 43 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne MCHR1 47 47 COc1cncc(NC(=O)NCc2ccc(CN3CCC(O)CC3)cc2)c1 ZINC000880559993 FE On-Demand Anodyne NAMPT 45 38 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)N2CCCc3ccccc32)C1 ZINC000880560005 EC On-Demand Anodyne AVPR2 33 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)N2CCCc3ccccc32)C1 ZINC000880560007 EC On-Demand Anodyne AVPR2 33 41 COC(=O)[C@@]1(O)CCN(Cc2noc(-c3ccc(OC)cc3)n2)C1 ZINC000880560013 EC On-Demand Anodyne S1PR1 15 41 COC(=O)[C@@]1(O)CCN(Cc2noc(-c3ccc(OC)cc3)n2)C1 ZINC000880560013 EC On-Demand Anodyne PDK1 40 34 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)N(C)C)c2ccccc2)C1 ZINC000880560016 DC On-Demand Anodyne NPY2R 50 37 COC(=O)[C@@]1(O)CCN([C@H](C(=O)N(C)C)c2ccccc2)C1 ZINC000880560017 DC On-Demand Anodyne NPY2R 50 37 COC(=O)[C@@]1(O)CCN(CCSc2ccc(Cl)cc2)C1 ZINC000880560024 DE On-Demand Anodyne CCR1 43 37 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2)C1 ZINC000880560034 CC On-Demand Mild LTA4H 41 37 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2)C1 ZINC000880560034 CC On-Demand Mild HRH3 17 47 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2)C1 ZINC000880560034 CC On-Demand Mild MMP13 20 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2)C1 ZINC000880560034 CC On-Demand Mild MMP9 15 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2)C1 ZINC000880560034 CC On-Demand Mild PSMB1 41 35 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne DRD4 18 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne HRH2 15 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne DRD3 19 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne LTA4H 22 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne HRH3 75 52 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne SIGMAR1 17 50 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne MMP13 26 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne CCR1 67 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne HTR5A 15 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne ADAM17 17 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne EBP 29 50 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne MMP9 18 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(Cl)cc2)C1 ZINC000880560051 DD On-Demand Anodyne EPHX2 22 50 COc1cncc(NC(=O)N(C)CCN2CCOCC2)c1 ZINC000880560063 CC On-Demand Anodyne CASR 55 51 COc1cncc(NC(=O)N(C)CCN2CCOCC2)c1 ZINC000880560063 CC On-Demand Anodyne EPHX2 19 43 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne SIGMAR1 28 55 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne MMP13 37 57 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne ADAM17 19 53 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne MMP2 15 41 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne MMP3 24 41 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne ABCB1 15 40 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne MMP9 31 57 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne MMP1 27 57 COC(=O)[C@@]1(O)CCN(CCc2ccc(OC)cc2)C1 ZINC000880560065 CC On-Demand Anodyne SLC12A5 30 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(C)ccc(C)c2C)C1 ZINC000880560066 EC On-Demand Anodyne ACOX1 47 32 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(C)ccc(C)c2C)C1 ZINC000880560066 EC On-Demand Anodyne ABCB1 51 39 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(C)ccc(C)c2C)C1 ZINC000880560067 EC On-Demand Anodyne ACOX1 47 32 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(C)ccc(C)c2C)C1 ZINC000880560067 EC On-Demand Anodyne ABCB1 51 39 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2cccs2)C1 ZINC000880560071 EC On-Demand Anodyne BMP1 16 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2cccs2)C1 ZINC000880560073 EC On-Demand Anodyne BMP1 16 41 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880560076 FE On-Demand Anodyne PDGFRB 34 41 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880560076 FE On-Demand Anodyne CCR3 19 40 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880560076 FE On-Demand Anodyne FAAH 17 43 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880560076 FE On-Demand Anodyne EPHX2 20 44 COc1cncc(NC(=O)NCC2(N3CCCC3)CCOCC2)c1 ZINC000880560083 ED On-Demand Anodyne HCN1 63 38 COc1cncc(NC(=O)NCC2(N3CCCC3)CCOCC2)c1 ZINC000880560083 ED On-Demand Anodyne HCN4 52 37 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)cc2F)C1 ZINC000880560088 ED On-Demand Anodyne AKR1B1 21 41 COc1cncc(NC(=O)N2CCCN(C(=O)CC3CCCC3)CC2)c1 ZINC000880560104 FF On-Demand Anodyne PDGFRB 48 37 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne LTA4H 68 45 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne HRH3 25 44 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne SIGMAR1 22 45 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne MMP13 21 53 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne ADAM17 21 53 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne MMP9 18 53 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne PSMB2 42 40 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne PSMB1 45 41 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2)C1 ZINC000880560106 CC On-Demand Anodyne SLC12A5 59 38 COc1cncc(NC(=O)NCCN2CCOC(C)(C)C2)c1 ZINC000880560111 DD On-Demand Anodyne DRD4 40 31 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2cccc(C(F)(F)F)c2)C1 ZINC000880560127 FD On-Demand Anodyne EPHX2 17 46 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2cccc(C(F)(F)F)c2)C1 ZINC000880560128 FD On-Demand Anodyne EPHX2 17 46 COc1cncc(NC(=O)N[C@H](C)Cn2cncn2)c1 ZINC000880560134 CC On-Demand Anodyne HIS3 82 38 COc1cncc(NC(=O)N[C@@H](C)Cn2cncn2)c1 ZINC000880560135 CC On-Demand Anodyne HIS3 82 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne HRH2 18 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne TACR1 25 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne SIGMAR1 17 47 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne CCR2 71 39 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne CACNA1G 21 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(F)(F)F)c2)C1 ZINC000880560141 DD On-Demand Anodyne SLC12A5 29 45 COc1cncc(NC(=O)NCc2ccc([C@@H](C)O)cc2)c1 ZINC000880560143 DE On-Demand Anodyne ROCK2 26 45 COc1cncc(NC(=O)NCc2ccc([C@H](C)O)cc2)c1 ZINC000880560144 DE On-Demand Anodyne ROCK2 26 45 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C(C)C)c1 ZINC000880560145 DH On-Demand Anodyne ROCK2 19 52 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C(C)C)c1 ZINC000880560145 DH On-Demand Anodyne NPY5R 24 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2ccccc2)C1 ZINC000880560147 DC On-Demand Anodyne AMP1_PLAFQ 23 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2ccccc2)C1 ZINC000880560147 DC On-Demand Anodyne SLC12A5 49 37 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2ccccc2)C1 ZINC000880560150 DC On-Demand Anodyne AMP1_PLAFQ 23 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2ccccc2)C1 ZINC000880560150 DC On-Demand Anodyne SLC12A5 49 37 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000880560152 EC On-Demand Anodyne DYRK2 55 32 COc1cncc(NC(=O)N2CCN([C@@H](C)C(=O)NC3CCCC3)CC2)c1 ZINC000880560159 GD On-Demand Anodyne PDGFRB 42 38 COc1cncc(NC(=O)N2CCN([C@H](C)C(=O)NC3CCCC3)CC2)c1 ZINC000880560160 GD On-Demand Anodyne PDGFRB 42 38 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(C(F)(F)F)c2)C1 ZINC000880560162 ED On-Demand Anodyne CCR2 41 38 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(C(F)(F)F)c2)C1 ZINC000880560162 ED On-Demand Anodyne EPHX2 20 45 COC(=O)[C@@]1(O)CCN([C@@H](C)c2nc(-c3cccs3)no2)C1 ZINC000880560163 DD On-Demand Anodyne ETHR 30 42 COC(=O)[C@@]1(O)CCN([C@H](C)c2nc(-c3cccs3)no2)C1 ZINC000880560166 DD On-Demand Anodyne ETHR 30 42 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccccc2Cl)C1 ZINC000880560189 ED On-Demand Anodyne KCNQ2 46 35 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccccc2Cl)C1 ZINC000880560190 ED On-Demand Anodyne KCNQ2 46 35 COc1cncc(NC(=O)N2CC[C@@H](N3CCCC3)C2)c1 ZINC000880560191 CD On-Demand Anodyne L3MBTL3 84 42 COc1cncc(NC(=O)N2CC[C@H](N3CCCC3)C2)c1 ZINC000880560192 CD On-Demand Anodyne L3MBTL3 84 42 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccsc3)CC2)c1 ZINC000880560203 FF On-Demand Anodyne NPBWR1 54 31 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C#N)cc2)C1 ZINC000880560211 DC On-Demand Mild HRH3 58 53 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C#N)cc2)C1 ZINC000880560211 DC On-Demand Mild MMP13 22 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C#N)cc2)C1 ZINC000880560211 DC On-Demand Mild MMP9 15 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(C#N)cc2)C1 ZINC000880560211 DC On-Demand Mild MEN1 51 42 COC(=O)[C@@]1(O)CCN(Cc2c(-c3ccccc3)nc3ccccn23)C1 ZINC000880560222 FE On-Demand Anodyne TSPO 16 48 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3cccc(C)c3)CC2)C1 ZINC000880560243 FC On-Demand Anodyne ADAM10 15 40 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne DRD2 15 46 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne LTA4H 48 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne HRH3 25 42 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne MMP13 25 45 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne ADAM17 19 44 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne MMP9 18 45 COC(=O)[C@@]1(O)CCN(CCOc2ccc(F)cc2)C1 ZINC000880560245 CC On-Demand Anodyne PSMB1 42 36 C/C=C\c1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560262 FD On-Demand Anodyne CCR1 42 37 C/C=C\c1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560262 FD On-Demand Anodyne ABCB1 47 38 C/C=C\c1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560263 FD On-Demand Anodyne CCR1 42 37 C/C=C\c1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560263 FD On-Demand Anodyne ABCB1 47 38 C/C=C/c1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560264 FD On-Demand Anodyne CCR1 42 37 C/C=C/c1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560264 FD On-Demand Anodyne ABCB1 47 38 C/C=C/c1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560265 FD On-Demand Anodyne CCR1 42 37 C/C=C/c1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)c(OC)c1 ZINC000880560265 FD On-Demand Anodyne ABCB1 47 38 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2cccc(C)c2)C1 ZINC000880560270 DC On-Demand Anodyne KCNK3 60 37 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2cccc(C)c2)C1 ZINC000880560270 DC On-Demand Anodyne KCNK9 49 35 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2cccc(C)c2)C1 ZINC000880560272 DC On-Demand Anodyne KCNK3 60 37 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2cccc(C)c2)C1 ZINC000880560272 DC On-Demand Anodyne KCNK9 49 35 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne DRD2 27 57 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne DRD1 17 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne DRD4 18 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne HTR2A 21 57 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne ADRA1B 15 43 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne DRD3 22 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne KCNH2 15 43 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne DRD5 15 54 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne LTA4H 22 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne HRH3 83 43 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne SIGMAR1 17 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne MMP13 26 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne HTR5A 19 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne ADAM17 17 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne MMP9 17 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(F)cc2)C1 ZINC000880560281 CD On-Demand Anodyne EPHX2 24 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(Cl)cccc2Cl)C1 ZINC000880560292 FD On-Demand Anodyne CCR1 43 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(Cl)cccc2Cl)C1 ZINC000880560292 FD On-Demand Anodyne ABCB1 63 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(Cl)cccc2Cl)C1 ZINC000880560293 FD On-Demand Anodyne CCR1 43 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(Cl)cccc2Cl)C1 ZINC000880560293 FD On-Demand Anodyne ABCB1 63 41 COc1cncc(NC(=O)N2CCN(CCN3[C@@H](C)CC[C@@H]3C)CC2)c1 ZINC000880560295 FE On-Demand Anodyne DRD4 42 32 COc1cncc(NC(=O)N2CCN(CCN3[C@@H](C)CC[C@@H]3C)CC2)c1 ZINC000880560295 FE On-Demand Anodyne PDGFRB 40 36 COc1cncc(NC(=O)N2CCN(CCN3[C@H](C)CC[C@H]3C)CC2)c1 ZINC000880560296 FE On-Demand Anodyne DRD4 42 32 COc1cncc(NC(=O)N2CCN(CCN3[C@H](C)CC[C@H]3C)CC2)c1 ZINC000880560296 FE On-Demand Anodyne PDGFRB 40 36 COc1cncc(NC(=O)N2CCN(CCN3[C@@H](C)CC[C@H]3C)CC2)c1 ZINC000880560297 FE On-Demand Anodyne DRD4 42 32 COc1cncc(NC(=O)N2CCN(CCN3[C@@H](C)CC[C@H]3C)CC2)c1 ZINC000880560297 FE On-Demand Anodyne PDGFRB 40 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560302 FD On-Demand Anodyne ACOX1 78 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560302 FD On-Demand Anodyne CCR1 44 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560302 FD On-Demand Anodyne ABCB1 77 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560305 FD On-Demand Anodyne ACOX1 78 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560305 FD On-Demand Anodyne CCR1 44 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(-c3ccccc3)cc2)C1 ZINC000880560305 FD On-Demand Anodyne ABCB1 77 45 COc1cncc(NC(=O)NCc2cccc(COC3CCOCC3)c2)c1 ZINC000880560306 FG On-Demand Anodyne ROCK2 39 46 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(CN3CCOCC3)cc2)C1 ZINC000880560308 GC On-Demand Anodyne EPHX2 18 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COCc2ccc(OC)cc2)C1 ZINC000880560311 EC On-Demand Anodyne MMP13 15 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COCc2ccc(OC)cc2)C1 ZINC000880560312 EC On-Demand Anodyne MMP13 15 40 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560314 GE On-Demand Anodyne KCNQ2 47 36 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560314 GE On-Demand Anodyne HCN1 58 34 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560314 GE On-Demand Anodyne HCN4 49 34 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560315 GE On-Demand Anodyne KCNQ2 47 36 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560315 GE On-Demand Anodyne HCN1 58 34 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560315 GE On-Demand Anodyne HCN4 49 34 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560316 GE On-Demand Anodyne KCNQ2 47 36 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560316 GE On-Demand Anodyne HCN1 58 34 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560316 GE On-Demand Anodyne HCN4 49 34 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560317 GE On-Demand Anodyne KCNQ2 47 36 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560317 GE On-Demand Anodyne HCN1 58 34 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560317 GE On-Demand Anodyne HCN4 49 34 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild HTR1A 52 52 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild DRD2 41 41 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild DRD4 43 37 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild HTR1D 16 52 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild HTR1B 20 52 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild DRD3 51 41 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild P2RY12 18 48 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild PDGFRB 59 46 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild HTR7 41 45 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild NPY2R 41 37 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild SSTR1 33 45 COc1cncc(NC(=O)N2CCN(c3ccccc3C#N)CC2)c1 ZINC000880560355 EE On-Demand Mild FAAH 19 46 CCCc1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880560365 CD On-Demand Anodyne MMP13 16 43 CCCc1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880560366 CD On-Demand Anodyne MMP13 16 43 COC(=O)[C@@]1(O)CCN(C[C@@H](O)CN(C)Cc2ccccc2)C1 ZINC000880560367 DC On-Demand Anodyne SLC12A5 42 35 COC(=O)[C@@]1(O)CCN(C[C@H](O)CN(C)Cc2ccccc2)C1 ZINC000880560368 DC On-Demand Anodyne SLC12A5 42 35 COc1ccc([C@@H]2CCN(C(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880560390 EG On-Demand Anodyne MMP13 15 41 COc1ccc([C@@H]2CCN(C(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880560390 EG On-Demand Anodyne MMP3 15 41 COc1ccc([C@@H]2CCN(C(=O)Nc3cncc(OC)c3)C2)cc1 ZINC000880560390 EG On-Demand Anodyne MMP1 16 41 COc1cncc(NC(=O)NCc2cc(OC)c(OC)cc2OC)c1 ZINC000880560393 EE On-Demand Anodyne PDGFRB 33 40 COc1cncc(NC(=O)NCc2cc(OC)c(OC)cc2OC)c1 ZINC000880560393 EE On-Demand Anodyne FLT4 17 40 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne PTAFR 22 43 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne SIGMAR1 15 44 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne MMP13 17 44 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne CHRNA7 49 40 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne FAAH 15 42 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne MMP9 15 44 COC(=O)[C@@]1(O)CCN(Cc2cccnc2)C1 ZINC000880560398 BC On-Demand Anodyne ACHP_LYMST 22 40 COC(=O)[C@@]1(O)CCN(Cc2ccn(-c3ccccc3)n2)C1 ZINC000880560401 DC On-Demand Anodyne SLC12A5 45 36 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne HTR1A 89 47 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne DRD2 65 45 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne DRD1 15 40 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne DRD4 51 41 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne HRH2 16 42 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne ADRA1D 43 42 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne HTR2A 60 51 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne HTR2C 43 46 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne SLC6A4 17 41 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne ADRA1A 45 42 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne ADRA1B 24 40 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne DRD3 92 48 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne HTR7 83 43 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne NPY1R 21 46 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne CCR3 52 51 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne CHRNA7 18 44 COc1cncc(NC(=O)NCCCN2CCN(c3ccncc3)CC2)c1 ZINC000880560402 FD On-Demand Anodyne QPCT 39 45 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne TSPO 40 31 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne MMP2 17 41 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne MMP3 21 41 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne ROCK2 33 40 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne NPY5R 34 42 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne MMP9 25 41 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne MMP12 16 41 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne MMP1 25 41 COc1cncc(NC(=O)N(Cc2ccccc2)C(C)C)c1 ZINC000880560412 CH On-Demand Anodyne PTGES 21 41 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)C2)c1 ZINC000880560419 CG On-Demand Anodyne EPHX2 32 44 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)C2)c1 ZINC000880560419 CG On-Demand Anodyne MCHR1 20 46 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)C2)c1 ZINC000880560419 CG On-Demand Anodyne ADAM10 29 43 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3)C2)c1 ZINC000880560419 CG On-Demand Anodyne SMO 22 43 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000880560420 CG On-Demand Anodyne EPHX2 32 44 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000880560420 CG On-Demand Anodyne MCHR1 20 46 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000880560420 CG On-Demand Anodyne ADAM10 29 43 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3)C2)c1 ZINC000880560420 CG On-Demand Anodyne SMO 22 43 COc1cncc(NC(=O)N2CCN(C(=O)c3c(F)cccc3Cl)CC2)c1 ZINC000880560426 GF On-Demand Anodyne FAAH 22 41 COc1cncc(NC(=O)N2CCN(C(=O)c3c(F)cccc3Cl)CC2)c1 ZINC000880560426 GF On-Demand Anodyne EPHX2 15 48 COc1cncc(NC(=O)N2CCN(C(=O)c3c(F)cccc3Cl)CC2)c1 ZINC000880560426 GF On-Demand Anodyne TYK2 24 40 CCOc1ccccc1NC(=O)[C@@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560436 ED On-Demand Anodyne HCN1 66 38 CCOc1ccccc1NC(=O)[C@@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560436 ED On-Demand Anodyne HCN4 52 38 CCOc1ccccc1NC(=O)[C@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560437 ED On-Demand Anodyne HCN1 66 38 CCOc1ccccc1NC(=O)[C@H](C)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880560437 ED On-Demand Anodyne HCN4 52 38 CCOc1ccccc1NC(=O)[C@@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560438 ED On-Demand Anodyne HCN1 66 38 CCOc1ccccc1NC(=O)[C@@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560438 ED On-Demand Anodyne HCN4 52 38 CCOc1ccccc1NC(=O)[C@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560439 ED On-Demand Anodyne HCN1 66 38 CCOc1ccccc1NC(=O)[C@H](C)N1CC[C@](O)(C(=O)OC)C1 ZINC000880560439 ED On-Demand Anodyne HCN4 52 38 CC[C@@H](C)c1ccc(NC(=O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880560444 ED On-Demand Anodyne SCN2A 15 41 CC[C@@H](C)c1ccc(NC(=O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880560445 ED On-Demand Anodyne SCN2A 15 41 COc1cncc(NC(=O)NC[C@H](O)C2CCCCC2)c1 ZINC000880560452 CE On-Demand Anodyne PRMT3 27 51 COc1cncc(NC(=O)NC[C@@H](O)C2CCCCC2)c1 ZINC000880560453 CE On-Demand Anodyne PRMT3 27 51 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880560455 EC On-Demand Anodyne RBP4 19 44 COc1cncc(NC(=O)N2CCN(Cc3cnc(C)s3)CC2)c1 ZINC000880560456 EE On-Demand Anodyne FAAH 17 45 COc1cncc(NC(=O)NCC2CCN(Cc3nc(C)c(C)o3)CC2)c1 ZINC000880560465 FF On-Demand Anodyne CCR3 38 42 COc1cncc(NC(=O)NCC2CCN(Cc3nc(C)c(C)o3)CC2)c1 ZINC000880560465 FF On-Demand Anodyne CACNA1I 59 36 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880560471 FD On-Demand Anodyne CPT1A 52 35 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880560471 FD On-Demand Anodyne CPT2 42 32 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880560471 FD On-Demand Anodyne RBP4 18 42 COc1cncc(NC(=O)N2CCC(c3nc(C)no3)CC2)c1 ZINC000880560473 DE On-Demand Anodyne SMO 38 53 COc1cncc(NC(=O)N2CCC(c3nc(C)no3)CC2)c1 ZINC000880560473 DE On-Demand Anodyne ETHR 48 38 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne CHRM2 15 44 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne DRD2 19 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne DRD4 44 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne SIGMAR1 73 42 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne FAAH 27 44 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne NPFFR1 43 38 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccccc3)CC2)C1 ZINC000880560486 FB On-Demand Anodyne SLC12A5 50 37 COC(=O)[C@@]1(O)CCN(C(c2ccccc2)c2ccccc2)C1 ZINC000880560487 DE On-Demand Anodyne OPRL1 41 55 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCOc2cccc(C)c2)C1 ZINC000880560488 FC On-Demand Anodyne MTNR1B 19 42 C=C(C)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880560489 DE On-Demand Mild EPHX2 43 41 C=C(C)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880560489 DE On-Demand Mild CXCR3 20 45 COc1cncc(NC(=O)N2CCC(CCN3CCOCC3)CC2)c1 ZINC000880560497 EE On-Demand Anodyne PDGFRB 37 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCOc2cccc(C)c2)C1 ZINC000880560501 FC On-Demand Anodyne MTNR1B 19 42 COc1cncc(NC(=O)N(Cc2ccccc2)CC2CCOCC2)c1 ZINC000880560502 FH On-Demand Anodyne CASR 26 41 COc1cncc(NC(=O)N(Cc2ccccc2)CC2CCOCC2)c1 ZINC000880560502 FH On-Demand Anodyne ROCK2 20 41 COc1cncc(NC(=O)N[C@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560507 FE On-Demand Anodyne CASR 50 47 COc1cncc(NC(=O)N[C@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560507 FE On-Demand Anodyne TACR2 15 47 COc1cncc(NC(=O)N[C@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560507 FE On-Demand Anodyne EPHX2 19 43 COc1cncc(NC(=O)N[C@@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560509 FE On-Demand Anodyne CASR 50 47 COc1cncc(NC(=O)N[C@@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560509 FE On-Demand Anodyne TACR2 15 47 COc1cncc(NC(=O)N[C@@H](CN2CCOCC2)c2ccccc2)c1 ZINC000880560509 FE On-Demand Anodyne EPHX2 19 43 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3)C2)c1 ZINC000880560510 DE On-Demand Anodyne CCR3 23 43 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3)C2)c1 ZINC000880560510 DE On-Demand Anodyne EPHX2 41 43 COc1cncc(NC(=O)N[C@@H]2CCN(c3ccccc3)C2)c1 ZINC000880560510 DE On-Demand Anodyne MCHR1 16 44 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3)C2)c1 ZINC000880560512 DE On-Demand Anodyne CCR3 23 43 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3)C2)c1 ZINC000880560512 DE On-Demand Anodyne EPHX2 41 43 COc1cncc(NC(=O)N[C@H]2CCN(c3ccccc3)C2)c1 ZINC000880560512 DE On-Demand Anodyne MCHR1 16 44 COc1cncc(NC(=O)N2CC[C@H](N3CCCCC3)C2)c1 ZINC000880560516 DE On-Demand Anodyne GALR2 44 32 COc1cncc(NC(=O)N2CC[C@H](N3CCCCC3)C2)c1 ZINC000880560516 DE On-Demand Anodyne L3MBTL3 83 41 COc1cncc(NC(=O)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000880560518 DE On-Demand Anodyne GALR2 44 32 COc1cncc(NC(=O)N2CC[C@@H](N3CCCCC3)C2)c1 ZINC000880560518 DE On-Demand Anodyne L3MBTL3 83 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560525 FD On-Demand Anodyne ACOX1 46 32 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560525 FD On-Demand Anodyne CCR1 60 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560525 FD On-Demand Anodyne ABCB1 53 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560529 FD On-Demand Anodyne ACOX1 46 32 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560529 FD On-Demand Anodyne CCR1 60 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)ccc2Cl)C1 ZINC000880560529 FD On-Demand Anodyne ABCB1 53 41 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880560543 FF On-Demand Anodyne ROCK1 28 42 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880560543 FF On-Demand Anodyne ROCK2 51 48 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2Cl)C1 ZINC000880560551 FD On-Demand Anodyne CCR1 77 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(Cl)cc2Cl)C1 ZINC000880560551 FD On-Demand Anodyne ABCB1 54 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2Cl)C1 ZINC000880560555 FD On-Demand Anodyne CCR1 77 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(Cl)cc2Cl)C1 ZINC000880560555 FD On-Demand Anodyne ABCB1 54 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC23CC4CC(CC(C4)C2)C3)C1 ZINC000880560564 FD On-Demand Anodyne EPHX2 47 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC23CC4CC(CC(C4)C2)C3)C1 ZINC000880560569 FD On-Demand Anodyne EPHX2 47 41 COc1cncc(NC(=O)NC[C@H]2CCCN(C)C2)c1 ZINC000880560571 CD On-Demand Anodyne CCR3 69 31 COc1cncc(NC(=O)NC[C@H]2CCCN(C)C2)c1 ZINC000880560571 CD On-Demand Anodyne CACNA1I 55 33 COc1cncc(NC(=O)NC[C@@H]2CCCN(C)C2)c1 ZINC000880560573 CD On-Demand Anodyne CCR3 69 31 COc1cncc(NC(=O)NC[C@@H]2CCCN(C)C2)c1 ZINC000880560573 CD On-Demand Anodyne CACNA1I 55 33 COc1cncc(NC(=O)NCCCCC#N)c1 ZINC000880560574 BD On-Demand Mild ADRB1 41 32 COc1cncc(NC(=O)N2CCN(Cc3cnn(C)c3)CC2)c1 ZINC000880560582 ED On-Demand Anodyne PDGFRB 44 34 COc1cncc(NC(=O)N2CCN(Cc3cnn(C)c3)CC2)c1 ZINC000880560582 ED On-Demand Anodyne FAAH 24 52 COc1cncc(NC(=O)N2CCC([C@H](O)c3ccc(F)cc3)CC2)c1 ZINC000880560584 FG On-Demand Anodyne S1PR2 28 42 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(Cl)cc3F)CC2)c1 ZINC000880560585 GF On-Demand Anodyne FAAH 18 40 COc1cncc(NC(=O)N2CCC([C@@H](O)c3ccc(F)cc3)CC2)c1 ZINC000880560586 FG On-Demand Anodyne S1PR2 28 42 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(Cl)c2)C1 ZINC000880560594 ED On-Demand Anodyne EPHX2 16 41 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(Cl)c2)C1 ZINC000880560594 ED On-Demand Anodyne MCHR1 32 44 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild HTR1A 40 49 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild HTR1B 17 49 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild P2RY12 15 45 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild PDGFRB 56 44 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild SSTR1 21 42 COc1cncc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c1 ZINC000880560596 FF On-Demand Mild TAAR1 18 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2F)C1 ZINC000880560599 DC On-Demand Anodyne ADRB2 23 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2F)C1 ZINC000880560599 DC On-Demand Anodyne CCR1 50 45 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2F)C1 ZINC000880560599 DC On-Demand Anodyne ABCB1 78 49 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2F)C1 ZINC000880560602 DC On-Demand Anodyne ADRB2 23 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2F)C1 ZINC000880560602 DC On-Demand Anodyne CCR1 50 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2F)C1 ZINC000880560602 DC On-Demand Anodyne ABCB1 78 49 COc1cncc(NC(=O)N(Cc2cccc(F)c2)C(C)C)c1 ZINC000880560610 DH On-Demand Anodyne ROCK1 20 41 COc1cncc(NC(=O)N(Cc2cccc(F)c2)C(C)C)c1 ZINC000880560610 DH On-Demand Anodyne ROCK2 33 56 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne ADRA1D 15 40 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne ADRA1A 32 40 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne ADRA1B 21 40 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne MMP13 24 44 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne CCR1 22 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne ADAM17 27 44 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2)C1 ZINC000880560614 EC On-Demand Anodyne MMP9 15 44 COc1cncc(NC(=O)N2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c1 ZINC000880560617 GF On-Demand Anodyne GRIN2B 25 42 COc1cncc(NC(=O)N2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c1 ZINC000880560617 GF On-Demand Anodyne HRH4 32 55 COc1cncc(NC(=O)N2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c1 ZINC000880560617 GF On-Demand Anodyne R1A_CVHSA 19 44 COc1cncc(NC(=O)N2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c1 ZINC000880560617 GF On-Demand Anodyne FPR2 23 43 COc1cncc(NC(=O)N2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)c1 ZINC000880560617 GF On-Demand Anodyne AKR1C3 19 45 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(CN3CCCC3)cc2)C1 ZINC000880560623 GC On-Demand Anodyne HRH3 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(CN3CCCC3)cc2)C1 ZINC000880560623 GC On-Demand Anodyne MCHR2 50 38 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(CN3CCCC3)cc2)C1 ZINC000880560623 GC On-Demand Anodyne NPFFR1 41 38 COc1cncc(NC(=O)NCCn2ccnc2C)c1 ZINC000880560624 CD On-Demand Anodyne QPCT 16 40 COc1cncc(NC(=O)N2CCN(CC(F)F)CC2)c1 ZINC000880560629 DD On-Demand Anodyne PDGFRB 46 36 COc1cncc(NC(=O)N2CCN(CC(F)F)CC2)c1 ZINC000880560629 DD On-Demand Anodyne S1PR2 27 40 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OC(C)C)C1 ZINC000880560631 CD On-Demand Anodyne CCR8 26 40 COc1cncc(NC(=O)NC2CCSCC2)c1 ZINC000880560637 CE On-Demand Anodyne EPHX2 49 36 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)F)cc2)C1 ZINC000880560640 DD On-Demand Anodyne MMP13 22 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)F)cc2)C1 ZINC000880560640 DD On-Demand Anodyne ADAM17 16 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(F)F)cc2)C1 ZINC000880560640 DD On-Demand Anodyne MMP9 18 44 COC(=O)[C@@]1(O)CCN(CCC(=O)N2CCN(c3ccccn3)CC2)C1 ZINC000880560643 FB On-Demand Anodyne DRD4 33 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(C)=O)c2)C1 ZINC000880560648 CC On-Demand Anodyne HTR1D 18 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(C)=O)c2)C1 ZINC000880560648 CC On-Demand Anodyne MCHR1 21 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(C)=O)c2)C1 ZINC000880560648 CC On-Demand Anodyne MCHR2 41 35 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(C)=O)c2)C1 ZINC000880560648 CC On-Demand Anodyne NPFFR1 41 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(C)=O)c2)C1 ZINC000880560648 CC On-Demand Anodyne SLC12A5 45 33 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCC(C)C)c2)C1 ZINC000880560654 ED On-Demand Anodyne DRD4 43 33 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCC(C)C)c2)C1 ZINC000880560654 ED On-Demand Anodyne HRH2 17 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCC(C)C)c2)C1 ZINC000880560654 ED On-Demand Anodyne CHRM3 17 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCC(C)C)c2)C1 ZINC000880560654 ED On-Demand Anodyne F3 68 35 COc1cncc(NC(=O)N2CCC[C@H]2c2nc3ccc(C)cc3[nH]2)c1 ZINC000880560670 FH On-Demand Anodyne PRCP 43 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2nc3ccc(C)cc3[nH]2)c1 ZINC000880560671 FH On-Demand Anodyne PRCP 43 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne DRD4 19 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne HRH2 41 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne SIGMAR1 43 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne MMP13 22 48 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne NPFFR2 28 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne ADAM17 44 49 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne FAAH 37 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne MMP9 17 48 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne MCHR2 50 33 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne FFAR1 39 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne CCR8 32 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne NPFFR1 39 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne SLC12A5 71 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccc3)c2)C1 ZINC000880560683 EE On-Demand Anodyne PDS 46 31 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne HRH2 29 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne DRD3 16 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne HRH3 41 43 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne EPHX2 27 52 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne GALR3 63 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880560689 EE On-Demand Anodyne PDS 45 42 COC(=O)[C@@]1(O)CCN(CC(=O)OCc2ccccc2)C1 ZINC000880560691 CC On-Demand Anodyne SIGMAR1 17 40 COC(=O)[C@@]1(O)CCN(CC(=O)OCc2ccccc2)C1 ZINC000880560691 CC On-Demand Anodyne CAPNS1 46 33 COC(=O)[C@@]1(O)CCN(CC(=O)OCc2ccccc2)C1 ZINC000880560691 CC On-Demand Anodyne SLC12A5 86 48 COc1cncc(NC(=O)N2CCCc3cc(OC)ccc3C2)c1 ZINC000880560707 EG On-Demand Anodyne CYP11B2 21 40 COc1cncc(NC(=O)N2CCCc3cc(OC)ccc3C2)c1 ZINC000880560707 EG On-Demand Anodyne MTNR1B 19 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2cccc(C(F)(F)F)c2)C1 ZINC000880560724 ED On-Demand Anodyne CCR2 44 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2cccc(C(F)(F)F)c2)C1 ZINC000880560729 ED On-Demand Anodyne CCR2 44 33 COc1cncc(NC(=O)NC2CCN(C(=O)Cc3ccccc3OC)CC2)c1 ZINC000880560737 GE On-Demand Anodyne SSTR5 26 40 COc1cncc(NC(=O)NC2CCN(C(=O)Cc3ccccc3OC)CC2)c1 ZINC000880560737 GE On-Demand Anodyne CCR3 32 44 COc1cncc(NC(=O)NC2CCN(C(=O)Cc3ccccc3OC)CC2)c1 ZINC000880560737 GE On-Demand Anodyne C3AR1 40 41 COc1cncc(NC(=O)NC2CCN(C(=O)Cc3ccccc3OC)CC2)c1 ZINC000880560737 GE On-Demand Anodyne EPHX2 60 54 COc1cncc(NC(=O)NC2CCN(C(=O)Cc3ccccc3OC)CC2)c1 ZINC000880560737 GE On-Demand Anodyne CCR8 20 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2c(C(C)C)cccc2C(C)C)C1 ZINC000880560747 FE On-Demand Anodyne SOAT1 65 46 COc1cncc(NC(=O)N(C)CCCOc2cccc(S(C)(=O)=O)c2)c1 ZINC000880560768 GE On-Demand Anodyne ROCK2 26 40 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne HTR1A 87 52 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne DRD2 72 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne DRD1 16 42 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne DRD4 51 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne HRH2 22 42 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne ADRA1D 37 40 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne HTR2A 46 49 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne HTR2C 29 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne ADRA1A 39 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne DRD3 97 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne HTR7 59 39 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne NPY1R 18 40 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne CCR3 40 46 COc1cncc(NC(=O)NCCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880560769 GD On-Demand Anodyne CHRNA7 22 49 COc1cncc(NC(=O)NCc2cccc(C(=O)NCCN(C)C)c2)c1 ZINC000880560773 FD On-Demand Anodyne DRD4 44 33 COc1cncc(NC(=O)NCc2cccc(C(=O)NCCN(C)C)c2)c1 ZINC000880560773 FD On-Demand Anodyne ROCK1 30 40 COc1cncc(NC(=O)NCc2cccc(C(=O)NCCN(C)C)c2)c1 ZINC000880560773 FD On-Demand Anodyne ROCK2 55 48 COCCN(CCCc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880560775 EG On-Demand Anodyne INHA 41 34 COCCN(CCCc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880560775 EG On-Demand Anodyne ROCK2 25 40 COCCN(CCCc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880560775 EG On-Demand Anodyne CRTM 40 36 COc1cncc(NC(=O)NCC(=O)NC2CCCC2)c1 ZINC000880560778 CD On-Demand Anodyne EPHX2 25 48 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000880560786 ED On-Demand Anodyne CCR8 40 41 COC(=O)[C@@]1(O)CCN(CCc2ccc3ccccc3c2)C1 ZINC000880560788 CD On-Demand Anodyne SIGMAR1 29 40 COC(=O)[C@@]1(O)CCN(CCc2ccc3ccccc3c2)C1 ZINC000880560788 CD On-Demand Anodyne MMP13 17 47 COC(=O)[C@@]1(O)CCN(CCc2ccc3ccccc3c2)C1 ZINC000880560788 CD On-Demand Anodyne ADAM17 16 47 COC(=O)[C@@]1(O)CCN(CCc2ccc3ccccc3c2)C1 ZINC000880560788 CD On-Demand Anodyne SLC12A5 55 36 COc1cncc(NC(=O)N(CCO)Cc2cc(Br)ccc2F)c1 ZINC000880560791 GG On-Demand Anodyne ROCK2 15 42 CC[C@H](C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1)c1ccccc1 ZINC000880560792 GG On-Demand Anodyne EPHX2 52 50 CC[C@H](C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1)c1ccccc1 ZINC000880560792 GG On-Demand Anodyne CXCR3 15 41 CC[C@@H](C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1)c1ccccc1 ZINC000880560793 GG On-Demand Anodyne EPHX2 52 50 CC[C@@H](C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1)c1ccccc1 ZINC000880560793 GG On-Demand Anodyne CXCR3 15 41 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne HTR1A 48 42 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne DRD2 39 42 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne DRD4 42 36 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne HTR1D 15 40 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne HTR1B 21 40 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne DRD3 54 39 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne HTR7 41 42 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne SCN2A 17 41 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne SOAT1 16 41 COc1cncc(NC(=O)NCc2ccccc2N2CCN(C(C)=O)CC2)c1 ZINC000880560795 GE On-Demand Anodyne SCN10A 32 41 COc1cncc(NC(=O)N(CCN(C)C)Cc2cccc(F)c2)c1 ZINC000880560803 EF On-Demand Anodyne ROCK1 24 58 COc1cncc(NC(=O)N(CCN(C)C)Cc2cccc(F)c2)c1 ZINC000880560803 EF On-Demand Anodyne ROCK2 37 58 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccc(C)cc3)CC2)c1 ZINC000880560804 FE On-Demand Anodyne PDGFRB 44 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)c(Br)c2)C1 ZINC000880560805 ED On-Demand Anodyne MMP13 15 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)c(Br)c2)C1 ZINC000880560805 ED On-Demand Anodyne MCHR2 46 34 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(C(F)(F)F)cc2)C1 ZINC000880560811 FD On-Demand Anodyne EPHX2 40 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(C(F)(F)F)cc2)C1 ZINC000880560811 FD On-Demand Anodyne TRPM8 45 39 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(C(F)(F)F)cc2)C1 ZINC000880560812 FD On-Demand Anodyne EPHX2 40 43 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(C(F)(F)F)cc2)C1 ZINC000880560812 FD On-Demand Anodyne TRPM8 45 39 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCc3ccco3)c2)C1 ZINC000880560813 FD On-Demand Anodyne DRD4 40 31 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)NCc3ccco3)c2)C1 ZINC000880560813 FD On-Demand Anodyne CHRM3 17 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne EDNRB 65 39 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne EDNRA 67 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne BMP1 42 33 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne HRH3 56 49 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne MMP13 15 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3c(c2)OCO3)C1 ZINC000880560816 DC On-Demand Anodyne EPHX2 18 47 COc1cncc(NC(=O)N2CCC(C(=O)NCCc3cccs3)CC2)c1 ZINC000880560825 GF On-Demand Anodyne MTNR1A 22 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne HTR1A 25 44 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne DRD2 27 44 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne DRD4 42 34 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne HRH2 37 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne HTR2A 24 44 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne ADRA1A 16 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne DRD3 31 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne AVPR1B 49 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne HTR7 22 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne HRH3 58 44 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne SIGMAR1 21 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne MMP13 15 44 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne CCR1 33 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne EBP 21 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(Cl)c2)C1 ZINC000880560827 DD On-Demand Anodyne EPHX2 26 44 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)cc3Cl)CC2)c1 ZINC000880560830 GF On-Demand Anodyne P2RX7 27 49 CCOc1ccccc1C(F)(F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880560845 FF On-Demand Anodyne HCN1 43 36 CCOc1ccccc1C(F)(F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880560845 FF On-Demand Anodyne HCN4 43 36 COc1cncc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880560857 FE On-Demand Anodyne ACACB 15 40 COc1cncc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880560857 FE On-Demand Anodyne CACNA1I 53 34 COc1cncc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880560859 FE On-Demand Anodyne ACACB 15 40 COc1cncc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880560859 FE On-Demand Anodyne CACNA1I 53 34 C/C(=C/C(=O)NCc1cn(C2CCC2)nn1)c1cccc(Cl)c1 ZINC000880560865 EG On-Demand Anodyne CACNA1I 42 38 C/C(=C\C(=O)NCc1cn(C2CCC2)nn1)c1cccc(Cl)c1 ZINC000880560866 EG On-Demand Anodyne CACNA1I 42 38 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccccc2)c2ccccc2)C1 ZINC000880560874 FD On-Demand Anodyne NPY2R 30 43 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccccc2)c2ccccc2)C1 ZINC000880560879 FD On-Demand Anodyne NPY2R 30 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2)C1 ZINC000880560892 CB On-Demand Anodyne SIGMAR1 23 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2)C1 ZINC000880560892 CB On-Demand Anodyne NPFFR1 43 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2)C1 ZINC000880560892 CB On-Demand Anodyne SLC12A5 66 41 COc1cncc(NC(=O)N2CCN(C(=O)C3CC3)CC2)c1 ZINC000880560898 DD On-Demand Anodyne PDGFRB 50 39 COc1cncc(NC(=O)NCCCS(=O)(=O)c2ccccc2)c1 ZINC000880560907 EE On-Demand Anodyne BMP1 24 45 COc1cncc(NC(=O)NCCCS(=O)(=O)c2ccccc2)c1 ZINC000880560907 EE On-Demand Anodyne QPCT 15 40 COc1cncc(NC(=O)NCCCS(=O)(=O)c2ccccc2)c1 ZINC000880560907 EE On-Demand Anodyne NAMPT 45 45 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3CC2)c1 ZINC000880560916 FF On-Demand Anodyne HTR2C 15 40 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3CC2)c1 ZINC000880560916 FF On-Demand Anodyne PDGFRB 45 40 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3CC2)c1 ZINC000880560916 FF On-Demand Anodyne CYP11B2 16 41 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3CC2)c1 ZINC000880560916 FF On-Demand Anodyne ABCB1 18 42 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3F)CC2)c1 ZINC000880560938 FE On-Demand Anodyne PDGFRB 42 38 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3F)CC2)c1 ZINC000880560938 FE On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3F)CC2)c1 ZINC000880560938 FE On-Demand Anodyne FAAH 21 44 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3F)CC2)c1 ZINC000880560938 FE On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N2CCC(C(=O)NC3CCCCC3)CC2)c1 ZINC000880560944 FF On-Demand Anodyne EPHX2 39 49 COc1cncc(NC(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000880560950 EH On-Demand Anodyne ROCK1 21 51 COc1cncc(NC(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000880560950 EH On-Demand Anodyne ROCK2 34 51 COc1cncc(NC(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000880560950 EH On-Demand Anodyne SCD1 20 42 COc1cncc(NC(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000880560950 EH On-Demand Anodyne SCD 32 42 COc1cncc(NC(=O)N2CCN(C(=O)N3CCCC3)CC2)c1 ZINC000880560952 ED On-Demand Anodyne PDGFRB 45 38 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(c3ccccc3OC)C2=O)C1 ZINC000880560955 EC On-Demand Anodyne HTR1A 41 39 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(Cl)cc2)C1 ZINC000880560956 CE On-Demand Anodyne CCR1 46 34 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(Cl)cc2)C1 ZINC000880560957 CE On-Demand Anodyne CCR1 46 34 COC(=O)[C@@]1(O)CCN([C@H]2CCN(c3ccccc3OC)C2=O)C1 ZINC000880560966 EC On-Demand Anodyne HTR1A 41 39 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne PIK3CA 31 41 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne ROCK2 17 40 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne MTOR 61 39 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne EPHX2 26 47 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne PIK3CG 32 41 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000880560969 FD On-Demand Anodyne NAMPT 49 47 COC(=O)[C@@]1(O)CCN(CCOc2cccc3ccccc23)C1 ZINC000880560974 DD On-Demand Anodyne HTR1A 24 42 COC(=O)[C@@]1(O)CCN(CCOc2cccc3ccccc23)C1 ZINC000880560974 DD On-Demand Anodyne HTR1B 17 41 COC(=O)[C@@]1(O)CCN(CCOc2cccc3ccccc23)C1 ZINC000880560974 DD On-Demand Anodyne ALB 24 40 COC(=O)[C@@]1(O)CCN(CCOc2cccc3ccccc23)C1 ZINC000880560974 DD On-Demand Anodyne MCL1 42 43 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C#N)C1 ZINC000880560980 CC On-Demand Mild ADRB1 41 32 CC(C)(C)OC(=O)N1CCC[C@H](OCC(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880560982 GE On-Demand Anodyne PREP 15 45 CC(C)(C)OC(=O)N1CCC[C@@H](OCC(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880560983 GE On-Demand Anodyne PREP 15 45 COc1ccc(OC2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880560986 FG On-Demand Anodyne PDGFRB 40 37 COc1ccc(OC2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880560986 FG On-Demand Anodyne PRSS2 57 32 COc1ccc(OC2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880560986 FG On-Demand Anodyne EPHX2 40 39 COc1ccc(OC2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880560986 FG On-Demand Anodyne SCD1 25 50 COC(=O)[C@@]1(O)CCN(CC(=O)NC2CCN(Cc3ccccc3C)CC2)C1 ZINC000880560991 GC On-Demand Anodyne DRD4 24 51 COC(=O)[C@@]1(O)CCN(CC(=O)NC2CCN(Cc3ccccc3C)CC2)C1 ZINC000880560991 GC On-Demand Anodyne SIGMAR1 22 49 COC(=O)[C@@]1(O)CCN(CC(=O)NC2CCN(Cc3ccccc3C)CC2)C1 ZINC000880560991 GC On-Demand Anodyne MCHR1 17 41 COC(=O)[C@@]1(O)CCN(CC(=O)NC2CCN(Cc3ccccc3C)CC2)C1 ZINC000880560991 GC On-Demand Anodyne CCR8 35 40 COc1cncc(NC(=O)N(Cc2cccnc2)C2CC2)c1 ZINC000880560996 CF On-Demand Anodyne CHRNA7 51 45 COc1cncc(NC(=O)N(Cc2cccnc2)C2CC2)c1 ZINC000880560996 CF On-Demand Anodyne ROCK2 33 55 COc1cncc(NC(=O)NC2(c3ccccc3)CC2)c1 ZINC000880560998 CF On-Demand Anodyne EPHX2 15 43 COc1cncc(NC(=O)N2CCN(C(=O)C(=O)N3CCCC3)CC2)c1 ZINC000880561002 FC On-Demand Anodyne PDGFRB 46 38 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3C)CC2)c1 ZINC000880561008 FE On-Demand Anodyne PDGFRB 45 39 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3C)CC2)c1 ZINC000880561008 FE On-Demand Anodyne FAAH 15 44 COc1cncc(NC(=O)N2CCN(C(=O)Cc3ccccc3C)CC2)c1 ZINC000880561008 FE On-Demand Anodyne P2RY14 42 33 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(C(F)(F)F)c2)C1 ZINC000880561021 FD On-Demand Anodyne EPHX2 23 43 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561026 GH On-Demand Anodyne CCR3 19 42 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561026 GH On-Demand Anodyne CPT1A 33 40 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561026 GH On-Demand Anodyne GRM5 19 61 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561026 GH On-Demand Anodyne SMO 36 47 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne HRH2 28 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne SIGMAR1 15 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne MMP13 15 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne ADAM17 15 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne FAAH 24 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(C)C)c2)C1 ZINC000880561030 CD On-Demand Anodyne CCR8 26 40 COc1cncc(NC(=O)NCC(=O)N2CCCCC2)c1 ZINC000880561039 CD On-Demand Anodyne PRMT3 19 49 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561041 GH On-Demand Anodyne CCR3 19 42 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561041 GH On-Demand Anodyne CPT1A 33 40 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561041 GH On-Demand Anodyne GRM5 19 61 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4ccc(F)cc4)no3)C2)c1 ZINC000880561041 GH On-Demand Anodyne SMO 36 47 COC(=O)[C@@]1(O)CCN(Cc2nccn2Cc2ccccc2)C1 ZINC000880561047 DD On-Demand Anodyne MMP13 15 40 COC(=O)[C@@]1(O)CCN(Cc2nccn2Cc2ccccc2)C1 ZINC000880561047 DD On-Demand Anodyne SLC12A5 60 37 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne HTR1A 83 48 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne DRD2 72 53 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne DRD4 44 45 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne ADRA1D 79 53 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne HTR1D 16 48 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne HTR1B 20 48 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne ADRA1A 70 53 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne ADRA1B 62 53 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne DRD3 74 43 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne HTR7 54 40 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne SSTR5 29 40 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne NPY1R 23 43 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne EPHX2 46 45 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne PDGFRA 29 41 COc1cncc(NC(=O)NC2CCN(c3ccccc3OC)CC2)c1 ZINC000880561066 FF On-Demand Anodyne CXCR3 16 42 COc1cncc(NC(=O)NCc2ccccc2OCCN(C)C)c1 ZINC000880561070 EE On-Demand Anodyne ROCK2 37 49 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne HTR1A 42 43 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne DRD4 21 47 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne HTR2A 23 45 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne DRD3 42 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne SIGMAR1 15 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne HTR5A 17 45 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne EBP 30 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc3ccccc23)C1 ZINC000880561074 EE On-Demand Anodyne MCL1 47 46 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561089 EC On-Demand Anodyne DRD4 41 32 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561089 EC On-Demand Anodyne MTNR1A 42 39 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561089 EC On-Demand Anodyne MTNR1B 40 39 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561089 EC On-Demand Anodyne ROCK2 35 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561089 EC On-Demand Anodyne CARM1 34 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561092 EC On-Demand Anodyne DRD4 41 32 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561092 EC On-Demand Anodyne MTNR1A 42 39 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561092 EC On-Demand Anodyne MTNR1B 40 39 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561092 EC On-Demand Anodyne ROCK2 35 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2cccc(OC)c2)C1 ZINC000880561092 EC On-Demand Anodyne CARM1 34 40 COC(=O)[C@@]1(O)CCN(CC[S@@](=O)c2ccccc2)C1 ZINC000880561094 CC On-Demand Anodyne SLC12A5 42 36 COc1ccc(C(=O)N2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561099 FE On-Demand Anodyne PDGFRB 54 42 COc1ccc(C(=O)N2CCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561099 FE On-Demand Anodyne FAAH 17 46 COC(=O)[C@@]1(O)CCN(CC[S@](=O)c2ccccc2)C1 ZINC000880561100 CC On-Demand Anodyne SLC12A5 42 36 COc1cncc(NC(=O)NCCC(=O)N2CCCCCC2)c1 ZINC000880561107 DE On-Demand Anodyne HRH2 19 43 CCOc1ccccc1OCCN1CC[C@@](O)(C(=O)OC)C1 ZINC000880561115 DD On-Demand Anodyne HTR7 18 44 CCOc1ccccc1OCCN1CC[C@@](O)(C(=O)OC)C1 ZINC000880561115 DD On-Demand Anodyne HCN1 65 39 CCOc1ccccc1OCCN1CC[C@@](O)(C(=O)OC)C1 ZINC000880561115 DD On-Demand Anodyne HCN4 54 38 COc1cncc(NC(=O)NC(C)(C)c2ccccc2OC)c1 ZINC000880561116 DG On-Demand Anodyne IMDH_CRYPV 56 42 CCOc1ccccc1OCCN1CC[C@](O)(C(=O)OC)C1 ZINC000880561117 DD On-Demand Anodyne HTR7 18 44 CCOc1ccccc1OCCN1CC[C@](O)(C(=O)OC)C1 ZINC000880561117 DD On-Demand Anodyne HCN1 65 39 CCOc1ccccc1OCCN1CC[C@](O)(C(=O)OC)C1 ZINC000880561117 DD On-Demand Anodyne HCN4 54 38 COc1cncc(NC(=O)N(C)[C@H](C)c2cccnc2)c1 ZINC000880561118 CF On-Demand Anodyne KCNA5 22 44 COc1cncc(NC(=O)N(C)[C@@H](C)c2cccnc2)c1 ZINC000880561121 CF On-Demand Anodyne KCNA5 22 44 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3C#N)CC2)c1 ZINC000880561128 FE On-Demand Mild DRD4 43 34 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3C#N)CC2)c1 ZINC000880561128 FE On-Demand Mild HTR1B 15 48 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3C#N)CC2)c1 ZINC000880561128 FE On-Demand Mild PDGFRB 47 40 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3C#N)CC2)c1 ZINC000880561128 FE On-Demand Mild SSTR1 21 48 COc1cncc(NC(=O)N2CCN(c3cccc(F)c3C#N)CC2)c1 ZINC000880561128 FE On-Demand Mild FAAH 17 41 COC(=O)[C@@]1(O)CCN(CCCOCCc2ccccc2)C1 ZINC000880561140 DD On-Demand Anodyne ADRA1B 20 40 COC(=O)[C@@]1(O)CCN(CCCOCCc2ccccc2)C1 ZINC000880561140 DD On-Demand Anodyne SLC6A3 15 43 COC(=O)[C@@]1(O)CCN(CCCOCCc2ccccc2)C1 ZINC000880561140 DD On-Demand Anodyne HRH3 18 46 COC(=O)[C@@]1(O)CCN(CCCOCCc2ccccc2)C1 ZINC000880561140 DD On-Demand Anodyne SIGMAR1 51 43 COC(=O)[C@@]1(O)CCN(CCCOCCc2ccccc2)C1 ZINC000880561140 DD On-Demand Anodyne SLC12A5 70 39 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc3ccccc3c2)C1 ZINC000880561159 CF On-Demand Anodyne CYP26A1 70 38 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc3ccccc3c2)C1 ZINC000880561162 CF On-Demand Anodyne CYP26A1 70 38 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CCCC2)C1 ZINC000880561165 FD On-Demand Anodyne KCNA3 52 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CCCC2)C1 ZINC000880561165 FD On-Demand Anodyne NPFFR1 39 44 COc1cncc(NC(=O)N[C@@H](C)C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561170 GF On-Demand Anodyne TAAR1 30 40 COc1cncc(NC(=O)N[C@H](C)C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561172 GF On-Demand Anodyne TAAR1 30 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561195 EC On-Demand Anodyne HTR7 16 49 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561195 EC On-Demand Anodyne BDKRB1 59 43 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561195 EC On-Demand Anodyne XIAP 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561195 EC On-Demand Anodyne BIRC3 27 41 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561195 EC On-Demand Anodyne BIRC2 41 38 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561196 EC On-Demand Anodyne HTR7 16 49 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561196 EC On-Demand Anodyne BDKRB1 59 43 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561196 EC On-Demand Anodyne XIAP 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561196 EC On-Demand Anodyne BIRC3 27 41 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561196 EC On-Demand Anodyne BIRC2 41 38 COc1cncc(NC(=O)N(CCN(C)C)Cc2cccc(C)c2)c1 ZINC000880561202 EF On-Demand Anodyne ROCK1 24 58 COc1cncc(NC(=O)N(CCN(C)C)Cc2cccc(C)c2)c1 ZINC000880561202 EF On-Demand Anodyne ROCK2 38 58 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(F)c(F)c2)C1 ZINC000880561203 EC On-Demand Anodyne CACNA1H 15 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(F)c(F)c2)C1 ZINC000880561205 EC On-Demand Anodyne CACNA1H 15 41 COc1cncc(NC(=O)N2CCN(CCCOCC(F)(F)F)CC2)c1 ZINC000880561215 GE On-Demand Anodyne PDGFRB 41 39 COC(=O)[C@@]1(O)CCN(CCCC2CCCC2)C1 ZINC000880561219 CD On-Demand Anodyne EBP 22 51 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccc(OCC(F)(F)F)c2)C1 ZINC000880561223 GC On-Demand Anodyne PDS 50 35 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C2CC2)C1 ZINC000880561235 EC On-Demand Anodyne OPRM1 15 44 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C2CC2)C1 ZINC000880561235 EC On-Demand Anodyne SIGMAR1 24 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C2CC2)C1 ZINC000880561235 EC On-Demand Anodyne CCR5 53 40 COC(=O)[C@@]1(O)CCN(CC(=O)N(Cc2ccccc2)C2CC2)C1 ZINC000880561235 EC On-Demand Anodyne SLC12A5 58 36 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561248 DC On-Demand Anodyne ANPEP 20 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561248 DC On-Demand Anodyne AMP1_PLAFQ 39 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561248 DC On-Demand Anodyne SLC12A5 58 37 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561250 DC On-Demand Anodyne ANPEP 20 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561250 DC On-Demand Anodyne AMP1_PLAFQ 39 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCc2ccccc2)C1 ZINC000880561250 DC On-Demand Anodyne SLC12A5 58 37 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CCOCC2)C1 ZINC000880561262 GC On-Demand Anodyne KCNA3 49 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CCOCC2)C1 ZINC000880561262 GC On-Demand Anodyne NPFFR1 28 42 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne HTR2A 26 44 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne TNF 35 43 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne PDGFRB 25 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne CASR 31 41 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne TACR2 15 44 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne MAPK14 18 44 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne SRC 27 42 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne KDR 18 45 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne ROCK2 19 45 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne ABCB1 15 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne MAPK9 15 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne MAP2K1 21 43 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne EPHX2 34 46 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne FLT3 25 45 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne MAPK12 20 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne AURKA 24 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne STK10 22 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne EPHA2 15 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne EPHA8 16 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne EPHA5 18 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne EPHA4 17 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne TIE1 20 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne DDR2 19 40 COc1cncc(NC(=O)NCc2ccccc2OCCN2CCOCC2)c1 ZINC000880561271 GE On-Demand Anodyne CDK8 22 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)F)c2)C1 ZINC000880561274 DD On-Demand Anodyne SIGMAR1 18 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)F)c2)C1 ZINC000880561274 DD On-Demand Anodyne CCR8 26 40 COc1cncc(NC(=O)NCc2ccc3c(c2)CCO3)c1 ZINC000880561275 CE On-Demand Anodyne ROCK2 25 43 COc1cncc(NC(=O)NC[C@H]2CCN(C(C)C)C2)c1 ZINC000880561276 CD On-Demand Anodyne CCR3 42 38 COc1cncc(NC(=O)NC[C@H]2CCN(C(C)C)C2)c1 ZINC000880561276 CD On-Demand Anodyne CACNA1I 41 35 COc1cncc(NC(=O)NC[C@@H]2CCN(C(C)C)C2)c1 ZINC000880561277 CD On-Demand Anodyne CCR3 42 38 COc1cncc(NC(=O)NC[C@@H]2CCN(C(C)C)C2)c1 ZINC000880561277 CD On-Demand Anodyne CACNA1I 41 35 COC(=O)[C@@]1(O)CCN(Cc2cnc(C)s2)C1 ZINC000880561278 CC On-Demand Anodyne MGEA5 33 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne LTA4H 22 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne SIGMAR1 18 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne MMP13 27 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne CHRNA7 43 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne ADAM17 39 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne FAAH 32 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne SLC6A5 24 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne MMP9 23 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccnc3)cc2)C1 ZINC000880561285 ED On-Demand Anodyne MMP1 17 46 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne LTA4H 40 51 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne MMP13 23 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne MMP14 15 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne MMP9 20 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne EPHX2 21 46 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C(F)(F)F)cc2)C1 ZINC000880561291 ED On-Demand Anodyne PSMB1 41 42 COc1cncc(NC(=O)N2CCN(c3cccnn3)CC2)c1 ZINC000880561310 DD On-Demand Anodyne PDGFRB 51 43 COc1cncc(NC(=O)N2CCN(C(=O)COc3ccc(C)cc3)CC2)c1 ZINC000880561311 GE On-Demand Anodyne PDGFRB 52 44 COc1cncc(NC(=O)NCc2ccc(N(C)C)c(F)c2)c1 ZINC000880561329 DF On-Demand Clean ROCK2 29 47 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880561337 ED On-Demand Anodyne ADRB2 28 45 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880561337 ED On-Demand Anodyne ADRB1 56 41 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880561337 ED On-Demand Anodyne ADRB3 27 44 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880561337 ED On-Demand Anodyne PDS 33 40 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880561338 ED On-Demand Anodyne ADRB2 28 45 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880561338 ED On-Demand Anodyne ADRB1 56 41 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880561338 ED On-Demand Anodyne ADRB3 27 44 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880561338 ED On-Demand Anodyne PDS 33 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccn3)cc2)C1 ZINC000880561357 ED On-Demand Anodyne SIGMAR1 17 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccn3)cc2)C1 ZINC000880561357 ED On-Demand Anodyne MMP13 19 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccn3)cc2)C1 ZINC000880561357 ED On-Demand Anodyne ADAM17 36 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccn3)cc2)C1 ZINC000880561357 ED On-Demand Anodyne FAAH 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccn3)cc2)C1 ZINC000880561357 ED On-Demand Anodyne MMP9 15 46 COC(=O)[C@@]1(O)CCN(CCOc2ccc(C#N)cc2OC)C1 ZINC000880561365 DC On-Demand Mild PDGFRB 15 45 COc1ccc(N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561373 FF On-Demand Clean EPHX2 51 42 COc1ccc(N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561373 FF On-Demand Clean PDK1 45 32 COc1ccc(N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561373 FF On-Demand Clean CXCR3 15 42 COc1ccc(N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561373 FF On-Demand Clean MCHR1 18 44 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc3c(c2)OCO3)c1 ZINC000880561379 EG On-Demand Anodyne EDNRB 75 42 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc3c(c2)OCO3)c1 ZINC000880561379 EG On-Demand Anodyne EDNRA 72 53 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc3c(c2)OCO3)c1 ZINC000880561381 EG On-Demand Anodyne EDNRB 75 42 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc3c(c2)OCO3)c1 ZINC000880561381 EG On-Demand Anodyne EDNRA 72 53 COc1cncc(NC(=O)NCCOC2CCCCC2)c1 ZINC000880561386 CF On-Demand Anodyne ADRB1 15 49 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(Cl)c2)C1 ZINC000880561390 FC On-Demand Anodyne DRD4 42 33 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(Cl)c2)C1 ZINC000880561390 FC On-Demand Anodyne HRH2 29 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(Cl)c2)C1 ZINC000880561390 FC On-Demand Anodyne AVPR1B 45 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000880561403 CB On-Demand Anodyne NPFFR1 45 44 COc1cncc(NC(=O)NCCCOc2ccccc2OC)c1 ZINC000880561407 EF On-Demand Anodyne ADRB1 44 34 COc1cncc(NC(=O)NCCCOc2ccccc2OC)c1 ZINC000880561407 EF On-Demand Anodyne HRH2 24 45 COc1cncc(NC(=O)NCCCOc2ccccc2OC)c1 ZINC000880561407 EF On-Demand Anodyne PDGFRA 43 35 COc1cncc(NC(=O)NCCCOc2ccccc2OC)c1 ZINC000880561407 EF On-Demand Anodyne QPCT 26 48 COc1cncc(NC(=O)NCCCOc2ccccc2OC)c1 ZINC000880561407 EF On-Demand Anodyne KCNK3 41 37 COC(=O)[C@@]1(O)CCN(CCCSc2ccccc2Cl)C1 ZINC000880561410 EE On-Demand Anodyne ADRA1A 15 41 COc1cncc(NC(=O)N[C@H](c2nc3ccccc3[nH]2)C(C)C)c1 ZINC000880561415 EG On-Demand Anodyne HPSE 22 41 COc1cncc(NC(=O)N[C@@H](c2nc3ccccc3[nH]2)C(C)C)c1 ZINC000880561416 EG On-Demand Anodyne HPSE 22 41 COc1cncc(NC(=O)NCC(=O)NC2CCCCC2)c1 ZINC000880561423 DD On-Demand Anodyne EPHX2 28 50 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561432 ED On-Demand Anodyne HTR7 18 54 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561432 ED On-Demand Anodyne SIGMAR1 17 42 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@H]2CCCc3ccccc32)C1 ZINC000880561432 ED On-Demand Anodyne BDKRB1 50 40 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561433 ED On-Demand Anodyne HTR7 18 54 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561433 ED On-Demand Anodyne SIGMAR1 17 42 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@@H]2CCCc3ccccc32)C1 ZINC000880561433 ED On-Demand Anodyne BDKRB1 50 40 COc1cncc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)c1 ZINC000880561437 EE On-Demand Anodyne PDGFRB 55 46 COc1cncc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)c1 ZINC000880561437 EE On-Demand Anodyne FAAH 25 42 COc1cncc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)c1 ZINC000880561437 EE On-Demand Anodyne RBP4 18 42 COc1cncc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)c1 ZINC000880561437 EE On-Demand Anodyne DGAT1 32 46 COc1cncc(NC(=O)N2CCN(c3ccc(Cl)cn3)CC2)c1 ZINC000880561437 EE On-Demand Anodyne NPBWR1 42 42 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)c1 ZINC000880561440 FF On-Demand Anodyne ROCK2 20 42 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)c1 ZINC000880561440 FF On-Demand Anodyne L3MBTL3 43 33 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)c1 ZINC000880561440 FF On-Demand Anodyne NAMPT 58 57 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3OC)CC2)c1 ZINC000880561442 GF On-Demand Anodyne PDGFRB 42 39 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3OC)CC2)c1 ZINC000880561442 GF On-Demand Anodyne RBP4 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)c2cn(CCC#N)c3ccccc23)C1 ZINC000880561449 FD On-Demand Mild CNR1 16 43 COC(=O)[C@@]1(O)CCN(CC(=O)c2cn(CCC#N)c3ccccc23)C1 ZINC000880561449 FD On-Demand Mild CNR2 23 43 COc1ccc(N2CCCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561460 FF On-Demand Clean PDGFRB 54 42 COc1ccc(N2CCCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561460 FF On-Demand Clean FAAH 15 45 COc1ccc(N2CCCN(C(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561460 FF On-Demand Clean GALR2 40 34 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne EDNRB 17 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne TACR1 26 47 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne NQO2 18 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne CCKAR 52 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne BRS3 27 42 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne NMBR 64 33 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne MC5R 32 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne MTNR1A 28 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne MTNR1B 19 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne GRPR 54 31 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne ECE1 48 36 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne MMP11 48 31 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne CCKBR 65 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne GHSR 54 37 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne MMP9 18 46 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne AANAT 54 33 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561461 FC On-Demand Anodyne KISS1R 53 32 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne EDNRB 17 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne TACR1 26 47 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne NQO2 18 43 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne CCKAR 52 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne BRS3 27 42 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne NMBR 64 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne MC5R 32 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne MTNR1A 28 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne MTNR1B 19 43 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne GRPR 54 31 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne ECE1 48 36 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne MMP11 48 31 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne CCKBR 65 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne GHSR 54 37 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne MMP9 18 46 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne AANAT 54 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2c[nH]c3ccccc23)C1 ZINC000880561463 FC On-Demand Anodyne KISS1R 53 32 COc1cncc(NC(=O)N[C@H](C)COc2ccccc2)c1 ZINC000880561467 DF On-Demand Anodyne ADRB1 16 43 COc1cncc(NC(=O)N[C@H](C)COc2ccccc2)c1 ZINC000880561467 DF On-Demand Anodyne MTNR1A 17 50 COc1cncc(NC(=O)N[C@H](C)COc2ccccc2)c1 ZINC000880561467 DF On-Demand Anodyne MTNR1B 22 50 COc1cncc(NC(=O)N[C@H](C)COc2ccccc2)c1 ZINC000880561467 DF On-Demand Anodyne PDS 48 36 COc1cncc(NC(=O)N[C@@H](C)COc2ccccc2)c1 ZINC000880561469 DF On-Demand Anodyne ADRB1 16 43 COc1cncc(NC(=O)N[C@@H](C)COc2ccccc2)c1 ZINC000880561469 DF On-Demand Anodyne MTNR1A 17 50 COc1cncc(NC(=O)N[C@@H](C)COc2ccccc2)c1 ZINC000880561469 DF On-Demand Anodyne MTNR1B 22 50 COc1cncc(NC(=O)N[C@@H](C)COc2ccccc2)c1 ZINC000880561469 DF On-Demand Anodyne PDS 48 36 COCCN(Cc1ccc(C#N)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880561473 EF On-Demand Mild ROCK2 17 40 COC(=O)[C@@]1(O)CCN([C@H](C(=O)NCc2ccccc2)c2ccccc2)C1 ZINC000880561474 FD On-Demand Anodyne SLC12A5 46 36 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)NCc2ccccc2)c2ccccc2)C1 ZINC000880561477 FD On-Demand Anodyne SLC12A5 46 36 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880561481 EI On-Demand Anodyne UL80 25 40 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880561481 EI On-Demand Anodyne CCR1 17 46 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880561481 EI On-Demand Anodyne SCN10A 34 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880561482 EI On-Demand Anodyne UL80 25 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880561482 EI On-Demand Anodyne CCR1 17 46 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880561482 EI On-Demand Anodyne SCN10A 34 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)N(C)Cc2ccccc2)C1 ZINC000880561485 DC On-Demand Anodyne SLC12A5 63 38 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)N(C)Cc2ccccc2)C1 ZINC000880561488 DC On-Demand Anodyne SLC12A5 63 38 COc1cncc(NC(=O)N(Cc2ccccc2F)C(C)C)c1 ZINC000880561497 DH On-Demand Anodyne COLA 21 40 O=C(NCc1cn(C2CCC2)nn1)c1ccc(Br)nc1 ZINC000880561499 EE On-Demand Anodyne CA14 18 47 COC(=O)[C@@]1(O)CCN([C@@H]2CCCC[C@H]2O)C1 ZINC000880561503 BB On-Demand Anodyne SLC18A3 31 42 CCCOc1cccc(CNC(=O)CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880561516 FC On-Demand Anodyne HRH2 29 41 CCCOc1cccc(CNC(=O)CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880561516 FC On-Demand Anodyne MMP13 18 43 CCCOc1cccc(CNC(=O)CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880561516 FC On-Demand Anodyne PDS 40 33 CCCOc1cccc(CNC(=O)CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880561518 FC On-Demand Anodyne HRH2 29 41 CCCOc1cccc(CNC(=O)CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880561518 FC On-Demand Anodyne MMP13 18 43 CCCOc1cccc(CNC(=O)CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880561518 FC On-Demand Anodyne PDS 40 33 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(C)cc3)CC2)c1 ZINC000880561520 FH On-Demand Anodyne PDGFRB 35 40 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(C)cc3)CC2)c1 ZINC000880561520 FH On-Demand Anodyne SLC18A3 42 44 COc1cncc(NC(=O)N2CCC(CC(=O)N3CCCC3)CC2)c1 ZINC000880561546 EE On-Demand Anodyne EPHX2 15 40 CCN(Cc1ccc(OC)cc1OC)C(=O)Nc1cncc(OC)c1 ZINC000880561547 EG On-Demand Anodyne PDGFRB 40 39 CCN(Cc1ccc(OC)cc1OC)C(=O)Nc1cncc(OC)c1 ZINC000880561547 EG On-Demand Anodyne ROCK2 20 45 O=C(NCc1cn(C2CCC2)nn1)c1cccnc1I ZINC000880561548 GD On-Demand Anodyne G2YM83_BOTF4 44 32 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880561551 FG On-Demand Anodyne ST14 47 33 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880561551 FG On-Demand Anodyne TMPRSS6 70 33 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880561552 FG On-Demand Anodyne ST14 47 33 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880561552 FG On-Demand Anodyne TMPRSS6 70 33 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne DRD4 42 32 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne MAPK14 35 51 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne CCR3 29 41 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne CHRNA7 15 41 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne ROCK1 29 40 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne ROCK2 50 48 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne MCHR1 20 42 COc1cncc(NC(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000880561559 EE On-Demand Anodyne NAMPT 38 40 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OCc2cccnc2)C1 ZINC000880561560 GE On-Demand Anodyne PTGER1 88 44 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccsc3)CC2)c1 ZINC000880561561 FF On-Demand Anodyne NPBWR1 75 32 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(C)c2)c1 ZINC000880561562 ED On-Demand Anodyne ADRB2 34 50 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(C)c2)c1 ZINC000880561562 ED On-Demand Anodyne ADRB1 55 50 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(C)c2)c1 ZINC000880561562 ED On-Demand Anodyne ADRB3 30 45 COc1cncc(NC(=O)NC[C@H](O)COc2cccc(C)c2)c1 ZINC000880561562 ED On-Demand Anodyne ACOX1 40 34 COc1cncc(NC(=O)N(Cc2ccc(O)c(OC)c2)C2CC2)c1 ZINC000880561563 EG On-Demand Anodyne ROCK2 22 50 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(C)c2)c1 ZINC000880561564 ED On-Demand Anodyne ADRB2 34 50 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(C)c2)c1 ZINC000880561564 ED On-Demand Anodyne ADRB1 55 50 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(C)c2)c1 ZINC000880561564 ED On-Demand Anodyne ADRB3 30 45 COc1cncc(NC(=O)NC[C@@H](O)COc2cccc(C)c2)c1 ZINC000880561564 ED On-Demand Anodyne ACOX1 40 34 COc1cncc(NC(=O)NCc2cc(C)ccc2OC)c1 ZINC000880561576 DF On-Demand Anodyne ROCK2 15 53 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccnc2)C1 ZINC000880561577 CB On-Demand Anodyne CHRNA7 43 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cccnc2)C1 ZINC000880561577 CB On-Demand Anodyne NAMPT 63 42 COCCN(CCc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880561580 EF On-Demand Anodyne ROCK2 27 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne ADRB2 19 50 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne ADRB1 22 50 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne HTR1A 17 51 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne SLC6A4 19 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne ACOX1 21 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561590 EC On-Demand Anodyne ABCB1 66 43 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne ADRB2 19 50 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne ADRB1 22 50 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne HTR1A 17 51 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne SLC6A4 19 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne ACOX1 21 41 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc3[nH]ccc23)C1 ZINC000880561591 EC On-Demand Anodyne ABCB1 66 43 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCC(F)(F)F)C1 ZINC000880561600 ED On-Demand Anodyne CCR8 23 42 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc(Cl)c2)C1 ZINC000880561601 CE On-Demand Anodyne OPRL1 19 44 COc1cncc(NC(=O)N2CCC(C(=O)N3CCCC3)CC2)c1 ZINC000880561602 ED On-Demand Anodyne EPHX2 17 41 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc(Cl)c2)C1 ZINC000880561605 CE On-Demand Anodyne OPRL1 19 44 COc1cncc(NC(=O)N2CCC[C@H](CNC(C)=O)C2)c1 ZINC000880561612 DD On-Demand Anodyne CCR3 21 47 COc1cncc(NC(=O)N2CCC[C@@H](CNC(C)=O)C2)c1 ZINC000880561615 DD On-Demand Anodyne CCR3 21 47 COc1cncc(NC(=O)N2CC[C@H](c3ccccc3C)C2)c1 ZINC000880561624 DG On-Demand Anodyne RBP4 49 38 COc1cncc(NC(=O)N2CC[C@@H](c3ccccc3C)C2)c1 ZINC000880561627 DG On-Demand Anodyne RBP4 49 38 COc1cncc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561631 DD On-Demand Anodyne CCR3 39 44 COc1cncc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561631 DD On-Demand Anodyne EPHX2 45 40 COc1cncc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561631 DD On-Demand Anodyne CXCR3 21 42 COc1cncc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561631 DD On-Demand Anodyne HPGDS 36 45 COc1cncc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561634 DD On-Demand Anodyne CCR3 39 44 COc1cncc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561634 DD On-Demand Anodyne EPHX2 45 40 COc1cncc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561634 DD On-Demand Anodyne CXCR3 21 42 COc1cncc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880561634 DD On-Demand Anodyne HPGDS 36 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(SC)c(OC)c2)C1 ZINC000880561641 DD On-Demand Anodyne MCHR2 40 32 COC(=O)[C@@]1(O)CCN(Cc2ccc3c(c2)CCC3)C1 ZINC000880561653 CD On-Demand Anodyne MCHR2 63 36 CC(C)(C)OC(=O)N[C@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561674 GG On-Demand Anodyne PGC 50 33 CC(C)(C)OC(=O)N[C@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561674 GG On-Demand Anodyne REN 64 36 CC(C)(C)OC(=O)N[C@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561674 GG On-Demand Anodyne FPR1 44 36 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561675 GG On-Demand Anodyne PGC 50 33 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561675 GG On-Demand Anodyne REN 64 36 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880561675 GG On-Demand Anodyne FPR1 44 36 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne HTR1A 71 42 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne DRD2 57 41 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne DRD4 40 40 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne ADRA1D 51 37 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne HTR2A 17 41 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne ADRA1A 49 39 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne ADRA1B 41 37 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne DRD3 65 39 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne HTR7 49 39 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne NPY1R 15 41 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne CCR3 42 41 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561683 FF On-Demand Anodyne SOAT1 15 41 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne HTR1A 71 42 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne DRD2 57 41 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne DRD4 40 40 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne ADRA1D 51 37 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne HTR2A 17 41 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne ADRA1A 49 39 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne ADRA1B 41 37 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne DRD3 65 39 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne HTR7 49 39 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne NPY1R 15 41 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne CCR3 42 41 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3OC)C2)c1 ZINC000880561684 FF On-Demand Anodyne SOAT1 15 41 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(F)(F)F)C1 ZINC000880561692 ED On-Demand Anodyne LTA4H 15 47 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(F)(F)F)C1 ZINC000880561692 ED On-Demand Anodyne RBP4 44 40 CCN(Cc1ccoc1)C(=O)Nc1cncc(OC)c1 ZINC000880561693 CF On-Demand Anodyne ROCK2 18 47 COc1cncc(NC(=O)NCc2cccc(CS(C)(=O)=O)c2)c1 ZINC000880561694 ED On-Demand Anodyne ROCK1 30 43 COc1cncc(NC(=O)NCc2cccc(CS(C)(=O)=O)c2)c1 ZINC000880561694 ED On-Demand Anodyne ROCK2 48 53 COc1cncc(NC(=O)NCc2cccc(CS(C)(=O)=O)c2)c1 ZINC000880561694 ED On-Demand Anodyne NAMPT 47 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2)C1 ZINC000880561699 CC On-Demand Anodyne LTA4H 20 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCC(F)(F)F)cc2)C1 ZINC000880561700 ED On-Demand Anodyne MMP13 22 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCC(F)(F)F)cc2)C1 ZINC000880561700 ED On-Demand Anodyne ADAM17 20 43 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2OC)C1 ZINC000880561703 CC On-Demand Anodyne MTNR1B 36 42 COc1cncc(NC(=O)N2CCN(C)c3ccccc3C2)c1 ZINC000880561713 DF On-Demand Anodyne PDGFRB 43 39 COc1cncc(NC(=O)N[C@@H](C)c2cc(OC)ccc2O)c1 ZINC000880561717 DF On-Demand Clean THRB 45 35 COc1cncc(NC(=O)N[C@H](C)c2cc(OC)ccc2O)c1 ZINC000880561719 DF On-Demand Clean THRB 45 35 COc1cncc(NC(=O)N2CCN(c3nccc(OC)n3)CC2)c1 ZINC000880561739 ED On-Demand Anodyne PDGFRB 53 41 COc1cncc(NC(=O)N2CCN(c3nccc(OC)n3)CC2)c1 ZINC000880561739 ED On-Demand Anodyne FAAH 21 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)N(Cc2ccccc2)C(C)C)C1 ZINC000880561741 ED On-Demand Anodyne SLC12A5 60 38 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)N(Cc2ccccc2)C(C)C)C1 ZINC000880561743 ED On-Demand Anodyne SLC12A5 60 38 COc1cncc(NC(=O)N2CCC(NC(=O)NC3CCCCC3)CC2)c1 ZINC000880561745 GF On-Demand Anodyne CCR3 15 40 COc1cncc(NC(=O)N2CCC(NC(=O)NC3CCCCC3)CC2)c1 ZINC000880561745 GF On-Demand Anodyne C3AR1 34 41 COc1cncc(NC(=O)N2CCC(NC(=O)NC3CCCCC3)CC2)c1 ZINC000880561745 GF On-Demand Anodyne EPHX2 52 49 COc1cncc(NC(=O)NCCCN2CCOC2=O)c1 ZINC000880561761 CD On-Demand Anodyne CCR3 27 42 COc1cncc(NC(=O)NCCCN2CCOC2=O)c1 ZINC000880561761 CD On-Demand Anodyne QPCT 27 40 COc1cncc(NC(=O)N2CCC(Oc3cccc(C#N)c3)CC2)c1 ZINC000880561762 FG On-Demand Mild CCR3 34 41 COc1cncc(NC(=O)N2CCC(Oc3cccc(C#N)c3)CC2)c1 ZINC000880561762 FG On-Demand Mild EPHX2 21 52 COc1cncc(NC(=O)N2CCC(Oc3cccc(C#N)c3)CC2)c1 ZINC000880561762 FG On-Demand Mild SCD1 15 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne DRD2 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne DRD4 35 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne CHRM3 21 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne SIGMAR1 69 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne MMP13 20 53 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne NPFFR2 33 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne ADAM17 17 53 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne FAAH 24 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne MMP9 19 53 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne MCHR2 56 39 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne NPFFR1 45 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3)cc2)C1 ZINC000880561765 DE On-Demand Anodyne SLC12A5 64 37 COc1cncc(NC(=O)NCC(=O)N2CCc3ccccc3C2)c1 ZINC000880561768 ED On-Demand Anodyne NOD1 15 41 COc1cncc(NC(=O)NCC(=O)N2CCc3ccccc3C2)c1 ZINC000880561768 ED On-Demand Anodyne NOD2 41 41 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(OC)cc2)c2ccccc2)C1 ZINC000880561772 GD On-Demand Anodyne OPRL1 15 44 COC(=O)[C@@]1(O)CCN([C@H](C(=O)Nc2ccc(OC)cc2)c2ccccc2)C1 ZINC000880561772 GD On-Demand Anodyne NPY2R 38 42 O=C(COC/C=C/c1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880561776 EE On-Demand Anodyne PREP 18 40 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(OC)cc2)c2ccccc2)C1 ZINC000880561777 GD On-Demand Anodyne OPRL1 15 44 COC(=O)[C@@]1(O)CCN([C@@H](C(=O)Nc2ccc(OC)cc2)c2ccccc2)C1 ZINC000880561777 GD On-Demand Anodyne NPY2R 38 42 O=C(COC/C=C\c1ccccc1)NCc1cn(C2CCC2)nn1 ZINC000880561780 EE On-Demand Anodyne PREP 18 40 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880561789 FF On-Demand Anodyne CCR3 15 44 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880561791 FF On-Demand Anodyne CCR3 15 44 COc1cncc(NC(=O)NCCCN2CCC[C@H]2C(=O)N(C)C)c1 ZINC000880561799 ED On-Demand Anodyne CCR3 39 44 COc1cncc(NC(=O)NCCCN2CCC[C@@H]2C(=O)N(C)C)c1 ZINC000880561800 ED On-Demand Anodyne CCR3 39 44 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne HTR1A 20 43 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne DRD2 25 42 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne DRD4 15 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne ADRA1D 20 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne HTR2A 15 43 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne ADRA1A 38 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne ADRA1B 27 43 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne OPRM1 21 48 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne DRD3 24 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne OPRD1 18 48 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne OPRK1 15 48 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne OPRL1 15 44 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne SLC6A3 20 49 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne LTA4H 15 42 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne SIGMAR1 74 53 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne EBP 31 43 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne FAAH 26 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2)C1 ZINC000880561811 CD On-Demand Anodyne SLC12A5 75 42 CC[C@@H](C)c1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880561817 DG On-Demand Anodyne CA14 16 45 COc1cncc(NC(=O)N[C@@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561830 GG On-Demand Anodyne CCR3 48 37 COc1cncc(NC(=O)N[C@@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561830 GG On-Demand Anodyne CCKBR 15 40 COc1cncc(NC(=O)N[C@@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561830 GG On-Demand Anodyne TAAR1 32 40 COc1cncc(NC(=O)N[C@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561831 GG On-Demand Anodyne CCR3 48 37 COc1cncc(NC(=O)N[C@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561831 GG On-Demand Anodyne CCKBR 15 40 COc1cncc(NC(=O)N[C@H](C)CC(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000880561831 GG On-Demand Anodyne TAAR1 32 40 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne SSTR5 49 38 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne CCR3 26 40 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne EPHX2 64 53 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne CXCR3 21 41 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne MCHR1 17 43 CCOc1ccc(C(=O)N2CCC(NC(=O)Nc3cncc(OC)c3)CC2)cc1 ZINC000880561841 GF On-Demand Anodyne PTR1 45 33 COC(=O)[C@@]1(O)CCN(CCCc2ccc(Cl)cc2)C1 ZINC000880561856 CD On-Demand Anodyne DRD4 20 49 COC(=O)[C@@]1(O)CCN(CCCc2ccc(Cl)cc2)C1 ZINC000880561856 CD On-Demand Anodyne SIGMAR1 28 41 COC(=O)[C@@]1(O)CCN(CCCc2ccc(Cl)cc2)C1 ZINC000880561856 CD On-Demand Anodyne MMP13 15 42 COC(=O)[C@@]1(O)CCN(CCCc2ccc(Cl)cc2)C1 ZINC000880561856 CD On-Demand Anodyne CCR1 66 42 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc4c(c3)OCO4)CC2)c1 ZINC000880561875 GD On-Demand Anodyne PDGFRB 35 41 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc4c(c3)OCO4)CC2)c1 ZINC000880561875 GD On-Demand Anodyne EDNRA 37 41 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc4c(c3)OCO4)CC2)c1 ZINC000880561875 GD On-Demand Anodyne BMP1 29 40 COc1cncc(NC(=O)N(C)CCCOc2ccc(S(C)(=O)=O)cc2)c1 ZINC000880561887 GE On-Demand Anodyne USP7 43 37 COc1cncc(NC(=O)N(C)CCCOc2ccc(S(C)(=O)=O)cc2)c1 ZINC000880561887 GE On-Demand Anodyne USP47 54 37 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880561888 GD On-Demand Anodyne P2RY1 43 34 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880561890 GD On-Demand Anodyne P2RY1 43 34 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880561892 EE On-Demand Anodyne TSPO 25 40 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880561892 EE On-Demand Anodyne ROCK2 42 43 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880561892 EE On-Demand Anodyne LIMK2 17 41 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1cncc(OC)c1 ZINC000880561892 EE On-Demand Anodyne NAMPT 23 40 COc1cncc(NC(=O)N2CCc3ccc(OC)cc3C2)c1 ZINC000880561909 DF On-Demand Anodyne HDAC6 30 41 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880561911 FF On-Demand Anodyne EPHX2 67 55 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880561911 FF On-Demand Anodyne CXCR3 18 42 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880561911 FF On-Demand Anodyne MCHR1 15 42 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880561911 FF On-Demand Anodyne SMO 23 41 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880561911 FF On-Demand Anodyne L3MBTL3 48 33 COC(=O)[C@@]1(O)CCN(CCN(C)c2ccccc2)C1 ZINC000880561916 CC On-Demand Anodyne SLC12A5 54 38 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(C)no3)C2)c1 ZINC000880561919 DE On-Demand Anodyne SMO 19 44 COc1cncc(NC(=O)N2CCC[C@H](c3nc(C)no3)C2)c1 ZINC000880561920 DE On-Demand Anodyne SMO 19 44 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne PDGFRB 47 38 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne CCR3 17 46 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne MTNR1B 15 47 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne NPY5R 17 41 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne EPHX2 40 45 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880561924 FG On-Demand Anodyne LIMK2 15 42 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2OC)c1 ZINC000880561929 EG On-Demand Anodyne TACR1 15 40 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2OC)c1 ZINC000880561929 EG On-Demand Anodyne CCR3 17 47 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2OC)c1 ZINC000880561929 EG On-Demand Anodyne CHRNA7 20 45 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2OC)c1 ZINC000880561929 EG On-Demand Anodyne ACKR3 64 33 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2OC)c1 ZINC000880561930 EG On-Demand Anodyne TACR1 15 40 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2OC)c1 ZINC000880561930 EG On-Demand Anodyne CCR3 17 47 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2OC)c1 ZINC000880561930 EG On-Demand Anodyne CHRNA7 20 45 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2OC)c1 ZINC000880561930 EG On-Demand Anodyne ACKR3 64 33 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880561932 ED On-Demand Anodyne MMP13 23 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880561932 ED On-Demand Anodyne ADAM17 34 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880561932 ED On-Demand Anodyne MMP9 15 47 COc1cncc(NC(=O)NC2CCN(C(=O)CC(C)C)CC2)c1 ZINC000880561944 EE On-Demand Anodyne EPHX2 51 57 COc1cncc(NC(=O)NC2CCN(C(=O)CC(C)C)CC2)c1 ZINC000880561944 EE On-Demand Anodyne CXCR3 16 41 COc1cncc(NC(=O)NC[C@H](c2cccc(F)c2)N2CCOCC2)c1 ZINC000880561945 FE On-Demand Anodyne CCR3 17 41 COc1cncc(NC(=O)NC[C@@H](c2cccc(F)c2)N2CCOCC2)c1 ZINC000880561947 FE On-Demand Anodyne CCR3 17 41 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne LTA4H 18 41 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne MMP13 30 45 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne ADAM17 17 45 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne MMP9 26 45 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne MMP1 17 45 COC(=O)[C@@]1(O)CCN(CCOCc2ccc(OC)cc2)C1 ZINC000880561963 DC On-Demand Anodyne SLC12A5 47 42 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne PDE3A 40 38 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne PDGFRB 55 40 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne CCR3 17 40 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne PDE3B 46 38 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne EPHX2 25 43 COc1cncc(NC(=O)N2CCC(Oc3c(OC)cccc3OC)CC2)c1 ZINC000880561968 GG On-Demand Anodyne SCD1 25 54 CCCN(CC)C(=O)Nc1cncc(OC)c1 ZINC000880561971 BE On-Demand Anodyne ROCK2 17 42 COC(=O)[C@@]1(O)CCN(CCn2ccccc2=O)C1 ZINC000880561979 CB On-Demand Anodyne SLC12A5 49 37 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cc3F)CC2)c1 ZINC000880561991 FE On-Demand Mild PDGFRB 49 46 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cc3F)CC2)c1 ZINC000880561991 FE On-Demand Mild NPY2R 57 40 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cc3F)CC2)c1 ZINC000880561991 FE On-Demand Mild SLC6A9 21 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)N(C)C)c2)C1 ZINC000880562016 DC On-Demand Anodyne CHRM3 15 40 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccsc3)oc2C)C1 ZINC000880562018 DD On-Demand Anodyne PPARG 27 43 COC(=O)[C@@]1(O)CCN(Cc2nc(-c3ccsc3)oc2C)C1 ZINC000880562018 DD On-Demand Anodyne PDE8B 65 38 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne F2 88 47 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne PLG 37 43 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne PRSS1 31 44 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne ACE 33 46 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne FKBP1A 56 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne OPRM1 31 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne OPRD1 18 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne CELA1 27 52 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne ELANE 38 45 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne CTRA_BOVIN 63 33 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne TRY1_BOVIN 106 45 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne NTSR1 83 36 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne NTSR2 55 32 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne CTSG 44 33 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne HLA-A 57 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne PREP 83 55 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne CELA2A 51 33 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne LGMN 92 52 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne KLK5 26 44 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne XIAP 47 46 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne BRCA1 61 32 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne TMPRSS11D 83 47 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880562021 GE On-Demand Anodyne TMPRSS6 15 44 COc1cncc(NC(=O)N(C)Cc2ccc(SC)c(OC)c2)c1 ZINC000880562028 EG On-Demand Anodyne ROCK2 18 44 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562029 GH On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562029 GH On-Demand Anodyne CPT1A 34 40 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562029 GH On-Demand Anodyne GRM5 24 55 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562029 GH On-Demand Anodyne SMO 35 48 COc1cncc(NC(=O)N2CCC[C@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562029 GH On-Demand Anodyne ETHR 41 47 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562030 GH On-Demand Anodyne CCR3 21 43 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562030 GH On-Demand Anodyne CPT1A 34 40 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562030 GH On-Demand Anodyne GRM5 24 55 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562030 GH On-Demand Anodyne SMO 35 48 COc1cncc(NC(=O)N2CCC[C@@H](c3nc(-c4cccc(F)c4)no3)C2)c1 ZINC000880562030 GH On-Demand Anodyne ETHR 41 47 CCOC(=O)N1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880562034 DD On-Demand Anodyne P2RY12 35 46 CCOC(=O)N1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880562034 DD On-Demand Anodyne PDGFRB 42 40 COC(=O)[C@@]1(O)CCN(CCOc2cccc(C#N)c2)C1 ZINC000880562102 CC On-Demand Mild DRD4 40 30 COC(=O)[C@@]1(O)CCN(CCOc2cccc(C#N)c2)C1 ZINC000880562102 CC On-Demand Mild CHRNA10 15 44 COC(=O)[C@@]1(O)CCN(CCOc2cccc(C#N)c2)C1 ZINC000880562102 CC On-Demand Mild MCHR1 22 41 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880562109 GD On-Demand Anodyne HTR1A 17 47 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880562109 GD On-Demand Anodyne DRD4 32 47 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880562109 GD On-Demand Anodyne DRD3 15 41 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne HTR7 28 52 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne MMP13 29 42 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne CCR1 17 50 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne ADAM17 20 42 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne MMP9 25 42 COC(=O)[C@@]1(O)CCN(CCNS(=O)(=O)c2ccccc2)C1 ZINC000880562112 EB On-Demand Anodyne SLC12A5 66 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)n2)C1 ZINC000880562115 CC On-Demand Anodyne ALS 71 32 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CC2)C1 ZINC000880562136 EC On-Demand Anodyne ADRA1A 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CC2)C1 ZINC000880562136 EC On-Demand Anodyne KCNA3 53 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCC2(c3ccccc3)CC2)C1 ZINC000880562136 EC On-Demand Anodyne NPFFR1 39 46 COc1cncc(NC(=O)N2CCN(C(=O)CCCc3ccccc3)CC2)c1 ZINC000880562148 GF On-Demand Anodyne PDGFRB 44 41 COc1cncc(NC(=O)N2CCN(C(=O)CCCc3ccccc3)CC2)c1 ZINC000880562148 GF On-Demand Anodyne PTAFR 18 43 COc1cncc(NC(=O)N2CCN(C(=O)CCCc3ccccc3)CC2)c1 ZINC000880562148 GF On-Demand Anodyne PREP 47 42 COc1cncc(NC(=O)N2CCN(C(=O)CCCc3ccccc3)CC2)c1 ZINC000880562148 GF On-Demand Anodyne FAAH 50 48 COC(=O)[C@@]1(O)CCN(Cc2ccccc2Oc2cccnc2)C1 ZINC000880562151 ED On-Demand Anodyne CCR8 41 49 COC(=O)[C@@]1(O)CCN(CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000880562168 CC On-Demand Bother ADRA1A 22 40 COC(=O)[C@@]1(O)CCN(CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000880562168 CC On-Demand Bother MMP9 15 44 COC(=O)[C@@]1(O)CCN(CCc2ccc([N+](=O)[O-])cc2)C1 ZINC000880562168 CC On-Demand Bother KCNJ1 38 54 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MAOB 23 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne LTA4H 58 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne HRH3 18 53 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne SIGMAR1 73 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP13 36 59 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne CACNA1B 23 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne ADAM17 62 59 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP2 18 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP14 21 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne FAAH 27 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne SLC6A5 38 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP9 28 59 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP10 17 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne ADAMTS4 28 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne MMP1 18 59 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne FFAR1 43 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne NPFFR1 44 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne SLC12A5 75 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)cc2)C1 ZINC000880562170 EE On-Demand Anodyne NOD2 40 37 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne PDGFRB 39 40 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne NQO2 44 41 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne RAF1 23 40 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne MTNR1A 98 44 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne MTNR1B 81 41 COc1cncc(NC(=O)NCCc2ccc(OC)cc2OC)c1 ZINC000880562171 EE On-Demand Anodyne CSF1R 16 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne HRH3 53 47 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP13 65 52 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne ADAM17 51 52 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP2 34 42 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP3 35 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP8 24 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP9 37 52 COC(=O)[C@@]1(O)CCN(CCCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562177 FC On-Demand Anodyne MMP1 35 46 COC(=O)[C@@]1(O)CCN(CCCOc2ccccc2C)C1 ZINC000880562183 CD On-Demand Anodyne ADRA1A 44 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562186 FC On-Demand Anodyne ADRB2 17 44 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562186 FC On-Demand Anodyne CCR1 42 38 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562186 FC On-Demand Anodyne ABCB1 71 45 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562187 FC On-Demand Anodyne ADRB2 17 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562187 FC On-Demand Anodyne CCR1 42 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2c(OC)cccc2OC)C1 ZINC000880562187 FC On-Demand Anodyne ABCB1 71 45 COc1cncc(NC(=O)N2CCC(C(=O)Nc3cccc(F)c3)CC2)c1 ZINC000880562188 FG On-Demand Anodyne CACNA1H 41 35 COc1cncc(NC(=O)N2CCC(C(=O)Nc3cccc(F)c3)CC2)c1 ZINC000880562188 FG On-Demand Anodyne CCR3 27 50 COc1cncc(NC(=O)N2CCC(C(=O)Nc3cccc(F)c3)CC2)c1 ZINC000880562188 FG On-Demand Anodyne EPHX2 26 42 COc1cncc(NC(=O)N2CCC(C(=O)Nc3cccc(F)c3)CC2)c1 ZINC000880562188 FG On-Demand Anodyne SCD1 18 43 COc1cncc(NC(=O)N2CCC(C(=O)Nc3cccc(F)c3)CC2)c1 ZINC000880562188 FG On-Demand Anodyne LIMK2 23 46 COc1cncc(NC(=O)N2CCN(C(=O)CC3CCCCC3)CC2)c1 ZINC000880562191 FF On-Demand Anodyne PDGFRB 50 39 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne HTR1A 27 43 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne DRD2 20 40 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne DRD4 44 36 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne DRD3 31 43 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne CCR3 16 42 COc1cncc(NC(=O)NCCC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880562196 GD On-Demand Anodyne SOAT1 15 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562200 FD On-Demand Anodyne ACOX1 69 34 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562200 FD On-Demand Anodyne ABCB1 49 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562200 FD On-Demand Anodyne PDS 48 43 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562201 FD On-Demand Anodyne ACOX1 69 34 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562201 FD On-Demand Anodyne ABCB1 49 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880562201 FD On-Demand Anodyne PDS 48 43 COc1cncc(NC(=O)NCc2cccc(OCC(F)F)c2)c1 ZINC000880562210 EG On-Demand Anodyne HRH2 20 42 COc1cncc(NC(=O)NCc2cccc(OCC(F)F)c2)c1 ZINC000880562210 EG On-Demand Anodyne ROCK1 41 46 COc1cncc(NC(=O)NCc2cccc(OCC(F)F)c2)c1 ZINC000880562210 EG On-Demand Anodyne ROCK2 58 55 COc1cncc(NC(=O)NCc2cccc(OCC(F)F)c2)c1 ZINC000880562210 EG On-Demand Anodyne NAMPT 40 41 COc1cncc(NC(=O)NCc2cccc(OCC(F)F)c2)c1 ZINC000880562210 EG On-Demand Anodyne PDS 94 45 COc1cncc(NC(=O)NCCCOC2CCCC2)c1 ZINC000880562217 CF On-Demand Anodyne HRH2 19 42 COc1cncc(NC(=O)NCCCOC2CCCC2)c1 ZINC000880562217 CF On-Demand Anodyne CCR3 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCOc2cccc(C)c2)C1 ZINC000880562228 FC On-Demand Anodyne HRH2 47 43 COC(=O)[C@@]1(O)CCN(Cc2cccnc2Cl)C1 ZINC000880562230 CC On-Demand Anodyne CCR8 24 40 COC(=O)[C@@]1(O)CCN(Cc2cccnc2Cl)C1 ZINC000880562230 CC On-Demand Anodyne G2YM83_BOTF4 44 33 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCO[C@H](C)c2ccccc2)C1 ZINC000880562233 FC On-Demand Anodyne ADRA1A 20 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCCCO[C@@H](C)c2ccccc2)C1 ZINC000880562234 FC On-Demand Anodyne ADRA1A 20 42 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne HTR1A 48 39 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne DRD2 40 39 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne DRD3 44 37 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne HTR4 18 42 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne HTR7 40 37 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2OC)C1 ZINC000880562243 CC On-Demand Anodyne HCN1 40 36 COC(=O)[C@@]1(O)CCN([C@H](C)CCc2ccccc2)C1 ZINC000880562246 CD On-Demand Anodyne ACE 44 36 COC(=O)[C@@]1(O)CCN([C@H](C)CCc2ccccc2)C1 ZINC000880562246 CD On-Demand Anodyne SLC12A5 67 41 COC(=O)[C@@]1(O)CCN([C@@H](C)CCc2ccccc2)C1 ZINC000880562247 CD On-Demand Anodyne ACE 44 36 COC(=O)[C@@]1(O)CCN([C@@H](C)CCc2ccccc2)C1 ZINC000880562247 CD On-Demand Anodyne SLC12A5 67 41 COc1cncc(NC(=O)NCc2cccc(N(C)C)c2)c1 ZINC000880562248 DE On-Demand Anodyne ROCK1 38 44 COc1cncc(NC(=O)NCc2cccc(N(C)C)c2)c1 ZINC000880562248 DE On-Demand Anodyne ROCK2 57 53 COc1cncc(NC(=O)NCc2cccc(N(C)C)c2)c1 ZINC000880562248 DE On-Demand Anodyne FLT4 17 40 COc1cncc(NC(=O)NCc2cccc(N(C)C)c2)c1 ZINC000880562248 DE On-Demand Anodyne NAMPT 40 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCC(F)(F)F)c2)C1 ZINC000880562250 ED On-Demand Anodyne HRH2 31 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCC(F)(F)F)c2)C1 ZINC000880562250 ED On-Demand Anodyne FAAH 22 40 COC(=O)[C@@]1(O)CCN(Cc2csc3ccccc23)C1 ZINC000880562253 CE On-Demand Anodyne FFAR2 63 36 COc1cncc(NC(=O)N(Cc2cccs2)C(C)C)c1 ZINC000880562256 DH On-Demand Anodyne ROCK2 15 48 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCCN(Cc3ccc(C)cc3)CC2)C1 ZINC000880562260 GC On-Demand Anodyne DRD4 15 41 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne HTR1A 21 43 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne DRD2 26 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne HTR2A 21 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne PPARG 15 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne HRH3 87 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne SIGMAR1 34 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne MMP13 22 49 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne HTR5A 21 44 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne ADAM17 26 45 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne EBP 36 40 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne MMP9 17 49 COC(=O)[C@@]1(O)CCN(CCCOc2ccc3ccccc3c2)C1 ZINC000880562273 EE On-Demand Anodyne EPHX2 22 40 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562275 EE On-Demand Anodyne MMP13 19 43 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562275 EE On-Demand Anodyne MMP2 24 43 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562275 EE On-Demand Anodyne MMP14 15 43 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562275 EE On-Demand Anodyne MMP9 17 43 COC(=O)[C@@]1(O)CCN([C@@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562275 EE On-Demand Anodyne EPHX2 47 40 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562276 EE On-Demand Anodyne MMP13 19 43 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562276 EE On-Demand Anodyne MMP2 24 43 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562276 EE On-Demand Anodyne MMP14 15 43 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562276 EE On-Demand Anodyne MMP9 17 43 COC(=O)[C@@]1(O)CCN([C@H](C)c2ccc(OC(F)(F)F)cc2)C1 ZINC000880562276 EE On-Demand Anodyne EPHX2 47 40 CCN(Cc1c(F)cccc1F)C(=O)Nc1cncc(OC)c1 ZINC000880562278 DG On-Demand Anodyne ROCK2 22 48 COc1cncc(NC(=O)NCCCCOCc2ccccc2)c1 ZINC000880562279 EG On-Demand Anodyne HRH2 22 43 COc1cncc(NC(=O)NCCCCOCc2ccccc2)c1 ZINC000880562279 EG On-Demand Anodyne CCR3 26 47 COc1cncc(NC(=O)NCc2ccc(OCC3CC3)nc2)c1 ZINC000880562280 EF On-Demand Anodyne ROCK2 15 40 O=C(NCc1cn(C2CCC2)nn1)c1cc(C(F)(F)F)ccc1F ZINC000880562282 EG On-Demand Anodyne CCR2 60 38 O=C(NCc1cn(C2CCC2)nn1)c1cc(C(F)(F)F)ccc1F ZINC000880562282 EG On-Demand Anodyne LIPG 42 34 COc1cncc(NC(=O)NCC2(c3ccccc3OC)CC2)c1 ZINC000880562283 EF On-Demand Anodyne KCNA3 44 38 COc1cncc(NC(=O)NCC2(c3ccccc3OC)CC2)c1 ZINC000880562283 EF On-Demand Anodyne NMBR 54 43 COc1cncc(NC(=O)NCC2(c3ccccc3OC)CC2)c1 ZINC000880562283 EF On-Demand Anodyne MTNR1B 18 41 COc1cncc(NC(=O)NCC2(c3ccccc3OC)CC2)c1 ZINC000880562283 EF On-Demand Anodyne GRPR 33 43 COc1cncc(NC(=O)NCC2(c3ccccc3OC)CC2)c1 ZINC000880562283 EF On-Demand Anodyne SOAT1 27 49 COc1cncc(NC(=O)N2CCC(NC(C)=O)CC2)c1 ZINC000880562291 CD On-Demand Anodyne EPHX2 27 42 COc1cncc(NC(=O)NC2CCN(CC(F)F)CC2)c1 ZINC000880562292 DD On-Demand Anodyne CCR3 47 43 COc1cncc(NC(=O)NC2CCN(CC(F)F)CC2)c1 ZINC000880562292 DD On-Demand Anodyne EPHX2 56 43 COc1cncc(NC(=O)NC2CCN(CC(F)F)CC2)c1 ZINC000880562292 DD On-Demand Anodyne CXCR3 22 45 COc1cncc(NC(=O)NC2CCN(CC(F)F)CC2)c1 ZINC000880562292 DD On-Demand Anodyne MCHR1 16 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCC#N)cc2)C1 ZINC000880562312 CC On-Demand Mild MMP13 28 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCC#N)cc2)C1 ZINC000880562312 CC On-Demand Mild ADAM17 37 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCC#N)cc2)C1 ZINC000880562312 CC On-Demand Mild MMP9 18 46 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2cccc(OC)c2)C1 ZINC000880562314 EC On-Demand Anodyne DRD4 44 34 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2cccc(OC)c2)C1 ZINC000880562314 EC On-Demand Anodyne MMP13 26 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2cccc(OC)c2)C1 ZINC000880562314 EC On-Demand Anodyne ADAM17 22 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2cccc(OC)c2)C1 ZINC000880562314 EC On-Demand Anodyne MMP9 21 44 COc1cncc(NC(=O)N2CCC(CNC(=O)OC(C)(C)C)CC2)c1 ZINC000880562325 FF On-Demand Anodyne CACNA1I 46 33 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCC(C)C)C1 ZINC000880562331 DD On-Demand Anodyne CCR8 24 55 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)C)cc2)C1 ZINC000880562345 CD On-Demand Anodyne MMP13 22 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)C)cc2)C1 ZINC000880562345 CD On-Demand Anodyne ADAM17 17 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)C)cc2)C1 ZINC000880562345 CD On-Demand Anodyne MMP9 18 44 COc1cncc(NC(=O)N2CCC[C@H](CNC(=O)C(C)C)C2)c1 ZINC000880562352 EE On-Demand Anodyne CCR3 24 47 COc1cncc(NC(=O)N2CCC[C@@H](CNC(=O)C(C)C)C2)c1 ZINC000880562353 EE On-Demand Anodyne CCR3 24 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(OC)c2Br)C1 ZINC000880562361 FD On-Demand Anodyne SLC9A1 55 30 COC(=O)[C@@]1(O)CCN(CCOc2cc(Cl)cc(Cl)c2)C1 ZINC000880562372 ED On-Demand Anodyne CACNA1I 47 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2cccc(Cl)c2)C1 ZINC000880562373 CC On-Demand Anodyne ADRB1 24 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2cccc(Cl)c2)C1 ZINC000880562376 CC On-Demand Anodyne ADRB1 24 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(I)cc2)C1 ZINC000880562379 FD On-Demand Anodyne SIGMAR1 22 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(I)cc2)C1 ZINC000880562379 FD On-Demand Anodyne MMP13 15 42 COC(=O)[C@@]1(O)CCN(Cc2ccc3ccccc3n2)C1 ZINC000880562382 CD On-Demand Anodyne ALOX5AP 41 38 COc1cncc(NC(=O)NCc2ccc(C(=O)N3C[C@H](C)O[C@H](C)C3)cc2)c1 ZINC000880562391 GF On-Demand Anodyne NAMPT 27 43 COc1cncc(NC(=O)NCc2ccc(C(=O)N3C[C@H](C)O[C@@H](C)C3)cc2)c1 ZINC000880562392 GF On-Demand Anodyne NAMPT 27 43 COc1cncc(NC(=O)NCc2ccc(C(=O)N3C[C@@H](C)O[C@H](C)C3)cc2)c1 ZINC000880562393 GF On-Demand Anodyne NAMPT 27 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)cc2)C1 ZINC000880562405 DC On-Demand Anodyne EPHX2 15 40 COc1cncc(NC(=O)NCC(=O)N2CCCc3ccccc32)c1 ZINC000880562406 EE On-Demand Anodyne AVPR2 44 46 COc1cncc(NC(=O)NCc2ccccc2COC(C)C)c1 ZINC000880562410 EG On-Demand Anodyne ROCK2 17 44 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880562434 FH On-Demand Anodyne PDGFRB 34 41 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880562434 FH On-Demand Anodyne SLC18A3 37 44 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880562434 FH On-Demand Anodyne FAAH 18 40 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880562434 FH On-Demand Anodyne SCN10A 43 40 COc1cncc(NC(=O)NCCOc2ccccc2C)c1 ZINC000880562448 DF On-Demand Anodyne ADRB1 43 33 COc1cncc(NC(=O)NCCOc2ccccc2C)c1 ZINC000880562448 DF On-Demand Anodyne HRH2 15 43 COc1cncc(NC(=O)NCCOc2ccccc2C)c1 ZINC000880562448 DF On-Demand Anodyne MTNR1A 36 43 COc1cncc(NC(=O)NCCOc2ccccc2C)c1 ZINC000880562448 DF On-Demand Anodyne MTNR1B 38 43 COc1cncc(NC(=O)N2CCN(C(=O)C3CCCCC3)CC2)c1 ZINC000880562453 EE On-Demand Anodyne PDGFRB 46 38 COc1cncc(NC(=O)NCCOC2CCCC2)c1 ZINC000880562455 CE On-Demand Anodyne ADRB1 15 49 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c1 ZINC000880562456 FG On-Demand Anodyne GRIN2B 20 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c1 ZINC000880562456 FG On-Demand Anodyne PDE4A 16 43 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c1 ZINC000880562456 FG On-Demand Anodyne CCR3 22 41 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c1 ZINC000880562456 FG On-Demand Anodyne EPHX2 23 40 COc1cncc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c1 ZINC000880562456 FG On-Demand Anodyne SCD1 42 51 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(F)cc2C(F)(F)F)C1 ZINC000880562526 GD On-Demand Anodyne P2RX7 42 46 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OCC#N)C1 ZINC000880562538 DD On-Demand Mild PTGER1 41 37 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562546 FE On-Demand Anodyne PGC 46 36 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562546 FE On-Demand Anodyne CACNA1B 15 43 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562546 FE On-Demand Anodyne REN 71 41 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562546 FE On-Demand Anodyne POLG_HCV1 38 44 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562546 FE On-Demand Anodyne FPR1 48 41 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562547 FE On-Demand Anodyne PGC 46 36 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562547 FE On-Demand Anodyne CACNA1B 15 43 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562547 FE On-Demand Anodyne REN 71 41 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562547 FE On-Demand Anodyne POLG_HCV1 38 44 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880562547 FE On-Demand Anodyne FPR1 48 41 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne PDGFRB 27 46 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne TRPV1 24 40 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne ROCK1 20 41 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne ROCK2 39 50 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne FLT4 18 46 COc1cncc(NC(=O)NCc2ccc(C)c(OC)c2)c1 ZINC000880562552 DF On-Demand Anodyne NAMPT 31 40 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne DRD4 46 35 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne PDGFRB 51 45 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne NPY2R 21 50 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne CYP11B2 15 43 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne FAAH 21 49 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne TAAR1 31 40 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(OC)c3)CC2)c1 ZINC000880562553 FE On-Demand Anodyne KCNK3 21 42 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880562558 DG On-Demand Anodyne BMP1 28 41 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880562558 DG On-Demand Anodyne ROCK1 17 42 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880562558 DG On-Demand Anodyne ROCK2 24 51 COC(=O)[C@@]1(O)CCN(CCSc2ccccc2)C1 ZINC000880562565 CD On-Demand Anodyne SLC12A5 49 37 COc1cncc(NC(=O)N[C@H]2CCc3cc(F)ccc32)c1 ZINC000880562578 DG On-Demand Anodyne TRPV1 18 53 COc1cncc(NC(=O)N[C@@H]2CCc3cc(F)ccc32)c1 ZINC000880562579 DG On-Demand Anodyne TRPV1 18 53 COC(=O)[C@@]1(O)CCN(CCOc2ccc(SC)cc2)C1 ZINC000880562585 DD On-Demand Anodyne LTA4H 42 37 COC(=O)[C@@]1(O)CCN(CCOc2ccc(SC)cc2)C1 ZINC000880562585 DD On-Demand Anodyne MMP13 18 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(SC)cc2)C1 ZINC000880562585 DD On-Demand Anodyne PSMB1 41 35 COC(=O)[C@@]1(O)CCN(CCOc2cccc(S(C)(=O)=O)c2)C1 ZINC000880562587 EC On-Demand Anodyne MMP13 23 48 COC(=O)[C@@]1(O)CCN(CCOc2cccc(S(C)(=O)=O)c2)C1 ZINC000880562587 EC On-Demand Anodyne ADAM17 24 48 COC(=O)[C@@]1(O)CCN(CCOc2cccc(S(C)(=O)=O)c2)C1 ZINC000880562587 EC On-Demand Anodyne MMP9 18 48 COC(=O)[C@@]1(O)CCN(CC(=O)N(C)CCCOc2ccccc2)C1 ZINC000880562592 FC On-Demand Anodyne LTA4H 28 41 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne HTR1D 30 46 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne HTR1B 28 41 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne PDGFRB 41 38 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne NMBR 69 35 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne GHSR 55 36 COc1cncc(NC(=O)N2CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)c1 ZINC000880562597 GE On-Demand Anodyne AKT1 36 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)c(F)c2)C1 ZINC000880562608 ED On-Demand Anodyne MMP13 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)c(F)c2)C1 ZINC000880562608 ED On-Demand Anodyne MCHR2 45 35 COc1cncc(NC(=O)NCCNC(=O)C2CC2)c1 ZINC000880562617 CC On-Demand Anodyne MTNR1A 28 43 COc1cncc(NC(=O)NCCNC(=O)C2CC2)c1 ZINC000880562617 CC On-Demand Anodyne MTNR1B 23 42 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562620 FF On-Demand Anodyne DRD4 41 33 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562620 FF On-Demand Anodyne NPY2R 23 46 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562620 FF On-Demand Anodyne GRM5 21 50 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562620 FF On-Demand Anodyne FAAH 22 43 COc1cncc(NC(=O)N2CCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562620 FF On-Demand Anodyne EPHX2 17 42 COc1cncc(NC(=O)N2CCN(C(=O)N3CCCCC3)CC2)c1 ZINC000880562634 ED On-Demand Anodyne PDGFRB 43 37 COC(=O)[C@@]1(O)CCN(CCCc2cccc3ccccc23)C1 ZINC000880562661 DE On-Demand Anodyne ADRA1A 22 40 COC(=O)[C@@]1(O)CCN(CCCc2cccc3ccccc23)C1 ZINC000880562661 DE On-Demand Anodyne ADRA1B 17 40 COC(=O)[C@@]1(O)CCN(CCCc2cccc3ccccc23)C1 ZINC000880562661 DE On-Demand Anodyne DRD3 16 42 COC(=O)[C@@]1(O)CCN(CCCc2cccc3ccccc23)C1 ZINC000880562661 DE On-Demand Anodyne SIGMAR1 30 52 COC(=O)[C@@]1(O)CCN(CCCc2cccc3ccccc23)C1 ZINC000880562661 DE On-Demand Anodyne EBP 56 52 COc1cncc(NC(=O)NCc2cccnc2N2CCN(C)CC2)c1 ZINC000880562664 FD On-Demand Anodyne HTR1A 18 41 COc1cncc(NC(=O)NCc2cccnc2N2CCN(C)CC2)c1 ZINC000880562664 FD On-Demand Anodyne TRPV1 17 41 COc1cncc(NC(=O)NCc2cccnc2N2CCN(C)CC2)c1 ZINC000880562664 FD On-Demand Anodyne SCN2A 17 42 COc1cncc(NC(=O)NCc2cccnc2N2CCN(C)CC2)c1 ZINC000880562664 FD On-Demand Anodyne SCN10A 33 42 COc1cncc(NC(=O)NCc2cccnc2N2CCN(C)CC2)c1 ZINC000880562664 FD On-Demand Anodyne NAMPT 42 37 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(C)c(OC)c3)CC2)c1 ZINC000880562665 GE On-Demand Anodyne PDGFRB 66 44 COc1cncc(NC(=O)N(C)CCCOc2ccc(F)cc2)c1 ZINC000880562680 EG On-Demand Anodyne ROCK2 28 40 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C#N)c2)C1 ZINC000880562706 DC On-Demand Mild HRH2 37 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C#N)c2)C1 ZINC000880562706 DC On-Demand Mild HRH3 42 42 COC(=O)[C@@]1(O)CCN(CCCOc2cccc(C#N)c2)C1 ZINC000880562706 DC On-Demand Mild MEN1 42 36 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne P2RY12 16 43 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne PDGFRB 58 44 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne GRIN2B 43 43 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne PTPN2 20 40 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne SIGMAR1 15 44 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne CCR3 29 47 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne CHRNA7 26 46 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne FAAH 21 46 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne PTPN1 18 40 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne EPHX2 27 40 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne MCHR1 17 41 COc1cncc(NC(=O)N2CCC(COc3ccccc3)CC2)c1 ZINC000880562728 EG On-Demand Anodyne DGAT1 21 44 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne DRD4 16 45 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne GRIN2B 26 45 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne SIGMAR1 18 48 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne CCR3 34 41 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne CHRNA7 29 45 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne C3AR1 52 52 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne EPHX2 57 53 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne MCHR1 21 45 COc1cncc(NC(=O)NC2CCN(C(=O)CCc3ccccc3)CC2)c1 ZINC000880562744 GF On-Demand Anodyne CCR8 52 39 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2C)C1 ZINC000880562753 CD On-Demand Anodyne ADRA1D 16 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2C)C1 ZINC000880562753 CD On-Demand Anodyne ADRA1A 31 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2C)C1 ZINC000880562753 CD On-Demand Anodyne ADRA1B 21 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2C)C1 ZINC000880562753 CD On-Demand Anodyne EBP 39 42 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne HRH3 15 42 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP13 65 52 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne ADAM17 52 52 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP2 35 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP3 33 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP8 24 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP14 26 41 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP9 38 52 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne MMP1 35 52 COC(=O)[C@@]1(O)CCN(CCOc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880562759 EC On-Demand Anodyne PSMB1 40 34 COc1cncc(NC(=O)N2CCC(NC(=O)C3CCCCC3)CC2)c1 ZINC000880562760 FF On-Demand Anodyne EPHX2 40 44 COC(=O)[C@@]1(O)CCN(Cc2cc(C)nc3ccccc23)C1 ZINC000880562772 DD On-Demand Anodyne ADAM17 103 47 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne DRD4 19 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne F10 16 40 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne SIGMAR1 19 44 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne NPY1R 32 43 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne CCKAR 45 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne CCR3 32 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne CHRNA7 22 44 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne CCKBR 63 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562780 EE On-Demand Anodyne MCHR1 18 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne TSHR 41 31 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne DRD4 19 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne F10 16 40 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne SIGMAR1 19 44 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne NPY1R 32 43 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne CCKAR 45 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne CCR3 32 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne CHRNA7 22 44 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne CCKBR 63 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)c1 ZINC000880562781 EE On-Demand Anodyne MCHR1 18 41 COc1cncc(NC(=O)N2CCC[C@H]2c2cccc(F)c2)c1 ZINC000880562782 DH On-Demand Anodyne GRIN2B 20 40 COc1cncc(NC(=O)N2CCC[C@H]2c2cccc(F)c2)c1 ZINC000880562782 DH On-Demand Anodyne CCR3 20 43 COc1cncc(NC(=O)N2CCC[C@@H]2c2cccc(F)c2)c1 ZINC000880562783 DH On-Demand Anodyne GRIN2B 20 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2cccc(F)c2)c1 ZINC000880562783 DH On-Demand Anodyne CCR3 20 43 COC(=O)[C@@]1(O)CCN(CCOc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880562787 ED On-Demand Anodyne MAOA 63 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880562787 ED On-Demand Anodyne ACHE 24 48 COC(=O)[C@@]1(O)CCN(CCOc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880562787 ED On-Demand Anodyne MAOB 52 49 COC(=O)[C@@]1(O)CCN(CCOc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880562787 ED On-Demand Anodyne BCHE 22 48 COc1cncc(NC(=O)N[C@H]2CCc3c(F)cccc32)c1 ZINC000880562789 DG On-Demand Anodyne TRPV1 21 43 COc1cncc(NC(=O)N[C@@H]2CCc3c(F)cccc32)c1 ZINC000880562790 DG On-Demand Anodyne TRPV1 21 43 COc1cncc(NC(=O)NCc2ccc(OC)c(OC)c2OC)c1 ZINC000880562793 EE On-Demand Anodyne PDGFRB 41 39 COc1cncc(NC(=O)NCc2ccc(OC)c(OC)c2OC)c1 ZINC000880562793 EE On-Demand Anodyne ROCK2 15 51 COc1cncc(NC(=O)NCc2ccc(OC)c(OC)c2OC)c1 ZINC000880562793 EE On-Demand Anodyne PDGFRA 42 37 COc1cncc(NC(=O)N2CCN(CC3CC3)CC2)c1 ZINC000880562796 CD On-Demand Anodyne PDGFRB 52 39 COc1cncc(NC(=O)N2CCN(CC3CC3)CC2)c1 ZINC000880562796 CD On-Demand Anodyne CCR3 20 47 COc1cncc(NC(=O)N2CCN(CC3CC3)CC2)c1 ZINC000880562796 CD On-Demand Anodyne FAAH 17 45 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562801 GF On-Demand Anodyne F2 43 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562801 GF On-Demand Anodyne GRIN2B 20 43 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562801 GF On-Demand Anodyne TRY1_BOVIN 49 34 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562801 GF On-Demand Anodyne PREP 53 56 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562801 GF On-Demand Anodyne TMPRSS11D 69 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562802 GF On-Demand Anodyne F2 43 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562802 GF On-Demand Anodyne GRIN2B 20 43 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562802 GF On-Demand Anodyne TRY1_BOVIN 49 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562802 GF On-Demand Anodyne PREP 53 56 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880562802 GF On-Demand Anodyne TMPRSS11D 69 41 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880562810 FD On-Demand Anodyne HCN1 50 34 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880562810 FD On-Demand Anodyne HCN4 42 34 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880562811 FD On-Demand Anodyne HCN1 50 34 CCOc1ccccc1[C@@H](CC)NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880562811 FD On-Demand Anodyne HCN4 42 34 CCOc1ccccc1[C@H](CC)NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880562812 FD On-Demand Anodyne HCN1 50 34 CCOc1ccccc1[C@H](CC)NC(=O)CN1CC[C@](O)(C(=O)OC)C1 ZINC000880562812 FD On-Demand Anodyne HCN4 42 34 CCOc1ccccc1[C@H](CC)NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880562813 FD On-Demand Anodyne HCN1 50 34 CCOc1ccccc1[C@H](CC)NC(=O)CN1CC[C@@](O)(C(=O)OC)C1 ZINC000880562813 FD On-Demand Anodyne HCN4 42 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)c(Cl)c2)C1 ZINC000880562818 ED On-Demand Anodyne MCHR1 20 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCCCC3)nc2)C1 ZINC000880562821 FC On-Demand Anodyne SLC27A1 47 40 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne DRD4 33 48 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne ACHE 18 43 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne HRH2 15 40 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne KCNH2 15 44 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne HTR4 22 41 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne SIGMAR1 27 56 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne SSTR5 78 44 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne CCR3 68 44 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne CHRNA7 16 46 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne SLC6A5 28 41 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne EPHX2 48 47 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne PDK1 55 47 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne CXCR3 34 54 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne MCHR1 65 57 COc1cncc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c1 ZINC000880562825 EE On-Demand Anodyne CCR8 19 43 COCCCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880562826 EH On-Demand Anodyne ROCK1 15 45 COCCCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880562826 EH On-Demand Anodyne ROCK2 32 45 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(O)c2)c1 ZINC000880562828 DE On-Demand Anodyne INHA 47 35 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(O)c2)c1 ZINC000880562828 DE On-Demand Anodyne ROCK2 24 48 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(O)c2)c1 ZINC000880562828 DE On-Demand Anodyne MT-ND1 17 40 COc1cncc(NC(=O)N[C@H]2CCCN(C)C2)c1 ZINC000880562829 CD On-Demand Anodyne CCR3 37 41 COc1cncc(NC(=O)N[C@@H]2CCCN(C)C2)c1 ZINC000880562830 CD On-Demand Anodyne CCR3 37 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(-c3csc(C)n3)c2)C1 ZINC000880562831 GD On-Demand Anodyne ACOX1 49 41 COc1cncc(NC(=O)NCCCNc2ccccn2)c1 ZINC000880562833 DE On-Demand Anodyne ADRB1 40 31 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2cc(Cl)ccc2OC)C1 ZINC000880562835 FC On-Demand Anodyne CPT1A 24 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(C)cc3)CC2)c1 ZINC000880562839 FE On-Demand Anodyne PDGFRB 49 45 COC(=O)[C@@]1(O)CCN([C@@H](C(N)=O)c2ccccc2)C1 ZINC000880562846 CB On-Demand Anodyne OPRL1 26 45 COC(=O)[C@@]1(O)CCN([C@H](C(N)=O)c2ccccc2)C1 ZINC000880562849 CB On-Demand Anodyne OPRL1 26 45 COc1cncc(NC(=O)N(C)Cc2ccc(C)cc2)c1 ZINC000880562850 CG On-Demand Anodyne ROCK2 26 49 COc1cncc(NC(=O)NC[C@@H](C)CN2CCCCC2)c1 ZINC000880562851 DE On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NC[C@H](C)CN2CCCCC2)c1 ZINC000880562852 DE On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562853 GG On-Demand Anodyne HRH3 24 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562853 GG On-Demand Anodyne NPY2R 21 44 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562853 GG On-Demand Anodyne GRM5 20 48 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562853 GG On-Demand Anodyne FAAH 21 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(Cl)c3)CC2)c1 ZINC000880562853 GG On-Demand Anodyne EPHX2 19 41 COc1cncc(NC(=O)NC[C@@H]2COc3ccccc3C2)c1 ZINC000880562862 DE On-Demand Anodyne ROCK2 29 41 COc1cncc(NC(=O)NC[C@H]2COc3ccccc3C2)c1 ZINC000880562863 DE On-Demand Anodyne ROCK2 29 41 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccccc2-c2ccccc2)C1 ZINC000880562870 FE On-Demand Anodyne CHRM3 22 46 COC(=O)[C@@]1(O)CCN(Cc2nc3ccccc3c(=O)n2C)C1 ZINC000880562876 DC On-Demand Anodyne HTR7 20 41 COC(=O)[C@@]1(O)CCN(Cc2nc3ccccc3c(=O)n2C)C1 ZINC000880562876 DC On-Demand Anodyne HIF1A 19 41 COc1cncc(NC(=O)N2CCN(CC(F)(F)F)CC2)c1 ZINC000880562883 DD On-Demand Anodyne PDGFRB 44 36 COc1cncc(NC(=O)N2CCN(CC(F)(F)F)CC2)c1 ZINC000880562883 DD On-Demand Anodyne FAAH 15 45 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)CN(C)C)c1 ZINC000880562884 EE On-Demand Anodyne NPY5R 20 40 COc1cncc(NC(=O)N[C@@H](Cc2ccccc2)CN(C)C)c1 ZINC000880562884 EE On-Demand Anodyne CYP3A4 16 40 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)CN(C)C)c1 ZINC000880562885 EE On-Demand Anodyne NPY5R 20 40 COc1cncc(NC(=O)N[C@H](Cc2ccccc2)CN(C)C)c1 ZINC000880562885 EE On-Demand Anodyne CYP3A4 16 40 COC(=O)[C@@]1(O)CCN(Cc2nc(C)c3ccccc3n2)C1 ZINC000880562887 DD On-Demand Anodyne ADAM17 63 36 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean PIK3CA 42 39 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean ROCK2 17 42 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean MTOR 72 39 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean EPHX2 22 40 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean FLT3 15 40 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean EPHB4 59 42 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean STAT6 61 38 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880562888 EE On-Demand Clean NAMPT 55 47 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Oc3ccccc3)cc2)C1 ZINC000880562890 FE On-Demand Anodyne LTA4H 62 53 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Oc3ccccc3)cc2)C1 ZINC000880562890 FE On-Demand Anodyne ACOX1 31 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Oc3ccccc3)cc2)C1 ZINC000880562890 FE On-Demand Anodyne FAAH 18 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Oc3ccccc3)cc2)C1 ZINC000880562890 FE On-Demand Anodyne EPHX2 17 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Oc3ccccc3)cc2)C1 ZINC000880562890 FE On-Demand Anodyne MCHR1 18 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880562911 GC On-Demand Anodyne HRH2 25 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880562911 GC On-Demand Anodyne GALR3 52 32 COC(=O)[C@@]1(O)CCN(CC(=O)NCCOc2cccc(C(F)(F)F)c2)C1 ZINC000880562911 GC On-Demand Anodyne PDS 44 41 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne HTR1A 17 48 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne DRD2 15 47 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne DRD4 46 35 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne SIGMAR1 42 55 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne MMP13 22 47 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne MTNR1A 40 49 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne MTNR1B 42 49 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne EBP 53 44 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne ABCB1 24 44 COC(=O)[C@@]1(O)CCN(CCCc2cccc(OC)c2)C1 ZINC000880562913 CD On-Demand Anodyne CRTM 49 33 COc1cncc(NC(=O)N[C@H]2COc3ccccc3C2)c1 ZINC000880562923 CE On-Demand Anodyne ROCK2 26 42 COc1cncc(NC(=O)N[C@@H]2COc3ccccc3C2)c1 ZINC000880562924 CE On-Demand Anodyne ROCK2 26 42 COc1cncc(NC(=O)NCCc2cc(OC)ccc2OC)c1 ZINC000880562927 EE On-Demand Anodyne NQO2 39 40 COc1cncc(NC(=O)NCCc2cc(OC)ccc2OC)c1 ZINC000880562927 EE On-Demand Anodyne RAF1 25 40 COc1cncc(NC(=O)NCCc2cc(OC)ccc2OC)c1 ZINC000880562927 EE On-Demand Anodyne MTNR1A 93 46 COc1cncc(NC(=O)NCCc2cc(OC)ccc2OC)c1 ZINC000880562927 EE On-Demand Anodyne MTNR1B 78 52 COc1cncc(NC(=O)NCCc2cc(OC)ccc2OC)c1 ZINC000880562927 EE On-Demand Anodyne QPCT 15 41 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne HTR1A 23 48 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne DRD2 27 43 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne DRD4 23 43 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne ACHE 21 40 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne ADRA1D 21 41 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne ADRA1A 38 41 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne ADRA1B 26 41 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne DRD3 35 43 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne LTA4H 44 38 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne HRH3 55 49 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne SIGMAR1 41 44 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne MMP13 21 52 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne ADAM17 19 50 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne PLA2G4B 69 34 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne MMP9 18 52 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne EPHX2 22 42 COC(=O)[C@@]1(O)CCN(CCCCOc2ccccc2)C1 ZINC000880562950 CD On-Demand Anodyne SLC12A5 55 37 COC(=O)[C@@]1(O)CCN(CCc2nc(-c3cccc(Cl)c3)no2)C1 ZINC000880562965 FD On-Demand Anodyne GRM5 18 48 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(F)c(Cl)c2)C1 ZINC000880562998 ED On-Demand Anodyne ERBB4 41 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(F)c(Cl)c2)C1 ZINC000880562998 ED On-Demand Anodyne MCHR1 43 44 O=C(CCCc1ccsc1)NCc1cn(C2CCC2)nn1 ZINC000880562999 DF On-Demand Anodyne PREP 17 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3)CC2)c1 ZINC000880563000 FE On-Demand Anodyne PDGFRB 42 44 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3)CC2)c1 ZINC000880563000 FE On-Demand Anodyne NPY2R 24 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3)CC2)c1 ZINC000880563000 FE On-Demand Anodyne FAAH 19 46 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3)CC2)c1 ZINC000880563000 FE On-Demand Anodyne SMO 22 42 COc1cncc(NC(=O)N[C@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000880563001 EF On-Demand Anodyne PDE4A 15 42 COc1cncc(NC(=O)N[C@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000880563001 EF On-Demand Anodyne ENPP1 57 33 COc1cncc(NC(=O)N[C@@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000880563002 EF On-Demand Anodyne PDE4A 15 42 COc1cncc(NC(=O)N[C@@H](C)c2ccc(OC)c(OC)c2)c1 ZINC000880563002 EF On-Demand Anodyne ENPP1 57 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccccc2Cc2ccccc2)C1 ZINC000880563014 GE On-Demand Anodyne SLC12A5 44 36 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccccc2Cc2ccccc2)C1 ZINC000880563015 GE On-Demand Anodyne SLC12A5 44 36 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne CPT1A 25 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne ROCK1 22 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne ROCK2 15 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne HDAC9 15 47 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne TRPA1 15 48 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000880563018 FD On-Demand Anodyne SLC12A5 22 41 COc1cncc(NC(=O)N(C)Cc2cc(OC)cc(OC)c2)c1 ZINC000880563020 EF On-Demand Anodyne ROCK2 23 49 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OC)c(OC)c2)C1 ZINC000880563025 FC On-Demand Anodyne ENPP1 70 34 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OC)c(OC)c2)C1 ZINC000880563028 FC On-Demand Anodyne ENPP1 70 34 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(C)cn3)CC2)c1 ZINC000880563031 FF On-Demand Anodyne NPY5R 15 41 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(C)cn3)CC2)c1 ZINC000880563031 FF On-Demand Anodyne EPHX2 25 42 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(C)cn3)CC2)c1 ZINC000880563031 FF On-Demand Anodyne LUCI_LUCLA 17 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2Cl)C1 ZINC000880563041 DC On-Demand Anodyne EPHB3 42 34 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne DRD4 42 33 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne HRH2 50 49 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne HTR2A 21 41 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne AVPR1B 25 40 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne LTA4H 18 41 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne CASR 31 42 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne MAPK14 17 40 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne SRC 24 45 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne CCR3 22 43 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne CHRNA7 17 41 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne AURKB 15 49 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne ROCK1 41 46 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne KDR 20 48 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne ROCK2 53 51 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne MAP2K1 15 40 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne EPHX2 37 52 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne FLT3 25 48 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne AURKA 21 49 COc1cncc(NC(=O)NCc2cccc(OCCN3CCOCC3)c2)c1 ZINC000880563045 GE On-Demand Anodyne NAMPT 46 43 COc1cncc(NC(=O)NCCN2CCc3sccc3C2)c1 ZINC000880563046 EE On-Demand Anodyne DRD4 42 33 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c1 ZINC000880563057 GF On-Demand Anodyne GRIN2B 23 49 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c1 ZINC000880563057 GF On-Demand Anodyne CCR3 61 47 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c1 ZINC000880563057 GF On-Demand Anodyne CACNA1G 40 45 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c1 ZINC000880563057 GF On-Demand Anodyne NAMPT 40 35 COc1cncc(NC(=O)N2CCCN(c3ccc(C)cc3)CC2)c1 ZINC000880563060 EG On-Demand Anodyne DRD4 24 40 COc1cncc(NC(=O)N2CCCN(c3ccc(C)cc3)CC2)c1 ZINC000880563060 EG On-Demand Anodyne PDGFRB 50 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000880563062 GD On-Demand Anodyne MCHR1 25 46 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000880563062 GD On-Demand Anodyne IMDH_CRYPV 22 42 COc1cncc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000880563065 EE On-Demand Anodyne ADRB2 27 42 COc1cncc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000880563065 EE On-Demand Anodyne ADRB1 59 42 COc1cncc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000880563065 EE On-Demand Anodyne ADRB3 20 42 COc1cncc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000880563066 EE On-Demand Anodyne ADRB2 27 42 COc1cncc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000880563066 EE On-Demand Anodyne ADRB1 59 42 COc1cncc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000880563066 EE On-Demand Anodyne ADRB3 20 42 COc1cncc(NC(=O)N2CCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880563069 FE On-Demand Mild PDGFRB 50 45 COc1cncc(NC(=O)N2CCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880563069 FE On-Demand Mild MLNR 29 42 COc1cncc(NC(=O)N2CCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880563069 FE On-Demand Mild FAAH 32 57 COc1cncc(NC(=O)N2CCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880563069 FE On-Demand Mild MCHR1 20 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)C1 ZINC000880563076 GD On-Demand Anodyne MPL 27 45 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne MMP13 20 43 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne MMP3 23 43 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne MMP9 20 43 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne PKM 15 41 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne TGM2 80 40 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne MMP1 23 48 COc1cncc(NC(=O)N2CCCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880563083 GE On-Demand Anodyne F13A1 97 45 COc1cncc(NC(=O)N(Cc2ccccc2OC)C2CC2)c1 ZINC000880563086 EG On-Demand Anodyne TSPO 44 38 COc1cncc(NC(=O)N(Cc2ccccc2OC)C2CC2)c1 ZINC000880563086 EG On-Demand Anodyne ROCK2 21 48 COc1cncc(NC(=O)N(Cc2ccccc2OC)C2CC2)c1 ZINC000880563086 EG On-Demand Anodyne MBTPS1 51 35 COc1cncc(NC(=O)N(Cc2cccc(F)c2)C2CC2)c1 ZINC000880563090 DG On-Demand Anodyne ROCK1 18 40 COc1cncc(NC(=O)N(Cc2cccc(F)c2)C2CC2)c1 ZINC000880563090 DG On-Demand Anodyne ROCK2 30 56 COC(=O)[C@@]1(O)CCN(CCc2nc(-c3ccccc3)no2)C1 ZINC000880563099 DC On-Demand Anodyne NPPA 19 42 COC(=O)[C@@]1(O)CCN([C@@H]2CCCc3ccccc32)C1 ZINC000880563122 CD On-Demand Anodyne OPRL1 20 45 COC(=O)[C@@]1(O)CCN([C@@H]2CCCc3ccccc32)C1 ZINC000880563122 CD On-Demand Anodyne HTR7 15 40 COC(=O)[C@@]1(O)CCN([C@H]2CCCc3ccccc32)C1 ZINC000880563123 CD On-Demand Anodyne OPRL1 20 45 COC(=O)[C@@]1(O)CCN([C@H]2CCCc3ccccc32)C1 ZINC000880563123 CD On-Demand Anodyne HTR7 15 40 COc1cncc(NC(=O)N2CCC[C@@H](C(=O)NCC3CC3)C2)c1 ZINC000880563136 ED On-Demand Anodyne CCR3 15 44 COc1cncc(NC(=O)N2CCC[C@H](C(=O)NCC3CC3)C2)c1 ZINC000880563137 ED On-Demand Anodyne CCR3 15 44 COc1cncc(NC(=O)N(Cc2ccc(C(N)=O)cc2)C2CC2)c1 ZINC000880563152 EE On-Demand Anodyne GIPR 45 42 CC(C)(C)OC(=O)N1CCC(CCC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880563166 GG On-Demand Anodyne GPR119 47 39 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR1A 47 60 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne ADRA1D 29 41 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR1D 22 60 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR1B 34 60 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR2A 16 43 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR2C 17 43 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne ADRA1A 23 41 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne ADRA1B 19 41 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne DRD3 46 38 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne PDGFRB 55 46 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne HTR7 38 48 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne FAAH 22 46 COc1cncc(NC(=O)N2CCN(c3ccccc3C)CC2)c1 ZINC000880563167 EF On-Demand Anodyne RBP4 17 45 COc1cncc(NC(=O)N(C)Cc2ccc(C(=O)NC3CC3)cc2)c1 ZINC000880563170 FF On-Demand Anodyne MAPK14 27 43 COc1cncc(NC(=O)N(C)Cc2ccc(C(=O)NC3CC3)cc2)c1 ZINC000880563170 FF On-Demand Anodyne ROCK2 15 41 COc1cncc(NC(=O)N(C)Cc2ccc(C(=O)NC3CC3)cc2)c1 ZINC000880563170 FF On-Demand Anodyne MCHR1 20 40 COc1cncc(NC(=O)N(C)Cc2ccc(C(=O)NC3CC3)cc2)c1 ZINC000880563170 FF On-Demand Anodyne GIPR 56 34 COC(=O)[C@@]1(O)CCN(CCc2ccc3c(c2)CCO3)C1 ZINC000880563178 CC On-Demand Anodyne KCNJ1 49 37 O=C(NCc1cn(C2CCC2)nn1)c1cnc2ccccn12 ZINC000880563183 CD On-Demand Anodyne EPHB3 22 43 COc1cncc(NC(=O)N(C)CCOc2ccccc2OC)c1 ZINC000880563193 EF On-Demand Anodyne TSPO 40 31 COc1cncc(NC(=O)N(C)CCOc2ccccc2OC)c1 ZINC000880563193 EF On-Demand Anodyne ROCK2 26 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563195 GC On-Demand Anodyne MMP13 20 41 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563195 GC On-Demand Anodyne MMP2 23 41 COC(=O)[C@@]1(O)CCN(Cc2cc(=O)oc3cc(OC)ccc23)C1 ZINC000880563206 EC On-Demand Anodyne CYP11B1 17 42 COC(=O)[C@@]1(O)CCN(Cc2cc(=O)oc3cc(OC)ccc23)C1 ZINC000880563206 EC On-Demand Anodyne MAOB 28 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2nc3ccc(F)cc3s2)C1 ZINC000880563222 FD On-Demand Anodyne CSNK1D 40 39 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2nc3ccc(F)cc3s2)C1 ZINC000880563223 FD On-Demand Anodyne CSNK1D 40 39 COC(=O)[C@@]1(O)CCN(CC(=O)NCCc2nc3ccccc3s2)C1 ZINC000880563233 FC On-Demand Anodyne ACOX1 49 33 COc1cncc(NC(=O)N2CCC(CNC(C)=O)CC2)c1 ZINC000880563234 DD On-Demand Anodyne CACNA1I 54 31 COc1cncc(NC(=O)N(C)Cc2ccc(OC)cc2OC)c1 ZINC000880563235 EF On-Demand Anodyne PDGFRB 40 40 COc1cncc(NC(=O)N(C)Cc2ccc(OC)cc2OC)c1 ZINC000880563235 EF On-Demand Anodyne ROCK2 19 43 COc1cncc(NC(=O)N(C)Cc2ccc(OC)cc2OC)c1 ZINC000880563235 EF On-Demand Anodyne CSF1R 16 40 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne DRD3 15 43 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne NPY1R 22 40 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne CCR3 22 40 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne CHRNA7 15 42 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne EPHX2 52 47 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne CXCR3 16 43 COc1cncc(NC(=O)NC2CCN(c3ccccc3)CC2)c1 ZINC000880563246 EF On-Demand Anodyne MCHR1 19 43 COc1cncc(NC(=O)N2CCC(NC(=O)C(C)C)CC2)c1 ZINC000880563248 DD On-Demand Anodyne EPHX2 25 41 CCCOc1ncccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880563251 DF On-Demand Anodyne ROCK2 16 43 CCCOc1ncccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880563251 DF On-Demand Anodyne SCN10A 27 43 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne HRH2 30 48 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne CCR3 29 40 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne NPFFR2 19 41 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne AURKB 20 40 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne ROCK1 31 45 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne ROCK2 44 48 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne FAAH 23 41 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne EPHX2 27 41 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne MCHR1 21 45 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne AURKA 19 41 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne NPFFR1 22 41 COc1cncc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c1 ZINC000880563252 FE On-Demand Anodyne NAMPT 46 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC)cc2)C1 ZINC000880563258 DC On-Demand Anodyne MMP9 17 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC)cc2)C1 ZINC000880563258 DC On-Demand Anodyne EPHX2 15 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC)cc2)C1 ZINC000880563258 DC On-Demand Anodyne CA9 20 42 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563259 EF On-Demand Anodyne EPHX2 55 49 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563259 EF On-Demand Anodyne CXCR3 17 41 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@@H](C)c2ccc(Cl)cc2Cl)C1 ZINC000880563263 GD On-Demand Anodyne CCR1 44 34 COC(=O)[C@@]1(O)CCN(CC(=O)N[C@H](C)c2ccc(Cl)cc2Cl)C1 ZINC000880563265 GD On-Demand Anodyne CCR1 44 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne TSHR 50 36 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne PDGFRB 16 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne LTA4H 59 53 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne MMP13 20 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne ADAM17 54 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne FAAH 15 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne MMP9 20 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne EPHX2 15 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563274 GD On-Demand Anodyne SLC12A5 68 41 COc1cncc(NC(=O)NCCc2cccc(OC)c2OC)c1 ZINC000880563275 EE On-Demand Anodyne NQO2 56 46 COc1cncc(NC(=O)NCCc2cccc(OC)c2OC)c1 ZINC000880563275 EE On-Demand Anodyne MTNR1A 96 49 COc1cncc(NC(=O)NCCc2cccc(OC)c2OC)c1 ZINC000880563275 EE On-Demand Anodyne MTNR1B 77 46 COc1cncc(NC(=O)NCCc2cccc(OC)c2OC)c1 ZINC000880563275 EE On-Demand Anodyne PDGFRA 45 38 COc1cncc(NC(=O)NCc2ccc(CS(C)(=O)=O)cc2)c1 ZINC000880563278 ED On-Demand Anodyne ROCK2 25 45 COc1cncc(NC(=O)NCc2ccc(CS(C)(=O)=O)cc2)c1 ZINC000880563278 ED On-Demand Anodyne CA9 21 40 COc1cncc(NC(=O)NCc2ccc(CS(C)(=O)=O)cc2)c1 ZINC000880563278 ED On-Demand Anodyne PRMT3 18 41 COc1cncc(NC(=O)NCc2ccc(CS(C)(=O)=O)cc2)c1 ZINC000880563278 ED On-Demand Anodyne NAMPT 54 43 COc1cncc(NC(=O)N2CCN(CC(C)C)CC2)c1 ZINC000880563283 CD On-Demand Anodyne PDGFRB 46 37 COC(=O)[C@@]1(O)CCN(Cc2cnc(Cl)s2)C1 ZINC000880563295 CC On-Demand Anodyne MGEA5 33 42 COc1cncc(NC(=O)N2CCC[C@H]2Cc2cccc(F)c2)c1 ZINC000880563300 EG On-Demand Anodyne CCR3 61 44 COc1cncc(NC(=O)N2CCC[C@H]2Cc2cccc(F)c2)c1 ZINC000880563300 EG On-Demand Anodyne CHRNA7 25 45 COc1cncc(NC(=O)N2CCC[C@H]2Cc2cccc(F)c2)c1 ZINC000880563300 EG On-Demand Anodyne ACKR3 52 34 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)c1 ZINC000880563301 EG On-Demand Anodyne CCR3 61 44 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)c1 ZINC000880563301 EG On-Demand Anodyne CHRNA7 25 45 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)c1 ZINC000880563301 EG On-Demand Anodyne ACKR3 52 34 COc1cncc(NC(=O)N2CCC(C(=O)NCC(F)(F)F)CC2)c1 ZINC000880563308 FE On-Demand Anodyne CACNA1G 35 41 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000880563309 FG On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000880563309 FG On-Demand Anodyne DPP7 23 41 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000880563309 FG On-Demand Anodyne L3MBTL3 41 32 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000880563309 FG On-Demand Anodyne HPGD 31 40 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000880563309 FG On-Demand Anodyne NAMPT 57 58 COC(=O)[C@@]1(O)CCN(CC[C@@H]2CCOC2=O)C1 ZINC000880563327 CB On-Demand Anodyne TRAR 41 31 COC(=O)[C@@]1(O)CCN(CC[C@H]2CCOC2=O)C1 ZINC000880563329 CB On-Demand Anodyne TRAR 41 31 COC(=O)[C@@]1(O)CCN(CCCc2ccc(C(F)(F)F)cc2)C1 ZINC000880563335 EE On-Demand Anodyne SLC12A5 22 40 COC(=O)[C@@]1(O)CCN(CC(=O)NC2(c3ccccc3)CCC2)C1 ZINC000880563341 EC On-Demand Anodyne ADRA1A 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2C(=O)c2ccccc2)C1 ZINC000880563347 GD On-Demand Anodyne ABCB1 15 42 COc1cncc(NC(=O)N2CCN(C(=O)c3ccsc3)CC2)c1 ZINC000880563356 EE On-Demand Anodyne NPBWR1 73 31 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@@H](c2ccccc2)c2cccs2)C1 ZINC000880563357 GD On-Demand Anodyne PRCP 21 41 COC(=O)[C@@]1(O)CCN(CCC(=O)N[C@H](c2ccccc2)c2cccs2)C1 ZINC000880563360 GD On-Demand Anodyne PRCP 21 41 COc1cncc(NC(=O)NCCCCOCCc2ccccc2)c1 ZINC000880563376 EG On-Demand Anodyne HRH2 24 42 COc1cncc(NC(=O)NCCCCOCCc2ccccc2)c1 ZINC000880563376 EG On-Demand Anodyne CCR3 24 46 COc1cncc(NC(=O)NCCCCOCCc2ccccc2)c1 ZINC000880563376 EG On-Demand Anodyne MTNR1B 28 42 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)cc2)c1 ZINC000880563377 ED On-Demand Anodyne ADRB2 35 45 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)cc2)c1 ZINC000880563377 ED On-Demand Anodyne ADRB1 65 44 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)cc2)c1 ZINC000880563377 ED On-Demand Anodyne GRIN1 24 41 COc1cncc(NC(=O)NC[C@@H](O)COc2ccc(F)cc2)c1 ZINC000880563377 ED On-Demand Anodyne ADRB3 36 43 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)cc2)c1 ZINC000880563378 ED On-Demand Anodyne ADRB2 35 45 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)cc2)c1 ZINC000880563378 ED On-Demand Anodyne ADRB1 65 44 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)cc2)c1 ZINC000880563378 ED On-Demand Anodyne GRIN1 24 41 COc1cncc(NC(=O)NC[C@H](O)COc2ccc(F)cc2)c1 ZINC000880563378 ED On-Demand Anodyne ADRB3 36 43 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne PDGFRB 43 43 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne MTNR1A 50 34 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne MTNR1B 44 41 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne ROCK2 19 64 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne FLT4 21 43 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne CSF1R 18 43 COc1cncc(NC(=O)NCc2ccc(OC)cc2OC)c1 ZINC000880563383 DE On-Demand Anodyne LUCI_LUCLA 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)c3ccc(C)cc3)cc2)C1 ZINC000880563388 GD On-Demand Anodyne MMP13 38 54 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)c3ccc(C)cc3)cc2)C1 ZINC000880563388 GD On-Demand Anodyne ADAM17 36 54 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)c3ccc(C)cc3)cc2)C1 ZINC000880563388 GD On-Demand Anodyne MMP2 24 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)c3ccc(C)cc3)cc2)C1 ZINC000880563388 GD On-Demand Anodyne MMP9 24 54 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NCCc2ccc3c(c2)OCCO3)C1 ZINC000880563399 GC On-Demand Anodyne BMP1 51 36 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NCCc2ccc3c(c2)OCCO3)C1 ZINC000880563401 GC On-Demand Anodyne BMP1 51 36 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc3c(c2)OCO3)C1 ZINC000880563404 EB On-Demand Anodyne EDNRB 43 39 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc3c(c2)OCO3)C1 ZINC000880563404 EB On-Demand Anodyne EDNRA 46 39 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc3c(c2)OCO3)C1 ZINC000880563404 EB On-Demand Anodyne BMP1 61 37 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc3c(c2)OCO3)C1 ZINC000880563404 EB On-Demand Anodyne NOS2 100 38 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc3c(c2)OCO3)C1 ZINC000880563404 EB On-Demand Anodyne MCHR1 19 46 COC(=O)[C@@]1(O)CCN(CCC(=O)NC(c2ccccc2)c2ccccc2)C1 ZINC000880563405 GD On-Demand Anodyne PRCP 25 46 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC)c(Cl)c2)C1 ZINC000880563416 EC On-Demand Anodyne ENPP1 69 34 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CHRM2 22 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CHRM1 17 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne DRD2 21 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne DRD4 47 47 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne ACHE 40 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne KCNH2 16 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CHRM3 29 44 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne LTA4H 18 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne SIGMAR1 69 51 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne SSTR5 57 38 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CCR3 27 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne SLC6A5 19 42 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne PDK1 41 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne MCHR1 45 52 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CACNA1G 24 43 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563423 GC On-Demand Anodyne CCR8 21 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CHRM2 22 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CHRM1 17 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne DRD2 21 48 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne DRD4 47 47 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne ACHE 40 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne KCNH2 16 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CHRM3 29 44 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne LTA4H 18 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne SIGMAR1 69 51 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne SSTR5 57 38 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CCR3 27 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne SLC6A5 19 42 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne PDK1 41 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne MCHR1 45 52 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CACNA1G 24 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)NC2CCN(Cc3ccccc3)CC2)C1 ZINC000880563425 GC On-Demand Anodyne CCR8 21 43 O=C(NCc1cn(C2CCC2)nn1)c1ccc(C(F)(F)F)cc1O ZINC000880563431 EF On-Demand Anodyne CCR2 55 35 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)c1 ZINC000880563437 GG On-Demand Anodyne F10 52 34 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)c1 ZINC000880563437 GG On-Demand Anodyne NPY5R 20 46 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)c1 ZINC000880563437 GG On-Demand Anodyne TYK2 33 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CC[C@](O)(C(=O)OC)C3)cc2)C1 ZINC000880563442 GB On-Demand Anodyne MMP13 19 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CC[C@](O)(C(=O)OC)C3)cc2)C1 ZINC000880563442 GB On-Demand Anodyne ADAM17 15 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CC[C@](O)(C(=O)OC)C3)cc2)C1 ZINC000880563442 GB On-Demand Anodyne MMP9 15 46 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CC[C@](O)(C(=O)OC)C3)cc2)C1 ZINC000880563442 GB On-Demand Anodyne MCHR2 44 34 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3=O)cc2)c1 ZINC000880563447 FF On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3=O)cc2)c1 ZINC000880563447 FF On-Demand Anodyne PROKR1 49 30 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3=O)cc2)c1 ZINC000880563447 FF On-Demand Anodyne NAMPT 41 42 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne DRD4 41 31 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne HRH2 20 42 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne DRD3 15 43 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne CCR3 39 40 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne FLT1 15 42 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne KDR 18 51 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne FAAH 18 44 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne FLT3 25 51 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne MCHR1 30 45 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne DDR2 19 40 COc1cncc(NC(=O)NCc2ccc(CN3CCN(C)CC3)cc2)c1 ZINC000880563452 FE On-Demand Anodyne NAMPT 51 39 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563453 GC On-Demand Anodyne PIK3CA 19 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563453 GC On-Demand Anodyne MTOR 40 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563453 GC On-Demand Anodyne PIK3CG 19 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563453 GC On-Demand Anodyne STAT6 52 35 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563454 GC On-Demand Anodyne PIK3CA 19 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563454 GC On-Demand Anodyne MTOR 40 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563454 GC On-Demand Anodyne PIK3CG 19 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563454 GC On-Demand Anodyne STAT6 52 35 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2cccnc2Cl)C1 ZINC000880563471 EC On-Demand Anodyne G2YM83_BOTF4 61 35 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2cccnc2Cl)C1 ZINC000880563474 EC On-Demand Anodyne G2YM83_BOTF4 61 35 COc1cncc(NC(=O)N(Cc2ccc(N(C)C)cc2)C2CC2)c1 ZINC000880563479 EG On-Demand Clean ROCK2 15 49 O=C(NCc1cn(C2CCC2)nn1)[C@@H](F)Cc1ccccc1 ZINC000880563480 DE On-Demand Anodyne ACE 44 36 O=C(NCc1cn(C2CCC2)nn1)[C@@H](F)Cc1ccccc1 ZINC000880563480 DE On-Demand Anodyne MME 49 36 O=C(NCc1cn(C2CCC2)nn1)[C@@H](F)Cc1ccccc1 ZINC000880563480 DE On-Demand Anodyne PREP 23 41 O=C(NCc1cn(C2CCC2)nn1)[C@H](F)Cc1ccccc1 ZINC000880563481 DE On-Demand Anodyne ACE 44 36 O=C(NCc1cn(C2CCC2)nn1)[C@H](F)Cc1ccccc1 ZINC000880563481 DE On-Demand Anodyne MME 49 36 O=C(NCc1cn(C2CCC2)nn1)[C@H](F)Cc1ccccc1 ZINC000880563481 DE On-Demand Anodyne PREP 23 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563487 FC On-Demand Anodyne PIK3CA 40 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563487 FC On-Demand Anodyne MTOR 83 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563487 FC On-Demand Anodyne EPHX2 15 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563487 FC On-Demand Anodyne PIK3CG 35 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880563487 FC On-Demand Anodyne STAT6 53 34 COc1cncc(NC(=O)N(CCO)Cc2ccccc2OC)c1 ZINC000880563491 EE On-Demand Anodyne TSPO 44 37 COc1cncc(NC(=O)N(CCO)Cc2ccccc2OC)c1 ZINC000880563491 EE On-Demand Anodyne ROCK2 24 47 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(Cl)cc2)C1 ZINC000880563495 ED On-Demand Anodyne CCR1 42 34 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(Cl)cc2)C1 ZINC000880563496 ED On-Demand Anodyne CCR1 42 34 COc1cncc(NC(=O)NCc2cccc(OCC(=O)N(C)C)c2)c1 ZINC000880563498 FD On-Demand Anodyne HRH2 19 41 COc1cncc(NC(=O)NCc2cccc(OCC(=O)N(C)C)c2)c1 ZINC000880563498 FD On-Demand Anodyne ROCK1 44 47 COc1cncc(NC(=O)NCc2cccc(OCC(=O)N(C)C)c2)c1 ZINC000880563498 FD On-Demand Anodyne ROCK2 63 54 COc1cncc(NC(=O)NCc2cccc(OCC(=O)N(C)C)c2)c1 ZINC000880563498 FD On-Demand Anodyne NAMPT 40 41 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000880563499 CF On-Demand Anodyne CHRNA7 16 44 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccn2)c1 ZINC000880563499 CF On-Demand Anodyne CPT1A 78 36 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000880563500 CF On-Demand Anodyne CHRNA7 16 44 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccn2)c1 ZINC000880563500 CF On-Demand Anodyne CPT1A 78 36 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne KCNQ2 32 41 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne ROCK1 25 57 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne MTNR1A 24 41 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne MTNR1B 28 43 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne ROCK2 26 57 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC)c2)c1 ZINC000880563503 DF On-Demand Anodyne F7 16 52 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne KCNQ2 32 41 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne ROCK1 25 57 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne MTNR1A 24 41 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne MTNR1B 28 43 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne ROCK2 26 57 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC)c2)c1 ZINC000880563504 DF On-Demand Anodyne F7 16 52 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)c(F)c2)c1 ZINC000880563510 FE On-Demand Clean NPY2R 59 36 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)c(F)c2)c1 ZINC000880563510 FE On-Demand Clean MTOR 44 38 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)c(F)c2)c1 ZINC000880563510 FE On-Demand Clean STAT6 42 31 COc1cncc(NC(=O)NCc2ccc(N3CCOCC3)c(F)c2)c1 ZINC000880563510 FE On-Demand Clean NAMPT 34 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc(-c3ccc(F)cc3)cs2)C1 ZINC000880563512 GD On-Demand Anodyne ROCK1 20 45 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2nccs2)C1 ZINC000880563514 CC On-Demand Anodyne MAP1 105 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2nccs2)C1 ZINC000880563515 CC On-Demand Anodyne MAP1 105 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000880563524 DB On-Demand Anodyne EDNRB 29 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000880563524 DB On-Demand Anodyne EDNRA 26 40 COc1cncc(NC(=O)NCCCCn2ccnc2)c1 ZINC000880563525 CD On-Demand Anodyne TBXAS1 49 45 COc1cncc(NC(=O)NCCCCn2ccnc2)c1 ZINC000880563525 CD On-Demand Anodyne QPCT 68 65 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3ccccc3C#N)cc2)C1 ZINC000880563533 EE On-Demand Mild AGTR1B 34 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(-c3ccccc3)cc2)C1 ZINC000880563535 FD On-Demand Anodyne LTA4H 28 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(-c3ccccc3)cc2)C1 ZINC000880563535 FD On-Demand Anodyne PRNP 43 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(-c3ccccc3)cc2)C1 ZINC000880563535 FD On-Demand Anodyne SLC1A2 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(-c3ccccc3)cc2)C1 ZINC000880563535 FD On-Demand Anodyne MCHR1 18 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Oc3ccccc3)c2)C1 ZINC000880563537 FE On-Demand Anodyne LTA4H 35 44 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Oc3ccccc3)c2)C1 ZINC000880563537 FE On-Demand Anodyne ACOX1 23 45 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Oc3ccccc3)c2)C1 ZINC000880563537 FE On-Demand Anodyne FAAH 20 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Oc3ccccc3)c2)C1 ZINC000880563537 FE On-Demand Anodyne EPHX2 19 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(Oc3ccccc3)c2)C1 ZINC000880563537 FE On-Demand Anodyne MCHR1 21 41 COC(=O)[C@@]1(O)CCN(Cc2cc3ccccc3o2)C1 ZINC000880563541 CD On-Demand Anodyne SIGMAR1 17 55 COc1cncc(NC(=O)N2CCC[C@@H](C(=O)Nc3ccc(Cl)cn3)C2)c1 ZINC000880563548 GG On-Demand Anodyne F10 50 33 COc1cncc(NC(=O)N2CCC[C@H](C(=O)Nc3ccc(Cl)cn3)C2)c1 ZINC000880563549 GG On-Demand Anodyne F10 50 33 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880563550 FF On-Demand Anodyne FAAH 15 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880563550 FF On-Demand Anodyne PARP1 22 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880563550 FF On-Demand Anodyne EPHX2 18 45 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@@H]2CCCO2)c1 ZINC000880563556 EG On-Demand Anodyne ROCK2 21 40 COc1cncc(NC(=O)N(Cc2ccccc2)C[C@H]2CCCO2)c1 ZINC000880563557 EG On-Demand Anodyne ROCK2 21 40 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563560 GE On-Demand Anodyne PDGFRB 57 45 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563560 GE On-Demand Anodyne HCN1 71 39 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563560 GE On-Demand Anodyne HCN4 57 38 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563560 GE On-Demand Anodyne KCNK3 46 45 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563560 GE On-Demand Anodyne KCNK9 35 45 COC(=O)[C@@]1(O)CCN(CCc2ccc(F)c(F)c2)C1 ZINC000880563564 CD On-Demand Anodyne ABCC1 107 42 COC(=O)[C@@]1(O)CCN(CCc2ccc(F)c(F)c2)C1 ZINC000880563564 CD On-Demand Anodyne ABCB1A 55 42 COc1cncc(NC(=O)NCc2cccc(OC)c2OC)c1 ZINC000880563571 DE On-Demand Anodyne PDGFRB 46 43 COc1cncc(NC(=O)NCc2cccc(OC)c2OC)c1 ZINC000880563571 DE On-Demand Anodyne MTNR1B 32 40 COc1cncc(NC(=O)NCc2cccc(OC)c2OC)c1 ZINC000880563571 DE On-Demand Anodyne ROCK2 27 61 COc1cncc(NC(=O)NCc2cccc(OC)c2OC)c1 ZINC000880563571 DE On-Demand Anodyne FLT4 27 43 COc1cncc(NC(=O)NCc2cccc(OC)c2OC)c1 ZINC000880563571 DE On-Demand Anodyne PDGFRA 48 39 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cc(Cl)c(OC)cc2OC)C1 ZINC000880563577 FC On-Demand Anodyne HTR4 48 41 COc1cncc(NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000880563578 DE On-Demand Anodyne TSPO 40 32 COc1cncc(NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000880563578 DE On-Demand Anodyne ROCK1 21 56 COc1cncc(NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000880563578 DE On-Demand Anodyne ROCK2 33 56 COc1cncc(NC(=O)N(CCO)Cc2ccccc2)c1 ZINC000880563578 DE On-Demand Anodyne PTGES 18 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)cn2)C1 ZINC000880563587 DC On-Demand Anodyne F10 52 35 COc1cncc(NC(=O)N(C)CCOc2cccc(C)c2)c1 ZINC000880563589 DF On-Demand Anodyne ROCK2 27 41 COc1cncc(NC(=O)N2CCCN(c3nccs3)CC2)c1 ZINC000880563590 EE On-Demand Anodyne PDGFRB 51 39 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563592 GC On-Demand Anodyne MMP13 21 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563592 GC On-Demand Anodyne MMP2 24 42 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563592 GC On-Demand Anodyne MMP14 20 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563592 GC On-Demand Anodyne MMP9 22 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563596 FD On-Demand Anodyne MMP13 20 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563596 FD On-Demand Anodyne P2RY1 68 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563596 FD On-Demand Anodyne MMP2 23 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563596 FD On-Demand Anodyne EPHX2 62 47 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000880563596 FD On-Demand Anodyne MCHR1 16 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cc(OC)c(Cl)cc2OC)C1 ZINC000880563602 FC On-Demand Anodyne HTR4 41 38 COc1cncc(NC(=O)N2CCC(CN3CCN(C)CC3)CC2)c1 ZINC000880563605 ED On-Demand Anodyne PDGFRB 42 36 COc1cncc(NC(=O)N2CCC(CN3CCN(C)CC3)CC2)c1 ZINC000880563605 ED On-Demand Anodyne CCR3 20 49 COc1cncc(NC(=O)NC2CCN(C(C)(C)C)CC2)c1 ZINC000880563606 DE On-Demand Anodyne EPHX2 48 41 COc1cncc(NC(=O)NC2CCN(C(C)(C)C)CC2)c1 ZINC000880563606 DE On-Demand Anodyne CXCR3 17 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3cccc(C)c3)s2)C1 ZINC000880563608 GD On-Demand Anodyne SCD 32 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3cccc(C)c3)s2)C1 ZINC000880563608 GD On-Demand Anodyne MGEA5 34 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(OC)c(OC)c2)C1 ZINC000880563617 EC On-Demand Anodyne ENPP1 84 41 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne HRH2 26 50 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne SCNN1A 25 42 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne MTNR1A 58 40 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne MTNR1B 49 40 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne PIK3CG 18 41 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne CA9 17 40 COc1ccc(OCCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880563632 EF On-Demand Anodyne QPCT 17 41 COc1cncc(NC(=O)N(C)CCc2ccc(F)cc2)c1 ZINC000880563638 DF On-Demand Anodyne ROCK2 24 41 COc1cncc(NC(=O)N(C)CCc2ccc(F)cc2)c1 ZINC000880563638 DF On-Demand Anodyne NPY5R 20 40 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cn3)CC2)c1 ZINC000880563639 ED On-Demand Mild PDGFRB 60 51 COc1cncc(NC(=O)N2CCN(c3ccc(C#N)cn3)CC2)c1 ZINC000880563639 ED On-Demand Mild DGAT1 31 43 CCC(=O)N1CCCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880563640 DD On-Demand Anodyne PDGFRB 43 36 COc1cncc(NC(=O)N2CCC(CC(=O)NC3CCCC3)CC2)c1 ZINC000880563641 FF On-Demand Anodyne EPHX2 24 42 COc1cncc(NC(=O)Nc2cnn(C[C@H]3CCCO3)c2)c1 ZINC000880563648 DE On-Demand Anodyne PANC 54 36 COc1cncc(NC(=O)Nc2cnn(C[C@@H]3CCCO3)c2)c1 ZINC000880563649 DE On-Demand Anodyne PANC 54 36 COc1cncc(NC(=O)N2CCN(Cc3cscn3)CC2)c1 ZINC000880563652 ED On-Demand Anodyne PDGFRB 40 35 COc1cncc(NC(=O)N2CCN(Cc3cscn3)CC2)c1 ZINC000880563652 ED On-Demand Anodyne FAAH 16 46 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne SSTR5 40 37 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne CCR3 48 48 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne EPHX2 50 41 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne PDK1 41 42 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne CXCR3 21 50 COc1cncc(NC(=O)NC2CCN(CC3CC3)CC2)c1 ZINC000880563655 DE On-Demand Anodyne MCHR1 17 48 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccc2Cl)c1 ZINC000880563665 EI On-Demand Anodyne CPT1A 51 35 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccc2Cl)c1 ZINC000880563666 EI On-Demand Anodyne CPT1A 51 35 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccc(F)cc2)c1 ZINC000880563667 EF On-Demand Anodyne ROCK1 18 54 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccc(F)cc2)c1 ZINC000880563667 EF On-Demand Anodyne ROCK2 33 54 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nccs2)C1 ZINC000880563674 CB On-Demand Anodyne MAP1 123 47 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(Cl)cn2)C1 ZINC000880563676 EC On-Demand Anodyne F10 51 34 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(Cl)cn2)C1 ZINC000880563679 EC On-Demand Anodyne F10 51 34 COc1cncc(NC(=O)N2CCN(CCc3cccs3)CC2)c1 ZINC000880563687 EF On-Demand Anodyne HTR1A 16 40 COc1cncc(NC(=O)N2CCN(CCc3cccs3)CC2)c1 ZINC000880563687 EF On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)N2CCN(CCc3cccs3)CC2)c1 ZINC000880563687 EF On-Demand Anodyne PDGFRB 46 36 COc1cncc(NC(=O)N2CCN(CCc3cccs3)CC2)c1 ZINC000880563687 EF On-Demand Anodyne FAAH 19 44 COc1cncc(NC(=O)N2CCC(N3CCCCC3)CC2)c1 ZINC000880563692 DF On-Demand Anodyne CHRM2 41 38 COc1cncc(NC(=O)N2CCC(N3CCCCC3)CC2)c1 ZINC000880563692 DF On-Demand Anodyne HRH3 22 44 COc1cncc(NC(=O)N2CCC(N3CCCCC3)CC2)c1 ZINC000880563692 DF On-Demand Anodyne GALR2 44 32 COc1cncc(NC(=O)N2CCC(N3CCCCC3)CC2)c1 ZINC000880563692 DF On-Demand Anodyne L3MBTL3 91 42 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne HTR4 43 39 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne SSTR5 41 37 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne CCR3 34 41 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne EPHX2 51 47 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne PDK1 40 33 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne CXCR3 20 46 COCCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880563693 DD On-Demand Anodyne MCHR1 23 48 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccc(F)cc3)C2)c1 ZINC000880563701 EF On-Demand Anodyne CCR3 90 45 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccc(F)cc3)C2)c1 ZINC000880563702 EF On-Demand Anodyne CCR3 90 45 COc1cncc(NC(=O)N2CCCN(c3ccccc3)CC2)c1 ZINC000880563703 EF On-Demand Anodyne HTR1A 16 52 COc1cncc(NC(=O)N2CCCN(c3ccccc3)CC2)c1 ZINC000880563703 EF On-Demand Anodyne PDGFRB 57 46 COc1cncc(NC(=O)N2CCCN(c3ccccc3)CC2)c1 ZINC000880563703 EF On-Demand Anodyne FAAH 22 48 COc1cncc(NC(=O)N2CCCN(c3ccccc3)CC2)c1 ZINC000880563703 EF On-Demand Anodyne ADAM10 34 41 COc1cncc(NC(=O)NCCCc2ccc(OC)c(OC)c2)c1 ZINC000880563706 EF On-Demand Anodyne INHA 58 36 COc1cncc(NC(=O)NCCCc2ccc(OC)c(OC)c2)c1 ZINC000880563706 EF On-Demand Anodyne MTNR1A 21 50 COc1cncc(NC(=O)NCCCc2ccc(OC)c(OC)c2)c1 ZINC000880563706 EF On-Demand Anodyne MTNR1B 22 50 COc1cncc(NC(=O)NCCCc2ccc(OC)c(OC)c2)c1 ZINC000880563706 EF On-Demand Anodyne QPCT 28 49 COc1cncc(NC(=O)NCCCc2ccc(OC)c(OC)c2)c1 ZINC000880563706 EF On-Demand Anodyne ENPP1 41 32 COc1cncc(NC(=O)N(C)Cc2cccc(C)c2)c1 ZINC000880563711 CG On-Demand Anodyne ROCK1 23 54 COc1cncc(NC(=O)N(C)Cc2cccc(C)c2)c1 ZINC000880563711 CG On-Demand Anodyne ROCK2 37 54 COc1cncc(NC(=O)N(C)Cc2cccc(C)c2)c1 ZINC000880563711 CG On-Demand Anodyne HSD17B2 23 47 COc1cncc(NC(=O)N[C@@H](C)c2ccc(N3CCOCC3)cc2)c1 ZINC000880563714 FF On-Demand Clean MTOR 46 39 COc1cncc(NC(=O)N[C@@H](C)c2ccc(N3CCOCC3)cc2)c1 ZINC000880563714 FF On-Demand Clean EPHB4 31 43 COc1cncc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)c1 ZINC000880563715 FF On-Demand Clean MTOR 46 39 COc1cncc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)c1 ZINC000880563715 FF On-Demand Clean EPHB4 31 43 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1)N1CCOCC1 ZINC000880563716 JF On-Demand Anodyne CNR2 15 53 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1)N1CCOCC1 ZINC000880563717 JF On-Demand Anodyne CNR2 15 53 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880563719 GG On-Demand Anodyne PDGFRB 45 44 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880563719 GG On-Demand Anodyne HRH3 25 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880563719 GG On-Demand Anodyne FAAH 20 42 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880563719 GG On-Demand Anodyne EPHX2 20 41 COc1cncc(NC(=O)N2CCCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880563719 GG On-Demand Anodyne SCN10A 31 41 COc1cncc(NC(=O)NC[C@@H](C)CN2CCCC2)c1 ZINC000880563720 CD On-Demand Anodyne HRH2 15 40 COc1cncc(NC(=O)NC[C@H](C)CN2CCCC2)c1 ZINC000880563721 CD On-Demand Anodyne HRH2 15 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)cc2C(F)(F)F)C1 ZINC000880563743 GD On-Demand Anodyne CACNA1I 41 32 COc1cncc(NC(=O)NCC2(c3ccc(F)cc3)CCOCC2)c1 ZINC000880563744 FG On-Demand Anodyne KCNA3 40 36 COc1cncc(NC(=O)NCC2(c3ccc(F)cc3)CCOCC2)c1 ZINC000880563744 FG On-Demand Anodyne SOAT1 19 41 COc1cncc(NC(=O)NCC2(c3ccc(F)cc3)CCOCC2)c1 ZINC000880563744 FG On-Demand Anodyne ICMT 36 42 COc1cncc(NC(=O)NC[C@H](OC)c2ccccc2)c1 ZINC000880563750 DF On-Demand Anodyne SOAT1 40 39 COc1cncc(NC(=O)NC[C@@H](OC)c2ccccc2)c1 ZINC000880563751 DF On-Demand Anodyne SOAT1 40 39 COc1cncc(NC(=O)N[C@H](C)CN2CCC[C@@H](C)C2)c1 ZINC000880563754 DE On-Demand Anodyne CCR3 77 38 COc1cncc(NC(=O)N[C@@H](C)CN2CCC[C@@H](C)C2)c1 ZINC000880563755 DE On-Demand Anodyne CCR3 77 38 COc1cncc(NC(=O)N[C@H](C)CN2CCC[C@H](C)C2)c1 ZINC000880563756 DE On-Demand Anodyne CCR3 77 38 COc1cncc(NC(=O)N[C@@H](C)CN2CCC[C@H](C)C2)c1 ZINC000880563757 DE On-Demand Anodyne CCR3 77 38 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)C1 ZINC000880563781 GD On-Demand Anodyne ROCK1 19 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)C1 ZINC000880563782 GD On-Demand Anodyne ROCK1 19 41 COc1cncc(NC(=O)N2CCC[C@H](N3CCCC3)C2)c1 ZINC000880563796 DE On-Demand Anodyne HRH3 18 40 COc1cncc(NC(=O)N2CCC[C@H](N3CCCC3)C2)c1 ZINC000880563796 DE On-Demand Anodyne L3MBTL3 54 36 COc1cncc(NC(=O)N2CCC[C@@H](N3CCCC3)C2)c1 ZINC000880563797 DE On-Demand Anodyne HRH3 18 40 COc1cncc(NC(=O)N2CCC[C@@H](N3CCCC3)C2)c1 ZINC000880563797 DE On-Demand Anodyne L3MBTL3 54 36 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne FKBP1A 41 40 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne DRD4 40 30 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne CCR3 18 54 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne CHRNA7 42 51 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne ROCK1 34 42 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne PREP 44 33 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne MTNR1A 22 40 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne MTNR1B 34 40 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne ROCK2 46 40 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne FAAH 18 41 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)c1 ZINC000880563805 EG On-Demand Anodyne ACKR3 54 30 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3O)CC2)c1 ZINC000880563815 FD On-Demand Anodyne PDGFRB 47 41 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3O)CC2)c1 ZINC000880563815 FD On-Demand Anodyne FAAH 15 44 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3ccc(F)cc3)CC2)C1 ZINC000880563816 FC On-Demand Anodyne CCR1 20 43 COc1cncc(NC(=O)NCCC(=O)NC2CCCCC2)c1 ZINC000880563832 DE On-Demand Anodyne EPHX2 24 49 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(C(C)(C)C)cc2)C1 ZINC000880563850 ED On-Demand Anodyne TRPV1 15 40 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne BMP1 19 41 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne CA1 36 44 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne MMP13 18 40 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne CCR3 15 46 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne MMP9 15 40 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne CA12 19 44 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne CA9 20 44 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne MMP1 15 40 COc1cncc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)c1 ZINC000880563855 ED On-Demand Anodyne NAMPT 42 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(C(F)(F)F)cc2)C1 ZINC000880563859 ED On-Demand Anodyne EPHX2 44 41 O=C(NCc1cn(C2CCC2)nn1)c1ccc(S(F)(F)(F)(F)F)cc1 ZINC000880563866 GJ On-Demand Reactive CA14 16 50 COc1cncc(NC(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000880563871 EE On-Demand Anodyne HRH2 19 47 COc1cncc(NC(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000880563871 EE On-Demand Anodyne EDNRB 72 38 COc1cncc(NC(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000880563871 EE On-Demand Anodyne EDNRA 72 40 COc1cncc(NC(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000880563871 EE On-Demand Anodyne BMP1 64 41 COC(=O)[C@@]1(O)CCN(CC(=O)c2cc(C)n(Cc3ccccc3)c2C)C1 ZINC000880563873 FD On-Demand Anodyne SLC12A5 58 36 COc1cncc(NC(=O)N[C@H](C)Cc2ccc(O)cc2)c1 ZINC000880563886 DF On-Demand Anodyne GRIA1 45 32 COc1cncc(NC(=O)N[C@@H](C)Cc2ccc(O)cc2)c1 ZINC000880563887 DF On-Demand Anodyne GRIA1 45 32 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne TSHR 48 33 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne LTA4H 35 55 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne CTSK 18 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne ADAM17 40 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne TIMP3 43 37 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne MMP2 16 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne MMP9 18 48 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne EPHX2 15 53 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne FFAR1 23 41 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563893 GE On-Demand Anodyne SLC12A5 67 38 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne TSHR 48 33 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne LTA4H 35 55 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne CTSK 18 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne ADAM17 40 48 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne TIMP3 43 37 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne MMP2 16 48 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne MMP9 18 48 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne EPHX2 15 53 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne FFAR1 23 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880563894 GE On-Demand Anodyne SLC12A5 67 38 COc1cncc(NC(=O)N2CCC[C@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000880563897 FF On-Demand Anodyne EPHX2 20 40 COc1cncc(NC(=O)N2CCC[C@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000880563897 FF On-Demand Anodyne LUCI_LUCLA 15 41 COc1cncc(NC(=O)N2CCC[C@@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000880563898 FF On-Demand Anodyne EPHX2 20 40 COc1cncc(NC(=O)N2CCC[C@@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000880563898 FF On-Demand Anodyne LUCI_LUCLA 15 41 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccnc2Cl)C1 ZINC000880563903 DC On-Demand Anodyne G2YM83_BOTF4 69 35 COc1cncc(NC(=O)N[C@@H](Cn2ccnc2)C(C)(C)C)c1 ZINC000880563912 DF On-Demand Anodyne QPCT 24 44 COc1cncc(NC(=O)N[C@H](Cn2ccnc2)C(C)(C)C)c1 ZINC000880563913 DF On-Demand Anodyne QPCT 24 44 COc1cncc(NC(=O)NCc2ccc(N3CCC(O)CC3)c(F)c2)c1 ZINC000880563915 FF On-Demand Clean NPY2R 54 35 COc1cncc(NC(=O)NCc2ccc(N3CCC(O)CC3)c(F)c2)c1 ZINC000880563915 FF On-Demand Clean CCR3 52 39 COc1cncc(NC(=O)NCCN(C)Cc2ccccc2)c1 ZINC000880563916 DE On-Demand Anodyne LTA4H 21 41 COc1cncc(NC(=O)NCCN(C)Cc2ccccc2)c1 ZINC000880563916 DE On-Demand Anodyne ROCK2 39 41 COc1cncc(NC(=O)NCCN(C)Cc2ccccc2)c1 ZINC000880563916 DE On-Demand Anodyne LIMK2 17 40 CCc1nc(CN2CCN(C(=O)Nc3cncc(OC)c3)CC2)cs1 ZINC000880563917 FE On-Demand Anodyne PDGFRB 43 35 CCc1nc(CN2CCN(C(=O)Nc3cncc(OC)c3)CC2)cs1 ZINC000880563917 FE On-Demand Anodyne FAAH 15 45 COc1cncc(NC(=O)N[C@@H]2CCN([C@H](C)c3ccccc3)C2)c1 ZINC000880563924 EG On-Demand Anodyne CCR3 20 40 COc1cncc(NC(=O)N[C@@H]2CCN([C@H](C)c3ccccc3)C2)c1 ZINC000880563924 EG On-Demand Anodyne EPHX2 35 40 COc1cncc(NC(=O)N[C@@H]2CCN([C@@H](C)c3ccccc3)C2)c1 ZINC000880563925 EG On-Demand Anodyne CCR3 20 40 COc1cncc(NC(=O)N[C@@H]2CCN([C@@H](C)c3ccccc3)C2)c1 ZINC000880563925 EG On-Demand Anodyne EPHX2 35 40 COc1cncc(NC(=O)N[C@H]2CCN([C@@H](C)c3ccccc3)C2)c1 ZINC000880563926 EG On-Demand Anodyne CCR3 20 40 COc1cncc(NC(=O)N[C@H]2CCN([C@@H](C)c3ccccc3)C2)c1 ZINC000880563926 EG On-Demand Anodyne EPHX2 35 40 COc1cncc(NC(=O)N[C@H]2CCN([C@H](C)c3ccccc3)C2)c1 ZINC000880563927 EG On-Demand Anodyne CCR3 20 40 COc1cncc(NC(=O)N[C@H]2CCN([C@H](C)c3ccccc3)C2)c1 ZINC000880563927 EG On-Demand Anodyne EPHX2 35 40 COCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880563937 DF On-Demand Anodyne ROCK1 19 47 COCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880563937 DF On-Demand Anodyne ROCK2 33 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)=O)cc2)C1 ZINC000880563969 CC On-Demand Anodyne MMP13 20 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)=O)cc2)C1 ZINC000880563969 CC On-Demand Anodyne ADAM17 16 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC(C)=O)cc2)C1 ZINC000880563969 CC On-Demand Anodyne MMP9 16 45 COc1cncc(NC(=O)NCc2cc(OC)c(OC)c(OC)c2)c1 ZINC000880563971 EE On-Demand Anodyne PDGFRB 22 43 COc1cncc(NC(=O)NCc2cc(OC)c(OC)c(OC)c2)c1 ZINC000880563971 EE On-Demand Anodyne ROCK2 21 47 COc1cncc(NC(=O)NCc2cc(OC)c(OC)c(OC)c2)c1 ZINC000880563971 EE On-Demand Anodyne FLT4 15 43 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(c3ccccc3F)CC2)C1 ZINC000880563972 FC On-Demand Anodyne HTR7 23 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3c(s2)CCCC3)C1 ZINC000880563982 EC On-Demand Anodyne SLC27A1 60 55 COc1cncc(NC(=O)N(C)Cc2cc(Cl)ccc2OC)c1 ZINC000880563984 EG On-Demand Anodyne TSPO 37 40 COc1cncc(NC(=O)N(C)Cc2cc(Cl)ccc2OC)c1 ZINC000880563984 EG On-Demand Anodyne CPT1A 43 37 COc1cncc(NC(=O)N(C)Cc2cc(Cl)ccc2OC)c1 ZINC000880563984 EG On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)N(C)Cc2cc(Cl)ccc2OC)c1 ZINC000880563984 EG On-Demand Anodyne CPT1B 41 35 COc1cncc(NC(=O)N(C)Cc2cc(Cl)ccc2OC)c1 ZINC000880563984 EG On-Demand Anodyne SCN10A 18 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(C)cc3s2)C1 ZINC000880563993 ED On-Demand Anodyne CSNK1D 48 51 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(C)cc3s2)C1 ZINC000880563993 ED On-Demand Anodyne ACOX1 40 31 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(C)cc3s2)C1 ZINC000880563993 ED On-Demand Anodyne SLC27A1 34 41 COc1cncc(NC(=O)NCc2ccnc(N3CCN(C)CC3)c2)c1 ZINC000880563998 FD On-Demand Anodyne ROCK2 24 45 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccoc3)CC2)c1 ZINC000880564000 EE On-Demand Anodyne EPHX2 54 49 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cc(OC)c(Cl)cc2OC)C1 ZINC000880564004 GD On-Demand Anodyne HTR4 49 39 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne PDGFRB 32 43 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne GRIN2B 46 43 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne CCR3 22 44 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne CHRNA7 30 40 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne TIMP3 49 34 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne FAAH 23 45 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne EPHX2 27 40 COc1cncc(NC(=O)N2CCC(OCc3ccccc3)CC2)c1 ZINC000880564006 EG On-Demand Anodyne SCD1 23 46 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(F)c(F)c2)C1 ZINC000880564007 DC On-Demand Anodyne MCHR1 21 42 COc1cncc(NC(=O)NC2CCN(CCN(C)C)CC2)c1 ZINC000880564008 DD On-Demand Anodyne CCR3 41 42 COc1cncc(NC(=O)NC2CCN(CCN(C)C)CC2)c1 ZINC000880564008 DD On-Demand Anodyne SLC6A5 21 44 COc1cncc(NC(=O)NC2CCN(CCN(C)C)CC2)c1 ZINC000880564008 DD On-Demand Anodyne EPHX2 51 48 COc1cncc(NC(=O)NC2CCN(CCN(C)C)CC2)c1 ZINC000880564008 DD On-Demand Anodyne CXCR3 20 46 COc1cncc(NC(=O)NC2CCN(CCN(C)C)CC2)c1 ZINC000880564008 DD On-Demand Anodyne MCHR1 21 49 COc1cncc(NC(=O)NC[C@H]2Cc3ccccc32)c1 ZINC000880564009 CF On-Demand Anodyne MTNR1A 27 50 COc1cncc(NC(=O)NC[C@H]2Cc3ccccc32)c1 ZINC000880564009 CF On-Demand Anodyne MTNR1B 31 46 COc1cncc(NC(=O)NC[C@@H]2Cc3ccccc32)c1 ZINC000880564011 CF On-Demand Anodyne MTNR1A 27 50 COc1cncc(NC(=O)NC[C@@H]2Cc3ccccc32)c1 ZINC000880564011 CF On-Demand Anodyne MTNR1B 31 46 COc1cncc(NC(=O)NC2C[C@@H](C(F)(F)F)C[C@H](C(F)(F)F)C2)c1 ZINC000880564012 GI On-Demand Anodyne EPHX2 44 37 COc1cncc(NC(=O)N[C@@H]2C[C@@H](C(F)(F)F)C[C@@H](C(F)(F)F)C2)c1 ZINC000880564014 GI On-Demand Anodyne EPHX2 44 37 COc1cncc(NC(=O)NCc2ccc(N3CCC(CO)CC3)cc2)c1 ZINC000880564015 FF On-Demand Clean CCR3 51 41 COc1cncc(NC(=O)NCc2ccc(N3CCC(CO)CC3)cc2)c1 ZINC000880564015 FF On-Demand Clean NAMPT 40 39 COc1cncc(NC(=O)NC2C[C@H](C(F)(F)F)C[C@@H](C(F)(F)F)C2)c1 ZINC000880564016 GI On-Demand Anodyne EPHX2 44 37 COC(=O)[C@@]1(O)CCN(CCCn2c(O)nc3ccccc32)C1 ZINC000880564019 DC On-Demand Anodyne EBP 22 41 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564020 DF On-Demand Anodyne EDNRB 56 38 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564020 DF On-Demand Anodyne EDNRA 53 38 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564020 DF On-Demand Anodyne KCNQ2 22 44 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564020 DF On-Demand Anodyne F7 17 43 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564022 DF On-Demand Anodyne EDNRB 56 38 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564022 DF On-Demand Anodyne EDNRA 53 38 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564022 DF On-Demand Anodyne KCNQ2 22 44 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)OCO3)c1 ZINC000880564022 DF On-Demand Anodyne F7 17 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccccc2-c2ccccc2)C1 ZINC000880564039 FD On-Demand Anodyne CHRM3 18 47 COc1cncc(NC(=O)NC[C@@H](O)CN2CCCCC2)c1 ZINC000880564051 DD On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NC[C@@H](O)CN2CCCCC2)c1 ZINC000880564051 DD On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)NC[C@H](O)CN2CCCCC2)c1 ZINC000880564053 DD On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NC[C@H](O)CN2CCCCC2)c1 ZINC000880564053 DD On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)NCc2ccc(OC(C)C)nc2)c1 ZINC000880564055 DF On-Demand Anodyne ROCK2 21 42 COc1cncc(NC(=O)NCCCOCCc2ccccc2)c1 ZINC000880564060 EF On-Demand Anodyne HRH2 29 45 COc1cncc(NC(=O)NCCCOCCc2ccccc2)c1 ZINC000880564060 EF On-Demand Anodyne CCR3 27 47 COc1cncc(NC(=O)NCCCOCCc2ccccc2)c1 ZINC000880564060 EF On-Demand Anodyne MTNR1B 30 43 COc1cncc(NC(=O)NCCCOCCc2ccccc2)c1 ZINC000880564060 EF On-Demand Anodyne ROCK2 19 42 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(OC)c1 ZINC000880564067 EG On-Demand Anodyne INHA 50 34 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(OC)c1 ZINC000880564067 EG On-Demand Anodyne ROCK2 22 50 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(OC)c1 ZINC000880564067 EG On-Demand Anodyne MT-ND1 23 42 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(OC)c1 ZINC000880564067 EG On-Demand Anodyne ENPP1 60 32 COc1ccc(OCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564072 DE On-Demand Anodyne HRH2 20 46 COc1ccc(OCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564072 DE On-Demand Anodyne RAF1 20 40 COc1ccc(OCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564072 DE On-Demand Anodyne MTNR1A 52 44 COc1ccc(OCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564072 DE On-Demand Anodyne MTNR1B 42 44 COc1ccc(OCCNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564072 DE On-Demand Anodyne PIK3CG 18 41 COc1cncc(NC(=O)NCCCN2C[C@H](C)O[C@H](C)C2)c1 ZINC000880564073 DD On-Demand Anodyne CCR3 33 46 COc1cncc(NC(=O)NCCCN2C[C@H](C)O[C@H](C)C2)c1 ZINC000880564073 DD On-Demand Anodyne QPCT 15 40 COc1cncc(NC(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)c1 ZINC000880564074 DD On-Demand Anodyne CCR3 33 46 COc1cncc(NC(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)c1 ZINC000880564074 DD On-Demand Anodyne QPCT 15 40 COc1cncc(NC(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)c1 ZINC000880564076 DD On-Demand Anodyne CCR3 33 46 COc1cncc(NC(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)c1 ZINC000880564076 DD On-Demand Anodyne QPCT 15 40 COc1cncc(NC(=O)NCc2ccnc(N3CCCCC3)c2)c1 ZINC000880564077 EF On-Demand Anodyne HRH2 17 41 COc1cncc(NC(=O)NCc2ccnc(N3CCCCC3)c2)c1 ZINC000880564077 EF On-Demand Anodyne ROCK2 25 46 COc1cncc(NC(=O)NCc2ccnc(N3CCCCC3)c2)c1 ZINC000880564077 EF On-Demand Anodyne GALR2 40 32 COc1cncc(NC(=O)NCc2ccnc(N3CCCCC3)c2)c1 ZINC000880564077 EF On-Demand Anodyne NAMPT 49 41 COc1cncc(NC(=O)N2CCN(c3ncnc4sccc34)CC2)c1 ZINC000880564079 FE On-Demand Anodyne PDGFRB 91 52 COc1cncc(NC(=O)N2CCN(c3ncnc4sccc34)CC2)c1 ZINC000880564079 FE On-Demand Anodyne LIMK2 20 49 CCOc1ccccc1NC(=O)CCN1CC[C@@](O)(C(=O)OC)C1 ZINC000880564081 ED On-Demand Anodyne HCN1 56 36 CCOc1ccccc1NC(=O)CCN1CC[C@@](O)(C(=O)OC)C1 ZINC000880564081 ED On-Demand Anodyne HCN4 43 35 CCOc1ccccc1NC(=O)CCN1CC[C@](O)(C(=O)OC)C1 ZINC000880564083 ED On-Demand Anodyne HCN1 56 36 CCOc1ccccc1NC(=O)CCN1CC[C@](O)(C(=O)OC)C1 ZINC000880564083 ED On-Demand Anodyne HCN4 43 35 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880564089 FD On-Demand Anodyne RBP4 19 43 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2cc(Cl)ccc2OC)C1 ZINC000880564093 FD On-Demand Anodyne RBP4 19 43 COc1cncc(NC(=O)N(C)[C@H](C)c2ccccc2F)c1 ZINC000880564098 DG On-Demand Anodyne NPY5R 33 40 COc1cncc(NC(=O)N(C)[C@@H](C)c2ccccc2F)c1 ZINC000880564100 DG On-Demand Anodyne NPY5R 33 40 COc1cncc(NC(=O)NCc2ccc(OCC(F)(F)F)nc2)c1 ZINC000880564102 FF On-Demand Anodyne ROCK2 15 42 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccc(C#N)cc2)c1 ZINC000880564104 FF On-Demand Mild ROCK2 23 49 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880564106 GC On-Demand Anodyne MTOR 54 38 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880564106 GC On-Demand Anodyne EPHX2 18 40 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(N3CCOCC3)cc2)C1 ZINC000880564106 GC On-Demand Anodyne STAT6 52 33 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(Cl)cc2)C1 ZINC000880564116 ED On-Demand Anodyne CCR1 42 38 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(Cl)cc2)C1 ZINC000880564116 ED On-Demand Anodyne EPHX2 16 41 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)c(F)c3)CC2)c1 ZINC000880564119 GE On-Demand Anodyne PDGFRB 44 38 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)c(F)c3)CC2)c1 ZINC000880564119 GE On-Demand Anodyne TAAR1 19 46 CC(C)(C)OC(=O)N1CCC(OCC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880564122 GE On-Demand Anodyne GPR119 42 40 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne TSHR 41 30 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne PDGFRB 38 43 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne MTNR1A 53 37 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne MTNR1B 49 45 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne ROCK2 21 64 COc1cncc(NC(=O)NCc2cc(OC)ccc2OC)c1 ZINC000880564124 DE On-Demand Anodyne FLT4 23 43 COc1ccc([C@@H](O)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564126 DD On-Demand Anodyne MTNR1A 19 40 COc1ccc([C@@H](O)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564126 DD On-Demand Anodyne ROCK2 16 40 COc1ccc([C@@H](O)CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564126 DD On-Demand Anodyne F7 15 41 COc1cncc(NC(=O)NCc2ccnc(OCC(F)(F)F)c2)c1 ZINC000880564132 FF On-Demand Anodyne ROCK2 22 45 COc1cncc(NC(=O)NCc2ccc(N3C[C@H](C)O[C@@H](C)C3)nc2)c1 ZINC000880564134 FE On-Demand Anodyne NAMPT 37 45 COc1cncc(NC(=O)NCc2ccc(N3C[C@H](C)O[C@H](C)C3)nc2)c1 ZINC000880564135 FE On-Demand Anodyne NAMPT 37 45 COc1cncc(NC(=O)NCc2ccc(N3C[C@@H](C)O[C@H](C)C3)nc2)c1 ZINC000880564136 FE On-Demand Anodyne NAMPT 37 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)OC(C)(C)C)cc2)C1 ZINC000880564139 ED On-Demand Anodyne NOD2 41 35 COc1cncc(NC(=O)N(CCc2ccccc2)CCN(C)C)c1 ZINC000880564141 EF On-Demand Anodyne ROCK1 16 49 COc1cncc(NC(=O)N(CCc2ccccc2)CCN(C)C)c1 ZINC000880564141 EF On-Demand Anodyne ROCK2 30 49 COc1cncc(NC(=O)NCCN2CCCCC2)c1 ZINC000880564142 CD On-Demand Anodyne DRD4 49 38 COc1cncc(NC(=O)NCCN2CCCCC2)c1 ZINC000880564142 CD On-Demand Anodyne HRH2 27 48 COc1cncc(NC(=O)NCCN2CCCCC2)c1 ZINC000880564142 CD On-Demand Anodyne CCR3 41 45 COc1cncc(NC(=O)NCCN2CCCCC2)c1 ZINC000880564142 CD On-Demand Anodyne CHRNA7 23 51 COc1cncc(NC(=O)NCCN2CCCCC2)c1 ZINC000880564142 CD On-Demand Anodyne EPHX2 16 40 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne HTR1A 37 43 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne DRD2 37 47 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne HRH2 23 42 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne HTR2A 21 51 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne DRD3 61 47 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne HTR7 40 48 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne CCR3 45 51 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne CHRNA7 16 46 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne ABCB1B 49 36 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne MTNR1A 18 40 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne MTNR1B 19 40 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne ABCB1 24 44 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne MCHR1 15 41 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne QPCT 29 41 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne NOD1 17 44 COc1cncc(NC(=O)NCCCN2CCc3ccccc3C2)c1 ZINC000880564168 EF On-Demand Anodyne NOD2 45 44 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne PDGFRB 40 41 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne MMP13 30 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne MMP3 35 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne FAAH 17 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne MMP9 25 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne TGM2 83 41 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne MMP1 31 46 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne F13A1 103 44 COc1cncc(NC(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880564174 GD On-Demand Anodyne NAMPT 40 36 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccccc3s2)C1 ZINC000880564180 EC On-Demand Anodyne CSNK1D 45 48 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccccc3s2)C1 ZINC000880564180 EC On-Demand Anodyne ACOX1 46 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccccc3s2)C1 ZINC000880564180 EC On-Demand Anodyne SLC27A1 36 54 COc1cncc(NC(=O)NC2CCN(C(=O)C3CC3)CC2)c1 ZINC000880564188 DD On-Demand Anodyne EPHX2 58 57 COc1cncc(NC(=O)NC2CCN(C(=O)C3CC3)CC2)c1 ZINC000880564188 DD On-Demand Anodyne CXCR3 17 41 CCCN(Cc1ccc(C#N)cc1)C(=O)Nc1cncc(OC)c1 ZINC000880564191 DG On-Demand Mild ROCK2 19 41 COc1cncc(NC(=O)NCc2ccc(OCCN(C)C)cc2)c1 ZINC000880564193 EE On-Demand Anodyne ROCK2 35 46 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564195 FD On-Demand Anodyne DRD4 22 48 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564195 FD On-Demand Anodyne PDGFRB 61 43 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564195 FD On-Demand Anodyne FAAH 26 57 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne ADRB1 43 35 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne HRH2 39 51 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne CCR3 18 46 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne MTNR1A 48 44 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne MTNR1B 51 44 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)NCCCOc2ccccc2)c1 ZINC000880564198 DF On-Demand Anodyne QPCT 15 40 COc1cncc(NC(=O)NCCc2ccc(C)o2)c1 ZINC000880564199 CE On-Demand Anodyne MTNR1A 44 37 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne DRD2 23 49 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne DRD4 47 37 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne HRH2 15 40 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne DRD3 38 50 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne HTR7 21 43 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne CCR3 30 44 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne ABCB1B 55 37 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne MTNR1A 24 42 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne MTNR1B 30 42 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne ABCB1 25 41 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne ABCG2 30 41 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne NOD1 17 46 COc1cncc(NC(=O)NCCN2CCc3ccccc3C2)c1 ZINC000880564200 EE On-Demand Anodyne NOD2 47 46 COC(=O)[C@@]1(O)CCN(CCc2nc3ccccc3n2C)C1 ZINC000880564209 DC On-Demand Anodyne GRM2 16 40 COc1cncc(NC(=O)N2CCN(C(C)C)CC2)c1 ZINC000880564211 CD On-Demand Anodyne PDGFRB 43 39 COc1cncc(NC(=O)N[C@H](C)c2ccc3c(c2)OCCO3)c1 ZINC000880564214 EF On-Demand Anodyne F7 17 49 COc1cncc(NC(=O)N[C@@H](C)c2ccc3c(c2)OCCO3)c1 ZINC000880564215 EF On-Demand Anodyne F7 17 49 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3C)CC2)c1 ZINC000880564220 FF On-Demand Anodyne DRD4 18 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3C)CC2)c1 ZINC000880564220 FF On-Demand Anodyne CCR3 19 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccccc3C)CC2)c1 ZINC000880564220 FF On-Demand Anodyne CCR8 71 40 COc1cncc(NC(=O)N(C)[C@H](C)c2ccc(F)cc2)c1 ZINC000880564221 DG On-Demand Anodyne NPY5R 33 45 COc1cncc(NC(=O)N(C)[C@@H](C)c2ccc(F)cc2)c1 ZINC000880564222 DG On-Demand Anodyne NPY5R 33 45 CCCNC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880564224 EF On-Demand Anodyne DRD4 46 35 CCCNC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880564224 EF On-Demand Anodyne ROCK1 28 41 CCCNC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880564224 EF On-Demand Anodyne RAF1 15 42 CCCNC(=O)c1cccc(CNC(=O)Nc2cncc(OC)c2)c1 ZINC000880564224 EF On-Demand Anodyne ROCK2 54 50 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne ADRB1 44 34 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne HRH2 17 42 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne MTNR1A 29 42 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne MTNR1B 32 42 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne PDGFRA 44 36 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne QPCT 19 44 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne ENPP1 40 31 COc1cncc(NC(=O)NCCOc2ccccc2OC)c1 ZINC000880564225 DE On-Demand Anodyne KCNK3 42 38 COc1cncc(NC(=O)NCc2cccc(N3CCCC3=O)c2)c1 ZINC000880564228 EF On-Demand Anodyne ROCK2 42 46 COc1cncc(NC(=O)N[C@@H](C)c2cccc(OC(F)F)c2)c1 ZINC000880564233 EH On-Demand Anodyne KCNQ2 32 40 COc1cncc(NC(=O)N[C@H](C)c2cccc(OC(F)F)c2)c1 ZINC000880564234 EH On-Demand Anodyne KCNQ2 32 40 COc1cncc(NC(=O)NCc2cccnc2OC(C)C)c1 ZINC000880564238 DF On-Demand Anodyne ROCK2 19 43 COc1cncc(NC(=O)NC2CCN(CC(C)C)CC2)c1 ZINC000880564241 DE On-Demand Anodyne EPHX2 50 41 COc1cncc(NC(=O)NC2CCN(CC(C)C)CC2)c1 ZINC000880564241 DE On-Demand Anodyne PDK1 41 42 COc1cncc(NC(=O)NC2CCN(CC(C)C)CC2)c1 ZINC000880564241 DE On-Demand Anodyne CXCR3 21 46 COc1cncc(NC(=O)NC2CCN(CC(C)C)CC2)c1 ZINC000880564241 DE On-Demand Anodyne MCHR1 17 48 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCO3)c1 ZINC000880564242 DE On-Demand Anodyne BMP1 49 37 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCO3)c1 ZINC000880564242 DE On-Demand Anodyne NOS2 69 33 COc1cncc(NC(=O)NCc2ccc3c(c2)OCCO3)c1 ZINC000880564242 DE On-Demand Anodyne ROCK2 29 45 COC(=O)[C@@]1(O)CCN(Cc2nc3cc(Cl)ccc3n2C)C1 ZINC000880564244 DD On-Demand Anodyne GRM2 18 42 CN1C[C@H](C(=O)NCc2cn(C3CCC3)nn2)c2ccccc2C1=O ZINC000880564250 ED On-Demand Anodyne P2RX7 42 36 CN1C[C@@H](C(=O)NCc2cn(C3CCC3)nn2)c2ccccc2C1=O ZINC000880564251 ED On-Demand Anodyne P2RX7 42 36 COc1cncc(NC(=O)N(C)CC(=O)Nc2c(C)cccc2C)c1 ZINC000880564254 EF On-Demand Anodyne ROCK2 20 40 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(OC(F)F)c2)c1 ZINC000880564256 FG On-Demand Anodyne ROCK2 15 43 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(OC(F)F)c2)c1 ZINC000880564256 FG On-Demand Anodyne MT-ND1 17 40 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne DRD2 28 40 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne DRD4 40 30 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne DRD3 51 40 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne NPY1R 19 42 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne CCR3 60 54 COc1cncc(NC(=O)NCCCCN2CCC(C)CC2)c1 ZINC000880564257 DF On-Demand Anodyne CHRNA7 17 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3nccn3C)cc2)C1 ZINC000880564270 ED On-Demand Anodyne MMP13 17 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3nccn3C)cc2)C1 ZINC000880564270 ED On-Demand Anodyne ADAM17 21 40 COc1cncc(NC(=O)NCc2c[nH]nc2C)c1 ZINC000880564275 CD On-Demand Anodyne ROCK2 20 47 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2nc3ccccc3s2)C1 ZINC000880564277 ED On-Demand Anodyne CSNK1D 27 40 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2nc3ccccc3s2)C1 ZINC000880564279 ED On-Demand Anodyne CSNK1D 27 40 COC(=O)[C@@]1(O)CCN([C@H](c2ccccc2)c2nc(-c3ccccc3)no2)C1 ZINC000880564280 GE On-Demand Anodyne NPY2R 17 45 COC(=O)[C@@]1(O)CCN([C@@H](c2ccccc2)c2nc(-c3ccccc3)no2)C1 ZINC000880564281 GE On-Demand Anodyne NPY2R 17 45 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne DRD4 34 52 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne LTA4H 19 42 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne SIGMAR1 19 49 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne CCR3 50 47 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne CHRNA7 23 43 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne NPY5R 17 50 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne CCKBR 47 38 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne EPHX2 55 48 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne PDK1 47 36 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne CXCR3 22 48 COc1cncc(NC(=O)NC2CCN(CC(=O)Nc3ccccc3)CC2)c1 ZINC000880564286 GE On-Demand Anodyne MCHR1 35 46 COc1cncc(NC(=O)NCCCn2cccn2)c1 ZINC000880564290 CD On-Demand Anodyne HRH2 15 40 COc1cncc(NC(=O)NCCCn2cccn2)c1 ZINC000880564290 CD On-Demand Anodyne CCR3 17 42 COc1cncc(NC(=O)NCCCn2cccn2)c1 ZINC000880564290 CD On-Demand Anodyne QPCT 31 47 COc1cncc(NC(=O)N[C@@H]2CCC[C@@H](C(F)(F)F)C2)c1 ZINC000880564291 DG On-Demand Anodyne EPHX2 47 41 COc1cncc(NC(=O)N[C@H]2CCC[C@H](C(F)(F)F)C2)c1 ZINC000880564292 DG On-Demand Anodyne EPHX2 47 41 COc1cncc(NC(=O)N[C@@H]2CCC[C@H](C(F)(F)F)C2)c1 ZINC000880564293 DG On-Demand Anodyne EPHX2 47 41 COc1cncc(NC(=O)N[C@H]2CCC[C@@H](C(F)(F)F)C2)c1 ZINC000880564294 DG On-Demand Anodyne EPHX2 47 41 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne PDGFRB 41 41 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne PTPN2 48 38 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne MMP3 15 40 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne FAAH 23 48 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne PTPN1 41 40 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne MMP1 16 40 COc1cncc(NC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)c1 ZINC000880564297 GD On-Demand Anodyne F13A1 62 37 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3cccc(C)c3C)CC2)c1 ZINC000880564298 GE On-Demand Anodyne FAAH 17 42 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3cccc(C)c3C)CC2)c1 ZINC000880564298 GE On-Demand Anodyne P2RY14 42 34 COc1cncc(NC(=O)NCCN2CCC(C)CC2)c1 ZINC000880564299 CD On-Demand Anodyne DRD4 46 35 COc1cncc(NC(=O)NCCN2CCC(C)CC2)c1 ZINC000880564299 CD On-Demand Anodyne CCR3 55 48 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)nc2)c1 ZINC000880564304 FD On-Demand Anodyne ROCK2 15 40 COc1cncc(NC(=O)NCc2ccc(N3CCN(C)CC3)nc2)c1 ZINC000880564304 FD On-Demand Anodyne NAMPT 45 39 COC(=O)[C@@]1(O)CCN(CCP(=O)(c2ccccc2)c2ccccc2)C1 ZINC000880564308 FD On-Demand Reactive SLC12A5 42 36 COc1cncc(NC(=O)N[C@H](C)c2ccc(NC(=O)C3CC3)cc2)c1 ZINC000880564315 FG On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)N[C@H](C)c2ccc(NC(=O)C3CC3)cc2)c1 ZINC000880564315 FG On-Demand Anodyne F7 23 48 COc1cncc(NC(=O)N[C@@H](C)c2ccc(NC(=O)C3CC3)cc2)c1 ZINC000880564316 FG On-Demand Anodyne ROCK2 19 41 COc1cncc(NC(=O)N[C@@H](C)c2ccc(NC(=O)C3CC3)cc2)c1 ZINC000880564316 FG On-Demand Anodyne F7 23 48 COc1cncc(NC(=O)NC[C@@H]2CCN(c3ccccc3)C2)c1 ZINC000880564323 EF On-Demand Anodyne CCR3 55 44 COc1cncc(NC(=O)NC[C@H]2CCN(c3ccccc3)C2)c1 ZINC000880564324 EF On-Demand Anodyne CCR3 55 44 COCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564326 EE On-Demand Anodyne PDGFRB 19 46 COCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564326 EE On-Demand Anodyne ROCK2 30 45 COCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564326 EE On-Demand Anodyne CA9 18 40 COCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cc1 ZINC000880564326 EE On-Demand Anodyne NAMPT 35 41 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne GRIN2B 27 43 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne MMP13 23 41 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne CCR3 19 43 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne FAAH 17 44 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne EPHX2 45 47 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne CACNA1G 46 39 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne SCD1 27 40 COc1cncc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000880564330 FF On-Demand Anodyne NAMPT 43 34 COc1cncc(NC(=O)NCc2cccnc2N(C)C)c1 ZINC000880564341 DD On-Demand Anodyne ROCK2 21 42 COc1cncc(NC(=O)N2CCN(c3cnccn3)CC2)c1 ZINC000880564342 DD On-Demand Anodyne PDGFRB 54 43 COc1cncc(NC(=O)N2CCN(c3cnccn3)CC2)c1 ZINC000880564342 DD On-Demand Anodyne FAAH 15 43 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564344 GE On-Demand Anodyne F2 28 40 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564344 GE On-Demand Anodyne GRIN2B 21 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564344 GE On-Demand Anodyne PREP 48 54 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564344 GE On-Demand Anodyne TMPRSS11D 62 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564345 GE On-Demand Anodyne F2 28 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564345 GE On-Demand Anodyne GRIN2B 21 46 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564345 GE On-Demand Anodyne PREP 48 54 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880564345 GE On-Demand Anodyne TMPRSS11D 62 40 COc1cncc(NC(=O)NC[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880564350 EE On-Demand Anodyne CCR3 53 42 COc1cncc(NC(=O)NC[C@@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880564350 EE On-Demand Anodyne CACNA1I 67 37 COc1cncc(NC(=O)NC[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880564351 EE On-Demand Anodyne CCR3 53 42 COc1cncc(NC(=O)NC[C@H]2CCN(CC(F)(F)F)C2)c1 ZINC000880564351 EE On-Demand Anodyne CACNA1I 67 37 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880564354 FF On-Demand Anodyne PDGFRB 28 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880564354 FF On-Demand Anodyne HRH3 24 40 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(F)c3)CC2)c1 ZINC000880564354 FF On-Demand Anodyne CCR3 17 41 COc1cncc(NC(=O)NCc2ccccc2CN(C)C(C)C)c1 ZINC000880564356 EG On-Demand Anodyne ROCK2 21 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(OC(F)(F)Cl)cc1 ZINC000880564363 FG On-Demand Anodyne CA14 16 47 COc1cncc(NC(=O)NCc2ccc(N3CCCCC3)nc2)c1 ZINC000880564373 EF On-Demand Anodyne HRH2 18 41 COc1cncc(NC(=O)NCc2ccc(N3CCCCC3)nc2)c1 ZINC000880564373 EF On-Demand Anodyne ROCK2 16 40 COc1cncc(NC(=O)NCc2ccc(N3CCCCC3)nc2)c1 ZINC000880564373 EF On-Demand Anodyne GALR2 41 32 COc1cncc(NC(=O)NCc2ccc(N3CCCCC3)nc2)c1 ZINC000880564373 EF On-Demand Anodyne NAMPT 54 42 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne DRD4 20 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne SIGMAR1 22 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne MMP13 25 50 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne ADAM17 17 50 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne FAAH 21 50 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne MMP9 21 47 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN(Cc3ccc(OC)cc3)CC2)C1 ZINC000880564394 GB On-Demand Anodyne MMP1 15 50 COc1cncc(NC(=O)NCCCCN2CCC[C@H](C)C2)c1 ZINC000880564416 DF On-Demand Anodyne HRH2 25 42 COc1cncc(NC(=O)NCCCCN2CCC[C@H](C)C2)c1 ZINC000880564416 DF On-Demand Anodyne CCR3 65 54 COc1cncc(NC(=O)NCCCCN2CCC[C@H](C)C2)c1 ZINC000880564416 DF On-Demand Anodyne EBP 15 43 COc1cncc(NC(=O)NCCCCN2CCC[C@@H](C)C2)c1 ZINC000880564417 DF On-Demand Anodyne HRH2 25 42 COc1cncc(NC(=O)NCCCCN2CCC[C@@H](C)C2)c1 ZINC000880564417 DF On-Demand Anodyne CCR3 65 54 COc1cncc(NC(=O)NCCCCN2CCC[C@@H](C)C2)c1 ZINC000880564417 DF On-Demand Anodyne EBP 15 43 COc1cncc(NC(=O)NCC(=O)NC(C)C)c1 ZINC000880564418 CC On-Demand Anodyne F7 25 44 COC(=O)[C@@]1(O)CCN(Cc2nc3ccccc3n2C)C1 ZINC000880564422 CC On-Demand Anodyne GRM2 26 48 CN1CCOc2ccc(C(=O)NCc3cn(C4CCC4)nn3)cc21 ZINC000880564423 ED On-Demand Anodyne CA14 16 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(F)cc3s2)C1 ZINC000880564425 FC On-Demand Anodyne CSNK1D 49 43 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(F)cc3s2)C1 ZINC000880564425 FC On-Demand Anodyne PIK3CA 19 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3ccc(F)cc3s2)C1 ZINC000880564425 FC On-Demand Anodyne SLC27A1 43 49 COc1cncc(NC(=O)NCc2ccc(N(C)C)nc2)c1 ZINC000880564429 DD On-Demand Anodyne ROCK2 25 44 COc1cncc(NC(=O)N2CCN(Cc3csc(C)n3)CC2)c1 ZINC000880564435 EE On-Demand Anodyne FAAH 16 47 COc1cncc(NC(=O)NCc2ccc(OC(C)C)c(OC)c2)c1 ZINC000880564439 EG On-Demand Anodyne ROCK2 29 52 COc1cncc(NC(=O)NCc2ccc(OC(C)C)c(OC)c2)c1 ZINC000880564439 EG On-Demand Anodyne FLT4 15 43 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCCCC[C@H]2c2ccc(OC)cc2)C1 ZINC000880564440 GD On-Demand Anodyne CPT1A 99 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCCCC[C@@H]2c2ccc(OC)cc2)C1 ZINC000880564443 GD On-Demand Anodyne CPT1A 99 40 COc1cncc(NC(=O)NC[C@@H](C)N2CCC[C@@H](C)C2)c1 ZINC000880564445 DE On-Demand Anodyne CCR3 44 34 COc1cncc(NC(=O)NC[C@H](C)N2CCC[C@@H](C)C2)c1 ZINC000880564446 DE On-Demand Anodyne CCR3 44 34 COc1cncc(NC(=O)NC[C@@H](C)N2CCC[C@H](C)C2)c1 ZINC000880564447 DE On-Demand Anodyne CCR3 44 34 COc1cncc(NC(=O)NC[C@H](C)N2CCC[C@H](C)C2)c1 ZINC000880564448 DE On-Demand Anodyne CCR3 44 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)C1 ZINC000880564457 GD On-Demand Anodyne SCD1 35 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)C1 ZINC000880564457 GD On-Demand Anodyne SCD 30 40 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)C1 ZINC000880564457 GD On-Demand Anodyne MGEA5 32 42 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)C1 ZINC000880564457 GD On-Demand Anodyne SLC27A1 41 38 COc1cncc(NC(=O)N2CCC[C@H]2c2ccsc2)c1 ZINC000880564459 DH On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccsc2)c1 ZINC000880564460 DH On-Demand Anodyne NPBWR1 81 34 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(C)c3)CC2)c1 ZINC000880564461 FF On-Demand Anodyne KCNK3 58 42 COc1cncc(NC(=O)N2CCCN(C(=O)c3cccc(C)c3)CC2)c1 ZINC000880564461 FF On-Demand Anodyne KCNK9 42 37 COc1cncc(NC(=O)N2CCN(c3nc(C)cs3)CC2)c1 ZINC000880564463 EE On-Demand Anodyne PDGFRB 44 37 COc1cncc(NC(=O)N2CCN(C(=O)C(C)(C)C)CC2)c1 ZINC000880564471 DD On-Demand Anodyne PDGFRB 40 38 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OC)c(Cl)c2)C1 ZINC000880564474 FD On-Demand Anodyne ENPP1 72 35 COc1cncc(NC(=O)NCc2ccc(N3CCCC3=O)cc2)c1 ZINC000880564478 EF On-Demand Anodyne F10 19 40 COc1cncc(NC(=O)NCc2ccc(N3CCCC3=O)cc2)c1 ZINC000880564478 EF On-Demand Anodyne CYP11B2 16 42 COc1cncc(NC(=O)NCCN2CCCCCC2)c1 ZINC000880564479 CE On-Demand Anodyne DRD4 49 38 COc1cncc(NC(=O)NCCN2CCCCCC2)c1 ZINC000880564479 CE On-Demand Anodyne HRH2 27 48 COc1cncc(NC(=O)NCCN2CCCCCC2)c1 ZINC000880564479 CE On-Demand Anodyne CCR3 41 45 COc1cncc(NC(=O)NCCN2CCCCCC2)c1 ZINC000880564479 CE On-Demand Anodyne CHRNA7 23 51 COc1cncc(NC(=O)NCCN2CCCCCC2)c1 ZINC000880564479 CE On-Demand Anodyne EPHX2 16 40 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne TSHR 54 33 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne LTA4H 62 52 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne MMP13 16 43 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne ADAM17 46 43 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne MMP9 18 43 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne EPHX2 15 44 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OCc3ccccc3)cc2)C1 ZINC000880564484 GE On-Demand Anodyne SLC12A5 73 42 COc1cncc(NC(=O)N(C)[C@H](C)c2ccccc2)c1 ZINC000880564488 CG On-Demand Anodyne NPY5R 39 46 COc1cncc(NC(=O)N(C)[C@@H](C)c2ccccc2)c1 ZINC000880564489 CG On-Demand Anodyne NPY5R 39 46 COc1cncc(NC(=O)NCCCOc2ccccc2F)c1 ZINC000880564490 DF On-Demand Anodyne ADRB1 44 34 COc1cncc(NC(=O)NCCCOc2ccccc2F)c1 ZINC000880564490 DF On-Demand Anodyne HRH2 23 43 COc1cncc(NC(=O)NCCCOc2ccccc2F)c1 ZINC000880564490 DF On-Demand Anodyne CCR3 18 40 COc1cncc(NC(=O)NCCCOc2ccccc2F)c1 ZINC000880564490 DF On-Demand Anodyne QPCT 19 42 COc1cncc(NC(=O)NC[C@@H](CO)Cc2ccccc2)c1 ZINC000880564491 DE On-Demand Anodyne ROCK2 22 41 COc1cncc(NC(=O)NC[C@H](CO)Cc2ccccc2)c1 ZINC000880564492 DE On-Demand Anodyne ROCK2 22 41 COc1cncc(NC(=O)NCc2cccc(OCCN(C)C)c2)c1 ZINC000880564495 EE On-Demand Anodyne HRH2 25 45 COc1cncc(NC(=O)NCc2cccc(OCCN(C)C)c2)c1 ZINC000880564495 EE On-Demand Anodyne ROCK1 44 45 COc1cncc(NC(=O)NCc2cccc(OCCN(C)C)c2)c1 ZINC000880564495 EE On-Demand Anodyne ROCK2 65 56 COc1cncc(NC(=O)NCc2cccc(OCCN(C)C)c2)c1 ZINC000880564495 EE On-Demand Anodyne NAMPT 40 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(OC)c2)C1 ZINC000880564503 CD On-Demand Anodyne MCHR2 40 34 COC(=O)[C@@]1(O)CCN(Cc2cccnc2C)C1 ZINC000880564518 CC On-Demand Anodyne ADAM17 15 42 COc1cncc(NC(=O)N(Cc2ccc(C(=O)NC3CC3)cc2)C2CC2)c1 ZINC000880564525 GG On-Demand Anodyne GCGR 31 42 COc1cncc(NC(=O)N(Cc2ccc(C(=O)NC3CC3)cc2)C2CC2)c1 ZINC000880564525 GG On-Demand Anodyne MAPK14 25 43 COc1cncc(NC(=O)N(Cc2ccc(C(=O)NC3CC3)cc2)C2CC2)c1 ZINC000880564525 GG On-Demand Anodyne GIPR 59 44 COC(=O)[C@@]1(O)CCN([C@H]2CCc3ccccc32)C1 ZINC000880564531 CD On-Demand Anodyne OPRL1 20 44 COC(=O)[C@@]1(O)CCN([C@@H]2CCc3ccccc32)C1 ZINC000880564535 CD On-Demand Anodyne OPRL1 20 44 COc1cncc(NC(=O)NCc2cccc(CN(C)C)c2)c1 ZINC000880564540 DE On-Demand Anodyne ROCK1 42 44 COc1cncc(NC(=O)NCc2cccc(CN(C)C)c2)c1 ZINC000880564540 DE On-Demand Anodyne ROCK2 63 53 COc1cncc(NC(=O)NCc2cccc(CN(C)C)c2)c1 ZINC000880564540 DE On-Demand Anodyne NAMPT 40 42 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880564550 FF On-Demand Anodyne PDGFRB 48 46 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880564550 FF On-Demand Anodyne FAAH 22 44 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880564550 FF On-Demand Anodyne SCN10A 28 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(Cl)cc3)CC2)c1 ZINC000880564550 FF On-Demand Anodyne AKR1C3 19 41 COc1cncc(NC(=O)N(C)Cc2ccc(C(F)(F)F)cc2)c1 ZINC000880564551 EH On-Demand Anodyne RAF1 21 40 COc1cncc(NC(=O)N(C)Cc2ccc(C(F)(F)F)cc2)c1 ZINC000880564551 EH On-Demand Anodyne ROCK2 17 44 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(COc3ccccc3)cc2)C1 ZINC000880564555 GD On-Demand Anodyne MMP13 19 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(COc3ccccc3)cc2)C1 ZINC000880564555 GD On-Demand Anodyne ADAM17 50 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(COc3ccccc3)cc2)C1 ZINC000880564555 GD On-Demand Anodyne MMP9 15 43 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccc(COc3ccccc3)cc2)C1 ZINC000880564555 GD On-Demand Anodyne SLC12A5 63 38 COc1cncc(NC(=O)N2CCC(C(=O)c3ccc(O)cc3)CC2)c1 ZINC000880564559 FF On-Demand Anodyne SLC18A3 40 44 COc1cncc(NC(=O)NCc2ccc(OC)c(OC(F)F)c2)c1 ZINC000880564561 FG On-Demand Anodyne ROCK2 27 51 COc1cncc(NC(=O)NCc2ccc(OC)c(OC(F)F)c2)c1 ZINC000880564561 FG On-Demand Anodyne DRTS_TRYCR 44 30 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)C(F)(F)F ZINC000880564571 GE On-Demand Anodyne REN 42 36 CNC(=O)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880564574 DC On-Demand Anodyne DRD4 18 41 CNC(=O)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880564574 DC On-Demand Anodyne EPHX2 47 40 CNC(=O)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880564574 DC On-Demand Anodyne PDK1 40 33 CNC(=O)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880564574 DC On-Demand Anodyne CXCR3 21 46 CNC(=O)CN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880564574 DC On-Demand Anodyne MCHR1 16 48 COC(=O)[C@@]1(O)CCN(Cc2cc3ccccc3n(C)c2=O)C1 ZINC000880564576 DC On-Demand Anodyne NPSR1 32 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(N)c2)C1 ZINC000880564578 CC On-Demand Anodyne MCHR2 44 34 COC(=O)[C@@]1(O)CCN(Cc2cccc(N)c2)C1 ZINC000880564578 CC On-Demand Anodyne SLC12A5 55 36 COC(=O)[C@@]1(O)CCN(Cc2cnc3ccccc3c2)C1 ZINC000880564582 CD On-Demand Anodyne ADAM17 31 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3cccc(C#N)c3)c(OC)c2)C1 ZINC000880564597 GE On-Demand Mild SLC12A5 17 41 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne HTR1A 18 60 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne DRD4 47 38 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne HTR1B 15 60 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne PDGFRB 62 48 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne CCKAR 33 42 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne MTNR1A 19 40 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne MTNR1B 29 40 COc1cncc(NC(=O)N2CCN(c3cccc(OC)c3)CC2)c1 ZINC000880564605 EE On-Demand Anodyne FAAH 29 52 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564610 FE On-Demand Anodyne DRD4 39 50 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564610 FE On-Demand Anodyne HRH2 19 40 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564610 FE On-Demand Anodyne SIGMAR1 23 42 COc1cncc(NC(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564610 FE On-Demand Anodyne CCR3 43 47 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564611 FE On-Demand Anodyne DRD4 39 50 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564611 FE On-Demand Anodyne HRH2 19 40 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564611 FE On-Demand Anodyne SIGMAR1 23 42 COc1cncc(NC(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)c1 ZINC000880564611 FE On-Demand Anodyne CCR3 43 47 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne DRD4 48 37 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne CASR 23 41 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne CCR3 29 43 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne PIK3CA 18 41 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne CHRNA7 16 48 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne MTOR 36 41 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne EPHX2 30 47 COc1cncc(NC(=O)NCCN2CCOCC2)c1 ZINC000880564614 CC On-Demand Anodyne PIK3CG 22 42 COc1cncc(NC(=O)NCc2csc(C)n2)c1 ZINC000880564635 CE On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne HTR1A 18 42 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne DRD4 31 47 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne PDGFRB 65 48 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne EBP 26 42 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne SSTR1 24 43 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne FAAH 27 46 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne DGAT1 30 45 COc1cncc(NC(=O)N2CCN(c3ccccn3)CC2)c1 ZINC000880564641 DD On-Demand Anodyne SLC11A2 26 41 COc1cncc(NC(=O)NC2CCCCC2)c1 ZINC000880564651 BF On-Demand Anodyne EPHX2 51 48 COc1cncc(NC(=O)NC2CCCCC2)c1 ZINC000880564651 BF On-Demand Anodyne PDGFRA 17 49 COc1cncc(NC(=O)N(C)Cc2ccccc2C)c1 ZINC000880564653 CG On-Demand Anodyne ROCK2 20 43 COc1cncc(NC(=O)N2CCN(CC(=O)N3CCc4ccccc43)CC2)c1 ZINC000880564658 GD On-Demand Anodyne DRD4 28 46 COc1cncc(NC(=O)N2CCN(C(C)=O)CC2)c1 ZINC000880564659 CC On-Demand Anodyne PDGFRB 48 40 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OC)cc2)C1 ZINC000880564662 DC On-Demand Anodyne MMP13 15 42 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OC)cc2)C1 ZINC000880564662 DC On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OC)cc2)C1 ZINC000880564662 DC On-Demand Anodyne MMP9 15 42 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2ccc(OC)cc2)C1 ZINC000880564662 DC On-Demand Anodyne CA9 19 40 COc1cncc(NC(=O)N2CCN(C(=O)COc3ccc(F)cc3)CC2)c1 ZINC000880564663 GD On-Demand Anodyne PDGFRB 53 39 COc1cncc(NC(=O)N2CCN(C(=O)COc3ccc(F)cc3)CC2)c1 ZINC000880564663 GD On-Demand Anodyne FAAH 19 42 COc1cncc(NC(=O)N2CCN(C(=O)COc3ccc(F)cc3)CC2)c1 ZINC000880564663 GD On-Demand Anodyne S1PR2 29 43 COC(=O)[C@@]1(O)CCN(CCc2cccnc2)C1 ZINC000880564665 CC On-Demand Anodyne CHRNA7 50 41 COC(=O)[C@@]1(O)CCN(CCc2cccnc2)C1 ZINC000880564665 CC On-Demand Anodyne ACHP_LYMST 28 41 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne DRD4 25 55 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne SIGMAR1 19 52 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne SSTR5 64 41 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne CCR3 43 42 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne CHRNA7 18 42 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne EPHX2 50 48 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne PDK1 48 35 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne CXCR3 26 49 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne MCHR1 38 49 COc1cncc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c1 ZINC000880564672 EE On-Demand Anodyne CCR8 15 41 COC(=O)[C@@]1(O)CCN(C[C@@H]2C[C@H]2c2ccccc2)C1 ZINC000880564686 CD On-Demand Anodyne SLC6A3 19 40 COC(=O)[C@@]1(O)CCN(C[C@@H]2C[C@H]2c2ccccc2)C1 ZINC000880564686 CD On-Demand Anodyne CCR5 37 41 O=C(COCc1cccnc1)NCc1cn(C2CCC2)nn1 ZINC000880564698 DD On-Demand Anodyne CHRNA7 45 37 O=C(COCc1cccnc1)NCc1cn(C2CCC2)nn1 ZINC000880564698 DD On-Demand Anodyne PREP 20 41 O=C(COCc1cccnc1)NCc1cn(C2CCC2)nn1 ZINC000880564698 DD On-Demand Anodyne NAMPT 48 38 COC(=O)[C@@]1(O)CCN(CC[C@H](O)c2ccccc2)C1 ZINC000880564735 CC On-Demand Anodyne OPRK1 16 44 COC(=O)[C@@]1(O)CCN(CC[C@H](O)c2ccccc2)C1 ZINC000880564735 CC On-Demand Anodyne OPRL1 23 42 COC(=O)[C@@]1(O)CCN(CC[C@H](O)c2ccccc2)C1 ZINC000880564735 CC On-Demand Anodyne SLC6A3 19 47 COC(=O)[C@@]1(O)CCN(CC[C@H](O)c2ccccc2)C1 ZINC000880564735 CC On-Demand Anodyne SLC12A5 42 36 COCCOc1ccc(CNC(=O)Nc2cncc(OC)c2)cn1 ZINC000880564737 ED On-Demand Anodyne ROCK2 25 43 COc1cncc(NC(=O)NCCCCN2CCCC[C@@H]2C)c1 ZINC000880564739 DF On-Demand Anodyne HRH2 19 41 COc1cncc(NC(=O)NCCCCN2CCCC[C@@H]2C)c1 ZINC000880564739 DF On-Demand Anodyne CCR3 41 43 COC(=O)[C@@]1(O)CCN(CC[C@@H](O)c2ccccc2)C1 ZINC000880564740 CC On-Demand Anodyne OPRK1 16 44 COC(=O)[C@@]1(O)CCN(CC[C@@H](O)c2ccccc2)C1 ZINC000880564740 CC On-Demand Anodyne OPRL1 23 42 COC(=O)[C@@]1(O)CCN(CC[C@@H](O)c2ccccc2)C1 ZINC000880564740 CC On-Demand Anodyne SLC6A3 19 47 COC(=O)[C@@]1(O)CCN(CC[C@@H](O)c2ccccc2)C1 ZINC000880564740 CC On-Demand Anodyne SLC12A5 42 36 COc1cncc(NC(=O)NCCCCN2CCCC[C@H]2C)c1 ZINC000880564741 DF On-Demand Anodyne HRH2 19 41 COc1cncc(NC(=O)NCCCCN2CCCC[C@H]2C)c1 ZINC000880564741 DF On-Demand Anodyne CCR3 41 43 COC(=O)[C@@]1(O)CCN(Cc2cccnc2OC)C1 ZINC000880564747 CC On-Demand Anodyne CCR8 27 40 COc1cncc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c1 ZINC000880564752 EG On-Demand Anodyne DRD4 40 32 COc1cncc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c1 ZINC000880564752 EG On-Demand Anodyne PDGFRB 36 41 COc1cncc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c1 ZINC000880564752 EG On-Demand Anodyne SLC18A3 48 47 COc1cncc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c1 ZINC000880564752 EG On-Demand Anodyne FAAH 15 43 COc1cncc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c1 ZINC000880564752 EG On-Demand Anodyne SCD1 16 45 COc1cncc(NC(=O)N(C)Cc2ccc(OC(F)F)c(OC)c2)c1 ZINC000880564769 FG On-Demand Anodyne ROCK2 16 43 COc1cncc(NC(=O)N(C)Cc2ccc(OC(F)F)c(OC)c2)c1 ZINC000880564769 FG On-Demand Anodyne MT-ND1 17 40 COCc1ccccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880564770 DF On-Demand Anodyne ROCK2 20 47 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)C1 ZINC000880564779 GC On-Demand Anodyne DRD4 23 42 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)C1 ZINC000880564779 GC On-Demand Anodyne SIGMAR1 18 41 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)C1 ZINC000880564779 GC On-Demand Anodyne KCNA3 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)C1 ZINC000880564779 GC On-Demand Anodyne CCR8 58 38 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)C1 ZINC000880564779 GC On-Demand Anodyne SHH 21 40 COc1cncc(NC(=O)NCc2cccnc2OCC(F)(F)F)c1 ZINC000880564786 FF On-Demand Anodyne TRPV1 16 40 COc1cncc(NC(=O)NCc2cccnc2OCC(F)(F)F)c1 ZINC000880564786 FF On-Demand Anodyne P2RY1 48 44 COc1cncc(NC(=O)NCc2cccnc2OCC(F)(F)F)c1 ZINC000880564786 FF On-Demand Anodyne SCN10A 24 52 COCC(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880564788 DC On-Demand Anodyne PDGFRB 47 37 COc1cncc(NC(=O)NCc2ccnc(N3CCCC3)c2)c1 ZINC000880564796 EE On-Demand Anodyne ROCK2 26 47 COc1cncc(NC(=O)NCc2ccnc(N3CCCC3)c2)c1 ZINC000880564796 EE On-Demand Anodyne NAMPT 45 40 COC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880564798 CC On-Demand Anodyne OPRL1 25 42 COC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880564798 CC On-Demand Anodyne NPY2R 18 43 COC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880564800 CC On-Demand Anodyne OPRL1 25 42 COC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880564800 CC On-Demand Anodyne NPY2R 18 43 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCN(C(=O)c3ccccc3)C2)C1 ZINC000880564809 EC On-Demand Anodyne CCR5 18 40 COCCOc1ncccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880564810 ED On-Demand Anodyne ROCK2 20 44 COCCOc1ncccc1CNC(=O)Nc1cncc(OC)c1 ZINC000880564810 ED On-Demand Anodyne SCN10A 36 43 CCN(Cc1cccs1)C(=O)Nc1cncc(OC)c1 ZINC000880564812 CG On-Demand Anodyne ROCK2 19 47 COC(=O)[C@@]1(O)CCN(C[C@H]2CCN(C(=O)c3ccccc3)C2)C1 ZINC000880564815 EC On-Demand Anodyne CCR5 18 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Cl)C1 ZINC000880564816 CD On-Demand Anodyne DRD4 42 33 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Cl)C1 ZINC000880564816 CD On-Demand Anodyne MMP13 16 42 COC(=O)[C@@]1(O)CCN(CCCCOc2c(OC)cccc2OC)C1 ZINC000880564817 FD On-Demand Anodyne HTR1A 50 37 COC(=O)[C@@]1(O)CCN(CCCCOc2c(OC)cccc2OC)C1 ZINC000880564817 FD On-Demand Anodyne DRD2 41 38 COC(=O)[C@@]1(O)CCN(CCCCOc2c(OC)cccc2OC)C1 ZINC000880564817 FD On-Demand Anodyne DRD3 49 38 COC(=O)[C@@]1(O)CCN(CCCCOc2c(OC)cccc2OC)C1 ZINC000880564817 FD On-Demand Anodyne SIGMAR1 18 46 COC(=O)[C@@]1(O)CCN(CCCCOc2c(OC)cccc2OC)C1 ZINC000880564817 FD On-Demand Anodyne EBP 32 46 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880564818 EE On-Demand Anodyne P2RY12 15 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880564818 EE On-Demand Anodyne PDGFRB 48 46 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880564818 EE On-Demand Anodyne NPY2R 26 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880564818 EE On-Demand Anodyne FAAH 23 48 COc1cncc(NC(=O)N2CCN(C(=O)c3ccccc3)CC2)c1 ZINC000880564818 EE On-Demand Anodyne SMO 32 44 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne PDGFRB 46 41 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne MTNR1A 15 50 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne MTNR1B 22 50 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne FAAH 18 47 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne NPY5R 16 41 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne EPHX2 42 43 COc1cncc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c1 ZINC000880564824 FF On-Demand Anodyne LIMK2 20 43 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cc2ccc3ccccc3c2)C1 ZINC000880564839 ED On-Demand Anodyne TRY2_BOVIN 46 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cc2ccc3ccccc3c2)C1 ZINC000880564841 ED On-Demand Anodyne TRY2_BOVIN 46 33 COc1cncc(NC(=O)N2CCCCCC2)c1 ZINC000880564842 BE On-Demand Anodyne PDGFRB 42 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)c(C)c2)C1 ZINC000880564854 CD On-Demand Anodyne MCHR2 45 35 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne DRD4 41 32 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne HRH2 17 41 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne DRD3 45 40 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne CASR 21 40 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne FGFR1 17 44 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne CCR3 46 50 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne CHRNA7 20 53 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne MAP2K1 18 43 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne EPHX2 33 47 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne PIK3CG 22 40 COc1cncc(NC(=O)NCCCN2CCOCC2)c1 ZINC000880564881 CC On-Demand Anodyne QPCT 28 42 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1C[C@H]1c1ccccc1 ZINC000880564890 CE On-Demand Anodyne EPHX2 18 41 CCCOc1cccc(CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880564923 CD On-Demand Anodyne HRH2 46 50 CCCOc1cccc(CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880564923 CD On-Demand Anodyne MMP13 18 53 CCCOc1cccc(CN2CC[C@@](O)(C(=O)OC)C2)c1 ZINC000880564923 CD On-Demand Anodyne ADAM17 17 53 CCCOc1cccc(CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880564924 CD On-Demand Anodyne HRH2 46 50 CCCOc1cccc(CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880564924 CD On-Demand Anodyne MMP13 18 53 CCCOc1cccc(CN2CC[C@](O)(C(=O)OC)C2)c1 ZINC000880564924 CD On-Demand Anodyne ADAM17 17 53 CCOC(=O)C1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880564927 DD On-Demand Anodyne PTR1 47 34 CCOc1ccc([C@@H]2CCCN2C(=O)Nc2cncc(OC)c2)cc1 ZINC000880564939 EH On-Demand Anodyne CHRNA7 15 43 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne HTR1A 55 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne DRD2 46 44 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne ADRA1A 42 39 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne DRD3 53 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne HTR7 40 38 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne SIGMAR1 29 51 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne EBP 43 51 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne CCR8 26 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2OC)C1 ZINC000880564942 CD On-Demand Anodyne MBTPS1 47 32 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccc2)c1 ZINC000880564950 CG On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N2CCC[C@H]2c2ccccc2)c1 ZINC000880564950 CG On-Demand Anodyne CPT1A 65 35 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccc2)c1 ZINC000880564951 CG On-Demand Anodyne CHRNA7 17 42 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccccc2)c1 ZINC000880564951 CG On-Demand Anodyne CPT1A 65 35 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2nc3c(s2)CCC3)C1 ZINC000880564957 EC On-Demand Anodyne SLC27A1 58 52 COc1cncc(NC(=O)N2CCN(c3cc(C#N)ccn3)CC2)c1 ZINC000880564961 ED On-Demand Mild PDGFRB 54 46 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880564963 EF On-Demand Anodyne EDNRB 65 37 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880564963 EF On-Demand Anodyne EDNRA 64 40 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880564963 EF On-Demand Anodyne BMP1 73 44 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880564963 EF On-Demand Anodyne NOS2 50 32 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(OC)c1 ZINC000880564963 EF On-Demand Anodyne ROCK2 19 47 O=C(Cc1ccc(Cl)c(F)c1)NCc1cn(C2CCC2)nn1 ZINC000880564964 DF On-Demand Anodyne P2RX7 65 41 O=C(Cc1ccc(Cl)c(F)c1)NCc1cn(C2CCC2)nn1 ZINC000880564964 DF On-Demand Anodyne MAP3K8 37 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2OC)C1 ZINC000880564975 FC On-Demand Anodyne HTR1A 40 38 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2OC)C1 ZINC000880564975 FC On-Demand Anodyne DRD2 31 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2OC)C1 ZINC000880564975 FC On-Demand Anodyne ADRA1A 40 37 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2OC)C1 ZINC000880564975 FC On-Demand Anodyne DRD3 42 38 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccccc2OC)C1 ZINC000880564975 FC On-Demand Anodyne HTR7 35 41 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3C2)c1 ZINC000880564976 EF On-Demand Anodyne ABCB1 22 47 COc1cncc(NC(=O)N2CCc3cc(OC)c(OC)cc3C2)c1 ZINC000880564976 EF On-Demand Anodyne ABCG2 32 42 COc1cncc(NC(=O)N2CCN(Cc3cc(C)on3)CC2)c1 ZINC000880564980 ED On-Demand Anodyne PDGFRB 44 35 COc1cncc(NC(=O)N2CCN(Cc3cc(C)on3)CC2)c1 ZINC000880564980 ED On-Demand Anodyne FAAH 21 49 COc1cncc(NC(=O)NC2CCC(C(F)(F)F)CC2)c1 ZINC000880564984 DG On-Demand Anodyne EPHX2 55 42 CC(C)(C)OC(=O)N1CCC[C@H](CC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880564987 GG On-Demand Anodyne GPR119 42 38 CC(C)(C)OC(=O)N1CCC[C@@H](CC(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880564988 GG On-Demand Anodyne GPR119 42 38 CCN1CC[C@H](CNC(=O)Nc2cncc(OC)c2)C1 ZINC000880564989 CD On-Demand Anodyne CCR3 52 43 CCN1CC[C@H](CNC(=O)Nc2cncc(OC)c2)C1 ZINC000880564989 CD On-Demand Anodyne CACNA1I 56 35 COc1cncc(NC(=O)N(C)Cc2ccccc2C(F)(F)F)c1 ZINC000880564993 EH On-Demand Anodyne ROCK2 21 43 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880564996 EC On-Demand Anodyne MMP13 27 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880564996 EC On-Demand Anodyne ADAM17 30 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880564996 EC On-Demand Anodyne MMP9 19 42 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccco3)CC2)c1 ZINC000880564997 EE On-Demand Anodyne EPHX2 50 47 COc1cncc(NC(=O)NC[C@H](c2ccccc2)N2CCOCC2)c1 ZINC000880565000 FE On-Demand Anodyne CASR 38 43 COc1cncc(NC(=O)NC[C@@H](c2ccccc2)N2CCOCC2)c1 ZINC000880565001 FE On-Demand Anodyne CASR 38 43 CCOC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880565004 DD On-Demand Anodyne EPHX2 55 54 CCOC(=O)N1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880565004 DD On-Demand Anodyne CXCR3 17 42 O=C(NCc1cn(C2CCC2)nn1)[C@@H](F)c1ccc(C(F)(F)F)cc1 ZINC000880565006 FG On-Demand Anodyne TRPV1 41 33 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne DRD2 15 45 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne DRD4 40 31 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne HRH2 55 57 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne CHRM3 15 46 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne SIGMAR1 17 40 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne MMP13 22 40 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne CCR3 45 43 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne CHRNA7 15 40 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne NPFFR2 30 44 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne ROCK1 33 41 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne ROCK2 51 50 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne FAAH 26 42 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne MCHR1 36 45 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne NPFFR1 39 44 COc1cncc(NC(=O)NCc2cccc(CN3CCCC3)c2)c1 ZINC000880565009 EG On-Demand Anodyne NAMPT 48 42 COc1cncc(NC(=O)N2CCN(C(=O)CCC3CCCC3)CC2)c1 ZINC000880565010 FF On-Demand Anodyne PDGFRB 48 40 COc1cncc(NC(=O)NCCCNC(C)=O)c1 ZINC000880565013 CC On-Demand Anodyne MTNR1A 65 44 COc1cncc(NC(=O)NCCCNC(C)=O)c1 ZINC000880565013 CC On-Demand Anodyne MTNR1B 63 44 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne LTA4H 34 46 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne TSPO 41 34 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne ROCK1 15 42 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne MTNR1A 18 40 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne MTNR1B 24 40 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne ROCK2 26 42 COc1cncc(NC(=O)N(C)CCCOc2ccccc2)c1 ZINC000880565014 DG On-Demand Anodyne TAAR1 17 41 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c1 ZINC000880565015 DG On-Demand Anodyne FKBP1A 58 42 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c1 ZINC000880565015 DG On-Demand Anodyne TACR1 15 41 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c1 ZINC000880565015 DG On-Demand Anodyne CCR3 36 51 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c1 ZINC000880565015 DG On-Demand Anodyne CHRNA7 38 46 COc1cncc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c1 ZINC000880565015 DG On-Demand Anodyne PREP 74 36 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c1 ZINC000880565016 DG On-Demand Anodyne FKBP1A 58 42 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c1 ZINC000880565016 DG On-Demand Anodyne TACR1 15 41 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c1 ZINC000880565016 DG On-Demand Anodyne CCR3 36 51 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c1 ZINC000880565016 DG On-Demand Anodyne CHRNA7 38 46 COc1cncc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c1 ZINC000880565016 DG On-Demand Anodyne PREP 74 36 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne HRH2 15 42 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne CCR3 35 42 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne ROCK1 32 42 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne MTNR1A 17 46 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne MTNR1B 18 46 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne ROCK2 51 51 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne EPHX2 17 40 COc1cncc(NC(=O)NCc2cccc(NC(=O)C3CCC3)c2)c1 ZINC000880565017 FG On-Demand Anodyne NAMPT 44 38 O=C(NCc1cn(C2CCC2)nn1)[C@H](F)c1ccc(C(F)(F)F)cc1 ZINC000880565018 FG On-Demand Anodyne TRPV1 41 33 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880565025 GD On-Demand Anodyne CPT1A 41 33 COC(=O)[C@@]1(O)CCN(CCC(=O)N2CCc3ccccc3C2)C1 ZINC000880565027 EC On-Demand Anodyne HTR7 18 48 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880565028 GD On-Demand Anodyne CPT1A 41 33 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCc3cn(C4CCC4)nn3)ccc21 ZINC000880565039 GG On-Demand Anodyne PANC 49 33 COc1cncc(NC(=O)N(C)CCOc2ccccc2)c1 ZINC000880565045 DF On-Demand Anodyne LTA4H 27 42 COc1cncc(NC(=O)N(C)CCOc2ccccc2)c1 ZINC000880565045 DF On-Demand Anodyne TSPO 41 33 COc1cncc(NC(=O)N(C)CCOc2ccccc2)c1 ZINC000880565045 DF On-Demand Anodyne ROCK2 27 41 COc1cncc(NC(=O)N2CCN(C3CCCC3)CC2)c1 ZINC000880565046 DE On-Demand Anodyne HRH3 28 44 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne PIK3CA 53 41 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne SCN2A 17 41 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne ROCK2 16 41 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne PIK3CD 15 41 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne MTOR 78 39 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne PIK3CG 43 41 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne SCN10A 34 52 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne PIK3CB 17 40 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne STAT6 41 39 COc1cncc(NC(=O)NCc2cccnc2N2CCOCC2)c1 ZINC000880565056 ED On-Demand Anodyne NAMPT 49 43 COC(=O)[C@@]1(O)CCN([C@@H](C#N)c2ccccc2)C1 ZINC000880565058 CC On-Demand Mild OPRL1 23 41 COC(=O)[C@@]1(O)CCN([C@@H](C#N)c2ccccc2)C1 ZINC000880565058 CC On-Demand Mild PTAFR 36 41 CCOC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880565062 DC On-Demand Anodyne OPRL1 26 43 CCOC(=O)[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880565062 DC On-Demand Anodyne NPY2R 23 41 CCOC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880565063 DC On-Demand Anodyne OPRL1 26 43 CCOC(=O)[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880565063 DC On-Demand Anodyne NPY2R 23 41 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne PDGFRB 35 41 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne EPHX2 33 44 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne MCHR1 26 49 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne ADAM10 23 41 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne SCD1 15 42 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne SMO 20 46 COc1cncc(NC(=O)N2CCC(c3ccccc3)CC2)c1 ZINC000880565068 DH On-Demand Anodyne MGEA5 25 42 COC(=O)[C@@]1(O)CCN([C@H](C#N)c2ccccc2)C1 ZINC000880565069 CC On-Demand Mild OPRL1 23 41 COC(=O)[C@@]1(O)CCN([C@H](C#N)c2ccccc2)C1 ZINC000880565069 CC On-Demand Mild PTAFR 36 41 COC(=O)[C@@]1(O)CCN(CCCCCn2c(C)nc3ccccc32)C1 ZINC000880565075 EE On-Demand Anodyne PDE6D 22 42 COc1cncc(NC(=O)NC[C@H](O)CN2CCc3ccccc3C2)c1 ZINC000880565076 FD On-Demand Anodyne NOD1 16 43 COc1cncc(NC(=O)NC[C@H](O)CN2CCc3ccccc3C2)c1 ZINC000880565076 FD On-Demand Anodyne NOD2 45 43 COC(=O)[C@@]1(O)CCN(CCN(Cc2ccccc2)S(C)(=O)=O)C1 ZINC000880565082 FC On-Demand Anodyne SLC12A5 60 37 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880565084 DH On-Demand Anodyne TRPM8 22 56 COc1cncc(NC(=O)NCCCn2nc(C)cc2C)c1 ZINC000880565086 DE On-Demand Anodyne QPCT 64 44 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cncc(OC)c1 ZINC000880565087 DH On-Demand Anodyne TRPM8 22 56 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccccc2)C1 ZINC000880565088 CC On-Demand Anodyne CYP2J2 47 33 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccccc2)C1 ZINC000880565088 CC On-Demand Anodyne SLC12A5 58 37 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne PIK3CA 40 39 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne ROCK2 19 45 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne MTOR 70 39 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne PIK3CB 16 40 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne EPHB4 47 41 COc1cncc(NC(=O)NCc2ccnc(N3CCOCC3)c2)c1 ZINC000880565091 ED On-Demand Anodyne NAMPT 45 44 COc1cncc(NC(=O)NCCCn2c(C)nc3ccccc32)c1 ZINC000880565104 EF On-Demand Anodyne CCR3 20 42 COc1cncc(NC(=O)NCCCn2c(C)nc3ccccc32)c1 ZINC000880565104 EF On-Demand Anodyne QPCT 46 42 COC(=O)[C@@]1(O)CCN(Cc2cnc(-c3ccccc3)nc2)C1 ZINC000880565117 DD On-Demand Anodyne SIGMAR1 28 40 COc1cncc(NC(=O)N2CCC(C(=O)NCC(C)C)CC2)c1 ZINC000880565134 EE On-Demand Anodyne MTNR1A 15 43 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCN(C)CC3)cc2)c1 ZINC000880565136 GD On-Demand Anodyne ROCK2 20 40 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCN(C)CC3)cc2)c1 ZINC000880565136 GD On-Demand Anodyne EPHX2 16 48 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCN(C)CC3)cc2)c1 ZINC000880565136 GD On-Demand Anodyne FLT3 15 42 COc1cncc(NC(=O)NCc2ccc(C(=O)N3CCN(C)CC3)cc2)c1 ZINC000880565136 GD On-Demand Anodyne NAMPT 46 48 COc1cncc(NC(=O)NCCCOCC2CC2)c1 ZINC000880565148 CE On-Demand Anodyne HRH2 17 41 COc1cncc(NC(=O)NCCCOCC2CC2)c1 ZINC000880565148 CE On-Demand Anodyne CCR3 33 43 COc1cncc(NC(=O)N2CCC(C(=O)N3CCN(C)CC3)CC2)c1 ZINC000880565155 FD On-Demand Anodyne PDGFRB 45 37 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccc(Br)cc2)C1 ZINC000880565158 FE On-Demand Anodyne DRD2 28 43 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccc(Br)cc2)C1 ZINC000880565158 FE On-Demand Anodyne ERG2 20 43 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccc(Br)cc2)C1 ZINC000880565158 FE On-Demand Anodyne CYP2J2 50 35 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HTR1A 25 40 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HRH2 40 52 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HTR2A 20 52 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HTR2C 18 41 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne DRD3 49 39 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HTR4 17 46 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HRH3 26 42 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne NPY1R 16 47 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne CCR3 53 52 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne CHRNA7 30 56 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne EBP 16 42 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne HNMT 46 32 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne MCHR1 16 49 COc1cncc(NC(=O)NCCCN2CCCCCC2)c1 ZINC000880565171 DE On-Demand Anodyne QPCT 30 43 COC(=O)[C@@]1(O)CCN(C[C@H](OC)c2ccccc2)C1 ZINC000880565175 CC On-Demand Anodyne ADRA1A 15 40 COC(=O)[C@@]1(O)CCN(C[C@@H](OC)c2ccccc2)C1 ZINC000880565178 CC On-Demand Anodyne ADRA1A 15 40 COc1cncc(NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000880565180 DD On-Demand Anodyne PDGFRB 62 46 COc1cncc(NC(=O)N2CCN(c3ncccn3)CC2)c1 ZINC000880565180 DD On-Demand Anodyne FAAH 20 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)Cc2ccccc2)C1 ZINC000880565182 EC On-Demand Anodyne SIGMAR1 21 41 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)Cc2ccccc2)C1 ZINC000880565182 EC On-Demand Anodyne MMP13 18 41 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)Cc2ccccc2)C1 ZINC000880565182 EC On-Demand Anodyne MMP9 17 41 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)Cc2ccccc2)C1 ZINC000880565182 EC On-Demand Anodyne SLC12A5 71 39 COc1cncc(NC(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)c1 ZINC000880565198 GE On-Demand Anodyne PDGFRB 44 37 COc1cncc(NC(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)c1 ZINC000880565198 GE On-Demand Anodyne BMP1 30 40 COc1cncc(NC(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)c1 ZINC000880565198 GE On-Demand Anodyne FAAH 27 52 COc1cncc(NC(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)c1 ZINC000880565198 GE On-Demand Anodyne MCHR1 33 50 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)c(F)c2)C1 ZINC000880565201 DD On-Demand Anodyne HRH3 20 40 COC(=O)[C@@]1(O)CCN(CCOc2ccc(Cl)c(F)c2)C1 ZINC000880565201 DD On-Demand Anodyne MMP13 16 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCCCC3)cc2)C1 ZINC000880565202 ED On-Demand Anodyne HRH3 34 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCCCC3)cc2)C1 ZINC000880565202 ED On-Demand Anodyne MMP13 18 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCCCC3)cc2)C1 ZINC000880565202 ED On-Demand Anodyne MMP9 15 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCCCC3)cc2)C1 ZINC000880565202 ED On-Demand Anodyne MCHR2 44 34 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCCCC3)cc2)C1 ZINC000880565202 ED On-Demand Anodyne NPFFR1 41 38 COC(=O)[C@@]1(O)CCN(C[C@@H](Cc2ccccc2)OC)C1 ZINC000880565208 CC On-Demand Anodyne OPRL1 15 42 COC(=O)[C@@]1(O)CCN(C[C@@H](Cc2ccccc2)OC)C1 ZINC000880565208 CC On-Demand Anodyne SIGMAR1 20 42 COC(=O)[C@@]1(O)CCN(C[C@@H](Cc2ccccc2)OC)C1 ZINC000880565208 CC On-Demand Anodyne SLC12A5 65 38 COC(=O)[C@@]1(O)CCN(C[C@H](Cc2ccccc2)OC)C1 ZINC000880565209 CC On-Demand Anodyne OPRL1 15 42 COC(=O)[C@@]1(O)CCN(C[C@H](Cc2ccccc2)OC)C1 ZINC000880565209 CC On-Demand Anodyne SIGMAR1 20 42 COC(=O)[C@@]1(O)CCN(C[C@H](Cc2ccccc2)OC)C1 ZINC000880565209 CC On-Demand Anodyne SLC12A5 65 38 CCCCCNC(=O)Nc1cncc(OC)c1 ZINC000880565214 BE On-Demand Anodyne ASAH1 57 32 COc1cncc(NC(=O)NCCCN2CCCC2=O)c1 ZINC000880565219 CD On-Demand Anodyne HRH2 17 41 COc1cncc(NC(=O)NCCCN2CCCC2=O)c1 ZINC000880565219 CD On-Demand Anodyne CCR3 29 43 COc1cncc(NC(=O)NCCCN2CCCC2=O)c1 ZINC000880565219 CD On-Demand Anodyne QPCT 28 41 COc1cncc(NC(=O)NCCCN2CCCC2=O)c1 ZINC000880565219 CD On-Demand Anodyne TYRO3 21 45 CCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880565223 CH On-Demand Anodyne INHA 41 33 CCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880565223 CH On-Demand Anodyne ROCK1 19 48 CCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880565223 CH On-Demand Anodyne ROCK2 32 48 CCCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880565223 CH On-Demand Anodyne PTGES 18 40 COc1cncc(NC(=O)NCCCn2ccnc2)c1 ZINC000880565235 CD On-Demand Anodyne TBXAS1 50 45 COc1cncc(NC(=O)NCCCn2ccnc2)c1 ZINC000880565235 CD On-Demand Anodyne QPCT 90 69 COc1cncc(NC(=O)NCCCn2ccnc2)c1 ZINC000880565235 CD On-Demand Anodyne NAMPT 22 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880565237 DC On-Demand Anodyne MMP13 37 50 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880565237 DC On-Demand Anodyne ADAM17 33 50 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880565237 DC On-Demand Anodyne MMP14 30 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(C)(=O)=O)cc2)C1 ZINC000880565237 DC On-Demand Anodyne MMP9 27 50 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cc2ccccc2)C1 ZINC000880565257 CC On-Demand Anodyne SIGMAR1 18 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cc2ccccc2)C1 ZINC000880565257 CC On-Demand Anodyne ABCB1 52 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cc2ccccc2)C1 ZINC000880565257 CC On-Demand Anodyne SLC12A5 66 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cc2ccccc2)C1 ZINC000880565259 CC On-Demand Anodyne SIGMAR1 18 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cc2ccccc2)C1 ZINC000880565259 CC On-Demand Anodyne ABCB1 52 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cc2ccccc2)C1 ZINC000880565259 CC On-Demand Anodyne SLC12A5 66 38 CCOC(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880565265 DD On-Demand Anodyne P2RY12 45 48 CCOC(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880565265 DD On-Demand Anodyne PDGFRB 46 42 CCOC(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880565265 DD On-Demand Anodyne TGM2 23 40 CCOC(=O)N1CCN(C(=O)Nc2cncc(OC)c2)CC1 ZINC000880565265 DD On-Demand Anodyne F13A1 28 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(-c3cccs3)cc2)C1 ZINC000880565282 DF On-Demand Anodyne HDAC1 17 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(C)(=O)=O)c2)C1 ZINC000880565284 DC On-Demand Anodyne MMP13 19 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(C)(=O)=O)c2)C1 ZINC000880565284 DC On-Demand Anodyne ADAM17 16 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(C)(=O)=O)c2)C1 ZINC000880565284 DC On-Demand Anodyne MMP9 15 46 COC(=O)[C@@]1(O)CCN(Cc2cccc(S(C)(=O)=O)c2)C1 ZINC000880565284 DC On-Demand Anodyne SLC12A5 26 45 COC(=O)[C@@]1(O)CCN(Cc2ccn(CCc3ccccc3)n2)C1 ZINC000880565291 ED On-Demand Anodyne SLC12A5 49 36 COC(=O)[C@@]1(O)CCN(CCCSCc2ccccc2)C1 ZINC000880565327 DD On-Demand Anodyne SLC12A5 70 39 COC(=O)[C@@]1(O)CCN(Cc2ccc(CF)cc2)C1 ZINC000880565335 CD On-Demand Anodyne MMP13 16 42 COCCN(Cc1cccs1)C(=O)Nc1cncc(OC)c1 ZINC000880565336 DF On-Demand Anodyne ROCK2 18 41 COc1cncc(NC(=O)N2CCN(CC(=O)NCc3ccccc3)CC2)c1 ZINC000880565338 GD On-Demand Anodyne HTR1A 16 43 COc1cncc(NC(=O)N2CCN(CC(=O)NCc3ccccc3)CC2)c1 ZINC000880565338 GD On-Demand Anodyne DRD2 15 43 COc1cncc(NC(=O)N2CCN(CC(=O)NCc3ccccc3)CC2)c1 ZINC000880565338 GD On-Demand Anodyne PDGFRB 60 42 COc1cncc(NC(=O)N2CCN(CC(=O)NCc3ccccc3)CC2)c1 ZINC000880565338 GD On-Demand Anodyne HTR7 27 43 COc1cncc(NC(=O)N2CCN(CC(=O)NCc3ccccc3)CC2)c1 ZINC000880565338 GD On-Demand Anodyne FAAH 29 51 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)c(Cl)c2)C1 ZINC000880565341 EE On-Demand Anodyne MMP13 15 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)c(Cl)c2)C1 ZINC000880565341 EE On-Demand Anodyne MCHR2 44 33 COc1cncc(NC(=O)N(C)Cc2ccccc2OC)c1 ZINC000880565344 DF On-Demand Anodyne TSPO 46 40 COc1cncc(NC(=O)N(C)Cc2ccccc2OC)c1 ZINC000880565344 DF On-Demand Anodyne ROCK2 24 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)OC(C)C)cc2)C1 ZINC000880565350 DD On-Demand Anodyne MMP13 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(C(=O)OC(C)C)cc2)C1 ZINC000880565350 DD On-Demand Anodyne NOD2 41 35 COc1cncc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880565362 EE On-Demand Anodyne F13A1 16 40 COc1cncc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880565362 EE On-Demand Anodyne GPR119 35 43 COc1ccc(CN(C(=O)Nc2cncc(OC)c2)C2CC2)cc1 ZINC000880565364 EG On-Demand Anodyne BMP1 41 33 COc1ccc(CN(C(=O)Nc2cncc(OC)c2)C2CC2)cc1 ZINC000880565364 EG On-Demand Anodyne ROCK2 19 52 COc1ccc(CN(C(=O)Nc2cncc(OC)c2)C2CC2)cc1 ZINC000880565364 EG On-Demand Anodyne GIPR 38 41 COc1cncc(NC(=O)N[C@@H](C)Cn2ccnc2)c1 ZINC000880565371 CD On-Demand Anodyne QPCT 28 46 COc1cncc(NC(=O)N[C@H](C)Cn2ccnc2)c1 ZINC000880565372 CD On-Demand Anodyne QPCT 28 46 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne CASR 21 40 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne CCR3 23 43 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne ROCK2 16 41 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne EPHX2 30 42 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne MCHR1 18 41 COc1cncc(NC(=O)NCc2ccccc2CN2CCOCC2)c1 ZINC000880565376 FE On-Demand Anodyne NAMPT 28 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cn2)C1 ZINC000880565378 CC On-Demand Anodyne MMP13 18 43 COc1cncc(NC(=O)N(Cc2ccccn2)C2CC2)c1 ZINC000880565382 CF On-Demand Anodyne ROCK2 20 46 COc1cncc(NC(=O)NCc2ccc(N3CCCC3)nc2)c1 ZINC000880565383 EE On-Demand Anodyne ROCK2 16 41 COc1cncc(NC(=O)NCc2ccc(N3CCCC3)nc2)c1 ZINC000880565383 EE On-Demand Anodyne NAMPT 52 42 CCN(Cc1ccccc1C)C(=O)Nc1cncc(OC)c1 ZINC000880565385 CG On-Demand Anodyne ROCK2 18 45 COC(=O)[C@@]1(O)CCN(Cc2ccc3c(c2)OCCO3)C1 ZINC000880565388 CC On-Demand Anodyne MCHR1 24 43 COC(=O)[C@@]1(O)CCN(Cc2ccc3c(c2)OCCO3)C1 ZINC000880565388 CC On-Demand Anodyne MCHR2 40 32 COC(=O)[C@@]1(O)CCN(Cc2ccccc2CN2CC[C@](O)(C(=O)OC)C2)C1 ZINC000880565395 GB On-Demand Anodyne SIGMAR1 17 43 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(OC)c2)C1 ZINC000880565409 DC On-Demand Anodyne DRD4 44 34 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(OC)c2)C1 ZINC000880565409 DC On-Demand Anodyne MTNR1A 33 47 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(OC)c2)C1 ZINC000880565409 DC On-Demand Anodyne MTNR1B 38 50 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(OC)c2)C1 ZINC000880565409 DC On-Demand Anodyne EPHX2 19 40 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccc(OC)c2)C1 ZINC000880565409 DC On-Demand Anodyne TAAR1 39 41 COc1cncc(NC(=O)N(C)CCOc2ccccc2C)c1 ZINC000880565426 DF On-Demand Anodyne ROCK2 28 41 CCN(Cc1ccc(Cl)s1)C(=O)Nc1cncc(OC)c1 ZINC000880565437 EH On-Demand Anodyne ROCK2 15 42 COc1cncc(NC(=O)NCCc2ccccc2OC)c1 ZINC000880565439 DE On-Demand Anodyne ADRB1 40 31 COc1cncc(NC(=O)NCCc2ccccc2OC)c1 ZINC000880565439 DE On-Demand Anodyne NQO2 50 40 COc1cncc(NC(=O)NCCc2ccccc2OC)c1 ZINC000880565439 DE On-Demand Anodyne MTNR1A 91 44 COc1cncc(NC(=O)NCCc2ccccc2OC)c1 ZINC000880565439 DE On-Demand Anodyne MTNR1B 77 43 COc1cncc(NC(=O)NCCc2ccccc2OC)c1 ZINC000880565439 DE On-Demand Anodyne ROCK2 15 47 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne DRD2 17 47 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne DRD4 40 31 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne ACHE 19 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne CHRM3 19 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne NPFFR2 34 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne CPT1A 44 31 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne PRNP 40 36 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne FAAH 15 48 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne TAAR1 45 35 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne NPFFR1 45 39 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne SLC12A5 47 34 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne NOD1 17 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne NOD2 45 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne KCNK3 106 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(=O)Nc3ccccc3)c2)C1 ZINC000880565446 FE On-Demand Anodyne KCNK9 61 39 C[C@H](NC(=O)OC(C)(C)C)[C@H](C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565449 FE On-Demand Anodyne REN 41 34 C[C@H](NC(=O)OC(C)(C)C)[C@H](C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565449 FE On-Demand Anodyne FPR1 41 35 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880565454 ED On-Demand Anodyne F2 46 38 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880565454 ED On-Demand Anodyne ELANE 40 34 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880565454 ED On-Demand Anodyne TMPRSS11D 60 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880565455 ED On-Demand Anodyne F2 46 38 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880565455 ED On-Demand Anodyne ELANE 40 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880565455 ED On-Demand Anodyne TMPRSS11D 60 34 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Cl)C1 ZINC000880565465 CD On-Demand Anodyne DRD4 42 33 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Cl)C1 ZINC000880565465 CD On-Demand Anodyne SIGMAR1 15 41 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Cl)C1 ZINC000880565465 CD On-Demand Anodyne MMP13 16 44 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Cl)C1 ZINC000880565465 CD On-Demand Anodyne ADAM17 15 44 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Cl)C1 ZINC000880565465 CD On-Demand Anodyne MTNR1B 25 41 COC(=O)[C@@]1(O)CCN(CCC(=O)OCc2ccccc2)C1 ZINC000880565469 DC On-Demand Anodyne SLC12A5 88 49 COC(=O)[C@@]1(O)CCN(Cc2cccc(NC(=O)OC(C)(C)C)c2)C1 ZINC000880565474 FE On-Demand Anodyne HRH2 20 41 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880565490 FF On-Demand Anodyne CCR3 35 40 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880565490 FF On-Demand Anodyne EPHX2 59 48 COc1cncc(NC(=O)NC2CCN(C(=O)c3ccccc3F)CC2)c1 ZINC000880565490 FF On-Demand Anodyne CXCR3 16 40 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565500 FE On-Demand Anodyne PDGFRB 50 39 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565500 FE On-Demand Anodyne NPY2R 19 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565500 FE On-Demand Anodyne S1PR2 28 41 COc1cncc(NC(=O)NCCOc2ccc(C)cc2)c1 ZINC000880565501 DF On-Demand Anodyne ADRB1 15 41 COc1cncc(NC(=O)NCCOc2ccc(C)cc2)c1 ZINC000880565501 DF On-Demand Anodyne HRH2 17 42 COc1cncc(NC(=O)NCCOc2ccc(C)cc2)c1 ZINC000880565501 DF On-Demand Anodyne MTNR1A 27 42 COc1cncc(NC(=O)NCCOc2ccc(C)cc2)c1 ZINC000880565501 DF On-Demand Anodyne MTNR1B 24 42 COc1cncc(NC(=O)N2CCC(CN3CCCCCC3)CC2)c1 ZINC000880565507 EG On-Demand Anodyne HTR4 19 42 COc1cncc(NC(=O)N2CCC(CN3CCCCCC3)CC2)c1 ZINC000880565507 EG On-Demand Anodyne PDGFRB 42 36 COc1cncc(NC(=O)N2CCC(CN3CCCCCC3)CC2)c1 ZINC000880565507 EG On-Demand Anodyne CCR3 26 49 COc1cncc(NC(=O)N2CCC(CO)CC2)c1 ZINC000880565509 CD On-Demand Anodyne PDGFRB 42 36 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne HTR1A 86 51 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne DRD2 68 44 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne DRD1 15 42 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne DRD4 50 44 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne HRH2 22 42 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne ADRA1D 42 42 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne HTR2A 52 49 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne HTR2C 36 44 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne ADRA1A 44 44 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne DRD3 89 44 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne HTR7 65 39 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne NPY1R 18 41 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne CCR3 43 49 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne CHRNA7 21 46 COc1cncc(NC(=O)NCCCN2CCN(c3ncccn3)CC2)c1 ZINC000880565511 FD On-Demand Anodyne QPCT 22 41 COc1cncc(NC(=O)N2CCC[C@@H](c3nc4ccccc4o3)C2)c1 ZINC000880565513 FH On-Demand Anodyne SMO 22 43 COc1cncc(NC(=O)N2CCC[C@H](c3nc4ccccc4o3)C2)c1 ZINC000880565515 FH On-Demand Anodyne SMO 22 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CC[C@](O)(C(=O)OC)C3)c2)C1 ZINC000880565524 GB On-Demand Anodyne CHRM3 17 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CC[C@](O)(C(=O)OC)C3)c2)C1 ZINC000880565524 GB On-Demand Anodyne SIGMAR1 41 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CC[C@](O)(C(=O)OC)C3)c2)C1 ZINC000880565524 GB On-Demand Anodyne MCHR2 60 36 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CC[C@](O)(C(=O)OC)C3)c2)C1 ZINC000880565524 GB On-Demand Anodyne SLC12A5 58 37 COc1cncc(NC(=O)NCc2ccc(N3CCCC3)cc2)c1 ZINC000880565526 EG On-Demand Clean ROCK2 21 43 COc1cncc(NC(=O)NCc2ccc(N3CCCC3)cc2)c1 ZINC000880565526 EG On-Demand Clean FLT3 15 40 COc1cncc(NC(=O)NCc2ccc(N3CCCC3)cc2)c1 ZINC000880565526 EG On-Demand Clean NAMPT 54 45 COc1cncc(NC(=O)NCCCN2CCCCCC2=O)c1 ZINC000880565529 DE On-Demand Anodyne HRH2 24 44 COc1cncc(NC(=O)NCCCN2CCCCCC2=O)c1 ZINC000880565529 DE On-Demand Anodyne CCR3 29 42 COc1cncc(NC(=O)NCCCN2CCCCCC2=O)c1 ZINC000880565529 DE On-Demand Anodyne QPCT 21 40 COc1cncc(NC(=O)NCCCN2CCCCCC2=O)c1 ZINC000880565529 DE On-Demand Anodyne TYRO3 20 44 COc1cncc(NC(=O)NCc2ccnn2C)c1 ZINC000880565533 CD On-Demand Anodyne HTR2A 30 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne DRD4 18 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne MAPK14 40 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne SSTR5 44 42 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne CCR3 32 46 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne MAPK13 59 34 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne MCHR1 25 46 COc1cncc(NC(=O)N2CCC(NC(=O)c3ccc(F)cc3)CC2)c1 ZINC000880565541 FF On-Demand Anodyne HPGDS 33 41 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(F)c2)c1 ZINC000880565542 DF On-Demand Anodyne ROCK2 21 45 COc1cncc(NC(=O)N2CCN(C(=O)c3ccco3)CC2)c1 ZINC000880565544 ED On-Demand Anodyne FAAH 19 43 COc1cncc(NC(=O)N2CCN(C(=O)c3ccco3)CC2)c1 ZINC000880565544 ED On-Demand Anodyne R1A_CVHSA 21 40 COC(=O)[C@@]1(O)CCN(CC(=O)NCc2ccccc2COc2ccccc2)C1 ZINC000880565551 GD On-Demand Anodyne ADAM17 51 37 COc1cncc(NC(=O)N2CCN(c3ccc(O)cc3)CC2)c1 ZINC000880565558 EE On-Demand Anodyne PDGFRB 53 41 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2)c1 ZINC000880565566 DD On-Demand Anodyne ADRB2 52 48 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2)c1 ZINC000880565566 DD On-Demand Anodyne ADRB1 76 52 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2)c1 ZINC000880565566 DD On-Demand Anodyne ADRB3 52 52 COc1cncc(NC(=O)NC[C@@H](O)COc2ccccc2)c1 ZINC000880565566 DD On-Demand Anodyne PDS 51 37 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2)c1 ZINC000880565567 DD On-Demand Anodyne ADRB2 52 48 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2)c1 ZINC000880565567 DD On-Demand Anodyne ADRB1 76 52 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2)c1 ZINC000880565567 DD On-Demand Anodyne ADRB3 52 52 COc1cncc(NC(=O)NC[C@H](O)COc2ccccc2)c1 ZINC000880565567 DD On-Demand Anodyne PDS 51 37 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565569 FF On-Demand Anodyne PRNP 52 37 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565569 FF On-Demand Anodyne TAAR1 47 38 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565569 FF On-Demand Anodyne KCNK3 119 46 COC(=O)[C@@]1(O)CCN([C@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565569 FF On-Demand Anodyne KCNK9 76 40 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565571 FF On-Demand Anodyne PRNP 52 37 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565571 FF On-Demand Anodyne TAAR1 47 38 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565571 FF On-Demand Anodyne KCNK3 119 46 COC(=O)[C@@]1(O)CCN([C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000880565571 FF On-Demand Anodyne KCNK9 76 40 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCCO3)c1 ZINC000880565573 EE On-Demand Anodyne BMP1 51 38 C[C@@H](CNC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565574 ED On-Demand Anodyne REN 54 36 C[C@@H](CNC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565574 ED On-Demand Anodyne FPR1 45 36 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565575 ED On-Demand Anodyne REN 63 37 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880565575 ED On-Demand Anodyne FPR1 45 37 COc1cncc(NC(=O)NCC2(c3ccccc3)CCOCC2)c1 ZINC000880565577 EF On-Demand Anodyne KCNA3 52 45 COc1cncc(NC(=O)NCC2(c3ccccc3)CCOCC2)c1 ZINC000880565577 EF On-Demand Anodyne NMBR 43 34 COc1cncc(NC(=O)NCC2(c3ccccc3)CCOCC2)c1 ZINC000880565577 EF On-Demand Anodyne SOAT1 28 46 COc1cncc(NC(=O)NCC2(c3ccccc3)CCOCC2)c1 ZINC000880565577 EF On-Demand Anodyne ICMT 79 41 COc1cncc(NC(=O)N[C@H](C)CN2CCCCC2)c1 ZINC000880565580 CE On-Demand Anodyne CCR3 48 34 COc1cncc(NC(=O)N[C@@H](C)CN2CCCCC2)c1 ZINC000880565582 CE On-Demand Anodyne CCR3 48 34 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2cccc(CN3CCSCC3)c2)C1 ZINC000880565588 GC On-Demand Anodyne NPFFR1 41 39 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCCO3)c1 ZINC000880565592 EF On-Demand Anodyne BMP1 61 37 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCCO3)c1 ZINC000880565592 EF On-Demand Anodyne ROCK2 18 45 COC(=O)[C@@]1(O)CCN(CCc2cc(Cl)cc(Cl)c2)C1 ZINC000880565611 DE On-Demand Anodyne CACNA1I 45 32 COc1cncc(NC(=O)N2CCc3ccccc3C2)c1 ZINC000880565612 CF On-Demand Anodyne HDAC6 33 41 COc1cncc(NC(=O)N2CCc3ccccc3C2)c1 ZINC000880565612 CF On-Demand Anodyne P2RY14 47 35 COc1cncc(NC(=O)N2CCc3ccccc3C2)c1 ZINC000880565612 CF On-Demand Anodyne NOD1 16 43 COc1cncc(NC(=O)N2CCc3ccccc3C2)c1 ZINC000880565612 CF On-Demand Anodyne NOD2 43 43 COC(=O)[C@@]1(O)CCN(Cc2cccc3c2OC(C)(C)C3)C1 ZINC000880565617 DD On-Demand Anodyne CCR8 21 50 CCOCCCNC(=O)Nc1cncc(OC)c1 ZINC000880565620 CD On-Demand Anodyne HRH2 16 41 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)cc(Br)c2)C1 ZINC000880565621 EE On-Demand Anodyne CACNA1I 41 34 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCCCC2)c1 ZINC000880565625 EE On-Demand Anodyne HCN1 68 42 COc1cncc(NC(=O)NCC2(N3CCOCC3)CCCCC2)c1 ZINC000880565625 EE On-Demand Anodyne HCN4 58 41 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)ccc2OCC2CC2)C1 ZINC000880565629 EE On-Demand Anodyne PTGER1 42 45 COc1cncc(NC(=O)N2CCN(C)CC2)c1 ZINC000880565643 CC On-Demand Anodyne HTR1B 15 50 COc1cncc(NC(=O)N2CCN(C)CC2)c1 ZINC000880565643 CC On-Demand Anodyne PDGFRB 50 39 COc1cncc(NC(=O)NC2CCN(C)CC2)c1 ZINC000880565652 CD On-Demand Anodyne EPHX2 50 41 COc1cncc(NC(=O)NC2CCN(C)CC2)c1 ZINC000880565652 CD On-Demand Anodyne CXCR3 18 43 CCCCNC(=O)Nc1cncc(OC)c1 ZINC000880565653 BE On-Demand Anodyne MTNR1B 26 40 COC(=O)[C@@]1(O)CCN(CCCn2ccnc2)C1 ZINC000880565666 CB On-Demand Anodyne TBXAS1 41 42 COC(=O)[C@@]1(O)CCN(CCCn2ccnc2)C1 ZINC000880565666 CB On-Demand Anodyne QPCT 36 40 COC(=O)[C@@]1(O)CCN([C@@H]2CCCN(Cc3ccccc3)C2=O)C1 ZINC000880565670 EC On-Demand Anodyne SLC12A5 63 36 COC(=O)[C@@]1(O)CCN([C@H]2CCCN(Cc3ccccc3)C2=O)C1 ZINC000880565671 EC On-Demand Anodyne SLC12A5 63 36 COc1cncc(NC(=O)N2CCN(CC(=O)N3CCCC3)CC2)c1 ZINC000880565674 EC On-Demand Anodyne PDGFRB 42 35 COC(=O)[C@@]1(O)CCN(Cc2nc3ccc(OC)cc3s2)C1 ZINC000880565692 DD On-Demand Anodyne CSNK1D 27 44 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCO3)c1 ZINC000880565701 DE On-Demand Anodyne EDNRB 60 37 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCO3)c1 ZINC000880565701 DE On-Demand Anodyne EDNRA 62 41 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCO3)c1 ZINC000880565701 DE On-Demand Anodyne BMP1 73 43 COc1cncc(NC(=O)N(C)Cc2ccc3c(c2)OCO3)c1 ZINC000880565701 DE On-Demand Anodyne ROCK2 18 45 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN([C@@H](C#N)c3cccs3)CC2)C1 ZINC000880565702 GC On-Demand Mild PTAFR 33 42 COC(=O)[C@@]1(O)CCN(CC(=O)N2CCN([C@H](C#N)c3cccs3)CC2)C1 ZINC000880565705 GC On-Demand Mild PTAFR 33 42 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne HTR1A 21 45 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne DRD2 26 44 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne DRD4 15 40 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne ADRA1D 20 41 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne HTR2A 16 46 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne ADRA1A 38 41 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne ADRA1B 28 43 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne OPRM1 21 48 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne DRD3 26 40 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne OPRD1 17 48 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne OPRL1 15 44 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne SLC6A3 18 49 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne SIGMAR1 75 50 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne EBP 31 40 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne FAAH 43 42 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne CES1 43 37 COC(=O)[C@@]1(O)CCN(CCCCc2ccccc2)C1 ZINC000880565707 CD On-Demand Anodyne SLC12A5 75 42 COC(=O)[C@@]1(O)CCN(CCCc2cccc(F)c2)C1 ZINC000880565724 CD On-Demand Anodyne HTR2A 15 41 COC(=O)[C@@]1(O)CCN(CCCc2cccc(F)c2)C1 ZINC000880565724 CD On-Demand Anodyne SIGMAR1 35 46 COC(=O)[C@@]1(O)CCN(CCCc2cccc(F)c2)C1 ZINC000880565724 CD On-Demand Anodyne CACNA1G 15 40 COC(=O)[C@@]1(O)CCN(CCCc2cccc(F)c2)C1 ZINC000880565724 CD On-Demand Anodyne SLC12A5 48 34 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne DRD4 40 30 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne HRH2 19 41 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne DRD3 45 38 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne NPY1R 19 44 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne CCR3 61 56 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne CHRNA7 17 45 COc1cncc(NC(=O)NCCCN2CCC(C)CC2)c1 ZINC000880565738 DE On-Demand Anodyne QPCT 19 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3C)CC2)c1 ZINC000880565745 EF On-Demand Anodyne DRD4 20 41 COc1cncc(NC(=O)N2CCN(Cc3ccccc3C)CC2)c1 ZINC000880565745 EF On-Demand Anodyne PDGFRB 47 38 COc1cncc(NC(=O)N2CCN(Cc3ccccc3C)CC2)c1 ZINC000880565745 EF On-Demand Anodyne CCR3 18 40 COc1cncc(NC(=O)N2CCN(Cc3ccccc3C)CC2)c1 ZINC000880565745 EF On-Demand Anodyne FAAH 31 53 COc1cncc(NC(=O)N2CCN(Cc3ccccc3C)CC2)c1 ZINC000880565745 EF On-Demand Anodyne P2RY14 42 33 O=C(NCc1cn(C2CCC2)nn1)c1ccccc1OC1CC1 ZINC000880565768 DE On-Demand Anodyne HCN1 65 39 O=C(NCc1cn(C2CCC2)nn1)c1ccccc1OC1CC1 ZINC000880565768 DE On-Demand Anodyne HCN4 55 39 COc1cncc(NC(=O)NC[C@H](c2ccc(F)cc2)N2CCOCC2)c1 ZINC000880565769 FE On-Demand Anodyne CCR3 21 47 COc1cncc(NC(=O)NC[C@@H](c2ccc(F)cc2)N2CCOCC2)c1 ZINC000880565770 FE On-Demand Anodyne CCR3 21 47 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne SIGMAR1 15 40 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne MMP13 23 41 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne ADAM17 21 41 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne MTNR1B 27 42 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne MMP9 20 41 COC(=O)[C@@]1(O)CCN(Cc2cc(OC)ccc2Br)C1 ZINC000880565772 ED On-Demand Anodyne MMP1 15 41 COc1cncc(NC(=O)NC2CC(C)(C)NC(C)(C)C2)c1 ZINC000880565814 DF On-Demand Anodyne ENV 20 40 COc1cncc(NC(=O)NC2CC(C)(C)NC(C)(C)C2)c1 ZINC000880565814 DF On-Demand Anodyne EZH2 46 37 COC(=O)[C@@]1(O)CCN(CCC(=O)NCc2ccc(OC)cc2OC)C1 ZINC000880565837 FC On-Demand Anodyne HTR7 18 40 COC(=O)[C@@]1(O)CCN(CCC(=O)NCc2ccc(OC)cc2OC)C1 ZINC000880565837 FC On-Demand Anodyne MTNR1A 45 40 COC(=O)[C@@]1(O)CCN(CCC(=O)NCc2ccc(OC)cc2OC)C1 ZINC000880565837 FC On-Demand Anodyne MTNR1B 36 40 COc1cncc(NC(=O)NCCNC(C)=O)c1 ZINC000880565856 CC On-Demand Anodyne MTNR1A 69 43 COc1cncc(NC(=O)NCCNC(C)=O)c1 ZINC000880565856 CC On-Demand Anodyne MTNR1B 65 43 COc1cncc(NC(=O)N2CCC(C)CC2)c1 ZINC000880565861 BE On-Demand Anodyne TRPC6 26 42 COc1cncc(NC(=O)N2CCC(C)CC2)c1 ZINC000880565861 BE On-Demand Anodyne TRPC3 23 42 CCN(Cc1ccncc1)C(=O)Nc1cncc(OC)c1 ZINC000880565868 CF On-Demand Anodyne ROCK1 15 41 CCN(Cc1ccncc1)C(=O)Nc1cncc(OC)c1 ZINC000880565868 CF On-Demand Anodyne ROCK2 22 50 COC(=O)[C@@]1(O)CCN(C[C@H](OC)c2ccc(Cl)cc2)C1 ZINC000880565873 DD On-Demand Anodyne CCR1 52 37 COC(=O)[C@@]1(O)CCN(C[C@@H](OC)c2ccc(Cl)cc2)C1 ZINC000880565875 DD On-Demand Anodyne CCR1 52 37 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne HTR1A 25 56 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne HTR1B 15 56 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne DRD3 20 42 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne PDGFRB 61 48 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne HTR7 22 43 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne FAAH 28 51 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne RBP4 21 40 COc1cncc(NC(=O)N2CCN(c3ccccc3)CC2)c1 ZINC000880565880 DE On-Demand Anodyne DGAT1 20 40 COC(=O)[C@@]1(O)CCN(Cc2cccc([N+](=O)[O-])c2Br)C1 ZINC000880565909 FD On-Demand Bother COLA 53 31 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880565924 EC On-Demand Anodyne MMP13 31 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880565924 EC On-Demand Anodyne ADAM17 33 44 COC(=O)[C@@]1(O)CCN(CCS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880565924 EC On-Demand Anodyne MMP9 20 44 COc1cncc(NC(=O)N2CCCCCCC2)c1 ZINC000880565957 CF On-Demand Anodyne PDGFRB 42 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2OC)C1 ZINC000880565990 CD On-Demand Anodyne CCR8 22 42 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(OC)c2)c1 ZINC000880565992 EF On-Demand Anodyne ROCK2 24 48 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(OC)c2)c1 ZINC000880565992 EF On-Demand Anodyne MT-ND1 24 47 COc1cncc(NC(=O)N(C)Cc2ccc(OC)c(OC)c2)c1 ZINC000880565992 EF On-Demand Anodyne ENPP1 56 33 COC(=O)[C@@]1(O)CCN(Cc2ccc(Br)c(C)c2)C1 ZINC000880566065 ED On-Demand Anodyne MCHR2 44 34 COC(=O)[C@@]1(O)CCN(CCc2c(C)nc3ccccn3c2=O)C1 ZINC000880566067 EC On-Demand Anodyne ADRA2A 31 50 COC(=O)[C@@]1(O)CCN(CCc2c(C)nc3ccccn3c2=O)C1 ZINC000880566067 EC On-Demand Anodyne ADRA2B 38 50 COC(=O)[C@@]1(O)CCN(CCc2c(C)nc3ccccn3c2=O)C1 ZINC000880566067 EC On-Demand Anodyne ADRA2C 21 50 COC(=O)[C@@]1(O)CCN(C[C@@H](O)Cc2cccc(Cl)c2)C1 ZINC000880566074 DC On-Demand Anodyne CCR1 41 35 COC(=O)[C@@]1(O)CCN(C[C@H](O)Cc2cccc(Cl)c2)C1 ZINC000880566076 DC On-Demand Anodyne CCR1 41 35 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne HTR1A 146 53 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne DRD2 100 52 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne DRD4 68 49 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne ADRA1D 67 46 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne HTR2A 80 52 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne HTR2C 33 42 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne SLC6A4 19 40 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne ADRA1A 89 46 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne HRH1 18 49 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne ADRA1B 63 46 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne DRD3 105 49 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne DRD5 21 45 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne HTR7 152 48 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne SIGMAR1 42 48 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne CCR1 41 42 COC(=O)[C@@]1(O)CCN(CCCN2CCN(c3ccccc3)CC2)C1 ZINC000880566079 EC On-Demand Anodyne SLC12A5 58 35 COC(=O)[C@@]1(O)CCN(Cc2cncc(OCc3ccccc3)c2)C1 ZINC000880566099 ED On-Demand Anodyne MMP13 17 46 COC(=O)[C@@]1(O)CCN(Cc2cncc(OCc3ccccc3)c2)C1 ZINC000880566099 ED On-Demand Anodyne ADAM17 46 46 COC(=O)[C@@]1(O)CCN(Cc2cncc(OCc3ccccc3)c2)C1 ZINC000880566099 ED On-Demand Anodyne FAAH 23 41 COC(=O)[C@@]1(O)CCN(Cc2cncc(OCc3ccccc3)c2)C1 ZINC000880566099 ED On-Demand Anodyne SLC12A5 66 37 COC(=O)[C@@]1(O)CCN(CCN(C)Cc2ccccc2)C1 ZINC000880566101 CC On-Demand Anodyne ACHE 17 41 COC(=O)[C@@]1(O)CCN(CCN(C)Cc2ccccc2)C1 ZINC000880566101 CC On-Demand Anodyne SIGMAR1 41 42 COC(=O)[C@@]1(O)CCN(CCN(C)Cc2ccccc2)C1 ZINC000880566101 CC On-Demand Anodyne SLC12A5 72 40 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne INHA 41 32 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne TSPO 41 32 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne ROCK1 21 45 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne ROCK2 37 55 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne NPY5R 32 41 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne PTGES 25 42 CCN(Cc1ccccc1)C(=O)Nc1cncc(OC)c1 ZINC000880566110 CG On-Demand Anodyne LIMK2 17 41 COC(=O)[C@@]1(O)CCN(C[C@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566116 EC On-Demand Anodyne DRD4 34 44 COC(=O)[C@@]1(O)CCN(C[C@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566116 EC On-Demand Anodyne SIGMAR1 57 40 COC(=O)[C@@]1(O)CCN(C[C@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566116 EC On-Demand Anodyne SLC12A5 62 37 COC(=O)[C@@]1(O)CCN(C[C@@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566118 EC On-Demand Anodyne DRD4 34 44 COC(=O)[C@@]1(O)CCN(C[C@@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566118 EC On-Demand Anodyne SIGMAR1 57 40 COC(=O)[C@@]1(O)CCN(C[C@@H]2CN(Cc3ccccc3)CCCO2)C1 ZINC000880566118 EC On-Demand Anodyne SLC12A5 62 37 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR1A 103 65 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne DRD2 73 45 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne DRD1 23 42 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne DRD4 42 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne ADRA1D 81 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR1D 25 65 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR1B 31 65 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR2A 29 51 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR2C 20 51 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne ADRA1A 75 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne ADRA1B 63 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne DRD3 78 44 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne PDGFRB 75 54 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne HTR7 64 56 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne NPY2R 40 39 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne SSTR1 44 37 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne FAAH 22 47 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne PDGFRA 15 48 COc1cncc(NC(=O)N2CCN(c3ccccc3OC)CC2)c1 ZINC000880566127 EE On-Demand Anodyne RBP4 24 51 COCCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566132 FC On-Demand Anodyne ADRB2 16 49 COCCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566132 FC On-Demand Anodyne ADRB1 38 49 COCCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566132 FC On-Demand Anodyne ACOX1 49 32 COCCc1ccc(OC[C@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566132 FC On-Demand Anodyne ABCB1 62 42 COCCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566133 FC On-Demand Anodyne ADRB2 16 49 COCCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566133 FC On-Demand Anodyne ADRB1 38 49 COCCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566133 FC On-Demand Anodyne ACOX1 49 32 COCCc1ccc(OC[C@@H](O)CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566133 FC On-Demand Anodyne ABCB1 62 42 COCCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566134 FC On-Demand Anodyne ADRB2 16 49 COCCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566134 FC On-Demand Anodyne ADRB1 38 49 COCCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566134 FC On-Demand Anodyne ACOX1 49 32 COCCc1ccc(OC[C@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566134 FC On-Demand Anodyne ABCB1 62 42 COCCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566135 FC On-Demand Anodyne ADRB2 16 49 COCCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566135 FC On-Demand Anodyne ADRB1 38 49 COCCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566135 FC On-Demand Anodyne ACOX1 49 32 COCCc1ccc(OC[C@@H](O)CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566135 FC On-Demand Anodyne ABCB1 62 42 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000880566140 EF On-Demand Anodyne HTR1B 17 59 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000880566140 EF On-Demand Anodyne PDGFRB 54 42 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000880566140 EF On-Demand Anodyne FAAH 17 43 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000880566140 EF On-Demand Anodyne S1PR2 27 41 COc1cncc(NC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 ZINC000880566140 EF On-Demand Anodyne FLT3 15 40 CCCN(CCC)C(=O)Nc1cncc(OC)c1 ZINC000880566147 CF On-Demand Anodyne ROCK2 17 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Br)c2)C1 ZINC000880566156 EE On-Demand Anodyne MMP13 15 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(Br)c2)C1 ZINC000880566156 EE On-Demand Anodyne MCHR2 44 33 COc1cncc(NC(=O)N(C)Cc2ccc(OC(F)F)cc2)c1 ZINC000880566166 EG On-Demand Anodyne ROCK2 15 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(N(C)C)cc2)C1 ZINC000880566176 CC On-Demand Clean MMP13 15 41 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne HTR1A 18 48 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne DRD2 32 44 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne DRD1 15 43 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne DRD4 21 45 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne HTR2A 16 45 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne ADRA1A 27 45 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne ADRA1B 21 45 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne DRD3 26 54 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne ERG2 20 42 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne HTR7 17 48 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne SIGMAR1 22 42 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne EBP 23 42 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne CYP2J2 57 41 COC(=O)[C@@]1(O)CCN(CCCC(=O)c2ccccc2)C1 ZINC000880566185 CD On-Demand Anodyne SLC12A5 45 36 COc1cncc(NC(=O)N2CCC[C@H]2c2nc3ccccc3s2)c1 ZINC000880566198 FI On-Demand Anodyne UL80 28 40 COc1cncc(NC(=O)N2CCC[C@H]2c2nc3ccccc3s2)c1 ZINC000880566198 FI On-Demand Anodyne CPT1A 62 37 COc1cncc(NC(=O)N2CCC[C@@H]2c2nc3ccccc3s2)c1 ZINC000880566199 FI On-Demand Anodyne UL80 28 40 COc1cncc(NC(=O)N2CCC[C@@H]2c2nc3ccccc3s2)c1 ZINC000880566199 FI On-Demand Anodyne CPT1A 62 37 COc1cncc(NC(=O)NC[C@@H](c2ccccc2)N(C)C)c1 ZINC000880566204 DF On-Demand Anodyne KCNA5 19 41 COc1cncc(NC(=O)NC[C@H](c2ccccc2)N(C)C)c1 ZINC000880566205 DF On-Demand Anodyne KCNA5 19 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne ACHE 18 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne HRH2 35 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne CHRM3 18 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne HRH3 25 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne SIGMAR1 46 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne MCHR2 58 36 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne NPFFR1 41 39 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCCCC3)c2)C1 ZINC000880566207 ED On-Demand Anodyne SLC12A5 55 36 COCCCNC(=O)Nc1cncc(OC)c1 ZINC000880566213 BD On-Demand Anodyne HRH2 17 43 COC(=O)[C@@]1(O)CCN(CCc2ccc(Cl)cc2)C1 ZINC000880566229 CD On-Demand Anodyne DRD4 19 43 COC(=O)[C@@]1(O)CCN(CCc2ccc(Cl)cc2)C1 ZINC000880566229 CD On-Demand Anodyne SIGMAR1 21 42 COC(=O)[C@@]1(O)CCN(CCc2ccc(Cl)cc2)C1 ZINC000880566229 CD On-Demand Anodyne MMP13 15 44 COC(=O)[C@@]1(O)CCN(CCc2ccc(Cl)cc2)C1 ZINC000880566229 CD On-Demand Anodyne CCR1 61 39 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCCN2C)C1 ZINC000880566248 BB On-Demand Anodyne CHRNA10 40 35 COC(=O)[C@@]1(O)CCN(C[C@H]2CCCN2C)C1 ZINC000880566251 BB On-Demand Anodyne CHRNA10 40 35 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)=O)c2)C1 ZINC000880566253 CC On-Demand Anodyne CHRM3 18 43 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)=O)c2)C1 ZINC000880566253 CC On-Demand Anodyne MCHR2 45 33 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)=O)c2)C1 ZINC000880566253 CC On-Demand Anodyne SLC12A5 45 33 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne CHRM2 26 45 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne DRD2 20 43 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne DRD4 55 43 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne ACHE 40 42 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne DRD3 17 43 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne SLC6A3 15 40 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne CHRM3 33 45 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne SIGMAR1 76 44 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne SLC18A3 29 44 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne MCHR1 16 41 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566254 DC On-Demand Anodyne SLC12A5 56 36 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne CHRM2 26 45 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne DRD2 20 43 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne DRD4 55 43 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne ACHE 40 42 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne DRD3 17 43 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne SLC6A3 15 40 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne CHRM3 33 45 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne SIGMAR1 76 44 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne SLC18A3 29 44 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne MCHR1 16 41 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccccc3)C2)C1 ZINC000880566255 DC On-Demand Anodyne SLC12A5 56 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(SC)cc2)C1 ZINC000880566260 EC On-Demand Anodyne ACOX1 50 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccc(SC)cc2)C1 ZINC000880566260 EC On-Demand Anodyne ABCB1 49 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(SC)cc2)C1 ZINC000880566262 EC On-Demand Anodyne ACOX1 50 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccc(SC)cc2)C1 ZINC000880566262 EC On-Demand Anodyne ABCB1 49 40 CCCCN(CCO)C(=O)Nc1cncc(OC)c1 ZINC000880566264 CD On-Demand Anodyne ROCK2 15 42 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(OC)cc2)C1 ZINC000880566266 DC On-Demand Anodyne MMP13 21 42 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(OC)cc2)C1 ZINC000880566266 DC On-Demand Anodyne MMP9 17 42 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR1A 42 61 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne DRD4 43 36 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR1D 18 61 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR1B 24 61 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR2A 15 43 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR2C 17 43 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne DRD3 54 39 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne PDGFRB 54 46 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne HTR7 35 47 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne NPY2R 101 38 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne SSTR1 19 42 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne FAAH 26 46 COc1cncc(NC(=O)N2CCN(c3ccccc3F)CC2)c1 ZINC000880566269 EF On-Demand Anodyne RBP4 22 47 COC(=O)[C@@]1(O)CCN(CCSCc2ccccc2)C1 ZINC000880566281 CD On-Demand Anodyne SIGMAR1 18 42 COC(=O)[C@@]1(O)CCN(CCSCc2ccccc2)C1 ZINC000880566281 CD On-Demand Anodyne SLC12A5 72 40 CCCCN(CC)C(=O)Nc1cncc(OC)c1 ZINC000880566307 CF On-Demand Anodyne ROCK2 16 41 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)cc(Cl)c2)C1 ZINC000880566314 DE On-Demand Anodyne CACNA1I 54 37 COc1cncc(NC(=O)NC2CCN(C(C)C)CC2)c1 ZINC000880566320 CE On-Demand Anodyne EPHX2 49 41 COc1cncc(NC(=O)NC2CCN(C(C)C)CC2)c1 ZINC000880566320 CE On-Demand Anodyne CXCR3 17 41 O=C(NCc1cn(C2CCC2)nn1)c1cc(=O)c2ccc(F)cc2o1 ZINC000880566340 EE On-Demand Anodyne KCNH2 15 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)c(OC)c2)C1 ZINC000880566348 CD On-Demand Anodyne SSTR5 40 38 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)c(OC)c2)C1 ZINC000880566348 CD On-Demand Anodyne MCHR2 49 34 COc1cncc(NC(=O)N2CCN(CC(=O)NC(C)C)CC2)c1 ZINC000880566360 EC On-Demand Anodyne PDGFRB 41 35 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne OPRK1 17 41 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne GRIN2B 54 51 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne SIGMAR1 29 42 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne TGM2 30 45 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne F13A1 38 45 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne CCR8 25 41 COC(=O)[C@@]1(O)CCN(CC2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880566362 GD On-Demand Anodyne SLC12A5 76 44 COC(=O)[C@@]1(O)CCN(CCCc2cccc(C)c2)C1 ZINC000880566366 CD On-Demand Anodyne SIGMAR1 28 40 COC(=O)[C@@]1(O)CCN(CCC(C#N)(c2ccccc2)c2ccccc2)C1 ZINC000880566371 FE On-Demand Mild CCR1 24 53 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880566374 EC On-Demand Anodyne MMP13 36 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880566374 EC On-Demand Anodyne ADAM17 31 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880566374 EC On-Demand Anodyne MMP9 31 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)N(C)C)cc2)C1 ZINC000880566374 EC On-Demand Anodyne MMP1 18 47 COc1cncc(NC(=O)NC2CCN(C(C)=O)CC2)c1 ZINC000880566377 CD On-Demand Anodyne EPHX2 62 54 COc1cncc(NC(=O)NC2CCN(C(C)=O)CC2)c1 ZINC000880566377 CD On-Demand Anodyne CXCR3 18 46 CCCN(CCO)C(=O)Nc1cncc(OC)c1 ZINC000880566378 CD On-Demand Anodyne ROCK2 17 43 COC(=O)[C@@]1(O)CCN(CCN(C)Cc2ccc(F)cc2)C1 ZINC000880566387 DC On-Demand Anodyne SIGMAR1 15 43 COc1cncc(NC(=O)N2CCN(c3ncccc3C#N)CC2)c1 ZINC000880566392 ED On-Demand Mild P2RY12 23 52 COc1cncc(NC(=O)N2CCN(c3ncccc3C#N)CC2)c1 ZINC000880566392 ED On-Demand Mild PDGFRB 65 46 COc1cncc(NC(=O)N2CCN(c3ncccc3C#N)CC2)c1 ZINC000880566392 ED On-Demand Mild TRPV1 15 62 COc1cncc(NC(=O)N2CCN(c3ncccc3C#N)CC2)c1 ZINC000880566392 ED On-Demand Mild FAAH 19 42 COc1cncc(NC(=O)N2CCN(c3ncccc3C#N)CC2)c1 ZINC000880566392 ED On-Demand Mild RBP4 15 42 CN(CCC(=O)NCc1cn(C2CCC2)nn1)C(=O)OCc1ccccc1 ZINC000880566415 FE On-Demand Anodyne PREP 36 47 COC(=O)[C@@]1(O)CCN(C[C@H](O)CCc2ccccc2)C1 ZINC000880566420 CC On-Demand Anodyne ABCB1 60 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)CCc2ccccc2)C1 ZINC000880566420 CC On-Demand Anodyne SLC12A5 61 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)CCc2ccccc2)C1 ZINC000880566421 CC On-Demand Anodyne ABCB1 60 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)CCc2ccccc2)C1 ZINC000880566421 CC On-Demand Anodyne SLC12A5 61 37 COC(=O)[C@@]1(O)CCN(CCc2cccc(OC(F)(F)F)c2)C1 ZINC000880566430 ED On-Demand Anodyne EPHX2 32 41 COC(=O)[C@@]1(O)CCN(Cc2cn(Cc3ccccc3)nn2)C1 ZINC000880566432 DC On-Demand Anodyne SIGMAR1 45 40 COC(=O)[C@@]1(O)CCN(Cc2cn(Cc3ccccc3)nn2)C1 ZINC000880566432 DC On-Demand Anodyne NPFFR2 31 40 COC(=O)[C@@]1(O)CCN(Cc2cn(Cc3ccccc3)nn2)C1 ZINC000880566432 DC On-Demand Anodyne NPFFR1 42 40 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3c(C)cccc3C)CC2)c1 ZINC000880566466 GE On-Demand Anodyne PDGFRB 43 36 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3c(C)cccc3C)CC2)c1 ZINC000880566466 GE On-Demand Anodyne ACOX1 45 34 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3c(C)cccc3C)CC2)c1 ZINC000880566466 GE On-Demand Anodyne FAAH 20 44 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3c(C)cccc3C)CC2)c1 ZINC000880566466 GE On-Demand Anodyne P2RY14 42 33 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Br)C1 ZINC000880566472 ED On-Demand Anodyne SIGMAR1 23 41 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Br)C1 ZINC000880566472 ED On-Demand Anodyne EBP 38 42 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne HRH2 31 47 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne CCR3 36 45 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne CHRNA7 16 43 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne NPFFR2 17 40 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne ROCK2 22 43 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne MCHR1 30 40 COc1cncc(NC(=O)NCc2ccccc2CN2CCCC2)c1 ZINC000880566475 EG On-Demand Anodyne NPFFR1 20 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)c(F)c2)C1 ZINC000880566491 CD On-Demand Anodyne CXCR3 21 40 COC(=O)[C@@]1(O)CCN(Cc2ccc3ncccc3c2)C1 ZINC000880566494 CD On-Demand Anodyne CCR3 15 44 COC(=O)[C@@]1(O)CCN(Cc2ccc3ncccc3c2)C1 ZINC000880566494 CD On-Demand Anodyne ADAM17 18 42 COC(=O)[C@@]1(O)CCN(Cc2ccc3ncccc3c2)C1 ZINC000880566494 CD On-Demand Anodyne MCHR2 45 33 COC(=O)[C@@]1(O)CCN(Cc2ccc3ncccc3c2)C1 ZINC000880566494 CD On-Demand Anodyne ABCG2 17 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(Cl)cc2C#N)C1 ZINC000880566498 CD On-Demand Mild TRPV4 45 37 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne HTR4 20 44 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne SSTR5 41 38 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne CCR3 30 41 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne EPHX2 52 43 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne PDK1 46 33 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne CXCR3 22 48 CCN1CCC(NC(=O)Nc2cncc(OC)c2)CC1 ZINC000880566499 CD On-Demand Anodyne MCHR1 18 50 COc1cncc(NC(=O)N(Cc2ccncc2)C2CC2)c1 ZINC000880566500 CF On-Demand Anodyne PDE4A 22 42 COc1cncc(NC(=O)N(Cc2ccncc2)C2CC2)c1 ZINC000880566500 CF On-Demand Anodyne ROCK2 15 51 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccccc2)c1 ZINC000880566505 EF On-Demand Anodyne ROCK1 23 57 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccccc2)c1 ZINC000880566505 EF On-Demand Anodyne ROCK2 35 57 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccccc2)c1 ZINC000880566505 EF On-Demand Anodyne PTGES 19 40 COc1cncc(NC(=O)N(CCN(C)C)Cc2ccccc2)c1 ZINC000880566505 EF On-Demand Anodyne LIMK2 17 43 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C2CC2)c1 ZINC000880566508 DG On-Demand Anodyne GCGR 16 42 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C2CC2)c1 ZINC000880566508 DG On-Demand Anodyne ROCK2 21 52 COc1cncc(NC(=O)N(Cc2ccc(F)cc2)C2CC2)c1 ZINC000880566508 DG On-Demand Anodyne GIPR 39 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CHRM2 19 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CHRM1 15 44 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne DRD2 29 57 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne DRD4 61 57 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne ACHE 45 46 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne DRD3 24 57 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne HTR4 25 46 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CHRM3 25 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne LTA4H 30 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne SIGMAR1 53 59 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne SSTR5 68 40 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CCR3 86 59 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CHRNA7 27 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne UTS2R 24 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne SLC18A3 21 42 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne MLNR 45 33 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne FAAH 24 44 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CCR2 20 44 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne SLC6A5 20 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne EPHX2 45 45 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne PDK1 50 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CXCR3 29 46 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne MCHR1 60 53 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CACNA1G 28 41 COc1cncc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566509 EE On-Demand Anodyne CCR8 24 46 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CHRM2 19 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CHRM1 15 44 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne DRD2 29 57 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne DRD4 61 57 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne ACHE 45 46 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne DRD3 24 57 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne HTR4 25 46 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CHRM3 25 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne LTA4H 30 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne SIGMAR1 53 59 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne SSTR5 68 40 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CCR3 86 59 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CHRNA7 27 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne UTS2R 24 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne SLC18A3 21 42 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne MLNR 45 33 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne FAAH 24 44 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CCR2 20 44 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne SLC6A5 20 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne EPHX2 45 45 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne PDK1 50 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CXCR3 29 46 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne MCHR1 60 53 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CACNA1G 28 41 COc1cncc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2)c1 ZINC000880566510 EE On-Demand Anodyne CCR8 24 46 COc1cncc(NC(=O)N[C@@H](CCSC)c2nnc3ccccn23)c1 ZINC000880566515 FF On-Demand Anodyne FPR1 29 42 COc1cncc(NC(=O)N[C@H](CCSC)c2nnc3ccccn23)c1 ZINC000880566516 FF On-Demand Anodyne FPR1 29 42 COc1cncc(NC(=O)NCCCOC2CCCCC2)c1 ZINC000880566517 DF On-Demand Anodyne HRH2 22 43 COC(=O)[C@@]1(O)CCN(CCCc2ccc(C)cc2)C1 ZINC000880566523 CD On-Demand Anodyne SIGMAR1 22 43 COC(=O)[C@@]1(O)CCN(CC(=O)NOCc2ccccc2)C1 ZINC000880566528 DB On-Demand Anodyne SLC12A5 77 47 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)c(Br)c2)C1 ZINC000880566532 ED On-Demand Anodyne MCHR2 44 34 COc1cncc(NC(=O)N2CCN(Cc3cn4ccccc4n3)CC2)c1 ZINC000880566535 FE On-Demand Anodyne DRD4 24 42 COc1cncc(NC(=O)N2CCN(Cc3cn4ccccc4n3)CC2)c1 ZINC000880566535 FE On-Demand Anodyne FAAH 23 50 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)ccc2Cl)C1 ZINC000880566536 EC On-Demand Anodyne CCR1 48 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(C)ccc2Cl)C1 ZINC000880566536 EC On-Demand Anodyne ABCB1 57 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)ccc2Cl)C1 ZINC000880566538 EC On-Demand Anodyne CCR1 48 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(C)ccc2Cl)C1 ZINC000880566538 EC On-Demand Anodyne ABCB1 57 42 COC(=O)[C@@]1(O)CCN(CCCN2CCCCC2)C1 ZINC000880566541 CC On-Demand Anodyne HRH3 15 40 COC(=O)[C@@]1(O)CCN(CCCN2CCCCC2)C1 ZINC000880566541 CC On-Demand Anodyne EBP 18 42 COc1cncc(NC(=O)N(Cc2ccccc2F)C2CC2)c1 ZINC000880566562 DG On-Demand Anodyne ROCK2 15 46 COC(=O)[C@@]1(O)CCN(Cc2nnc(-c3ccc(Cl)cc3)n2C)C1 ZINC000880566566 FD On-Demand Anodyne HSD11B1 25 42 COC(=O)[C@@]1(O)CCN(Cc2nnc(-c3ccc(Cl)cc3)n2C)C1 ZINC000880566566 FD On-Demand Anodyne CCR1 40 38 COc1cncc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)c1 ZINC000880566573 FF On-Demand Clean CASR 19 40 COc1cncc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)c1 ZINC000880566573 FF On-Demand Clean ROCK2 16 41 COc1cncc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)c1 ZINC000880566573 FF On-Demand Clean EPHB4 73 44 COc1cncc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)c1 ZINC000880566573 FF On-Demand Clean STAT6 48 35 COC(=O)[C@@]1(O)CCN(Cc2ccc(F)c(Cl)c2)C1 ZINC000880566574 CD On-Demand Anodyne CXCR3 24 42 COc1cncc(NC(=O)NCc2nc(C)cs2)c1 ZINC000880566587 CE On-Demand Anodyne ROCK2 17 40 COCC[C@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880566588 CD On-Demand Anodyne OPRL1 26 50 COCC[C@@H](c1ccccc1)N1CC[C@](O)(C(=O)OC)C1 ZINC000880566589 CD On-Demand Anodyne OPRL1 26 50 COCC[C@@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880566590 CD On-Demand Anodyne OPRL1 26 50 COCC[C@H](c1ccccc1)N1CC[C@@](O)(C(=O)OC)C1 ZINC000880566591 CD On-Demand Anodyne OPRL1 26 50 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne HTR1A 22 40 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne DRD2 30 40 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne DRD4 43 39 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne ACHE 34 48 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne HRH2 33 42 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne PDGFRB 56 41 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne LTA4H 16 41 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne SIGMAR1 46 45 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne CCR3 26 49 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne NPFFR2 27 42 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne FAAH 45 64 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne MCHR1 31 46 COc1cncc(NC(=O)N2CCCN(Cc3ccccc3)CC2)c1 ZINC000880566604 EF On-Demand Anodyne NPFFR1 36 42 COC(=O)[C@@]1(O)CCN(CCCc2ccncc2)C1 ZINC000880566607 CC On-Demand Anodyne SIGMAR1 19 42 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc3c(c2)OCCO3)c1 ZINC000880566622 FG On-Demand Anodyne EDNRB 45 36 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc3c(c2)OCCO3)c1 ZINC000880566622 FG On-Demand Anodyne EDNRA 38 47 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc3c(c2)OCCO3)c1 ZINC000880566623 FG On-Demand Anodyne EDNRB 45 36 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc3c(c2)OCCO3)c1 ZINC000880566623 FG On-Demand Anodyne EDNRA 38 47 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Cl)C1 ZINC000880566625 CD On-Demand Anodyne ADRA1A 22 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Cl)C1 ZINC000880566625 CD On-Demand Anodyne ADRA1B 17 40 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Cl)C1 ZINC000880566625 CD On-Demand Anodyne SIGMAR1 24 42 COC(=O)[C@@]1(O)CCN(CCCc2ccccc2Cl)C1 ZINC000880566625 CD On-Demand Anodyne EBP 32 41 COc1cncc(NC(=O)N2CCCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880566632 FF On-Demand Mild PDGFRB 42 45 COc1cncc(NC(=O)N2CCCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880566632 FF On-Demand Mild MLNR 19 40 COc1cncc(NC(=O)N2CCCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880566632 FF On-Demand Mild FAAH 26 53 COc1cncc(NC(=O)N2CCCN(Cc3ccc(C#N)cc3)CC2)c1 ZINC000880566632 FF On-Demand Mild MCHR1 17 43 COC(=O)[C@@]1(O)CCN(CC[C@@H](C)OCc2ccccc2)C1 ZINC000880566636 DD On-Demand Anodyne SLC12A5 77 43 COC(=O)[C@@]1(O)CCN(CC[C@H](C)OCc2ccccc2)C1 ZINC000880566637 DD On-Demand Anodyne SLC12A5 77 43 COc1cncc(NC(=O)NC[C@@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566643 EF On-Demand Anodyne ROCK1 34 43 COc1cncc(NC(=O)NC[C@@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566643 EF On-Demand Anodyne MTNR1B 33 42 COc1cncc(NC(=O)NC[C@@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566643 EF On-Demand Anodyne ROCK2 48 43 COc1cncc(NC(=O)NC[C@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566644 EF On-Demand Anodyne ROCK1 34 43 COc1cncc(NC(=O)NC[C@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566644 EF On-Demand Anodyne MTNR1B 33 42 COc1cncc(NC(=O)NC[C@H](c2cccc(OC)c2)N(C)C)c1 ZINC000880566644 EF On-Demand Anodyne ROCK2 48 43 COC(=O)[C@@]1(O)CCN(CCCOCc2ccccc2)C1 ZINC000880566650 CD On-Demand Anodyne UGCG 40 35 COC(=O)[C@@]1(O)CCN(CCCOCc2ccccc2)C1 ZINC000880566650 CD On-Demand Anodyne SIGMAR1 41 40 COC(=O)[C@@]1(O)CCN(CCCOCc2ccccc2)C1 ZINC000880566650 CD On-Demand Anodyne GBA 20 40 COC(=O)[C@@]1(O)CCN(CCCOCc2ccccc2)C1 ZINC000880566650 CD On-Demand Anodyne GBA2 50 40 COC(=O)[C@@]1(O)CCN(CCCOCc2ccccc2)C1 ZINC000880566650 CD On-Demand Anodyne SLC12A5 80 44 COc1cncc(NC(=O)N2CCN(Cc3ccco3)CC2)c1 ZINC000880566651 DE On-Demand Anodyne PDGFRB 48 36 COc1cncc(NC(=O)N2CCN(Cc3ccco3)CC2)c1 ZINC000880566651 DE On-Demand Anodyne FAAH 24 50 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne HRH2 31 50 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne HRH3 23 43 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne CCR3 48 39 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne F2R 41 32 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne NPFFR2 26 42 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne ROCK2 26 43 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne FAAH 15 43 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne FLT3 15 42 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne MCHR1 40 44 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne NPFFR1 35 42 COc1cncc(NC(=O)NCc2ccc(CN3CCCC3)cc2)c1 ZINC000880566668 EG On-Demand Anodyne NAMPT 56 45 COc1cccc(C2=NO[C@H](C(=O)NCc3cn(C4CCC4)nn3)C2)c1 ZINC000880566671 FD On-Demand Anodyne LUCI_PHOPY 19 41 COc1cccc(C2=NO[C@@H](C(=O)NCc3cn(C4CCC4)nn3)C2)c1 ZINC000880566672 FD On-Demand Anodyne LUCI_PHOPY 19 41 COc1cncc(NC(=O)NCCn2ccnc2)c1 ZINC000880566686 CD On-Demand Anodyne TBXAS1 46 42 COc1cncc(NC(=O)NCCn2ccnc2)c1 ZINC000880566686 CD On-Demand Anodyne QPCT 47 60 COc1cncc(NC(=O)NCCc2ccc(OC(F)F)cc2)c1 ZINC000880566687 EG On-Demand Anodyne RAF1 24 41 COc1cncc(NC(=O)NCCc2ccc(OC(F)F)cc2)c1 ZINC000880566687 EG On-Demand Anodyne PTGDR 15 40 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne HRH2 23 40 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne PDGFRB 55 39 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne PTAFR 29 48 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne CCR3 18 41 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne CHRNA7 56 44 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne FAAH 41 59 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne S1PR2 17 42 COc1cncc(NC(=O)N2CCN(Cc3cccnc3)CC2)c1 ZINC000880566699 ED On-Demand Anodyne MCHR1 17 43 COc1cncc(NC(=O)N2CCC(c3nc4ccccc4[nH]3)CC2)c1 ZINC000880566718 FG On-Demand Anodyne HTR2B 15 59 COc1cncc(NC(=O)N2CCC(c3nc4ccccc4[nH]3)CC2)c1 ZINC000880566718 FG On-Demand Anodyne SMO 33 47 COc1cncc(NC(=O)NC2CCN(C3CC3)CC2)c1 ZINC000880566724 CD On-Demand Anodyne EPHX2 48 40 COc1cncc(NC(=O)NC2CCN(C3CC3)CC2)c1 ZINC000880566724 CD On-Demand Anodyne CXCR3 18 42 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne F2 88 47 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne PLG 37 43 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne PRSS1 31 44 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne ACE 33 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne FKBP1A 56 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne OPRM1 31 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne OPRD1 18 40 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne CELA1 27 52 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne ELANE 38 45 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne CTRA_BOVIN 63 33 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne TRY1_BOVIN 106 45 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne NTSR1 83 36 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne NTSR2 55 32 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne CTSG 44 33 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne HLA-A 57 34 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne PREP 83 55 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne CELA2A 51 33 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne LGMN 92 52 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne KLK5 26 44 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne XIAP 47 46 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne BRCA1 61 32 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne TMPRSS11D 83 47 O=C(NCc1cn(C2CCC2)nn1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880566732 GE On-Demand Anodyne TMPRSS6 15 44 COC(=O)[C@@]1(O)CCN(Cc2cncn2Cc2ccccc2)C1 ZINC000880566734 DD On-Demand Anodyne CYP11B1 15 54 COC(=O)[C@@]1(O)CCN(Cc2cncn2Cc2ccccc2)C1 ZINC000880566734 DD On-Demand Anodyne SLC12A5 58 37 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)(C)C)c2)C1 ZINC000880566756 CE On-Demand Anodyne MCHR2 44 33 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)(C)C)c2)C1 ZINC000880566756 CE On-Demand Anodyne SLC12A5 55 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne CYP19A1 15 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne MME 52 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne ANPEP 48 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne TBXAS1 54 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne FCER2 72 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne CYP27B1 46 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne NPFFR1 42 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566758 GF On-Demand Anodyne GPR142 53 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne CYP19A1 15 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne MME 52 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne ANPEP 48 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne TBXAS1 54 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne FCER2 72 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne CYP27B1 46 37 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne NPFFR1 42 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566759 GF On-Demand Anodyne GPR142 53 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne CYP19A1 15 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne MME 52 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne ANPEP 48 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne TBXAS1 54 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne FCER2 72 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne CYP27B1 46 37 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne NPFFR1 42 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566760 GF On-Demand Anodyne GPR142 53 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne CYP19A1 15 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne MME 52 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne ANPEP 48 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne TBXAS1 54 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne FCER2 72 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne CYP27B1 46 37 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne NPFFR1 42 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566761 GF On-Demand Anodyne GPR142 53 41 COC(=O)[C@@]1(O)CCN(Cc2oc(-c3ccccc3)nc2C)C1 ZINC000880566777 DD On-Demand Anodyne PDE8B 61 38 C=CCN(CC=C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566782 DE On-Demand Mild TBXAS1 39 40 C=CCN(CC=C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566782 DE On-Demand Mild CYP27B1 49 33 C=CCN(CC=C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566783 DE On-Demand Mild TBXAS1 39 40 C=CCN(CC=C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566783 DE On-Demand Mild CYP27B1 49 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC[C@@H]1COc2ccccc2O1 ZINC000880566792 GE On-Demand Anodyne ADRA2B 15 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC[C@H]1COc2ccccc2O1 ZINC000880566793 GE On-Demand Anodyne ADRA2B 15 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC[C@H]1COc2ccccc2O1 ZINC000880566794 GE On-Demand Anodyne ADRA2B 15 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC[C@@H]1COc2ccccc2O1 ZINC000880566795 GE On-Demand Anodyne ADRA2B 15 40 COC(=O)[C@@]1(O)CCN([C@@H]2CCC[C@H]2O)C1 ZINC000880566806 BB On-Demand Anodyne SLC18A3 26 40 COc1cncc(NC(=O)N(C)Cc2ccccc2N2CCCC2)c1 ZINC000880566828 EG On-Demand Anodyne KCNQ2 74 41 COc1cncc(NC(=O)N2CCCN(C(C)=O)CC2)c1 ZINC000880566849 CD On-Demand Anodyne PDGFRB 45 38 COC(=O)[C@@]1(O)CCN(Cc2cc(O)cc(C(F)(F)F)c2)C1 ZINC000880566855 DD On-Demand Anodyne TACR1 18 42 COc1cncc(NC(=O)N2CCN(c3ccncc3)CC2)c1 ZINC000880566856 DD On-Demand Anodyne PDGFRB 55 42 COc1cncc(NC(=O)N2CCN(c3ccncc3)CC2)c1 ZINC000880566856 DD On-Demand Anodyne FAAH 18 46 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCc3ccccc3C2)C1 ZINC000880566859 CD On-Demand Anodyne PTGIR 42 32 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCc3ccccc3C2)C1 ZINC000880566859 CD On-Demand Anodyne SIGMAR1 17 46 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCc3ccccc3C2)C1 ZINC000880566859 CD On-Demand Anodyne PREP 26 41 COC(=O)[C@@]1(O)CCN(C[C@H]2CCc3ccccc3C2)C1 ZINC000880566865 CD On-Demand Anodyne PTGIR 42 32 COC(=O)[C@@]1(O)CCN(C[C@H]2CCc3ccccc3C2)C1 ZINC000880566865 CD On-Demand Anodyne SIGMAR1 17 46 COC(=O)[C@@]1(O)CCN(C[C@H]2CCc3ccccc3C2)C1 ZINC000880566865 CD On-Demand Anodyne PREP 26 41 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne DRD4 47 36 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne LTA4H 37 46 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne HRH3 18 47 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne SIGMAR1 16 42 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne MMP13 17 49 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne MTNR1A 36 46 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne MTNR1B 39 46 COC(=O)[C@@]1(O)CCN(CCOc2cccc(OC)c2)C1 ZINC000880566877 CC On-Demand Anodyne EPHX2 19 40 COc1cncc(NC(=O)N(C)Cc2cnn(C)c2)c1 ZINC000880566880 CD On-Demand Anodyne ROCK2 18 42 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(F)cc2)C1 ZINC000880566884 CD On-Demand Anodyne DRD2 31 47 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(F)cc2)C1 ZINC000880566884 CD On-Demand Anodyne DRD4 15 50 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(F)cc2)C1 ZINC000880566884 CD On-Demand Anodyne HTR2A 18 50 COC(=O)[C@@]1(O)CCN(CCC(=O)c2ccc(F)cc2)C1 ZINC000880566884 CD On-Demand Anodyne ERG2 21 47 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566896 FD On-Demand Anodyne ADRB2 21 40 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566896 FD On-Demand Anodyne CCR1 44 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566896 FD On-Demand Anodyne ABCB1 79 50 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566898 FD On-Demand Anodyne ADRB2 21 40 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566898 FD On-Demand Anodyne CCR1 44 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2ccccc2C(F)(F)F)C1 ZINC000880566898 FD On-Demand Anodyne ABCB1 79 50 COC(=O)/C=C\c1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566906 EC On-Demand Anodyne MMP13 19 43 COC(=O)/C=C\c1ccc(OCCN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880566906 EC On-Demand Anodyne MMP9 15 43 COC(=O)/C=C\c1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566909 EC On-Demand Anodyne MMP13 19 43 COC(=O)/C=C\c1ccc(OCCN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880566909 EC On-Demand Anodyne MMP9 15 43 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(C)cc2)C1 ZINC000880566912 EC On-Demand Anodyne ADRA1A 16 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(C)cc2)C1 ZINC000880566912 EC On-Demand Anodyne MMP13 27 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(C)cc2)C1 ZINC000880566912 EC On-Demand Anodyne ADAM17 29 42 COC(=O)[C@@]1(O)CCN(CCCS(=O)(=O)c2ccc(C)cc2)C1 ZINC000880566912 EC On-Demand Anodyne MMP9 18 42 COC(=O)[C@@]1(O)CCN(CCC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880566926 FD On-Demand Anodyne GPR119 28 41 COC(=O)[C@@]1(O)CCN(Cc2ccc(CO)cc2)C1 ZINC000880566929 CC On-Demand Anodyne MMP13 17 44 COc1cncc(NC(=O)N[C@H](C)CCc2ccc(O)cc2)c1 ZINC000880566930 DF On-Demand Anodyne ADRB1 18 43 COc1cncc(NC(=O)N[C@H](C)CCc2ccc(O)cc2)c1 ZINC000880566930 DF On-Demand Anodyne ADRB3 16 43 COc1cncc(NC(=O)N[C@H](C)CCc2ccc(O)cc2)c1 ZINC000880566930 DF On-Demand Anodyne CCR3 40 31 COc1cncc(NC(=O)N[C@H](C)CCc2ccc(O)cc2)c1 ZINC000880566930 DF On-Demand Anodyne GRIA1 46 32 COc1cncc(NC(=O)N[C@@H](C)CCc2ccc(O)cc2)c1 ZINC000880566931 DF On-Demand Anodyne ADRB1 18 43 COc1cncc(NC(=O)N[C@@H](C)CCc2ccc(O)cc2)c1 ZINC000880566931 DF On-Demand Anodyne ADRB3 16 43 COc1cncc(NC(=O)N[C@@H](C)CCc2ccc(O)cc2)c1 ZINC000880566931 DF On-Demand Anodyne CCR3 40 31 COc1cncc(NC(=O)N[C@@H](C)CCc2ccc(O)cc2)c1 ZINC000880566931 DF On-Demand Anodyne GRIA1 46 32 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(=O)OC(C)(C)C)C1 ZINC000880566933 FD On-Demand Anodyne HCN1 61 33 COC(=O)[C@@]1(O)CCN(CCOc2ccccc2C(=O)OC(C)(C)C)C1 ZINC000880566933 FD On-Demand Anodyne HCN4 48 32 COc1cncc(NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000880566934 EF On-Demand Anodyne PDGFRB 53 41 COc1cncc(NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000880566934 EF On-Demand Anodyne CCKAR 31 40 COc1cncc(NC(=O)N2CCN(c3cccc(C)c3)CC2)c1 ZINC000880566934 EF On-Demand Anodyne FAAH 21 46 C[C@@]1(C(=O)NCc2cn(C3CCC3)nn2)CCN(C(=O)OCc2ccccc2)C1 ZINC000880566936 GF On-Demand Anodyne PREP 40 50 C[C@@]1(C(=O)NCc2cn(C3CCC3)nn2)CCN(C(=O)OCc2ccccc2)C1 ZINC000880566936 GF On-Demand Anodyne SLC12A5 53 35 COC(=O)[C@@]1(O)CCN(Cc2ccc(C#N)cc2C(F)(F)F)C1 ZINC000880566983 ED On-Demand Mild ABL2 43 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC1CCCCC1 ZINC000880566992 EF On-Demand Anodyne TBXAS1 41 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC1CCCCC1 ZINC000880566993 EF On-Demand Anodyne TBXAS1 41 38 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880566995 GF On-Demand Anodyne TRY1_BOVIN 22 43 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880566995 GF On-Demand Anodyne REN 70 37 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880566995 GF On-Demand Anodyne FPR1 47 38 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)c1ccccc1 ZINC000880566995 GF On-Demand Anodyne Q82323_9DELA 40 30 CCN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566997 DE On-Demand Anodyne CYP19A1 16 41 CCN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566997 DE On-Demand Anodyne TBXAS1 65 44 CCN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566997 DE On-Demand Anodyne CYP24A1 42 34 CCN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566997 DE On-Demand Anodyne CYP26A1 48 35 CCN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880566997 DE On-Demand Anodyne CYP27B1 55 34 CCN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566998 DE On-Demand Anodyne CYP19A1 16 41 CCN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566998 DE On-Demand Anodyne TBXAS1 65 44 CCN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566998 DE On-Demand Anodyne CYP24A1 42 34 CCN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566998 DE On-Demand Anodyne CYP26A1 48 35 CCN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880566998 DE On-Demand Anodyne CYP27B1 55 34 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)nc2)C1 ZINC000880567004 ED On-Demand Anodyne ADAM17 17 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OCc3ccccc3)nc2)C1 ZINC000880567004 ED On-Demand Anodyne SLC12A5 69 38 COC(=O)[C@@]1(O)CCN(CCC(=O)Nc2cccnc2)C1 ZINC000880567022 CC On-Demand Anodyne CHRNA7 25 42 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HTR1A 25 40 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne DRD4 43 33 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HRH2 40 52 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HTR2A 20 52 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HTR2C 18 41 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne DRD3 49 39 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HTR4 17 46 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HRH3 26 42 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne NPY1R 16 47 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne CCR3 53 52 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne CHRNA7 30 56 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne EBP 16 42 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne HNMT 46 32 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne MCHR1 16 49 COc1cncc(NC(=O)NCCCN2CCCCC2)c1 ZINC000880567031 CE On-Demand Anodyne QPCT 30 43 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne SIGMAR1 36 48 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP13 44 56 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne ADAM17 24 56 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP2 17 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP3 27 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP8 15 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP9 37 56 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MMP1 34 56 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne MCHR1 18 44 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne PROKR1 58 32 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2)C1 ZINC000880567035 CC On-Demand Anodyne NOD2 33 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567036 FF On-Demand Anodyne TBXAS1 59 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567036 FF On-Demand Anodyne AMP1_PLAFQ 31 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567036 FF On-Demand Anodyne CYP24A1 40 38 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567036 FF On-Demand Anodyne CYP27B1 52 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567038 FF On-Demand Anodyne TBXAS1 59 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567038 FF On-Demand Anodyne AMP1_PLAFQ 31 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567038 FF On-Demand Anodyne CYP24A1 40 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCCCc1ccccc1 ZINC000880567038 FF On-Demand Anodyne CYP27B1 52 38 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2ccc(Cl)cc2Cl)C1 ZINC000880567043 ED On-Demand Anodyne CCR1 43 33 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2ccc(Cl)cc2Cl)C1 ZINC000880567049 ED On-Demand Anodyne CCR1 43 33 COC(=O)[C@@]1(O)CCN(C[C@H]2CC(c3ccc(Cl)cc3)=NO2)C1 ZINC000880567055 ED On-Demand Anodyne LUCI_PHOPY 65 44 COC(=O)[C@@]1(O)CCN(C[C@@H]2CC(c3ccc(Cl)cc3)=NO2)C1 ZINC000880567057 ED On-Demand Anodyne LUCI_PHOPY 65 44 CCC(CC)[C@@H](CNC(=O)c1cc(-c2cccnc2)nc2ccccc12)N1CCOCC1 ZINC000880567064 II On-Demand Anodyne TACR3 49 46 CCC(CC)[C@H](CNC(=O)c1cc(-c2cccnc2)nc2ccccc12)N1CCOCC1 ZINC000880567065 II On-Demand Anodyne TACR3 49 46 CC[C@@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567066 EG On-Demand Anodyne CCR5 18 40 CC[C@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567067 EG On-Demand Anodyne CCR5 18 40 CC[C@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567068 EG On-Demand Anodyne CCR5 18 40 CC[C@@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567070 EG On-Demand Anodyne CCR5 18 40 COC(=O)[C@@]1(O)CCN(CCOC(=O)Cc2ccccc2)C1 ZINC000880567084 DC On-Demand Anodyne LTA4H 31 41 COC(=O)[C@@]1(O)CCN(CCOC(=O)Cc2ccccc2)C1 ZINC000880567084 DC On-Demand Anodyne SIGMAR1 26 40 COC(=O)[C@@]1(O)CCN(CCOC(=O)Cc2ccccc2)C1 ZINC000880567084 DC On-Demand Anodyne SLC12A5 76 42 COC(=O)[C@@]1(O)CCN(Cc2ccc3c(c2)COC3)C1 ZINC000880567087 CC On-Demand Anodyne MCHR2 70 37 COC(=O)[C@@]1(O)CCN(CCSc2cccc(OC)c2)C1 ZINC000880567090 DD On-Demand Anodyne DRD4 45 34 COC(=O)[C@@]1(O)CCN(CCSc2cccc(OC)c2)C1 ZINC000880567090 DD On-Demand Anodyne MTNR1A 24 49 COC(=O)[C@@]1(O)CCN(CCSc2cccc(OC)c2)C1 ZINC000880567090 DD On-Demand Anodyne MTNR1B 30 49 C=C(C)CN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567097 EF On-Demand Mild TBXAS1 40 40 C=C(C)CN(CC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567097 EF On-Demand Mild CYP27B1 43 31 C=C(C)CN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567099 EF On-Demand Mild TBXAS1 40 40 C=C(C)CN(CC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567099 EF On-Demand Mild CYP27B1 43 31 COc1cncc(NC(=O)NC[C@H](Cc2ccccc2)N(C)C)c1 ZINC000880567108 EE On-Demand Anodyne ROCK2 24 40 COc1cncc(NC(=O)NC[C@H](Cc2ccccc2)N(C)C)c1 ZINC000880567108 EE On-Demand Anodyne NPY5R 21 44 COc1cncc(NC(=O)NC[C@@H](Cc2ccccc2)N(C)C)c1 ZINC000880567109 EE On-Demand Anodyne ROCK2 24 40 COc1cncc(NC(=O)NC[C@@H](Cc2ccccc2)N(C)C)c1 ZINC000880567109 EE On-Demand Anodyne NPY5R 21 44 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCO3)c1 ZINC000880567144 DE On-Demand Anodyne EDNRB 56 38 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCO3)c1 ZINC000880567144 DE On-Demand Anodyne EDNRA 57 40 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCO3)c1 ZINC000880567144 DE On-Demand Anodyne BMP1 70 43 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCO3)c1 ZINC000880567144 DE On-Demand Anodyne NOS2 72 40 COc1cncc(NC(=O)NCCc2ccc3c(c2)OCO3)c1 ZINC000880567144 DE On-Demand Anodyne MCHR1 15 49 COC(=O)[C@@]1(O)CCN(CC[C@@](C#N)(C(C)=O)c2ccccc2)C1 ZINC000880567151 ED On-Demand Mild CCR1 20 49 COC(=O)[C@@]1(O)CCN(CC[C@@](C#N)(C(C)=O)c2ccccc2)C1 ZINC000880567151 ED On-Demand Mild SLC12A5 40 34 COC(=O)[C@@]1(O)CCN(CC[C@](C#N)(C(C)=O)c2ccccc2)C1 ZINC000880567153 ED On-Demand Mild CCR1 20 49 COC(=O)[C@@]1(O)CCN(CC[C@](C#N)(C(C)=O)c2ccccc2)C1 ZINC000880567153 ED On-Demand Mild SLC12A5 40 34 C[C@@H]1CCCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880567157 EE On-Demand Anodyne TBXAS1 40 40 C[C@@H]1CCCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880567164 EE On-Demand Anodyne TBXAS1 40 40 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880567165 ED On-Demand Mild MMP13 20 41 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880567165 ED On-Demand Mild MMP2 26 42 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880567165 ED On-Demand Mild MMP14 19 42 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880567165 ED On-Demand Mild MMP9 22 42 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(OC(F)(F)F)cc2)C1 ZINC000880567165 ED On-Demand Mild EPHX2 43 38 COC(=O)[C@@]1(O)CCN(C[C@H]2CCc3ccccc32)C1 ZINC000880567182 CD On-Demand Anodyne SIGMAR1 20 46 COC(=O)[C@@]1(O)CCN(C[C@H]2CCc3ccccc32)C1 ZINC000880567182 CD On-Demand Anodyne EBP 17 40 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCc3ccccc32)C1 ZINC000880567183 CD On-Demand Anodyne SIGMAR1 20 46 COC(=O)[C@@]1(O)CCN(C[C@@H]2CCc3ccccc32)C1 ZINC000880567183 CD On-Demand Anodyne EBP 17 40 O=C(NCc1cn(C2CCC2)nn1)C(F)(F)Cc1ccccc1 ZINC000880567188 DE On-Demand Anodyne PREP 19 41 COC(=O)[C@@]1(O)CCN(C[C@@H](O)CN2CCN(c3ccc(OC)cc3)CC2)C1 ZINC000880567200 GB On-Demand Clean ABCB1 42 42 COC(=O)[C@@]1(O)CCN(C[C@H](O)CN2CCN(c3ccc(OC)cc3)CC2)C1 ZINC000880567204 GB On-Demand Clean ABCB1 42 42 COC(=O)[C@@]1(O)CCN(Cc2cc(Cl)nc3ccccc23)C1 ZINC000880567207 DD On-Demand Anodyne ADAM17 65 39 COc1cncc(NC(=O)N2CCC[C@H]2c2cccnc2)c1 ZINC000880567211 CF On-Demand Anodyne CHRNA7 32 50 COc1cncc(NC(=O)N2CCC[C@@H]2c2cccnc2)c1 ZINC000880567212 CF On-Demand Anodyne CHRNA7 32 50 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(Cl)c2)C1 ZINC000880567217 CD On-Demand Anodyne PDE5A 48 39 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(Cl)c2)C1 ZINC000880567217 CD On-Demand Anodyne SIGMAR1 15 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)c(Cl)c2)C1 ZINC000880567217 CD On-Demand Anodyne PDE6A 41 32 COc1cncc(NC(=O)N2CCN(Cc3ccsc3)CC2)c1 ZINC000880567218 EF On-Demand Anodyne PDGFRB 43 35 COc1cncc(NC(=O)N2CCN(Cc3ccsc3)CC2)c1 ZINC000880567218 EF On-Demand Anodyne FAAH 29 53 COc1cncc(NC(=O)N2CCN(Cc3ccsc3)CC2)c1 ZINC000880567218 EF On-Demand Anodyne NPBWR1 43 30 COC(=O)[C@@]1(O)CCN(CC2(O)CCC(c3ccccc3)CC2)C1 ZINC000880567223 ED On-Demand Anodyne SIGMAR1 18 41 COC(=O)[C@@]1(O)CCN(CC2(O)CCC(c3ccccc3)CC2)C1 ZINC000880567223 ED On-Demand Anodyne SLC12A5 42 35 COc1cncc(NC(=O)NCc2ccc(OC(F)F)c(OC)c2)c1 ZINC000880567227 FG On-Demand Anodyne ROCK2 27 51 COC(=O)[C@@]1(O)CCN(CC#Cc2ccccc2)C1 ZINC000880567234 CC On-Demand Mild SLC12A5 62 38 COC(=O)[C@@]1(O)CCN(Cc2cnn(Cc3ccccc3)c2)C1 ZINC000880567243 DD On-Demand Anodyne SIGMAR1 51 39 COC(=O)[C@@]1(O)CCN(Cc2cnn(Cc3ccccc3)c2)C1 ZINC000880567243 DD On-Demand Anodyne NPFFR1 43 39 COC(=O)[C@@]1(O)CCN(Cc2cnn(Cc3ccccc3)c2)C1 ZINC000880567243 DD On-Demand Anodyne SLC12A5 46 36 COc1cncc(NC(=O)N2CCN(Cc3cccs3)CC2)c1 ZINC000880567244 EF On-Demand Anodyne PDGFRB 43 36 COc1cncc(NC(=O)N2CCN(Cc3cccs3)CC2)c1 ZINC000880567244 EF On-Demand Anodyne FAAH 25 50 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@@H]3CCCO3)cc2)C1 ZINC000880567247 ED On-Demand Anodyne HRH3 15 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@@H]3CCCO3)cc2)C1 ZINC000880567247 ED On-Demand Anodyne MMP13 24 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@@H]3CCCO3)cc2)C1 ZINC000880567247 ED On-Demand Anodyne ADAM17 20 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@H]3CCCO3)cc2)C1 ZINC000880567248 ED On-Demand Anodyne HRH3 15 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@H]3CCCO3)cc2)C1 ZINC000880567248 ED On-Demand Anodyne MMP13 24 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC[C@H]3CCCO3)cc2)C1 ZINC000880567248 ED On-Demand Anodyne ADAM17 20 40 COc1cncc(NC(=O)N2CCN(Cc3ccncc3)CC2)c1 ZINC000880567255 ED On-Demand Anodyne PDGFRB 54 37 COc1cncc(NC(=O)N2CCN(Cc3ccncc3)CC2)c1 ZINC000880567255 ED On-Demand Anodyne FAAH 36 59 COc1cncc(NC(=O)N2CCN(Cc3ccncc3)CC2)c1 ZINC000880567255 ED On-Demand Anodyne MCHR1 22 46 COc1cncc(NC(=O)N2CCN(Cc3cc(C)no3)CC2)c1 ZINC000880567260 ED On-Demand Anodyne FAAH 16 45 COc1cncc(NC(=O)N2CCN(c3cccc(O)c3)CC2)c1 ZINC000880567278 EE On-Demand Anodyne PDGFRB 53 41 COc1cncc(NC(=O)N2CCN(c3cccc(O)c3)CC2)c1 ZINC000880567278 EE On-Demand Anodyne FAAH 18 46 COC(=O)[C@@]1(O)CCN(CCCc2ccsc2)C1 ZINC000880567279 CD On-Demand Anodyne SLC12A5 15 40 COc1cncc(NC(=O)NCCN(C)c2ccccc2)c1 ZINC000880567282 DE On-Demand Anodyne MTNR1A 26 45 COc1cncc(NC(=O)NCCN(C)c2ccccc2)c1 ZINC000880567282 DE On-Demand Anodyne MTNR1B 24 45 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR1A 56 45 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne DRD2 48 45 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne DRD4 43 39 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR1D 30 42 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR1B 30 42 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR2A 35 49 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR2C 21 40 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne DRD3 57 42 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne PDGFRB 57 42 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne HTR7 44 41 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne SIGMAR1 44 50 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne CCR3 25 46 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne CHRNA7 29 40 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne FAAH 45 55 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne ABCB1 47 41 COc1cncc(NC(=O)N2CCN(CCc3ccccc3)CC2)c1 ZINC000880567286 EE On-Demand Anodyne ABCG2 27 40 COC(=O)[C@@]1(O)CCN([C@@H](C#N)c2ccc(Cl)cc2)C1 ZINC000880567293 CD On-Demand Mild CCR1 23 42 COC(=O)[C@@]1(O)CCN([C@H](C#N)c2ccc(Cl)cc2)C1 ZINC000880567298 CD On-Demand Mild CCR1 23 42 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP19A1 22 42 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP11B1 43 40 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne TBXAS1 65 44 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP11B2 22 40 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP24A1 44 36 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP26A1 33 42 CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567311 CD On-Demand Anodyne CYP27B1 57 36 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP19A1 22 42 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP11B1 43 40 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne TBXAS1 65 44 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP11B2 22 40 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP24A1 44 36 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP26A1 33 42 CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567312 CD On-Demand Anodyne CYP27B1 57 36 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567342 FF On-Demand Anodyne ADRB2 23 45 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567342 FF On-Demand Anodyne ADRB1 49 33 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567343 FF On-Demand Anodyne ADRB2 23 45 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567343 FF On-Demand Anodyne ADRB1 49 33 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567344 FF On-Demand Anodyne ADRB2 23 45 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567344 FF On-Demand Anodyne ADRB1 49 33 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567345 FF On-Demand Anodyne ADRB2 23 45 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1F ZINC000880567345 FF On-Demand Anodyne ADRB1 49 33 COC(=O)[C@@]1(O)CCN(CC#Cc2ccc(F)cc2)C1 ZINC000880567346 CC On-Demand Mild GRIN2C 17 45 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880567366 GE On-Demand Anodyne PDGFRB 60 39 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880567366 GE On-Demand Anodyne FAAH 18 46 COc1cncc(NC(=O)N2CCN(CC(=O)Nc3ccc(F)cc3)CC2)c1 ZINC000880567366 GE On-Demand Anodyne S1PR2 27 40 COc1cncc(NC(=O)N[C@@H](CN(C)C)c2ccccc2)c1 ZINC000880567376 DF On-Demand Anodyne ROCK1 15 46 COc1cncc(NC(=O)N[C@@H](CN(C)C)c2ccccc2)c1 ZINC000880567376 DF On-Demand Anodyne ROCK2 19 46 COc1cncc(NC(=O)N[C@@H](CN(C)C)c2ccccc2)c1 ZINC000880567376 DF On-Demand Anodyne PAK4 53 40 COc1cncc(NC(=O)N[C@@H](CN(C)C)c2ccccc2)c1 ZINC000880567376 DF On-Demand Anodyne UTS2 48 36 COc1cncc(NC(=O)N[C@H](CN(C)C)c2ccccc2)c1 ZINC000880567377 DF On-Demand Anodyne ROCK1 15 46 COc1cncc(NC(=O)N[C@H](CN(C)C)c2ccccc2)c1 ZINC000880567377 DF On-Demand Anodyne ROCK2 19 46 COc1cncc(NC(=O)N[C@H](CN(C)C)c2ccccc2)c1 ZINC000880567377 DF On-Demand Anodyne PAK4 53 40 COc1cncc(NC(=O)N[C@H](CN(C)C)c2ccccc2)c1 ZINC000880567377 DF On-Demand Anodyne UTS2 48 36 COc1cncc(NC(=O)N2CCC[C@H]2c2ccc(F)cc2)c1 ZINC000880567384 DH On-Demand Anodyne CCR3 17 44 COc1cncc(NC(=O)N2CCC[C@@H]2c2ccc(F)cc2)c1 ZINC000880567385 DH On-Demand Anodyne CCR3 17 44 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2ccc(Cl)cc2)C1 ZINC000880567410 CC On-Demand Anodyne CCR1 60 36 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2ccc(Cl)cc2)C1 ZINC000880567413 CC On-Demand Anodyne CCR1 60 36 COc1cncc(NC(=O)N2CCN(c3ccc(C(C)=O)cc3F)CC2)c1 ZINC000880567416 FF On-Demand Anodyne HTR1B 15 48 COc1cncc(NC(=O)N2CCN(c3ccc(C(C)=O)cc3F)CC2)c1 ZINC000880567416 FF On-Demand Anodyne PDGFRB 55 41 COc1cncc(NC(=O)N2CCN(c3ccc(C(C)=O)cc3F)CC2)c1 ZINC000880567416 FF On-Demand Anodyne NPY2R 86 39 COc1cncc(NC(=O)N2CCN(c3ccc(C(C)=O)cc3F)CC2)c1 ZINC000880567416 FF On-Demand Anodyne SLC6A9 17 42 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567426 FD On-Demand Anodyne ACOX1 51 31 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567426 FD On-Demand Anodyne CCR1 46 39 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567426 FD On-Demand Anodyne ABCB1 40 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567426 FD On-Demand Anodyne CACNA1I 42 36 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567427 FD On-Demand Anodyne ACOX1 51 31 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567427 FD On-Demand Anodyne CCR1 46 39 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567427 FD On-Demand Anodyne ABCB1 40 37 COC(=O)[C@@]1(O)CCN(C[C@H](O)COc2cc(Cl)cc(Cl)c2)C1 ZINC000880567427 FD On-Demand Anodyne CACNA1I 42 36 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)N[C@H](C)c2ccccc2)C1 ZINC000880567429 DC On-Demand Anodyne OPRL1 21 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)N[C@H](C)c2ccccc2)C1 ZINC000880567430 DC On-Demand Anodyne OPRL1 21 41 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne CYP19A1 35 43 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne CYP11B1 48 43 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne TBXAS1 41 44 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne CYP11B2 25 43 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne CYP24A1 49 35 COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567440 BD On-Demand Anodyne CYP27B1 66 35 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne CYP19A1 35 43 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne CYP11B1 48 43 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne TBXAS1 41 44 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne CYP11B2 25 43 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne CYP24A1 49 35 COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567441 BD On-Demand Anodyne CYP27B1 66 35 CCOC(=O)[C@]1(c2ccccc2)C[C@H]1N1CC[C@@](O)(C(=O)OC)C1 ZINC000880567442 EC On-Demand Anodyne KCNA3 15 44 CCOC(=O)[C@]1(c2ccccc2)C[C@H]1N1CC[C@@](O)(C(=O)OC)C1 ZINC000880567442 EC On-Demand Anodyne SLC12A5 60 38 CCOC(=O)[C@]1(c2ccccc2)C[C@H]1N1CC[C@](O)(C(=O)OC)C1 ZINC000880567443 EC On-Demand Anodyne KCNA3 15 44 CCOC(=O)[C@]1(c2ccccc2)C[C@H]1N1CC[C@](O)(C(=O)OC)C1 ZINC000880567443 EC On-Demand Anodyne SLC12A5 60 38 CCOC(=O)[C@]1(c2ccccc2)C[C@@H]1N1CC[C@](O)(C(=O)OC)C1 ZINC000880567444 EC On-Demand Anodyne KCNA3 15 44 CCOC(=O)[C@]1(c2ccccc2)C[C@@H]1N1CC[C@](O)(C(=O)OC)C1 ZINC000880567444 EC On-Demand Anodyne SLC12A5 60 38 CCOC(=O)[C@]1(c2ccccc2)C[C@@H]1N1CC[C@@](O)(C(=O)OC)C1 ZINC000880567445 EC On-Demand Anodyne KCNA3 15 44 CCOC(=O)[C@]1(c2ccccc2)C[C@@H]1N1CC[C@@](O)(C(=O)OC)C1 ZINC000880567445 EC On-Demand Anodyne SLC12A5 60 38 COC(=O)[C@@]1(O)CCN(CCCC2CCC2)C1 ZINC000880567446 BD On-Demand Anodyne EBP 21 48 CCN1CCC(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567504 FD On-Demand Anodyne SIGMAR1 15 41 CCN1CCC(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567505 FD On-Demand Anodyne SIGMAR1 15 41 CC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567512 FC On-Demand Anodyne TBXAS1 58 42 CC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567512 FC On-Demand Anodyne PTAFR 34 45 CC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567512 FC On-Demand Anodyne CYP24A1 46 35 CC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567512 FC On-Demand Anodyne CYP27B1 61 35 CC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567513 FC On-Demand Anodyne TBXAS1 58 42 CC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567513 FC On-Demand Anodyne PTAFR 34 45 CC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567513 FC On-Demand Anodyne CYP24A1 46 35 CC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567513 FC On-Demand Anodyne CYP27B1 61 35 CN(Cc1ccc(Cl)s1)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567526 GH On-Demand Anodyne TBXAS1 28 40 CN(Cc1ccc(Cl)s1)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567527 GH On-Demand Anodyne TBXAS1 28 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)NC3CC3)cc2)C1 ZINC000880567570 FC On-Demand Anodyne MMP13 34 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)NC3CC3)cc2)C1 ZINC000880567570 FC On-Demand Anodyne ADAM17 23 45 COC(=O)[C@@]1(O)CCN(Cc2ccc(S(=O)(=O)NC3CC3)cc2)C1 ZINC000880567570 FC On-Demand Anodyne MMP9 24 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(C)c(F)c2)C1 ZINC000880567574 CD On-Demand Anodyne MCHR2 44 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567575 DC On-Demand Anodyne TBXAS1 54 39 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567575 DC On-Demand Anodyne CYP24A1 42 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567575 DC On-Demand Anodyne CYP27B1 55 33 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567576 DC On-Demand Anodyne TBXAS1 54 39 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567576 DC On-Demand Anodyne CYP24A1 42 33 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCNC1=O ZINC000880567576 DC On-Demand Anodyne CYP27B1 55 33 COC(=O)[C@@]1(O)CCN(CCOCc2ccccc2)C1 ZINC000880567582 CC On-Demand Anodyne SIGMAR1 33 40 COC(=O)[C@@]1(O)CCN(CCOCc2ccccc2)C1 ZINC000880567582 CC On-Demand Anodyne SLC12A5 82 46 C[C@@H]1CCCC[C@H]1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567591 EF On-Demand Anodyne CYP27B1 43 32 C[C@@H]1CCCC[C@@H]1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567592 EF On-Demand Anodyne CYP27B1 43 32 C[C@@H]1CCCC[C@@H]1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567593 EF On-Demand Anodyne CYP27B1 43 32 C[C@@H]1CCCC[C@H]1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567594 EF On-Demand Anodyne CYP27B1 43 32 COC(=O)[C@@]1(O)CCN(CCCCc2cccc(Cl)c2)C1 ZINC000880567596 DE On-Demand Anodyne HTR1A 19 44 COC(=O)[C@@]1(O)CCN(CCCCc2cccc(Cl)c2)C1 ZINC000880567596 DE On-Demand Anodyne DRD2 18 41 COC(=O)[C@@]1(O)CCN(CCCCc2cccc(Cl)c2)C1 ZINC000880567596 DE On-Demand Anodyne HTR2A 18 41 COC(=O)[C@@]1(O)CCN(CCCCc2cccc(Cl)c2)C1 ZINC000880567596 DE On-Demand Anodyne SIGMAR1 29 41 COC(=O)[C@@]1(O)CCN(CCCCc2cccc(Cl)c2)C1 ZINC000880567596 DE On-Demand Anodyne CCR1 34 41 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567609 EF On-Demand Anodyne ADRB2 50 53 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567609 EF On-Demand Anodyne ADRB1 62 53 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567609 EF On-Demand Anodyne ADRB3 48 41 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567609 EF On-Demand Anodyne TBXAS1 30 46 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567610 EF On-Demand Anodyne ADRB2 50 53 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567610 EF On-Demand Anodyne ADRB1 62 53 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567610 EF On-Demand Anodyne ADRB3 48 41 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567610 EF On-Demand Anodyne TBXAS1 30 46 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567611 EF On-Demand Anodyne ADRB2 50 53 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567611 EF On-Demand Anodyne ADRB1 62 53 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567611 EF On-Demand Anodyne ADRB3 48 41 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567611 EF On-Demand Anodyne TBXAS1 30 46 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567612 EF On-Demand Anodyne ADRB2 50 53 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567612 EF On-Demand Anodyne ADRB1 62 53 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567612 EF On-Demand Anodyne ADRB3 48 41 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1 ZINC000880567612 EF On-Demand Anodyne TBXAS1 30 46 C#CCCOc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880567613 DE On-Demand Mild CA14 19 45 N#CCc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567616 GF On-Demand Mild ADRB2 39 45 N#CCc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567616 GF On-Demand Mild ADRB1 56 45 N#CCc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567616 GF On-Demand Mild ADRB3 42 40 N#CCc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567617 GF On-Demand Mild ADRB2 39 45 N#CCc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567617 GF On-Demand Mild ADRB1 56 45 N#CCc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567617 GF On-Demand Mild ADRB3 42 40 N#CCc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567618 GF On-Demand Mild ADRB2 39 45 N#CCc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567618 GF On-Demand Mild ADRB1 56 45 N#CCc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567618 GF On-Demand Mild ADRB3 42 40 N#CCc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567619 GF On-Demand Mild ADRB2 39 45 N#CCc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567619 GF On-Demand Mild ADRB1 56 45 N#CCc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880567619 GF On-Demand Mild ADRB3 42 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Br)C1 ZINC000880567646 ED On-Demand Anodyne MMP13 23 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Br)C1 ZINC000880567646 ED On-Demand Anodyne ADAM17 18 42 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Br)C1 ZINC000880567646 ED On-Demand Anodyne MTNR1B 27 40 COC(=O)[C@@]1(O)CCN(Cc2ccc(OC)cc2Br)C1 ZINC000880567646 ED On-Demand Anodyne MMP9 19 42 COC(=O)[C@@]1(O)CCN(Cc2ccc3oc(=O)n(C)c3c2)C1 ZINC000880567662 DC On-Demand Anodyne MCHR2 47 35 COC(=O)[C@@]1(O)CCN(C[C@@H]2CC[C@@H](c3ccccc3)C2)C1 ZINC000880567664 DE On-Demand Anodyne SIGMAR1 16 42 CNS(=O)(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880567672 EB On-Demand Anodyne MMP13 37 48 CNS(=O)(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880567672 EB On-Demand Anodyne ADAM17 30 48 CNS(=O)(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880567672 EB On-Demand Anodyne MMP9 26 48 CNS(=O)(=O)c1ccc(CN2CC[C@@](O)(C(=O)OC)C2)cc1 ZINC000880567672 EB On-Demand Anodyne MMP1 16 48 CNS(=O)(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880567673 EB On-Demand Anodyne MMP13 37 48 CNS(=O)(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880567673 EB On-Demand Anodyne ADAM17 30 48 CNS(=O)(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880567673 EB On-Demand Anodyne MMP9 26 48 CNS(=O)(=O)c1ccc(CN2CC[C@](O)(C(=O)OC)C2)cc1 ZINC000880567673 EB On-Demand Anodyne MMP1 16 48 COC(=O)[C@@]1(O)CCN(Cc2nc3cc(C)ccc3s2)C1 ZINC000880567679 DD On-Demand Anodyne AKR1B1 15 41 COC(=O)[C@@]1(O)CCN(Cc2nc3cc(C)ccc3s2)C1 ZINC000880567679 DD On-Demand Anodyne ACOX1 52 31 CC(C)c1ccccc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567690 FH On-Demand Anodyne TBXAS1 49 42 CC(C)c1ccccc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567690 FH On-Demand Anodyne SOAT1 40 38 CC(C)c1ccccc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567690 FH On-Demand Anodyne CYP27B1 43 31 CC(C)c1ccccc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567691 FH On-Demand Anodyne TBXAS1 49 42 CC(C)c1ccccc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567691 FH On-Demand Anodyne SOAT1 40 38 CC(C)c1ccccc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567691 FH On-Demand Anodyne CYP27B1 43 31 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567706 DD On-Demand Anodyne TBXAS1 50 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567706 DD On-Demand Anodyne PTAFR 24 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567706 DD On-Demand Anodyne CYP24A1 41 34 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567706 DD On-Demand Anodyne CYP27B1 54 34 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567707 DD On-Demand Anodyne TBXAS1 50 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567707 DD On-Demand Anodyne PTAFR 24 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567707 DD On-Demand Anodyne CYP24A1 41 34 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880567707 DD On-Demand Anodyne CYP27B1 54 34 COC(=O)[C@@]1(O)CCN(C[C@H](OC)c2ccc(F)cc2)C1 ZINC000880567714 CD On-Demand Anodyne LEF 32 44 COC(=O)[C@@]1(O)CCN(C[C@@H](OC)c2ccc(F)cc2)C1 ZINC000880567716 CD On-Demand Anodyne LEF 32 44 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CC1 ZINC000880567721 CD On-Demand Anodyne TBXAS1 58 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CC1 ZINC000880567721 CD On-Demand Anodyne CYP27B1 40 33 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CC1 ZINC000880567722 CD On-Demand Anodyne TBXAS1 58 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CC1 ZINC000880567722 CD On-Demand Anodyne CYP27B1 40 33 COC(=O)[C@@]1(O)CCN(C[C@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000880567729 ED On-Demand Anodyne TACR2 65 37 COC(=O)[C@@]1(O)CCN(C[C@@H](O)c2ccc(Cl)c(Cl)c2)C1 ZINC000880567732 ED On-Demand Anodyne TACR2 65 37 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild CYP19A1 19 41 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild CYP11B1 35 41 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild TBXAS1 38 42 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild CYP11B2 18 41 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild CYP24A1 41 32 C=C(C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567739 BF On-Demand Mild CYP27B1 53 32 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild CYP19A1 19 41 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild CYP11B1 35 41 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild TBXAS1 38 42 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild CYP11B2 18 41 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild CYP24A1 41 32 C=C(C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567740 BF On-Demand Mild CYP27B1 53 32 Cc1cccc(C(C)C)c1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567749 GI On-Demand Anodyne TBXAS1 38 40 Cc1cccc(C(C)C)c1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567749 GI On-Demand Anodyne SOAT1 53 42 Cc1cccc(C(C)C)c1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567750 GI On-Demand Anodyne TBXAS1 38 40 Cc1cccc(C(C)C)c1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567750 GI On-Demand Anodyne SOAT1 53 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880567761 FF On-Demand Anodyne DPP8 15 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880567761 FF On-Demand Anodyne CYP27B1 43 32 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880567762 FF On-Demand Anodyne DPP8 15 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880567762 FF On-Demand Anodyne CYP27B1 43 32 COC(=O)[C@@]1(O)CCN(CC(=O)c2c[nH]c3ccc(F)cc23)C1 ZINC000880567767 DD On-Demand Anodyne MPO 77 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567769 EF On-Demand Anodyne TBXAS1 62 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567769 EF On-Demand Anodyne PTAFR 30 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567769 EF On-Demand Anodyne CYP24A1 43 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567769 EF On-Demand Anodyne CYP27B1 56 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567770 EF On-Demand Anodyne TBXAS1 62 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567770 EF On-Demand Anodyne PTAFR 30 43 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567770 EF On-Demand Anodyne CYP24A1 43 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCCC1 ZINC000880567770 EF On-Demand Anodyne CYP27B1 56 35 COC(=O)[C@@]1(O)CCN(CC(=O)Nc2ccc(Cl)c(F)c2)C1 ZINC000880567776 ED On-Demand Anodyne ENV 45 40 COC(=O)C1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567780 FD On-Demand Anodyne TBXAS1 44 38 COC(=O)C1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567780 FD On-Demand Anodyne PTAFR 19 41 COC(=O)C1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567780 FD On-Demand Anodyne CYP27B1 40 34 COC(=O)C1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567781 FD On-Demand Anodyne TBXAS1 44 38 COC(=O)C1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567781 FD On-Demand Anodyne PTAFR 19 41 COC(=O)C1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567781 FD On-Demand Anodyne CYP27B1 40 34 Cc1ccccc1[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880567782 GG On-Demand Anodyne REN 55 36 Cc1ccccc1[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880567782 GG On-Demand Anodyne FPR1 43 35 Cc1ccccc1[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880567783 GG On-Demand Anodyne REN 55 36 Cc1ccccc1[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880567783 GG On-Demand Anodyne FPR1 43 35 CC(C)(C)OC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567806 DF On-Demand Anodyne TBXAS1 56 42 CC(C)(C)OC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567806 DF On-Demand Anodyne CYP24A1 49 37 CC(C)(C)OC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567806 DF On-Demand Anodyne CYP26A1 99 41 CC(C)(C)OC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567806 DF On-Demand Anodyne CYP27B1 65 37 CC(C)(C)OC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567807 DF On-Demand Anodyne TBXAS1 56 42 CC(C)(C)OC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567807 DF On-Demand Anodyne CYP24A1 49 37 CC(C)(C)OC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567807 DF On-Demand Anodyne CYP26A1 99 41 CC(C)(C)OC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567807 DF On-Demand Anodyne CYP27B1 65 37 CCOC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567808 GD On-Demand Anodyne P2RY12 114 44 CCOC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567808 GD On-Demand Anodyne TBXAS1 49 41 CCOC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567808 GD On-Demand Anodyne PTAFR 33 42 CCOC(=O)N1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567808 GD On-Demand Anodyne CYP27B1 44 33 CCOC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567809 GD On-Demand Anodyne P2RY12 114 44 CCOC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567809 GD On-Demand Anodyne TBXAS1 49 41 CCOC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567809 GD On-Demand Anodyne PTAFR 33 42 CCOC(=O)N1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880567809 GD On-Demand Anodyne CYP27B1 44 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)Nc1ccc2c(c1)OCCCO2 ZINC000880567810 GG On-Demand Anodyne NOS2 69 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)Nc1ccc2c(c1)OCCCO2 ZINC000880567810 GG On-Demand Anodyne QPCT 35 44 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)Nc1ccc2c(c1)OCCCO2 ZINC000880567811 GG On-Demand Anodyne NOS2 69 33 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)Nc1ccc2c(c1)OCCCO2 ZINC000880567811 GG On-Demand Anodyne QPCT 35 44 CC[C@H](C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567822 DE On-Demand Anodyne TBXAS1 58 42 CC[C@H](C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567822 DE On-Demand Anodyne CYP27B1 40 33 CC[C@H](C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567823 DE On-Demand Anodyne TBXAS1 58 42 CC[C@H](C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567823 DE On-Demand Anodyne CYP27B1 40 33 CN(C)CCc1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880567825 EE On-Demand Anodyne CA14 16 45 COC(=O)[C@@]1(O)CCN(Cc2nnc(-c3cccc4ccccc34)o2)C1 ZINC000880567827 FD On-Demand Anodyne ALOX15 52 36 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCc2ccccc2)C1 ZINC000880567854 EE On-Demand Anodyne PTGER1 48 41 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCc2ccccc2)C1 ZINC000880567854 EE On-Demand Anodyne SIGMAR1 24 40 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCc2ccccc2)C1 ZINC000880567854 EE On-Demand Anodyne ADAM17 19 42 COC(=O)[C@@]1(O)CCN(Cc2ccccc2OCc2ccccc2)C1 ZINC000880567854 EE On-Demand Anodyne SLC12A5 70 40 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1F ZINC000880567855 GG On-Demand Anodyne CYP26A1 42 33 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1F ZINC000880567856 GG On-Demand Anodyne CYP26A1 42 33 N#Cc1ccc(C(=O)NCc2cn(C3CCC3)nn2)o1 ZINC000880567858 CD On-Demand Mild CSF1R 21 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC(=O)NCC(F)(F)F ZINC000880567891 FD On-Demand Anodyne CYP27B1 46 34 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC(=O)NCC(F)(F)F ZINC000880567892 FD On-Demand Anodyne CYP27B1 46 34 COCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567903 DD On-Demand Anodyne TBXAS1 52 42 COCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567903 DD On-Demand Anodyne CYP24A1 41 37 COCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880567903 DD On-Demand Anodyne CYP27B1 52 37 COCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567904 DD On-Demand Anodyne TBXAS1 52 42 COCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567904 DD On-Demand Anodyne CYP24A1 41 37 COCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880567904 DD On-Demand Anodyne CYP27B1 52 37 CC(C)(C)NC(=O)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568033 ED On-Demand Anodyne TBXAS1 44 40 CC(C)(C)NC(=O)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568033 ED On-Demand Anodyne CYP26A1 55 36 CC(C)(C)NC(=O)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568033 ED On-Demand Anodyne CYP27B1 46 34 CC(C)(C)NC(=O)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568034 ED On-Demand Anodyne TBXAS1 44 40 CC(C)(C)NC(=O)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568034 ED On-Demand Anodyne CYP26A1 55 36 CC(C)(C)NC(=O)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568034 ED On-Demand Anodyne CYP27B1 46 34 O=C(NCc1cn(C2CCC2)nn1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568066 GD On-Demand Anodyne CELA1 19 42 O=C(NCc1cn(C2CCC2)nn1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568066 GD On-Demand Anodyne PREP 48 52 O=C(NCc1cn(C2CCC2)nn1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568066 GD On-Demand Anodyne LGMN 71 41 O=C(NCc1cn(C2CCC2)nn1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568066 GD On-Demand Anodyne KLK5 23 40 O=C(NCc1cn(C2CCC2)nn1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568066 GD On-Demand Anodyne TMPRSS11D 68 38 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568067 GD On-Demand Anodyne CELA1 19 42 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568067 GD On-Demand Anodyne PREP 48 52 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568067 GD On-Demand Anodyne LGMN 71 41 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568067 GD On-Demand Anodyne KLK5 23 40 O=C(NCc1cn(C2CCC2)nn1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880568067 GD On-Demand Anodyne TMPRSS11D 68 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(C(C)C)c2)C1 ZINC000880568079 CD On-Demand Anodyne MCHR2 42 33 COC(=O)[C@@]1(O)CCN(C[C@@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568083 EC On-Demand Anodyne DRD4 23 40 COC(=O)[C@@]1(O)CCN(C[C@@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568083 EC On-Demand Anodyne SIGMAR1 61 41 COC(=O)[C@@]1(O)CCN(C[C@@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568083 EC On-Demand Anodyne NPFFR1 44 40 COC(=O)[C@@]1(O)CCN(C[C@@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568083 EC On-Demand Anodyne SLC12A5 62 38 COC(=O)[C@@]1(O)CCN(C[C@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568085 EC On-Demand Anodyne DRD4 23 40 COC(=O)[C@@]1(O)CCN(C[C@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568085 EC On-Demand Anodyne SIGMAR1 61 41 COC(=O)[C@@]1(O)CCN(C[C@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568085 EC On-Demand Anodyne NPFFR1 44 40 COC(=O)[C@@]1(O)CCN(C[C@]2(O)CCN(Cc3ccccc3)C2)C1 ZINC000880568085 EC On-Demand Anodyne SLC12A5 62 38 C[C@@H]1C[C@@H](C)CN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568095 EF On-Demand Anodyne TBXAS1 45 42 C[C@@H]1C[C@@H](C)CN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568095 EF On-Demand Anodyne CYP27B1 49 33 C[C@H]1C[C@@H](C)CN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568096 EF On-Demand Anodyne TBXAS1 45 42 C[C@H]1C[C@@H](C)CN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568096 EF On-Demand Anodyne CYP27B1 49 33 C[C@@H]1C[C@@H](C)CN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568097 EF On-Demand Anodyne TBXAS1 45 42 C[C@@H]1C[C@@H](C)CN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568097 EF On-Demand Anodyne CYP27B1 49 33 C[C@H]1C[C@@H](C)CN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568098 EF On-Demand Anodyne TBXAS1 45 42 C[C@H]1C[C@@H](C)CN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568098 EF On-Demand Anodyne CYP27B1 49 33 COC(=O)[C@@]1(O)CCN(CCCc2c(F)cccc2F)C1 ZINC000880568100 CD On-Demand Anodyne ADRA1A 43 38 COC(=O)[C@@]1(O)CCN(CCc2nsc3ccccc23)C1 ZINC000880568105 DD On-Demand Anodyne HTR1A 19 41 COC(=O)[C@@]1(O)CCN(CCc2nsc3ccccc23)C1 ZINC000880568105 DD On-Demand Anodyne DRD2 25 41 CCOC(=O)C1=C(CN[C@@H](Cn2ccnc2)c2ccccc2)NC(=O)N[C@@H]1C ZINC000880568107 GD On-Demand Anodyne TBXAS1 20 40 CCOC(=O)C1=C(CN[C@H](Cn2ccnc2)c2ccccc2)NC(=O)N[C@@H]1C ZINC000880568108 GD On-Demand Anodyne TBXAS1 20 40 CCOC(=O)C1=C(CN[C@H](Cn2ccnc2)c2ccccc2)NC(=O)N[C@H]1C ZINC000880568109 GD On-Demand Anodyne TBXAS1 20 40 CCOC(=O)C1=C(CN[C@@H](Cn2ccnc2)c2ccccc2)NC(=O)N[C@H]1C ZINC000880568110 GD On-Demand Anodyne TBXAS1 20 40 COC(=O)[C@@]1(O)CCN(CC[C@H]2CCc3ccccc32)C1 ZINC000880568190 CD On-Demand Anodyne SIGMAR1 25 54 COC(=O)[C@@]1(O)CCN(CC[C@H]2CCc3ccccc32)C1 ZINC000880568190 CD On-Demand Anodyne EBP 36 54 COC(=O)[C@@]1(O)CCN(CC[C@@H]2CCc3ccccc32)C1 ZINC000880568191 CD On-Demand Anodyne SIGMAR1 25 54 COC(=O)[C@@]1(O)CCN(CC[C@@H]2CCc3ccccc32)C1 ZINC000880568191 CD On-Demand Anodyne EBP 36 54 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)(F)F)c2)C1 ZINC000880568197 DD On-Demand Anodyne SIGMAR1 15 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)(F)F)c2)C1 ZINC000880568197 DD On-Demand Anodyne MMP2 21 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)(F)F)c2)C1 ZINC000880568197 DD On-Demand Anodyne MMP14 18 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC(F)(F)F)c2)C1 ZINC000880568197 DD On-Demand Anodyne CCR8 25 40 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568199 FF On-Demand Anodyne ADRB2 45 48 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568199 FF On-Demand Anodyne ADRB1 61 48 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568199 FF On-Demand Anodyne CYP19A1 18 47 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568199 FF On-Demand Anodyne ADRB3 43 42 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568199 FF On-Demand Anodyne ABCB1 15 40 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568200 FF On-Demand Anodyne ADRB2 45 48 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568200 FF On-Demand Anodyne ADRB1 61 48 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568200 FF On-Demand Anodyne CYP19A1 18 47 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568200 FF On-Demand Anodyne ADRB3 43 42 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568200 FF On-Demand Anodyne ABCB1 15 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568201 FF On-Demand Anodyne ADRB2 45 48 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568201 FF On-Demand Anodyne ADRB1 61 48 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568201 FF On-Demand Anodyne CYP19A1 18 47 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568201 FF On-Demand Anodyne ADRB3 43 42 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568201 FF On-Demand Anodyne ABCB1 15 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568202 FF On-Demand Anodyne ADRB2 45 48 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568202 FF On-Demand Anodyne ADRB1 61 48 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568202 FF On-Demand Anodyne CYP19A1 18 47 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568202 FF On-Demand Anodyne ADRB3 43 42 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccc(F)cc1 ZINC000880568202 FF On-Demand Anodyne ABCB1 15 40 COC(=O)[C@@]1(O)CCN(CCc2ccc(C#N)cc2)C1 ZINC000880568208 CC On-Demand Mild SLC12A5 19 42 COC(=O)[C@@]1(O)CCN(CCc2ccc(C#N)cc2)C1 ZINC000880568208 CC On-Demand Mild KCNJ1 39 52 COc1ccccc1[C@H](C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568215 GG On-Demand Anodyne CYP19A1 15 45 COc1ccccc1[C@H](C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568215 GG On-Demand Anodyne TBXAS1 34 40 COc1ccccc1[C@H](C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568215 GG On-Demand Anodyne CYP27B1 40 35 COc1ccccc1[C@H](C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568216 GG On-Demand Anodyne CYP19A1 15 45 COc1ccccc1[C@H](C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568216 GG On-Demand Anodyne TBXAS1 34 40 COc1ccccc1[C@H](C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568216 GG On-Demand Anodyne CYP27B1 40 35 COC(=O)[C@@]1(O)CCN(CCCC2CC2)C1 ZINC000880568222 BC On-Demand Anodyne EBP 18 43 COC(=O)[C@@]1(O)CCN(CCCN(C)c2ccccc2)C1 ZINC000880568235 CD On-Demand Anodyne SIGMAR1 15 41 COC(=O)[C@@]1(O)CCN(CCCN(C)c2ccccc2)C1 ZINC000880568235 CD On-Demand Anodyne SLC12A5 52 37 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCC1 ZINC000880568236 DE On-Demand Anodyne TBXAS1 54 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCC1 ZINC000880568237 DE On-Demand Anodyne TBXAS1 54 41 COC(=O)[C@@]1(O)CCN(C[C@H](C)c2ccc(OC)cc2)C1 ZINC000880568297 CD On-Demand Anodyne MMP13 23 40 COC(=O)[C@@]1(O)CCN(C[C@H](C)c2ccc(OC)cc2)C1 ZINC000880568297 CD On-Demand Anodyne MMP9 21 40 COC(=O)[C@@]1(O)CCN(C[C@@H](C)c2ccc(OC)cc2)C1 ZINC000880568299 CD On-Demand Anodyne MMP13 23 40 COC(=O)[C@@]1(O)CCN(C[C@@H](C)c2ccc(OC)cc2)C1 ZINC000880568299 CD On-Demand Anodyne MMP9 21 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568301 EG On-Demand Anodyne CNR1 18 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568301 EG On-Demand Anodyne TBXAS1 50 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568301 EG On-Demand Anodyne CNR2 22 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568301 EG On-Demand Anodyne EPHX2 17 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568302 EG On-Demand Anodyne CNR1 18 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568302 EG On-Demand Anodyne TBXAS1 50 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568302 EG On-Demand Anodyne CNR2 22 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCCC1 ZINC000880568302 EG On-Demand Anodyne EPHX2 17 40 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568309 GE On-Demand Anodyne ACE 19 40 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568309 GE On-Demand Anodyne FKBP1A 83 43 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568309 GE On-Demand Anodyne TBXAS1 23 40 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568310 GE On-Demand Anodyne ACE 19 40 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568310 GE On-Demand Anodyne FKBP1A 83 43 CCOC(=O)[C@@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568310 GE On-Demand Anodyne TBXAS1 23 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCOCC3)c2)C1 ZINC000880568317 EC On-Demand Anodyne SIGMAR1 41 38 COC(=O)[C@@]1(O)CCN(Cc2cccc(CN3CCOCC3)c2)C1 ZINC000880568317 EC On-Demand Anodyne MCHR2 45 35 COC(=O)[C@@]1(O)CCN(Cc2ccnc(C)c2)C1 ZINC000880568321 CC On-Demand Anodyne MCHR2 44 33 COC(=O)[C@@]1(O)CCN(CCCC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880568328 FE On-Demand Anodyne GPR119 27 42 CC(C)(C)OC(=O)N1CSC[C@H]1C(=O)NCc1cn(C2CCC2)nn1 ZINC000880568331 FD On-Demand Anodyne CACNA1B 19 42 COC(=O)[C@@]1(O)CCN(Cc2cccc(OC)c2Cl)C1 ZINC000880568359 CD On-Demand Anodyne CCR8 31 42 O=C(c1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1)N1CCCC1 ZINC000880568367 FH On-Demand Anodyne TBXAS1 45 41 O=C(c1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1)N1CCCC1 ZINC000880568367 FH On-Demand Anodyne CYP27B1 41 36 O=C(c1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1)N1CCCC1 ZINC000880568368 FH On-Demand Anodyne TBXAS1 45 41 O=C(c1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1)N1CCCC1 ZINC000880568368 FH On-Demand Anodyne CYP27B1 41 36 COC(=O)[C@@]1(O)CCN(Cc2ccc(CN3CCOCC3)cc2)C1 ZINC000880568379 EC On-Demand Anodyne MMP13 19 43 O=C(Cc1cc2cc(Cl)ccc2[nH]1)NCc1cn(C2CCC2)nn1 ZINC000880568397 EF On-Demand Anodyne PYGL 72 41 CCOC(=O)C1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568402 GE On-Demand Anodyne TBXAS1 34 42 CCOC(=O)C1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568402 GE On-Demand Anodyne PTAFR 19 41 CCOC(=O)C1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568403 GE On-Demand Anodyne TBXAS1 34 42 CCOC(=O)C1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568403 GE On-Demand Anodyne PTAFR 19 41 CCCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568406 DF On-Demand Anodyne TBXAS1 55 43 CCCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568406 DF On-Demand Anodyne SOAT1 38 40 CCCCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568406 DF On-Demand Anodyne CYP27B1 50 34 CCCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568407 DF On-Demand Anodyne TBXAS1 55 43 CCCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568407 DF On-Demand Anodyne SOAT1 38 40 CCCCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568407 DF On-Demand Anodyne CYP27B1 50 34 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccn3)c2)C1 ZINC000880568421 ED On-Demand Anodyne HRH2 35 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccn3)c2)C1 ZINC000880568421 ED On-Demand Anodyne ADAM17 21 41 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccn3)c2)C1 ZINC000880568421 ED On-Demand Anodyne FAAH 24 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCc3ccccn3)c2)C1 ZINC000880568421 ED On-Demand Anodyne CCR8 31 42 CCCN(CCC)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568437 EF On-Demand Anodyne TBXAS1 51 41 CCCN(CCC)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568438 EF On-Demand Anodyne TBXAS1 51 41 COC(=O)[C@@]1(O)CCN([C@H](C)C(=O)Nc2c(C)cccc2Cl)C1 ZINC000880568447 ED On-Demand Anodyne CXCL8 17 40 COC(=O)[C@@]1(O)CCN([C@@H](C)C(=O)Nc2c(C)cccc2Cl)C1 ZINC000880568449 ED On-Demand Anodyne CXCL8 17 40 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCC(C)C)c2)C1 ZINC000880568460 DD On-Demand Anodyne HRH2 32 45 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCC(C)C)c2)C1 ZINC000880568460 DD On-Demand Anodyne ADAM17 17 44 COC(=O)[C@@]1(O)CCN(Cc2cccc(OCC(C)C)c2)C1 ZINC000880568460 DD On-Demand Anodyne PDS 59 32 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccc(OC)cc3)C2=O)C1 ZINC000880568461 EC On-Demand Anodyne MMP1 21 44 COC(=O)[C@@]1(O)CCN([C@@H]2CCN(Cc3ccc(OC)cc3)C2=O)C1 ZINC000880568461 EC On-Demand Anodyne PROKR1 60 32 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccc(OC)cc3)C2=O)C1 ZINC000880568462 EC On-Demand Anodyne MMP1 21 44 COC(=O)[C@@]1(O)CCN([C@H]2CCN(Cc3ccc(OC)cc3)C2=O)C1 ZINC000880568462 EC On-Demand Anodyne PROKR1 60 32 C#CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568469 CC On-Demand Mild TBXAS1 51 41 C#CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568469 CC On-Demand Mild CYP27B1 41 34 C#CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568470 CC On-Demand Mild TBXAS1 51 41 C#CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568470 CC On-Demand Mild CYP27B1 41 34 C=CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568482 CD On-Demand Mild TBXAS1 46 41 C=CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568482 CD On-Demand Mild CYP24A1 43 36 C=CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568482 CD On-Demand Mild CYP27B1 56 36 C=CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568483 CD On-Demand Mild TBXAS1 46 41 C=CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568483 CD On-Demand Mild CYP24A1 43 36 C=CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568483 CD On-Demand Mild CYP27B1 56 36 c1ccc([C@H](Cn2ccnc2)NC[C@H]2CCCO2)cc1 ZINC000880568484 CE On-Demand Anodyne TNK2 40 33 c1ccc([C@H](Cn2ccnc2)NC[C@@H]2CCCO2)cc1 ZINC000880568485 CE On-Demand Anodyne TNK2 40 33 c1ccc([C@@H](Cn2ccnc2)NC[C@H]2CCCO2)cc1 ZINC000880568486 CE On-Demand Anodyne TNK2 40 33 c1ccc([C@@H](Cn2ccnc2)NC[C@@H]2CCCO2)cc1 ZINC000880568487 CE On-Demand Anodyne TNK2 40 33 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cn(C2CCC2)nn1)C1CCC1 ZINC000880568497 FE On-Demand Anodyne REN 42 37 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne CYP19A1 30 44 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne CYP11B1 45 44 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne TBXAS1 43 44 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne CYP11B2 22 44 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne CYP24A1 45 34 FCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568508 BF On-Demand Anodyne CYP27B1 60 34 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne CYP19A1 30 44 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne CYP11B1 45 44 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne TBXAS1 43 44 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne CYP11B2 22 44 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne CYP24A1 45 34 FCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568509 BF On-Demand Anodyne CYP27B1 60 34 COC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568510 CE On-Demand Anodyne CYP19A1 25 44 COC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568510 CE On-Demand Anodyne TBXAS1 74 45 COC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568510 CE On-Demand Anodyne CYP24A1 54 38 COC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568510 CE On-Demand Anodyne CYP26A1 102 42 COC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568510 CE On-Demand Anodyne CYP27B1 74 38 COC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568511 CE On-Demand Anodyne CYP19A1 25 44 COC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568511 CE On-Demand Anodyne TBXAS1 74 45 COC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568511 CE On-Demand Anodyne CYP24A1 54 38 COC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568511 CE On-Demand Anodyne CYP26A1 102 42 COC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568511 CE On-Demand Anodyne CYP27B1 74 38 CCSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568518 CF On-Demand Anodyne CYP19A1 15 40 CCSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568518 CF On-Demand Anodyne CYP11B1 35 40 CCSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568518 CF On-Demand Anodyne TBXAS1 24 40 CCSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568518 CF On-Demand Anodyne CYP11B2 19 40 CCSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568519 CF On-Demand Anodyne CYP19A1 15 40 CCSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568519 CF On-Demand Anodyne CYP11B1 35 40 CCSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568519 CF On-Demand Anodyne TBXAS1 24 40 CCSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568519 CF On-Demand Anodyne CYP11B2 19 40 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568522 EF On-Demand Anodyne TBXAS1 57 41 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568522 EF On-Demand Anodyne PTAFR 24 45 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568522 EF On-Demand Anodyne CYP24A1 43 36 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568522 EF On-Demand Anodyne CYP26A1 57 35 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568522 EF On-Demand Anodyne CYP27B1 56 36 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568523 EF On-Demand Anodyne TBXAS1 57 41 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568523 EF On-Demand Anodyne PTAFR 24 45 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568523 EF On-Demand Anodyne CYP24A1 43 36 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568523 EF On-Demand Anodyne CYP26A1 57 35 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880568523 EF On-Demand Anodyne CYP27B1 56 36 COC(=O)CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568526 EC On-Demand Anodyne TBXAS1 56 40 COC(=O)CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568526 EC On-Demand Anodyne CYP26A1 85 39 COC(=O)CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568526 EC On-Demand Anodyne CYP27B1 44 38 COC(=O)CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568527 EC On-Demand Anodyne TBXAS1 56 40 COC(=O)CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568527 EC On-Demand Anodyne CYP26A1 85 39 COC(=O)CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568527 EC On-Demand Anodyne CYP27B1 44 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568537 ED On-Demand Anodyne TBXAS1 51 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568537 ED On-Demand Anodyne CYP24A1 44 36 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568537 ED On-Demand Anodyne CYP27B1 57 36 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568538 ED On-Demand Anodyne TBXAS1 51 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568538 ED On-Demand Anodyne CYP24A1 44 36 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC(F)(F)F ZINC000880568538 ED On-Demand Anodyne CYP27B1 57 36 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880568557 GF On-Demand Anodyne PREP 15 48 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880568557 GF On-Demand Anodyne GPR119 40 37 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880568558 GF On-Demand Anodyne PREP 15 48 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cn(C3CCC3)nn2)CC1 ZINC000880568558 GF On-Demand Anodyne GPR119 40 37 CCCCNC(=O)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568559 ED On-Demand Anodyne TBXAS1 43 41 CCCCNC(=O)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568560 ED On-Demand Anodyne TBXAS1 43 41 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP19A1 31 53 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP11B1 52 45 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne TBXAS1 29 51 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne HTR7 16 40 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP11B2 28 41 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne HMOX1 41 42 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne HMOX2 26 41 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP24A1 43 42 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP26A1 96 38 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne QPCT 24 42 COc1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568563 EG On-Demand Anodyne CYP27B1 62 42 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP19A1 31 53 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP11B1 52 45 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne TBXAS1 29 51 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne HTR7 16 40 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP11B2 28 41 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne HMOX1 41 42 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne HMOX2 26 41 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP24A1 43 42 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP26A1 96 38 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne QPCT 24 42 COc1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568564 EG On-Demand Anodyne CYP27B1 62 42 CC(C)(C(=O)NCc1cn(C2CCC2)nn1)[C@@H](O)c1cc(Cl)cc(Cl)c1 ZINC000880568567 GH On-Demand Anodyne CACNA1I 40 34 CC(C)(C(=O)NCc1cn(C2CCC2)nn1)[C@H](O)c1cc(Cl)cc(Cl)c1 ZINC000880568568 GH On-Demand Anodyne CACNA1I 40 34 CCCn1nccc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568571 FE On-Demand Anodyne TBXAS1 35 41 CCCn1nccc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568572 FE On-Demand Anodyne TBXAS1 35 41 C[C@H](CCc1ccc(F)cc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880568582 EG On-Demand Anodyne CCR3 71 33 C[C@@H](CCc1ccc(F)cc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880568583 EG On-Demand Anodyne CCR3 71 33 FCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568585 BE On-Demand Anodyne CYP19A1 32 44 FCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568585 BE On-Demand Anodyne CYP11B1 45 44 FCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568585 BE On-Demand Anodyne TBXAS1 34 44 FCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568585 BE On-Demand Anodyne CYP11B2 22 44 FCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568585 BE On-Demand Anodyne CYP27B1 50 32 FCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568586 BE On-Demand Anodyne CYP19A1 32 44 FCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568586 BE On-Demand Anodyne CYP11B1 45 44 FCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568586 BE On-Demand Anodyne TBXAS1 34 44 FCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568586 BE On-Demand Anodyne CYP11B2 22 44 FCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568586 BE On-Demand Anodyne CYP27B1 50 32 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP19A1 28 43 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP11B1 43 44 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne TBXAS1 60 52 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP11B2 21 44 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne HMOX1 37 43 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP17A1 16 40 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne HMOX2 53 43 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP24A1 48 40 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne QPCT 45 43 c1ccc([C@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568624 CF On-Demand Anodyne CYP27B1 65 40 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP19A1 28 43 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP11B1 43 44 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne TBXAS1 60 52 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP11B2 21 44 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne HMOX1 37 43 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP17A1 16 40 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne HMOX2 53 43 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP24A1 48 40 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne QPCT 45 43 c1ccc([C@@H](Cn2ccnc2)NCCCn2ccnc2)cc1 ZINC000880568625 CF On-Demand Anodyne CYP27B1 65 40 O[C@@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568631 EG On-Demand Anodyne CYP11B1 31 43 O[C@@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568631 EG On-Demand Anodyne TBXAS1 29 43 O[C@@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568631 EG On-Demand Anodyne CYP11B2 15 43 O[C@@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568631 EG On-Demand Anodyne HMOX1 41 53 O[C@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568632 EG On-Demand Anodyne CYP11B1 31 43 O[C@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568632 EG On-Demand Anodyne TBXAS1 29 43 O[C@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568632 EG On-Demand Anodyne CYP11B2 15 43 O[C@H](CCc1ccccc1)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568632 EG On-Demand Anodyne HMOX1 41 53 O[C@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568633 EG On-Demand Anodyne CYP11B1 31 43 O[C@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568633 EG On-Demand Anodyne TBXAS1 29 43 O[C@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568633 EG On-Demand Anodyne CYP11B2 15 43 O[C@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568633 EG On-Demand Anodyne HMOX1 41 53 O[C@@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568634 EG On-Demand Anodyne CYP11B1 31 43 O[C@@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568634 EG On-Demand Anodyne TBXAS1 29 43 O[C@@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568634 EG On-Demand Anodyne CYP11B2 15 43 O[C@@H](CCc1ccccc1)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568634 EG On-Demand Anodyne HMOX1 41 53 CCCOc1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880568636 EI On-Demand Anodyne TBXAS1 22 44 CCCOc1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880568636 EI On-Demand Anodyne HMOX2 17 40 CCCOc1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880568637 EI On-Demand Anodyne TBXAS1 22 44 CCCOc1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880568637 EI On-Demand Anodyne HMOX2 17 40 CC(C)(C)OC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568654 FD On-Demand Anodyne TBXAS1 44 39 CC(C)(C)OC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568654 FD On-Demand Anodyne CYP24A1 42 37 CC(C)(C)OC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568654 FD On-Demand Anodyne CYP26A1 67 36 CC(C)(C)OC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568654 FD On-Demand Anodyne CYP27B1 54 37 CC(C)(C)OC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568655 FD On-Demand Anodyne TBXAS1 44 39 CC(C)(C)OC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568655 FD On-Demand Anodyne CYP24A1 42 37 CC(C)(C)OC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568655 FD On-Demand Anodyne CYP26A1 67 36 CC(C)(C)OC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568655 FD On-Demand Anodyne CYP27B1 54 37 CN(C)[S@](C)(=O)=NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568656 ED On-Demand Anodyne TBXAS1 37 42 CN(C)[S@](C)(=O)=NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568659 ED On-Demand Anodyne TBXAS1 37 42 CC(C)(C)C(=O)NNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568666 ED On-Demand Reactive TBXAS1 48 41 CC(C)(C)C(=O)NNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568666 ED On-Demand Reactive CYP26A1 50 37 CC(C)(C)C(=O)NNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568666 ED On-Demand Reactive CYP27B1 47 36 CC(C)(C)C(=O)NNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568667 ED On-Demand Reactive TBXAS1 48 41 CC(C)(C)C(=O)NNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568667 ED On-Demand Reactive CYP26A1 50 37 CC(C)(C)C(=O)NNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568667 ED On-Demand Reactive CYP27B1 47 36 c1ccc([C@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568677 CE On-Demand Anodyne CYP19A1 23 43 c1ccc([C@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568677 CE On-Demand Anodyne CYP11B1 46 43 c1ccc([C@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568677 CE On-Demand Anodyne TBXAS1 37 43 c1ccc([C@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568677 CE On-Demand Anodyne CYP11B2 22 43 c1ccc([C@@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568678 CE On-Demand Anodyne CYP19A1 23 43 c1ccc([C@@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568678 CE On-Demand Anodyne CYP11B1 46 43 c1ccc([C@@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568678 CE On-Demand Anodyne TBXAS1 37 43 c1ccc([C@@H](Cn2ccnc2)NCCn2cccn2)cc1 ZINC000880568678 CE On-Demand Anodyne CYP11B2 22 43 CCOCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568688 DD On-Demand Anodyne TBXAS1 46 39 CCOCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568689 DD On-Demand Anodyne TBXAS1 46 39 COc1ccccc1[C@H](C)N(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568702 GG On-Demand Anodyne CYP26A1 69 36 COc1ccccc1[C@H](C)N(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568704 GG On-Demand Anodyne CYP26A1 69 36 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP19A1 22 40 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP11B1 32 40 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne TBXAS1 67 46 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP11B2 16 40 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP24A1 50 36 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP26A1 62 40 CCOC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568730 CD On-Demand Anodyne CYP27B1 67 36 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP19A1 22 40 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP11B1 32 40 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne TBXAS1 67 46 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP11B2 16 40 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP24A1 50 36 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP26A1 62 40 CCOC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568731 CD On-Demand Anodyne CYP27B1 67 36 N#CCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568732 CD On-Demand Mild TBXAS1 49 41 N#CCCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568732 CD On-Demand Mild CYP27B1 46 34 N#CCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568733 CD On-Demand Mild TBXAS1 49 41 N#CCCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568733 CD On-Demand Mild CYP27B1 46 34 C[C@@H]1Cc2cc(C(=O)NCc3cn(C4CCC4)nn3)ccc2O1 ZINC000880568736 DE On-Demand Anodyne CA14 16 42 C[C@H]1Cc2cc(C(=O)NCc3cn(C4CCC4)nn3)ccc2O1 ZINC000880568737 DE On-Demand Anodyne CA14 16 42 O=C(NCc1cn(C2CCC2)nn1)c1cccc(SC(F)(F)F)c1 ZINC000880568740 FH On-Demand Anodyne CCR2 43 37 CCOC(=O)CN(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568741 ED On-Demand Anodyne TBXAS1 46 41 CCOC(=O)CN(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568741 ED On-Demand Anodyne CYP27B1 41 34 CCOC(=O)CN(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568742 ED On-Demand Anodyne TBXAS1 46 41 CCOC(=O)CN(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568742 ED On-Demand Anodyne CYP27B1 41 34 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne CYP19A1 22 42 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne CYP11B1 39 42 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne TBXAS1 39 45 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne CYP11B2 19 42 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne SOAT1 24 41 CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568747 CG On-Demand Anodyne CYP17A1 17 42 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne CYP19A1 22 42 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne CYP11B1 39 42 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne TBXAS1 39 45 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne CYP11B2 19 42 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne SOAT1 24 41 CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568748 CG On-Demand Anodyne CYP17A1 17 42 CCCCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568750 DF On-Demand Anodyne TBXAS1 58 43 CCCCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568750 DF On-Demand Anodyne CYP24A1 41 36 CCCCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568750 DF On-Demand Anodyne CYP26A1 40 37 CCCCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568750 DF On-Demand Anodyne CYP27B1 52 36 CCCCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568751 DF On-Demand Anodyne TBXAS1 58 43 CCCCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568751 DF On-Demand Anodyne CYP24A1 41 36 CCCCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568751 DF On-Demand Anodyne CYP26A1 40 37 CCCCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568751 DF On-Demand Anodyne CYP27B1 52 36 c1ccc([C@@H](Cn2ccnc2)NCCCN2CCOCC2)cc1 ZINC000880568756 DD On-Demand Anodyne CASR 45 37 c1ccc([C@H](Cn2ccnc2)NCCCN2CCOCC2)cc1 ZINC000880568757 DD On-Demand Anodyne CASR 45 37 CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568758 CD On-Demand Anodyne CYP19A1 21 41 CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568758 CD On-Demand Anodyne TBXAS1 67 44 CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568758 CD On-Demand Anodyne CYP24A1 49 39 CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568758 CD On-Demand Anodyne CYP26A1 71 40 CNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568758 CD On-Demand Anodyne CYP27B1 66 39 CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568759 CD On-Demand Anodyne CYP19A1 21 41 CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568759 CD On-Demand Anodyne TBXAS1 67 44 CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568759 CD On-Demand Anodyne CYP24A1 49 39 CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568759 CD On-Demand Anodyne CYP26A1 71 40 CNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568759 CD On-Demand Anodyne CYP27B1 66 39 NS(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568761 DC On-Demand Anodyne TBXAS1 39 41 NS(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568761 DC On-Demand Anodyne CYP24A1 40 31 NS(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568761 DC On-Demand Anodyne CYP27B1 52 30 NS(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568762 DC On-Demand Anodyne TBXAS1 39 41 NS(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568762 DC On-Demand Anodyne CYP24A1 40 31 NS(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568762 DC On-Demand Anodyne CYP27B1 52 30 CC(C)(C)OC(=O)N1CC(CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568776 FG On-Demand Anodyne CYP26A1 43 34 CC(C)(C)OC(=O)N1CC(CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568776 FG On-Demand Anodyne CYP27B1 40 33 CC(C)(C)OC(=O)N1CC(CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568777 FG On-Demand Anodyne CYP26A1 43 34 CC(C)(C)OC(=O)N1CC(CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880568777 FG On-Demand Anodyne CYP27B1 40 33 C#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568786 BE On-Demand Mild CYP19A1 19 41 C#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568786 BE On-Demand Mild CYP11B1 37 41 C#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568786 BE On-Demand Mild TBXAS1 25 41 C#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568786 BE On-Demand Mild CYP11B2 18 41 C#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568787 BE On-Demand Mild CYP19A1 19 41 C#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568787 BE On-Demand Mild CYP11B1 37 41 C#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568787 BE On-Demand Mild TBXAS1 25 41 C#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568787 BE On-Demand Mild CYP11B2 18 41 ICCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568792 FG On-Demand Reactive CYP19A1 23 42 ICCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568792 FG On-Demand Reactive CYP11B1 39 42 ICCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568792 FG On-Demand Reactive TBXAS1 34 42 ICCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568792 FG On-Demand Reactive CYP11B2 19 42 ICCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568793 FG On-Demand Reactive CYP19A1 23 42 ICCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568793 FG On-Demand Reactive CYP11B1 39 42 ICCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568793 FG On-Demand Reactive TBXAS1 34 42 ICCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568793 FG On-Demand Reactive CYP11B2 19 42 CCOC(=O)c1c(CN[C@@H](Cn2ccnc2)c2ccccc2)n[nH]c1C ZINC000880568794 FF On-Demand Anodyne TBXAS1 32 40 CCOC(=O)c1c(CN[C@H](Cn2ccnc2)c2ccccc2)n[nH]c1C ZINC000880568795 FF On-Demand Anodyne TBXAS1 32 40 CN(C[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568802 FE On-Demand Anodyne CYP26A1 51 34 CN(C[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568802 FE On-Demand Anodyne CYP27B1 42 35 CN(C[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568803 FE On-Demand Anodyne CYP26A1 51 34 CN(C[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568803 FE On-Demand Anodyne CYP27B1 42 35 CN(C[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568804 FE On-Demand Anodyne CYP26A1 51 34 CN(C[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568804 FE On-Demand Anodyne CYP27B1 42 35 CN(C[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568805 FE On-Demand Anodyne CYP26A1 51 34 CN(C[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)OC(C)(C)C ZINC000880568805 FE On-Demand Anodyne CYP27B1 42 35 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP19A1 19 41 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP11B1 36 41 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne TBXAS1 43 42 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP11B2 18 41 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP24A1 49 38 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP26A1 51 36 CC(C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568816 CD On-Demand Anodyne CYP27B1 66 38 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP19A1 19 41 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP11B1 36 41 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne TBXAS1 43 42 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP11B2 18 41 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP24A1 49 38 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP26A1 51 36 CC(C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568817 CD On-Demand Anodyne CYP27B1 66 38 COC(=O)C1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568834 CE On-Demand Anodyne CYP19A1 22 45 COC(=O)C1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568834 CE On-Demand Anodyne TBXAS1 56 41 COC(=O)C1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568834 CE On-Demand Anodyne CYP26A1 107 40 COC(=O)C1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568834 CE On-Demand Anodyne CYP27B1 47 38 COC(=O)C1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568835 CE On-Demand Anodyne CYP19A1 22 45 COC(=O)C1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568835 CE On-Demand Anodyne TBXAS1 56 41 COC(=O)C1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568835 CE On-Demand Anodyne CYP26A1 107 40 COC(=O)C1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568835 CE On-Demand Anodyne CYP27B1 47 38 CSc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568836 GG On-Demand Anodyne ADRB2 33 47 CSc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568836 GG On-Demand Anodyne ADRB1 44 47 CSc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568837 GG On-Demand Anodyne ADRB2 33 47 CSc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568837 GG On-Demand Anodyne ADRB1 44 47 CSc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568838 GG On-Demand Anodyne ADRB2 33 47 CSc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568838 GG On-Demand Anodyne ADRB1 44 47 CSc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568839 GG On-Demand Anodyne ADRB2 33 47 CSc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568839 GG On-Demand Anodyne ADRB1 44 47 O=C(Cc1ccc2cccnc2c1)NCc1cn(C2CCC2)nn1 ZINC000880568840 DE On-Demand Anodyne CDK5 26 43 O=C(Cc1ccc2cccnc2c1)NCc1cn(C2CCC2)nn1 ZINC000880568840 DE On-Demand Anodyne SUCNR1 52 37 c1ccc([C@@H](Cn2ccnc2)NCc2cccc(CN3CCOCC3)c2)cc1 ZINC000880568859 GG On-Demand Anodyne CYP11B1 30 41 c1ccc([C@@H](Cn2ccnc2)NCc2cccc(CN3CCOCC3)c2)cc1 ZINC000880568859 GG On-Demand Anodyne CYP11B2 16 41 c1ccc([C@H](Cn2ccnc2)NCc2cccc(CN3CCOCC3)c2)cc1 ZINC000880568860 GG On-Demand Anodyne CYP11B1 30 41 c1ccc([C@H](Cn2ccnc2)NCc2cccc(CN3CCOCC3)c2)cc1 ZINC000880568860 GG On-Demand Anodyne CYP11B2 16 41 Cn1cncc1CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568867 DF On-Demand Anodyne TBXAS1 22 40 Cn1cncc1CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568868 DF On-Demand Anodyne TBXAS1 22 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)Nc1ccc(N2CCCC2)cc1 ZINC000880568889 GG On-Demand Anodyne KCNQ2 42 50 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)Nc1ccc(N2CCCC2)cc1 ZINC000880568890 GG On-Demand Anodyne KCNQ2 42 50 CC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568914 CD On-Demand Anodyne TBXAS1 67 46 CC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568914 CD On-Demand Anodyne CYP24A1 48 36 CC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568914 CD On-Demand Anodyne CYP27B1 63 36 CC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568915 CD On-Demand Anodyne TBXAS1 67 46 CC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568915 CD On-Demand Anodyne CYP24A1 48 36 CC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568915 CD On-Demand Anodyne CYP27B1 63 36 N#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568920 BE On-Demand Mild CYP19A1 24 43 N#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568920 BE On-Demand Mild CYP11B1 41 42 N#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568920 BE On-Demand Mild TBXAS1 29 42 N#CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568920 BE On-Demand Mild CYP11B2 20 42 N#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568921 BE On-Demand Mild CYP19A1 24 43 N#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568921 BE On-Demand Mild CYP11B1 41 42 N#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568921 BE On-Demand Mild TBXAS1 29 42 N#CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568921 BE On-Demand Mild CYP11B2 20 42 O=C(c1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568922 GI On-Demand Anodyne TBXAS1 42 37 O=C(c1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568922 GI On-Demand Anodyne DPP7 40 35 O=C(c1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568922 GI On-Demand Anodyne CYP27B1 48 31 O=C(c1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568923 GI On-Demand Anodyne TBXAS1 42 37 O=C(c1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568923 GI On-Demand Anodyne DPP7 40 35 O=C(c1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1)N1CCCCC1 ZINC000880568923 GI On-Demand Anodyne CYP27B1 48 31 N#CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568934 CF On-Demand Mild CYP19A1 15 40 N#CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568934 CF On-Demand Mild TBXAS1 26 40 N#CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568935 CF On-Demand Mild CYP19A1 15 40 N#CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568935 CF On-Demand Mild TBXAS1 26 40 COC(=O)CN(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568936 ED On-Demand Anodyne TBXAS1 50 39 COC(=O)CN(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568936 ED On-Demand Anodyne CYP26A1 101 38 COC(=O)CN(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568937 ED On-Demand Anodyne TBXAS1 50 39 COC(=O)CN(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568937 ED On-Demand Anodyne CYP26A1 101 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568949 EF On-Demand Anodyne CNR1 18 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568949 EF On-Demand Anodyne TBXAS1 50 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568949 EF On-Demand Anodyne CNR2 22 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568949 EF On-Demand Anodyne EPHX2 17 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568950 EF On-Demand Anodyne CNR1 18 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568950 EF On-Demand Anodyne TBXAS1 50 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568950 EF On-Demand Anodyne CNR2 22 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCCC1 ZINC000880568950 EF On-Demand Anodyne EPHX2 17 40 CCOC(=O)N1CCC(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568951 GD On-Demand Anodyne P2RY12 71 39 CCOC(=O)N1CCC(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568951 GD On-Demand Anodyne TBXAS1 34 40 CCOC(=O)N1CCC(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568951 GD On-Demand Anodyne CCR8 25 40 CCOC(=O)N1CCC(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568952 GD On-Demand Anodyne P2RY12 71 39 CCOC(=O)N1CCC(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568952 GD On-Demand Anodyne TBXAS1 34 40 CCOC(=O)N1CCC(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880568952 GD On-Demand Anodyne CCR8 25 40 C[C@@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568955 EC On-Demand Anodyne TBXAS1 46 41 C[C@@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568955 EC On-Demand Anodyne CYP26A1 54 33 C[C@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568956 EC On-Demand Anodyne TBXAS1 46 41 C[C@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568956 EC On-Demand Anodyne CYP26A1 54 33 C[C@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568957 EC On-Demand Anodyne TBXAS1 46 41 C[C@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568957 EC On-Demand Anodyne CYP26A1 54 33 C[C@@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568958 EC On-Demand Anodyne TBXAS1 46 41 C[C@@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N(C)C ZINC000880568958 EC On-Demand Anodyne CYP26A1 54 33 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC1(c2ccccc2)CC1 ZINC000880568960 FG On-Demand Anodyne NPFFR1 24 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC1(c2ccccc2)CC1 ZINC000880568961 FG On-Demand Anodyne NPFFR1 24 40 CCOC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568962 CE On-Demand Anodyne TBXAS1 67 45 CCOC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568962 CE On-Demand Anodyne CYP24A1 48 37 CCOC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568962 CE On-Demand Anodyne CYP26A1 82 39 CCOC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568962 CE On-Demand Anodyne CYP27B1 64 37 CCOC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568963 CE On-Demand Anodyne TBXAS1 67 45 CCOC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568963 CE On-Demand Anodyne CYP24A1 48 37 CCOC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568963 CE On-Demand Anodyne CYP26A1 82 39 CCOC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568963 CE On-Demand Anodyne CYP27B1 64 37 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne CYP19A1 30 44 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne CYP11B1 47 44 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne TBXAS1 52 44 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne CYP11B2 24 44 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne CYP24A1 42 33 OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568966 BD On-Demand Anodyne CYP27B1 55 33 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne CYP19A1 30 44 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne CYP11B1 47 44 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne TBXAS1 52 44 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne CYP11B2 24 44 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne CYP24A1 42 33 OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568967 BD On-Demand Anodyne CYP27B1 55 33 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne CYP19A1 18 46 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne TBXAS1 38 46 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne BMP1 50 36 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne MMP12 16 40 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne CYP24A1 32 40 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne CYP26A1 95 37 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne QPCT 23 40 COc1ccc(CN(C)C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568973 GF On-Demand Anodyne CYP27B1 46 40 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne CYP19A1 18 46 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne TBXAS1 38 46 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne BMP1 50 36 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne MMP12 16 40 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne CYP24A1 32 40 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne CYP26A1 95 37 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne QPCT 23 40 COc1ccc(CN(C)C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880568974 GF On-Demand Anodyne CYP27B1 46 40 CC(C)(C)NC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568983 FD On-Demand Anodyne TBXAS1 42 40 CC(C)(C)NC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568983 FD On-Demand Anodyne CYP26A1 42 37 CC(C)(C)NC(=O)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568983 FD On-Demand Anodyne CYP27B1 47 35 CC(C)(C)NC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568984 FD On-Demand Anodyne TBXAS1 42 40 CC(C)(C)NC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568984 FD On-Demand Anodyne CYP26A1 42 37 CC(C)(C)NC(=O)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568984 FD On-Demand Anodyne CYP27B1 47 35 C=CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568994 CH On-Demand Mild CYP11B1 36 41 C=CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568994 CH On-Demand Mild TBXAS1 30 41 C=CCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880568994 CH On-Demand Mild CYP11B2 18 41 C=CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568995 CH On-Demand Mild CYP11B1 36 41 C=CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568995 CH On-Demand Mild TBXAS1 30 41 C=CCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880568995 CH On-Demand Mild CYP11B2 18 41 c1ccc(COCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569003 EH On-Demand Anodyne CYP11B1 34 43 c1ccc(COCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569003 EH On-Demand Anodyne TBXAS1 32 43 c1ccc(COCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569003 EH On-Demand Anodyne CYP11B2 18 43 c1ccc(COCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569003 EH On-Demand Anodyne QPCT 18 41 c1ccc(COCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569004 EH On-Demand Anodyne CYP11B1 34 43 c1ccc(COCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569004 EH On-Demand Anodyne TBXAS1 32 43 c1ccc(COCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569004 EH On-Demand Anodyne CYP11B2 18 43 c1ccc(COCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569004 EH On-Demand Anodyne QPCT 18 41 c1ccc([C@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569040 DG On-Demand Anodyne TBXAS1 26 40 c1ccc([C@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569040 DG On-Demand Anodyne HRH3 22 40 c1ccc([C@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569040 DG On-Demand Anodyne HNMT 93 40 c1ccc([C@@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569041 DG On-Demand Anodyne TBXAS1 26 40 c1ccc([C@@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569041 DG On-Demand Anodyne HRH3 22 40 c1ccc([C@@H](Cn2ccnc2)NCCCN2CCCCC2)cc1 ZINC000880569041 DG On-Demand Anodyne HNMT 93 40 CCc1nnc(CN[C@@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569055 DF On-Demand Anodyne CYP11B1 21 40 CCc1nnc(CN[C@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569056 DF On-Demand Anodyne CYP11B1 21 40 c1ccc(COCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569063 DG On-Demand Anodyne CYP19A1 20 45 c1ccc(COCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569063 DG On-Demand Anodyne CYP11B1 46 45 c1ccc(COCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569063 DG On-Demand Anodyne TBXAS1 34 45 c1ccc(COCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569063 DG On-Demand Anodyne CYP11B2 24 45 c1ccc(COCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569063 DG On-Demand Anodyne QPCT 15 40 c1ccc(COCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569064 DG On-Demand Anodyne CYP19A1 20 45 c1ccc(COCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569064 DG On-Demand Anodyne CYP11B1 46 45 c1ccc(COCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569064 DG On-Demand Anodyne TBXAS1 34 45 c1ccc(COCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569064 DG On-Demand Anodyne CYP11B2 24 45 c1ccc(COCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569064 DG On-Demand Anodyne QPCT 15 40 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569084 GF On-Demand Anodyne TNF 31 44 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569084 GF On-Demand Anodyne TBXAS1 51 39 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569084 GF On-Demand Anodyne MAPK14 28 44 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569084 GF On-Demand Anodyne CTSV 40 31 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569085 GF On-Demand Anodyne TNF 31 44 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569085 GF On-Demand Anodyne TBXAS1 51 39 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569085 GF On-Demand Anodyne MAPK14 28 44 Cn1nc(C(C)(C)C)cc1NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569085 GF On-Demand Anodyne CTSV 40 31 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569086 EF On-Demand Anodyne CYP19A1 17 44 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569086 EF On-Demand Anodyne CYP11B1 32 44 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569086 EF On-Demand Anodyne HMOX1 29 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569086 EF On-Demand Anodyne CYP24A1 21 42 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569086 EF On-Demand Anodyne CYP27B1 28 42 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569088 EF On-Demand Anodyne CYP19A1 17 44 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569088 EF On-Demand Anodyne CYP11B1 32 44 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569088 EF On-Demand Anodyne HMOX1 29 40 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569088 EF On-Demand Anodyne CYP24A1 21 42 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569088 EF On-Demand Anodyne CYP27B1 28 42 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569090 EF On-Demand Anodyne CYP19A1 17 44 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569090 EF On-Demand Anodyne CYP11B1 32 44 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569090 EF On-Demand Anodyne HMOX1 29 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569090 EF On-Demand Anodyne CYP24A1 21 42 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569090 EF On-Demand Anodyne CYP27B1 28 42 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569091 EF On-Demand Anodyne CYP19A1 17 44 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569091 EF On-Demand Anodyne CYP11B1 32 44 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569091 EF On-Demand Anodyne HMOX1 29 40 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569091 EF On-Demand Anodyne CYP24A1 21 42 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccc(F)cc1 ZINC000880569091 EF On-Demand Anodyne CYP27B1 28 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)Nc1nc2c(s1)CCCC2 ZINC000880569094 GG On-Demand Anodyne SLC27A1 37 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)Nc1nc2c(s1)CCCC2 ZINC000880569096 GG On-Demand Anodyne SLC27A1 37 41 O=C(NCCCN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569098 EE On-Demand Anodyne TBXAS1 59 43 O=C(NCCCN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569098 EE On-Demand Anodyne CYP24A1 42 34 O=C(NCCCN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569098 EE On-Demand Anodyne CYP27B1 56 34 Cc1sc(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)c(C)c1C ZINC000880569099 FH On-Demand Anodyne TBXAS1 42 41 O=C(NCCCN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569100 EE On-Demand Anodyne TBXAS1 59 43 O=C(NCCCN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569100 EE On-Demand Anodyne CYP24A1 42 34 O=C(NCCCN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569100 EE On-Demand Anodyne CYP27B1 56 34 CCOc1ccccc1NC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569102 GH On-Demand Anodyne TBXAS1 37 40 CCOc1ccccc1NC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569102 GH On-Demand Anodyne CYP26A1 54 37 Cc1sc(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)c(C)c1C ZINC000880569103 FH On-Demand Anodyne TBXAS1 42 41 CCOc1ccccc1NC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569104 GH On-Demand Anodyne TBXAS1 37 40 CCOc1ccccc1NC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569104 GH On-Demand Anodyne CYP26A1 54 37 c1ccc([C@@H](Cn2ccnc2)NCc2ccc3c(c2)OCCO3)cc1 ZINC000880569116 EG On-Demand Anodyne CYP19A1 16 45 c1ccc([C@@H](Cn2ccnc2)NCc2ccc3c(c2)OCCO3)cc1 ZINC000880569116 EG On-Demand Anodyne NOS2 96 35 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569122 GH On-Demand Anodyne TBXAS1 34 40 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569122 GH On-Demand Anodyne CYP26A1 94 38 c1ccc([C@H](Cn2ccnc2)NCc2ccc3c(c2)OCCO3)cc1 ZINC000880569123 EG On-Demand Anodyne CYP19A1 16 45 c1ccc([C@H](Cn2ccnc2)NCc2ccc3c(c2)OCCO3)cc1 ZINC000880569123 EG On-Demand Anodyne NOS2 96 35 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569126 GH On-Demand Anodyne TBXAS1 34 40 C[C@@H](c1ccc(F)cc1)N(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569126 GH On-Demand Anodyne CYP26A1 94 38 CCOc1cc(CN[C@H](Cn2ccnc2)c2ccccc2)ccc1[N+](=O)[O-] ZINC000880569130 FH On-Demand Bother CYP19A1 16 43 CCOc1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)ccc1[N+](=O)[O-] ZINC000880569131 FH On-Demand Bother CYP19A1 16 43 CC[C@@H](Nc1cccnc1Cl)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880569138 EF On-Demand Anodyne G2YM83_BOTF4 58 33 CC[C@H](Nc1cccnc1Cl)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880569139 EF On-Demand Anodyne G2YM83_BOTF4 58 33 NC(=S)c1ccc(C(=O)NCc2cn(C3CCC3)nn2)cc1 ZINC000880569151 DD On-Demand Anodyne CA14 22 52 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880569152 GG On-Demand Anodyne CYP11B1 38 41 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880569152 GG On-Demand Anodyne CYP11B2 18 41 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne ADRB2 50 55 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne ADRB1 79 55 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne ADRB3 63 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne TBXAS1 29 43 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne ABCB1 17 45 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne CYP26A1 84 34 CC(=O)Nc1ccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569153 GF On-Demand Anodyne QPCT 24 41 c1ccc([C@H](Cn2ccnc2)NCc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880569154 GG On-Demand Anodyne CYP11B1 38 41 c1ccc([C@H](Cn2ccnc2)NCc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880569154 GG On-Demand Anodyne CYP11B2 18 41 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne ADRB2 50 55 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne ADRB1 79 55 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne ADRB3 63 46 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne TBXAS1 29 43 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne ABCB1 17 45 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne CYP26A1 84 34 CC(=O)Nc1ccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569155 GF On-Demand Anodyne QPCT 24 41 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne ADRB2 50 55 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne ADRB1 79 55 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne ADRB3 63 46 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne TBXAS1 29 43 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne ABCB1 17 45 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne CYP26A1 84 34 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569157 GF On-Demand Anodyne QPCT 24 41 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne ADRB2 50 55 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne ADRB1 79 55 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne ADRB3 63 46 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne TBXAS1 29 43 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne ABCB1 17 45 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne CYP26A1 84 34 CC(=O)Nc1ccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880569159 GF On-Demand Anodyne QPCT 24 41 FC(F)COCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569160 CE On-Demand Anodyne TBXAS1 26 41 FC(F)COCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569161 CE On-Demand Anodyne TBXAS1 26 41 CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569165 CC On-Demand Anodyne CYP19A1 23 42 CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569165 CC On-Demand Anodyne TBXAS1 64 45 CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569165 CC On-Demand Anodyne CYP24A1 43 35 CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569165 CC On-Demand Anodyne CYP26A1 41 38 CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569165 CC On-Demand Anodyne CYP27B1 56 35 CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569167 CC On-Demand Anodyne CYP19A1 23 42 CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569167 CC On-Demand Anodyne TBXAS1 64 45 CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569167 CC On-Demand Anodyne CYP24A1 43 35 CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569167 CC On-Demand Anodyne CYP26A1 41 38 CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569167 CC On-Demand Anodyne CYP27B1 56 35 CCOC(=O)c1nc(CN[C@@H](Cn2ccnc2)c2ccccc2)cs1 ZINC000880569173 FG On-Demand Anodyne TBXAS1 33 40 CCOC(=O)c1nc(CN[C@H](Cn2ccnc2)c2ccccc2)cs1 ZINC000880569176 FG On-Demand Anodyne TBXAS1 33 40 COCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569178 CG On-Demand Anodyne TBXAS1 40 42 COCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569178 CG On-Demand Anodyne CYP24A1 44 33 COCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569178 CG On-Demand Anodyne CYP27B1 59 33 COCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569180 CG On-Demand Anodyne TBXAS1 40 42 COCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569180 CG On-Demand Anodyne CYP24A1 44 33 COCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569180 CG On-Demand Anodyne CYP27B1 59 33 O=[N+]([O-])c1cnn(CCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569182 EE On-Demand Bother CYP19A1 17 42 O=[N+]([O-])c1cnn(CCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569184 EE On-Demand Bother CYP19A1 17 42 C[S@@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569185 CD On-Demand Anodyne CYP19A1 20 40 C[S@@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569185 CD On-Demand Anodyne CYP11B1 39 40 C[S@@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569185 CD On-Demand Anodyne TBXAS1 38 41 C[S@@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569185 CD On-Demand Anodyne CYP11B2 21 40 C[S@@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569185 CD On-Demand Anodyne CYP27B1 47 31 N#CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569186 CC On-Demand Mild TBXAS1 53 41 N#CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569186 CC On-Demand Mild CYP27B1 42 35 C[S@@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569187 CD On-Demand Anodyne CYP19A1 20 40 C[S@@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569187 CD On-Demand Anodyne CYP11B1 39 40 C[S@@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569187 CD On-Demand Anodyne TBXAS1 38 41 C[S@@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569187 CD On-Demand Anodyne CYP11B2 21 40 C[S@@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569187 CD On-Demand Anodyne CYP27B1 47 31 C[S@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569188 CD On-Demand Anodyne CYP19A1 20 40 C[S@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569188 CD On-Demand Anodyne CYP11B1 39 40 C[S@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569188 CD On-Demand Anodyne TBXAS1 38 41 C[S@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569188 CD On-Demand Anodyne CYP11B2 21 40 C[S@](=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569188 CD On-Demand Anodyne CYP27B1 47 31 C[S@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569189 CD On-Demand Anodyne CYP19A1 20 40 C[S@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569189 CD On-Demand Anodyne CYP11B1 39 40 C[S@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569189 CD On-Demand Anodyne TBXAS1 38 41 C[S@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569189 CD On-Demand Anodyne CYP11B2 21 40 C[S@](=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569189 CD On-Demand Anodyne CYP27B1 47 31 c1ccc([C@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569190 DG On-Demand Anodyne CYP19A1 15 42 c1ccc([C@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569190 DG On-Demand Anodyne CYP11B1 38 43 c1ccc([C@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569190 DG On-Demand Anodyne TBXAS1 30 42 c1ccc([C@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569190 DG On-Demand Anodyne CYP11B2 19 42 c1ccc([C@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569190 DG On-Demand Anodyne HMOX1 48 39 N#CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569191 CC On-Demand Mild TBXAS1 53 41 N#CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569191 CC On-Demand Mild CYP27B1 42 35 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569193 DG On-Demand Anodyne CYP19A1 15 42 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569193 DG On-Demand Anodyne CYP11B1 38 43 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569193 DG On-Demand Anodyne TBXAS1 30 42 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569193 DG On-Demand Anodyne CYP11B2 19 42 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccncc2)cc1 ZINC000880569193 DG On-Demand Anodyne HMOX1 48 39 CC[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569194 CG On-Demand Anodyne CYP19A1 16 41 CC[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569194 CG On-Demand Anodyne CYP11B1 37 41 CC[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569194 CG On-Demand Anodyne TBXAS1 26 41 CC[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569194 CG On-Demand Anodyne CYP11B2 20 41 CC[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569194 CG On-Demand Anodyne CYP27B1 48 32 CC[C@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569196 CG On-Demand Anodyne CYP19A1 16 41 CC[C@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569196 CG On-Demand Anodyne CYP11B1 37 41 CC[C@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569196 CG On-Demand Anodyne TBXAS1 26 41 CC[C@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569196 CG On-Demand Anodyne CYP11B2 20 41 CC[C@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569196 CG On-Demand Anodyne CYP27B1 48 32 CC[C@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569198 CG On-Demand Anodyne CYP19A1 16 41 CC[C@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569198 CG On-Demand Anodyne CYP11B1 37 41 CC[C@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569198 CG On-Demand Anodyne TBXAS1 26 41 CC[C@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569198 CG On-Demand Anodyne CYP11B2 20 41 CC[C@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569198 CG On-Demand Anodyne CYP27B1 48 32 CC[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569199 CG On-Demand Anodyne CYP19A1 16 41 CC[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569199 CG On-Demand Anodyne CYP11B1 37 41 CC[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569199 CG On-Demand Anodyne TBXAS1 26 41 CC[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569199 CG On-Demand Anodyne CYP11B2 20 41 CC[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569199 CG On-Demand Anodyne CYP27B1 48 32 COc1ccc(C)cc1CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569201 DH On-Demand Anodyne CYP19A1 24 42 COc1ccc(C)cc1CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569201 DH On-Demand Anodyne QPCT 24 42 COc1ccc(C)cc1CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569203 DH On-Demand Anodyne CYP19A1 24 42 COc1ccc(C)cc1CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569203 DH On-Demand Anodyne QPCT 24 42 CCOC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569206 DF On-Demand Anodyne CYP19A1 15 40 CCOC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569206 DF On-Demand Anodyne TBXAS1 72 50 CCOC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569206 DF On-Demand Anodyne CYP24A1 51 36 CCOC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569206 DF On-Demand Anodyne CYP26A1 88 40 CCOC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569206 DF On-Demand Anodyne CYP27B1 68 36 CCOC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569208 DF On-Demand Anodyne CYP19A1 15 40 CCOC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569208 DF On-Demand Anodyne TBXAS1 72 50 CCOC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569208 DF On-Demand Anodyne CYP24A1 51 36 CCOC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569208 DF On-Demand Anodyne CYP26A1 88 40 CCOC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569208 DF On-Demand Anodyne CYP27B1 68 36 CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880569210 GE On-Demand Anodyne GPR119 33 43 CN(C)S(=O)(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569211 DD On-Demand Anodyne CYP24A1 40 32 CN(C)S(=O)(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569211 DD On-Demand Anodyne CYP27B1 52 31 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880569212 GE On-Demand Anodyne GPR119 33 43 CN(C)S(=O)(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569213 DD On-Demand Anodyne CYP24A1 40 32 CN(C)S(=O)(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569213 DD On-Demand Anodyne CYP27B1 52 31 CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880569214 GE On-Demand Anodyne GPR119 33 43 CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880569216 GE On-Demand Anodyne GPR119 33 43 C=C(CC)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569234 CG On-Demand Mild CYP11B1 33 40 C=C(CC)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569234 CG On-Demand Mild TBXAS1 38 41 C=C(CC)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569234 CG On-Demand Mild CYP11B2 18 40 C=C(CC)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569234 CG On-Demand Mild CYP27B1 47 31 C=C(CC)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569236 CG On-Demand Mild CYP11B1 33 40 C=C(CC)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569236 CG On-Demand Mild TBXAS1 38 41 C=C(CC)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569236 CG On-Demand Mild CYP11B2 18 40 C=C(CC)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569236 CG On-Demand Mild CYP27B1 47 31 CN(CCC#N)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569238 ED On-Demand Mild CYP26A1 80 35 CN(CCC#N)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569244 ED On-Demand Mild CYP26A1 80 35 O=C1[C@@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569247 FG On-Demand Anodyne CYP11B1 25 42 O=C1[C@@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569247 FG On-Demand Anodyne TBXAS1 17 42 O=C1[C@@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569247 FG On-Demand Anodyne CYP11B2 15 42 O=C1[C@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569249 FG On-Demand Anodyne CYP11B1 25 42 O=C1[C@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569249 FG On-Demand Anodyne TBXAS1 17 42 O=C1[C@H](N[C@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569249 FG On-Demand Anodyne CYP11B2 15 42 CC(C)(C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569250 DE On-Demand Anodyne TBXAS1 60 43 CC(C)(C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569250 DE On-Demand Anodyne CYP24A1 41 35 CC(C)(C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569250 DE On-Demand Anodyne CYP26A1 64 37 CC(C)(C)NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569250 DE On-Demand Anodyne CYP27B1 53 35 O=C1[C@@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569251 FG On-Demand Anodyne CYP11B1 25 42 O=C1[C@@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569251 FG On-Demand Anodyne TBXAS1 17 42 O=C1[C@@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569251 FG On-Demand Anodyne CYP11B2 15 42 CC(C)(C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569252 DE On-Demand Anodyne TBXAS1 60 43 CC(C)(C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569252 DE On-Demand Anodyne CYP24A1 41 35 CC(C)(C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569252 DE On-Demand Anodyne CYP26A1 64 37 CC(C)(C)NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569252 DE On-Demand Anodyne CYP27B1 53 35 O=C1[C@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569254 FG On-Demand Anodyne CYP11B1 25 42 O=C1[C@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569254 FG On-Demand Anodyne TBXAS1 17 42 O=C1[C@H](N[C@@H](Cn2ccnc2)c2ccccc2)CCCN1Cc1ccccc1 ZINC000880569254 FG On-Demand Anodyne CYP11B2 15 42 O=[N+]([O-])c1ccn(CCN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880569257 EE On-Demand Bother CYP19A1 17 40 O=[N+]([O-])c1ccn(CCN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880569259 EE On-Demand Bother CYP19A1 17 40 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne CYP19A1 31 45 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne CYP11B1 49 47 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne TBXAS1 55 48 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne CYP11B2 24 47 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne HMOX1 36 40 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne HMOX2 48 39 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne CYP24A1 49 37 c1ccc([C@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569263 CE On-Demand Anodyne CYP27B1 67 37 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne CYP19A1 31 45 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne CYP11B1 49 47 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne TBXAS1 55 48 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne CYP11B2 24 47 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne HMOX1 36 40 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne HMOX2 48 39 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne CYP24A1 49 37 c1ccc([C@@H](Cn2ccnc2)NCCn2ccnc2)cc1 ZINC000880569265 CE On-Demand Anodyne CYP27B1 67 37 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC1CCC1 ZINC000880569268 DE On-Demand Anodyne TBXAS1 41 39 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC1CCC1 ZINC000880569269 DE On-Demand Anodyne TBXAS1 41 39 C[C@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N1CCCCC1 ZINC000880569271 GD On-Demand Anodyne DPP7 46 36 C[C@@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N1CCCCC1 ZINC000880569272 GD On-Demand Anodyne DPP7 46 36 C[C@@H](NC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)C(=O)N1CCCCC1 ZINC000880569273 GD On-Demand Anodyne DPP7 46 36 C[C@H](NC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)C(=O)N1CCCCC1 ZINC000880569274 GD On-Demand Anodyne DPP7 46 36 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCCCO3)cc1 ZINC000880569275 GE On-Demand Anodyne BMP1 65 36 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne BMP1 79 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP13 47 43 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP2 30 40 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP3 33 43 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP8 29 43 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP9 40 40 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP12 30 43 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)C(F)F)cc2)cc1 ZINC000880569276 GF On-Demand Anodyne MMP1 33 43 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccs2)cc1 ZINC000880569279 EE On-Demand Anodyne BMP1 28 40 COc1ccc(CN(CCO)CCC(=O)N2CCc3sccc3C2)cc1 ZINC000880569282 FF On-Demand Anodyne BMP1 46 36 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne MMP13 36 47 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne ROCK1 42 42 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne MTNR1A 90 45 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne MTNR1B 80 45 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne MMP3 16 46 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne ROCK2 47 42 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne CA9 15 40 COc1ccc(CN(CCO)CC(=O)NCc2cccc(OC)c2)cc1 ZINC000880569288 FD On-Demand Anodyne PDS 50 40 COc1ccc(CN(CCO)CC(=O)NCC(=O)N2CCCC2)cc1 ZINC000880569300 EC On-Demand Anodyne MMP13 20 43 COc1ccc(CN(CCO)CC(=O)NCC(=O)N2CCCC2)cc1 ZINC000880569300 EC On-Demand Anodyne MMP3 22 43 COc1ccc(CN(CCO)CC(=O)NCC(=O)N2CCCC2)cc1 ZINC000880569300 EC On-Demand Anodyne DPP7 21 41 COc1ccc(CN(CCO)CC(=O)NCC(=O)N2CCCC2)cc1 ZINC000880569300 EC On-Demand Anodyne MMP1 24 43 COc1ccc(CN(CCO)Cc2cc(F)ccc2OC)cc1 ZINC000880569305 DF On-Demand Anodyne TSPO 32 42 CC[C@H](C)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569310 CD On-Demand Anodyne MMP13 16 41 CC[C@H](C)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569310 CD On-Demand Anodyne MMP3 23 41 CC[C@H](C)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569310 CD On-Demand Anodyne MMP8 19 41 CC[C@H](C)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569310 CD On-Demand Anodyne MMP12 22 41 CC[C@H](C)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569310 CD On-Demand Anodyne MMP1 28 41 COc1ccc(CN(CCO)C[C@@H](O)c2ccc(F)cc2)cc1 ZINC000880569313 DE On-Demand Anodyne AOC3 18 48 COc1ccc(CN(CCO)C[C@H](O)c2ccc(F)cc2)cc1 ZINC000880569314 DE On-Demand Anodyne AOC3 18 48 COc1ccc(CN(CCO)Cc2nc3ccccc3s2)cc1 ZINC000880569317 EG On-Demand Anodyne LUCI_PHOPE 30 48 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne LTA4H 52 50 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne BMP1 34 43 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP13 24 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne HDAC8 17 43 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MTNR1A 25 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MTNR1B 30 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP2 19 44 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP3 34 44 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP8 17 44 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne NPY5R 29 46 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP9 31 44 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP12 25 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne CA9 16 43 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne MMP1 34 44 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2)cc1 ZINC000880569318 DE On-Demand Anodyne RORC 16 45 COc1ccc(CN(CCO)CC(=O)Nc2cccc(NC(C)=O)c2)cc1 ZINC000880569322 FE On-Demand Anodyne LTA4H 18 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(NC(C)=O)c2)cc1 ZINC000880569322 FE On-Demand Anodyne MTNR1A 50 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(NC(C)=O)c2)cc1 ZINC000880569322 FE On-Demand Anodyne MTNR1B 48 42 FC(F)OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569323 CE On-Demand Anodyne CYP19A1 24 41 FC(F)OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569323 CE On-Demand Anodyne CYP11B1 40 41 FC(F)OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569323 CE On-Demand Anodyne TBXAS1 33 43 FC(F)OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569323 CE On-Demand Anodyne CYP11B2 20 41 FC(F)OCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569323 CE On-Demand Anodyne CYP27B1 48 30 FC(F)OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569324 CE On-Demand Anodyne CYP19A1 24 41 FC(F)OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569324 CE On-Demand Anodyne CYP11B1 40 41 FC(F)OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569324 CE On-Demand Anodyne TBXAS1 33 43 FC(F)OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569324 CE On-Demand Anodyne CYP11B2 20 41 FC(F)OCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569324 CE On-Demand Anodyne CYP27B1 48 30 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP13 18 45 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP3 20 45 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP8 15 45 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP9 23 41 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP12 22 45 CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569326 CC On-Demand Anodyne MMP1 31 45 COc1ccc(CN(CCO)Cc2ccc(OC(F)F)cc2)cc1 ZINC000880569327 EG On-Demand Anodyne SLC18A2 20 40 Cn1nc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1Cl ZINC000880569328 DF On-Demand Anodyne CYP27B1 40 33 Cn1nc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1Cl ZINC000880569329 DF On-Demand Anodyne CYP27B1 40 33 COc1ccc(CN(CCO)Cc2csc(NC(C)=O)n2)cc1 ZINC000880569335 EE On-Demand Anodyne AOC3 18 44 CC(C)(C)OC(=O)N1CC(CCN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880569342 FG On-Demand Anodyne CYP27B1 40 33 CC(C)(C)OC(=O)N1CC(CCN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880569343 FG On-Demand Anodyne CYP27B1 40 33 COc1ccc(CN(CCO)Cc2cc([N+](=O)[O-])ccc2OC)cc1 ZINC000880569344 EF On-Demand Bother TBXA2R 15 42 COc1ccc(CN(CCO)Cc2cc([N+](=O)[O-])ccc2OC)cc1 ZINC000880569344 EF On-Demand Bother BMP1 24 40 COc1ccc(CN(CCO)Cc2cc([N+](=O)[O-])ccc2OC)cc1 ZINC000880569344 EF On-Demand Bother MMP8 24 45 COc1ccc(CN(CCO)Cc2cc([N+](=O)[O-])ccc2OC)cc1 ZINC000880569344 EF On-Demand Bother MMP1 19 45 COc1ccc(CN(CCO)Cc2nc(-c3ccccn3)no2)cc1 ZINC000880569345 EE On-Demand Anodyne LUCI_PHOPE 31 43 COc1ccc(CN(CCO)C[C@H](O)COc2ccc(F)cc2)cc1 ZINC000880569346 EE On-Demand Anodyne GRIN1 23 52 COc1ccc(CN(CCO)C[C@@H](O)COc2ccc(F)cc2)cc1 ZINC000880569347 EE On-Demand Anodyne GRIN1 23 52 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne BMP1 66 38 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP13 35 46 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP2 18 41 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP3 26 43 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP8 18 41 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP9 34 41 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP12 27 43 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccccc2)cc1 ZINC000880569357 FE On-Demand Anodyne MMP1 31 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne PDGFRB 16 43 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne LTA4H 25 43 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne ROCK1 24 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne MTNR1A 54 49 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne MTNR1B 52 51 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne ROCK2 29 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne TAAR1 33 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(OC)c2)cc1 ZINC000880569362 EE On-Demand Anodyne KCNK3 46 35 COc1ccc(CN(CCO)C[C@@H](O)c2ccccc2)cc1 ZINC000880569365 DE On-Demand Anodyne AOC3 26 47 COc1ccc(CN(CCO)C[C@H](O)c2ccccc2)cc1 ZINC000880569366 DE On-Demand Anodyne AOC3 26 47 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C2SCCCS2)cc1 ZINC000880569367 HK On-Demand Mild GRM5 15 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C2SCCCS2)cc1 ZINC000880569367 HK On-Demand Mild KCNK3 61 42 COc1ccc(CN(CCO)Cc2cccc(C(=O)NCc3ccco3)c2)cc1 ZINC000880569368 GG On-Demand Anodyne MMP13 19 43 COc1ccc(CN(CCO)Cc2cccc(C(=O)NCc3ccco3)c2)cc1 ZINC000880569368 GG On-Demand Anodyne ROCK2 23 42 CCC(CC)[C@H](CNC(=O)COc1ccc2c(C)cc(=O)oc2c1)N1CCOCC1 ZINC000880569369 HF On-Demand Anodyne MAOA 65 56 CCC(CC)[C@H](CNC(=O)COc1ccc2c(C)cc(=O)oc2c1)N1CCOCC1 ZINC000880569369 HF On-Demand Anodyne MAOB 37 56 CCC(CC)[C@@H](CNC(=O)COc1ccc2c(C)cc(=O)oc2c1)N1CCOCC1 ZINC000880569370 HF On-Demand Anodyne MAOA 65 56 CCC(CC)[C@@H](CNC(=O)COc1ccc2c(C)cc(=O)oc2c1)N1CCOCC1 ZINC000880569370 HF On-Demand Anodyne MAOB 37 56 CC/C=C\CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569384 CH On-Demand Anodyne CYP11B1 39 42 CC/C=C\CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569384 CH On-Demand Anodyne TBXAS1 24 42 CC/C=C\CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569384 CH On-Demand Anodyne CYP11B2 19 42 CC/C=C/CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569385 CH On-Demand Anodyne CYP11B1 39 42 CC/C=C/CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569385 CH On-Demand Anodyne TBXAS1 24 42 CC/C=C/CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569385 CH On-Demand Anodyne CYP11B2 19 42 CC/C=C\CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569386 CH On-Demand Anodyne CYP11B1 39 42 CC/C=C\CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569386 CH On-Demand Anodyne TBXAS1 24 42 CC/C=C\CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569386 CH On-Demand Anodyne CYP11B2 19 42 CC/C=C/CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569387 CH On-Demand Anodyne CYP11B1 39 42 CC/C=C/CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569387 CH On-Demand Anodyne TBXAS1 24 42 CC/C=C/CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569387 CH On-Demand Anodyne CYP11B2 19 42 c1ccc([C@H](Cn2ccnc2)NCCc2cncs2)cc1 ZINC000880569394 CF On-Demand Anodyne CYP11B1 42 40 c1ccc([C@H](Cn2ccnc2)NCCc2cncs2)cc1 ZINC000880569394 CF On-Demand Anodyne CYP11B2 20 40 c1ccc([C@@H](Cn2ccnc2)NCCc2cncs2)cc1 ZINC000880569395 CF On-Demand Anodyne CYP11B1 42 40 c1ccc([C@@H](Cn2ccnc2)NCCc2cncs2)cc1 ZINC000880569395 CF On-Demand Anodyne CYP11B2 20 40 O=S(=O)(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569398 FF On-Demand Anodyne CYP19A1 17 43 O=S(=O)(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569398 FF On-Demand Anodyne CYP11B1 35 43 O=S(=O)(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569398 FF On-Demand Anodyne TBXAS1 31 43 O=S(=O)(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569398 FF On-Demand Anodyne CYP11B2 18 43 O=S(=O)(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569399 FF On-Demand Anodyne CYP19A1 17 43 O=S(=O)(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569399 FF On-Demand Anodyne CYP11B1 35 43 O=S(=O)(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569399 FF On-Demand Anodyne TBXAS1 31 43 O=S(=O)(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569399 FF On-Demand Anodyne CYP11B2 18 43 CN(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569401 EG On-Demand Anodyne CYP19A1 18 43 CN(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569401 EG On-Demand Anodyne CYP11B1 38 43 CN(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569401 EG On-Demand Anodyne TBXAS1 33 43 CN(CCN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569401 EG On-Demand Anodyne CYP11B2 19 43 CN(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569402 EG On-Demand Anodyne CYP19A1 18 43 CN(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569402 EG On-Demand Anodyne CYP11B1 38 43 CN(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569402 EG On-Demand Anodyne TBXAS1 33 43 CN(CCN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569402 EG On-Demand Anodyne CYP11B2 19 43 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne CYP19A1 28 45 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne CYP11B1 46 40 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne TBXAS1 26 48 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne CYP11B2 28 40 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne HMOX2 26 43 COc1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569415 EG On-Demand Anodyne CYP27B1 47 37 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne CYP19A1 28 45 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne CYP11B1 46 40 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne TBXAS1 26 48 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne CYP11B2 28 40 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne HMOX2 26 43 COc1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880569416 EG On-Demand Anodyne CYP27B1 47 37 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCN(c2cnccn2)CC1 ZINC000880569417 GD On-Demand Anodyne PTAFR 32 44 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCN(c2cnccn2)CC1 ZINC000880569418 GD On-Demand Anodyne PTAFR 32 44 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild CYP19A1 18 40 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild CYP11B1 34 40 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild TBXAS1 39 41 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild CYP11B2 19 40 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild CYP24A1 42 33 C=C(C)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569430 CG On-Demand Mild CYP27B1 55 33 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild CYP19A1 18 40 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild CYP11B1 34 40 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild TBXAS1 39 41 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild CYP11B2 19 40 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild CYP24A1 42 33 C=C(C)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569431 CG On-Demand Mild CYP27B1 55 33 Cn1cc(-c2ccc(C(=O)NCc3cn(C4CCC4)nn3)cc2)cn1 ZINC000880569444 EE On-Demand Anodyne CA14 15 45 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne CYP19A1 19 40 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne CYP11B1 36 40 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne TBXAS1 37 41 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne CYP11B2 19 40 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne HMOX1 30 40 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne CYP24A1 42 34 CC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569447 CD On-Demand Anodyne CYP27B1 54 34 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne CYP19A1 19 40 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne CYP11B1 36 40 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne TBXAS1 37 41 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne CYP11B2 19 40 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne HMOX1 30 40 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne CYP24A1 42 34 CC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569448 CD On-Demand Anodyne CYP27B1 54 34 CN(C)[C@@H](CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569457 GF On-Demand Anodyne TBXAS1 37 40 CN(C)[C@@H](CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569457 GF On-Demand Anodyne CYP26A1 50 35 CN(C)[C@@H](CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569457 GF On-Demand Anodyne CYP27B1 42 35 CN(C)[C@@H](CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569458 GF On-Demand Anodyne TBXAS1 37 40 CN(C)[C@@H](CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569458 GF On-Demand Anodyne CYP26A1 50 35 CN(C)[C@@H](CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880569458 GF On-Demand Anodyne CYP27B1 42 35 COc1ccc(CN(CCO)CCC(=O)N2CCN(c3ncccn3)CC2)cc1 ZINC000880569472 GD On-Demand Anodyne BMP1 16 40 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2C(C)C)cc1 ZINC000880569493 FG On-Demand Anodyne SOAT1 16 40 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2C(C)C)cc1 ZINC000880569493 FG On-Demand Anodyne NPY5R 15 40 COc1ccc(CN(CCO)CC(=O)NC2CCCCCC2)cc1 ZINC000880569497 EE On-Demand Anodyne MMP13 18 42 COc1ccc(CN(CCO)CC(=O)NC2CCCCCC2)cc1 ZINC000880569497 EE On-Demand Anodyne MMP3 23 42 COc1ccc(CN(CCO)CC(=O)NC2CCCCCC2)cc1 ZINC000880569497 EE On-Demand Anodyne MMP9 17 42 COc1ccc(CN(CCO)CC(=O)NC2CCCCCC2)cc1 ZINC000880569497 EE On-Demand Anodyne EPHX2 15 48 COc1ccc(CN(CCO)CC(=O)NC2CCCCCC2)cc1 ZINC000880569497 EE On-Demand Anodyne MMP1 20 42 COc1ccc(CN(CCO)Cc2coc(-c3ccccc3)n2)cc1 ZINC000880569500 EG On-Demand Anodyne PPARA 18 42 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2)cc1 ZINC000880569505 ED On-Demand Anodyne ADRB2 23 48 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2)cc1 ZINC000880569505 ED On-Demand Anodyne ADRB1 34 48 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2)cc1 ZINC000880569505 ED On-Demand Anodyne GRIN1 21 49 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2)cc1 ZINC000880569505 ED On-Demand Anodyne ADRB3 25 48 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2)cc1 ZINC000880569505 ED On-Demand Anodyne ABCB1 19 42 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2)cc1 ZINC000880569506 ED On-Demand Anodyne ADRB2 23 48 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2)cc1 ZINC000880569506 ED On-Demand Anodyne ADRB1 34 48 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2)cc1 ZINC000880569506 ED On-Demand Anodyne GRIN1 21 49 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2)cc1 ZINC000880569506 ED On-Demand Anodyne ADRB3 25 48 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2)cc1 ZINC000880569506 ED On-Demand Anodyne ABCB1 19 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880569509 FE On-Demand Anodyne EDNRB 72 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880569509 FE On-Demand Anodyne EDNRA 70 46 COc1ccc(CN(CCO)CCC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880569509 FE On-Demand Anodyne BMP1 86 42 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother CACNA1C 45 43 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother BMP1 30 41 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother CACNA1D 73 43 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother MMP8 18 43 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother MMP9 17 43 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother MMP1 18 43 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2)cc1 ZINC000880569510 DF On-Demand Bother NR1D1 30 44 COc1ccc(CN(CCO)Cc2cccc(C(=O)N(C)C)c2)cc1 ZINC000880569511 EE On-Demand Anodyne HSD17B2 22 43 COc1ccc(CN(CCO)C[C@@H](O)c2cccc(F)c2)cc1 ZINC000880569518 DE On-Demand Anodyne AOC3 20 44 COc1ccc(CN(CCO)C[C@H](O)c2cccc(F)c2)cc1 ZINC000880569519 DE On-Demand Anodyne AOC3 20 44 COc1ccc(CN(CCO)Cc2nc(-c3ccc(F)cc3)no2)cc1 ZINC000880569521 FF On-Demand Anodyne LUCI_PHOPE 28 40 COc1ccc(CN(CCO)Cc2csc([N+](=O)[O-])c2)cc1 ZINC000880569534 DF On-Demand Bother NR1D1 36 47 COC(=O)C1CCN(C(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880569535 FC On-Demand Anodyne CACNA1G 23 41 COC(=O)C1CCN(C(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880569535 FC On-Demand Anodyne PTR1 49 39 COC(=O)c1sccc1NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569539 GD On-Demand Anodyne FAS 47 56 COc1ccc(CN(CCO)CC(=O)Nc2c(C)cccc2C(C)C)cc1 ZINC000880569541 FH On-Demand Anodyne SOAT1 36 45 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CC2)cc1 ZINC000880569542 DC On-Demand Anodyne MMP13 29 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CC2)cc1 ZINC000880569542 DC On-Demand Anodyne MMP3 33 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CC2)cc1 ZINC000880569542 DC On-Demand Anodyne MMP8 20 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CC2)cc1 ZINC000880569542 DC On-Demand Anodyne MMP12 18 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CC2)cc1 ZINC000880569542 DC On-Demand Anodyne MMP1 27 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2N2CCCC2=O)cc1 ZINC000880569546 GE On-Demand Anodyne KCNQ2 56 41 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880569547 DF On-Demand Bother MMP2 19 52 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880569547 DF On-Demand Bother MMP8 37 52 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880569547 DF On-Demand Bother MMP9 22 52 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880569547 DF On-Demand Bother MMP1 28 52 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880569547 DF On-Demand Bother NR1D1 22 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne LTA4H 55 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne BMP1 33 47 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne HDAC8 19 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne MTNR1A 17 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne MTNR1B 22 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne MMP3 25 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne NPY5R 24 43 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne MMP9 23 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne CA9 15 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2)cc1 ZINC000880569555 EF On-Demand Anodyne MMP1 26 41 CCN(CC)C(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569558 CD On-Demand Anodyne HCRTR2 17 48 COc1ccc(CN(CCO)CCOc2ccccc2[N+](=O)[O-])cc1 ZINC000880569562 EE On-Demand Bother COLA 19 40 O=C(CCc1cccc2ccccc12)NCc1cn(C2CCC2)nn1 ZINC000880569592 EG On-Demand Anodyne MTNR1A 17 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569599 CE On-Demand Anodyne CYP11B1 35 42 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569599 CE On-Demand Anodyne CYP11B2 18 42 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569599 CE On-Demand Anodyne CYP27B1 44 33 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569600 CE On-Demand Anodyne CYP11B1 35 42 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569600 CE On-Demand Anodyne CYP11B2 18 42 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569600 CE On-Demand Anodyne CYP27B1 44 33 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569601 CE On-Demand Anodyne CYP11B1 35 42 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569601 CE On-Demand Anodyne CYP11B2 18 42 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569601 CE On-Demand Anodyne CYP27B1 44 33 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569602 CE On-Demand Anodyne CYP11B1 35 42 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569602 CE On-Demand Anodyne CYP11B2 18 42 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C(F)(F)F ZINC000880569602 CE On-Demand Anodyne CYP27B1 44 33 c1ccc([C@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569603 DI On-Demand Anodyne CYP19A1 17 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569603 DI On-Demand Anodyne CYP11B1 40 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569603 DI On-Demand Anodyne TBXAS1 22 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569603 DI On-Demand Anodyne CYP11B2 18 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569603 DI On-Demand Anodyne HMOX1 41 35 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569604 DI On-Demand Anodyne CYP19A1 17 40 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569604 DI On-Demand Anodyne CYP11B1 40 40 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569604 DI On-Demand Anodyne TBXAS1 22 40 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569604 DI On-Demand Anodyne CYP11B2 18 40 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(C3CC3)cc2)cc1 ZINC000880569604 DI On-Demand Anodyne HMOX1 41 35 CSc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1Br ZINC000880569605 GG On-Demand Anodyne CA14 15 43 FC(F)(F)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569629 DH On-Demand Anodyne CYP11B1 27 40 FC(F)(F)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569629 DH On-Demand Anodyne CYP11B2 15 40 FC(F)(F)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569630 DH On-Demand Anodyne CYP11B1 27 40 FC(F)(F)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569630 DH On-Demand Anodyne CYP11B2 15 40 COC(=O)c1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1C ZINC000880569635 EE On-Demand Anodyne CA14 20 42 COC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880569636 CD On-Demand Anodyne CYP19A1 18 44 COC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880569636 CD On-Demand Anodyne TBXAS1 23 40 COC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880569638 CD On-Demand Anodyne CYP19A1 18 44 COC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880569638 CD On-Demand Anodyne TBXAS1 23 40 C[C@H]1CC(=O)N[C@@H](C(=O)NCc2cn(C3CCC3)nn2)C1 ZINC000880569644 CC On-Demand Anodyne TRHR 50 35 C[C@@]1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569649 DH On-Demand Anodyne CYP11B1 24 40 C[C@@]1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569649 DH On-Demand Anodyne TBXAS1 18 40 C[C@@]1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569650 DH On-Demand Anodyne CYP11B1 24 40 C[C@@]1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569650 DH On-Demand Anodyne TBXAS1 18 40 C[C@]1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569651 DH On-Demand Anodyne CYP11B1 24 40 C[C@]1(CN[C@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569651 DH On-Demand Anodyne TBXAS1 18 40 C[C@]1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569652 DH On-Demand Anodyne CYP11B1 24 40 C[C@]1(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1(Cl)Cl ZINC000880569652 DH On-Demand Anodyne TBXAS1 18 40 C=CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569657 CE On-Demand Mild TBXAS1 25 40 C=CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569657 CE On-Demand Mild CYP27B1 43 31 C=CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569658 CE On-Demand Mild TBXAS1 25 40 C=CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569658 CE On-Demand Mild CYP27B1 43 31 CNC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569659 CD On-Demand Anodyne CYP19A1 16 40 CNC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569659 CD On-Demand Anodyne TBXAS1 67 45 CNC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569659 CD On-Demand Anodyne CYP24A1 57 40 CNC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569659 CD On-Demand Anodyne CYP26A1 65 39 CNC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569659 CD On-Demand Anodyne CYP27B1 78 40 CNC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569660 CD On-Demand Anodyne CYP19A1 16 40 CNC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569660 CD On-Demand Anodyne TBXAS1 67 45 CNC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569660 CD On-Demand Anodyne CYP24A1 57 40 CNC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569660 CD On-Demand Anodyne CYP26A1 65 39 CNC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569660 CD On-Demand Anodyne CYP27B1 78 40 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)NC(=O)NCC(F)(F)F ZINC000880569661 GD On-Demand Anodyne CYP27B1 47 36 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)NC(=O)NCC(F)(F)F ZINC000880569662 GD On-Demand Anodyne CYP27B1 47 36 c1ccc([C@H](Cn2ccnc2)NC[C@@H]2COc3ccccc3O2)cc1 ZINC000880569668 EG On-Demand Anodyne ADRA2B 15 42 c1ccc([C@@H](Cn2ccnc2)NC[C@@H]2COc3ccccc3O2)cc1 ZINC000880569669 EG On-Demand Anodyne ADRA2B 15 42 c1ccc([C@H](Cn2ccnc2)NC[C@H]2COc3ccccc3O2)cc1 ZINC000880569670 EG On-Demand Anodyne ADRA2B 15 42 c1ccc([C@@H](Cn2ccnc2)NC[C@H]2COc3ccccc3O2)cc1 ZINC000880569671 EG On-Demand Anodyne ADRA2B 15 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569685 EC On-Demand Reactive TBXAS1 49 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569685 EC On-Demand Reactive CCR5 21 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569685 EC On-Demand Reactive CYP27B1 48 31 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569686 EC On-Demand Reactive TBXAS1 49 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569686 EC On-Demand Reactive CCR5 21 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NNC(=O)C1CC1 ZINC000880569686 EC On-Demand Reactive CYP27B1 48 31 COc1ccc(CN(CCO)C[C@@H](O)COc2cccc(C)c2)cc1 ZINC000880569691 EE On-Demand Anodyne GRIN1 19 43 COc1ccc(CN(CCO)C[C@H](O)COc2cccc(C)c2)cc1 ZINC000880569692 EE On-Demand Anodyne GRIN1 19 43 COc1ccc(CN(CCO)CCCNC(C)=O)cc1 ZINC000880569697 CD On-Demand Anodyne MTNR1A 104 47 COc1ccc(CN(CCO)CCCNC(C)=O)cc1 ZINC000880569697 CD On-Demand Anodyne MTNR1B 90 48 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2F)cc1 ZINC000880569706 FE On-Demand Anodyne GNRHR 18 40 COc1ccc(CN(CCO)Cc2ccc(-n3cccn3)cc2)cc1 ZINC000880569711 EF On-Demand Anodyne AMP1_PLAFQ 43 36 COc1ccc(CN(CCO)Cc2ccc(Cl)nc2)cc1 ZINC000880569716 DF On-Demand Anodyne Q8WSF8_APLCA 26 40 COc1ccc(CN(CCO)Cc2ccc(Cl)nc2)cc1 ZINC000880569716 DF On-Demand Anodyne NACHRBETA2 32 40 COc1ccc(CN(CCO)CC(=O)NC2CC2)cc1 ZINC000880569717 CC On-Demand Anodyne MMP13 18 41 COc1ccc(CN(CCO)CC(=O)NC2CC2)cc1 ZINC000880569717 CC On-Demand Anodyne MMP3 27 41 COc1ccc(CN(CCO)CC(=O)NC2CC2)cc1 ZINC000880569717 CC On-Demand Anodyne MMP8 15 41 COc1ccc(CN(CCO)CC(=O)NC2CC2)cc1 ZINC000880569717 CC On-Demand Anodyne MMP12 16 41 COc1ccc(CN(CCO)CC(=O)NC2CC2)cc1 ZINC000880569717 CC On-Demand Anodyne MMP1 24 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne BMP1 72 38 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne MMP13 23 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne MMP3 28 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne MMP8 20 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne MMP12 24 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(C)C)cc1 ZINC000880569733 EC On-Demand Anodyne MMP1 31 41 COc1ccc(CN(CCO)Cc2ccc(Cl)s2)cc1 ZINC000880569734 DG On-Demand Anodyne NR1D1 35 42 COc1ccc(CN(CCO)CC(=O)N2CCCC2)cc1 ZINC000880569735 CD On-Demand Anodyne MMP13 22 41 COc1ccc(CN(CCO)CC(=O)N2CCCC2)cc1 ZINC000880569735 CD On-Demand Anodyne DPP7 15 41 COc1ccc(CN(CCO)CC(=O)N2CCCC2)cc1 ZINC000880569735 CD On-Demand Anodyne MMP1 24 41 COc1ccc(CN(CCO)Cc2ccccc2[N+](=O)[O-])cc1 ZINC000880569739 DF On-Demand Bother COLA 122 49 COc1ccc(CN(CCO)Cc2cnn(-c3ccccc3)c2)cc1 ZINC000880569742 EF On-Demand Anodyne GRM4 17 41 COc1ccc(CN(CCO)CCC(=O)N2CCCCC2)cc1 ZINC000880569743 DD On-Demand Anodyne MMP13 15 42 COc1ccc(CN(CCO)CCC(=O)N2CCCCC2)cc1 ZINC000880569743 DD On-Demand Anodyne DPP7 20 42 COc1ccc(CN(CCO)CCC(=O)N2CCCCC2)cc1 ZINC000880569743 DD On-Demand Anodyne MMP1 17 42 CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569744 CC On-Demand Anodyne MMP13 15 44 CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569744 CC On-Demand Anodyne MMP3 17 44 CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569744 CC On-Demand Anodyne MMP9 19 40 CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569744 CC On-Demand Anodyne MMP12 22 44 CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569744 CC On-Demand Anodyne MMP1 22 44 CCN(C(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880569746 EF On-Demand Anodyne MMP9 15 41 COc1ccc(CN(CCO)CC(=O)NCc2cccs2)cc1 ZINC000880569750 ED On-Demand Anodyne BMP1 41 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(O)cc2)cc1 ZINC000880569751 ED On-Demand Anodyne LTA4H 32 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(O)cc2)cc1 ZINC000880569751 ED On-Demand Anodyne MTNR1B 19 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(O)cc2)cc1 ZINC000880569751 ED On-Demand Anodyne NPY5R 15 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(O)cc2)cc1 ZINC000880569751 ED On-Demand Anodyne MMP12 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(O)cc2)cc1 ZINC000880569751 ED On-Demand Anodyne CA9 18 44 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569763 GD On-Demand Anodyne MMP13 15 45 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569763 GD On-Demand Anodyne MMP3 19 45 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569763 GD On-Demand Anodyne MMP8 19 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569763 GD On-Demand Anodyne DPP7 40 45 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569763 GD On-Demand Anodyne MMP1 24 45 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569764 GD On-Demand Anodyne MMP13 15 45 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569764 GD On-Demand Anodyne MMP3 19 45 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569764 GD On-Demand Anodyne MMP8 19 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569764 GD On-Demand Anodyne DPP7 40 45 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(=O)N2CCCCC2)cc1 ZINC000880569764 GD On-Demand Anodyne MMP1 24 45 COC(=O)c1cc(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)c(C)[nH]1 ZINC000880569770 FF On-Demand Anodyne TBXAS1 40 38 COC(=O)c1cc(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)c(C)[nH]1 ZINC000880569770 FF On-Demand Anodyne CYP27B1 40 33 COC(=O)c1cc(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)c(C)[nH]1 ZINC000880569771 FF On-Demand Anodyne TBXAS1 40 38 COC(=O)c1cc(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)c(C)[nH]1 ZINC000880569771 FF On-Demand Anodyne CYP27B1 40 33 C#CCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569773 CG On-Demand Mild TBXAS1 26 41 C#CCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569774 CG On-Demand Mild TBXAS1 26 41 CCOC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569782 CD On-Demand Anodyne MMP1 15 40 CCOC(=O)c1ncc(CN[C@@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569785 FG On-Demand Anodyne CYP11B1 16 40 CCOC(=O)c1ncc(CN[C@@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569785 FG On-Demand Anodyne TBXAS1 38 40 CCOC(=O)c1ncc(CN[C@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569786 FG On-Demand Anodyne CYP11B1 16 40 CCOC(=O)c1ncc(CN[C@H](Cn2ccnc2)c2ccccc2)s1 ZINC000880569786 FG On-Demand Anodyne TBXAS1 38 40 COc1ccc(CN(CCO)CC(=O)N2CCc3ccccc3C2)cc1 ZINC000880569787 FE On-Demand Anodyne HDAC6 19 40 COc1ccc(CN(CCO)CC(=O)N2CCc3ccccc3C2)cc1 ZINC000880569787 FE On-Demand Anodyne NOD1 15 45 COc1ccc(CN(CCO)CC(=O)N2CCc3ccccc3C2)cc1 ZINC000880569787 FE On-Demand Anodyne NOD2 44 45 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCN(Cc2ccco2)CC1 ZINC000880569791 GE On-Demand Anodyne PTAFR 20 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCN(Cc2ccco2)CC1 ZINC000880569792 GE On-Demand Anodyne PTAFR 20 40 CC(C)(C)OC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569801 EG On-Demand Anodyne TBXAS1 54 42 CC(C)(C)OC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569801 EG On-Demand Anodyne CYP24A1 52 38 CC(C)(C)OC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569801 EG On-Demand Anodyne CYP26A1 87 37 CC(C)(C)OC(=O)NCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569801 EG On-Demand Anodyne CYP27B1 70 38 CC(C)(C)OC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569802 EG On-Demand Anodyne TBXAS1 54 42 CC(C)(C)OC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569802 EG On-Demand Anodyne CYP24A1 52 38 CC(C)(C)OC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569802 EG On-Demand Anodyne CYP26A1 87 37 CC(C)(C)OC(=O)NCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569802 EG On-Demand Anodyne CYP27B1 70 38 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCC2(CC1)OCCO2 ZINC000880569813 FD On-Demand Anodyne PTAFR 17 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCC2(CC1)OCCO2 ZINC000880569814 FD On-Demand Anodyne PTAFR 17 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)Nc1nc2c(s1)CCC2 ZINC000880569855 FF On-Demand Anodyne SLC27A1 33 46 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)Nc1nc2c(s1)CCC2 ZINC000880569856 FF On-Demand Anodyne SLC27A1 33 46 FCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569857 CF On-Demand Anodyne CYP19A1 24 42 FCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569857 CF On-Demand Anodyne CYP11B1 39 42 FCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569857 CF On-Demand Anodyne TBXAS1 36 42 FCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569857 CF On-Demand Anodyne CYP11B2 19 42 FCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880569857 CF On-Demand Anodyne CYP27B1 40 33 FCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569858 CF On-Demand Anodyne CYP19A1 24 42 FCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569858 CF On-Demand Anodyne CYP11B1 39 42 FCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569858 CF On-Demand Anodyne TBXAS1 36 42 FCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569858 CF On-Demand Anodyne CYP11B2 19 42 FCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880569858 CF On-Demand Anodyne CYP27B1 40 33 COC(=O)C1(NC(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CCCCC1 ZINC000880569859 GE On-Demand Anodyne CYP26A1 41 34 COC(=O)C1(NC(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CCCCC1 ZINC000880569860 GE On-Demand Anodyne CYP26A1 41 34 O=C(NCc1cn(C2CCC2)nn1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880569861 FG On-Demand Anodyne C3AR1 42 44 O=C(NCc1cn(C2CCC2)nn1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880569861 FG On-Demand Anodyne NAMPT 41 37 O=C(NCc1cn(C2CCC2)nn1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880569862 FG On-Demand Anodyne C3AR1 42 44 O=C(NCc1cn(C2CCC2)nn1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880569862 FG On-Demand Anodyne NAMPT 41 37 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne CYP11B1 37 44 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne ADRB3 21 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne TBXAS1 39 44 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne CYP11B2 19 44 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne HMOX1 35 41 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569877 DF On-Demand Anodyne CYP27B1 45 37 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne CYP11B1 37 44 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne ADRB3 21 40 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne TBXAS1 39 44 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne CYP11B2 19 44 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne HMOX1 35 41 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569878 DF On-Demand Anodyne CYP27B1 45 37 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne CYP11B1 37 44 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne ADRB3 21 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne TBXAS1 39 44 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne CYP11B2 19 44 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne HMOX1 35 41 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569879 DF On-Demand Anodyne CYP27B1 45 37 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne CYP11B1 37 44 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne ADRB3 21 40 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne TBXAS1 39 44 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne CYP11B2 19 44 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne HMOX1 35 41 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cc1ccccc1 ZINC000880569880 DF On-Demand Anodyne CYP27B1 45 37 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2OC)cc1 ZINC000880569886 FE On-Demand Anodyne TSPO 43 35 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2OC)cc1 ZINC000880569886 FE On-Demand Anodyne MBTPS1 47 41 COc1ccc(CN(CCO)CC(=O)NC(C)C)cc1 ZINC000880569895 CD On-Demand Anodyne MMP13 19 43 COc1ccc(CN(CCO)CC(=O)NC(C)C)cc1 ZINC000880569895 CD On-Demand Anodyne MMP3 27 43 COc1ccc(CN(CCO)CC(=O)NC(C)C)cc1 ZINC000880569895 CD On-Demand Anodyne MMP8 21 43 COc1ccc(CN(CCO)CC(=O)NC(C)C)cc1 ZINC000880569895 CD On-Demand Anodyne MMP12 24 43 COc1ccc(CN(CCO)CC(=O)NC(C)C)cc1 ZINC000880569895 CD On-Demand Anodyne MMP1 32 43 Cc1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)n(C)n1 ZINC000880569903 CE On-Demand Anodyne TBXAS1 24 40 Cc1cc(CN[C@H](Cn2ccnc2)c2ccccc2)n(C)n1 ZINC000880569904 CE On-Demand Anodyne TBXAS1 24 40 COc1ccc(CN(CCO)CCC(=O)Nc2sccc2C#N)cc1 ZINC000880569915 FE On-Demand Mild VIPR1 25 47 COc1ccc(CN(CCO)CC(=O)NC(C)(C)C)cc1 ZINC000880569921 CD On-Demand Anodyne MMP13 16 43 COc1ccc(CN(CCO)CC(=O)NC(C)(C)C)cc1 ZINC000880569921 CD On-Demand Anodyne MMP3 22 45 COc1ccc(CN(CCO)CC(=O)NC(C)(C)C)cc1 ZINC000880569921 CD On-Demand Anodyne MMP9 22 41 COc1ccc(CN(CCO)CC(=O)NC(C)(C)C)cc1 ZINC000880569921 CD On-Demand Anodyne MMP12 21 43 COc1ccc(CN(CCO)CC(=O)NC(C)(C)C)cc1 ZINC000880569921 CD On-Demand Anodyne MMP1 27 43 COc1ccc(CN(CCO)CC(=O)Nc2cc(C)no2)cc1 ZINC000880569936 DD On-Demand Anodyne BMP1 63 37 CCCCNC(=O)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569943 ED On-Demand Anodyne BMP1 41 37 CCCCNC(=O)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569943 ED On-Demand Anodyne MMP3 18 41 CCCCNC(=O)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569943 ED On-Demand Anodyne MMP12 18 41 COc1ccc(CN(CCO)CC(=O)N2CCCC[C@@H]2C)cc1 ZINC000880569947 DD On-Demand Anodyne FKBP1A 21 40 COc1ccc(CN(CCO)CC(=O)N2CCCC[C@H]2C)cc1 ZINC000880569948 DD On-Demand Anodyne FKBP1A 21 40 COc1ccc(CN(CCO)Cc2cccc(NC(C)=O)c2)cc1 ZINC000880569950 EF On-Demand Anodyne BMP1 46 36 COc1ccc(CN(CCO)Cc2cccc(NC(C)=O)c2)cc1 ZINC000880569950 EF On-Demand Anodyne ROCK1 22 42 COc1ccc(CN(CCO)Cc2cccc(NC(C)=O)c2)cc1 ZINC000880569950 EF On-Demand Anodyne MTNR1A 59 43 COc1ccc(CN(CCO)Cc2cccc(NC(C)=O)c2)cc1 ZINC000880569950 EF On-Demand Anodyne MTNR1B 57 43 COc1ccc(CN(CCO)Cc2cccc(NC(C)=O)c2)cc1 ZINC000880569950 EF On-Demand Anodyne ROCK2 27 42 COc1ccc(CN(CCO)CC(=O)N(C)c2ccccc2)cc1 ZINC000880569951 EE On-Demand Anodyne TSPO 23 41 COc1ccc(CN(CCO)CC(=O)N2CCCCCC2)cc1 ZINC000880569952 DD On-Demand Anodyne MMP13 19 42 COc1ccc(CN(CCO)CC(=O)N2CCCCCC2)cc1 ZINC000880569952 DD On-Demand Anodyne MMP3 18 42 COc1ccc(CN(CCO)CC(=O)N2CCCCCC2)cc1 ZINC000880569952 DD On-Demand Anodyne DPP7 22 42 COc1ccc(CN(CCO)CC(=O)N2CCCCCC2)cc1 ZINC000880569952 DD On-Demand Anodyne MMP1 22 42 COc1ccc(CN(CCO)CC(=O)N(C)C2CCCCC2)cc1 ZINC000880569954 EE On-Demand Anodyne AVPR1B 15 40 COc1ccc(CN(CCO)Cc2ccc(OC)c([N+](=O)[O-])c2)cc1 ZINC000880569955 EF On-Demand Bother BMP1 25 41 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne BMP1 58 41 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP13 38 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP2 24 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP3 28 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP8 22 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP9 37 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP12 30 42 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccccc2)cc1 ZINC000880569959 ED On-Demand Anodyne MMP1 32 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C)c2)cc1 ZINC000880569960 EE On-Demand Anodyne MTNR1A 28 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C)c2)cc1 ZINC000880569960 EE On-Demand Anodyne MTNR1B 30 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C)c2)cc1 ZINC000880569960 EE On-Demand Anodyne AKR1C2 16 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C)c2)cc1 ZINC000880569960 EE On-Demand Anodyne KCNK3 69 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C)c2)cc1 ZINC000880569960 EE On-Demand Anodyne KCNK9 55 35 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne BMP1 55 40 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne MMP13 18 41 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne MMP3 24 41 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne MMP8 17 41 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne MMP12 24 41 COc1ccc(CN(CCO)CC(=O)NCC(C)C)cc1 ZINC000880569964 CD On-Demand Anodyne MMP1 30 41 COc1ccc(CN(CCO)CC(N)=O)cc1 ZINC000880569969 BB On-Demand Anodyne MMP12 19 41 COc1ccc(CN(CCO)C[C@@H](O)COc2ccc(C#N)cc2)cc1 ZINC000880569970 FD On-Demand Mild GRIN1 18 45 COc1ccc(CN(CCO)C[C@H](O)COc2ccc(C#N)cc2)cc1 ZINC000880569971 FD On-Demand Mild GRIN1 18 45 COC(=O)CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569973 DB On-Demand Anodyne MMP12 16 42 COC(=O)CNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569973 DB On-Demand Anodyne MMP1 16 42 COC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569979 CC On-Demand Anodyne MMP13 21 44 COC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569979 CC On-Demand Anodyne MMP3 21 44 COC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569979 CC On-Demand Anodyne MMP9 26 40 COC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569979 CC On-Demand Anodyne MMP12 25 44 COC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880569979 CC On-Demand Anodyne MMP1 30 44 COc1ccc(CN(CCO)C[C@H](O)c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880569987 GD On-Demand Anodyne BMP1 52 43 COc1ccc(CN(CCO)C[C@@H](O)c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880569988 GD On-Demand Anodyne BMP1 52 43 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne CYP19A1 18 41 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne CYP11B1 46 41 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne LTA4H 18 50 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne TBXAS1 25 47 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne CYP11B2 22 41 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne CYP2C19 22 40 CCCOc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570009 EI On-Demand Anodyne CYP26A1 41 34 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne CYP19A1 18 41 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne CYP11B1 46 41 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne LTA4H 18 50 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne TBXAS1 25 47 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne CYP11B2 22 41 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne CYP2C19 22 40 CCCOc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880570010 EI On-Demand Anodyne CYP26A1 41 34 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570011 DE On-Demand Anodyne TBXAS1 61 41 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570011 DE On-Demand Anodyne PTAFR 26 45 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570011 DE On-Demand Anodyne CYP24A1 44 36 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570011 DE On-Demand Anodyne CYP26A1 58 36 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570011 DE On-Demand Anodyne CYP27B1 57 36 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570012 DE On-Demand Anodyne TBXAS1 61 41 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570012 DE On-Demand Anodyne PTAFR 26 45 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570012 DE On-Demand Anodyne CYP24A1 44 36 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570012 DE On-Demand Anodyne CYP26A1 58 36 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880570012 DE On-Demand Anodyne CYP27B1 57 36 C[C@@H]1NC(=O)N(CCN[C@H](Cn2ccnc2)c2ccccc2)C1=O ZINC000880570013 ED On-Demand Anodyne CYP27B1 47 32 C[C@@H]1NC(=O)N(CCN[C@@H](Cn2ccnc2)c2ccccc2)C1=O ZINC000880570016 ED On-Demand Anodyne CYP27B1 47 32 C[C@@H](CBr)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570018 DG On-Demand Reactive CYP11B1 33 40 C[C@@H](CBr)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570018 DG On-Demand Reactive TBXAS1 21 40 C[C@@H](CBr)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570018 DG On-Demand Reactive CYP11B2 18 40 C[C@@H](CBr)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570018 DG On-Demand Reactive CYP27B1 43 31 C[C@@H](CBr)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570021 DG On-Demand Reactive CYP11B1 33 40 C[C@@H](CBr)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570021 DG On-Demand Reactive TBXAS1 21 40 C[C@@H](CBr)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570021 DG On-Demand Reactive CYP11B2 18 40 C[C@@H](CBr)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570021 DG On-Demand Reactive CYP27B1 43 31 C#CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570061 CF On-Demand Mild TBXAS1 25 40 C#CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570062 CF On-Demand Mild TBXAS1 25 40 CC(C)(C)C(=O)N1CCC(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570065 FG On-Demand Anodyne GRIN2B 21 43 CC(C)(C)C(=O)N1CCC(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570065 FG On-Demand Anodyne TBXAS1 43 38 CC(C)(C)C(=O)N1CCC(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570065 FG On-Demand Anodyne CYP26A1 45 35 CC(C)(C)C(=O)N1CCC(CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570065 FG On-Demand Anodyne CYP27B1 40 33 CC(C)(C)C(=O)N1CCC(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570066 FG On-Demand Anodyne GRIN2B 21 43 CC(C)(C)C(=O)N1CCC(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570066 FG On-Demand Anodyne TBXAS1 43 38 CC(C)(C)C(=O)N1CCC(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570066 FG On-Demand Anodyne CYP26A1 45 35 CC(C)(C)C(=O)N1CCC(CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880570066 FG On-Demand Anodyne CYP27B1 40 33 CCOC(=O)c1csc(CN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570071 FG On-Demand Anodyne TBXAS1 35 40 CCOC(=O)c1csc(CN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570072 FG On-Demand Anodyne TBXAS1 35 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(Cl)c2)cc1 ZINC000880570089 EF On-Demand Anodyne LTA4H 20 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(Cl)c2)cc1 ZINC000880570089 EF On-Demand Anodyne MMP1 15 42 COc1ccc(CN(CCO)Cc2nc3ccccc3[nH]2)cc1 ZINC000880570094 DF On-Demand Anodyne CXCR4 35 42 COc1ccc(CN(CCO)Cc2nc3ccccc3[nH]2)cc1 ZINC000880570094 DF On-Demand Anodyne ALKBH3 26 40 COc1ccc(CN(CCO)CC2CCCC2)cc1 ZINC000880570103 CF On-Demand Anodyne SLC18A2 19 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C)c(F)c2)cc1 ZINC000880570104 EF On-Demand Anodyne LTA4H 22 41 COc1ccc(CN(CCO)Cc2csc(C3CCCC3)n2)cc1 ZINC000880570106 EH On-Demand Anodyne AVPR1B 18 45 COc1ccc(CN(CCO)CCOc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880570109 EE On-Demand Bother MMP2 17 49 COc1ccc(CN(CCO)CCOc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880570109 EE On-Demand Bother MMP8 34 49 COc1ccc(CN(CCO)CCOc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880570109 EE On-Demand Bother MMP9 24 49 COc1ccc(CN(CCO)CCOc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880570109 EE On-Demand Bother MMP1 25 49 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne BMP1 94 41 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP13 30 43 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP3 18 43 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP8 15 40 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP9 32 43 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP12 24 40 COc1ccc(CN(CCO)Cc2cccc(S(=O)(=O)N(C)C)c2)cc1 ZINC000880570111 GD On-Demand Anodyne MMP1 28 43 CCOC(=O)[C@@H]1CCCCN1C(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570117 GD On-Demand Anodyne FKBP1A 95 48 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N3CCCC3)o2)cc1 ZINC000880570120 GE On-Demand Anodyne LPL 26 42 COc1ccc(CN(CCO)CCOc2cccc(C#N)c2)cc1 ZINC000880570125 EE On-Demand Mild SQLE 41 35 CCOC(=O)N1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570126 GD On-Demand Anodyne MMP13 21 45 CCOC(=O)N1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570126 GD On-Demand Anodyne MMP3 21 45 CCOC(=O)N1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570126 GD On-Demand Anodyne MMP9 19 45 CCOC(=O)N1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570126 GD On-Demand Anodyne MCHR1 18 43 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(F)c2)cc1 ZINC000880570128 EF On-Demand Anodyne BMP1 20 40 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(F)c2)cc1 ZINC000880570128 EF On-Demand Anodyne AURKB 24 40 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(F)c2)cc1 ZINC000880570128 EF On-Demand Anodyne MTNR1A 21 40 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(F)c2)cc1 ZINC000880570128 EF On-Demand Anodyne MTNR1B 23 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(F)cc2)cc1 ZINC000880570132 EF On-Demand Anodyne LTA4H 35 48 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(F)cc2)cc1 ZINC000880570132 EF On-Demand Anodyne BMP1 19 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(F)cc2)cc1 ZINC000880570132 EF On-Demand Anodyne MTNR1B 15 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(F)cc2)cc1 ZINC000880570132 EF On-Demand Anodyne NPY5R 17 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(F)cc2)cc1 ZINC000880570132 EF On-Demand Anodyne CA9 15 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)[C@H]1CC[C@@H](C(F)(F)F)CC1 ZINC000880570133 GI On-Demand Anodyne TBXAS1 42 39 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)[C@H]1CC[C@@H](C(F)(F)F)CC1 ZINC000880570134 GI On-Demand Anodyne TBXAS1 42 39 COC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570142 CD On-Demand Anodyne BMP1 45 38 COC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570142 CD On-Demand Anodyne MMP13 15 40 COC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570142 CD On-Demand Anodyne MMP3 15 40 COC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570142 CD On-Demand Anodyne MMP12 20 40 COC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570142 CD On-Demand Anodyne MMP1 24 40 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP13 18 41 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP3 24 41 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP8 15 40 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP9 17 41 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP12 18 40 COc1ccc(CN(CCO)CC(=O)NC2CCCC2)cc1 ZINC000880570147 DD On-Demand Anodyne MMP1 21 41 C=CCNC(=O)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570148 DC On-Demand Mild MMP3 17 41 C=CCNC(=O)NC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570148 DC On-Demand Mild MMP12 18 41 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2C)cc1 ZINC000880570153 EE On-Demand Anodyne BMP1 41 34 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2C)cc1 ZINC000880570153 EE On-Demand Anodyne MMP13 18 40 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2C)cc1 ZINC000880570153 EE On-Demand Anodyne MMP9 21 40 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2C)cc1 ZINC000880570153 EE On-Demand Anodyne MMP12 20 40 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2C)cc1 ZINC000880570153 EE On-Demand Anodyne MMP1 23 40 COc1ccc(CN(CCO)Cc2cccc(C(=O)N3CCCCC3)c2)cc1 ZINC000880570154 GG On-Demand Anodyne TRY2_BOVIN 43 34 COc1ccc(CN(CCO)Cc2cccc(C(=O)N3CCCCC3)c2)cc1 ZINC000880570154 GG On-Demand Anodyne PARP1 15 42 COc1ccc(CN(CCO)Cc2cccc(C(=O)N3CCCCC3)c2)cc1 ZINC000880570154 GG On-Demand Anodyne DPP7 20 41 COc1ccc(CN(CCO)Cc2cccc(C(=O)N3CCCCC3)c2)cc1 ZINC000880570154 GG On-Demand Anodyne HPGD 31 43 COc1ccc(CN(CCO)CC(=O)N2CCCCC2)cc1 ZINC000880570155 DD On-Demand Anodyne MMP13 19 42 COc1ccc(CN(CCO)CC(=O)N2CCCCC2)cc1 ZINC000880570155 DD On-Demand Anodyne MMP3 18 42 COc1ccc(CN(CCO)CC(=O)N2CCCCC2)cc1 ZINC000880570155 DD On-Demand Anodyne DPP7 22 42 COc1ccc(CN(CCO)CC(=O)N2CCCCC2)cc1 ZINC000880570155 DD On-Demand Anodyne MMP1 22 42 COc1ccc(CN(CCO)Cc2noc(-c3ccccc3)n2)cc1 ZINC000880570156 EF On-Demand Anodyne PPARG 15 43 COc1ccc(CN(CCO)Cc2noc(-c3ccccc3)n2)cc1 ZINC000880570156 EF On-Demand Anodyne PPARA 19 40 COc1ccc(CN(CCO)CCC(=O)NC2CCCC2)cc1 ZINC000880570166 DD On-Demand Anodyne BMP1 20 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCC(F)(F)F)cc1 ZINC000880570168 FC On-Demand Anodyne MMP12 16 41 COC(=O)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570170 DF On-Demand Anodyne CYP19A1 22 42 COC(=O)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570170 DF On-Demand Anodyne TBXAS1 73 45 COC(=O)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570170 DF On-Demand Anodyne CYP24A1 51 37 COC(=O)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570170 DF On-Demand Anodyne CYP26A1 94 41 COC(=O)CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570170 DF On-Demand Anodyne CYP27B1 68 37 COC(=O)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570171 DF On-Demand Anodyne CYP19A1 22 42 COC(=O)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570171 DF On-Demand Anodyne TBXAS1 73 45 COC(=O)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570171 DF On-Demand Anodyne CYP24A1 51 37 COC(=O)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570171 DF On-Demand Anodyne CYP26A1 94 41 COC(=O)CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570171 DF On-Demand Anodyne CYP27B1 68 37 COc1ccc(CN(CCO)Cc2cccc3cccnc23)cc1 ZINC000880570174 DG On-Demand Anodyne PDE4C 17 40 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne PPARG 15 40 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne PPARA 17 40 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne LTA4H 44 50 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne ERG2 17 41 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne ESRRG 48 38 COc1ccc(CN(CCO)CCOc2ccccc2)cc1 ZINC000880570177 DF On-Demand Anodyne TAAR1 15 40 CC(C)(C)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570178 DE On-Demand Anodyne TBXAS1 55 41 CC(C)(C)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570178 DE On-Demand Anodyne CYP24A1 49 38 CC(C)(C)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570178 DE On-Demand Anodyne CYP26A1 50 38 CC(C)(C)CNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570178 DE On-Demand Anodyne CYP27B1 65 38 CC(C)(C)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570179 DE On-Demand Anodyne TBXAS1 55 41 CC(C)(C)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570179 DE On-Demand Anodyne CYP24A1 49 38 CC(C)(C)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570179 DE On-Demand Anodyne CYP26A1 50 38 CC(C)(C)CNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570179 DE On-Demand Anodyne CYP27B1 65 38 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCCO3)cc1 ZINC000880570184 FD On-Demand Anodyne EDNRB 40 38 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCCO3)cc1 ZINC000880570184 FD On-Demand Anodyne EDNRA 36 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCCO3)cc1 ZINC000880570184 FD On-Demand Anodyne BMP1 70 36 CCCS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570187 DD On-Demand Anodyne MMP13 18 40 CCCS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570187 DD On-Demand Anodyne MMP3 15 40 CCCS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570187 DD On-Demand Anodyne MMP12 20 40 CCCS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570187 DD On-Demand Anodyne MMP1 17 40 C#CCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570193 CD On-Demand Mild TBXAS1 52 41 C#CCNC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570193 CD On-Demand Mild CYP27B1 42 36 C#CCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570194 CD On-Demand Mild TBXAS1 52 41 C#CCNC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570194 CD On-Demand Mild CYP27B1 42 36 c1ccc([C@@H](Cn2ccnc2)NCCCc2ccsc2)cc1 ZINC000880570199 DH On-Demand Anodyne CYP11B1 29 41 c1ccc([C@H](Cn2ccnc2)NCCCc2ccsc2)cc1 ZINC000880570200 DH On-Demand Anodyne CYP11B1 29 41 Cn1ncc(CN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570201 CD On-Demand Anodyne TBXAS1 28 40 Cn1ncc(CN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570202 CD On-Demand Anodyne TBXAS1 28 40 CC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570204 CF On-Demand Anodyne CYP19A1 19 42 CC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570204 CF On-Demand Anodyne CYP11B1 38 44 CC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570204 CF On-Demand Anodyne CYP11B2 19 44 CC[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570204 CF On-Demand Anodyne CYP27B1 48 33 CC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570206 CF On-Demand Anodyne CYP19A1 19 42 CC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570206 CF On-Demand Anodyne CYP11B1 38 44 CC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570206 CF On-Demand Anodyne CYP11B2 19 44 CC[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)OC ZINC000880570206 CF On-Demand Anodyne CYP27B1 48 33 O=S1(=O)CCCN1CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570207 ED On-Demand Anodyne TBXAS1 27 40 O=S1(=O)CCCN1CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570208 ED On-Demand Anodyne TBXAS1 27 40 CN1C(=O)CCc2cc(CN[C@@H](Cn3ccnc3)c3ccccc3)ccc21 ZINC000880570209 FG On-Demand Anodyne CYP11B1 25 41 CN1C(=O)CCc2cc(CN[C@@H](Cn3ccnc3)c3ccccc3)ccc21 ZINC000880570209 FG On-Demand Anodyne CYP11B2 17 41 CN1C(=O)CCc2cc(CN[C@H](Cn3ccnc3)c3ccccc3)ccc21 ZINC000880570210 FG On-Demand Anodyne CYP11B1 25 41 CN1C(=O)CCc2cc(CN[C@H](Cn3ccnc3)c3ccccc3)ccc21 ZINC000880570210 FG On-Demand Anodyne CYP11B2 17 41 CCC[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570212 CE On-Demand Anodyne TBXAS1 30 42 CCC[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570212 CE On-Demand Anodyne HMOX1 30 41 CCC[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570212 CE On-Demand Anodyne CYP27B1 43 32 CCC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570213 CE On-Demand Anodyne TBXAS1 30 42 CCC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570213 CE On-Demand Anodyne HMOX1 30 41 CCC[C@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570213 CE On-Demand Anodyne CYP27B1 43 32 CCC[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570214 CE On-Demand Anodyne TBXAS1 30 42 CCC[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570214 CE On-Demand Anodyne HMOX1 30 41 CCC[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570214 CE On-Demand Anodyne CYP27B1 43 32 CCC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570215 CE On-Demand Anodyne TBXAS1 30 42 CCC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570215 CE On-Demand Anodyne HMOX1 30 41 CCC[C@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570215 CE On-Demand Anodyne CYP27B1 43 32 FCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570239 CG On-Demand Anodyne CYP19A1 21 41 FCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570239 CG On-Demand Anodyne CYP11B1 37 41 FCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570239 CG On-Demand Anodyne TBXAS1 38 44 FCCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570239 CG On-Demand Anodyne CYP11B2 18 41 FCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570240 CG On-Demand Anodyne CYP19A1 21 41 FCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570240 CG On-Demand Anodyne CYP11B1 37 41 FCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570240 CG On-Demand Anodyne TBXAS1 38 44 FCCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570240 CG On-Demand Anodyne CYP11B2 18 41 FC(F)(Br)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570241 EG On-Demand Anodyne CYP19A1 18 41 FC(F)(Br)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570241 EG On-Demand Anodyne CYP11B1 37 41 FC(F)(Br)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570241 EG On-Demand Anodyne TBXAS1 31 41 FC(F)(Br)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570241 EG On-Demand Anodyne CYP11B2 18 41 FC(F)(Br)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570241 EG On-Demand Anodyne CYP27B1 54 32 FC(F)(Br)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570242 EG On-Demand Anodyne CYP19A1 18 41 FC(F)(Br)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570242 EG On-Demand Anodyne CYP11B1 37 41 FC(F)(Br)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570242 EG On-Demand Anodyne TBXAS1 31 41 FC(F)(Br)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570242 EG On-Demand Anodyne CYP11B2 18 41 FC(F)(Br)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570242 EG On-Demand Anodyne CYP27B1 54 32 O=C(NCc1cn(C2CCC2)nn1)c1cccc(Oc2ccc(Cl)cn2)c1 ZINC000880570243 GH On-Demand Anodyne DRD4 41 34 COc1ccc(CN(CCO)C[C@@H](O)c2ccc(F)c(F)c2)cc1 ZINC000880570259 EF On-Demand Anodyne AOC3 16 42 COc1ccc(CN(CCO)C[C@H](O)c2ccc(F)c(F)c2)cc1 ZINC000880570261 EF On-Demand Anodyne AOC3 16 42 COc1cc(C)nc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570264 DG On-Demand Anodyne CYP19A1 19 41 COc1cc(C)nc(CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570266 DG On-Demand Anodyne CYP19A1 19 41 Cc1oncc1CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570276 CF On-Demand Anodyne CYP11B1 49 41 Cc1oncc1CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570276 CF On-Demand Anodyne CYP11B2 25 41 Cc1oncc1CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570278 CF On-Demand Anodyne CYP11B1 49 41 Cc1oncc1CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570278 CF On-Demand Anodyne CYP11B2 25 41 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne BMP1 47 40 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne MMP13 24 41 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne MMP3 25 41 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne MMP8 21 41 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne MMP12 24 41 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C(C)C)cc1 ZINC000880570287 DE On-Demand Anodyne MMP1 28 41 CN(C)C(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570292 DE On-Demand Anodyne TBXAS1 63 45 CN(C)C(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570292 DE On-Demand Anodyne CYP24A1 40 35 CN(C)C(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570292 DE On-Demand Anodyne CYP26A1 101 37 CN(C)C(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570292 DE On-Demand Anodyne CYP27B1 52 35 CN(C)C(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570293 DE On-Demand Anodyne TBXAS1 63 45 CN(C)C(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570293 DE On-Demand Anodyne CYP24A1 40 35 CN(C)C(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570293 DE On-Demand Anodyne CYP26A1 101 37 CN(C)C(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570293 DE On-Demand Anodyne CYP27B1 52 35 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne CYP19A1 26 41 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne CYP11B1 41 41 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne TBXAS1 31 41 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne CYP11B2 22 41 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne CYP24A1 46 34 CO[C@@H](C)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570294 CE On-Demand Anodyne CYP27B1 61 34 COc1ccc(CN(CCO)CC(=O)N2CCOCC2)cc1 ZINC000880570295 DC On-Demand Anodyne BMP1 26 41 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne CYP19A1 26 41 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne CYP11B1 41 41 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne TBXAS1 31 41 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne CYP11B2 22 41 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne CYP24A1 46 34 CO[C@@H](C)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570298 CE On-Demand Anodyne CYP27B1 61 34 COc1ccc(CN(CCO)CCC(=O)N2CCN(c3ccccn3)CC2)cc1 ZINC000880570300 GD On-Demand Anodyne DRD4 28 41 COc1ccc(CN(CCO)CCC(=O)N2CCN(c3ccccn3)CC2)cc1 ZINC000880570300 GD On-Demand Anodyne EBP 21 42 COc1ccc(CN(CCO)CCC(=O)N2CCN(c3ccccn3)CC2)cc1 ZINC000880570300 GD On-Demand Anodyne SSTR1 47 37 COc1ccc(CN(CCO)CC(=O)NCC2CC2)cc1 ZINC000880570302 CD On-Demand Anodyne MMP13 18 40 COc1ccc(CN(CCO)CC(=O)NCC2CC2)cc1 ZINC000880570302 CD On-Demand Anodyne MMP3 22 40 COc1ccc(CN(CCO)CC(=O)NCC2CC2)cc1 ZINC000880570302 CD On-Demand Anodyne MMP8 15 40 COc1ccc(CN(CCO)CC(=O)NCC2CC2)cc1 ZINC000880570302 CD On-Demand Anodyne MMP12 16 40 COc1ccc(CN(CCO)CC(=O)NCC2CC2)cc1 ZINC000880570302 CD On-Demand Anodyne MMP1 21 40 COc1ccc(CN(CCO)Cc2cccc(OC)c2)cc1 ZINC000880570309 DF On-Demand Anodyne G6PC 26 41 COc1ccc(CN(CCO)Cc2cccc(OC)c2)cc1 ZINC000880570309 DF On-Demand Anodyne ROCK1 30 43 COc1ccc(CN(CCO)Cc2cccc(OC)c2)cc1 ZINC000880570309 DF On-Demand Anodyne ROCK2 36 43 COc1ccc(CN(CCO)Cc2cccc(OC)c2)cc1 ZINC000880570309 DF On-Demand Anodyne AOC3 15 47 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne BMP1 30 43 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne MMP13 19 40 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne MMP3 15 40 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne MMP12 20 40 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne ACR 50 41 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880570312 EE On-Demand Anodyne MMP1 24 41 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C[C@H](O)c1ccccc1 ZINC000880570315 FF On-Demand Anodyne TBXAS1 34 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C[C@H](O)c1ccccc1 ZINC000880570315 FF On-Demand Anodyne CYP27B1 44 33 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C[C@H](O)c1ccccc1 ZINC000880570316 FF On-Demand Anodyne TBXAS1 34 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C[C@H](O)c1ccccc1 ZINC000880570316 FF On-Demand Anodyne CYP27B1 44 33 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C[C@@H](O)c1ccccc1 ZINC000880570317 FF On-Demand Anodyne TBXAS1 34 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)C[C@@H](O)c1ccccc1 ZINC000880570317 FF On-Demand Anodyne CYP27B1 44 33 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C[C@@H](O)c1ccccc1 ZINC000880570318 FF On-Demand Anodyne TBXAS1 34 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)C[C@@H](O)c1ccccc1 ZINC000880570318 FF On-Demand Anodyne CYP27B1 44 33 CCOC(=O)C1CCN(C(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570326 GD On-Demand Anodyne PTR1 46 36 COc1ccc(CN(CCO)CC(=O)c2cn(CCC#N)c3ccccc23)cc1 ZINC000880570337 GG On-Demand Mild CNR1 15 45 COc1ccc(CN(CCO)CC(=O)c2cn(CCC#N)c3ccccc23)cc1 ZINC000880570337 GG On-Demand Mild CNR2 21 54 COc1ccc(CN(CCO)CCS(C)(=O)=O)cc1 ZINC000880570339 CC On-Demand Anodyne BMP1 46 38 COc1ccc(CN(CCO)CCS(C)(=O)=O)cc1 ZINC000880570339 CC On-Demand Anodyne MMP13 18 43 COc1ccc(CN(CCO)CCS(C)(=O)=O)cc1 ZINC000880570339 CC On-Demand Anodyne MMP3 15 40 COc1ccc(CN(CCO)CCS(C)(=O)=O)cc1 ZINC000880570339 CC On-Demand Anodyne MMP12 21 43 COc1ccc(CN(CCO)CCS(C)(=O)=O)cc1 ZINC000880570339 CC On-Demand Anodyne MMP1 17 40 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)c2cccs2)cc1 ZINC000880570341 EE On-Demand Anodyne BMP1 48 39 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2cccs2)cc1 ZINC000880570342 EE On-Demand Anodyne BMP1 48 39 C#CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570343 CC On-Demand Mild MMP12 18 41 COC(=O)c1cccc(CN(CCO)Cc2ccc(OC)cc2)c1 ZINC000880570354 EE On-Demand Anodyne BMP1 46 39 COC(=O)c1cccc(CN(CCO)Cc2ccc(OC)cc2)c1 ZINC000880570354 EE On-Demand Anodyne MMP13 24 42 COc1ccc(CN(CCO)CCC(=O)N2CCOCC2)cc1 ZINC000880570358 DC On-Demand Anodyne BMP1 41 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2cccs2)cc1 ZINC000880570366 GD On-Demand Anodyne BMP1 55 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(F)c2)cc1 ZINC000880570368 EE On-Demand Anodyne LTA4H 20 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(F)c2)cc1 ZINC000880570368 EE On-Demand Anodyne BMP1 20 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(F)c2)cc1 ZINC000880570368 EE On-Demand Anodyne AURKB 38 44 COc1ccc(CN(CCO)CC(=O)Nc2cccc(F)c2)cc1 ZINC000880570368 EE On-Demand Anodyne AURKA 20 40 COc1ccc(CN(CCO)Cc2nnc(-c3ccccc3)o2)cc1 ZINC000880570369 EF On-Demand Anodyne PPARA 21 41 COc1ccc(CN(CCO)CC(=O)NCC2CCCCC2)cc1 ZINC000880570370 EE On-Demand Anodyne MMP3 20 44 CNC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570373 CC On-Demand Anodyne BMP1 31 42 CNC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570373 CC On-Demand Anodyne MMP3 15 42 CNC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570373 CC On-Demand Anodyne MMP12 21 42 CNC(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880570373 CC On-Demand Anodyne MMP1 24 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne ACHE 16 50 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne ROCK1 30 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne MTNR1A 38 41 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne MTNR1B 36 41 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne ROCK2 36 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cccc(OC)c2)cc1 ZINC000880570378 FE On-Demand Anodyne HSD17B2 27 51 c1ccc([C@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570381 CC On-Demand Anodyne CYP19A1 22 40 c1ccc([C@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570381 CC On-Demand Anodyne CYP11B1 36 40 c1ccc([C@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570381 CC On-Demand Anodyne TBXAS1 27 40 c1ccc([C@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570381 CC On-Demand Anodyne CYP11B2 17 40 c1ccc([C@@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570382 CC On-Demand Anodyne CYP19A1 22 40 c1ccc([C@@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570382 CC On-Demand Anodyne CYP11B1 36 40 c1ccc([C@@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570382 CC On-Demand Anodyne TBXAS1 27 40 c1ccc([C@@H](Cn2ccnc2)NCCn2cnnn2)cc1 ZINC000880570382 CC On-Demand Anodyne CYP11B2 17 40 COC(=O)c1occc1CN(CCO)Cc1ccc(OC)cc1 ZINC000880570384 DE On-Demand Anodyne MMP12 18 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC(C)(C)C)cc1 ZINC000880570385 ED On-Demand Anodyne MMP13 21 43 COc1ccc(CN(CCO)CC(=O)NC(=O)NC(C)(C)C)cc1 ZINC000880570385 ED On-Demand Anodyne MMP3 21 43 COc1ccc(CN(CCO)CC(=O)NC(=O)NC(C)(C)C)cc1 ZINC000880570385 ED On-Demand Anodyne MMP8 15 43 COc1ccc(CN(CCO)CC(=O)NC(=O)NC(C)(C)C)cc1 ZINC000880570385 ED On-Demand Anodyne MMP12 22 43 COc1ccc(CN(CCO)CC(=O)NC(=O)NC(C)(C)C)cc1 ZINC000880570385 ED On-Demand Anodyne MMP1 26 43 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne HRH3 15 41 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne MMP13 19 40 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne SLC18A3 16 42 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne DPP7 16 40 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne MMP1 19 40 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne L3MBTL3 62 38 COc1ccc(CN(CCO)Cc2ccc(C(=O)N3CCCC3)cc2)cc1 ZINC000880570388 FF On-Demand Anodyne HPGD 21 43 COc1ccc(CN(CCO)CC(=O)NCc2ccc3c(c2)OCO3)cc1 ZINC000880570390 FD On-Demand Anodyne EDNRB 89 41 COc1ccc(CN(CCO)CC(=O)NCc2ccc3c(c2)OCO3)cc1 ZINC000880570390 FD On-Demand Anodyne EDNRA 88 43 COc1ccc(CN(CCO)CC(=O)NCc2ccc3c(c2)OCO3)cc1 ZINC000880570390 FD On-Demand Anodyne BMP1 82 46 COc1ccc(CN(CCO)CC(=O)NCc2ccc3c(c2)OCO3)cc1 ZINC000880570390 FD On-Demand Anodyne NOS2 97 37 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne BMP1 69 46 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP13 47 47 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP2 25 41 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP3 27 44 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP8 28 44 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP9 43 47 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP12 28 44 COc1ccc(CN(CCO)CCOc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880570391 GD On-Demand Anodyne MMP1 35 47 COc1ccc(CN(CCO)CC(=O)Nc2cc(C)cc(C)c2)cc1 ZINC000880570412 EF On-Demand Anodyne MMP9 15 40 COc1ccc(CN(CCO)CC(=O)Nc2cc(C)cc(C)c2)cc1 ZINC000880570412 EF On-Demand Anodyne MMP12 15 40 COc1ccc(CN(CCO)CC(=O)Nc2cc(C)cc(C)c2)cc1 ZINC000880570412 EF On-Demand Anodyne MMP1 17 40 COc1ccc(CN(CCO)CCS(=O)(=O)C(C)C)cc1 ZINC000880570420 DD On-Demand Anodyne BMP1 42 40 COc1ccc(CN(CCO)CCCS(N)(=O)=O)cc1 ZINC000880570427 DC On-Demand Anodyne MMP13 21 41 COc1ccc(CN(CCO)CCCS(N)(=O)=O)cc1 ZINC000880570427 DC On-Demand Anodyne MMP3 17 41 COc1ccc(CN(CCO)CCCS(N)(=O)=O)cc1 ZINC000880570427 DC On-Demand Anodyne MMP12 22 41 COc1ccc(CN(CCO)CCCS(N)(=O)=O)cc1 ZINC000880570427 DC On-Demand Anodyne MMP1 21 41 COc1ccc(CN(CCO)CC(=O)Nc2nc3c(s2)CCC3)cc1 ZINC000880570429 FE On-Demand Anodyne CSNK1D 18 40 COc1ccc(CN(CCO)CC(=O)Nc2nc3c(s2)CCC3)cc1 ZINC000880570429 FE On-Demand Anodyne SLC27A1 39 43 COc1ccc(CN(CCO)CC(=O)N(C(C)C)C2CCCC2)cc1 ZINC000880570431 EF On-Demand Anodyne AVPR1B 15 41 CCOC[C@H](O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570435 CC On-Demand Anodyne GRIN1 15 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C(C)=O)c2)cc1 ZINC000880570437 FE On-Demand Anodyne LTA4H 21 41 O=C(Cc1ccc(Br)cc1Cl)NCc1cn(C2CCC2)nn1 ZINC000880570448 GG On-Demand Anodyne P2RX7 42 40 COc1ccc(CN(CCO)Cc2nc(O)c3ccc(Cl)cc3n2)cc1 ZINC000880570449 FF On-Demand Anodyne HRP1_PLAFA 23 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2C#N)cc1 ZINC000880570453 FE On-Demand Mild VIPR1 22 41 COc1ccc(CN(CCO)CCCNC(=O)C(F)(F)F)cc1 ZINC000880570454 ED On-Demand Anodyne MTNR1A 18 42 COc1ccc(CN(CCO)Cc2ccn(C(C)C)n2)cc1 ZINC000880570458 DE On-Demand Anodyne PROKR1 41 30 COc1ccc(CN(CCO)Cc2csc(CS(C)(=O)=O)n2)cc1 ZINC000880570460 FD On-Demand Anodyne AVPR1B 15 41 COc1ccc(CN(CCO)Cc2nc3ccccc3c(=O)n2C)cc1 ZINC000880570461 FD On-Demand Anodyne TSPO 17 41 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880570468 FG On-Demand Anodyne CYP27B1 44 33 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc2C1 ZINC000880570469 FG On-Demand Anodyne CYP27B1 44 33 COc1ccc(CN(CCO)CC(=O)Nc2nncs2)cc1 ZINC000880570470 DC On-Demand Anodyne CA9 15 40 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(C)ccc23)cc1 ZINC000880570475 FG On-Demand Anodyne CYP11B1 15 42 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(C)ccc23)cc1 ZINC000880570475 FG On-Demand Anodyne MAOB 36 40 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(NC(C)=O)ccc23)cc1 ZINC000880570487 GF On-Demand Anodyne CYP11B1 15 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCCC3)cc2)cc1 ZINC000880570493 GF On-Demand Anodyne LTA4H 26 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCCC3)cc2)cc1 ZINC000880570493 GF On-Demand Anodyne KCNQ2 17 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cn2)cc1 ZINC000880570497 EE On-Demand Anodyne KLKB1 20 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cn2)cc1 ZINC000880570497 EE On-Demand Anodyne F10 53 37 COc1ccc(CN(CCO)CC(=O)Nc2cc(OC)cc(OC)c2)cc1 ZINC000880570512 FE On-Demand Anodyne LTA4H 19 40 COc1ccc(CN(CCO)CC(=O)Nc2cc(OC)cc(OC)c2)cc1 ZINC000880570512 FE On-Demand Anodyne MTNR1B 28 41 COc1ccc(CN(CCO)CC(=O)Nc2cc(OC)cc(OC)c2)cc1 ZINC000880570512 FE On-Demand Anodyne MMP12 16 41 COc1ccc(CN(CCO)CC(=O)Nc2cc(OC)cc(OC)c2)cc1 ZINC000880570512 FE On-Demand Anodyne CA9 16 40 COc1ccc(CN(CCO)CC(=O)Nc2cc(OC)cc(OC)c2)cc1 ZINC000880570512 FE On-Demand Anodyne MMP1 17 41 Brc1ncn(CCN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570513 FE On-Demand Anodyne CYP19A1 18 40 Brc1ncn(CCN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570513 FE On-Demand Anodyne CYP11B1 43 40 Brc1ncn(CCN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570513 FE On-Demand Anodyne TBXAS1 28 40 Brc1ncn(CCN[C@@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570513 FE On-Demand Anodyne CYP11B2 20 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2cccc(OC)c2)cc1 ZINC000880570514 GD On-Demand Anodyne BMP1 45 36 COc1ccc(CN(CCO)CCS(=O)(=O)c2cccc(OC)c2)cc1 ZINC000880570514 GD On-Demand Anodyne MMP3 16 40 Brc1ncn(CCN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570515 FE On-Demand Anodyne CYP19A1 18 40 Brc1ncn(CCN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570515 FE On-Demand Anodyne CYP11B1 43 40 Brc1ncn(CCN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570515 FE On-Demand Anodyne TBXAS1 28 40 Brc1ncn(CCN[C@H](Cn2ccnc2)c2ccccc2)n1 ZINC000880570515 FE On-Demand Anodyne CYP11B2 20 40 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne CYP19A1 15 40 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne CYP11B1 34 40 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne TBXAS1 37 41 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne CYP11B2 19 40 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne CYP24A1 41 33 C[C@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570527 CD On-Demand Anodyne CYP27B1 54 33 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne CYP19A1 15 40 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne CYP11B1 34 40 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne TBXAS1 37 41 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne CYP11B2 19 40 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne CYP24A1 41 33 C[C@@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570528 CD On-Demand Anodyne CYP27B1 54 33 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne CYP19A1 15 40 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne CYP11B1 34 40 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne TBXAS1 37 41 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne CYP11B2 19 40 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne CYP24A1 41 33 C[C@@H](CO)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570529 CD On-Demand Anodyne CYP27B1 54 33 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne CYP19A1 15 40 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne CYP11B1 34 40 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne TBXAS1 37 41 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne CYP11B2 19 40 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne CYP24A1 41 33 C[C@H](CO)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570530 CD On-Demand Anodyne CYP27B1 54 33 COc1ccc(CN(CCO)[C@H]2C=CCCC2)cc1 ZINC000880570539 CF On-Demand Anodyne SLC18A2 21 41 COc1ccc(CN(CCO)[C@@H]2C=CCCC2)cc1 ZINC000880570540 CF On-Demand Anodyne SLC18A2 21 41 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)(C)C)cc1 ZINC000880570555 EC On-Demand Reactive MMP12 18 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)(C)C)cc1 ZINC000880570555 EC On-Demand Reactive MMP1 18 40 COC[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570571 CD On-Demand Anodyne CYP19A1 18 43 COC[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570571 CD On-Demand Anodyne CYP27B1 40 34 COC[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570573 CD On-Demand Anodyne CYP19A1 18 43 COC[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570573 CD On-Demand Anodyne CYP27B1 40 34 O=C(NCc1cn(C2CCC2)nn1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880570584 EE On-Demand Anodyne GABRA1 15 49 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2C(F)(F)F)cc1 ZINC000880570592 GG On-Demand Anodyne BMP1 22 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2Cl)cc1 ZINC000880570597 FG On-Demand Anodyne CA9 15 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne BMP1 64 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP13 29 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne CA4 19 46 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MTNR1B 22 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP2 20 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP3 24 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP8 27 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP9 34 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP12 25 42 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne CA9 19 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570600 GD On-Demand Anodyne MMP1 30 42 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2F)cc1 ZINC000880570601 EE On-Demand Anodyne GRIN1 18 41 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2F)cc1 ZINC000880570602 EE On-Demand Anodyne GRIN1 18 41 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccc(OC)cc2)cc1 ZINC000880570603 FE On-Demand Anodyne MMP12 15 40 COc1ccc(CN(CCO)CC(=O)NCc2ccc(C)cc2)cc1 ZINC000880570605 EE On-Demand Anodyne MMP13 16 40 COc1ccc(CN(CCO)CC(=O)NCc2ccc(C)cc2)cc1 ZINC000880570605 EE On-Demand Anodyne MMP12 17 40 COc1ccc(CN(CCO)CC(=O)NCc2ccc(C)cc2)cc1 ZINC000880570605 EE On-Demand Anodyne CA9 15 44 COc1ccc(CN(CCO)Cc2nc(-c3ccco3)no2)cc1 ZINC000880570618 EE On-Demand Anodyne ADORA2A 16 41 CCOC(=O)N1CCN(C(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570619 GC On-Demand Anodyne BMP1 19 42 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP19A1 29 42 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP11B1 43 41 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne TBXAS1 74 50 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP11B2 23 41 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP24A1 48 36 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP26A1 50 36 CC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570624 BD On-Demand Anodyne CYP27B1 64 36 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP19A1 29 42 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP11B1 43 41 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne TBXAS1 74 50 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP11B2 23 41 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP24A1 48 36 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP26A1 50 36 CC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570625 BD On-Demand Anodyne CYP27B1 64 36 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne LTA4H 27 40 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne MMP13 20 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne MMP3 22 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne NPY5R 15 40 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne MMP9 25 42 COc1ccc(CN(CCO)CC(=O)N(C)Cc2ccccc2)cc1 ZINC000880570626 EE On-Demand Anodyne MMP1 24 42 C=CCNC(=O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880570627 CC On-Demand Mild MMP12 16 41 COc1ccc(CN(CCO)C[C@@H](O)CN2CCCC2)cc1 ZINC000880570630 DC On-Demand Anodyne SLC18A2 18 43 COc1ccc(CN(CCO)C[C@H](O)CN2CCCC2)cc1 ZINC000880570631 DC On-Demand Anodyne SLC18A2 18 43 COc1ccc(CN(CCO)CCOc2cccc([N+](=O)[O-])c2)cc1 ZINC000880570632 EE On-Demand Bother CACNA1D 46 39 COc1ccc(CN(CCO)CCOc2cccc([N+](=O)[O-])c2)cc1 ZINC000880570632 EE On-Demand Bother MMP9 15 41 COc1ccc(CN(CCO)CCOc2cccc([N+](=O)[O-])c2)cc1 ZINC000880570632 EE On-Demand Bother ACR 18 44 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne PPARA 17 41 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne BMP1 40 41 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne TSPO 27 44 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP13 40 44 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MTNR1A 49 36 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MTNR1B 49 35 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP2 20 46 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP3 31 46 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP8 19 46 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP9 36 46 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP12 24 40 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne CA9 18 44 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne MMP1 37 46 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2)cc1 ZINC000880570640 ED On-Demand Anodyne PDS 53 39 COc1ccc(CN(CCO)CC(=O)NCCc2ccc(F)cc2)cc1 ZINC000880570660 FD On-Demand Anodyne MTNR1A 46 38 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C)cc1 ZINC000880570661 EE On-Demand Anodyne ADRB2 15 43 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C)cc1 ZINC000880570661 EE On-Demand Anodyne GRIN1 16 40 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C)cc1 ZINC000880570661 EE On-Demand Anodyne ABCB1 30 40 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C)cc1 ZINC000880570662 EE On-Demand Anodyne ADRB2 15 43 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C)cc1 ZINC000880570662 EE On-Demand Anodyne GRIN1 16 40 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C)cc1 ZINC000880570662 EE On-Demand Anodyne ABCB1 30 40 COc1ccc(CN(CCO)CC(=O)N(C)C2CC2)cc1 ZINC000880570665 CD On-Demand Anodyne ERG7 16 42 COc1ccc(CN(CCO)C[C@H](O)COC(C)(C)C)cc1 ZINC000880570672 DD On-Demand Anodyne GRIN1 15 41 COc1ccc(CN(CCO)C[C@@H](O)COC(C)(C)C)cc1 ZINC000880570673 DD On-Demand Anodyne GRIN1 15 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(C)C)cc1 ZINC000880570688 DD On-Demand Anodyne MMP13 16 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(C)C)cc1 ZINC000880570688 DD On-Demand Anodyne MMP3 22 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(C)C)cc1 ZINC000880570688 DD On-Demand Anodyne MMP8 20 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(C)C)cc1 ZINC000880570688 DD On-Demand Anodyne MMP12 22 41 COc1ccc(CN(CCO)CC(=O)N[C@@H](C)C(C)C)cc1 ZINC000880570688 DD On-Demand Anodyne MMP1 26 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(C)C)cc1 ZINC000880570689 DD On-Demand Anodyne MMP13 16 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(C)C)cc1 ZINC000880570689 DD On-Demand Anodyne MMP3 22 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(C)C)cc1 ZINC000880570689 DD On-Demand Anodyne MMP8 20 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(C)C)cc1 ZINC000880570689 DD On-Demand Anodyne MMP12 22 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)C(C)C)cc1 ZINC000880570689 DD On-Demand Anodyne MMP1 26 41 CCN1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570692 ED On-Demand Anodyne DRD4 15 46 CCN1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570692 ED On-Demand Anodyne LTA4H 19 41 CCN1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570692 ED On-Demand Anodyne SIGMAR1 23 54 CCN1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570692 ED On-Demand Anodyne PDK1 41 36 CCN1CCC(NC(=O)CN(CCO)Cc2ccc(OC)cc2)CC1 ZINC000880570692 ED On-Demand Anodyne MCHR1 29 49 COc1ccc(CN(CCO)CCC(=O)NC(C)C)cc1 ZINC000880570700 CD On-Demand Anodyne BMP1 42 40 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne CYP19A1 21 41 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne CYP11B1 35 41 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne TBXAS1 40 44 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne CYP11B2 18 41 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne HMOX1 35 40 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne CYP24A1 40 32 O[C@@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570702 DG On-Demand Anodyne CYP27B1 53 32 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne CYP19A1 21 41 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne CYP11B1 35 41 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne TBXAS1 40 44 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne CYP11B2 18 41 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne HMOX1 35 40 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne CYP24A1 40 32 O[C@@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570703 DG On-Demand Anodyne CYP27B1 53 32 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne CYP19A1 21 41 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne CYP11B1 35 41 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne TBXAS1 40 44 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne CYP11B2 18 41 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne HMOX1 35 40 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne CYP24A1 40 32 O[C@H](CCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570704 DG On-Demand Anodyne CYP27B1 53 32 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne CYP19A1 21 41 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne CYP11B1 35 41 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne TBXAS1 40 44 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne CYP11B2 18 41 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne HMOX1 35 40 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne CYP24A1 40 32 O[C@H](CCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880570705 DG On-Demand Anodyne CYP27B1 53 32 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2OC)cc1 ZINC000880570708 FD On-Demand Anodyne MTNR1A 41 37 COc1ccc(CN(CCO)CC(=O)NCc2ccccc2OC)cc1 ZINC000880570708 FD On-Demand Anodyne MBTPS1 58 42 COc1ccc(CN(CCO)Cc2cccc([N+](=O)[O-])c2C)cc1 ZINC000880570709 EF On-Demand Bother COLA 60 40 CON(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570762 DD On-Demand Anodyne CYP19A1 15 40 CON(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570762 DD On-Demand Anodyne TBXAS1 58 41 CON(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570762 DD On-Demand Anodyne CYP24A1 47 38 CON(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570762 DD On-Demand Anodyne CYP26A1 112 40 CON(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570762 DD On-Demand Anodyne CYP27B1 63 38 CON(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570763 DD On-Demand Anodyne CYP19A1 15 40 CON(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570763 DD On-Demand Anodyne TBXAS1 58 41 CON(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570763 DD On-Demand Anodyne CYP24A1 47 38 CON(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570763 DD On-Demand Anodyne CYP26A1 112 40 CON(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570763 DD On-Demand Anodyne CYP27B1 63 38 CC(C)(C)OC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570770 EG On-Demand Anodyne TBXAS1 58 42 CC(C)(C)OC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570770 EG On-Demand Anodyne CYP24A1 52 38 CC(C)(C)OC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570770 EG On-Demand Anodyne CYP26A1 116 39 CC(C)(C)OC(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570770 EG On-Demand Anodyne CYP27B1 70 38 CC(C)(C)OC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570771 EG On-Demand Anodyne TBXAS1 58 42 CC(C)(C)OC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570771 EG On-Demand Anodyne CYP24A1 52 38 CC(C)(C)OC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570771 EG On-Demand Anodyne CYP26A1 116 39 CC(C)(C)OC(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570771 EG On-Demand Anodyne CYP27B1 70 38 CC(C)(C)[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570776 CF On-Demand Anodyne CYP11B1 28 40 CC(C)(C)[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570776 CF On-Demand Anodyne TBXAS1 35 40 CC(C)(C)[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570776 CF On-Demand Anodyne CYP11B2 17 40 CC(C)(C)[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570776 CF On-Demand Anodyne CYP24A1 40 35 CC(C)(C)[C@@H](O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570776 CF On-Demand Anodyne CYP27B1 51 35 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne BMP1 51 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP13 43 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP2 22 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP3 33 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP8 20 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP9 39 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP12 27 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne CA9 18 42 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne MMP1 37 46 COc1ccc(CN(CCO)CC(=O)NC(=O)NCc2ccccc2)cc1 ZINC000880570779 FD On-Demand Anodyne PDS 51 38 CC(C)(C)[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570780 CF On-Demand Anodyne CYP11B1 28 40 CC(C)(C)[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570780 CF On-Demand Anodyne TBXAS1 35 40 CC(C)(C)[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570780 CF On-Demand Anodyne CYP11B2 17 40 CC(C)(C)[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570780 CF On-Demand Anodyne CYP24A1 40 35 CC(C)(C)[C@@H](O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570780 CF On-Demand Anodyne CYP27B1 51 35 COc1ccc(CN(CCO)Cc2ccc(-n3ccnc3)cc2)cc1 ZINC000880570795 EF On-Demand Anodyne NOS2 15 44 COc1ccc(CN(CCO)Cc2ccc(-n3ccnc3)cc2)cc1 ZINC000880570795 EF On-Demand Anodyne CYP2C19 19 47 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne MMP13 18 42 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne MMP3 21 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne MMP9 17 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne MMP1 19 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne GPR119 41 38 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570800 FF On-Demand Anodyne NR1D1 21 42 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne MMP13 18 42 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne MMP3 21 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne MMP9 17 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne MMP1 19 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne GPR119 41 38 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880570802 FF On-Demand Anodyne NR1D1 21 42 COc1ccc(CN(CCO)CCC(=O)N(C)c2ccccc2)cc1 ZINC000880570813 EF On-Demand Anodyne TSPO 17 41 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880570816 GE On-Demand Anodyne BMP1 47 37 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880570816 GE On-Demand Anodyne MMP13 28 47 COc1ccc(CN(CCO)CCCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880570816 GE On-Demand Anodyne MMP1 25 41 COc1ccc(CN(CCO)CCOc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880570827 GD On-Demand Anodyne BMP1 51 38 COc1ccc(CN(CCO)CCNS(C)(=O)=O)cc1 ZINC000880570834 DC On-Demand Anodyne MMP13 23 41 COc1ccc(CN(CCO)CCNS(C)(=O)=O)cc1 ZINC000880570834 DC On-Demand Anodyne MMP3 16 41 COc1ccc(CN(CCO)CCNS(C)(=O)=O)cc1 ZINC000880570834 DC On-Demand Anodyne MMP12 21 41 COc1ccc(CN(CCO)CCNS(C)(=O)=O)cc1 ZINC000880570834 DC On-Demand Anodyne MMP1 25 41 COc1ccc(CN(CCO)C[C@@H](O)c2cccc(Cl)c2)cc1 ZINC000880570835 EF On-Demand Anodyne ADRB1 22 42 COc1ccc(CN(CCO)C[C@@H](O)c2cccc(Cl)c2)cc1 ZINC000880570835 EF On-Demand Anodyne ADRB3 37 42 COc1ccc(CN(CCO)C[C@@H](O)c2cccc(Cl)c2)cc1 ZINC000880570835 EF On-Demand Anodyne AOC3 23 44 COc1ccc(CN(CCO)C[C@H](O)c2cccc(Cl)c2)cc1 ZINC000880570837 EF On-Demand Anodyne ADRB1 22 42 COc1ccc(CN(CCO)C[C@H](O)c2cccc(Cl)c2)cc1 ZINC000880570837 EF On-Demand Anodyne ADRB3 37 42 COc1ccc(CN(CCO)C[C@H](O)c2cccc(Cl)c2)cc1 ZINC000880570837 EF On-Demand Anodyne AOC3 23 44 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(C#N)c2)cc1 ZINC000880570840 FE On-Demand Mild MTNR1B 15 40 COc1ccc(CN(CCO)Cc2cnc(Cl)s2)cc1 ZINC000880570844 DF On-Demand Anodyne NR1D1 23 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne MMP13 18 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne MMP3 21 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne MMP9 26 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne MMP12 25 41 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne CA9 19 43 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Br)cc1 ZINC000880570848 GF On-Demand Anodyne MMP1 28 41 COc1ccc(CN(CCO)CCC(=O)Nc2sc3c(c2C#N)CCC3)cc1 ZINC000880570859 GF On-Demand Mild VIPR1 40 72 COc1ccc(CN(CCO)Cc2ccc3c(c2)OCCO3)cc1 ZINC000880570864 EE On-Demand Anodyne EDNRA 33 42 COc1ccc(CN(CCO)Cc2ccc3c(c2)OCCO3)cc1 ZINC000880570864 EE On-Demand Anodyne BMP1 69 41 COc1ccc(CN(CCO)CC(=O)OCc2ccccc2)cc1 ZINC000880570875 EE On-Demand Anodyne MMP3 20 41 COc1ccc(CN(CCO)CC(=O)OCc2ccccc2)cc1 ZINC000880570875 EE On-Demand Anodyne MMP9 20 41 COc1ccc(CN(CCO)CC(=O)OCc2ccccc2)cc1 ZINC000880570875 EE On-Demand Anodyne MMP1 20 41 COc1ccc(CN(CCO)CC(=O)OCc2ccccc2)cc1 ZINC000880570875 EE On-Demand Anodyne SLC12A5 21 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(SC)cc2)cc1 ZINC000880570882 FF On-Demand Anodyne LTA4H 26 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(SC)cc2)cc1 ZINC000880570882 FF On-Demand Anodyne BMP1 16 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(SC)cc2)cc1 ZINC000880570882 FF On-Demand Anodyne CA9 15 42 COc1ccc(CN(CCO)CCc2cccnc2)cc1 ZINC000880570884 CE On-Demand Anodyne PTAFR 26 42 COc1ccc(CN(CCO)CCc2cccnc2)cc1 ZINC000880570884 CE On-Demand Anodyne CYP11B2 20 43 COc1ccc(CN(CCO)CCc2cccnc2)cc1 ZINC000880570884 CE On-Demand Anodyne NR1D1 39 51 O=C(Cc1cccc2ncccc12)NCc1cn(C2CCC2)nn1 ZINC000880570885 DE On-Demand Anodyne CDK5 24 42 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2Cl)cc1 ZINC000880570897 GD On-Demand Reactive ECR 24 41 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2Cl)cc1 ZINC000880570897 GD On-Demand Reactive MMP9 17 45 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2Cl)cc1 ZINC000880570897 GD On-Demand Reactive MMP1 18 45 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2Cl)cc1 ZINC000880570897 GD On-Demand Reactive E3UJZ5_SPOLI 20 41 COc1cccc(C(C)(C)C(=O)NCc2cn(C3CCC3)nn2)c1 ZINC000880570901 EF On-Demand Anodyne DRD4 40 30 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880570903 FE On-Demand Anodyne LTA4H 30 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880570903 FE On-Demand Anodyne CA9 15 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(F)cc2F)cc1 ZINC000880570904 FE On-Demand Anodyne SOAT1 26 45 COc1ccc(CN(CCO)CC(=O)N2CCC[C@H](NC(C)=O)C2)cc1 ZINC000880570914 FC On-Demand Anodyne BIRC2 15 40 COc1ccc(CN(CCO)CC(=O)N2CCC[C@@H](NC(C)=O)C2)cc1 ZINC000880570915 FC On-Demand Anodyne BIRC2 15 40 COC(=O)[C@@](C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570919 DD On-Demand Anodyne CYP19A1 23 41 COC(=O)[C@@](C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570919 DD On-Demand Anodyne TBXAS1 57 41 COC(=O)[C@@](C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570919 DD On-Demand Anodyne CYP24A1 53 41 COC(=O)[C@@](C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570919 DD On-Demand Anodyne CYP26A1 102 45 COC(=O)[C@@](C)(O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570919 DD On-Demand Anodyne CYP27B1 72 41 COc1ccc(CN(CCO)CC(=O)NCCc2c(F)cccc2F)cc1 ZINC000880570921 GE On-Demand Anodyne MTNR1A 70 41 COc1ccc(CN(CCO)CC(=O)NCCc2c(F)cccc2F)cc1 ZINC000880570921 GE On-Demand Anodyne MTNR1B 60 41 COC(=O)[C@@](C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570922 DD On-Demand Anodyne CYP19A1 23 41 COC(=O)[C@@](C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570922 DD On-Demand Anodyne TBXAS1 57 41 COC(=O)[C@@](C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570922 DD On-Demand Anodyne CYP24A1 53 41 COC(=O)[C@@](C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570922 DD On-Demand Anodyne CYP26A1 102 45 COC(=O)[C@@](C)(O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570922 DD On-Demand Anodyne CYP27B1 72 41 C[C@@H](O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570933 CE On-Demand Anodyne TBXAS1 40 45 C[C@@H](O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570933 CE On-Demand Anodyne CYP27B1 48 31 C[C@@H](O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570936 CE On-Demand Anodyne TBXAS1 40 45 C[C@@H](O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570936 CE On-Demand Anodyne CYP27B1 48 31 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(OC[C@H]3CCCO3)cc2)cc1 ZINC000880570937 GH On-Demand Anodyne HMOX1 49 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(OC[C@@H]3CCCO3)cc2)cc1 ZINC000880570938 GH On-Demand Anodyne HMOX1 49 40 c1ccc([C@H](Cn2ccnc2)NCc2ccc(OC[C@H]3CCCO3)cc2)cc1 ZINC000880570939 GH On-Demand Anodyne HMOX1 49 40 c1ccc([C@@H](Cn2ccnc2)NCc2ccc(OC[C@@H]3CCCO3)cc2)cc1 ZINC000880570940 GH On-Demand Anodyne HMOX1 49 40 O=C(Cc1ccc2cnccc2c1)NCc1cn(C2CCC2)nn1 ZINC000880570944 DE On-Demand Anodyne NAMPT 55 39 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cn1cccn1 ZINC000880570947 DD On-Demand Anodyne CYP27B1 40 34 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)Cn1cccn1 ZINC000880570948 DD On-Demand Anodyne CYP27B1 40 34 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cn1cccn1 ZINC000880570949 DD On-Demand Anodyne CYP27B1 40 34 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)Cn1cccn1 ZINC000880570950 DD On-Demand Anodyne CYP27B1 40 34 CN(Cc1ccc(N(C)C)cc1)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880570958 GF On-Demand Clean TBXAS1 36 40 CN(Cc1ccc(N(C)C)cc1)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880570959 GF On-Demand Clean TBXAS1 36 40 Cc1cnc(CN[C@@H](Cn2ccnc2)c2ccccc2)o1 ZINC000880570960 CF On-Demand Anodyne CYP11B1 43 37 Cc1cnc(CN[C@H](Cn2ccnc2)c2ccccc2)o1 ZINC000880570961 CF On-Demand Anodyne CYP11B1 43 37 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne ADRB2 33 43 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne ADRB1 44 42 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne ADRB3 37 40 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne TBXAS1 30 47 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne ABCB1 25 45 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne CYP24A1 42 34 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne CYP26A1 60 34 CC(=O)c1cccc(OC[C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570982 GF On-Demand Anodyne CYP27B1 55 34 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne ADRB2 33 43 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne ADRB1 44 42 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne ADRB3 37 40 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne TBXAS1 30 47 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne ABCB1 25 45 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne CYP24A1 42 34 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne CYP26A1 60 34 CC(=O)c1cccc(OC[C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570983 GF On-Demand Anodyne CYP27B1 55 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne ADRB2 33 43 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne ADRB1 44 42 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne ADRB3 37 40 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne TBXAS1 30 47 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne ABCB1 25 45 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne CYP24A1 42 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne CYP26A1 60 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570984 GF On-Demand Anodyne CYP27B1 55 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne ADRB2 33 43 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne ADRB1 44 42 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne ADRB3 37 40 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne TBXAS1 30 47 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne ABCB1 25 45 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne CYP24A1 42 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne CYP26A1 60 34 CC(=O)c1cccc(OC[C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880570985 GF On-Demand Anodyne CYP27B1 55 34 CC(C)(C)OC(=O)N1CC[C@@H](CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880570995 FG On-Demand Anodyne GRIN2B 20 42 CC(C)(C)OC(=O)N1CC[C@H](CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880570996 FG On-Demand Anodyne GRIN2B 20 42 CC(C)(C)OC(=O)N1CC[C@H](CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880570997 FG On-Demand Anodyne GRIN2B 20 42 CC(C)(C)OC(=O)N1CC[C@@H](CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880570998 FG On-Demand Anodyne GRIN2B 20 42 c1ccc([C@H](Cn2ccnc2)NCc2ccc3c(c2)CCC3)cc1 ZINC000880571005 DH On-Demand Anodyne HMOX1 40 33 c1ccc([C@@H](Cn2ccnc2)NCc2ccc3c(c2)CCC3)cc1 ZINC000880571006 DH On-Demand Anodyne HMOX1 40 33 O=C(NCc1cn(C2CCC2)nn1)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880571026 GE On-Demand Anodyne CA14 19 43 O=C(NCc1cn(C2CCC2)nn1)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880571026 GE On-Demand Anodyne CCR2 61 38 CN(C)S(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571037 ED On-Demand Anodyne TBXAS1 30 40 CN(C)S(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571037 ED On-Demand Anodyne CYP27B1 42 30 CN(C)S(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571038 ED On-Demand Anodyne TBXAS1 30 40 CN(C)S(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571038 ED On-Demand Anodyne CYP27B1 42 30 COc1ccc(CN(CCO)Cc2cn(-c3ccccc3)nn2)cc1 ZINC000880571039 EE On-Demand Anodyne FIMH 21 42 COc1ccc(CN(CCO)CCC(=O)C2CC2)cc1 ZINC000880571042 CD On-Demand Anodyne SLC18A2 19 40 COc1ccc(CN(CCO)Cc2ccc3ccccc3n2)cc1 ZINC000880571048 DG On-Demand Anodyne ALOX5 21 41 COc1ccc(CN(CCO)Cc2ccc3ccccc3n2)cc1 ZINC000880571048 DG On-Demand Anodyne CYSLTR1 63 46 CS(=O)(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571053 DC On-Demand Anodyne TBXAS1 47 40 CS(=O)(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571053 DC On-Demand Anodyne CYP24A1 47 32 CS(=O)(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571053 DC On-Demand Anodyne CYP27B1 62 32 CS(=O)(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571054 DC On-Demand Anodyne TBXAS1 47 40 CS(=O)(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571054 DC On-Demand Anodyne CYP24A1 47 32 CS(=O)(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571054 DC On-Demand Anodyne CYP27B1 62 32 C[C@@H](c1ccc(F)c(F)c1)N(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571055 GH On-Demand Anodyne CYP26A1 91 35 C[C@@H](c1ccc(F)c(F)c1)N(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571058 GH On-Demand Anodyne CYP26A1 91 35 COc1ccc(CN(CCO)CC(=O)NCc2ccccn2)cc1 ZINC000880571062 ED On-Demand Anodyne BMP1 19 43 COc1ccc(CN(CCO)CC(=O)NCc2ccccn2)cc1 ZINC000880571062 ED On-Demand Anodyne MMP12 21 40 COC(=O)c1sccc1CN(CCO)Cc1ccc(OC)cc1 ZINC000880571063 EF On-Demand Anodyne FAS 34 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne BMP1 45 40 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne MMP13 27 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne MMP3 21 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne MMP8 16 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne MMP12 27 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne CA9 19 42 COc1ccc(CN(CCO)CCS(N)(=O)=O)cc1 ZINC000880571065 CB On-Demand Anodyne MMP1 26 42 COc1ccc(CN(CCO)CC2CCC2)cc1 ZINC000880571067 BE On-Demand Anodyne SLC18A2 22 42 O=c1cc(CN[C@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571077 GI On-Demand Anodyne CYP19A1 29 47 O=c1cc(CN[C@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571077 GI On-Demand Anodyne CYP11B1 36 44 O=c1cc(CN[C@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571077 GI On-Demand Anodyne CYP11B2 21 44 O=c1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571080 GI On-Demand Anodyne CYP19A1 29 47 O=c1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571080 GI On-Demand Anodyne CYP11B1 36 44 O=c1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)c2cc3c(cc2o1)CCC3 ZINC000880571080 GI On-Demand Anodyne CYP11B2 21 44 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571082 DE On-Demand Anodyne TBXAS1 62 42 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571082 DE On-Demand Anodyne PTAFR 30 43 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571082 DE On-Demand Anodyne CYP24A1 43 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571082 DE On-Demand Anodyne CYP27B1 56 35 COc1ccc(CN(CCO)[C@@H](C)C(=O)NNC(=O)CC(C)C)cc1 ZINC000880571083 FD On-Demand Reactive BMP1 34 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571084 DE On-Demand Anodyne TBXAS1 62 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571084 DE On-Demand Anodyne PTAFR 30 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571084 DE On-Demand Anodyne CYP24A1 43 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCCC1 ZINC000880571084 DE On-Demand Anodyne CYP27B1 56 35 COc1ccc(CN(CCO)[C@H](C)C(=O)NNC(=O)CC(C)C)cc1 ZINC000880571085 FD On-Demand Reactive BMP1 34 40 N#CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571086 CF On-Demand Mild CYP19A1 19 41 N#CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571086 CF On-Demand Mild CYP11B1 34 40 N#CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571086 CF On-Demand Mild TBXAS1 29 41 N#CCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571086 CF On-Demand Mild CYP11B2 18 40 COc1ccc(CN(CCO)CC[C@H]2CCOC2=O)cc1 ZINC000880571091 CD On-Demand Anodyne TRAR 45 31 COc1ccc(CN(CCO)CC[C@@H]2CCOC2=O)cc1 ZINC000880571092 CD On-Demand Anodyne TRAR 45 31 N#CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571095 CF On-Demand Mild CYP19A1 19 41 N#CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571095 CF On-Demand Mild CYP11B1 34 40 N#CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571095 CF On-Demand Mild TBXAS1 29 41 N#CCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571095 CF On-Demand Mild CYP11B2 18 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571096 CD On-Demand Anodyne TBXAS1 64 43 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571096 CD On-Demand Anodyne PTAFR 31 44 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571096 CD On-Demand Anodyne CYP24A1 46 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571096 CD On-Demand Anodyne CYP27B1 61 35 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne LTA4H 38 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne BMP1 27 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MTNR1A 23 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MTNR1B 25 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MMP3 16 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne NPY5R 20 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MMP9 17 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MMP12 18 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne CA9 22 48 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne MMP1 21 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571097 EE On-Demand Anodyne RORC 16 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571098 CD On-Demand Anodyne TBXAS1 64 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571098 CD On-Demand Anodyne PTAFR 31 44 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571098 CD On-Demand Anodyne CYP24A1 46 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCC1 ZINC000880571098 CD On-Demand Anodyne CYP27B1 61 35 COc1ccc(CN(CCO)CC(=O)NCc2ccc(F)cc2)cc1 ZINC000880571099 ED On-Demand Anodyne MMP13 15 40 COc1ccc(CN(CCO)CC(=O)NCc2ccc(F)cc2)cc1 ZINC000880571099 ED On-Demand Anodyne MMP12 15 40 COc1ccc(CN(CCO)CC(=O)NCc2ccc(F)cc2)cc1 ZINC000880571099 ED On-Demand Anodyne CA9 15 44 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571112 GD On-Demand Anodyne TBXAS1 45 39 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571112 GD On-Demand Anodyne PTAFR 33 45 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571112 GD On-Demand Anodyne CYP27B1 44 33 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C(=O)N(C)C)c2)cc1 ZINC000880571113 GD On-Demand Anodyne LTA4H 21 41 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C(=O)N(C)C)c2)cc1 ZINC000880571113 GD On-Demand Anodyne MTNR1A 31 40 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C(=O)N(C)C)c2)cc1 ZINC000880571113 GD On-Demand Anodyne MTNR1B 33 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571114 GD On-Demand Anodyne TBXAS1 45 39 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571114 GD On-Demand Anodyne PTAFR 33 45 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCN(C(=O)C2CC2)CC1 ZINC000880571114 GD On-Demand Anodyne CYP27B1 44 33 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880571115 FD On-Demand Anodyne EDNRB 79 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880571115 FD On-Demand Anodyne EDNRA 78 46 COc1ccc(CN(CCO)CC(=O)Nc2ccc3c(c2)OCO3)cc1 ZINC000880571115 FD On-Demand Anodyne BMP1 83 42 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccc(C)cc2)cc1 ZINC000880571119 FD On-Demand Reactive UTS2 16 42 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571139 GG On-Demand Anodyne TBXAS1 32 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571139 GG On-Demand Anodyne SSTR4 51 36 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571139 GG On-Demand Anodyne SSTR5 41 36 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571141 GG On-Demand Anodyne TBXAS1 32 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571141 GG On-Demand Anodyne SSTR4 51 36 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880571141 GG On-Demand Anodyne SSTR5 41 36 c1ccc([C@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571143 CD On-Demand Anodyne CYP19A1 22 41 c1ccc([C@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571143 CD On-Demand Anodyne CYP11B1 39 41 c1ccc([C@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571143 CD On-Demand Anodyne TBXAS1 29 41 c1ccc([C@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571143 CD On-Demand Anodyne HIS3 48 37 c1ccc([C@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571143 CD On-Demand Anodyne CYP11B2 19 41 c1ccc([C@@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571145 CD On-Demand Anodyne CYP19A1 22 41 c1ccc([C@@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571145 CD On-Demand Anodyne CYP11B1 39 41 c1ccc([C@@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571145 CD On-Demand Anodyne TBXAS1 29 41 c1ccc([C@@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571145 CD On-Demand Anodyne HIS3 48 37 c1ccc([C@@H](Cn2ccnc2)NCCn2cncn2)cc1 ZINC000880571145 CD On-Demand Anodyne CYP11B2 19 41 COc1ccc(CN(CCO)Cc2csc(C3CC3)n2)cc1 ZINC000880571146 DG On-Demand Anodyne AVPR1B 17 44 COc1ccc(CN(CCO)CC(=O)NCC2CCC2)cc1 ZINC000880571157 DD On-Demand Anodyne MMP3 21 41 COc1ccc(CN(CCO)CC(=O)NCC2CCC2)cc1 ZINC000880571157 DD On-Demand Anodyne MMP9 15 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne BMP1 24 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne MMP13 29 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne MMP3 31 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne MMP8 21 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne EPHX2 21 49 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne MMP12 18 40 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCC2)cc1 ZINC000880571161 ED On-Demand Anodyne MMP1 27 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571162 CD On-Demand Anodyne TBXAS1 64 43 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571162 CD On-Demand Anodyne PTAFR 31 44 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571162 CD On-Demand Anodyne CYP24A1 46 35 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571162 CD On-Demand Anodyne CYP27B1 61 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571163 CD On-Demand Anodyne TBXAS1 64 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571163 CD On-Demand Anodyne PTAFR 31 44 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571163 CD On-Demand Anodyne CYP24A1 46 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N1CCCC1 ZINC000880571163 CD On-Demand Anodyne CYP27B1 61 35 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cc2)cc1 ZINC000880571166 EF On-Demand Anodyne LTA4H 31 53 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cc2)cc1 ZINC000880571166 EF On-Demand Anodyne BMP1 19 45 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cc2)cc1 ZINC000880571166 EF On-Demand Anodyne NPY5R 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cc2)cc1 ZINC000880571166 EF On-Demand Anodyne CA9 16 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)cc2)cc1 ZINC000880571166 EF On-Demand Anodyne RORC 15 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(C#N)cc2)cc1 ZINC000880571170 FD On-Demand Mild MMP13 20 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(C#N)cc2)cc1 ZINC000880571170 FD On-Demand Mild MMP1 17 40 Cc1nnc(N2CCN(C(=O)c3cc4ccccc4cc3F)CC2)n1C ZINC000880571194 FE On-Demand Anodyne CCKAR 41 38 C=CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571199 BF On-Demand Mild CYP19A1 21 44 C=CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571199 BF On-Demand Mild CYP11B1 42 44 C=CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571199 BF On-Demand Mild TBXAS1 28 44 C=CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571199 BF On-Demand Mild CYP11B2 20 44 C=CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571199 BF On-Demand Mild CYP27B1 49 32 C=CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571200 BF On-Demand Mild CYP19A1 21 44 C=CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571200 BF On-Demand Mild CYP11B1 42 44 C=CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571200 BF On-Demand Mild TBXAS1 28 44 C=CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571200 BF On-Demand Mild CYP11B2 20 44 C=CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571200 BF On-Demand Mild CYP27B1 49 32 CO/C(=C/c1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880571201 DE On-Demand Anodyne PREP 15 40 CO/C(=C\c1ccccc1)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880571202 DE On-Demand Anodyne PREP 15 40 COc1ccc(CN(CCO)CC(=O)NC2CCC3(CC2)OCCO3)cc1 ZINC000880571212 GD On-Demand Anodyne C5AR1 28 42 Cc1nnc(N2CCN(C(=O)c3cc4cc(F)ccc4[nH]c3=O)CC2)n1C ZINC000880571216 FD On-Demand Anodyne HRH4 21 49 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne LTA4H 45 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne BMP1 28 45 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne MTNR1A 15 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne MTNR1B 20 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne NPY5R 19 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne MMP12 17 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne CA9 19 47 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(OC)cc2)cc1 ZINC000880571217 FF On-Demand Anodyne MMP1 15 40 COc1ccc(CN(CCO)CCC(=O)NCC2CCCCC2)cc1 ZINC000880571218 EF On-Demand Anodyne BMP1 24 46 COc1ccc(CN(CCO)CCC(=O)NCC2CCCCC2)cc1 ZINC000880571218 EF On-Demand Anodyne MMP3 15 42 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne CYP19A1 15 47 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne CYP11B1 17 46 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne MAOA 49 35 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne ACHE 15 47 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne MAOB 47 44 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(OC)ccc23)cc1 ZINC000880571224 FF On-Demand Anodyne HSD17B3 21 40 COc1ccc(CN(CCO)CC(=O)Nc2ccccc2Cl)cc1 ZINC000880571232 EF On-Demand Anodyne CA9 15 43 COc1ccc(CN(CCO)CC(=O)N(C)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571234 FE On-Demand Bother MMP2 15 48 COc1ccc(CN(CCO)CC(=O)N(C)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571234 FE On-Demand Bother MMP8 31 48 COc1ccc(CN(CCO)CC(=O)N(C)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571234 FE On-Demand Bother MMP9 19 48 COc1ccc(CN(CCO)CC(=O)N(C)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571234 FE On-Demand Bother MMP1 24 48 COc1ccc(CN(CCO)CC(=O)Nc2cccc(C(=O)NC3CC3)c2)cc1 ZINC000880571235 GE On-Demand Anodyne MCHR1 25 44 COc1ccc(CN(CCO)CC(=O)N(C)Cc2cnn(C)c2)cc1 ZINC000880571242 EC On-Demand Anodyne PLA2G7 51 38 COc1ccc(CN(CCO)CC(=O)N2CCc3ccc([N+](=O)[O-])cc32)cc1 ZINC000880571249 GD On-Demand Bother MMP8 22 42 COc1ccc(CN(CCO)CC(=O)N2CCc3ccc([N+](=O)[O-])cc32)cc1 ZINC000880571249 GD On-Demand Bother MMP9 16 42 COc1ccc(CN(CCO)CC(=O)N2CCc3ccc([N+](=O)[O-])cc32)cc1 ZINC000880571249 GD On-Demand Bother MMP1 19 42 COc1ccc(CN(CCO)CC(=O)NNC(=O)C2CC2)cc1 ZINC000880571250 DC On-Demand Reactive MMP13 32 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C2CC2)cc1 ZINC000880571250 DC On-Demand Reactive MMP3 47 38 COc1ccc(CN(CCO)CC(=O)NNC(=O)C2CC2)cc1 ZINC000880571250 DC On-Demand Reactive MMP12 19 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C2CC2)cc1 ZINC000880571250 DC On-Demand Reactive MMP1 43 40 COc1ccc(CN(CCO)CCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1 ZINC000880571258 GB On-Demand Anodyne MAOB 15 47 COc1ccc(CN(CCO)Cc2nc(C)c3ccccc3n2)cc1 ZINC000880571267 EF On-Demand Anodyne TSPO 17 42 COc1ccc(CN(CCO)Cc2cc(C)nc3ccccc23)cc1 ZINC000880571268 EH On-Demand Anodyne TSPO 21 44 COc1ccc(CN(CCO)Cc2cc(C)nc3ccccc23)cc1 ZINC000880571268 EH On-Demand Anodyne ADAM17 79 39 COc1ccc(CN(CCO)CCC(=O)Nc2ccccc2C(F)(F)F)cc1 ZINC000880571270 GH On-Demand Anodyne BMP1 26 40 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA2 91 53 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne BMP1 56 45 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA6 19 41 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA1 79 53 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA7 58 50 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP13 32 42 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA13 21 41 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA4 55 50 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA14 44 44 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP2 18 47 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP3 26 42 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP8 20 47 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP9 32 47 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP12 27 42 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA12 60 53 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CA9 71 53 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne MMP1 29 47 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CAH_METTE 19 41 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne CYNT 24 42 COc1ccc(CN(CCO)CCc2ccc(S(N)(=O)=O)cc2)cc1 ZINC000880571279 FD On-Demand Anodyne NCE103 20 50 COc1ccc(CN(CCO)C[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000880571280 FD On-Demand Anodyne NR1D1 22 44 COc1ccc(CN(CCO)C[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000880571281 FD On-Demand Anodyne NR1D1 22 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCOCC3)cc2)cc1 ZINC000880571282 GD On-Demand Anodyne LTA4H 23 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCOCC3)cc2)cc1 ZINC000880571282 GD On-Demand Anodyne MTOR 56 39 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCOCC3)cc2)cc1 ZINC000880571282 GD On-Demand Anodyne PIK3CB 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(N3CCOCC3)cc2)cc1 ZINC000880571282 GD On-Demand Anodyne EPHB4 58 37 COc1ccc(CN(CCO)C[C@H](O)c2ccc(C#N)cc2)cc1 ZINC000880571285 EE On-Demand Mild AOC3 16 48 COc1ccc(CN(CCO)C[C@@H](O)c2ccc(C#N)cc2)cc1 ZINC000880571286 EE On-Demand Mild AOC3 16 48 Cc1nnc(N2CCN(C(=O)c3csc(NC4CCCCC4)n3)CC2)n1C ZINC000880571290 GE On-Demand Anodyne TRPC6 64 45 Cc1nnc(N2CCN(C(=O)c3csc(NC4CCCCC4)n3)CC2)n1C ZINC000880571290 GE On-Demand Anodyne TRPC3 58 45 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880571291 FF On-Demand Anodyne LTA4H 38 42 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880571291 FF On-Demand Anodyne BMP1 19 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880571291 FF On-Demand Anodyne MTNR1B 16 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C(C)=O)cc2)cc1 ZINC000880571291 FF On-Demand Anodyne CA9 15 42 Cc1nnc(N2CCN(C(=O)CC[C@@H]3CCc4ccccc43)CC2)n1C ZINC000880571295 FE On-Demand Anodyne SSTR1 44 42 Cc1nnc(N2CCN(C(=O)CC[C@H]3CCc4ccccc43)CC2)n1C ZINC000880571296 FE On-Demand Anodyne SSTR1 44 42 COc1ccc(CN(CCO)CCCN2CCOCC2)cc1 ZINC000880571297 DD On-Demand Anodyne HRH3 15 42 COc1ccc(CN(CCO)CCCN2CCOCC2)cc1 ZINC000880571297 DD On-Demand Anodyne SIGMAR1 18 44 COc1ccc(CN(CCO)CCCN2CCOCC2)cc1 ZINC000880571297 DD On-Demand Anodyne PTGDS 19 42 COc1ccc(CN(CCO)CC(=O)NCC#N)cc1 ZINC000880571299 CC On-Demand Mild MMP12 16 42 COc1ccc(CN(CCO)Cc2nc(O)c3cc(Cl)ccc3n2)cc1 ZINC000880571303 FF On-Demand Anodyne HRP1_PLAFA 18 42 COc1ccc(CN(CCO)Cc2cc(=O)c(O)co2)cc1 ZINC000880571310 DD On-Demand Anodyne DAO 23 43 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne LTA4H 38 43 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne BMP1 43 48 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP13 28 41 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne HDAC8 16 41 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP2 26 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP3 32 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP8 27 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne NPY5R 28 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP9 38 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP12 27 41 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne CA12 20 40 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne CA9 21 40 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne MMP1 35 44 COc1ccc(CN(CCO)CC(=O)NC(=O)Nc2ccccc2)cc1 ZINC000880571313 FD On-Demand Anodyne RORC 18 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C#N)cc2)cc1 ZINC000880571315 ED On-Demand Mild LTA4H 25 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C#N)cc2)cc1 ZINC000880571315 ED On-Demand Mild CA12 15 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C#N)cc2)cc1 ZINC000880571315 ED On-Demand Mild CA9 20 41 COc1ccc(CN(CCO)Cc2cnc(OC)c(Cl)c2)cc1 ZINC000880571320 EF On-Demand Anodyne PDE6A 40 31 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne CA2 26 52 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne LTA4H 24 46 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne BMP1 75 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne CA1 24 52 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP13 53 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne CA4 31 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP2 37 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP3 44 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP8 42 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP9 53 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP12 31 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne CA12 18 52 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne CA9 27 52 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne MMP1 52 47 COc1ccc(CN(CCO)CC(=O)Nc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880571324 GD On-Demand Anodyne RORC 35 43 COc1ccc(CN(CCO)CC(=O)Nc2sccc2C#N)cc1 ZINC000880571325 EE On-Demand Mild VIPR1 17 41 COc1ccc(CN(CCO)CCc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571328 EF On-Demand Bother MMP8 30 48 COc1ccc(CN(CCO)CCc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571328 EF On-Demand Bother MMP9 18 48 COc1ccc(CN(CCO)CCc2ccc([N+](=O)[O-])cc2)cc1 ZINC000880571328 EF On-Demand Bother MMP1 23 48 COc1ccc(CN(CCO)CC(=O)Nc2cc(C)nn2C(C)(C)C)cc1 ZINC000880571331 FE On-Demand Anodyne PROKR1 47 31 COc1ccc(CN(CCO)CC(=O)Nc2c(C)cccc2C)cc1 ZINC000880571334 EF On-Demand Anodyne MMP12 18 40 COc1ccc(CN(CCO)Cc2csc(N(C(C)=O)C3CC3)n2)cc1 ZINC000880571340 GF On-Demand Anodyne AVPR1B 15 42 O=C(NCc1cn(C2CCC2)nn1)c1ccc(C(F)(F)Br)nc1 ZINC000880571417 GF On-Demand Anodyne CA14 18 46 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)NC1CCCC1 ZINC000880571418 EF On-Demand Anodyne TBXAS1 53 39 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)NC1CCCC1 ZINC000880571419 EF On-Demand Anodyne TBXAS1 53 39 c1ccc([C@H](Cn2ccnc2)NCCN2CCOCC2)cc1 ZINC000880571420 DD On-Demand Anodyne CASR 46 38 c1ccc([C@@H](Cn2ccnc2)NCCN2CCOCC2)cc1 ZINC000880571421 DD On-Demand Anodyne CASR 46 38 CCOCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571424 CF On-Demand Anodyne TBXAS1 35 40 CCOCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571425 CF On-Demand Anodyne TBXAS1 35 40 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571435 ED On-Demand Anodyne TBXAS1 45 39 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571435 ED On-Demand Anodyne PTAFR 21 43 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571435 ED On-Demand Anodyne CYP26A1 43 34 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571435 ED On-Demand Anodyne CYP27B1 46 35 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571436 ED On-Demand Anodyne TBXAS1 45 39 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571436 ED On-Demand Anodyne PTAFR 21 43 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571436 ED On-Demand Anodyne CYP26A1 43 34 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCOCC1 ZINC000880571436 ED On-Demand Anodyne CYP27B1 46 35 O=C(CCN[C@@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc21 ZINC000880571446 FG On-Demand Anodyne CYP27B1 40 33 O=C(CCN[C@H](Cn1ccnc1)c1ccccc1)N1CCc2ccccc21 ZINC000880571447 FG On-Demand Anodyne CYP27B1 40 33 CS(=O)(=O)c1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571450 GF On-Demand Anodyne TBXAS1 22 44 CS(=O)(=O)c1cccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571450 GF On-Demand Anodyne HMOX2 17 40 CS(=O)(=O)c1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571451 GF On-Demand Anodyne TBXAS1 22 44 CS(=O)(=O)c1cccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571451 GF On-Demand Anodyne HMOX2 17 40 CC(C)(C)OC(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571472 EF On-Demand Anodyne TBXAS1 64 41 CC(C)(C)OC(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571472 EF On-Demand Anodyne CYP24A1 56 39 CC(C)(C)OC(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571472 EF On-Demand Anodyne CYP26A1 102 38 CC(C)(C)OC(=O)NCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571472 EF On-Demand Anodyne CYP27B1 76 39 CC(C)(C)OC(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571473 EF On-Demand Anodyne TBXAS1 64 41 CC(C)(C)OC(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571473 EF On-Demand Anodyne CYP24A1 56 39 CC(C)(C)OC(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571473 EF On-Demand Anodyne CYP26A1 102 38 CC(C)(C)OC(=O)NCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571473 EF On-Demand Anodyne CYP27B1 76 39 COC(=O)c1oc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1C ZINC000880571478 EG On-Demand Anodyne TBXAS1 41 39 COC(=O)c1oc(CN[C@@H](Cn2ccnc2)c2ccccc2)cc1C ZINC000880571478 EG On-Demand Anodyne CYP27B1 43 32 COC(=O)c1oc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1C ZINC000880571479 EG On-Demand Anodyne TBXAS1 41 39 COC(=O)c1oc(CN[C@H](Cn2ccnc2)c2ccccc2)cc1C ZINC000880571479 EG On-Demand Anodyne CYP27B1 43 32 CC(C)(C)CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571489 EF On-Demand Anodyne TBXAS1 50 41 CC(C)(C)CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571489 EF On-Demand Anodyne CYP24A1 41 36 CC(C)(C)CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571489 EF On-Demand Anodyne CYP26A1 49 37 CC(C)(C)CCNC(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571489 EF On-Demand Anodyne CYP27B1 52 36 CC(C)(C)CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571490 EF On-Demand Anodyne TBXAS1 50 41 CC(C)(C)CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571490 EF On-Demand Anodyne CYP24A1 41 36 CC(C)(C)CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571490 EF On-Demand Anodyne CYP26A1 49 37 CC(C)(C)CCNC(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571490 EF On-Demand Anodyne CYP27B1 52 36 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne PDGFRB 15 43 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne LTA4H 27 41 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne ROCK1 23 40 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne MTNR1A 47 49 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne MTNR1B 47 49 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne ROCK2 27 40 COc1ccc(CN(CCO)CCC(=O)Nc2cccc(OC)c2)cc1 ZINC000880571507 FF On-Demand Anodyne TAAR1 32 40 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)s1 ZINC000880571511 EF On-Demand Anodyne NR1D1 18 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne LTA4H 31 45 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne MTNR1A 27 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne MTNR1B 30 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne NPY5R 16 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne MMP12 16 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne CA9 21 45 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne MMP1 16 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(NC(C)=O)cc2)cc1 ZINC000880571512 FE On-Demand Anodyne RORC 18 43 COc1ccc(CN(CCO)CCCS(=O)(=O)N(C)C)cc1 ZINC000880571514 EC On-Demand Anodyne MMP12 17 40 COc1ccc(CN(CCO)C[C@H](O)COc2cccc3[nH]ccc23)cc1 ZINC000880571516 FE On-Demand Anodyne ADRB1 19 49 COc1ccc(CN(CCO)C[C@@H](O)COc2cccc3[nH]ccc23)cc1 ZINC000880571517 FE On-Demand Anodyne ADRB1 19 49 COC(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1F ZINC000880571518 EF On-Demand Anodyne BMP1 28 41 COc1ccc(CN(CCO)[C@H]2CCCN(C(C)C)C2=O)cc1 ZINC000880571519 DD On-Demand Anodyne SLC18A2 20 40 COc1ccc(CN(CCO)[C@@H]2CCCN(C(C)C)C2=O)cc1 ZINC000880571520 DD On-Demand Anodyne SLC18A2 20 40 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne PTAFR 28 41 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne BMP1 17 44 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne KCNA5 15 44 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne MMP13 35 47 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne MMP3 16 48 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne MMP9 24 47 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne MMP12 17 41 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne HCRTR2 15 50 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne MMP1 24 47 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne NAMPT 57 43 COc1ccc(CN(CCO)CC(=O)NCc2cccnc2)cc1 ZINC000880571522 ED On-Demand Anodyne NR1D1 31 45 CNC(=O)[C@@H](NC(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880571526 GD On-Demand Anodyne MMP2 22 41 CNC(=O)[C@@H](NC(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880571526 GD On-Demand Anodyne MMP3 35 43 CNC(=O)[C@@H](NC(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880571526 GD On-Demand Anodyne MTTP 47 37 CNC(=O)[C@@H](NC(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880571526 GD On-Demand Anodyne MMP9 28 41 CNC(=O)[C@@H](NC(=O)CN(CCO)Cc1ccc(OC)cc1)c1ccccc1 ZINC000880571526 GD On-Demand Anodyne MMP1 43 46 COc1ccc(CN(CCO)CCCCS(C)(=O)=O)cc1 ZINC000880571528 DD On-Demand Anodyne BMP1 40 37 COC[C@@H](O)CN(CCO)Cc1ccc(OC)cc1 ZINC000880571535 CC On-Demand Anodyne GRIN1 15 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(F)c(F)c2)cc1 ZINC000880571536 FE On-Demand Anodyne LTA4H 21 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(F)c(F)c2)cc1 ZINC000880571536 FE On-Demand Anodyne BMP1 19 40 COc1ccc(CN(CCO)CC(=O)NCCc2cccc3cccnc23)cc1 ZINC000880571543 GE On-Demand Anodyne NQO2 29 42 COc1ccc(CN(CCO)CC(=O)NCCc2cccc3cccnc23)cc1 ZINC000880571543 GE On-Demand Anodyne MTNR1A 71 45 COc1ccc(CN(CCO)CC(=O)NCCc2cccc3cccnc23)cc1 ZINC000880571543 GE On-Demand Anodyne MTNR1B 49 40 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne CYP19A1 21 40 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne CYP11B1 28 44 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne TBXAS1 44 41 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne HMOX1 37 41 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne HMOX2 48 40 COc1ccc(CN(CCO)CCCn2ccnc2)cc1 ZINC000880571546 CD On-Demand Anodyne QPCT 38 52 COc1ccc(CN(CCO)CC(=O)Nc2nnc(C(C)(C)C)s2)cc1 ZINC000880571548 GE On-Demand Anodyne CA2 18 45 COc1ccc(CN(CCO)CC(=O)Nc2nnc(C(C)(C)C)s2)cc1 ZINC000880571548 GE On-Demand Anodyne CSNK1D 21 40 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne LTA4H 34 49 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne HRH3 55 55 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne SIGMAR1 35 47 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne EBP 48 42 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne PSMB2 39 40 COc1ccc(CN(CCO)CCN2CCCCC2)cc1 ZINC000880571549 CD On-Demand Anodyne PSMB1 42 40 COc1ccc(CN(CCO)CC(=O)NC2CCN(C(C)=O)CC2)cc1 ZINC000880571552 FC On-Demand Anodyne SIGMAR1 15 48 COc1ccc(CN(CCO)CC(=O)NC2CCN(C(C)=O)CC2)cc1 ZINC000880571552 FC On-Demand Anodyne EPHX2 21 46 COc1ccc(CN(CCO)CC(=O)NC2CCN(C(C)=O)CC2)cc1 ZINC000880571552 FC On-Demand Anodyne MCHR1 18 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C#N)cc2)cc1 ZINC000880571553 FE On-Demand Mild BMP1 16 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(C#N)cc2)cc1 ZINC000880571553 FE On-Demand Mild CA9 17 41 COc1ccc(CN(CCO)CC(=O)NCc2ccc(N(C)C)cc2)cc1 ZINC000880571554 FD On-Demand Clean CA9 15 43 COc1ccc(CN(CCO)CC(=O)NCc2cc(F)cc(F)c2)cc1 ZINC000880571557 FE On-Demand Anodyne CA9 15 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2cccc(C)c2)cc1 ZINC000880571558 FD On-Demand Reactive CTSL 17 43 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2cccc(C)c2)cc1 ZINC000880571558 FD On-Demand Reactive KCNK3 58 42 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2cccc(C)c2)cc1 ZINC000880571558 FD On-Demand Reactive KCNK9 42 36 COc1ccc(CN(CCO)CC(=O)Nc2cccnc2Cl)cc1 ZINC000880571562 EE On-Demand Anodyne G2YM83_BOTF4 63 32 COc1ccc(CN(CCO)CC(=O)Nc2nnc(C(C)C)s2)cc1 ZINC000880571567 FE On-Demand Anodyne CA2 15 45 COc1ccc(CN(CCO)CC(=O)Nc2nnc(C(C)C)s2)cc1 ZINC000880571567 FE On-Demand Anodyne CSNK1D 17 40 COc1ccc(CN(CCO)CCn2ccnc2)cc1 ZINC000880571568 CD On-Demand Anodyne CYP11B1 34 45 COc1ccc(CN(CCO)CCn2ccnc2)cc1 ZINC000880571568 CD On-Demand Anodyne TBXAS1 37 44 COc1ccc(CN(CCO)CCn2ccnc2)cc1 ZINC000880571568 CD On-Demand Anodyne CYP11B2 21 40 COc1ccc(CN(CCO)CCn2ccnc2)cc1 ZINC000880571568 CD On-Demand Anodyne QPCT 28 48 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(O)ccc23)cc1 ZINC000880571573 FF On-Demand Anodyne CYP11B1 15 44 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(O)ccc23)cc1 ZINC000880571573 FF On-Demand Anodyne MAOB 37 42 COc1ccc(CN(CCO)Cc2cc(=O)oc3cc(O)ccc23)cc1 ZINC000880571573 FF On-Demand Anodyne HSD17B3 41 52 COc1ccc(CN(CCO)CC(=O)NCc2cccc(C)c2)cc1 ZINC000880571575 EE On-Demand Anodyne MMP13 30 42 COc1ccc(CN(CCO)CC(=O)NCc2cccc(C)c2)cc1 ZINC000880571575 EE On-Demand Anodyne MTNR1A 50 37 COc1ccc(CN(CCO)CC(=O)NCc2cccc(C)c2)cc1 ZINC000880571575 EE On-Demand Anodyne MTNR1B 46 37 COc1ccc(CN(CCO)CC(=O)N(C)CC(=O)Nc2ccc(C)cc2)cc1 ZINC000880571576 GD On-Demand Anodyne LTA4H 28 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne LTA4H 19 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne MTNR1B 26 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne CA9 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne HCRTR2 16 50 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne ENPP1 83 39 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC)c(OC)c2)cc1 ZINC000880571577 FE On-Demand Anodyne DRTS_TRYCR 45 32 COc1ccc(CN(CCO)Cc2nc(-c3ccc4c(c3)OCO4)no2)cc1 ZINC000880571579 GE On-Demand Anodyne EDNRB 54 41 COc1ccc(CN(CCO)Cc2nc(-c3ccc4c(c3)OCO4)no2)cc1 ZINC000880571579 GE On-Demand Anodyne EDNRA 58 41 COc1ccc(CN(CCO)Cc2nc(-c3ccc4c(c3)OCO4)no2)cc1 ZINC000880571579 GE On-Demand Anodyne BMP1 59 36 COc1ccc(CN(CCO)Cc2nc(-c3ccc4c(c3)OCO4)no2)cc1 ZINC000880571579 GE On-Demand Anodyne GSK3A 19 44 COc1ccc(CN(CCO)CC(=O)N(C2CCCC2)C2CC2)cc1 ZINC000880571580 EE On-Demand Anodyne AVPR1B 15 43 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C(=O)N(C)C)cc2)cc1 ZINC000880571581 GD On-Demand Anodyne LTA4H 30 48 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C(=O)N(C)C)cc2)cc1 ZINC000880571581 GD On-Demand Anodyne NPY5R 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C(=O)N(C)C)cc2)cc1 ZINC000880571581 GD On-Demand Anodyne CA9 15 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCCC2)cc1 ZINC000880571582 FD On-Demand Anodyne BMP1 22 42 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCCC2)cc1 ZINC000880571582 FD On-Demand Anodyne MMP3 28 41 COc1ccc(CN(CCO)CC(=O)NC(=O)NC2CCCCC2)cc1 ZINC000880571582 FD On-Demand Anodyne EPHX2 26 51 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne AVPR1B 15 40 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne BMP1 109 46 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP13 57 50 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne ADAM17 22 44 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP2 29 44 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP3 39 50 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP8 36 50 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP9 55 45 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP12 34 50 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)cc2)cc1 ZINC000880571587 GD On-Demand Anodyne MMP1 50 50 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C)c(C)c2)cc1 ZINC000880571588 EF On-Demand Anodyne LTA4H 20 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C)c(C)c2)cc1 ZINC000880571588 EF On-Demand Anodyne CA9 15 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(C)c(C)c2)cc1 ZINC000880571588 EF On-Demand Anodyne ENPP1 59 32 COc1ccc(CN(CCO)CC(=O)NCC(=O)c2ccccc2)cc1 ZINC000880571589 FD On-Demand Anodyne LTA4H 17 40 COc1ccc(CN(CCO)CC(=O)NCC(=O)c2ccccc2)cc1 ZINC000880571589 FD On-Demand Anodyne MMP3 19 41 COc1ccc(CN(CCO)CC(=O)NCC(=O)c2ccccc2)cc1 ZINC000880571589 FD On-Demand Anodyne MMP9 18 41 COc1ccc(CN(CCO)CC(=O)NCC(=O)c2ccccc2)cc1 ZINC000880571589 FD On-Demand Anodyne MMP1 20 41 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC(F)F)cc2)cc1 ZINC000880571593 GF On-Demand Anodyne LTA4H 28 42 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC(F)F)cc2)cc1 ZINC000880571593 GF On-Demand Anodyne NPY5R 19 40 COc1ccc(CN(CCO)CC(=O)Nc2ccc(OC(F)F)cc2)cc1 ZINC000880571593 GF On-Demand Anodyne CA9 15 41 COc1ccc(CN(CCO)CC(=O)NC2CCN(C(C)C)CC2)cc1 ZINC000880571594 FD On-Demand Anodyne MCHR1 19 45 C[C@@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571615 EF On-Demand Anodyne CYP27B1 43 32 C[C@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571616 EF On-Demand Anodyne CYP27B1 43 32 C[C@@H]1CCCCN1C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571617 EF On-Demand Anodyne CYP27B1 43 32 C[C@H]1CCCCN1C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571618 EF On-Demand Anodyne CYP27B1 43 32 CSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571624 CF On-Demand Anodyne CYP19A1 23 42 CSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571624 CF On-Demand Anodyne CYP11B1 40 42 CSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571624 CF On-Demand Anodyne TBXAS1 28 42 CSCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571624 CF On-Demand Anodyne CYP11B2 20 42 CSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571625 CF On-Demand Anodyne CYP19A1 23 42 CSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571625 CF On-Demand Anodyne CYP11B1 40 42 CSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571625 CF On-Demand Anodyne TBXAS1 28 42 CSCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571625 CF On-Demand Anodyne CYP11B2 20 42 CNS(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571635 DD On-Demand Anodyne TBXAS1 32 40 CNS(=O)(=O)CCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571635 DD On-Demand Anodyne CYP27B1 47 30 CNS(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571636 DD On-Demand Anodyne TBXAS1 32 40 CNS(=O)(=O)CCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571636 DD On-Demand Anodyne CYP27B1 47 30 FC(F)(F)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571641 CG On-Demand Anodyne CYP19A1 19 41 FC(F)(F)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571641 CG On-Demand Anodyne CYP11B1 37 43 FC(F)(F)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571641 CG On-Demand Anodyne TBXAS1 31 41 FC(F)(F)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571641 CG On-Demand Anodyne CYP11B2 18 43 FC(F)(F)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571641 CG On-Demand Anodyne CYP27B1 43 30 FC(F)(F)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571642 CG On-Demand Anodyne CYP19A1 19 41 FC(F)(F)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571642 CG On-Demand Anodyne CYP11B1 37 43 FC(F)(F)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571642 CG On-Demand Anodyne TBXAS1 31 41 FC(F)(F)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571642 CG On-Demand Anodyne CYP11B2 18 43 FC(F)(F)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571642 CG On-Demand Anodyne CYP27B1 43 30 CS(=O)(=O)c1ccc(OCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571646 GG On-Demand Anodyne TBXAS1 27 44 CS(=O)(=O)c1ccc(OCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571646 GG On-Demand Anodyne CYP17A1 16 40 CS(=O)(=O)c1ccc(OCCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571646 GG On-Demand Anodyne CYP26A1 54 33 CS(=O)(=O)c1ccc(OCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571647 GG On-Demand Anodyne TBXAS1 27 44 CS(=O)(=O)c1ccc(OCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571647 GG On-Demand Anodyne CYP17A1 16 40 CS(=O)(=O)c1ccc(OCCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571647 GG On-Demand Anodyne CYP26A1 54 33 FC(F)(F)COc1ccc(CN[C@@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571654 GH On-Demand Anodyne CYP11B1 34 40 FC(F)(F)COc1ccc(CN[C@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571655 GH On-Demand Anodyne CYP11B1 34 40 CN(C)S(=O)(=O)c1cccc(CN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571660 GF On-Demand Anodyne CYP11B1 19 40 CN(C)S(=O)(=O)c1cccc(CN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571661 GF On-Demand Anodyne CYP11B1 19 40 COC(=O)/C(C)=C/CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571662 CE On-Demand Anodyne CYP19A1 18 40 COC(=O)/C(C)=C/CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571662 CE On-Demand Anodyne TBXAS1 54 41 COC(=O)/C(C)=C/CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571662 CE On-Demand Anodyne CYP24A1 52 36 COC(=O)/C(C)=C/CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571662 CE On-Demand Anodyne CYP27B1 72 36 COC(=O)/C(C)=C/CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571663 CE On-Demand Anodyne CYP19A1 18 40 COC(=O)/C(C)=C/CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571663 CE On-Demand Anodyne TBXAS1 54 41 COC(=O)/C(C)=C/CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571663 CE On-Demand Anodyne CYP24A1 52 36 COC(=O)/C(C)=C/CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571663 CE On-Demand Anodyne CYP27B1 72 36 COC(=O)/C(C)=C\CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571664 CE On-Demand Anodyne CYP19A1 18 40 COC(=O)/C(C)=C\CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571664 CE On-Demand Anodyne TBXAS1 54 41 COC(=O)/C(C)=C\CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571664 CE On-Demand Anodyne CYP24A1 52 36 COC(=O)/C(C)=C\CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571664 CE On-Demand Anodyne CYP27B1 72 36 COC(=O)/C(C)=C\CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571665 CE On-Demand Anodyne CYP19A1 18 40 COC(=O)/C(C)=C\CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571665 CE On-Demand Anodyne TBXAS1 54 41 COC(=O)/C(C)=C\CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571665 CE On-Demand Anodyne CYP24A1 52 36 COC(=O)/C(C)=C\CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571665 CE On-Demand Anodyne CYP27B1 72 36 C[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)CS(C)(=O)=O ZINC000880571668 DD On-Demand Anodyne TBXAS1 29 40 C[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)CS(C)(=O)=O ZINC000880571668 DD On-Demand Anodyne CYP27B1 41 34 C[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)CS(C)(=O)=O ZINC000880571669 DD On-Demand Anodyne TBXAS1 29 40 C[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)CS(C)(=O)=O ZINC000880571669 DD On-Demand Anodyne CYP27B1 41 34 C#CCN1CCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880571671 FC On-Demand Mild PTAFR 34 44 C#CCN1CCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)CC1 ZINC000880571672 FC On-Demand Mild PTAFR 34 44 c1ccc([C@@H](Cn2ccnc2)NCCN2CCCCC2)cc1 ZINC000880571683 CF On-Demand Anodyne HNMT 62 35 c1ccc([C@H](Cn2ccnc2)NCCN2CCCCC2)cc1 ZINC000880571684 CF On-Demand Anodyne HNMT 62 35 FC(F)C(F)(F)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571692 DG On-Demand Anodyne CYP11B1 31 40 FC(F)C(F)(F)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571692 DG On-Demand Anodyne CYP11B2 17 40 FC(F)C(F)(F)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571692 DG On-Demand Anodyne CYP27B1 48 31 FC(F)C(F)(F)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571693 DG On-Demand Anodyne CYP11B1 31 40 FC(F)C(F)(F)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571693 DG On-Demand Anodyne CYP11B2 17 40 FC(F)C(F)(F)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571693 DG On-Demand Anodyne CYP27B1 48 31 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1C#N ZINC000880571694 DD On-Demand Mild CA14 17 41 COc1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1C#N ZINC000880571694 DD On-Demand Mild SLC5A7 35 41 CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571695 CE On-Demand Anodyne CYP19A1 21 41 CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571695 CE On-Demand Anodyne CYP11B1 41 41 CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571695 CE On-Demand Anodyne TBXAS1 35 43 CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571695 CE On-Demand Anodyne CYP11B2 22 41 CCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571695 CE On-Demand Anodyne CYP27B1 42 30 CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571696 CE On-Demand Anodyne CYP19A1 21 41 CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571696 CE On-Demand Anodyne CYP11B1 41 41 CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571696 CE On-Demand Anodyne TBXAS1 35 43 CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571696 CE On-Demand Anodyne CYP11B2 22 41 CCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571696 CE On-Demand Anodyne CYP27B1 42 30 OCCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571697 CD On-Demand Anodyne TBXAS1 39 41 OCCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571697 CD On-Demand Anodyne CYP24A1 46 31 OCCOCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571697 CD On-Demand Anodyne CYP27B1 63 31 OCCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571698 CD On-Demand Anodyne TBXAS1 39 41 OCCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571698 CD On-Demand Anodyne CYP24A1 46 31 OCCOCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571698 CD On-Demand Anodyne CYP27B1 63 31 COc1ccc(CN(CCO)CC(=O)Nc2c(C)cc(C)cc2C)cc1 ZINC000880571705 FG On-Demand Anodyne FFAR4 19 40 COc1ccc(CN(CCO)CC(=O)Nc2sc(C)c(C)c2C#N)cc1 ZINC000880571718 FF On-Demand Mild VIPR1 24 46 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne BMP1 75 41 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP13 57 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne ADAM17 18 42 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP2 38 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP3 35 42 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP8 27 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP14 20 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne ALOX15 42 43 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP9 49 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP12 34 44 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP7 17 41 COc1ccc(CN(CCO)CCNS(=O)(=O)c2ccccc2)cc1 ZINC000880571724 FD On-Demand Anodyne MMP1 41 44 COc1ccc(CN(CCO)CCn2cc([N+](=O)[O-])ccc2=O)cc1 ZINC000880571725 ED On-Demand Bother MMP8 19 42 COc1ccc(CN(CCO)CCn2cc([N+](=O)[O-])ccc2=O)cc1 ZINC000880571725 ED On-Demand Bother MMP1 16 42 COc1ccc(CN(CCO)CC(=O)NCCC(C)(C)C)cc1 ZINC000880571726 DE On-Demand Anodyne MMP12 15 40 COc1ccc(CN(CCO)CCC2CC2)cc1 ZINC000880571730 BE On-Demand Anodyne SLC18A2 23 41 COc1ccc(CN(CCO)Cc2cncc(Br)c2)cc1 ZINC000880571736 FF On-Demand Anodyne CYP11B2 20 41 COc1ccc(CN(CCO)CC(=O)Nc2nccs2)cc1 ZINC000880571739 DD On-Demand Anodyne MAP1 121 43 COC(=O)c1cccc(NC(=O)CN(CCO)Cc2ccc(OC)cc2)c1 ZINC000880571745 FD On-Demand Anodyne LTA4H 20 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive BMP1 28 42 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP13 23 41 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP3 26 44 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP8 15 44 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP9 30 44 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP12 23 41 COc1ccc(CN(CCO)CC(=O)NNC(=O)c2ccccc2)cc1 ZINC000880571748 FC On-Demand Reactive MMP1 30 44 COc1ccc(CN(CCO)CC[C@@H]2CCCN2C)cc1 ZINC000880571754 CD On-Demand Anodyne HRH1 26 45 COc1ccc(CN(CCO)CC[C@@H]2CCCN2C)cc1 ZINC000880571754 CD On-Demand Anodyne SLC18A2 61 45 COc1ccc(CN(CCO)CC[C@@H]2CCCN2C)cc1 ZINC000880571754 CD On-Demand Anodyne SIGMAR1 17 40 COc1ccc(CN(CCO)CC[C@@H]2CCCN2C)cc1 ZINC000880571754 CD On-Demand Anodyne CHRNA10 69 43 COc1ccc(CN(CCO)CC[C@@H]2CCCN2C)cc1 ZINC000880571754 CD On-Demand Anodyne ACKR3 75 39 COc1ccc(CN(CCO)CC[C@H]2CCCN2C)cc1 ZINC000880571755 CD On-Demand Anodyne HRH1 26 45 COc1ccc(CN(CCO)CC[C@H]2CCCN2C)cc1 ZINC000880571755 CD On-Demand Anodyne SLC18A2 61 45 COc1ccc(CN(CCO)CC[C@H]2CCCN2C)cc1 ZINC000880571755 CD On-Demand Anodyne SIGMAR1 17 40 COc1ccc(CN(CCO)CC[C@H]2CCCN2C)cc1 ZINC000880571755 CD On-Demand Anodyne CHRNA10 69 43 COc1ccc(CN(CCO)CC[C@H]2CCCN2C)cc1 ZINC000880571755 CD On-Demand Anodyne ACKR3 75 39 COc1ccc(CN(CCO)Cc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880571766 FF On-Demand Anodyne HRH3 16 47 COc1ccc(CN(CCO)Cc2ccc(CN3CCOCC3)cc2)cc1 ZINC000880571766 FF On-Demand Anodyne SIGMAR1 21 49 COc1ccc(CN(CCO)CCC(=O)c2ccccc2)cc1 ZINC000880571768 DF On-Demand Anodyne MMP1 17 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)N(C)C)s2)cc1 ZINC000880571776 GE On-Demand Anodyne NR1D1 15 41 COc1ccc(CN(CCO)C[C@@H](O)CN(C)C2CC2)cc1 ZINC000880571784 DC On-Demand Anodyne SLC18A2 21 42 COc1ccc(CN(CCO)C[C@H](O)CN(C)C2CC2)cc1 ZINC000880571785 DC On-Demand Anodyne SLC18A2 21 42 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne ACHE 16 53 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne LTA4H 29 47 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne HRP1_PLAFA 18 44 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne HRH3 73 52 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne SIGMAR1 36 53 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne EBP 45 43 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne HNMT 40 33 COc1ccc(CN(CCO)CCCN2CCCCC2)cc1 ZINC000880571791 DE On-Demand Anodyne PSMB1 41 39 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive BMP1 53 39 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive MMP13 16 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive MMP3 22 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive MMP8 20 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive MMP12 26 40 COc1ccc(CN(CCO)CC(=O)NNC(=O)C(C)C)cc1 ZINC000880571796 DC On-Demand Reactive MMP1 27 40 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C#N)cc1 ZINC000880571800 FD On-Demand Mild ADRB1 57 40 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C#N)cc1 ZINC000880571800 FD On-Demand Mild CASR 46 48 COc1ccc(CN(CCO)C[C@@H](O)COc2ccccc2C#N)cc1 ZINC000880571800 FD On-Demand Mild CYP2D6 18 48 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C#N)cc1 ZINC000880571801 FD On-Demand Mild ADRB1 57 40 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C#N)cc1 ZINC000880571801 FD On-Demand Mild CASR 46 48 COc1ccc(CN(CCO)C[C@H](O)COc2ccccc2C#N)cc1 ZINC000880571801 FD On-Demand Mild CYP2D6 18 48 Cc1nnc(N2CCN(C(=O)c3cc(F)c(F)cc3Cl)CC2)n1C ZINC000880571808 FE On-Demand Anodyne P2RX7 22 41 COc1ccc(CN(CCO)CCOCC2CCC2)cc1 ZINC000880571809 CE On-Demand Anodyne SLC18A2 22 41 COc1ccc(CN(CCO)C[C@H](O)C2CC2)cc1 ZINC000880571813 CD On-Demand Anodyne SLC18A2 23 44 COc1ccc(CN(CCO)C[C@@H](O)C2CC2)cc1 ZINC000880571814 CD On-Demand Anodyne SLC18A2 23 44 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne BMP1 62 42 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP13 35 44 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP2 21 45 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP3 28 45 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP8 21 45 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP9 38 45 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP12 30 44 COc1ccc(CN(CCO)CCS(=O)(=O)Cc2ccccc2)cc1 ZINC000880571815 FE On-Demand Anodyne MMP1 33 45 COc1ccc(CN(CCO)CCC(=O)N2CCCC2)cc1 ZINC000880571828 DD On-Demand Anodyne MMP13 17 40 COc1ccc(CN(CCO)CCC(=O)N2CCCC2)cc1 ZINC000880571828 DD On-Demand Anodyne DPP7 15 40 COc1ccc(CN(CCO)CCC(=O)N2CCCC2)cc1 ZINC000880571828 DD On-Demand Anodyne MMP1 19 40 COc1ccc(CN(CCO)CCOCc2ccccc2)cc1 ZINC000880571831 DF On-Demand Anodyne G6PC 24 40 COc1ccc(CN(CCO)CCc2c(C)nc3ccccn3c2=O)cc1 ZINC000880571838 FE On-Demand Anodyne ADRA2A 22 41 COc1ccc(CN(CCO)CCc2c(C)nc3ccccn3c2=O)cc1 ZINC000880571838 FE On-Demand Anodyne ADRA2B 26 41 COc1ccc(CN(CCO)C[C@H](OC)c2ccccc2)cc1 ZINC000880571847 DF On-Demand Anodyne AOC3 25 47 COc1ccc(CN(CCO)C[C@@H](OC)c2ccccc2)cc1 ZINC000880571848 DF On-Demand Anodyne AOC3 25 47 COc1ccc(CN(CCO)Cc2cncn2Cc2ccccc2)cc1 ZINC000880571852 FF On-Demand Anodyne CYP11B1 23 60 COc1ccc(CN(CCO)Cc2cncn2Cc2ccccc2)cc1 ZINC000880571852 FF On-Demand Anodyne CYP11B2 19 60 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne CYP19A1 24 40 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne CYP11B1 36 40 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne TBXAS1 37 42 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne CYP11B2 20 40 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne CYP24A1 45 34 COCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571857 CE On-Demand Anodyne CYP27B1 60 34 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne CYP19A1 24 40 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne CYP11B1 36 40 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne TBXAS1 37 42 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne CYP11B2 20 40 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne CYP24A1 45 34 COCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571858 CE On-Demand Anodyne CYP27B1 60 34 O=C(NCc1cn(C2CCC2)nn1)C(=O)c1cc(Cl)cc(Cl)c1 ZINC000880571859 FF On-Demand Anodyne CACNA1I 51 34 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571879 FF On-Demand Anodyne CYP11B1 25 40 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571879 FF On-Demand Anodyne TBXAS1 22 46 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571880 FF On-Demand Anodyne CYP11B1 25 40 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571880 FF On-Demand Anodyne TBXAS1 22 46 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571881 FF On-Demand Anodyne CYP11B1 25 40 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571881 FF On-Demand Anodyne TBXAS1 22 46 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571882 FF On-Demand Anodyne CYP11B1 25 40 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COCc1ccccc1 ZINC000880571882 FF On-Demand Anodyne TBXAS1 22 46 COc1cccc(S(=O)(=O)CCN[C@@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571883 GF On-Demand Anodyne CYP19A1 20 41 COc1cccc(S(=O)(=O)CCN[C@H](Cn2ccnc2)c2ccccc2)c1 ZINC000880571884 GF On-Demand Anodyne CYP19A1 20 41 O=C1CCC(=O)N1CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571885 DD On-Demand Anodyne CYP11B1 42 39 O=C1CCC(=O)N1CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571885 DD On-Demand Anodyne TBXAS1 54 44 O=C1CCC(=O)N1CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571886 DD On-Demand Anodyne CYP11B1 42 39 O=C1CCC(=O)N1CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571886 DD On-Demand Anodyne TBXAS1 54 44 c1ccc([C@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571891 CG On-Demand Anodyne CYP19A1 16 40 c1ccc([C@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571891 CG On-Demand Anodyne CYP11B1 34 40 c1ccc([C@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571891 CG On-Demand Anodyne TBXAS1 28 40 c1ccc([C@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571891 CG On-Demand Anodyne CYP11B2 19 40 c1ccc([C@@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571892 CG On-Demand Anodyne CYP19A1 16 40 c1ccc([C@@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571892 CG On-Demand Anodyne CYP11B1 34 40 c1ccc([C@@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571892 CG On-Demand Anodyne TBXAS1 28 40 c1ccc([C@@H](Cn2ccnc2)NCCC2CC2)cc1 ZINC000880571892 CG On-Demand Anodyne CYP11B2 19 40 CC(=O)c1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OC(C)C ZINC000880571899 FF On-Demand Anodyne CA14 17 42 CC(=O)c1cc(C(=O)NCc2cn(C3CCC3)nn2)ccc1OC(C)C ZINC000880571899 FF On-Demand Anodyne SLC5A7 34 41 CCN(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571900 DE On-Demand Anodyne TBXAS1 61 42 CCN(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571900 DE On-Demand Anodyne CYP26A1 96 37 CCN(C)C(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880571900 DE On-Demand Anodyne CYP27B1 42 35 CCN(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571901 DE On-Demand Anodyne TBXAS1 61 42 CCN(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571901 DE On-Demand Anodyne CYP26A1 96 37 CCN(C)C(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880571901 DE On-Demand Anodyne CYP27B1 42 35 O[C@@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1Cl ZINC000880571908 FG On-Demand Anodyne ADRB2 26 45 O[C@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1Cl ZINC000880571909 FG On-Demand Anodyne ADRB2 26 45 O[C@H](CN[C@@H](Cn1ccnc1)c1ccccc1)COc1ccccc1Cl ZINC000880571910 FG On-Demand Anodyne ADRB2 26 45 O[C@@H](CN[C@H](Cn1ccnc1)c1ccccc1)COc1ccccc1Cl ZINC000880571911 FG On-Demand Anodyne ADRB2 26 45 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC(=O)N1CCCC1 ZINC000880571915 FC On-Demand Anodyne TBXAS1 45 39 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC(=O)N1CCCC1 ZINC000880571915 FC On-Demand Anodyne CYP27B1 46 35 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC(=O)N1CCCC1 ZINC000880571916 FC On-Demand Anodyne TBXAS1 45 39 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC(=O)N1CCCC1 ZINC000880571916 FC On-Demand Anodyne CYP27B1 46 35 CS(=O)(=O)c1ccc([C@@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571917 GE On-Demand Anodyne ADRB3 63 49 CS(=O)(=O)c1ccc([C@@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571918 GE On-Demand Anodyne ADRB3 63 49 CS(=O)(=O)c1ccc([C@H](O)CN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571919 GE On-Demand Anodyne ADRB3 63 49 CS(=O)(=O)c1ccc([C@H](O)CN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571920 GE On-Demand Anodyne ADRB3 63 49 c1ccc([C@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571923 BF On-Demand Anodyne CYP19A1 27 41 c1ccc([C@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571923 BF On-Demand Anodyne CYP11B1 45 41 c1ccc([C@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571923 BF On-Demand Anodyne TBXAS1 31 41 c1ccc([C@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571923 BF On-Demand Anodyne CYP11B2 25 41 c1ccc([C@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571923 BF On-Demand Anodyne CYP27B1 42 30 c1ccc([C@@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571924 BF On-Demand Anodyne CYP19A1 27 41 c1ccc([C@@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571924 BF On-Demand Anodyne CYP11B1 45 41 c1ccc([C@@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571924 BF On-Demand Anodyne TBXAS1 31 41 c1ccc([C@@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571924 BF On-Demand Anodyne CYP11B2 25 41 c1ccc([C@@H](Cn2ccnc2)NCC2CC2)cc1 ZINC000880571924 BF On-Demand Anodyne CYP27B1 42 30 CS(=O)(=O)c1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571930 GF On-Demand Anodyne CYP19A1 16 42 CS(=O)(=O)c1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571930 GF On-Demand Anodyne TBXAS1 27 46 CS(=O)(=O)c1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571930 GF On-Demand Anodyne CYP17A1 17 41 CS(=O)(=O)c1ccc(OCCN[C@@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571930 GF On-Demand Anodyne CYP26A1 40 32 CS(=O)(=O)c1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571931 GF On-Demand Anodyne CYP19A1 16 42 CS(=O)(=O)c1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571931 GF On-Demand Anodyne TBXAS1 27 46 CS(=O)(=O)c1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571931 GF On-Demand Anodyne CYP17A1 17 41 CS(=O)(=O)c1ccc(OCCN[C@H](Cn2ccnc2)c2ccccc2)cc1 ZINC000880571931 GF On-Demand Anodyne CYP26A1 40 32 O=C(NCc1cn(C2CCC2)nn1)c1ccc(CF)cc1 ZINC000880571936 CE On-Demand Anodyne CA14 16 48 Cn1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571937 CE On-Demand Anodyne CYP11B1 40 40 Cn1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571937 CE On-Demand Anodyne TBXAS1 20 40 Cn1cc(CN[C@@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571937 CE On-Demand Anodyne CYP11B2 18 40 Cn1cc(CN[C@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571938 CE On-Demand Anodyne CYP11B1 40 40 Cn1cc(CN[C@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571938 CE On-Demand Anodyne TBXAS1 20 40 Cn1cc(CN[C@H](Cn2ccnc2)c2ccccc2)cn1 ZINC000880571938 CE On-Demand Anodyne CYP11B2 18 40 c1ccc([C@H](Cn2ccnc2)NCCCCCn2cccn2)cc1 ZINC000880571945 DG On-Demand Anodyne TBXAS1 43 45 c1ccc([C@@H](Cn2ccnc2)NCCCCCn2cccn2)cc1 ZINC000880571946 DG On-Demand Anodyne TBXAS1 43 45 COc1ccc(CN(CCO)Cc2cncc(F)c2)cc1 ZINC000880571961 CE On-Demand Anodyne CYP11B2 19 41 Cc1nnc(N2CCN(C(=O)c3cc(=O)c4ccccc4o3)CC2)n1C ZINC000880571962 FD On-Demand Anodyne TNKS 26 48 COc1ccc(CN(CCO)Cc2cncc(C)c2)cc1 ZINC000880571966 CE On-Demand Anodyne CYP11B1 15 45 COc1ccc(CN(CCO)Cc2cncc(C)c2)cc1 ZINC000880571966 CE On-Demand Anodyne CYP11B2 23 45 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne BMP1 52 39 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne ACACA 19 40 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne ACACB 16 40 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP2 23 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP3 34 43 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP8 21 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne NPY5R 27 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP9 33 41 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP12 27 43 COc1ccc(CN(CCO)CC(=O)N[C@H](C)c2ccccc2)cc1 ZINC000880571973 EE On-Demand Anodyne MMP1 39 41 COc1ccc(CN(CCO)CCC(=O)N2CCN(C)CC2)cc1 ZINC000880571990 EC On-Demand Anodyne BMP1 39 45 CCCOc1ccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880571994 FD On-Demand Anodyne HTR1D 15 40 CCCOc1ccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880571994 FD On-Demand Anodyne HTR1B 18 40 CCCOc1ccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880571994 FD On-Demand Anodyne PLA2G4B 74 34 COc1ccc(CN(CCO)Cc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880571998 EE On-Demand Anodyne BMP1 85 40 COc1ccc(CN(CCO)Cc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880571998 EE On-Demand Anodyne MMP13 29 42 COc1ccc(CN(CCO)Cc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880571998 EE On-Demand Anodyne MMP3 18 42 COc1ccc(CN(CCO)Cc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880571998 EE On-Demand Anodyne MMP9 29 42 COc1ccc(CN(CCO)Cc2cccc(S(C)(=O)=O)c2)cc1 ZINC000880571998 EE On-Demand Anodyne MMP1 26 42 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MTNR1A 15 40 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MMP2 17 44 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MMP3 27 44 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MMP8 16 44 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MMP9 28 44 COc1ccc(CN(CCO)CC(=O)NOCc2ccccc2)cc1 ZINC000880572019 ED On-Demand Anodyne MMP1 29 44 Cc1nnc(N2CCN(C(=O)c3cccc(-n4cnnn4)c3)CC2)n1C ZINC000880572023 FC On-Demand Anodyne HPGD 42 37 Cc1nnc(N2CCN(C(=O)c3cccc(-n4cnnn4)c3)CC2)n1C ZINC000880572023 FC On-Demand Anodyne KCNJ1 50 36 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne GRIN2B 29 40 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne MMP13 24 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne SLC18A3 21 51 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne MMP3 28 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne MMP9 27 46 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne MMP7 20 41 COc1ccc(CN(CCO)C[C@@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572038 FF On-Demand Anodyne MMP1 27 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne GRIN2B 29 40 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne MMP13 24 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne SLC18A3 21 51 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne MMP3 28 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne MMP9 27 46 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne MMP7 20 41 COc1ccc(CN(CCO)C[C@H]2CCN(C(=O)c3ccccc3)C2)cc1 ZINC000880572039 FF On-Demand Anodyne MMP1 27 46 COc1ccc(CN(CCO)CC[C@H](O)c2ccccc2)cc1 ZINC000880572045 DF On-Demand Anodyne AOC3 21 40 COc1ccc(CN(CCO)CC[C@@H](O)c2ccccc2)cc1 ZINC000880572046 DF On-Demand Anodyne AOC3 21 40 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne BMP1 92 41 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP13 73 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP2 42 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP3 51 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP8 37 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP14 19 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP9 63 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP12 33 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP7 35 45 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne CA9 20 40 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne MMP1 61 46 CNS(=O)(=O)c1ccc(CN(CCO)Cc2ccc(OC)cc2)cc1 ZINC000880572055 FD On-Demand Anodyne FFAR4 19 40 Cc1nnc(N2CCN(C(=O)COc3cccc(C(F)(F)F)c3)CC2)n1C ZINC000880572063 GD On-Demand Anodyne HTR1D 15 43 Cc1nnc(N2CCN(C(=O)COc3cccc(C(F)(F)F)c3)CC2)n1C ZINC000880572063 GD On-Demand Anodyne HTR1B 18 43 Cc1nnc(N2CCN(C(=O)COc3cccc(C(F)(F)F)c3)CC2)n1C ZINC000880572063 GD On-Demand Anodyne LIPG 42 33 Cc1nnc(N2CCN(C(=O)COc3cccc(C(F)(F)F)c3)CC2)n1C ZINC000880572063 GD On-Demand Anodyne PDS 41 37 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne BMP1 50 38 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne MMP13 28 43 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne MMP3 20 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne MMP8 20 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne MMP12 24 40 COc1ccc(CN(CCO)CCS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880572064 FE On-Demand Anodyne MMP1 26 42 CCc1nc2ccccc2n1CC(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880572065 FD On-Demand Anodyne HRH1 26 44 COc1ccc(CN(CCO)CC(=O)Nc2ccc(Cl)nc2)cc1 ZINC000880572117 EE On-Demand Anodyne LTA4H 21 40 COc1ccc(CN(CCO)Cc2nc(-c3ccccc3F)no2)cc1 ZINC000880572121 FF On-Demand Anodyne LUCI_PHOPE 30 46 COc1ccc(CN(CCO)C[C@H](OC)C2CCC2)cc1 ZINC000880572146 CE On-Demand Anodyne SLC18A2 21 41 COc1ccc(CN(CCO)C[C@@H](OC)C2CCC2)cc1 ZINC000880572147 CE On-Demand Anodyne SLC18A2 21 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC1CC1 ZINC000880572149 CD On-Demand Anodyne TBXAS1 49 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NCC1CC1 ZINC000880572149 CD On-Demand Anodyne CYP27B1 41 34 COc1ccc(CN(CCO)CCOC2CCC2)cc1 ZINC000880572150 CE On-Demand Anodyne SLC18A2 20 43 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC1CC1 ZINC000880572152 CD On-Demand Anodyne TBXAS1 49 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NCC1CC1 ZINC000880572152 CD On-Demand Anodyne CYP27B1 41 34 O=C(CCc1cccnc1Cl)NCc1cn(C2CCC2)nn1 ZINC000880572176 DE On-Demand Anodyne SUCNR1 40 36 CC#CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572188 BE On-Demand Mild CYP19A1 27 43 CC#CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572188 BE On-Demand Mild CYP11B1 49 43 CC#CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572188 BE On-Demand Mild TBXAS1 33 43 CC#CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572188 BE On-Demand Mild CYP11B2 25 43 CC#CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572188 BE On-Demand Mild CYP27B1 48 31 CC#CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572191 BE On-Demand Mild CYP19A1 27 43 CC#CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572191 BE On-Demand Mild CYP11B1 49 43 CC#CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572191 BE On-Demand Mild TBXAS1 33 43 CC#CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572191 BE On-Demand Mild CYP11B2 25 43 CC#CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572191 BE On-Demand Mild CYP27B1 48 31 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N[C@H](c1ccccc1)C1CC1 ZINC000880572193 FG On-Demand Anodyne TBXAS1 42 40 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N[C@@H](c1ccccc1)C1CC1 ZINC000880572196 FG On-Demand Anodyne TBXAS1 42 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N[C@@H](c1ccccc1)C1CC1 ZINC000880572197 FG On-Demand Anodyne TBXAS1 42 40 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N[C@H](c1ccccc1)C1CC1 ZINC000880572198 FG On-Demand Anodyne TBXAS1 42 40 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880572214 GF On-Demand Mild REN 54 35 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880572214 GF On-Demand Mild FPR1 40 35 COc1ccc(CN(CCO)CCC2CCC2)cc1 ZINC000880572216 CF On-Demand Anodyne SLC18A2 27 44 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880572217 GF On-Demand Mild REN 54 35 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cn(C2CCC2)nn1 ZINC000880572217 GF On-Demand Mild FPR1 40 35 COc1ccc(CN(CCO)Cc2nc(=O)n(C)[nH]2)cc1 ZINC000880572221 CC On-Demand Anodyne PROKR1 41 30 CCN(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572227 CD On-Demand Anodyne TBXAS1 59 43 CCN(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572227 CD On-Demand Anodyne CYP26A1 55 35 CCN(C)C(=O)CN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572227 CD On-Demand Anodyne CYP27B1 45 33 CCN(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572229 CD On-Demand Anodyne TBXAS1 59 43 CCN(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572229 CD On-Demand Anodyne CYP26A1 55 35 CCN(C)C(=O)CN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572229 CD On-Demand Anodyne CYP27B1 45 33 O=S(=O)(CCCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880572232 FG On-Demand Anodyne TBXAS1 33 40 O=S(=O)(CCCN[C@@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880572232 FG On-Demand Anodyne CYP27B1 42 30 O=S(=O)(CCCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880572233 FG On-Demand Anodyne TBXAS1 33 40 O=S(=O)(CCCN[C@H](Cn1ccnc1)c1ccccc1)c1ccccc1 ZINC000880572233 FG On-Demand Anodyne CYP27B1 42 30 COCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572250 CF On-Demand Anodyne TBXAS1 38 41 COCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572250 CF On-Demand Anodyne CYP24A1 44 33 COCCCCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572250 CF On-Demand Anodyne CYP27B1 59 33 COCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572251 CF On-Demand Anodyne TBXAS1 38 41 COCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572251 CF On-Demand Anodyne CYP24A1 44 33 COCCCCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572251 CF On-Demand Anodyne CYP27B1 59 33 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC(C1CC1)C1CC1 ZINC000880572257 EF On-Demand Anodyne TBXAS1 54 41 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)NC(C1CC1)C1CC1 ZINC000880572257 EF On-Demand Anodyne CYP27B1 41 34 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC(C1CC1)C1CC1 ZINC000880572258 EF On-Demand Anodyne TBXAS1 54 41 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)NC(C1CC1)C1CC1 ZINC000880572258 EF On-Demand Anodyne CYP27B1 41 34 O=C(CN[C@@H](Cn1ccnc1)c1ccccc1)N(C1CCCC1)C1CC1 ZINC000880572274 FG On-Demand Anodyne TBXAS1 41 39 O=C(CN[C@H](Cn1ccnc1)c1ccccc1)N(C1CCCC1)C1CC1 ZINC000880572275 FG On-Demand Anodyne TBXAS1 41 39 CC(C)(C)OC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572278 DF On-Demand Anodyne TBXAS1 59 41 CC(C)(C)OC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572278 DF On-Demand Anodyne CYP24A1 47 39 CC(C)(C)OC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572278 DF On-Demand Anodyne CYP26A1 113 40 CC(C)(C)OC(=O)CCN[C@@H](Cn1ccnc1)c1ccccc1 ZINC000880572278 DF On-Demand Anodyne CYP27B1 61 39 CC(C)(C)OC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572279 DF On-Demand Anodyne TBXAS1 59 41 CC(C)(C)OC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572279 DF On-Demand Anodyne CYP24A1 47 39 CC(C)(C)OC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572279 DF On-Demand Anodyne CYP26A1 113 40 CC(C)(C)OC(=O)CCN[C@H](Cn1ccnc1)c1ccccc1 ZINC000880572279 DF On-Demand Anodyne CYP27B1 61 39 CCOC(=O)[C@@H]1CCCN(C(=O)CN[C@@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880572285 GE On-Demand Anodyne TBXAS1 23 40 CCOC(=O)[C@@H]1CCCN(C(=O)CN[C@H](Cn2ccnc2)c2ccccc2)C1 ZINC000880572288 GE On-Demand Anodyne TBXAS1 23 40 COc1ccc(CN(CCO)C[C@@H]2CCC[C@H](O)C2)cc1 ZINC000880572356 CE On-Demand Anodyne SLC18A2 21 40 COc1ccc(CN(CCO)C[C@H]2CCC[C@H](O)C2)cc1 ZINC000880572357 CE On-Demand Anodyne SLC18A2 21 40 COc1ccc(CN(CCO)C[C@@H]2CCC[C@@H](O)C2)cc1 ZINC000880572358 CE On-Demand Anodyne SLC18A2 21 40 COc1ccc(CN(CCO)C[C@H]2CCC[C@@H](O)C2)cc1 ZINC000880572359 CE On-Demand Anodyne SLC18A2 21 40 COc1ccc(CN(CCO)Cc2ccc(C#N)s2)cc1 ZINC000880572362 DF On-Demand Mild NR1D1 28 64 COc1ccc(CN(CCO)Cc2ccc([N+](=O)[O-])c(F)c2)cc1 ZINC000880572363 EF On-Demand Bother BMP1 22 41 COc1ccc(CN(CCO)CC(=O)NCC(C)(C)C)cc1 ZINC000880572368 DD On-Demand Anodyne MMP3 15 41 COc1ccc(CN(CCO)CC(=O)NCC(C)(C)C)cc1 ZINC000880572368 DD On-Demand Anodyne MMP12 18 41 COc1ccc(CN(CCO)CC(=O)NCC(C)(C)C)cc1 ZINC000880572368 DD On-Demand Anodyne MMP1 15 41 COc1ccc(CN(CCO)C[C@@H](O)c2ccc(Cl)cc2)cc1 ZINC000880572370 EF On-Demand Anodyne AOC3 19 48 COc1ccc(CN(CCO)C[C@H](O)c2ccc(Cl)cc2)cc1 ZINC000880572371 EF On-Demand Anodyne AOC3 19 48 COc1ccc(CN(CCO)CCC(=O)Nc2cccnc2)cc1 ZINC000880572372 ED On-Demand Anodyne NR1D1 15 41 CNS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880572373 DC On-Demand Anodyne MMP13 24 43 CNS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880572373 DC On-Demand Anodyne MMP3 18 41 CNS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880572373 DC On-Demand Anodyne MMP8 16 43 CNS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880572373 DC On-Demand Anodyne MMP12 24 43 CNS(=O)(=O)CCN(CCO)Cc1ccc(OC)cc1 ZINC000880572373 DC On-Demand Anodyne MMP1 26 41 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne AVPR1B 20 41 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne BMP1 82 39 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP13 74 44 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP2 48 44 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP3 59 44 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP8 42 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP14 19 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP9 64 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP12 31 42 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP7 44 43 COc1ccc(CN(CCO)Cc2ccc(S(=O)(=O)NC3CC3)cc2)cc1 ZINC000880572374 GE On-Demand Anodyne MMP1 62 44 COc1ccc(CN(CCO)CC2CCC3(CC2)OCCO3)cc1 ZINC000880572387 EE On-Demand Anodyne C5AR1 20 40 COc1ccc(CN(CCO)CCS(=O)(=O)N(C)C)cc1 ZINC000880572396 DC On-Demand Anodyne MMP12 17 42 COc1ccc(CN(CCO)C[C@@H](O)CC2CCCC2)cc1 ZINC000880572405 DE On-Demand Anodyne SLC18A2 21 43 COc1ccc(CN(CCO)C[C@H](O)CC2CCCC2)cc1 ZINC000880572406 DE On-Demand Anodyne SLC18A2 21 43 COc1ccc(CN(CCO)Cc2cccc(CN3CCOCC3)c2)cc1 ZINC000880572408 FF On-Demand Anodyne SIGMAR1 22 46 Cc1nnc(N2CCN(C(=O)Cn3ccc(C(F)(F)F)n3)CC2)n1C ZINC000880572410 FC On-Demand Anodyne CCR1 24 41 COc1ccc(CN(CCO)CCCN2CCN(C(C)C)CC2)cc1 ZINC000880572411 ED On-Demand Anodyne HRP1_PLAFA 18 44 COc1ccc(CN(CCO)CCCN2CCN(C(C)C)CC2)cc1 ZINC000880572411 ED On-Demand Anodyne HRH3 15 42 COc1ccc(CN(CCO)C[C@@H](O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880572417 EE On-Demand Bother MMP8 21 45 COc1ccc(CN(CCO)C[C@@H](O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880572417 EE On-Demand Bother MMP1 17 45 COc1ccc(CN(CCO)C[C@H](O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880572418 EE On-Demand Bother MMP8 21 45 COc1ccc(CN(CCO)C[C@H](O)c2ccc([N+](=O)[O-])cc2)cc1 ZINC000880572418 EE On-Demand Bother MMP1 17 45 COc1ccc(CN(CCO)CC2CN(C(=O)OC(C)(C)C)C2)cc1 ZINC000880572426 FE On-Demand Anodyne MMP3 15 42 COc1ccc(CN(CCO)CC(=O)N=[S@@](C)(=O)N(C)C)cc1 ZINC000880572428 EC On-Demand Anodyne MMP3 15 40 COc1ccc(CN(CCO)CC(=O)N=[S@@](C)(=O)N(C)C)cc1 ZINC000880572428 EC On-Demand Anodyne MMP12 17 40 COc1ccc(CN(CCO)CC(=O)N=[S@](C)(=O)N(C)C)cc1 ZINC000880572429 EC On-Demand Anodyne MMP3 15 40 COc1ccc(CN(CCO)CC(=O)N=[S@](C)(=O)N(C)C)cc1 ZINC000880572429 EC On-Demand Anodyne MMP12 17 40 COc1ccc(CN(CCO)CC2CCN(C(=O)C(C)(C)C)CC2)cc1 ZINC000880572460 FF On-Demand Anodyne MMP1 15 40 COc1ccc(CN(CCO)Cc2nnc(-c3ccc(Cl)cc3)n2C)cc1 ZINC000880572464 GG On-Demand Anodyne HSD11B1 18 40 COc1ccc(CN(CCO)CCC(=O)N2CCc3ccccc3C2)cc1 ZINC000880572465 FE On-Demand Anodyne BMP1 46 36 COc1ccc(CN(CCO)CCC(=O)N2CCc3ccccc3C2)cc1 ZINC000880572465 FE On-Demand Anodyne HDAC6 15 40 COc1ccc(CN(CCO)CCC(=O)N2CCc3ccccc3C2)cc1 ZINC000880572465 FE On-Demand Anodyne NOD1 15 44 COc1ccc(CN(CCO)CCC(=O)N2CCc3ccccc3C2)cc1 ZINC000880572465 FE On-Demand Anodyne NOD2 42 44 COc1ccc(CN(CCO)Cc2cc(Cl)cc(S(N)(=O)=O)c2)cc1 ZINC000880572466 GD On-Demand Anodyne CA2 20 43 COc1ccc(CN(CCO)Cc2cc(Cl)cc(S(N)(=O)=O)c2)cc1 ZINC000880572466 GD On-Demand Anodyne CA1 18 43 COc1ccc(CN(CCO)Cc2cc(Cl)cc(S(N)(=O)=O)c2)cc1 ZINC000880572466 GD On-Demand Anodyne CA12 23 43 COc1ccc(CN(CCO)Cc2cc(Cl)cc(S(N)(=O)=O)c2)cc1 ZINC000880572466 GD On-Demand Anodyne CA9 26 43 COc1ccc(CN(CCO)CC(=O)Nc2ccccn2)cc1 ZINC000880572468 DD On-Demand Anodyne MMP3 16 42 COc1ccc(CN(CCO)Cc2cn(Cc3ccccc3)nn2)cc1 ZINC000880572474 FE On-Demand Anodyne FIMH 17 45 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne MMP13 26 42 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne MMP3 32 42 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne MMP9 22 42 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne MMP7 25 42 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne MMP1 28 42 COc1ccc(CN(CCO)C[C@@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572507 EC On-Demand Anodyne NR1D1 26 49 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne MMP13 26 42 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne MMP3 32 42 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne MMP9 22 42 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne MMP7 25 42 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne MMP1 28 42 COc1ccc(CN(CCO)C[C@H]2CCN(S(C)(=O)=O)C2)cc1 ZINC000880572508 EC On-Demand Anodyne NR1D1 26 49 COc1ccc(CN(CCO)CCC(=O)C(C)C)cc1 ZINC000880572515 CE On-Demand Anodyne BMP1 43 39 COc1ccc(CN(CCO)Cc2cncc(Cl)c2)cc1 ZINC000880572516 DF On-Demand Anodyne CYP11B2 19 41 Cc1nnc(N2CCN(C(=O)COc3ccccc3-c3ccccc3)CC2)n1C ZINC000880572517 GF On-Demand Anodyne PLA2G1B 42 35 COc1ccc(CN(CCO)CC(=O)N=S(C)(C)=O)cc1 ZINC000880572519 DC On-Demand Anodyne MMP13 17 42 COc1ccc(CN(CCO)CC(=O)N=S(C)(C)=O)cc1 ZINC000880572519 DC On-Demand Anodyne MMP12 20 42 COc1ccc(CN(CCO)CC(=O)N=S(C)(C)=O)cc1 ZINC000880572519 DC On-Demand Anodyne MMP1 18 42 Cc1nnc(N2CCN(C(=O)COc3cccc(Br)c3)CC2)n1C ZINC000880572522 GD On-Demand Anodyne HTR1D 17 45 Cc1nnc(N2CCN(C(=O)COc3cccc(Br)c3)CC2)n1C ZINC000880572522 GD On-Demand Anodyne HTR1B 19 45 CNC(=O)CCCN(CCO)Cc1ccc(OC)cc1 ZINC000880572524 CD On-Demand Anodyne MMP3 15 40 CNC(=O)CCCN(CCO)Cc1ccc(OC)cc1 ZINC000880572524 CD On-Demand Anodyne MMP12 20 40 CNC(=O)CCCN(CCO)Cc1ccc(OC)cc1 ZINC000880572524 CD On-Demand Anodyne MMP1 20 40 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne PTGER2 18 45 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne BMP1 44 40 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP13 27 42 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP2 18 47 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP3 24 47 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP8 17 47 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP9 31 47 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP12 24 42 COc1ccc(CN(CCO)CCN(Cc2ccccc2)S(C)(=O)=O)cc1 ZINC000880572541 GD On-Demand Anodyne MMP1 28 47 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(N(C)C)cc2)cc1 ZINC000880572550 FF On-Demand Anodyne LTA4H 35 40 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(N(C)C)cc2)cc1 ZINC000880572550 FF On-Demand Anodyne BMP1 20 41 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(N(C)C)cc2)cc1 ZINC000880572550 FF On-Demand Anodyne MTNR1B 17 44 COc1ccc(CN(CCO)CCC(=O)Nc2ccc(N(C)C)cc2)cc1 ZINC000880572550 FF On-Demand Anodyne CA9 15 42 Cc1nnc(N2CCN(C(=O)c3cc(S(C)(=O)=O)ccc3Cl)CC2)n1C ZINC000880572556 GD On-Demand Anodyne SLC6A9 45 46 COc1ccc(CN(CCO)Cc2cncc(OC)c2)cc1 ZINC000880572561 DE On-Demand Anodyne CYP11B1 16 44 COc1ccc(CN(CCO)Cc2cncc(OC)c2)cc1 ZINC000880572561 DE On-Demand Anodyne CYP11B2 24 44 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne PTGS2 22 48 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne BMP1 76 48 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP13 51 46 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP2 29 41 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP3 39 46 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP8 29 46 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP9 50 42 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP12 32 46 COc1ccc(CN(CCO)Cc2ccc(S(C)(=O)=O)cc2)cc1 ZINC000880572568 EE On-Demand Anodyne MMP1 47 46 Cc1nnc(N2CCN(C(=O)COc3ccc4c(c3)CCC4)CC2)n1C ZINC000880572594 FD On-Demand Anodyne HTR1D 16 45 Cc1nnc(N2CCN(C(=O)COc3ccc4c(c3)CCC4)CC2)n1C ZINC000880572594 FD On-Demand Anodyne HTR1B 19 45 Cc1nnc(N2CCN(C(=O)COc3ccc4ccc(=O)oc4c3)CC2)n1C ZINC000880572597 GC On-Demand Anodyne MAOA 49 38 Cc1nnc(N2CCN(C(=O)COc3ccc4ccc(=O)oc4c3)CC2)n1C ZINC000880572597 GC On-Demand Anodyne HTR1D 15 44 Cc1nnc(N2CCN(C(=O)COc3ccc4ccc(=O)oc4c3)CC2)n1C ZINC000880572597 GC On-Demand Anodyne HTR1B 19 44 COc1ccc(CN(CCO)C[C@H](OC)c2ccc(F)cc2)cc1 ZINC000880572618 EG On-Demand Anodyne AOC3 20 48 COc1ccc(CN(CCO)C[C@@H](OC)c2ccc(F)cc2)cc1 ZINC000880572619 EG On-Demand Anodyne AOC3 20 48 COc1ccc(CN(CCO)Cc2cncc3ccccc23)cc1 ZINC000880572631 DG On-Demand Anodyne CYP11B2 15 49 CC(=O)c1cccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880572633 FD On-Demand Anodyne DRD4 42 33 CC(=O)c1cccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880572633 FD On-Demand Anodyne HTR1D 17 44 CC(=O)c1cccc(OCC(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880572633 FD On-Demand Anodyne HTR1B 19 44 Cc1nnc(N2CCN(C(=O)[C@@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572659 GD On-Demand Anodyne PREP 42 61 Cc1nnc(N2CCN(C(=O)[C@@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572659 GD On-Demand Anodyne SFRP1 23 40 Cc1nnc(N2CCN(C(=O)[C@@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572659 GD On-Demand Anodyne WNT3 33 40 Cc1nnc(N2CCN(C(=O)[C@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572660 GD On-Demand Anodyne PREP 42 61 Cc1nnc(N2CCN(C(=O)[C@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572660 GD On-Demand Anodyne SFRP1 23 40 Cc1nnc(N2CCN(C(=O)[C@H]3CCCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880572660 GD On-Demand Anodyne WNT3 33 40 Cc1cc(C)c2cc(C(=O)N3CCN(c4nnc(C)n4C)CC3)[nH]c2c1 ZINC000880572677 FE On-Demand Anodyne HRH4 29 44 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne ACE 35 42 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne P2RY12 48 37 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CELA1 15 44 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne ELANE 30 42 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne MME 17 42 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CTRA_BOVIN 41 31 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CASP3 15 44 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne KLK3 75 36 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CTSB 64 45 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne TRY2_BOVIN 58 34 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne PAPA1_CARPA 73 36 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CYSP_TRYCR 53 38 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CTSK 40 45 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CTSL 47 38 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CAPNS1 64 38 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne LGMN 15 41 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CTSS 21 45 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CAPN1 83 41 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne CAPN2 128 39 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne PLAU 20 40 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne TGM2 38 44 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne NPR 67 34 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne PSMB5 42 38 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne Q6PRC7_IXORI 62 42 Cc1nnc(N2CCN(C(=O)[C@H](C)NC(=O)OCc3ccccc3)CC2)n1C ZINC000880572688 GD On-Demand Anodyne SLC12A5 42 32 Cc1nn(CC(=O)N2CCN(c3nnc(C)n3C)CC2)c(C)c1Cl ZINC000880572714 FC On-Demand Anodyne CCR1 27 53 CCOC(=O)Nc1ccc(C(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880572721 FD On-Demand Anodyne ACR 40 33 COc1ccc(CN(CCO)CC(=O)NC2CCN(S(C)(=O)=O)CC2)cc1 ZINC000880572723 GC On-Demand Anodyne MMP3 42 39 COc1ccc(CN(CCO)CC(=O)NC2CCN(S(C)(=O)=O)CC2)cc1 ZINC000880572723 GC On-Demand Anodyne EPHX2 17 42 COc1ccc(CN(CCO)CC(=O)NC2CCN(S(C)(=O)=O)CC2)cc1 ZINC000880572723 GC On-Demand Anodyne MMP1 40 39 COc1ccc(CN(CCO)CC(=O)NC2CCN(S(C)(=O)=O)CC2)cc1 ZINC000880572723 GC On-Demand Anodyne RORC 17 42 COc1ccc(CN(CCO)CCc2ccc(C(N)=O)cc2)cc1 ZINC000880572727 ED On-Demand Anodyne BMP1 19 41 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880572756 GD On-Demand Anodyne P2RY12 63 35 Cc1nnc(N2CCN(C(=O)Cc3c[nH]c4cc(F)ccc34)CC2)n1C ZINC000880572767 FD On-Demand Anodyne MPO 48 36 COC(=O)CCN(CC(=O)OC(C)(C)C)Cc1nc2ccccc2[nH]1 ZINC000880572773 EE On-Demand Anodyne CACNA1G 22 40 COc1ccc(CN(CCO)CCCC2CC2)cc1 ZINC000880572802 CF On-Demand Anodyne SLC18A2 22 40 Cc1nnc(N2CCN(C(=O)c3cc4c(Cl)c(Cl)ccc4[nH]3)CC2)n1C ZINC000880572809 GF On-Demand Anodyne HRH4 34 67 Cc1nnc(N2CCN(C(=O)C[C@@H](c3ccccc3)N3CCOC3=O)CC2)n1C ZINC000880572832 GD On-Demand Anodyne PTAFR 22 56 Cc1nnc(N2CCN(C(=O)C[C@H](c3ccccc3)N3CCOC3=O)CC2)n1C ZINC000880572833 GD On-Demand Anodyne PTAFR 22 56 Cc1nnc(N2CCN(C(=O)COc3cccnc3)CC2)n1C ZINC000880572835 DC On-Demand Anodyne HTR1B 15 40 Cc1nnc(N2CCN(C(=O)COc3cccnc3)CC2)n1C ZINC000880572835 DC On-Demand Anodyne CPT1A 15 40 CCC(=O)N1CSC[C@@H]1C(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880572845 FC On-Demand Anodyne PREP 15 40 CCC(=O)N1CSC[C@H]1C(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880572846 FC On-Demand Anodyne PREP 15 40 COc1ccc(CC(=O)N2CCN(c3nnc(C)n3C)CC2)cc1F ZINC000880572848 ED On-Demand Anodyne CCR1 19 40 COc1ccc(CC(=O)N2CCN(c3nnc(C)n3C)CC2)cc1F ZINC000880572848 ED On-Demand Anodyne KCNJ1 40 36 COc1ccc(CN(CCO)Cc2nc(O)c3c(n2)CCOC3)cc1 ZINC000880572850 ED On-Demand Anodyne TNKS2 22 40 Cc1nnc(N2CCN(C(=O)c3cc4ccccc4c(Cl)n3)CC2)n1C ZINC000880572912 FE On-Demand Anodyne CCKAR 40 40 Cc1nnc(N2CCN(C(=O)[C@@H](C)Oc3cccc(CO)c3)CC2)n1C ZINC000880572917 FC On-Demand Anodyne TRY2_BOVIN 52 34 Cc1nnc(N2CCN(C(=O)[C@H](C)Oc3cccc(CO)c3)CC2)n1C ZINC000880572918 FC On-Demand Anodyne TRY2_BOVIN 52 34 Cc1nnc(N2CCN(C(=O)c3ccc(C(F)(F)F)cc3O)CC2)n1C ZINC000880572928 FD On-Demand Anodyne SLC6A9 25 40 Cc1nnc(N2CCN(C(=O)c3cc(N4CCOC4=O)ccc3F)CC2)n1C ZINC000880572934 GD On-Demand Anodyne PARP1 40 34 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne PTAFR 15 41 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CTSB 46 40 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CYSP_TRYCR 41 36 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CTSK 27 40 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CAPNS1 56 32 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CAPN1 62 34 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne CAPN2 100 34 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne TGM2 31 41 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne NPR 62 35 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne Q6PRC7_IXORI 42 35 Cc1nnc(N2CCN(C(=O)CNC(=O)OCc3ccccc3)CC2)n1C ZINC000880572971 FC On-Demand Anodyne SLC12A5 51 33 CCCCSCC(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880572984 DD On-Demand Anodyne EST1_PIG 43 37 COc1ccc(CN(CCO)C[C@@H](O)C[C@@H](O)c2ccccc2)cc1 ZINC000880572986 ED On-Demand Anodyne AOC3 18 40 COc1ccc(CN(CCO)C[C@@H](O)C[C@H](O)c2ccccc2)cc1 ZINC000880572987 ED On-Demand Anodyne AOC3 18 40 COc1ccc(CN(CCO)C[C@H](O)C[C@H](O)c2ccccc2)cc1 ZINC000880572988 ED On-Demand Anodyne AOC3 18 40 COc1ccc(CN(CCO)C[C@H](O)C[C@@H](O)c2ccccc2)cc1 ZINC000880572989 ED On-Demand Anodyne AOC3 18 40 Cc1nnc(N2CCN(C(=O)c3cn(C)c4ccccc34)CC2)n1C ZINC000880572993 ED On-Demand Anodyne TPSAB1 18 45 Cc1nnc(N2CCN(C(=O)c3cc4ccc(C(C)C)cc4[nH]3)CC2)n1C ZINC000880573001 FF On-Demand Anodyne GRIN2B 16 40 Cc1nnc(N2CCN(C(=O)c3cc4ccc(C(C)C)cc4[nH]3)CC2)n1C ZINC000880573001 FF On-Demand Anodyne HRH4 35 51 COC(=O)Nc1ccc(C(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880573019 FD On-Demand Anodyne PDGFRB 42 35 Cc1nnc(N2CCN(C(=O)[C@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573038 ED On-Demand Anodyne MC4R 47 47 Cc1nnc(N2CCN(C(=O)[C@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573038 ED On-Demand Anodyne MC3R 21 40 Cc1nnc(N2CCN(C(=O)[C@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573038 ED On-Demand Anodyne MC5R 29 41 Cc1nnc(N2CCN(C(=O)[C@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573038 ED On-Demand Anodyne AKT1 20 45 Cc1nnc(N2CCN(C(=O)[C@@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573039 ED On-Demand Anodyne MC4R 47 47 Cc1nnc(N2CCN(C(=O)[C@@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573039 ED On-Demand Anodyne MC3R 21 40 Cc1nnc(N2CCN(C(=O)[C@@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573039 ED On-Demand Anodyne MC5R 29 41 Cc1nnc(N2CCN(C(=O)[C@@H](C)Cc3ccc(F)cc3)CC2)n1C ZINC000880573039 ED On-Demand Anodyne AKT1 20 45 COc1ccc(CN(CCO)CC(C)=O)cc1 ZINC000880573046 BD On-Demand Anodyne MMP12 17 42 COc1ccc(CN(CCO)CC(C)=O)cc1 ZINC000880573046 BD On-Demand Anodyne MMP1 17 42 COC(=O)CCN(CC(=O)OC(C)(C)C)[C@H](C)c1cccnc1 ZINC000880573115 DE On-Demand Anodyne KCNA5 23 47 COC(=O)CCN(CC(=O)OC(C)(C)C)[C@@H](C)c1cccnc1 ZINC000880573116 DE On-Demand Anodyne KCNA5 23 47 COc1ccc(CN(CCO)Cc2ccc(C)c([N+](=O)[O-])c2)cc1 ZINC000880573131 EF On-Demand Bother BMP1 15 46 COc1ccc(CN(CCO)Cc2ccc(C)c([N+](=O)[O-])c2)cc1 ZINC000880573131 EF On-Demand Bother NR1D1 20 41 COc1ccc(CN(CCO)CC(=O)NC2CCN(C)CC2)cc1 ZINC000880573135 EC On-Demand Anodyne SIGMAR1 17 49 COc1ccc(CN(CCO)CC(=O)NC2CCN(C)CC2)cc1 ZINC000880573135 EC On-Demand Anodyne SLC6A5 31 41 COc1ccc(CN(CCO)CC(=O)NC2CCN(C)CC2)cc1 ZINC000880573135 EC On-Demand Anodyne MCHR1 19 45 Cc1nnc(N2CCN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)CC2)n1C ZINC000880573137 GD On-Demand Anodyne REN 24 40 Cc1nnc(N2CCN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)CC2)n1C ZINC000880573137 GD On-Demand Anodyne FPR1 47 36 Cc1nnc(N2CCN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)CC2)n1C ZINC000880573138 GD On-Demand Anodyne REN 24 40 Cc1nnc(N2CCN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)CC2)n1C ZINC000880573138 GD On-Demand Anodyne FPR1 47 36 Cc1nnc(N2CCN(C(=O)c3csc(C4CC4)n3)CC2)n1C ZINC000880573139 ED On-Demand Anodyne TRPC6 42 40 Cc1nnc(N2CCN(C(=O)c3csc(C4CC4)n3)CC2)n1C ZINC000880573139 ED On-Demand Anodyne TRPC3 35 40 Cc1nnc(N2CCN(C(=O)CSc3ccc([N+](=O)[O-])cc3)CC2)n1C ZINC000880573184 GD On-Demand Bother SSTR1 37 40 Cc1nnc(N2CCN(C(=O)c3[nH]c4ccccc4c3Cl)CC2)n1C ZINC000880573187 FE On-Demand Anodyne HRH4 17 44 Cc1nnc(N2CCN(C(=O)c3[nH]c4ccc(F)cc4c3Cl)CC2)n1C ZINC000880573215 GE On-Demand Anodyne HRH4 19 41 Cc1nnc(N2CCN(C(=O)C3CCN(C(=O)OC(C)(C)C)CC3)CC2)n1C ZINC000880573216 GD On-Demand Anodyne GPR119 41 42 Cc1nnc(N2CCN(C(=O)c3ccccc3-n3cnnn3)CC2)n1C ZINC000880573248 FC On-Demand Anodyne KCNJ1 53 34 Cc1nnc(N2CCN(C(=O)COc3ccc4c(c3)CCC(=O)N4)CC2)n1C ZINC000880573273 GC On-Demand Anodyne DRD2 15 43 Cc1nnc(N2CCN(C(=O)COc3ccc4c(c3)CCC(=O)N4)CC2)n1C ZINC000880573273 GC On-Demand Anodyne HTR1D 16 41 Cc1nnc(N2CCN(C(=O)COc3ccc4c(c3)CCC(=O)N4)CC2)n1C ZINC000880573273 GC On-Demand Anodyne HTR1B 19 41 COc1cccc(OC)c1C(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880573280 ED On-Demand Anodyne SSTR1 40 33 COc1cccc(OC)c1C(=O)N1CCN(c2nnc(C)n2C)CC1 ZINC000880573280 ED On-Demand Anodyne ALS 42 36 Cc1nnc(N2CCN(C(=O)C(=O)NCCCc3ccccc3)CC2)n1C ZINC000880573305 FC On-Demand Anodyne AMP1_PLAFQ 22 41 Cc1nnc(N2CCN(C(=O)CSc3ccc4ccccc4c3)CC2)n1C ZINC000880573364 GF On-Demand Anodyne TRY2_BOVIN 40 31 Cc1nnc(N2CCN(C(=O)COc3cccc(C#N)c3)CC2)n1C ZINC000880573371 EC On-Demand Mild HTR1D 15 47 Cc1nnc(N2CCN(C(=O)COc3cccc(C#N)c3)CC2)n1C ZINC000880573371 EC On-Demand Mild HTR1B 18 47 Cc1nnc(N2CCN(C(=O)COc3ccc(C(C)C)cc3)CC2)n1C ZINC000880573406 FD On-Demand Anodyne HTR1D 15 40 Cc1nnc(N2CCN(C(=O)COc3ccc(C(C)C)cc3)CC2)n1C ZINC000880573406 FD On-Demand Anodyne HTR1B 17 40 Cc1nnc(N2CCN(C(=O)c3cccc(Cl)c3O)CC2)n1C ZINC000880573445 ED On-Demand Anodyne P2RX7 41 42 Cc1nnc(N2CCN(C(=O)c3ccccc3C(C)(C)C)CC2)n1C ZINC000880573455 EE On-Demand Anodyne SCD1 21 44 Cc1nnc(N2CCN(C(=O)c3ccccc3C(C)(C)C)CC2)n1C ZINC000880573455 EE On-Demand Anodyne SCD 19 43 Cc1nnc(N2CCN(C(=O)c3cc4occc4[nH]3)CC2)n1C ZINC000880573462 DD On-Demand Anodyne HRH4 30 41 Cc1nnc(N2CCN(C(=O)c3ccccc3N3CCOCC3)CC2)n1C ZINC000880573464 FC On-Demand Anodyne SLC6A9 15 42 Cc1nnc(N2CCN(C(=O)c3ccccc3N3CCOCC3)CC2)n1C ZINC000880573464 FC On-Demand Anodyne AKR1C3 15 42 Cc1ccc(N2CCCC2)c(C(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880573486 FD On-Demand Anodyne HCRTR1 43 43 Cc1ccc(N2CCCC2)c(C(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880573486 FD On-Demand Anodyne SLC6A9 22 45 Cc1ccc(N2CCCC2)c(C(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880573486 FD On-Demand Anodyne HCRTR2 25 43 NC(=O)COc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880573635 EF On-Demand Anodyne HRH3 34 46 NC(=O)COc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880573635 EF On-Demand Anodyne CPT1A 41 36 NC(=O)COc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880573636 EF On-Demand Anodyne HRH3 34 46 NC(=O)COc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880573636 EF On-Demand Anodyne CPT1A 41 36 CNc1nc(C(=O)N2CCN(c3nnc(C)n3C)CC2)cs1 ZINC000880573743 DC On-Demand Anodyne TRPC6 63 45 CNc1nc(C(=O)N2CCN(c3nnc(C)n3C)CC2)cs1 ZINC000880573743 DC On-Demand Anodyne TRPC3 56 45 Cc1nnc(N2CCN(C(=O)c3csc(Cl)n3)CC2)n1C ZINC000880573763 ED On-Demand Anodyne TRPC6 45 39 O=S(=O)(CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880573773 FF On-Demand Anodyne SLC6A1 47 34 O=S(=O)(CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880573774 FF On-Demand Anodyne SLC6A1 47 34 Cc1nnc(N2CCN(C(=O)[C@@H](F)Cc3ccccc3)CC2)n1C ZINC000880573802 ED On-Demand Anodyne TRY2_BOVIN 55 33 Cc1nnc(N2CCN(C(=O)[C@H](F)Cc3ccccc3)CC2)n1C ZINC000880573803 ED On-Demand Anodyne TRY2_BOVIN 55 33 CC(C)(C)CCN(CCCC(=O)O)CCc1ccccc1 ZINC000880573808 CH On-Demand Anodyne CES1 52 40 CC(C)(C)CCN(CCCC(=O)O)CCc1ccccc1 ZINC000880573808 CH On-Demand Anodyne FFAR1 40 40 Cc1nnc(N2CCN(C(=O)c3ccccc3OC3CC3)CC2)n1C ZINC000880573850 ED On-Demand Anodyne SCD1 45 40 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1ccccc1 ZINC000880573853 EF On-Demand Anodyne SIGMAR1 20 44 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1ccccc1 ZINC000880573853 EF On-Demand Anodyne PREP 29 40 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1ccccc1 ZINC000880573854 EF On-Demand Anodyne SIGMAR1 20 44 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1ccccc1 ZINC000880573854 EF On-Demand Anodyne PREP 29 40 Cc1nnc(N2CCN(C(=O)[C@@H]3C[C@H]3c3ccccc3)CC2)n1C ZINC000880573857 ED On-Demand Anodyne NPBWR1 60 32 c1ccc2[nH]c(CN3CCCC[C@H](C4CCOCC4)C3)nc2c1 ZINC000880573868 DH On-Demand Anodyne KCNN3 30 40 c1ccc2[nH]c(CN3CCCC[C@@H](C4CCOCC4)C3)nc2c1 ZINC000880573869 DH On-Demand Anodyne KCNN3 30 40 c1csc(-c2noc(CN3CCCC[C@H](C4CCOCC4)C3)n2)c1 ZINC000880573883 EH On-Demand Anodyne ETHR 31 41 c1csc(-c2noc(CN3CCCC[C@@H](C4CCOCC4)C3)n2)c1 ZINC000880573884 EH On-Demand Anodyne ETHR 31 41 c1cc(CCN2CCCC[C@@H](C3CCOCC3)C2)ccn1 ZINC000880573894 CG On-Demand Anodyne L3MBTL3 31 41 c1cc(CCN2CCCC[C@H](C3CCOCC3)C2)ccn1 ZINC000880573895 CG On-Demand Anodyne L3MBTL3 31 41 Cc1nnc(N2CCN(C(=O)c3ccc(-c4ccccc4)n3C)CC2)n1C ZINC000880573937 FE On-Demand Anodyne SMO 32 42 O[C@@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccc(F)cc1 ZINC000880573954 DG On-Demand Anodyne SLC6A3 18 40 O[C@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccc(F)cc1 ZINC000880573955 DG On-Demand Anodyne SLC6A3 18 40 O[C@@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccc(F)cc1 ZINC000880573957 DG On-Demand Anodyne SLC6A3 18 40 O[C@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccc(F)cc1 ZINC000880573958 DG On-Demand Anodyne SLC6A3 18 40 Cc1nnc(N2CCN(C(=O)COCc3cccnc3)CC2)n1C ZINC000880573970 EC On-Demand Anodyne PTAFR 15 41 Cc1nnc(N2CCN(C(=O)COCc3cccnc3)CC2)n1C ZINC000880573970 EC On-Demand Anodyne CHRNA7 41 35 Cc1nnc(N2CCN(C(=O)[C@H](O)c3cccnc3)CC2)n1C ZINC000880573986 DB On-Demand Anodyne PTAFR 16 44 Cc1nnc(N2CCN(C(=O)[C@@H](O)c3cccnc3)CC2)n1C ZINC000880573989 DB On-Demand Anodyne PTAFR 16 44 CC(C)(C)CCN(CCC(=O)O)CCc1ccccc1 ZINC000880574045 CG On-Demand Anodyne MME 19 40 CC(C)(C)CCN(CCC(=O)O)CCc1ccccc1 ZINC000880574045 CG On-Demand Anodyne CES1 41 39 CC(C)(C)CCN(CCC(=O)O)CCc1ccccc1 ZINC000880574045 CG On-Demand Anodyne FFAR1 52 44 Cc1nnc(N2CCN(C(=O)CCCn3ccnc3)CC2)n1C ZINC000880574046 DC On-Demand Anodyne TBXAS1 44 41 C#CCCOc1ccc(C(=O)N2CCN(c3nnc(C)n3C)CC2)cc1 ZINC000880574049 FD On-Demand Mild HRH3 17 43 Cc1nnc(N2CCN(C(=O)c3ncccc3Oc3ccccc3)CC2)n1C ZINC000880574087 GE On-Demand Anodyne CCR8 21 40 CC(C)(C)CCN(CCc1ccccc1)CC(=O)NCC#N ZINC000880574088 DF On-Demand Mild PAPA1_CARPA 45 40 CC(C)(C)CCN(CCc1ccccc1)CC(=O)NCC#N ZINC000880574088 DF On-Demand Mild CTSL 22 41 CC(C)(C)CCN(CCc1ccccc1)CC(=O)NCC#N ZINC000880574088 DF On-Demand Mild CTSS 19 43 CC(=O)Nc1cccc(CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574094 EH On-Demand Anodyne CCR3 52 39 CC(=O)Nc1cccc(CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574094 EH On-Demand Anodyne EPHX2 19 41 CC(=O)Nc1cccc(CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574094 EH On-Demand Anodyne MCHR1 33 43 CC(=O)Nc1cccc(CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574095 EH On-Demand Anodyne CCR3 52 39 CC(=O)Nc1cccc(CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574095 EH On-Demand Anodyne EPHX2 19 41 CC(=O)Nc1cccc(CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574095 EH On-Demand Anodyne MCHR1 33 43 COC(=O)CCN(CC(=O)OC(C)(C)C)Cc1ccc(C#N)s1 ZINC000880574127 EE On-Demand Mild NR1D1 19 42 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574162 DG On-Demand Anodyne SLC6A1 50 34 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574162 DG On-Demand Anodyne CHRNA7 17 43 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574162 DG On-Demand Anodyne EPHX2 22 40 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574163 DG On-Demand Anodyne SLC6A1 50 34 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574163 DG On-Demand Anodyne CHRNA7 17 43 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574163 DG On-Demand Anodyne EPHX2 22 40 O=[S@](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574180 EG On-Demand Anodyne SLC6A1 53 41 O=[S@@](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574181 EG On-Demand Anodyne SLC6A1 53 41 O=[S@@](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574182 EG On-Demand Anodyne SLC6A1 53 41 O=[S@](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574183 EG On-Demand Anodyne SLC6A1 53 41 c1ccc(-c2nc(CN3CCCC[C@@H](C4CCOCC4)C3)no2)cc1 ZINC000880574186 EH On-Demand Anodyne PDE8B 17 41 c1ccc(-c2nc(CN3CCCC[C@H](C4CCOCC4)C3)no2)cc1 ZINC000880574187 EH On-Demand Anodyne PDE8B 17 41 O[C@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574212 EF On-Demand Anodyne ADRB2 20 48 O[C@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574212 EF On-Demand Anodyne ADRB1 23 44 O[C@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574212 EF On-Demand Anodyne CPT1A 51 36 O[C@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574212 EF On-Demand Anodyne ABCB1 68 47 O[C@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574216 EF On-Demand Anodyne ADRB2 20 48 O[C@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574216 EF On-Demand Anodyne ADRB1 23 44 O[C@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574216 EF On-Demand Anodyne CPT1A 51 36 O[C@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574216 EF On-Demand Anodyne ABCB1 68 47 O[C@@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574219 EF On-Demand Anodyne ADRB2 20 48 O[C@@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574219 EF On-Demand Anodyne ADRB1 23 44 O[C@@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574219 EF On-Demand Anodyne CPT1A 51 36 O[C@@H](COc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574219 EF On-Demand Anodyne ABCB1 68 47 O[C@@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574221 EF On-Demand Anodyne ADRB2 20 48 O[C@@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574221 EF On-Demand Anodyne ADRB1 23 44 O[C@@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574221 EF On-Demand Anodyne CPT1A 51 36 O[C@@H](COc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574221 EF On-Demand Anodyne ABCB1 68 47 Cc1nnc(N2CCN(C(=O)[C@H]3CCCN3C(=O)C(F)(F)F)CC2)n1C ZINC000880574227 FC On-Demand Anodyne WNT3 40 31 Cc1nnc(N2CCN(C(=O)[C@@H]3CCCN3C(=O)C(F)(F)F)CC2)n1C ZINC000880574228 FC On-Demand Anodyne WNT3 40 31 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild PRNP 51 35 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild KDR 46 39 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild ABCB1B 24 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild GRM4 44 45 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild NR1H4 17 43 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild GRM5 20 43 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild ABCB1 15 41 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild ABCG2 32 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild SMO 37 45 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild KCNK3 126 52 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1OC ZINC000880574260 JK On-Demand Mild KCNK9 86 44 N#Cc1ccnc(N2CCN(C(=O)/C=C\c3ccccc3F)CC2)c1 ZINC000880574295 EE On-Demand Mild ITGAL 40 31 N#Cc1ccnc(N2CCN(C(=O)/C=C\c3cc(C(F)(F)F)ccc3Cl)CC2)c1 ZINC000880574325 HH On-Demand Mild ITGAL 45 32 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574356 EH On-Demand Anodyne SLC6A1 113 37 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574356 EH On-Demand Anodyne CHRNA7 19 46 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574356 EH On-Demand Anodyne TERT 16 43 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574357 EH On-Demand Anodyne SLC6A1 113 37 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574357 EH On-Demand Anodyne CHRNA7 19 46 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1 ZINC000880574357 EH On-Demand Anodyne TERT 16 43 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574365 GF On-Demand Anodyne ADRB2 15 45 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574365 GF On-Demand Anodyne HTR1A 17 41 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574365 GF On-Demand Anodyne ABCB1 61 47 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574366 GF On-Demand Anodyne ADRB2 15 45 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574366 GF On-Demand Anodyne HTR1A 17 41 COc1cccc(OC)c1OC[C@@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574366 GF On-Demand Anodyne ABCB1 61 47 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574367 GF On-Demand Anodyne ADRB2 15 45 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574367 GF On-Demand Anodyne HTR1A 17 41 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574367 GF On-Demand Anodyne ABCB1 61 47 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574368 GF On-Demand Anodyne ADRB2 15 45 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574368 GF On-Demand Anodyne HTR1A 17 41 COc1cccc(OC)c1OC[C@H](O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574368 GF On-Demand Anodyne ABCB1 61 47 C/C(=C/C(=O)N1CCN(c2nnc(C)n2C)CC1)c1ccccc1C(F)(F)F ZINC000880574495 GF On-Demand Anodyne RBP4 47 34 C/C(=C/C(=O)N1CCN(c2nnc(C)n2C)CC1)c1ccccc1C(F)(F)F ZINC000880574495 GF On-Demand Anodyne SCD1 23 42 C/C(=C/C(=O)N1CCN(c2nnc(C)n2C)CC1)c1ccccc1C(F)(F)F ZINC000880574495 GF On-Demand Anodyne SCD 23 41 Cc1nnc(N2CCN(C(=O)[C@@H](O)Cc3ccccc3Cl)CC2)n1C ZINC000880574498 FD On-Demand Anodyne MC4R 45 37 Cc1nnc(N2CCN(C(=O)[C@H](O)Cc3ccccc3Cl)CC2)n1C ZINC000880574499 FD On-Demand Anodyne MC4R 45 37 Cc1nnc(N2CCN(C(=O)c3ccnc(Br)c3)CC2)n1C ZINC000880574502 FD On-Demand Anodyne HPGD 42 36 COC(=O)CCN(CC(=O)OC(C)(C)C)C[C@H]1CCCN1C ZINC000880574544 DD On-Demand Anodyne ACKR3 59 30 COC(=O)CCN(CC(=O)OC(C)(C)C)C[C@@H]1CCCN1C ZINC000880574545 DD On-Demand Anodyne ACKR3 59 30 Cc1nnc(N2CCN(C(=O)c3cc(C(F)(F)F)ccc3F)CC2)n1C ZINC000880574546 FE On-Demand Anodyne SLC6A9 31 40 Cc1nnc(N2CCN(C(=O)c3cc(C(F)(F)F)ccc3F)CC2)n1C ZINC000880574546 FE On-Demand Anodyne PARP1 47 36 Cc1nnc(N2CCN(C(=O)c3cc(C(F)(F)F)ccc3F)CC2)n1C ZINC000880574546 FE On-Demand Anodyne LIPG 47 33 Cc1nnc(N2CCN(C(=O)c3c[nH]nc3-c3cccc(Cl)c3)CC2)n1C ZINC000880574550 GE On-Demand Anodyne P2RX7 23 40 Cc1nnc(N2CCN(C(=O)c3c[nH]nc3-c3cccc(Cl)c3)CC2)n1C ZINC000880574550 GE On-Demand Anodyne CCKAR 16 40 Cc1nnc(N2CCN(C(=O)c3cccc(Cl)c3[N+](=O)[O-])CC2)n1C ZINC000880574552 FD On-Demand Bother P2RX7 34 44 Cc1nnc(N2CCN(C(=O)c3ccccc3OCC(C)C)CC2)n1C ZINC000880574587 FE On-Demand Anodyne ABCB1 40 38 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne ESR1 85 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne ESR2 56 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne LTA4H 53 43 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne CA7 21 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne HRH3 44 45 NS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574672 GE On-Demand Anodyne PSMB1 44 39 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne ESR1 85 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne ESR2 56 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne LTA4H 53 43 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne CA7 21 40 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne HRH3 44 45 NS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574673 GE On-Demand Anodyne PSMB1 44 39 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1F ZINC000880574704 EH On-Demand Anodyne SLC6A1 84 37 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1ccccc1F ZINC000880574704 EH On-Demand Anodyne CHRNA7 16 40 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1F ZINC000880574705 EH On-Demand Anodyne SLC6A1 84 37 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1ccccc1F ZINC000880574705 EH On-Demand Anodyne CHRNA7 16 40 CC(=O)Nc1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574719 FG On-Demand Anodyne EPHX2 20 42 CC(=O)Nc1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574721 FG On-Demand Anodyne EPHX2 20 42 COC(=O)CCN(CC(=O)OC(C)(C)C)Cc1cc2ccccc2n(C)c1=O ZINC000880574727 GE On-Demand Anodyne NPSR1 34 43 N#CCc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574747 FG On-Demand Mild ABCB1 24 40 N#CCc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574751 FG On-Demand Mild ABCB1 24 40 N#CCc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574755 FG On-Demand Mild ABCB1 24 40 N#CCc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574758 FG On-Demand Mild ABCB1 24 40 Cc1nnc(N2CCN(C(=O)[C@H]3CC(=O)N(c4ccc(F)cc4)C3)CC2)n1C ZINC000880574762 GC On-Demand Anodyne SSTR1 53 38 Cc1nnc(N2CCN(C(=O)[C@@H]3CC(=O)N(c4ccc(F)cc4)C3)CC2)n1C ZINC000880574772 GC On-Demand Anodyne SSTR1 53 38 Cc1nnc(N2CCN(C(=O)c3cccnc3F)CC2)n1C ZINC000880574774 DC On-Demand Anodyne P2RX7 20 40 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574797 GG On-Demand Anodyne HRH3 17 44 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574797 GG On-Demand Anodyne ACOX1 43 32 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574797 GG On-Demand Anodyne ABCB1 53 47 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574798 GG On-Demand Anodyne HRH3 17 44 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574798 GG On-Demand Anodyne ACOX1 43 32 CC(=O)c1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574798 GG On-Demand Anodyne ABCB1 53 47 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574799 GG On-Demand Anodyne HRH3 17 44 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574799 GG On-Demand Anodyne ACOX1 43 32 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574799 GG On-Demand Anodyne ABCB1 53 47 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574800 GG On-Demand Anodyne HRH3 17 44 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574800 GG On-Demand Anodyne ACOX1 43 32 CC(=O)c1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574800 GG On-Demand Anodyne ABCB1 53 47 N#Cc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880574846 CH On-Demand Mild HRH3 24 45 N#Cc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880574847 CH On-Demand Mild HRH3 24 45 O[C@@H](COCc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574910 EG On-Demand Anodyne ABCB1 35 42 O[C@@H](COCc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574911 EG On-Demand Anodyne ABCB1 35 42 O[C@H](COCc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880574912 EG On-Demand Anodyne ABCB1 35 42 O[C@H](COCc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880574913 EG On-Demand Anodyne ABCB1 35 42 N#Cc1cccc(CNC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574919 FF On-Demand Mild CCR3 15 41 N#Cc1cccc(CNC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880574919 FF On-Demand Mild MCHR1 26 40 N#Cc1cccc(CNC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574920 FF On-Demand Mild CCR3 15 41 N#Cc1cccc(CNC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880574920 FF On-Demand Mild MCHR1 26 40 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CHRM2 17 42 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CHRM1 15 42 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne SLC6A1 50 33 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CHRM4 15 42 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CHRM5 19 42 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CHRM3 25 42 C[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574961 DG On-Demand Anodyne CYP2J2 44 33 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CHRM2 17 42 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CHRM1 15 42 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne SLC6A1 50 33 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CHRM4 15 42 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CHRM5 19 42 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CHRM3 25 42 C[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880574964 DG On-Demand Anodyne CYP2J2 44 33 O=C(c1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1)N1CCCC1 ZINC000880574972 FH On-Demand Anodyne HRH3 30 48 O=C(c1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1)N1CCCC1 ZINC000880574972 FH On-Demand Anodyne L3MBTL3 88 52 O=C(c1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1)N1CCCC1 ZINC000880574973 FH On-Demand Anodyne HRH3 30 48 O=C(c1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1)N1CCCC1 ZINC000880574973 FH On-Demand Anodyne L3MBTL3 88 52 O[C@@H]1CCCC[C@H]1N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575093 CF On-Demand Anodyne SLC18A3 37 54 O[C@@H]1CCCC[C@H]1N1CCCC[C@H](C2CCOCC2)C1 ZINC000880575094 CF On-Demand Anodyne SLC18A3 37 54 c1cncc(CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575097 CG On-Demand Anodyne CHRNA7 36 42 c1cncc(CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575098 CG On-Demand Anodyne CHRNA7 36 42 O[C@@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575099 DG On-Demand Anodyne OPRK1 18 42 O[C@@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575099 DG On-Demand Anodyne SLC6A3 15 41 O[C@@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575099 DG On-Demand Anodyne SLC18A3 15 42 O[C@@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575100 DG On-Demand Anodyne OPRK1 18 42 O[C@@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575100 DG On-Demand Anodyne SLC6A3 15 41 O[C@@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575100 DG On-Demand Anodyne SLC18A3 15 42 O[C@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575101 DG On-Demand Anodyne OPRK1 18 42 O[C@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575101 DG On-Demand Anodyne SLC6A3 15 41 O[C@H](CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575101 DG On-Demand Anodyne SLC18A3 15 42 O[C@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575102 DG On-Demand Anodyne OPRK1 18 42 O[C@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575102 DG On-Demand Anodyne SLC6A3 15 41 O[C@H](CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575102 DG On-Demand Anodyne SLC18A3 15 42 COc1cccc(C2=NO[C@H](C(=O)N3CCN(c4nnc(C)n4C)CC3)C2)c1 ZINC000880575114 GC On-Demand Anodyne LUCI_PHOPY 16 41 COc1cccc(C2=NO[C@@H](C(=O)N3CCN(c4nnc(C)n4C)CC3)C2)c1 ZINC000880575115 GC On-Demand Anodyne LUCI_PHOPY 16 41 c1nc(CN2CCCC[C@H](C3CCOCC3)C2)cs1 ZINC000880575226 CG On-Demand Anodyne SCN5A 43 35 c1nc(CN2CCCC[C@@H](C3CCOCC3)C2)cs1 ZINC000880575227 CG On-Demand Anodyne SCN5A 43 35 CC(=O)c1cccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575236 GG On-Demand Anodyne ACOX1 55 34 CC(=O)c1cccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575236 GG On-Demand Anodyne ABCB1 62 55 CC(=O)c1cccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575237 GG On-Demand Anodyne ACOX1 55 34 CC(=O)c1cccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575237 GG On-Demand Anodyne ABCB1 62 55 CC(=O)c1cccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575238 GG On-Demand Anodyne ACOX1 55 34 CC(=O)c1cccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575238 GG On-Demand Anodyne ABCB1 62 55 CC(=O)c1cccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575239 GG On-Demand Anodyne ACOX1 55 34 CC(=O)c1cccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575239 GG On-Demand Anodyne ABCB1 62 55 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NNC(=O)c1ccccc1 ZINC000880575307 FD On-Demand Reactive SLC6A1 54 35 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NNC(=O)c1ccccc1 ZINC000880575308 FD On-Demand Reactive SLC6A1 54 35 Cc1nnc(N2CCN(C(=O)c3cc(O)c4ccccc4c3)CC2)n1C ZINC000880575397 FD On-Demand Anodyne SMO 29 41 Cc1nnc(N2CCN(C(=O)CN(C)C(=O)OCc3ccccc3)CC2)n1C ZINC000880575417 GD On-Demand Anodyne Q6PRC7_IXORI 43 36 Cc1nnc(N2CCN(C(=O)CN(C)C(=O)OCc3ccccc3)CC2)n1C ZINC000880575417 GD On-Demand Anodyne SLC12A5 64 36 CS(=O)(=O)c1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575457 GF On-Demand Anodyne CASR 26 49 CS(=O)(=O)c1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575457 GF On-Demand Anodyne EPHX2 18 40 CS(=O)(=O)c1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575458 GF On-Demand Anodyne CASR 26 49 CS(=O)(=O)c1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575458 GF On-Demand Anodyne EPHX2 18 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne ADRB2 15 48 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne ADRB1 41 48 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne ADRB3 20 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne ACOX1 57 37 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne ABCB1 43 41 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575469 GF On-Demand Anodyne EPHX2 19 43 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne ADRB2 15 48 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne ADRB1 41 48 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne ADRB3 20 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne ACOX1 57 37 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne ABCB1 43 41 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575470 GF On-Demand Anodyne EPHX2 19 43 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne ADRB2 15 48 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne ADRB1 41 48 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne ADRB3 20 40 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne ACOX1 57 37 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne ABCB1 43 41 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575471 GF On-Demand Anodyne EPHX2 19 43 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne ADRB2 15 48 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne ADRB1 41 48 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne ADRB3 20 40 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne ACOX1 57 37 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne ABCB1 43 41 CC(=O)Nc1ccc(OC[C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575472 GF On-Demand Anodyne EPHX2 19 43 Cc1nnc(N2CCN(C(=O)[C@@H]3CSCN3C(=O)OC(C)(C)C)CC2)n1C ZINC000880575541 GD On-Demand Anodyne PREP 16 40 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1nccs1 ZINC000880575553 DF On-Demand Anodyne MAP1 87 53 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1nccs1 ZINC000880575554 DF On-Demand Anodyne MAP1 87 53 C[C@@H](C(=O)Nc1nccs1)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575572 EF On-Demand Anodyne MAP1 74 39 C[C@@H](C(=O)Nc1nccs1)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575572 EF On-Demand Anodyne GCK 20 42 C[C@H](C(=O)Nc1nccs1)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880575573 EF On-Demand Anodyne MAP1 74 39 C[C@H](C(=O)Nc1nccs1)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880575573 EF On-Demand Anodyne GCK 20 42 C[C@H](C(=O)Nc1nccs1)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575574 EF On-Demand Anodyne MAP1 74 39 C[C@H](C(=O)Nc1nccs1)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575574 EF On-Demand Anodyne GCK 20 42 C[C@@H](C(=O)Nc1nccs1)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880575575 EF On-Demand Anodyne MAP1 74 39 C[C@@H](C(=O)Nc1nccs1)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880575575 EF On-Demand Anodyne GCK 20 42 COc1cccc(C(C)(C)C(=O)N2CCN(c3nnc(C)n3C)CC2)c1 ZINC000880575595 FD On-Demand Anodyne DRD4 43 34 Oc1nc(CN2CCCC[C@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575662 GI On-Demand Anodyne PIM1 20 53 Oc1nc(CN2CCCC[C@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575662 GI On-Demand Anodyne PIM2 15 53 Oc1nc(CN2CCCC[C@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575662 GI On-Demand Anodyne CDC7 21 53 Oc1nc(CN2CCCC[C@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575662 GI On-Demand Anodyne PIM3 25 53 Oc1nc(CN2CCCC[C@@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575663 GI On-Demand Anodyne PIM1 20 53 Oc1nc(CN2CCCC[C@@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575663 GI On-Demand Anodyne PIM2 15 53 Oc1nc(CN2CCCC[C@@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575663 GI On-Demand Anodyne CDC7 21 53 Oc1nc(CN2CCCC[C@@H](C3CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880575663 GI On-Demand Anodyne PIM3 25 53 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575708 GE On-Demand Anodyne CASR 52 40 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575708 GE On-Demand Anodyne CCR5 22 42 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575708 GE On-Demand Anodyne PGA5 42 31 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575708 GE On-Demand Anodyne BIRC2 51 39 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575709 GE On-Demand Anodyne CASR 52 40 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575709 GE On-Demand Anodyne CCR5 22 42 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575709 GE On-Demand Anodyne PGA5 42 31 CNC(=O)[C@@H](NC(=O)CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880575709 GE On-Demand Anodyne BIRC2 51 39 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1ccc(F)cc1 ZINC000880575725 EF On-Demand Anodyne CCR3 48 35 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1ccc(F)cc1 ZINC000880575725 EF On-Demand Anodyne WNT3A 50 42 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1ccc(F)cc1 ZINC000880575726 EF On-Demand Anodyne CCR3 48 35 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1ccc(F)cc1 ZINC000880575726 EF On-Demand Anodyne WNT3A 50 42 CS(=O)(=O)c1cccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575785 GF On-Demand Anodyne ESR1 57 38 CS(=O)(=O)c1cccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575785 GF On-Demand Anodyne ESR2 40 38 CS(=O)(=O)c1cccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575785 GF On-Demand Anodyne LTA4H 33 41 CS(=O)(=O)c1cccc(OCCN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575786 GF On-Demand Anodyne ESR1 57 38 CS(=O)(=O)c1cccc(OCCN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575786 GF On-Demand Anodyne ESR2 40 38 CS(=O)(=O)c1cccc(OCCN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575786 GF On-Demand Anodyne LTA4H 33 41 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880575803 GG On-Demand Anodyne EPHX2 23 45 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880575804 GG On-Demand Anodyne EPHX2 23 45 NC(=O)c1ccc(NC(=O)CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880575805 FF On-Demand Anodyne TERT 15 40 NC(=O)c1ccc(NC(=O)CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880575806 FF On-Demand Anodyne TERT 15 40 Cc1ccc(F)c2[nH]c(C(=O)N3CCN(c4nnc(C)n4C)CC3)cc12 ZINC000880575892 FE On-Demand Anodyne HRH4 37 62 COc1ccccc1NC(=O)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880575902 EG On-Demand Anodyne DRD4 23 43 COc1ccccc1NC(=O)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880575903 EG On-Demand Anodyne DRD4 23 43 N#Cc1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575908 EG On-Demand Mild CASR 20 48 N#Cc1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575908 EG On-Demand Mild CCR3 22 44 N#Cc1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880575908 EG On-Demand Mild MCHR1 46 45 N#Cc1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575909 EG On-Demand Mild CASR 20 48 N#Cc1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575909 EG On-Demand Mild CCR3 22 44 N#Cc1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880575909 EG On-Demand Mild MCHR1 46 45 Cc1nnc(N2CCN(C(=O)c3cccc([C@H]4CCCN(C)C4)c3)CC2)n1C ZINC000880576035 GD On-Demand Anodyne L3MBTL3 41 38 Cc1nnc(N2CCN(C(=O)c3cccc([C@@H]4CCCN(C)C4)c3)CC2)n1C ZINC000880576036 GD On-Demand Anodyne L3MBTL3 41 38 Cc1nnc(N2CCN(C(=O)[C@H]3CCC[C@@H]3c3ccccc3)CC2)n1C ZINC000880576050 FE On-Demand Anodyne NPBWR1 60 32 Cc1nnc(N2CCN(C(=O)[C@@H]3CCC[C@@H]3c3ccccc3)CC2)n1C ZINC000880576051 FE On-Demand Anodyne NPBWR1 60 32 Cc1nnc(N2CCN(C(=O)[C@H]3CCC[C@H]3c3ccccc3)CC2)n1C ZINC000880576052 FE On-Demand Anodyne NPBWR1 60 32 Cc1nnc(N2CCN(C(=O)[C@@H]3CCC[C@H]3c3ccccc3)CC2)n1C ZINC000880576053 FE On-Demand Anodyne NPBWR1 60 32 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1cccnc1 ZINC000880576054 EE On-Demand Anodyne CHRNA7 47 35 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCc1cccnc1 ZINC000880576054 EE On-Demand Anodyne NAMPT 92 45 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1cccnc1 ZINC000880576055 EE On-Demand Anodyne CHRNA7 47 35 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCc1cccnc1 ZINC000880576055 EE On-Demand Anodyne NAMPT 92 45 Cc1nnc(N2CCN(C(=O)CCc3cccc4ccccc34)CC2)n1C ZINC000880576065 FF On-Demand Anodyne SSTR1 26 48 Cc1nnc(N2CCN(C(=O)[C@@H](Cc3cccnc3)C3CCCC3)CC2)n1C ZINC000880576066 GE On-Demand Anodyne C3AR1 44 44 Cc1nnc(N2CCN(C(=O)[C@H](Cc3cccnc3)C3CCCC3)CC2)n1C ZINC000880576067 GE On-Demand Anodyne C3AR1 44 44 Cc1nnc(N2CCN(C(=O)c3cccc(Oc4ccccn4)c3)CC2)n1C ZINC000880576072 GE On-Demand Anodyne CFTR 17 42 C#CC1(F)CN(C(=O)Nc2ccc(C(=O)OC)nc2)C1 ZINC000880576127 CD On-Demand Mild EPHX2 29 41 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1cccnc1Cl ZINC000880576168 FG On-Demand Anodyne G2YM83_BOTF4 63 32 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1cccnc1Cl ZINC000880576169 FG On-Demand Anodyne G2YM83_BOTF4 63 32 Cc1nnc(N2CCN(C(=O)c3cccc(OC(C)(C)C)c3)CC2)n1C ZINC000880576197 FE On-Demand Anodyne DRD4 41 32 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne ESR1 87 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne ESR2 58 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne LTA4H 52 43 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne HRH3 53 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne PSMB2 41 39 CS(=O)(=O)c1ccc(OCCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576230 GF On-Demand Anodyne PSMB1 45 39 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne ESR1 87 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne ESR2 58 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne LTA4H 52 43 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne HRH3 53 45 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne PSMB2 41 39 CS(=O)(=O)c1ccc(OCCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576232 GF On-Demand Anodyne PSMB1 45 39 N#CCOc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576259 EH On-Demand Mild HRH3 24 45 N#CCOc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576263 EH On-Demand Mild HRH3 24 45 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NNC(=O)c1ccc(F)cc1 ZINC000880576300 GE On-Demand Reactive WNT3A 58 38 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NNC(=O)c1ccc(F)cc1 ZINC000880576302 GE On-Demand Reactive WNT3A 58 38 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA2 29 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA1 30 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA7 15 41 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne HRH3 17 46 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA4 17 40 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA12 20 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne CA9 24 41 NS(=O)(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576432 FE On-Demand Anodyne L3MBTL3 30 40 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA2 29 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA1 30 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA7 15 41 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne HRH3 17 46 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA4 17 40 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA12 20 42 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne CA9 24 41 NS(=O)(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576434 FE On-Demand Anodyne L3MBTL3 30 40 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NCC(=O)c1ccccc1 ZINC000880576488 FF On-Demand Anodyne SLC6A1 53 34 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NCC(=O)c1ccccc1 ZINC000880576489 FF On-Demand Anodyne SLC6A1 53 34 CC(=O)Oc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880576532 EH On-Demand Anodyne HRH3 26 42 CC(=O)Oc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880576535 EH On-Demand Anodyne HRH3 26 42 c1cc(CCCN2CCCC[C@H](C3CCOCC3)C2)ccn1 ZINC000880576579 DH On-Demand Anodyne SIGMAR1 15 42 c1cc(CCCN2CCCC[C@H](C3CCOCC3)C2)ccn1 ZINC000880576579 DH On-Demand Anodyne L3MBTL3 20 41 c1cc(CCCN2CCCC[C@@H](C3CCOCC3)C2)ccn1 ZINC000880576581 DH On-Demand Anodyne SIGMAR1 15 42 c1cc(CCCN2CCCC[C@@H](C3CCOCC3)C2)ccn1 ZINC000880576581 DH On-Demand Anodyne L3MBTL3 20 41 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1cccnc1 ZINC000880576584 EF On-Demand Anodyne CHRNA7 43 47 O=C(CCN1CCCC[C@H](C2CCOCC2)C1)Nc1cccnc1 ZINC000880576584 EF On-Demand Anodyne NAMPT 33 41 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1cccnc1 ZINC000880576586 EF On-Demand Anodyne CHRNA7 43 47 O=C(CCN1CCCC[C@@H](C2CCOCC2)C1)Nc1cccnc1 ZINC000880576586 EF On-Demand Anodyne NAMPT 33 41 Cc1nnc(N2CCN(C(=O)c3csc(Br)n3)CC2)n1C ZINC000880576651 FD On-Demand Anodyne TRPC6 41 39 O=C(NCCC1(CO)CCC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880576719 EG On-Demand Anodyne PDE4D 15 42 Cc1nnc(N2CCN(C(=O)c3cc4sccc4nc3Cl)CC2)n1C ZINC000880576748 GE On-Demand Anodyne HRH4 16 40 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1ccc(C(=O)OC)nc1)C2 ZINC000880576780 FE On-Demand Anodyne P2RY14 42 31 Cc1nnc(N2CCN(C(=O)Cc3cc4cc(Cl)ccc4[nH]3)CC2)n1C ZINC000880576782 FE On-Demand Anodyne HRH4 16 44 C[C@H](C(=O)Nc1cccnc1Cl)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880576792 FH On-Demand Anodyne G2YM83_BOTF4 59 34 C[C@H](C(=O)Nc1cccnc1Cl)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880576795 FH On-Demand Anodyne G2YM83_BOTF4 59 34 O=S(=O)(CCN1CCCC[C@H](C2CCOCC2)C1)Cc1ccccc1 ZINC000880576878 FG On-Demand Anodyne SLC6A1 47 34 O=S(=O)(CCN1CCCC[C@@H](C2CCOCC2)C1)Cc1ccccc1 ZINC000880576879 FG On-Demand Anodyne SLC6A1 47 34 O[C@@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576906 DH On-Demand Anodyne SLC6A1 59 41 O[C@@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576906 DH On-Demand Anodyne SLC6A3 15 47 O[C@@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576906 DH On-Demand Anodyne CCR5 24 40 O[C@@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576908 DH On-Demand Anodyne SLC6A1 59 41 O[C@@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576908 DH On-Demand Anodyne SLC6A3 15 47 O[C@@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576908 DH On-Demand Anodyne CCR5 24 40 O[C@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576910 DH On-Demand Anodyne SLC6A1 59 41 O[C@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576910 DH On-Demand Anodyne SLC6A3 15 47 O[C@H](CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576910 DH On-Demand Anodyne CCR5 24 40 O[C@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576912 DH On-Demand Anodyne SLC6A1 59 41 O[C@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576912 DH On-Demand Anodyne SLC6A3 15 47 O[C@H](CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880576912 DH On-Demand Anodyne CCR5 24 40 C[C@@H](c1ccc(S(C)(=O)=O)cc1)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880577007 FH On-Demand Anodyne CHRM2 16 43 C[C@@H](c1ccc(S(C)(=O)=O)cc1)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880577008 FH On-Demand Anodyne CHRM2 16 43 CC(=O)[C@](C#N)(CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577073 FH On-Demand Mild SLC6A1 70 35 CC(=O)[C@@](C#N)(CCN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577074 FH On-Demand Mild SLC6A1 70 35 CC(=O)[C@@](C#N)(CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577075 FH On-Demand Mild SLC6A1 70 35 CC(=O)[C@](C#N)(CCN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577076 FH On-Demand Mild SLC6A1 70 35 c1cncc(CCN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880577255 CG On-Demand Anodyne CHRNA7 44 35 c1cncc(CCN2CCCC[C@@H](C3CCOCC3)C2)c1 ZINC000880577255 CG On-Demand Anodyne ACHP_LYMST 24 40 c1cncc(CCN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880577258 CG On-Demand Anodyne CHRNA7 44 35 c1cncc(CCN2CCCC[C@H](C3CCOCC3)C2)c1 ZINC000880577258 CG On-Demand Anodyne ACHP_LYMST 24 40 O=[N+]([O-])c1ccc([C@@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880577262 EG On-Demand Bother KCNJ1 19 41 O=[N+]([O-])c1ccc([C@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880577265 EG On-Demand Bother KCNJ1 19 41 O=[N+]([O-])c1ccc([C@@H](O)CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880577268 EG On-Demand Bother KCNJ1 19 41 O=[N+]([O-])c1ccc([C@H](O)CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880577272 EG On-Demand Bother KCNJ1 19 41 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N[C@H](CO)CCF)ccn2)CC1 ZINC000880577290 GD On-Demand Anodyne GPR119 35 42 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N[C@@H](CO)CCF)ccn2)CC1 ZINC000880577293 GD On-Demand Anodyne GPR119 35 42 NC(=O)[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577313 ED On-Demand Anodyne CHRM2 21 41 NC(=O)[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577313 ED On-Demand Anodyne CHRM3 33 41 NC(=O)[C@@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577313 ED On-Demand Anodyne CYP2J2 45 31 NC(=O)[C@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577314 ED On-Demand Anodyne CHRM2 21 41 NC(=O)[C@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577314 ED On-Demand Anodyne CHRM3 33 41 NC(=O)[C@](O)(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577314 ED On-Demand Anodyne CYP2J2 45 31 NC(=O)[C@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577316 ED On-Demand Anodyne CHRM2 21 41 NC(=O)[C@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577316 ED On-Demand Anodyne CHRM3 33 41 NC(=O)[C@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577316 ED On-Demand Anodyne CYP2J2 45 31 NC(=O)[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577317 ED On-Demand Anodyne CHRM2 21 41 NC(=O)[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577317 ED On-Demand Anodyne CHRM3 33 41 NC(=O)[C@@](O)(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1 ZINC000880577317 ED On-Demand Anodyne CYP2J2 45 31 O=C1c2ccccc2C(=O)N1OCCCN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880577370 GG On-Demand Anodyne SLC6A1 45 35 O=C1c2ccccc2C(=O)N1OCCCN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880577370 GG On-Demand Anodyne HRH3 25 40 O=C1c2ccccc2C(=O)N1OCCCN1CCCC[C@H](C2CCOCC2)C1 ZINC000880577371 GG On-Demand Anodyne SLC6A1 45 35 O=C1c2ccccc2C(=O)N1OCCCN1CCCC[C@H](C2CCOCC2)C1 ZINC000880577371 GG On-Demand Anodyne HRH3 25 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@]3(C2)CC3(F)F)N1Cc1ccccc1 ZINC000880577375 GE On-Demand Anodyne PREP 41 38 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@]3(C2)CC3(F)F)N1Cc1ccccc1 ZINC000880577376 GE On-Demand Anodyne PREP 41 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]2C[C@H]1C2(C)C ZINC000880577419 FF On-Demand Anodyne CELA1 29 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]2C[C@H]1C2(C)C ZINC000880577419 FF On-Demand Anodyne CELA2A 41 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]2C[C@H]1C2(C)C ZINC000880577420 FF On-Demand Anodyne CELA1 29 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]2C[C@H]1C2(C)C ZINC000880577420 FF On-Demand Anodyne CELA2A 41 34 O=C(CC[C@@H]1CCc2ccccc21)NCCC1(CO)CCC1 ZINC000880577443 DG On-Demand Anodyne NQO2 18 41 O=C(CC[C@H]1CCc2ccccc21)NCCC1(CO)CCC1 ZINC000880577444 DG On-Demand Anodyne NQO2 18 41 O=C(N[C@@H](CO)CCF)c1cnc2cc[nH]c2c1 ZINC000880577491 CD On-Demand Anodyne AKT1 49 30 O=C(N[C@H](CO)CCF)c1cnc2cc[nH]c2c1 ZINC000880577492 CD On-Demand Anodyne AKT1 49 30 OCc1ccc(CN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880577541 DG On-Demand Anodyne HRH3 20 40 OCc1ccc(CN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880577542 DG On-Demand Anodyne HRH3 20 40 CS(=O)(=O)C1CCC(C(=O)NCCc2ccc3c(c2)OC(F)(F)O3)CC1 ZINC000880577622 GE On-Demand Anodyne MTNR1A 19 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(=O)n3ccccc3n1)C2 ZINC000880577645 FE On-Demand Anodyne MTNR1A 35 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(=O)n3ccccc3n1)C2 ZINC000880577645 FE On-Demand Anodyne MTNR1B 34 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2ncsc2C2CC2)CC1 ZINC000880577699 GH On-Demand Anodyne SIRT3 48 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2ncsc2C2CC2)CC1 ZINC000880577699 GH On-Demand Anodyne SIRT2 49 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2ncsc2C2CC2)CC1 ZINC000880577699 GH On-Demand Anodyne SIRT1 48 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@H]2CCc3nncn3CC2)CC1 ZINC000880577709 GE On-Demand Anodyne SIRT3 26 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@H]2CCc3nncn3CC2)CC1 ZINC000880577709 GE On-Demand Anodyne SIRT2 25 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@H]2CCc3nncn3CC2)CC1 ZINC000880577709 GE On-Demand Anodyne SIRT1 24 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@@H]2CCc3nncn3CC2)CC1 ZINC000880577712 GE On-Demand Anodyne SIRT3 26 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@@H]2CCc3nncn3CC2)CC1 ZINC000880577712 GE On-Demand Anodyne SIRT2 25 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)[C@@H]2CCc3nncn3CC2)CC1 ZINC000880577712 GE On-Demand Anodyne SIRT1 24 42 O=C(NCCC[C@H]1CC1(Cl)Cl)c1coc(-c2ccccn2)n1 ZINC000880577747 EG On-Demand Anodyne TBXA2R 28 40 O=C(NCCC[C@@H]1CC1(Cl)Cl)c1coc(-c2ccccn2)n1 ZINC000880577748 EG On-Demand Anodyne TBXA2R 28 40 COC(=O)c1cccc(NC(=O)CN2CCCC[C@H](C3CCOCC3)C2)n1 ZINC000880577790 GE On-Demand Anodyne CASR 46 37 COC(=O)c1cccc(NC(=O)CN2CCCC[C@@H](C3CCOCC3)C2)n1 ZINC000880577791 GE On-Demand Anodyne CASR 46 37 O=C(CN1CCCC[C@H](C2CCOCC2)C1)N1CCN(c2cnccn2)CC1 ZINC000880577792 GD On-Demand Anodyne MAPK1 19 40 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)N1CCN(c2cnccn2)CC1 ZINC000880577793 GD On-Demand Anodyne MAPK1 19 40 O=C(N[C@@H](CO)CCF)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880577809 CD On-Demand Anodyne MPO 58 36 O=C(N[C@H](CO)CCF)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880577810 CD On-Demand Anodyne MPO 58 36 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne ACE 24 46 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne CTRA_BOVIN 59 31 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne KLK3 62 31 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne CTSG 40 31 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne CTSK 16 43 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne PREP 25 42 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne CELA2A 48 31 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne LGMN 74 43 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne CAPN1 35 41 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne KLK5 40 40 O=C(N[C@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577824 FD On-Demand Anodyne Q9NAW4_PLAFA 46 55 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne ACE 24 46 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne CTRA_BOVIN 59 31 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne KLK3 62 31 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne CTSG 40 31 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne CTSK 16 43 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne PREP 25 42 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne CELA2A 48 31 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne LGMN 74 43 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne CAPN1 35 41 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne KLK5 40 40 O=C(N[C@@H](CO)CCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880577825 FD On-Demand Anodyne Q9NAW4_PLAFA 46 55 Cc1ncc(CC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)o1 ZINC000880577885 FF On-Demand Anodyne SIRT3 34 44 Cc1ncc(CC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)o1 ZINC000880577885 FF On-Demand Anodyne SIRT2 30 44 Cc1ncc(CC(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)o1 ZINC000880577885 FF On-Demand Anodyne SIRT1 30 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne GRIN2B 47 34 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne ACACB 19 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne SIRT3 54 37 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne SIRT2 57 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne SIRT1 54 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880577915 FG On-Demand Anodyne SFRP1 44 36 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2c[nH]cc2C2CC2)CC1 ZINC000880577923 FH On-Demand Anodyne SIRT3 26 43 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2c[nH]cc2C2CC2)CC1 ZINC000880577923 FH On-Demand Anodyne SIRT2 25 43 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2c[nH]cc2C2CC2)CC1 ZINC000880577923 FH On-Demand Anodyne SIRT1 25 43 O=C(NCCC1(CO)CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880577970 DE On-Demand Anodyne MPO 40 38 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@]2(C1)CC2(F)F ZINC000880577980 DI On-Demand Anodyne EBP 19 51 Cc1nc(C(C)C)ncc1C(=O)NCc1cc(=O)n2ccccc2n1 ZINC000880577981 ED On-Demand Anodyne POLR1A 66 36 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@]2(C1)CC2(F)F ZINC000880577982 DI On-Demand Anodyne EBP 19 51 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@@]2(C1)CC2(F)F ZINC000880577985 DI On-Demand Anodyne EBP 19 51 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@@]2(C1)CC2(F)F ZINC000880577986 DI On-Demand Anodyne EBP 19 51 O=C(NCC[C@@]1(O)CCCOC1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880578040 ED On-Demand Anodyne PLD2 44 38 O=C(NCC[C@]1(O)CCCOC1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880578052 ED On-Demand Anodyne PLD2 44 38 O[C@@H]1CCC[C@H]1N1CCCC[C@H](C2CCOCC2)C1 ZINC000880578179 CE On-Demand Anodyne SLC18A3 36 53 O[C@@H]1CCC[C@H]1N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880578180 CE On-Demand Anodyne SLC18A3 36 53 CC[C@@H](NC(=O)Nc1ccc(C(=O)OC)nc1)c1cccc(OC)c1OC ZINC000880578227 FG On-Demand Anodyne PDGFRA 40 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H](c2ccccc2)O1 ZINC000880578247 GF On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H](c2ccccc2)O1 ZINC000880578247 GF On-Demand Anodyne PAPA1_CARPA 43 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H](c2ccccc2)O1 ZINC000880578247 GF On-Demand Anodyne CACNA1B 18 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H](c2ccccc2)O1 ZINC000880578247 GF On-Demand Anodyne REN 60 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H](c2ccccc2)O1 ZINC000880578247 GF On-Demand Anodyne FPR1 47 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H](c2ccccc2)O1 ZINC000880578251 GF On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H](c2ccccc2)O1 ZINC000880578251 GF On-Demand Anodyne PAPA1_CARPA 43 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H](c2ccccc2)O1 ZINC000880578251 GF On-Demand Anodyne CACNA1B 18 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H](c2ccccc2)O1 ZINC000880578251 GF On-Demand Anodyne REN 60 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H](c2ccccc2)O1 ZINC000880578251 GF On-Demand Anodyne FPR1 47 39 Cc1cnc(Cl)c(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880578337 GH On-Demand Anodyne CACNA1I 53 36 Cc1cnc(Cl)c(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880578337 GH On-Demand Anodyne SIRT3 46 45 Cc1cnc(Cl)c(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880578337 GH On-Demand Anodyne SIRT2 43 45 Cc1cnc(Cl)c(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1 ZINC000880578337 GH On-Demand Anodyne SIRT1 45 45 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](CO)CCF)C2 ZINC000880578339 CD On-Demand Anodyne NQO2 28 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](CO)CCF)C2 ZINC000880578341 CD On-Demand Anodyne NQO2 28 41 COc1ccccc1-c1ccc(C(=O)NCCC[C@@H]2CC2(Cl)Cl)c(O)n1 ZINC000880578353 GI On-Demand Anodyne KCNA3 40 34 COc1ccccc1-c1ccc(C(=O)NCCC[C@H]2CC2(Cl)Cl)c(O)n1 ZINC000880578354 GI On-Demand Anodyne KCNA3 40 34 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880578370 FG On-Demand Anodyne SIRT3 29 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880578370 FG On-Demand Anodyne SIRT2 29 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880578370 FG On-Demand Anodyne SIRT1 29 42 Cc1nc(C(C)C)ncc1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880578414 GH On-Demand Anodyne SIRT3 41 43 Cc1nc(C(C)C)ncc1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880578414 GH On-Demand Anodyne SIRT2 42 43 Cc1nc(C(C)C)ncc1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880578414 GH On-Demand Anodyne SIRT1 43 43 O=C(NCC[C@@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578467 GD On-Demand Anodyne CTRA_BOVIN 48 30 O=C(NCC[C@@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578467 GD On-Demand Anodyne LGMN 62 38 O=C(NCC[C@@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578467 GD On-Demand Anodyne Q9NAW4_PLAFA 35 40 O=C(NCC[C@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578469 GD On-Demand Anodyne CTRA_BOVIN 48 30 O=C(NCC[C@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578469 GD On-Demand Anodyne LGMN 62 38 O=C(NCC[C@]1(O)CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578469 GD On-Demand Anodyne Q9NAW4_PLAFA 35 40 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cncc3[nH]ccc23)CC1 ZINC000880578522 FG On-Demand Anodyne ACACB 15 43 O=C(N[C@@H](CO)CCF)c1cc2ccccc2cc1F ZINC000880578571 CE On-Demand Anodyne PIN1 43 40 O=C(N[C@H](CO)CCF)c1cc2ccccc2cc1F ZINC000880578572 CE On-Demand Anodyne PIN1 43 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H](CO)CCF ZINC000880578585 DD On-Demand Anodyne KCNQ2 57 36 O=C(Cc1ccccc1N1CCCC1=O)N[C@H](CO)CCF ZINC000880578586 DD On-Demand Anodyne KCNQ2 57 36 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NOCc1ccccc1 ZINC000880578650 EF On-Demand Anodyne PREP 31 40 O=C(CN1CCCC[C@H](C2CCOCC2)C1)NOCc1ccccc1 ZINC000880578650 EF On-Demand Anodyne SLC12A5 59 36 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NOCc1ccccc1 ZINC000880578651 EF On-Demand Anodyne PREP 31 40 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)NOCc1ccccc1 ZINC000880578651 EF On-Demand Anodyne SLC12A5 59 36 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(C3CC3)o2)CC1 ZINC000880578671 FG On-Demand Anodyne SIRT3 45 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(C3CC3)o2)CC1 ZINC000880578671 FG On-Demand Anodyne SIRT2 42 45 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(C3CC3)o2)CC1 ZINC000880578671 FG On-Demand Anodyne SIRT1 44 45 Oc1nc(CN2CCCC[C@H](C3CCOCC3)C2)nc2c1COCC2 ZINC000880578701 EE On-Demand Anodyne WNT3A 52 32 Oc1nc(CN2CCCC[C@@H](C3CCOCC3)C2)nc2c1COCC2 ZINC000880578702 EE On-Demand Anodyne WNT3A 52 32 O=C(CN1CCCC[C@H](C2CCOCC2)C1)c1ccccc1F ZINC000880578723 DH On-Demand Anodyne SLC6A1 91 42 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)c1ccccc1F ZINC000880578725 DH On-Demand Anodyne SLC6A1 91 42 O[C@@H](Cc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880578751 DG On-Demand Anodyne TACR2 39 40 O[C@@H](Cc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880578751 DG On-Demand Anodyne ABCB1 29 41 O[C@@H](Cc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880578753 DG On-Demand Anodyne TACR2 39 40 O[C@@H](Cc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880578753 DG On-Demand Anodyne ABCB1 29 41 O[C@H](Cc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880578755 DG On-Demand Anodyne TACR2 39 40 O[C@H](Cc1ccccc1)CN1CCCC[C@H](C2CCOCC2)C1 ZINC000880578755 DG On-Demand Anodyne ABCB1 29 41 O[C@H](Cc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880578757 DG On-Demand Anodyne TACR2 39 40 O[C@H](Cc1ccccc1)CN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880578757 DG On-Demand Anodyne ABCB1 29 41 C[C@@H](CCO)N(C)C(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880578802 GD On-Demand Anodyne GPR119 35 43 C[C@H](CCO)N(C)C(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880578804 GD On-Demand Anodyne GPR119 35 43 COc1ccccc1-c1ccc(C(=O)NCCC2(CO)CCC2)c(O)n1 ZINC000880578825 FF On-Demand Anodyne KCNA3 45 38 NC(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880578835 EF On-Demand Anodyne HRH3 17 43 NC(=O)c1ccc(CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880578835 EF On-Demand Anodyne L3MBTL3 34 40 NC(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880578836 EF On-Demand Anodyne HRH3 17 43 NC(=O)c1ccc(CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880578836 EF On-Demand Anodyne L3MBTL3 34 40 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne CELA1 20 42 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne PREP 26 42 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne LGMN 47 37 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne SLC12A5 65 36 O=C(NCCC1(CO)CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880578847 GE On-Demand Anodyne Q9NAW4_PLAFA 38 45 O=C(CN1CCCC[C@H](C2CCOCC2)C1)Nc1nnc(-c2ccco2)o1 ZINC000880578923 FF On-Demand Anodyne CHRNA7 16 41 O=C(CN1CCCC[C@@H](C2CCOCC2)C1)Nc1nnc(-c2ccco2)o1 ZINC000880578924 FF On-Demand Anodyne CHRNA7 16 41 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(C)(C)C ZINC000880578994 DF On-Demand Anodyne KCNQ2 63 37 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@@]2(C1)CC2(F)F ZINC000880579087 DF On-Demand Anodyne HPGD 44 41 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@]2(C1)CC2(F)F ZINC000880579089 DF On-Demand Anodyne HPGD 44 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880579259 GH On-Demand Anodyne SIRT3 61 49 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880579259 GH On-Demand Anodyne SIRT2 61 49 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880579259 GH On-Demand Anodyne SIRT1 59 49 CCn1ncc(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1C1CC1 ZINC000880579271 GH On-Demand Anodyne SIRT3 18 40 CCn1ncc(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1C1CC1 ZINC000880579271 GH On-Demand Anodyne SIRT2 21 40 CCn1ncc(C(=O)N2CCC(CCNC(=O)OC(C)(C)C)CC2)c1C1CC1 ZINC000880579271 GH On-Demand Anodyne SIRT1 19 40 O=[N+]([O-])c1ccc(S(=O)(=O)CCN2CCCC[C@H](C3CCOCC3)C2)cc1 ZINC000880579445 GF On-Demand Bother KCNJ1 21 40 O=[N+]([O-])c1ccc(S(=O)(=O)CCN2CCCC[C@@H](C3CCOCC3)C2)cc1 ZINC000880579446 GF On-Demand Bother KCNJ1 21 40 C=CC(C)(C)CC(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579538 EH On-Demand Mild SIRT3 18 40 C=CC(C)(C)CC(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579538 EH On-Demand Mild SIRT2 21 40 C=CC(C)(C)CC(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579538 EH On-Demand Mild SIRT1 19 40 Cc1nnc(N2CCN(C(=O)c3cc4c(C5CC5)cccc4[nH]3)CC2)n1C ZINC000880579626 FE On-Demand Anodyne GRIN2B 24 41 Cc1nnc(N2CCN(C(=O)c3cc4c(C5CC5)cccc4[nH]3)CC2)n1C ZINC000880579626 FE On-Demand Anodyne HRH4 29 50 O=c1ccc([N+](=O)[O-])cn1CCN1CCCC[C@H](C2CCOCC2)C1 ZINC000880579633 EE On-Demand Bother KCNJ1 18 40 O=c1ccc([N+](=O)[O-])cn1CCN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880579634 EE On-Demand Bother KCNJ1 18 40 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579687 FH On-Demand Anodyne SLC6A1 49 34 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579687 FH On-Demand Anodyne TACR2 22 40 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579687 FH On-Demand Anodyne L3MBTL3 72 37 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579690 FH On-Demand Anodyne SLC6A1 49 34 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579690 FH On-Demand Anodyne TACR2 22 40 O=C(c1ccccc1)N1CC[C@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579690 FH On-Demand Anodyne L3MBTL3 72 37 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579691 FH On-Demand Anodyne SLC6A1 49 34 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579691 FH On-Demand Anodyne TACR2 22 40 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@@H](C3CCOCC3)C2)C1 ZINC000880579691 FH On-Demand Anodyne L3MBTL3 72 37 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579692 FH On-Demand Anodyne SLC6A1 49 34 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579692 FH On-Demand Anodyne TACR2 22 40 O=C(c1ccccc1)N1CC[C@@H](CN2CCCC[C@H](C3CCOCC3)C2)C1 ZINC000880579692 FH On-Demand Anodyne L3MBTL3 72 37 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H](CO)CCF)N1Cc1ccccc1 ZINC000880579727 EC On-Demand Anodyne TRY1_BOVIN 42 31 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H](CO)CCF)N1Cc1ccccc1 ZINC000880579727 EC On-Demand Anodyne XIAP 47 35 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H](CO)CCF)N1Cc1ccccc1 ZINC000880579730 EC On-Demand Anodyne TRY1_BOVIN 42 31 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H](CO)CCF)N1Cc1ccccc1 ZINC000880579730 EC On-Demand Anodyne XIAP 47 35 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579734 GG On-Demand Anodyne SIRT3 18 40 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579734 GG On-Demand Anodyne SIRT2 21 40 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579734 GG On-Demand Anodyne SIRT1 19 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579735 GG On-Demand Anodyne SIRT3 18 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579735 GG On-Demand Anodyne SIRT2 21 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579735 GG On-Demand Anodyne SIRT1 19 40 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579737 GG On-Demand Anodyne SIRT3 18 40 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579737 GG On-Demand Anodyne SIRT2 21 40 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(CCNC(=O)OC(C)(C)C)CC1 ZINC000880579737 GG On-Demand Anodyne SIRT1 19 40 CC(C)(C)OC(=O)NCCC1CCN(C(=O)COC2CC2)CC1 ZINC000880579763 EE On-Demand Anodyne SIRT3 18 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)COC2CC2)CC1 ZINC000880579763 EE On-Demand Anodyne SIRT2 21 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)COC2CC2)CC1 ZINC000880579763 EE On-Demand Anodyne SIRT1 23 41 C[C@@H](NC(=O)c1cccn2nccc12)C(C)(C)C ZINC000880579795 BE On-Demand Anodyne JAK3 19 53 C[C@@H](NC(=O)c1cccn2nccc12)C(C)(C)C ZINC000880579795 BE On-Demand Anodyne JAK1 16 53 C[C@@H](NC(=O)c1cccn2nccc12)C(C)(C)C ZINC000880579795 BE On-Demand Anodyne TYK2 20 53 O=c1c2ccccc2ncn1CCN1CCCC[C@@H](C2CCOCC2)C1 ZINC000880579809 FF On-Demand Anodyne HNMT 75 34 O=c1c2ccccc2ncn1CCN1CCCC[C@H](C2CCOCC2)C1 ZINC000880579810 FF On-Demand Anodyne HNMT 75 34 C[C@H](CCO)N(C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880579885 CD On-Demand Anodyne MPO 70 37 C[C@@H](CCO)N(C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880579886 CD On-Demand Anodyne MPO 70 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579932 DE On-Demand Anodyne PAPA1_CARPA 39 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579932 DE On-Demand Anodyne CTSK 17 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579932 DE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579932 DE On-Demand Anodyne FPR1 48 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579933 DE On-Demand Anodyne PAPA1_CARPA 39 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579933 DE On-Demand Anodyne CTSK 17 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579933 DE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C(C)(C)C ZINC000880579933 DE On-Demand Anodyne FPR1 48 39 O=[N+]([O-])c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880580013 FE On-Demand Bother HRH3 21 41 O=[N+]([O-])c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880580014 FE On-Demand Bother HRH3 21 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cccn3nccc23)CC1 ZINC000880580044 FG On-Demand Anodyne SIRT3 25 40 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cccn3nccc23)CC1 ZINC000880580044 FG On-Demand Anodyne SIRT2 27 40 CC(C)(C)OC(=O)NCCC1CCN(C(=O)c2cccn3nccc23)CC1 ZINC000880580044 FG On-Demand Anodyne SIRT1 24 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H](C)CCO ZINC000880580114 DD On-Demand Anodyne PAPA1_CARPA 34 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H](C)CCO ZINC000880580114 DD On-Demand Anodyne CTSK 16 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@@H](C)CCO ZINC000880580115 DD On-Demand Anodyne PAPA1_CARPA 34 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@@H](C)CCO ZINC000880580115 DD On-Demand Anodyne CTSK 16 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@@H](C)CCO ZINC000880580116 DD On-Demand Anodyne PAPA1_CARPA 34 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@@H](C)CCO ZINC000880580116 DD On-Demand Anodyne CTSK 16 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H](C)CCO ZINC000880580117 DD On-Demand Anodyne PAPA1_CARPA 34 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H](C)CCO ZINC000880580117 DD On-Demand Anodyne CTSK 16 48 C[C@H](CCO)N(C)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880580122 DD On-Demand Anodyne KCNQ2 62 34 C[C@@H](CCO)N(C)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880580123 DD On-Demand Anodyne KCNQ2 62 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CC2(CCC2)C1 ZINC000880580144 EE On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CC2(CCC2)C1 ZINC000880580146 EE On-Demand Anodyne PAPA1_CARPA 34 42 CN(CCN1C[C@H](O)CC2(CCOCC2)C1)Cc1ccc(F)cc1 ZINC000880580278 EE On-Demand Anodyne TACR3 16 40 CN(CCN1C[C@@H](O)CC2(CCOCC2)C1)Cc1ccc(F)cc1 ZINC000880580279 EE On-Demand Anodyne TACR3 16 40 CC(C)(C)OC(=O)N1CCC(CCCN2C[C@@H](O)CC3(CCOCC3)C2)CC1 ZINC000880580400 GG On-Demand Anodyne GPR119 25 41 CC(C)(C)OC(=O)N1CCC(CCCN2C[C@H](O)CC3(CCOCC3)C2)CC1 ZINC000880580401 GG On-Demand Anodyne GPR119 25 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880580472 FE On-Demand Anodyne PREP 50 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880580472 FE On-Demand Anodyne SLC12A5 56 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880580472 FE On-Demand Anodyne Q9NAW4_PLAFA 27 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880580473 FE On-Demand Anodyne PREP 50 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880580473 FE On-Demand Anodyne SLC12A5 56 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880580473 FE On-Demand Anodyne Q9NAW4_PLAFA 27 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880580474 FE On-Demand Anodyne PREP 50 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880580474 FE On-Demand Anodyne SLC12A5 56 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880580474 FE On-Demand Anodyne Q9NAW4_PLAFA 27 41 CO[C@@H](CN1C[C@@H](O)CC2(CCOCC2)C1)c1ccc(F)cc1 ZINC000880580527 DE On-Demand Anodyne LEF 26 43 CO[C@@H](CN1C[C@H](O)CC2(CCOCC2)C1)c1ccc(F)cc1 ZINC000880580528 DE On-Demand Anodyne LEF 26 43 N#Cc1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880580602 DD On-Demand Mild KCNJ1 17 47 N#Cc1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880580603 DD On-Demand Mild KCNJ1 17 47 O=C(NC1CC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880580613 DF On-Demand Anodyne GABRA1 18 42 O=C(NC1CC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880580613 DF On-Demand Anodyne MPO 41 36 O=C(NC1CC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880580613 DF On-Demand Anodyne GABRA2 16 42 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)c(F)c1 ZINC000880580672 FE On-Demand Anodyne ENV 47 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)c(F)c1 ZINC000880580673 FE On-Demand Anodyne ENV 47 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)c1c[nH]c2ccc(F)cc12 ZINC000880580758 EE On-Demand Anodyne MPO 63 34 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)c1c[nH]c2ccc(F)cc12 ZINC000880580759 EE On-Demand Anodyne MPO 63 34 N#Cc1ccccc1OC[C@H](O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880580901 ED On-Demand Mild ADRB1 59 36 N#Cc1ccccc1OC[C@H](O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880580901 ED On-Demand Mild ABCB1 40 36 N#Cc1ccccc1OC[C@H](O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880580902 ED On-Demand Mild ADRB1 59 36 N#Cc1ccccc1OC[C@H](O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880580902 ED On-Demand Mild ABCB1 40 36 N#Cc1ccccc1OC[C@@H](O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880580903 ED On-Demand Mild ADRB1 59 36 N#Cc1ccccc1OC[C@@H](O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880580903 ED On-Demand Mild ABCB1 40 36 N#Cc1ccccc1OC[C@@H](O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880580904 ED On-Demand Mild ADRB1 59 36 N#Cc1ccccc1OC[C@@H](O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880580904 ED On-Demand Mild ABCB1 40 36 NC(=O)[C@@H]1CC[C@H](C(=O)NC2CC3(CCC3)C2)N1Cc1ccccc1 ZINC000880580925 ED On-Demand Anodyne SIGMAR1 18 42 O[C@H]1CN(C[C@H]2COc3ccccc3O2)CC2(CCOCC2)C1 ZINC000880581071 DD On-Demand Anodyne ADRA2B 18 41 O[C@@H]1CN(C[C@H]2COc3ccccc3O2)CC2(CCOCC2)C1 ZINC000880581072 DD On-Demand Anodyne ADRA2B 18 41 O[C@H]1CN(C[C@@H]2COc3ccccc3O2)CC2(CCOCC2)C1 ZINC000880581073 DD On-Demand Anodyne ADRA2B 18 41 O[C@@H]1CN(C[C@@H]2COc3ccccc3O2)CC2(CCOCC2)C1 ZINC000880581074 DD On-Demand Anodyne ADRA2B 18 41 O=C(NC1CC2(CCC2)C1)c1cccn2nccc12 ZINC000880581115 CE On-Demand Anodyne JAK3 18 40 O=C(NC1CC2(CCC2)C1)c1cccn2nccc12 ZINC000880581115 CE On-Demand Anodyne TYK2 21 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880581174 FG On-Demand Anodyne RBP4 43 34 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880581175 FG On-Demand Anodyne RBP4 43 34 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880581176 FG On-Demand Anodyne RBP4 43 34 O[C@@H]1CN(Cc2ccc(CN3CCCCC3)cc2)CC2(CCOCC2)C1 ZINC000880581229 FG On-Demand Anodyne HRH3 21 49 O[C@H]1CN(Cc2ccc(CN3CCCCC3)cc2)CC2(CCOCC2)C1 ZINC000880581230 FG On-Demand Anodyne HRH3 21 49 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild CHRM1 16 47 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild DRD4 26 43 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild KCNH2 17 45 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild CHRM3 25 47 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild SIGMAR1 28 50 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild SSTR5 46 36 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild CCR3 64 48 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild MLNR 38 41 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild MCHR1 67 48 CC(C)(C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1)c1ccc(F)cc1F ZINC000880581296 GH On-Demand Mild CACNA1G 36 43 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild DRD4 27 44 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild CHRM3 15 41 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild SIGMAR1 20 44 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild SSTR5 48 39 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild CCR3 34 44 N#Cc1cccc(CN2CCC(NC(=O)c3ncsc3C3CC3)CC2)c1 ZINC000880581300 FG On-Demand Mild MCHR1 50 49 CN(C)[C@@H](CNC(=O)CN1C[C@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880581301 GD On-Demand Anodyne OPRK1 21 40 CN(C)[C@@H](CNC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880581302 GD On-Demand Anodyne OPRK1 21 40 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild DRD2 17 48 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild DRD4 46 52 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild ACHE 24 45 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild DRD3 15 45 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild KCNH2 15 42 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild HTR4 23 45 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild CHRM3 21 42 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild SIGMAR1 27 48 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild SSTR5 64 48 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild CCR3 48 45 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild PDE4B 48 34 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild UTS2R 19 41 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild MLNR 22 45 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild CXCR3 31 42 Cc1cnc(Cl)c(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880581307 FG On-Demand Mild MCHR1 72 53 CN(CCN1CCCCC1)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880581324 EE On-Demand Anodyne HRH3 15 47 CN(CCN1CCCCC1)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880581324 EE On-Demand Anodyne SIGMAR1 15 41 O=C(c1cnc2cc[nH]c2c1)N1CC[C@]2(C1)CC2(F)F ZINC000880581331 CE On-Demand Anodyne ACACA 17 49 O=C(c1cnc2cc[nH]c2c1)N1CC[C@@]2(C1)CC2(F)F ZINC000880581332 CE On-Demand Anodyne ACACA 17 49 COCc1ccnc(NC(=O)[C@H]2CO[C@@H](CCC(=O)OC(C)(C)C)C2)c1 ZINC000880581359 FF On-Demand Anodyne TYK2 44 33 COCc1ccnc(NC(=O)[C@@H]2CO[C@@H](CCC(=O)OC(C)(C)C)C2)c1 ZINC000880581360 FF On-Demand Anodyne TYK2 44 33 COCc1ccnc(NC(=O)[C@H]2CO[C@H](CCC(=O)OC(C)(C)C)C2)c1 ZINC000880581361 FF On-Demand Anodyne TYK2 44 33 COCc1ccnc(NC(=O)[C@@H]2CO[C@H](CCC(=O)OC(C)(C)C)C2)c1 ZINC000880581362 FF On-Demand Anodyne TYK2 44 33 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild DRD4 28 51 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild CHRM3 18 44 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild SIGMAR1 20 49 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild SSTR5 60 37 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild CCR3 41 44 N#Cc1cccc(CN2CCC(NC(=O)c3cccc4nsnc34)CC2)c1 ZINC000880581368 GF On-Demand Mild MCHR1 44 47 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2ccc(F)cc2s1 ZINC000880581372 GE On-Demand Anodyne CSNK1D 45 42 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2ccc(F)cc2s1 ZINC000880581372 GE On-Demand Anodyne SLC27A1 40 49 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2ccc(F)cc2s1 ZINC000880581374 GE On-Demand Anodyne CSNK1D 45 42 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2ccc(F)cc2s1 ZINC000880581374 GE On-Demand Anodyne SLC27A1 40 49 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581388 GD On-Demand Mild DRD4 21 42 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581388 GD On-Demand Mild SIGMAR1 21 48 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581388 GD On-Demand Mild CCR3 29 45 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581388 GD On-Demand Mild MLNR 16 44 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581388 GD On-Demand Mild MCHR1 40 47 N#Cc1cccc(CN2CCC(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581390 GD On-Demand Mild DRD4 21 42 N#Cc1cccc(CN2CCC(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581390 GD On-Demand Mild SIGMAR1 21 48 N#Cc1cccc(CN2CCC(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581390 GD On-Demand Mild CCR3 29 45 N#Cc1cccc(CN2CCC(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581390 GD On-Demand Mild MLNR 16 44 N#Cc1cccc(CN2CCC(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880581390 GD On-Demand Mild MCHR1 40 47 COCc1ccnc(NC(=O)c2ncsc2C2CC2)c1 ZINC000880581391 CF On-Demand Anodyne MAP1 95 39 COCc1ccnc(NC(=O)c2ncsc2C2CC2)c1 ZINC000880581391 CF On-Demand Anodyne TYK2 43 35 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild DRD4 26 46 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild SIGMAR1 20 47 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild SSTR5 48 41 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild CCR3 35 43 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild PRKCD 49 43 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild MLNR 16 40 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild PRKCQ 64 43 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild MCHR1 46 45 N#Cc1cccc(CN2CCC(NC(=O)c3cncc4[nH]ccc34)CC2)c1 ZINC000880581395 FF On-Demand Mild HPGDS 47 34 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2c(s1)CCC2 ZINC000880581399 FD On-Demand Anodyne SLC27A1 48 52 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2c(s1)CCC2 ZINC000880581400 FD On-Demand Anodyne SLC27A1 48 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(COC)ccn1 ZINC000880581430 FE On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(COC)ccn1 ZINC000880581430 FE On-Demand Anodyne FPR1 44 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(COC)ccn1 ZINC000880581431 FE On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(COC)ccn1 ZINC000880581431 FE On-Demand Anodyne FPR1 44 36 N#Cc1cccc(NC(=O)CCN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880581488 ED On-Demand Mild CCR3 15 41 N#Cc1cccc(NC(=O)CCN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880581488 ED On-Demand Mild MCHR1 41 44 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild DRD4 26 44 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild CHRM3 19 42 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild SIGMAR1 28 48 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild SSTR5 49 37 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild CCR3 39 46 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild MLNR 20 43 C=CC(C)(C)CC(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880581497 EG On-Demand Mild MCHR1 66 55 N#Cc1cccc(NC(=O)CCN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880581503 ED On-Demand Mild CCR3 15 41 N#Cc1cccc(NC(=O)CCN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880581503 ED On-Demand Mild MCHR1 41 44 CN(CCN1CCCCC1)C(=O)c1cccn2nccc12 ZINC000880581530 CD On-Demand Anodyne HNMT 19 40 CC(C)(C)OC(=O)N1CCC(CCN2C[C@H](O)CC3(CCOCC3)C2)CC1 ZINC000880581538 GF On-Demand Anodyne GPR119 27 40 CC(C)(C)OC(=O)N1CCC(CCN2C[C@@H](O)CC3(CCOCC3)C2)CC1 ZINC000880581539 GF On-Demand Anodyne GPR119 27 40 Cn1nc2c(c1C(=O)NC1CCN(Cc3cccc(C#N)c3)CC1)CSCC2 ZINC000880581540 GE On-Demand Mild DRD4 25 43 Cn1nc2c(c1C(=O)NC1CCN(Cc3cccc(C#N)c3)CC1)CSCC2 ZINC000880581540 GE On-Demand Mild SIGMAR1 17 41 Cn1nc2c(c1C(=O)NC1CCN(Cc3cccc(C#N)c3)CC1)CSCC2 ZINC000880581540 GE On-Demand Mild SSTR5 44 38 Cn1nc2c(c1C(=O)NC1CCN(Cc3cccc(C#N)c3)CC1)CSCC2 ZINC000880581540 GE On-Demand Mild CCR3 29 43 Cn1nc2c(c1C(=O)NC1CCN(Cc3cccc(C#N)c3)CC1)CSCC2 ZINC000880581540 GE On-Demand Mild MCHR1 43 44 CN(CCN1CCCCC1)C(=O)c1cncc2[nH]ccc12 ZINC000880581547 CE On-Demand Anodyne HPGDS 15 43 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild DRD4 21 40 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild SIGMAR1 16 40 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild SSTR5 47 36 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild CCR3 27 41 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild MAPKAPK2 18 42 N#Cc1cccc(CN2CCC(NC(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880581570 GF On-Demand Mild MCHR1 38 43 CC(=O)c1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880581572 ED On-Demand Anodyne CASR 16 42 CC(=O)c1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880581572 ED On-Demand Anodyne EPHX2 20 41 CC(=O)c1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880581573 ED On-Demand Anodyne CASR 16 42 CC(=O)c1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880581573 ED On-Demand Anodyne EPHX2 20 41 CN(CCN1CCCCC1)C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880581588 EE On-Demand Anodyne HRH3 15 47 CN(CCN1CCCCC1)C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880581589 EE On-Demand Anodyne HRH3 15 47 CC(C)(C(=O)N1CC[C@@]2(C1)CC2(F)F)c1ccc(C(F)(F)F)cc1 ZINC000880581637 EI On-Demand Anodyne EPHX2 17 42 CC(C)(C(=O)N1CC[C@]2(C1)CC2(F)F)c1ccc(C(F)(F)F)cc1 ZINC000880581638 EI On-Demand Anodyne EPHX2 17 42 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild DRD4 23 44 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild CHRM3 19 46 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild SIGMAR1 25 48 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild CCR3 32 46 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild MLNR 16 43 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880581685 ED On-Demand Mild MCHR1 53 53 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild DRD4 23 44 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild CHRM3 19 46 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild SIGMAR1 25 48 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild CCR3 32 46 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild MLNR 16 43 N#Cc1cccc(CN2CCC(NC(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880581686 ED On-Demand Mild MCHR1 53 53 CN(CCN1CCCCC1)C(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880581723 DG On-Demand Anodyne SLC6A1 52 34 CN(CCN1CCCCC1)C(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880581723 DG On-Demand Anodyne SIGMAR1 27 41 CN(CCN1CCCCC1)C(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880581723 DG On-Demand Anodyne TACR3 34 40 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880581903 DE On-Demand Anodyne CYP2J2 48 34 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880581906 DE On-Demand Anodyne CYP2J2 48 34 COCc1ccnc(NC(=O)C2CCC(S(C)(=O)=O)CC2)c1 ZINC000880581951 ED On-Demand Anodyne TYK2 60 44 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581997 FE On-Demand Anodyne CASR 20 45 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581997 FE On-Demand Anodyne CSNK1D 42 46 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581997 FE On-Demand Anodyne SLC27A1 32 54 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581999 FE On-Demand Anodyne CASR 20 45 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581999 FE On-Demand Anodyne CSNK1D 42 46 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2ccccc2s1 ZINC000880581999 FE On-Demand Anodyne SLC27A1 32 54 CN(CCN1CCCCC1)C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880582009 EE On-Demand Anodyne PLD2 45 38 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild DRD4 26 42 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild CHRM3 15 44 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild SIGMAR1 24 48 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild CCR3 34 46 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild MLNR 16 43 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild MCHR1 56 53 N#Cc1cccc(CN2CCC(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880582017 GD On-Demand Mild CACNA1G 15 41 N#Cc1cccc2c1CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880582029 DH On-Demand Mild SSTR1 33 42 N#Cc1cccc2c1CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880582031 DH On-Demand Mild SSTR1 33 42 O=C(Nc1ccccc1)c1cccc(CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880582036 GG On-Demand Anodyne KCNK3 78 40 O=C(Nc1ccccc1)c1cccc(CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880582038 GG On-Demand Anodyne KCNK3 78 40 COCc1ccnc(NC(=O)[C@@H]2CCc3nncn3CC2)c1 ZINC000880582071 DD On-Demand Anodyne TYK2 55 39 COCc1ccnc(NC(=O)[C@H]2CCc3nncn3CC2)c1 ZINC000880582072 DD On-Demand Anodyne TYK2 55 39 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA2 52 42 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA1 53 42 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA7 28 41 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA4 33 41 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA12 38 42 NS(=O)(=O)c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582101 FC On-Demand Anodyne CA9 43 41 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA2 52 42 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA1 53 42 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA7 28 41 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA4 33 41 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA12 38 42 NS(=O)(=O)c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582102 FC On-Demand Anodyne CA9 43 41 CN(CCN1CCCCC1)C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880582108 FD On-Demand Anodyne SLC6A1 76 34 CN(CCN1CCCCC1)C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880582108 FD On-Demand Anodyne HRH3 21 54 CN(CCN1CCCCC1)C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880582108 FD On-Demand Anodyne SIGMAR1 40 43 CN(CCN1CCCCC1)C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880582108 FD On-Demand Anodyne AMY2 46 33 CN(CCN1CCCCC1)C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880582108 FD On-Demand Anodyne CACNA1G 21 40 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild DRD4 32 46 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild ACHE 22 41 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild KCNH2 15 44 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild HTR4 18 41 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild CHRM3 27 46 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild SIGMAR1 24 44 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild SSTR5 70 40 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild CCR3 43 46 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild MLNR 27 47 Cn1nnc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)n1 ZINC000880582118 EC On-Demand Mild MCHR1 69 49 CCOc1ccccc1NC(=O)CCN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582161 FE On-Demand Anodyne HCN1 44 36 CCOc1ccccc1NC(=O)CCN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582163 FE On-Demand Anodyne HCN1 44 36 O[C@@H]1CN(CCc2ccccc2)CC2(CCOCC2)C1 ZINC000880582174 CE On-Demand Anodyne SIGMAR1 24 43 O[C@H]1CN(CCc2ccccc2)CC2(CCOCC2)C1 ZINC000880582176 CE On-Demand Anodyne SIGMAR1 24 43 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild DRD2 17 46 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild DRD4 45 52 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild ACHE 25 44 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild KCNH2 17 49 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild CHRM3 26 47 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild SIGMAR1 29 47 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild SSTR5 65 44 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild CCR3 44 48 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild MLNR 20 45 Cc1coc(C(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)c1 ZINC000880582207 DF On-Demand Mild MCHR1 72 58 O[C@@H]1CN(C[C@H]2CC(c3ccc(Cl)cc3)=NO2)CC2(CCOCC2)C1 ZINC000880582225 FF On-Demand Anodyne LUCI_PHOPY 59 42 O[C@H]1CN(C[C@H]2CC(c3ccc(Cl)cc3)=NO2)CC2(CCOCC2)C1 ZINC000880582227 FF On-Demand Anodyne LUCI_PHOPY 59 42 O[C@@H]1CN(C[C@@H]2CC(c3ccc(Cl)cc3)=NO2)CC2(CCOCC2)C1 ZINC000880582229 FF On-Demand Anodyne LUCI_PHOPY 59 42 O[C@H]1CN(C[C@@H]2CC(c3ccc(Cl)cc3)=NO2)CC2(CCOCC2)C1 ZINC000880582230 FF On-Demand Anodyne LUCI_PHOPY 59 42 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild DRD4 32 49 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild ACHE 17 44 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild KCNH2 15 45 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild CHRM3 18 43 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild SIGMAR1 21 50 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild SSTR5 65 42 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild CCR3 42 45 N#Cc1cccc(CN2CCC(NC(=O)c3cccn4nccc34)CC2)c1 ZINC000880582250 FF On-Demand Mild MCHR1 56 49 CN(CCN1CCCCC1)C(=O)c1cnc2cc[nH]c2c1 ZINC000880582290 CE On-Demand Anodyne TACR2 20 42 CN(CCN1CCCCC1)C(=O)c1cnc2cc[nH]c2c1 ZINC000880582290 CE On-Demand Anodyne HRH3 18 43 CN(CCN1CCCCC1)C(=O)c1cnc2cc[nH]c2c1 ZINC000880582290 CE On-Demand Anodyne HNMT 55 38 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)OCc1ccccc1 ZINC000880582297 ED On-Demand Anodyne SLC12A5 59 35 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)OCc1ccccc1 ZINC000880582298 ED On-Demand Anodyne SLC12A5 59 35 O[C@@H]1CN(Cc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880582320 CE On-Demand Anodyne SIGMAR1 16 41 O[C@H]1CN(Cc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880582321 CE On-Demand Anodyne SIGMAR1 16 41 C[C@@H](C(=O)Nc1nc2ccccc2s1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582335 GE On-Demand Anodyne CASR 15 42 C[C@H](C(=O)Nc1nc2ccccc2s1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582336 GE On-Demand Anodyne CASR 15 42 C[C@@H](C(=O)Nc1nc2ccccc2s1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582337 GE On-Demand Anodyne CASR 15 42 C[C@H](C(=O)Nc1nc2ccccc2s1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582338 GE On-Demand Anodyne CASR 15 42 COCc1ccnc(NC(=O)[C@@H]2C[C@]2(C)c2ccccc2)c1 ZINC000880582339 CG On-Demand Anodyne TYK2 45 33 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582340 GH On-Demand Anodyne PRNP 41 37 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582340 GH On-Demand Anodyne KCNK3 89 39 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582340 GH On-Demand Anodyne KCNK9 41 38 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582342 GH On-Demand Anodyne PRNP 41 37 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582342 GH On-Demand Anodyne KCNK3 89 39 C[C@@H](c1cccc(NC(=O)c2ccccc2)c1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582342 GH On-Demand Anodyne KCNK9 41 38 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild DRD4 32 45 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild ACHE 23 40 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild HRH2 30 40 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild KCNH2 15 43 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild CHRM3 23 45 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild SIGMAR1 35 53 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild SSTR5 79 41 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild CCR3 45 50 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild MLNR 24 44 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild SLC6A5 24 40 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild MCHR1 79 57 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild CACNA1G 15 40 N#Cc1cccc(CN2CCC(NC(=O)COC3CC3)CC2)c1 ZINC000880582474 DD On-Demand Mild CCR8 15 48 CN(CCN1CCCCC1)C(=O)c1cccc2nsnc12 ZINC000880582488 DE On-Demand Anodyne HNMT 37 40 O[C@H](COc1ccccc1C(F)(F)F)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582515 GE On-Demand Anodyne ABCB1 42 38 O[C@H](COc1ccccc1C(F)(F)F)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582516 GE On-Demand Anodyne ABCB1 42 38 O[C@@H](COc1ccccc1C(F)(F)F)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582517 GE On-Demand Anodyne ABCB1 42 38 O[C@@H]1CN(C[C@@H](O)COc2ccccc2C(F)(F)F)CC2(CCOCC2)C1 ZINC000880582518 GE On-Demand Anodyne ABCB1 42 38 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild CHRM2 17 44 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild DRD4 32 44 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild CHRM3 29 51 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild SIGMAR1 44 49 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild CCR3 55 49 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild MLNR 19 42 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild SLC6A5 19 40 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild MCHR1 67 50 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild CACNA1G 18 42 N#Cc1cccc(CN2CCC(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880582519 GH On-Demand Mild CCR8 21 51 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880582528 GF On-Demand Anodyne EPHX2 26 45 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880582529 GF On-Demand Anodyne EPHX2 26 45 COCc1ccnc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582557 EF On-Demand Anodyne RAF1 18 48 COCc1ccnc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582557 EF On-Demand Anodyne FAAH 16 45 COCc1ccnc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582557 EF On-Demand Anodyne TYK2 46 43 COCc1ccnc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582558 EF On-Demand Anodyne RAF1 18 48 COCc1ccnc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582558 EF On-Demand Anodyne FAAH 16 45 COCc1ccnc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880582558 EF On-Demand Anodyne TYK2 46 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc2c(s1)CCCC2 ZINC000880582566 FD On-Demand Anodyne SLC27A1 55 52 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc2c(s1)CCCC2 ZINC000880582567 FD On-Demand Anodyne SLC27A1 55 52 Cc1cccc(C(=O)NNC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880582581 FC On-Demand Reactive KCNK3 43 34 Cc1cccc(C(=O)NNC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880582582 FC On-Demand Reactive KCNK3 43 34 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)CC2)c1 ZINC000880582621 FE On-Demand Mild DRD4 18 40 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)CC2)c1 ZINC000880582621 FE On-Demand Mild SIGMAR1 19 43 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)CC2)c1 ZINC000880582621 FE On-Demand Mild CCR3 27 44 N#Cc1cccc(CN2CCC(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)CC2)c1 ZINC000880582621 FE On-Demand Mild MCHR1 43 49 N#Cc1ccc(Cl)cc1NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880582635 FE On-Demand Mild TRPV4 41 33 N#Cc1ccc(Cl)cc1NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880582637 FE On-Demand Mild TRPV4 41 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582655 FH On-Demand Anodyne PAPA1_CARPA 39 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582655 FH On-Demand Anodyne CTSK 20 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582655 FH On-Demand Anodyne CTSL 21 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582655 FH On-Demand Anodyne FPR1 54 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582658 FH On-Demand Anodyne PAPA1_CARPA 39 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582658 FH On-Demand Anodyne CTSK 20 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582658 FH On-Demand Anodyne CTSL 21 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C)c(SC)c1 ZINC000880582658 FH On-Demand Anodyne FPR1 54 41 O=c1cc(CN2C[C@@H](O)CC3(CCOCC3)C2)c2ccc(O)cc2o1 ZINC000880582669 ED On-Demand Anodyne HSD17B3 30 46 O[C@@H]1CN(Cc2ccc(F)cc2Cl)CC2(CCOCC2)C1 ZINC000880582670 DF On-Demand Anodyne P2RX7 54 42 O=c1cc(CN2C[C@H](O)CC3(CCOCC3)C2)c2ccc(O)cc2o1 ZINC000880582671 ED On-Demand Anodyne HSD17B3 30 46 O[C@H]1CN(Cc2ccc(F)cc2Cl)CC2(CCOCC2)C1 ZINC000880582672 DF On-Demand Anodyne P2RX7 54 42 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild DRD4 28 50 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild KCNH2 15 44 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild HTR4 16 40 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild CHRM3 16 41 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild SIGMAR1 18 44 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild SSTR5 64 42 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild CCR3 41 42 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild PDE4B 54 36 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild MLNR 15 40 Cc1nc(C(C)C)ncc1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880582688 GG On-Demand Mild MCHR1 56 47 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild DRD4 34 46 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild ACHE 29 43 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild KCNH2 15 43 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild CHRM3 16 41 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild SIGMAR1 22 46 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild SSTR5 53 39 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild CCR3 41 45 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild MLNR 23 45 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild CXCR3 15 40 N#Cc1cccc(CN2CCC(NC(=O)c3ncccc3-c3ccccn3)CC2)c1 ZINC000880582732 GG On-Demand Mild MCHR1 49 47 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880582741 GE On-Demand Anodyne P2RY1 54 38 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880582741 GE On-Demand Anodyne EPHX2 64 46 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880582743 GE On-Demand Anodyne P2RY1 54 38 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880582743 GE On-Demand Anodyne EPHX2 64 46 CCOC(=O)Nc1ccc(C(=O)NC[C@@H](C(CC)CC)N2CCOCC2)cc1 ZINC000880582812 GG On-Demand Anodyne F3 75 34 CCOC(=O)Nc1ccc(C(=O)NC[C@H](C(CC)CC)N2CCOCC2)cc1 ZINC000880582814 GG On-Demand Anodyne F3 75 34 CS(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582824 FD On-Demand Anodyne MMP13 47 42 CS(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582824 FD On-Demand Anodyne ADAM17 23 42 CS(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582824 FD On-Demand Anodyne MMP8 15 40 CS(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582824 FD On-Demand Anodyne MMP1 25 41 CS(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582825 FD On-Demand Anodyne MMP13 47 42 CS(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582825 FD On-Demand Anodyne ADAM17 23 42 CS(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582825 FD On-Demand Anodyne MMP8 15 40 CS(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880582825 FD On-Demand Anodyne MMP1 25 41 COCc1ccnc(NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)c1 ZINC000880582836 FD On-Demand Anodyne TYK2 51 35 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880582885 GD On-Demand Anodyne MAPK1 22 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880582886 GD On-Demand Anodyne MAPK1 22 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@]2(C1)CC2(F)F ZINC000880582901 GF On-Demand Anodyne PREP 46 47 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@]2(C1)CC2(F)F ZINC000880582901 GF On-Demand Anodyne SLC12A5 66 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@]2(C1)CC2(F)F ZINC000880582902 GF On-Demand Anodyne PREP 46 47 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@]2(C1)CC2(F)F ZINC000880582902 GF On-Demand Anodyne SLC12A5 66 36 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild DRD4 30 43 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild ACHE 15 42 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild KCNH2 15 43 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild SIGMAR1 19 43 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild SSTR5 73 37 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild CCR3 39 43 N#Cc1cccc(CN2CCC(NC(=O)c3coc(-c4ccccn4)n3)CC2)c1 ZINC000880582961 GG On-Demand Mild MCHR1 44 45 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nccs1 ZINC000880582998 DC On-Demand Anodyne MAP1 96 45 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nccs1 ZINC000880582999 DC On-Demand Anodyne MAP1 96 45 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(C(F)(F)F)cc1 ZINC000880583011 FF On-Demand Anodyne EPHX2 36 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(C(F)(F)F)cc1 ZINC000880583013 FF On-Demand Anodyne EPHX2 36 43 N#Cc1cccc(CN2CCC(NC(=O)c3cnc(CC4CC4)s3)CC2)c1 ZINC000880583014 GG On-Demand Mild DRD4 26 43 N#Cc1cccc(CN2CCC(NC(=O)c3cnc(CC4CC4)s3)CC2)c1 ZINC000880583014 GG On-Demand Mild SIGMAR1 24 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc(CC4CC4)s3)CC2)c1 ZINC000880583014 GG On-Demand Mild SSTR5 50 40 N#Cc1cccc(CN2CCC(NC(=O)c3cnc(CC4CC4)s3)CC2)c1 ZINC000880583014 GG On-Demand Mild CCR3 42 50 N#Cc1cccc(CN2CCC(NC(=O)c3cnc(CC4CC4)s3)CC2)c1 ZINC000880583014 GG On-Demand Mild MCHR1 52 46 CC1(C)CC[C@@H](CC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)OC1 ZINC000880583035 FG On-Demand Mild DRD4 23 43 CC1(C)CC[C@@H](CC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)OC1 ZINC000880583035 FG On-Demand Mild SIGMAR1 24 48 CC1(C)CC[C@@H](CC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)OC1 ZINC000880583035 FG On-Demand Mild CCR3 35 44 CC1(C)CC[C@@H](CC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)OC1 ZINC000880583035 FG On-Demand Mild MLNR 15 41 CC1(C)CC[C@@H](CC(=O)NC2CCN(Cc3cccc(C#N)c3)CC2)OC1 ZINC000880583035 FG On-Demand Mild MCHR1 57 52 CN(CCN1CCCCC1)C(=O)c1ncccc1-c1ccccn1 ZINC000880583039 DF On-Demand Anodyne HRH3 15 46 CN(CCN1CCCCC1)C(=O)c1ncccc1-c1ccccn1 ZINC000880583039 DF On-Demand Anodyne HNMT 38 43 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild DRD4 21 41 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild SIGMAR1 18 41 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild SSTR5 52 37 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild CCR3 29 42 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild MLNR 29 44 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583094 GF On-Demand Mild MCHR1 43 46 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild DRD4 21 41 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild SIGMAR1 18 41 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild SSTR5 52 37 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild CCR3 29 42 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild MLNR 29 44 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583095 GF On-Demand Mild MCHR1 43 46 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild DRD4 21 41 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild SIGMAR1 18 41 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild SSTR5 52 37 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild CCR3 29 42 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild MLNR 29 44 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583096 GF On-Demand Mild MCHR1 43 46 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild DRD4 21 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild SIGMAR1 18 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild SSTR5 52 37 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild CCR3 29 42 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild MLNR 29 44 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC1CCN(Cc2cccc(C#N)c2)CC1 ZINC000880583098 GF On-Demand Mild MCHR1 43 46 CSc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583116 EH On-Demand Anodyne HTR1F 23 43 CSc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583116 EH On-Demand Anodyne MAPK14 17 40 CSc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583116 EH On-Demand Anodyne KCNK3 42 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(C#N)c2C1 ZINC000880583151 FE On-Demand Mild PAPA1_CARPA 36 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(C#N)c2C1 ZINC000880583152 FE On-Demand Mild PAPA1_CARPA 36 41 O=C1NCC[C@H]1CC(=O)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880583168 EE On-Demand Anodyne PREP 47 34 O=C1NCC[C@@H]1CC(=O)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880583169 EE On-Demand Anodyne PREP 47 34 CC(C)(C(=O)N1Cc2cccc(C#N)c2C1)c1ccc(F)cc1F ZINC000880583170 EH On-Demand Mild AR 25 42 O=C(COC1CC1)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880583199 DF On-Demand Anodyne CPT1A 77 35 O=C(COC1CC1)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880583199 DF On-Demand Anodyne CPT2 40 32 CSc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583209 EH On-Demand Anodyne HTR1F 23 43 CSc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583209 EH On-Demand Anodyne MAPK14 17 40 CSc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1C ZINC000880583209 EH On-Demand Anodyne KCNK3 42 35 C[C@H](C(=O)Nc1nccs1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880583307 ED On-Demand Anodyne MAP1 60 34 C[C@@H](C(=O)Nc1nccs1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880583308 ED On-Demand Anodyne MAP1 60 34 C[C@@H](C(=O)Nc1nccs1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880583310 ED On-Demand Anodyne MAP1 60 34 C[C@H](C(=O)Nc1nccs1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880583312 ED On-Demand Anodyne MAP1 60 34 O[C@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583341 DE On-Demand Anodyne UGCG 48 36 O[C@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583341 DE On-Demand Anodyne GBA 28 41 O[C@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583341 DE On-Demand Anodyne GBA2 64 41 O[C@@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583342 DE On-Demand Anodyne UGCG 48 36 O[C@@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583342 DE On-Demand Anodyne GBA 28 41 O[C@@H]1CN(CCCOCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583342 DE On-Demand Anodyne GBA2 64 41 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCCCC2)nc1 ZINC000880583354 GD On-Demand Anodyne SLC27A1 52 39 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCCCC2)nc1 ZINC000880583356 GD On-Demand Anodyne SLC27A1 52 39 O[C@H]1CN(CCCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583376 DF On-Demand Anodyne OPRM1 15 41 O[C@H]1CN(CCCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583376 DF On-Demand Anodyne SIGMAR1 32 44 O[C@@H]1CN(CCCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583378 DF On-Demand Anodyne OPRM1 15 41 O[C@@H]1CN(CCCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880583378 DF On-Demand Anodyne SIGMAR1 32 44 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NOCc1ccccc1 ZINC000880583400 ED On-Demand Anodyne SLC12A5 42 35 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NOCc1ccccc1 ZINC000880583401 ED On-Demand Anodyne SLC12A5 42 35 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(F)c(Cl)c1 ZINC000880583428 FE On-Demand Anodyne ERBB4 49 38 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(F)c(Cl)c1 ZINC000880583428 FE On-Demand Anodyne MCHR1 32 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(F)c(Cl)c1 ZINC000880583429 FE On-Demand Anodyne ERBB4 49 38 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(F)c(Cl)c1 ZINC000880583429 FE On-Demand Anodyne MCHR1 32 43 CN(CC(=O)NC(C)(C)C)C(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c([N+](=O)[O-])c2)cc1 ZINC000880583441 JG On-Demand Bother LIMK2 33 43 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880583466 EH On-Demand Anodyne PREP 48 35 CC[C@@H](C(=O)OC(C)(C)C)N(C)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880583483 FF On-Demand Anodyne KCNQ2 43 34 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)N1CCc2ccccc2C1 ZINC000880583496 FD On-Demand Anodyne HTR7 15 40 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)N1CCc2ccccc2C1 ZINC000880583497 FD On-Demand Anodyne HTR7 15 40 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild DRD4 29 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild ACHE 17 41 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild CHRM3 17 44 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild SIGMAR1 22 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild SSTR5 75 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild CCR3 37 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild JAK1 17 40 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild MLNR 25 41 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild SLC6A5 29 41 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild CXCR3 27 42 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild MCHR1 63 46 N#Cc1cccc(CN2CCC(NC(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880583531 FF On-Demand Mild HPGDS 36 40 O[C@@H]1CN(Cc2ccc3c(c2)COC3)CC2(CCOCC2)C1 ZINC000880583537 DE On-Demand Anodyne MCHR2 44 34 O[C@H]1CN(Cc2ccc3c(c2)COC3)CC2(CCOCC2)C1 ZINC000880583539 DE On-Demand Anodyne MCHR2 44 34 COCc1ccnc(NC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880583550 FH On-Demand Anodyne INHA 55 41 COCc1ccnc(NC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880583550 FH On-Demand Anodyne ENPP1 57 35 N#CC(CCN1C[C@H](O)CC2(CCOCC2)C1)(c1ccccc1)c1ccccc1 ZINC000880583570 GH On-Demand Mild CHRM3 43 30 N#CC(CCN1C[C@@H](O)CC2(CCOCC2)C1)(c1ccccc1)c1ccccc1 ZINC000880583574 GH On-Demand Mild CHRM3 43 30 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3C[C@H]3C3CC3)CC2)c1 ZINC000880583596 EG On-Demand Mild DRD4 21 42 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3C[C@H]3C3CC3)CC2)c1 ZINC000880583596 EG On-Demand Mild SIGMAR1 27 49 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3C[C@H]3C3CC3)CC2)c1 ZINC000880583596 EG On-Demand Mild CCR3 33 47 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3C[C@H]3C3CC3)CC2)c1 ZINC000880583596 EG On-Demand Mild MLNR 16 42 N#Cc1cccc(CN2CCC(NC(=O)C[C@@H]3C[C@H]3C3CC3)CC2)c1 ZINC000880583596 EG On-Demand Mild MCHR1 49 54 CCCOc1cccc(CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880583617 DF On-Demand Anodyne HRH2 27 41 CCCOc1cccc(CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880583618 DF On-Demand Anodyne HRH2 27 41 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880583635 FG On-Demand Anodyne CACNA1I 42 33 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880583635 FG On-Demand Anodyne SIRT3 41 36 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880583635 FG On-Demand Anodyne SIRT2 47 36 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880583635 FG On-Demand Anodyne SIRT1 42 36 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cc(C(F)F)[nH]n2)CC1 ZINC000880583635 FG On-Demand Anodyne GPR119 46 46 CSc1cc(NC(=O)C2CCC(S(C)(=O)=O)CC2)ccc1C ZINC000880583646 EG On-Demand Anodyne EPHX2 20 42 COCCc1ccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583653 GD On-Demand Anodyne ADRB1 15 45 COCCc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583657 GD On-Demand Anodyne ADRB1 15 45 COCCc1ccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583662 GD On-Demand Anodyne ADRB1 15 45 COCCc1ccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583666 GD On-Demand Anodyne ADRB1 15 45 Cc1c(NC(=O)COC2CC2)cnn1-c1ccc(F)cc1F ZINC000880583668 DF On-Demand Anodyne MAPK14 22 45 C[C@H](C(=O)Nc1cccnc1Cl)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880583830 FD On-Demand Anodyne G2YM83_BOTF4 68 34 C[C@H](C(=O)Nc1cccnc1Cl)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880583831 FD On-Demand Anodyne G2YM83_BOTF4 68 34 O[C@H]1CN(Cc2ccc(-n3ccnc3)cc2)CC2(CCOCC2)C1 ZINC000880583859 EE On-Demand Anodyne CYP2C19 15 41 O[C@@H]1CN(Cc2ccc(-n3ccnc3)cc2)CC2(CCOCC2)C1 ZINC000880583860 EE On-Demand Anodyne CYP2C19 15 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCc1ccc2c(c1)OCO2 ZINC000880583867 FC On-Demand Anodyne NOS2 99 38 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCc1ccc2c(c1)OCO2 ZINC000880583868 FC On-Demand Anodyne NOS2 99 38 CSc1cc(NC(=O)COC2CC2)ccc1C ZINC000880583873 CF On-Demand Anodyne TIMP3 49 32 O=C(Nc1ccccc1)c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583885 GG On-Demand Anodyne PRNP 50 40 O=C(Nc1ccccc1)c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583885 GG On-Demand Anodyne NOD1 18 42 O=C(Nc1ccccc1)c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583885 GG On-Demand Anodyne NOD2 48 40 O=C(Nc1ccccc1)c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583885 GG On-Demand Anodyne KCNK3 49 37 O=C(Nc1ccccc1)c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583886 GG On-Demand Anodyne PRNP 50 40 O=C(Nc1ccccc1)c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583886 GG On-Demand Anodyne NOD1 18 42 O=C(Nc1ccccc1)c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583886 GG On-Demand Anodyne NOD2 48 40 O=C(Nc1ccccc1)c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880583886 GG On-Demand Anodyne KCNK3 49 37 O=C(CCCN1C[C@@H](O)CC2(CCOCC2)C1)c1ccc(Br)cc1 ZINC000880583924 GG On-Demand Anodyne CYP2J2 51 36 O=C(CCCN1C[C@H](O)CC2(CCOCC2)C1)c1ccc(Br)cc1 ZINC000880583925 GG On-Demand Anodyne CYP2J2 51 36 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne GRIN2B 18 40 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne CACNA1I 51 35 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne SIRT3 46 39 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne SIRT2 50 39 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne SIRT1 48 39 Cc1coc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880583930 EG On-Demand Anodyne GPR119 49 48 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCCC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880583950 GG On-Demand Anodyne GPR119 40 44 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCCC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880583951 GG On-Demand Anodyne GPR119 40 44 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCCC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880583952 GG On-Demand Anodyne GPR119 40 44 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCCC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880583953 GG On-Demand Anodyne GPR119 40 44 CSc1cc(NC(=O)c2ncsc2C2CC2)ccc1C ZINC000880584021 DI On-Demand Anodyne MAP1 71 36 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NC(=O)Nc1ccccc1 ZINC000880584047 ED On-Demand Anodyne EPHX2 19 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NC(=O)Nc1ccccc1 ZINC000880584048 ED On-Demand Anodyne EPHX2 19 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880584068 GD On-Demand Anodyne EPHX2 19 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880584069 GD On-Demand Anodyne EPHX2 19 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(Oc2ccccc2)cc1 ZINC000880584070 GG On-Demand Anodyne LTA4H 44 48 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(Oc2ccccc2)cc1 ZINC000880584070 GG On-Demand Anodyne EPHX2 18 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(Oc2ccccc2)cc1 ZINC000880584071 GG On-Demand Anodyne LTA4H 44 48 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(Oc2ccccc2)cc1 ZINC000880584071 GG On-Demand Anodyne EPHX2 18 40 CC(C)(C)OC(=O)N1CCC(CCNC(=O)[C@H]2CCc3nncn3CC2)CC1 ZINC000880584099 GE On-Demand Anodyne GPR119 38 43 CC(C)(C)OC(=O)N1CCC(CCNC(=O)[C@@H]2CCc3nncn3CC2)CC1 ZINC000880584101 GE On-Demand Anodyne GPR119 38 43 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne GRIN2B 19 40 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne CACNA1I 50 35 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne SIRT3 44 40 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne SIRT2 47 40 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne SIRT1 42 40 Cc1ncc(CC(=O)NCCC2CCN(C(=O)OC(C)(C)C)CC2)o1 ZINC000880584123 FF On-Demand Anodyne GPR119 58 47 O[C@@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584189 EE On-Demand Anodyne CHRM2 15 43 O[C@@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584189 EE On-Demand Anodyne CHRM3 16 43 O[C@@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584189 EE On-Demand Anodyne SIGMAR1 54 39 O[C@@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584189 EE On-Demand Anodyne SLC18A3 25 43 O[C@@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584190 EE On-Demand Anodyne CHRM2 15 43 O[C@@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584190 EE On-Demand Anodyne CHRM3 16 43 O[C@@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584190 EE On-Demand Anodyne SIGMAR1 54 39 O[C@@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584190 EE On-Demand Anodyne SLC18A3 25 43 O[C@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584191 EE On-Demand Anodyne CHRM2 15 43 O[C@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584191 EE On-Demand Anodyne CHRM3 16 43 O[C@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584191 EE On-Demand Anodyne SIGMAR1 54 39 O[C@H]1CN([C@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584191 EE On-Demand Anodyne SLC18A3 25 43 O[C@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584192 EE On-Demand Anodyne CHRM2 15 43 O[C@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584192 EE On-Demand Anodyne CHRM3 16 43 O[C@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584192 EE On-Demand Anodyne SIGMAR1 54 39 O[C@H]1CN([C@@H]2CCN(Cc3ccccc3)C2)CC2(CCOCC2)C1 ZINC000880584192 EE On-Demand Anodyne SLC18A3 25 43 O[C@@H]1CN(C[C@H]2CN(Cc3ccccc3)CCCO2)CC2(CCOCC2)C1 ZINC000880584214 FE On-Demand Anodyne DRD4 15 43 O[C@H]1CN(C[C@H]2CN(Cc3ccccc3)CCCO2)CC2(CCOCC2)C1 ZINC000880584215 FE On-Demand Anodyne DRD4 15 43 O[C@H]1CN(C[C@@H]2CN(Cc3ccccc3)CCCO2)CC2(CCOCC2)C1 ZINC000880584216 FE On-Demand Anodyne DRD4 15 43 O[C@@H]1CN(C[C@@H]2CN(Cc3ccccc3)CCCO2)CC2(CCOCC2)C1 ZINC000880584217 FE On-Demand Anodyne DRD4 15 43 N#Cc1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880584325 ED On-Demand Mild CCR3 15 40 N#Cc1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880584325 ED On-Demand Mild MCHR1 45 44 N#Cc1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880584329 ED On-Demand Mild CCR3 15 40 N#Cc1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880584329 ED On-Demand Mild MCHR1 45 44 CN(CCN1CCCCC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880584346 EE On-Demand Anodyne SLC6A4 17 42 CN(CCN1CCCCC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880584346 EE On-Demand Anodyne MPO 51 46 O[C@@H]1CN(CCc2ccc(F)c(F)c2)CC2(CCOCC2)C1 ZINC000880584347 DE On-Demand Anodyne ABCC1 61 36 O[C@H]1CN(CCc2ccc(F)c(F)c2)CC2(CCOCC2)C1 ZINC000880584349 DE On-Demand Anodyne ABCC1 61 36 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCc1ccc(Cl)cc1 ZINC000880584411 FD On-Demand Anodyne DPOL_VZVD 40 37 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCc1ccc(Cl)cc1 ZINC000880584412 FD On-Demand Anodyne DPOL_VZVD 40 37 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2c[nH]cc2C2CC2)CC1 ZINC000880584437 FH On-Demand Anodyne CACNA1I 42 33 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2c[nH]cc2C2CC2)CC1 ZINC000880584437 FH On-Demand Anodyne GPR119 38 44 CSc1cc(NC(=O)[C@@H]2CCc3nncn3CC2)ccc1C ZINC000880584521 DF On-Demand Anodyne EPHX2 19 41 CSc1cc(NC(=O)[C@H]2CCc3nncn3CC2)ccc1C ZINC000880584522 DF On-Demand Anodyne EPHX2 19 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)cc1 ZINC000880584616 EE On-Demand Anodyne EPHX2 18 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)cc1 ZINC000880584617 EE On-Demand Anodyne EPHX2 18 40 O=[N+]([O-])c1ccc(CCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584622 DE On-Demand Bother KCNJ1 33 49 O=[N+]([O-])c1ccc(CCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584624 DE On-Demand Bother KCNJ1 33 49 COc1ccc(NC(=O)[C@H](C)N2C[C@H](O)CC3(CCOCC3)C2)cc1OC ZINC000880584665 GD On-Demand Anodyne ENPP1 68 33 COc1ccc(NC(=O)[C@H](C)N2C[C@@H](O)CC3(CCOCC3)C2)cc1OC ZINC000880584667 GD On-Demand Anodyne ENPP1 68 33 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584680 GF On-Demand Anodyne ROCK1 20 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584680 GF On-Demand Anodyne SPHK2 44 31 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584680 GF On-Demand Anodyne HDAC9 15 44 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880584682 FF On-Demand Anodyne EPHX2 20 42 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880584682 FF On-Demand Anodyne MCHR1 16 48 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584683 GF On-Demand Anodyne ROCK1 20 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584683 GF On-Demand Anodyne SPHK2 44 31 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1nc(-c2ccccc2)cs1 ZINC000880584683 GF On-Demand Anodyne HDAC9 15 44 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880584684 FF On-Demand Anodyne EPHX2 20 42 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880584684 FF On-Demand Anodyne MCHR1 16 48 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880584704 GD On-Demand Anodyne SSTR4 50 35 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880584704 GD On-Demand Anodyne SSTR5 41 35 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880584705 GD On-Demand Anodyne SSTR4 50 35 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCc2[nH]c3ccccc3c2C1 ZINC000880584705 GD On-Demand Anodyne SSTR5 41 35 N#Cc1cccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880584866 EE On-Demand Mild EPHX2 19 41 N#Cc1cccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880584868 EE On-Demand Mild EPHX2 19 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCCOc1ccc2c(c1)OCO2 ZINC000880584909 GC On-Demand Anodyne EDNRA 21 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCCOc1ccc2c(c1)OCO2 ZINC000880584913 GC On-Demand Anodyne EDNRA 21 40 CS(=O)(=O)c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584914 GD On-Demand Anodyne HRH3 28 46 CS(=O)(=O)c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584914 GD On-Demand Anodyne MMP13 46 43 CS(=O)(=O)c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584914 GD On-Demand Anodyne ADAM17 24 43 CS(=O)(=O)c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584914 GD On-Demand Anodyne MMP3 31 41 CS(=O)(=O)c1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584914 GD On-Demand Anodyne EPHX2 15 40 CS(=O)(=O)c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584916 GD On-Demand Anodyne HRH3 28 46 CS(=O)(=O)c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584916 GD On-Demand Anodyne MMP13 46 43 CS(=O)(=O)c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584916 GD On-Demand Anodyne ADAM17 24 43 CS(=O)(=O)c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584916 GD On-Demand Anodyne MMP3 31 41 CS(=O)(=O)c1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584916 GD On-Demand Anodyne EPHX2 15 40 O=C(c1ncccc1-c1ccccn1)N1CCC[C@@H](F)C1 ZINC000880584921 CF On-Demand Anodyne MAP3K12 29 40 O=C(c1ncccc1-c1ccccn1)N1CCC[C@H](F)C1 ZINC000880584923 CF On-Demand Anodyne MAP3K12 29 40 N#Cc1ccc(CNC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584952 ED On-Demand Mild CTSC 15 40 N#Cc1ccc(CNC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880584954 ED On-Demand Mild CTSC 15 40 Oc1nc(CN2C[C@H](O)CC3(CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880584973 FE On-Demand Anodyne CDC7 16 49 Oc1nc(CN2C[C@H](O)CC3(CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880584973 FE On-Demand Anodyne PIM3 18 52 Oc1nc(CN2C[C@@H](O)CC3(CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880584974 FE On-Demand Anodyne CDC7 16 49 Oc1nc(CN2C[C@@H](O)CC3(CCOCC3)C2)nc2c1oc1ccccc12 ZINC000880584974 FE On-Demand Anodyne PIM3 18 52 N#Cc1c(NC(=O)CCN2C[C@@H](O)CC3(CCOCC3)C2)sc2c1CCC2 ZINC000880585000 GE On-Demand Mild VIPR1 29 46 N#Cc1c(NC(=O)CCN2C[C@H](O)CC3(CCOCC3)C2)sc2c1CCC2 ZINC000880585001 GE On-Demand Mild VIPR1 29 46 Cc1nc(C(C)C)ncc1C(=O)Nc1cnn(-c2ccc(F)cc2F)c1C ZINC000880585043 FH On-Demand Anodyne MAPK14 15 42 CC(C)(C)OC(=O)N1CCC(CCNC(=O)C[C@@H]2CCNC2=O)CC1 ZINC000880585050 FD On-Demand Anodyne GPR119 34 46 CC(C)(C)OC(=O)N1CCC(CCNC(=O)C[C@H]2CCNC2=O)CC1 ZINC000880585051 FD On-Demand Anodyne GPR119 34 46 CC(C)(C)OC(=O)N1CCC(CCNC(=O)COC2CC2)CC1 ZINC000880585052 EE On-Demand Anodyne GPR119 39 48 CC(C)(C(=O)N1CCC[C@@H](F)C1)c1ccc(F)cc1F ZINC000880585104 CG On-Demand Anodyne DPP4 15 41 CC(C)(C(=O)N1CCC[C@H](F)C1)c1ccc(F)cc1F ZINC000880585128 CG On-Demand Anodyne DPP4 15 41 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585188 FD On-Demand Anodyne ADRB1 21 46 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585188 FD On-Demand Anodyne HTR1A 16 51 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585188 FD On-Demand Anodyne SLC6A4 19 43 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880585190 FD On-Demand Anodyne ADRB1 21 46 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880585190 FD On-Demand Anodyne HTR1A 16 51 O[C@H](COc1cccc2[nH]ccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880585190 FD On-Demand Anodyne SLC6A4 19 43 O[C@@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585192 FD On-Demand Anodyne ADRB1 21 46 O[C@@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585192 FD On-Demand Anodyne HTR1A 16 51 O[C@@H](COc1cccc2[nH]ccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585192 FD On-Demand Anodyne SLC6A4 19 43 O[C@@H]1CN(C[C@@H](O)COc2cccc3[nH]ccc23)CC2(CCOCC2)C1 ZINC000880585193 FD On-Demand Anodyne ADRB1 21 46 O[C@@H]1CN(C[C@@H](O)COc2cccc3[nH]ccc23)CC2(CCOCC2)C1 ZINC000880585193 FD On-Demand Anodyne HTR1A 16 51 O[C@@H]1CN(C[C@@H](O)COc2cccc3[nH]ccc23)CC2(CCOCC2)C1 ZINC000880585193 FD On-Demand Anodyne SLC6A4 19 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(Oc2ccccc2)c1 ZINC000880585195 GG On-Demand Anodyne EPHX2 24 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(Oc2ccccc2)c1 ZINC000880585197 GG On-Demand Anodyne EPHX2 24 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585217 GD On-Demand Anodyne MTOR 61 36 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585217 GD On-Demand Anodyne EPHX2 20 47 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585217 GD On-Demand Anodyne STAT6 53 32 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585219 GD On-Demand Anodyne MTOR 61 36 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585219 GD On-Demand Anodyne EPHX2 20 47 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880585219 GD On-Demand Anodyne STAT6 53 32 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccnc1Cl ZINC000880585223 ED On-Demand Anodyne G2YM83_BOTF4 67 33 O=[N+]([O-])c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880585225 DD On-Demand Bother KCNJ1 25 53 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccnc1Cl ZINC000880585226 ED On-Demand Anodyne G2YM83_BOTF4 67 33 O=[N+]([O-])c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880585227 DD On-Demand Bother KCNJ1 25 53 CSc1cc(NC(=O)Cc2c(Br)cnn2C)ccc1C ZINC000880585306 FG On-Demand Anodyne IMDH_CRYPV 24 42 COc1cc(CN2C[C@@H](O)CC3(CCOCC3)C2)ccc1Cl ZINC000880585328 EF On-Demand Anodyne DRD4 15 40 COc1cc(CN2C[C@H](O)CC3(CCOCC3)C2)ccc1Cl ZINC000880585329 EF On-Demand Anodyne DRD4 15 40 CCOc1cc(CN2C[C@@H](O)CC3(CCOCC3)C2)ccc1[N+](=O)[O-] ZINC000880585403 FE On-Demand Bother SSTR5 56 37 CCOc1cc(CN2C[C@H](O)CC3(CCOCC3)C2)ccc1[N+](=O)[O-] ZINC000880585404 FE On-Demand Bother SSTR5 56 37 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)cc1 ZINC000880585409 FF On-Demand Anodyne EPHX2 20 41 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)Nc1ccc(Cl)cc1 ZINC000880585410 FF On-Demand Anodyne EPHX2 20 41 COC(=O)[C@@H]1CN(C(=O)c2cnc(CC3CC3)s2)C[C@H]1C1CC1 ZINC000880585506 EE On-Demand Anodyne PTR1 44 32 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC[C@@H](F)C1 ZINC000880585536 DH On-Demand Anodyne L3MBTL3 43 35 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC[C@H](F)C1 ZINC000880585538 DH On-Demand Anodyne L3MBTL3 43 35 O[C@@H]1CN(CCCOc2cccc(Cl)c2)CC2(CCOCC2)C1 ZINC000880585539 EF On-Demand Anodyne HRH3 19 45 O[C@@H]1CN(CCCOc2cccc(Cl)c2)CC2(CCOCC2)C1 ZINC000880585539 EF On-Demand Anodyne EPHX2 21 45 O[C@H]1CN(CCCOc2cccc(Cl)c2)CC2(CCOCC2)C1 ZINC000880585541 EF On-Demand Anodyne HRH3 19 45 O[C@H]1CN(CCCOc2cccc(Cl)c2)CC2(CCOCC2)C1 ZINC000880585541 EF On-Demand Anodyne EPHX2 21 45 COC(=O)[C@@H]1CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@H]1C1CC1 ZINC000880585572 FE On-Demand Anodyne SSTR1 47 35 COC(=O)[C@@H]1CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@H]1C1CC1 ZINC000880585574 FE On-Demand Anodyne SSTR1 47 35 COC(=O)c1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880585578 FD On-Demand Anodyne CASR 17 45 COC(=O)c1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880585578 FD On-Demand Anodyne EPHX2 21 44 COC(=O)c1cccc(NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880585578 FD On-Demand Anodyne HIF1A 15 44 COC(=O)c1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880585579 FD On-Demand Anodyne CASR 17 45 COC(=O)c1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880585579 FD On-Demand Anodyne EPHX2 21 44 COC(=O)c1cccc(NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880585579 FD On-Demand Anodyne HIF1A 15 44 O[C@H]1CN(Cc2ccccc2Oc2cccnc2)CC2(CCOCC2)C1 ZINC000880585582 FG On-Demand Anodyne CCR8 16 41 O[C@@H]1CN(Cc2ccccc2Oc2cccnc2)CC2(CCOCC2)C1 ZINC000880585584 FG On-Demand Anodyne CCR8 16 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)OCc1ccccc1 ZINC000880585769 DD On-Demand Anodyne SLC12A5 64 36 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)OCc1ccccc1 ZINC000880585771 DD On-Demand Anodyne SLC12A5 64 36 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H](F)C2)N1Cc1ccccc1 ZINC000880585773 ED On-Demand Anodyne PREP 107 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H](F)C2)N1Cc1ccccc1 ZINC000880585773 ED On-Demand Anodyne DPP7 24 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H](F)C2)N1Cc1ccccc1 ZINC000880585775 ED On-Demand Anodyne PREP 107 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H](F)C2)N1Cc1ccccc1 ZINC000880585775 ED On-Demand Anodyne DPP7 24 40 O[C@H](COc1cccc(C(F)(F)F)c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585781 GE On-Demand Anodyne PDS 41 35 O[C@H](COc1cccc(C(F)(F)F)c1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880585783 GE On-Demand Anodyne PDS 41 35 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880585785 GE On-Demand Anodyne PDS 41 35 O[C@@H]1CN(C[C@@H](O)COc2cccc(C(F)(F)F)c2)CC2(CCOCC2)C1 ZINC000880585787 GE On-Demand Anodyne PDS 41 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](F)C1 ZINC000880585943 DD On-Demand Anodyne POLG_HCV1 22 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](F)C1 ZINC000880585944 DD On-Demand Anodyne POLG_HCV1 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](F)C1 ZINC000880585945 DD On-Demand Anodyne POLG_HCV1 22 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](F)C1 ZINC000880585946 DD On-Demand Anodyne POLG_HCV1 22 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@H](F)C1 ZINC000880585976 EH On-Demand Anodyne RBP4 51 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@H](F)C1 ZINC000880585976 EH On-Demand Anodyne SFRP1 74 33 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@H](F)C1 ZINC000880585976 EH On-Demand Anodyne WNT3 50 30 O=C(CCCN1C[C@@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880585977 DF On-Demand Anodyne CYP2J2 58 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@@H](F)C1 ZINC000880585978 EH On-Demand Anodyne RBP4 51 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@@H](F)C1 ZINC000880585978 EH On-Demand Anodyne SFRP1 74 33 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@@H](F)C1 ZINC000880585978 EH On-Demand Anodyne WNT3 50 30 O=C(CCCN1C[C@H](O)CC2(CCOCC2)C1)c1ccccc1 ZINC000880585980 DF On-Demand Anodyne CYP2J2 58 41 CN(CCN1CCCCC1)C(=O)c1ccc(CN2CCOCC2)o1 ZINC000880586014 ED On-Demand Anodyne HRH3 26 49 Cn1c(=O)c(CN2C[C@@H](O)CC3(CCOCC3)C2)cc2ccccc21 ZINC000880586021 ED On-Demand Anodyne NPSR1 32 45 Cn1c(=O)c(CN2C[C@H](O)CC3(CCOCC3)C2)cc2ccccc21 ZINC000880586025 ED On-Demand Anodyne NPSR1 32 45 O[C@@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586114 DE On-Demand Anodyne LTA4H 22 40 O[C@@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586114 DE On-Demand Anodyne HRH3 35 47 O[C@@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586114 DE On-Demand Anodyne EPHX2 20 45 O[C@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586115 DE On-Demand Anodyne LTA4H 22 40 O[C@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586115 DE On-Demand Anodyne HRH3 35 47 O[C@H]1CN(CCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586115 DE On-Demand Anodyne EPHX2 20 45 C[C@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880586126 GE On-Demand Mild MLYCD 19 42 C[C@@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880586127 GE On-Demand Mild MLYCD 19 42 C[C@@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880586128 GE On-Demand Mild MLYCD 19 42 C[C@H](C(=O)N(CCC#N)c1ccc(F)cc1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880586129 GE On-Demand Mild MLYCD 19 42 CCN(CCNC(=O)Nc1ccc(C(=O)OC)nc1)C(C)C ZINC000880586148 DD On-Demand Anodyne DOT1L 42 32 O[C@@H]1CN(CCCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586161 DF On-Demand Anodyne HRH3 21 52 O[C@@H]1CN(CCCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586161 DF On-Demand Anodyne EPHX2 23 44 O[C@H]1CN(CCCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586162 DF On-Demand Anodyne HRH3 21 52 O[C@H]1CN(CCCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880586162 DF On-Demand Anodyne EPHX2 23 44 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CCC[C@H](F)C3)ccn2)CC1 ZINC000880586173 GF On-Demand Anodyne GPR119 47 48 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CCC[C@@H](F)C3)ccn2)CC1 ZINC000880586174 GF On-Demand Anodyne GPR119 47 48 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cnc(C3CC3)o2)CC1 ZINC000880586210 FG On-Demand Anodyne CACNA1I 45 34 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cnc(C3CC3)o2)CC1 ZINC000880586210 FG On-Demand Anodyne SIRT3 49 40 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cnc(C3CC3)o2)CC1 ZINC000880586210 FG On-Demand Anodyne SIRT2 50 40 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cnc(C3CC3)o2)CC1 ZINC000880586210 FG On-Demand Anodyne SIRT1 49 40 CC(C)(C)OC(=O)N1CCC(CCNC(=O)c2cnc(C3CC3)o2)CC1 ZINC000880586210 FG On-Demand Anodyne GPR119 54 44 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne HTR1A 54 48 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne DRD2 28 48 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne DRD4 27 42 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne HTR2A 38 48 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne DRD3 32 42 O[C@@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586299 FE On-Demand Anodyne HTR7 60 44 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne HTR1A 54 48 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne DRD2 28 48 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne DRD4 27 42 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne HTR2A 38 48 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne DRD3 32 42 O[C@H]1CN(CCCN2CCN(c3ccccc3)CC2)CC2(CCOCC2)C1 ZINC000880586300 FE On-Demand Anodyne HTR7 60 44 Cc1c(NC(=O)C[C@@H]2CCNC2=O)cnn1-c1ccc(F)cc1F ZINC000880586301 ED On-Demand Anodyne MAPK14 17 44 Cc1c(NC(=O)C[C@H]2CCNC2=O)cnn1-c1ccc(F)cc1F ZINC000880586302 ED On-Demand Anodyne MAPK14 17 44 CCC(CC)[C@H](CNC(=O)c1ccc(NC(=O)OC(C)(C)C)cc1)N1CCOCC1 ZINC000880586320 HH On-Demand Anodyne F3 43 31 CCC(CC)[C@@H](CNC(=O)c1ccc(NC(=O)OC(C)(C)C)cc1)N1CCOCC1 ZINC000880586321 HH On-Demand Anodyne F3 43 31 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCN(c2cnccn2)CC1 ZINC000880586335 GB On-Demand Anodyne MAPK1 17 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCN(c2cnccn2)CC1 ZINC000880586336 GB On-Demand Anodyne MAPK1 17 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCCOc1cccc(Cl)c1 ZINC000880586497 GD On-Demand Anodyne AVPR1B 37 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCCOc1cccc(Cl)c1 ZINC000880586498 GD On-Demand Anodyne AVPR1B 37 40 O[C@H]1CN(CCOc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586521 EG On-Demand Anodyne ALB 21 41 O[C@H]1CN(CCOc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586521 EG On-Demand Anodyne MCL1 31 41 O[C@@H]1CN(CCOc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586522 EG On-Demand Anodyne ALB 21 41 O[C@@H]1CN(CCOc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586522 EG On-Demand Anodyne MCL1 31 41 O[C@@H]1CN(CCOc2ccc(C(F)(F)F)cc2)CC2(CCOCC2)C1 ZINC000880586597 FF On-Demand Anodyne LTA4H 21 46 O[C@H]1CN(CCOc2ccc(C(F)(F)F)cc2)CC2(CCOCC2)C1 ZINC000880586598 FF On-Demand Anodyne LTA4H 21 46 O=C(c1ccc(OC(F)F)c(Br)c1)N1CCC[C@@H](F)C1 ZINC000880586603 FH On-Demand Anodyne L3MBTL3 50 40 O=C(c1ccc(OC(F)F)c(Br)c1)N1CCC[C@H](F)C1 ZINC000880586604 FH On-Demand Anodyne L3MBTL3 50 40 N#Cc1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880586624 EE On-Demand Mild HRH3 27 44 N#Cc1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880586624 EE On-Demand Mild MEN1 45 42 N#Cc1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880586625 EE On-Demand Mild HRH3 27 44 N#Cc1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880586625 EE On-Demand Mild MEN1 45 42 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@H](F)C1 ZINC000880586692 CE On-Demand Anodyne MAP3K12 30 41 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@@H](F)C1 ZINC000880586693 CE On-Demand Anodyne MAP3K12 30 41 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCc1cccnc1 ZINC000880586715 DC On-Demand Anodyne NAMPT 66 45 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCc1cccnc1 ZINC000880586716 DC On-Demand Anodyne NAMPT 66 45 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@H](F)C3)cc2)N1 ZINC000880586735 CE On-Demand Anodyne L3MBTL3 52 39 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H](F)C3)cc2)N1 ZINC000880586736 CE On-Demand Anodyne L3MBTL3 52 39 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@H](F)C3)cc2)N1 ZINC000880586737 CE On-Demand Anodyne L3MBTL3 52 39 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H](F)C3)cc2)N1 ZINC000880586738 CE On-Demand Anodyne L3MBTL3 52 39 C[C@@H](C(=O)N1CCN(c2ccccc2)CC1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880586826 GD On-Demand Anodyne ADAM10 40 44 C[C@@H](C(=O)N1CCN(c2ccccc2)CC1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880586827 GD On-Demand Anodyne ADAM10 40 44 O[C@@H]1CN(CCCc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586935 EH On-Demand Anodyne EBP 37 41 O[C@H]1CN(CCCc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880586936 EH On-Demand Anodyne EBP 37 41 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587037 GD On-Demand Anodyne ESR1 22 41 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587037 GD On-Demand Anodyne MMP13 45 39 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587037 GD On-Demand Anodyne ADAM17 17 40 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587038 GD On-Demand Anodyne ESR1 22 41 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587038 GD On-Demand Anodyne MMP13 45 39 CN(C)S(=O)(=O)c1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880587038 GD On-Demand Anodyne ADAM17 17 40 Cc1cccc(C(C)C)c1NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880587039 EF On-Demand Anodyne SOAT1 39 40 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne PRSS1 23 42 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne F10 16 42 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne FCER2 43 35 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne TRY2_BOVIN 54 37 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne CACNA1B 30 43 COC(=O)c1cccc(CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587067 CD On-Demand Anodyne NPR 42 32 O=C(c1ccc(CN2C[C@@H](O)CC3(CCOCC3)C2)cc1)N1CCCC1 ZINC000880587101 FE On-Demand Anodyne L3MBTL3 63 46 O=C(c1ccc(CN2C[C@H](O)CC3(CCOCC3)C2)cc1)N1CCCC1 ZINC000880587102 FE On-Demand Anodyne L3MBTL3 63 46 C[C@@H](NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1)c1ccc(Cl)cc1 ZINC000880587109 FE On-Demand Anodyne PRCP 15 41 C[C@@H](NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1)c1ccc(Cl)cc1 ZINC000880587110 FE On-Demand Anodyne PRCP 15 41 C[C@H](NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1)c1ccc(Cl)cc1 ZINC000880587111 FE On-Demand Anodyne PRCP 15 41 C[C@H](NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1)c1ccc(Cl)cc1 ZINC000880587112 FE On-Demand Anodyne PRCP 15 41 COc1cc2c(cc1OC)CN(C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)CC2 ZINC000880587171 GD On-Demand Anodyne SLC18A2 47 36 COc1cc2c(cc1OC)CN(C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)CC2 ZINC000880587171 GD On-Demand Anodyne ABCB1 15 48 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)NC(=O)Nc1ccccc1 ZINC000880587229 FD On-Demand Anodyne EPHX2 19 41 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)NC(=O)Nc1ccccc1 ZINC000880587230 FD On-Demand Anodyne EPHX2 19 41 COC(=O)c1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587310 CD On-Demand Anodyne CACNA1B 33 44 COC(=O)c1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587310 CD On-Demand Anodyne ACR 57 35 COc1ccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587313 CD On-Demand Anodyne MMP3 15 42 COc1ccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587313 CD On-Demand Anodyne MMP8 20 42 COc1ccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587313 CD On-Demand Anodyne MMP12 15 42 COc1ccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587313 CD On-Demand Anodyne MMP1 16 42 COc1ccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587313 CD On-Demand Anodyne AOC3 16 40 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2cccc(C#Cc3ccccn3)c2)C1 ZINC000880587331 HI On-Demand Mild GRM5 22 51 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2cccc(C#Cc3ccccn3)c2)C1 ZINC000880587331 HI On-Demand Mild GPR119 23 43 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)Nc2cccc(C#Cc3ccccn3)c2)C1 ZINC000880587333 HI On-Demand Mild GRM5 22 51 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)Nc2cccc(C#Cc3ccccn3)c2)C1 ZINC000880587333 HI On-Demand Mild GPR119 23 43 CC(=O)Nc1nc(CN(C)[C@@H](CC(C)C)C(N)=O)cs1 ZINC000880587444 CD On-Demand Anodyne AOC3 19 47 CCOC(=O)N1CCN(C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)CC1 ZINC000880587469 EC On-Demand Anodyne CHRNA3 16 40 COc1ccc(-c2nc(CN(C)[C@@H](CC(C)C)C(N)=O)cs2)cc1 ZINC000880587516 EG On-Demand Anodyne AVPR1B 21 49 Cc1c(CN(C)[C@@H](CC(C)C)C(N)=O)cccc1[N+](=O)[O-] ZINC000880587518 CE On-Demand Bother COLA 121 42 COc1ccc(-c2nc(CN(C)[C@@H](CC(C)C)C(N)=O)cs2)cc1OC ZINC000880587530 GG On-Demand Anodyne DCK 37 41 C[C@@H]1Cc2ccccc2N1C(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587597 ED On-Demand Anodyne DRD4 28 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587597 ED On-Demand Anodyne TPP2 54 34 C[C@@H]1Cc2ccccc2N1C(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587607 ED On-Demand Anodyne DRD4 28 48 C[C@@H]1Cc2ccccc2N1C(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587607 ED On-Demand Anodyne TPP2 54 34 Cc1ccccc1CCNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880587641 DD On-Demand Anodyne NPR 65 36 COc1ccc(OCCCN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587646 DE On-Demand Anodyne FDPS 15 43 Cc1ccc(CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587650 DD On-Demand Anodyne TPSAB1 15 43 O=C(NCc1ccco1)c1cccc(CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880587713 GF On-Demand Anodyne CHRM3 15 40 O=C(NCc1ccco1)c1cccc(CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880587714 GF On-Demand Anodyne CHRM3 15 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCC(Cc2ccccc2)CC1 ZINC000880587744 GE On-Demand Anodyne GRIN2B 79 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCC(Cc2ccccc2)CC1 ZINC000880587744 GE On-Demand Anodyne CCR3 28 41 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCC(Cc2ccccc2)CC1 ZINC000880587747 GE On-Demand Anodyne GRIN2B 79 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCC(Cc2ccccc2)CC1 ZINC000880587747 GE On-Demand Anodyne CCR3 28 41 O[C@@H]1CN(Cc2ccccc2)CC2(CCOCC2)C1 ZINC000880587817 CE On-Demand Anodyne SIGMAR1 51 40 O[C@H]1CN(Cc2ccccc2)CC2(CCOCC2)C1 ZINC000880587819 CE On-Demand Anodyne SIGMAR1 51 40 Cc1oc(-c2ccccc2)nc1CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587877 EG On-Demand Anodyne PPARG 52 41 Cc1oc(-c2ccccc2)nc1CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587877 EG On-Demand Anodyne PPARA 54 39 Cc1oc(-c2ccccc2)nc1CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587877 EG On-Demand Anodyne PDE8B 78 49 Cc1oc(-c2ccccc2)nc1CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587879 EG On-Demand Anodyne PPARG 52 41 Cc1oc(-c2ccccc2)nc1CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587879 EG On-Demand Anodyne PPARA 54 39 Cc1oc(-c2ccccc2)nc1CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587879 EG On-Demand Anodyne PDE8B 78 49 CC(=O)c1cccc(OC[C@@H](O)CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587897 ED On-Demand Anodyne ABCB1 17 45 CC(=O)c1cccc(OC[C@H](O)CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880587899 ED On-Demand Anodyne ABCB1 17 45 COc1ccc(CN(C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)C2CC2)cc1 ZINC000880587920 FE On-Demand Anodyne BMP1 40 35 Cc1oc(-c2ccccc2)nc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880587943 DF On-Demand Anodyne PPARG 84 46 Cc1oc(-c2ccccc2)nc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880587943 DF On-Demand Anodyne PPARA 92 46 Cc1oc(-c2ccccc2)nc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880587943 DF On-Demand Anodyne PDE8B 59 34 COc1ccc(CN(C)C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587950 ED On-Demand Anodyne CACNA1B 27 40 COc1ccc(CN(C)C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880587950 ED On-Demand Anodyne MMP1 18 41 O[C@H](COc1ccccc1F)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587974 ED On-Demand Anodyne ABCB1 42 39 O[C@H](COc1ccccc1F)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880587975 ED On-Demand Anodyne ABCB1 42 39 O[C@@H](COc1ccccc1F)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880587976 ED On-Demand Anodyne ABCB1 42 39 O[C@@H]1CN(C[C@@H](O)COc2ccccc2F)CC2(CCOCC2)C1 ZINC000880587978 ED On-Demand Anodyne ABCB1 42 39 O[C@@H]1CN(CCOCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880588032 ED On-Demand Anodyne LTA4H 20 40 O[C@H]1CN(CCOCCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880588036 ED On-Demand Anodyne LTA4H 20 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne ACE 39 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne OPRM1 58 55 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne OPRD1 51 55 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MME 110 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne ANPEP 71 43 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne TACR1 24 52 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MC4R 40 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CMA1 26 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne FCER2 112 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne TACR2 18 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne RNPEP 30 43 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne KLK3 83 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CTSB 63 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne TRY2_BOVIN 47 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne PAPA1_CARPA 67 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CYSP_TRYCR 50 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CCKAR 40 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CTSL 49 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CACNA1B 51 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne F2R 41 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne NPFFR2 56 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne TIMP3 50 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne C3AR1 36 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne HLA-A 18 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne TACR3 15 45 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MC3R 48 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MC5R 43 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CAPNS1 76 44 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP2 31 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP3 46 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP8 37 46 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne HLA-DRB1 90 45 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne REN 35 46 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne REN1 52 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne FURIN 52 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CAPN1 111 44 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP9 35 46 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne CAPN2 119 44 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne ACE2 63 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MC1R 65 39 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne LAP3 21 43 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP7 38 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne MMP1 52 47 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne FPR1 81 48 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne NPR 94 44 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne AMP1_PLAFQ 29 43 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne PSMB5 42 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne BLA1_STEMA 44 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne KISS1R 80 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne QRFPR 52 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne NPFFR1 74 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588073 ED On-Demand Anodyne GPR142 55 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne ACE 39 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne OPRM1 58 55 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne OPRD1 51 55 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MME 110 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne ANPEP 71 43 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne TACR1 24 52 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MC4R 40 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CMA1 26 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne FCER2 112 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne TACR2 18 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne RNPEP 30 43 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne KLK3 83 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CTSB 63 42 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne TRY2_BOVIN 47 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne PAPA1_CARPA 67 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CYSP_TRYCR 50 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CCKAR 40 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CTSL 49 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CACNA1B 51 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne F2R 41 42 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne NPFFR2 56 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne TIMP3 50 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne C3AR1 36 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne HLA-A 18 41 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne TACR3 15 45 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MC3R 48 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MC5R 43 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CAPNS1 76 44 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP2 31 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP3 46 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP8 37 46 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne HLA-DRB1 90 45 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne REN 35 46 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne REN1 52 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne FURIN 52 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CAPN1 111 44 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP9 35 46 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne CAPN2 119 44 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne ACE2 63 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MC1R 65 39 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne LAP3 21 43 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP7 38 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne MMP1 52 47 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne FPR1 81 48 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne NPR 94 44 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne AMP1_PLAFQ 29 43 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne PSMB5 42 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne BLA1_STEMA 44 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne KISS1R 80 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne QRFPR 52 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne NPFFR1 74 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588076 ED On-Demand Anodyne GPR142 55 34 C[C@H](C(=O)N(C)Cc1ccccc1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588081 ED On-Demand Anodyne TACR1 18 41 C[C@@H](C(=O)N(C)Cc1ccccc1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588083 ED On-Demand Anodyne TACR1 18 41 C[C@H](C(=O)N(C)Cc1ccccc1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588084 ED On-Demand Anodyne TACR1 18 41 C[C@@H](C(=O)N(C)Cc1ccccc1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588086 ED On-Demand Anodyne TACR1 18 41 CCC[C@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588148 EE On-Demand Anodyne CAPNS1 42 31 CCC[C@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588148 EE On-Demand Anodyne CAPN2 59 38 CCC[C@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588148 EE On-Demand Anodyne NPR 45 35 CCC[C@@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588151 EE On-Demand Anodyne CAPNS1 42 31 CCC[C@@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588151 EE On-Demand Anodyne CAPN2 59 38 CCC[C@@H](NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880588151 EE On-Demand Anodyne NPR 45 35 O[C@@H]1CN(Cc2csc(Nc3ccccc3)n2)CC2(CCOCC2)C1 ZINC000880588163 FG On-Demand Anodyne SPHK2 62 33 O[C@@H]1CN(Cc2csc(Nc3ccccc3)n2)CC2(CCOCC2)C1 ZINC000880588163 FG On-Demand Anodyne SPHK1 49 35 O[C@H]1CN(Cc2csc(Nc3ccccc3)n2)CC2(CCOCC2)C1 ZINC000880588166 FG On-Demand Anodyne SPHK2 62 33 O[C@H]1CN(Cc2csc(Nc3ccccc3)n2)CC2(CCOCC2)C1 ZINC000880588166 FG On-Demand Anodyne SPHK1 49 35 O[C@H]1CN(CCOC(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588174 GH On-Demand Anodyne SLC6A4 22 47 O[C@H]1CN(CCOC(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588174 GH On-Demand Anodyne SLC6A3 60 49 O[C@@H]1CN(CCOC(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588175 GH On-Demand Anodyne SLC6A4 22 47 O[C@@H]1CN(CCOC(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588175 GH On-Demand Anodyne SLC6A3 60 49 CC(=O)c1ccccc1OCCN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588215 EE On-Demand Anodyne HCN1 61 38 CC(=O)c1ccccc1OCCN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588215 EE On-Demand Anodyne HCN4 40 31 CC(=O)c1ccccc1OCCN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588216 EE On-Demand Anodyne HCN1 61 38 CC(=O)c1ccccc1OCCN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588216 EE On-Demand Anodyne HCN4 40 31 CC(=O)c1ccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588244 FD On-Demand Anodyne ABCB1 31 40 Cc1cccc(CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880588274 DD On-Demand Anodyne ANPEP 18 51 Cc1cccc(CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880588274 DD On-Demand Anodyne KISS1R 47 31 CCOc1ccccc1NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588283 ED On-Demand Anodyne HCN1 44 37 CCOc1ccccc1NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588283 ED On-Demand Anodyne HCN4 40 32 CS(=O)(=O)Nc1cc2ccccc2cc1C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880588284 II On-Demand Mild KCNK3 49 35 CS(=O)(=O)Nc1cc2ccccc2cc1C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880588284 II On-Demand Mild KCNK9 43 34 CCOc1ccccc1NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588285 ED On-Demand Anodyne HCN1 44 37 CCOc1ccccc1NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588285 ED On-Demand Anodyne HCN4 40 32 CC(=O)c1ccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588287 FD On-Demand Anodyne ABCB1 31 40 CC(=O)c1ccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588290 FD On-Demand Anodyne ABCB1 31 40 CC(=O)c1ccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588293 FD On-Demand Anodyne ABCB1 31 40 O[C@H](COc1ccc(F)cc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588369 ED On-Demand Anodyne ABCB1 19 44 O[C@H](COc1ccc(F)cc1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588371 ED On-Demand Anodyne ABCB1 19 44 O[C@@H](COc1ccc(F)cc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588373 ED On-Demand Anodyne ABCB1 19 44 O[C@@H]1CN(C[C@@H](O)COc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880588375 ED On-Demand Anodyne ABCB1 19 44 O[C@H](COc1ccc(Cl)cc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588383 GF On-Demand Anodyne CCR1 44 39 O[C@H](COc1ccc(Cl)cc1Cl)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588385 GF On-Demand Anodyne CCR1 44 39 O[C@@H](COc1ccc(Cl)cc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588387 GF On-Demand Anodyne CCR1 44 39 O[C@@H]1CN(C[C@@H](O)COc2ccc(Cl)cc2Cl)CC2(CCOCC2)C1 ZINC000880588389 GF On-Demand Anodyne CCR1 44 39 O[C@@H]1CN(Cc2nc(-c3cccc(Cl)c3)no2)CC2(CCOCC2)C1 ZINC000880588462 FF On-Demand Anodyne GRM5 16 44 O[C@H]1CN(Cc2nc(-c3cccc(Cl)c3)no2)CC2(CCOCC2)C1 ZINC000880588465 FF On-Demand Anodyne GRM5 16 44 Cc1ccccc1CN1CCC(NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)CC1 ZINC000880588478 GD On-Demand Anodyne SIGMAR1 17 45 Cc1ccccc1CN1CCC(NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)CC1 ZINC000880588478 GD On-Demand Anodyne CACNA1B 18 42 CN(Cc1ccc(F)cc1)C(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588505 FD On-Demand Anodyne TACR3 23 43 CN(Cc1ccc(F)cc1)C(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588505 FD On-Demand Anodyne WNT3A 41 34 CN(Cc1ccc(F)cc1)C(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588507 FD On-Demand Anodyne TACR3 23 43 CN(Cc1ccc(F)cc1)C(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588507 FD On-Demand Anodyne WNT3A 41 34 Cc1cccc(NC(=O)[C@H](C)N2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880588521 EE On-Demand Anodyne CCKAR 15 40 Cc1cccc(NC(=O)[C@@H](C)N2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880588523 EE On-Demand Anodyne CCKAR 15 40 Cc1cccc(NC(=O)[C@H](C)N2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880588525 EE On-Demand Anodyne CCKAR 15 40 Cc1cccc(NC(=O)[C@@H](C)N2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880588527 EE On-Demand Anodyne CCKAR 15 40 C[C@H](C(=O)Nc1ccccc1C(F)(F)F)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588533 GF On-Demand Anodyne RBP4 49 33 C[C@H](C(=O)Nc1ccccc1C(F)(F)F)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588535 GF On-Demand Anodyne RBP4 49 33 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588536 GD On-Demand Anodyne CHRM2 15 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588536 GD On-Demand Anodyne DRD4 32 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588536 GD On-Demand Anodyne SIGMAR1 53 37 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588537 GD On-Demand Anodyne CHRM2 15 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588537 GD On-Demand Anodyne DRD4 32 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N1CCN(Cc2ccccc2)CC1 ZINC000880588537 GD On-Demand Anodyne SIGMAR1 53 37 O[C@H](COc1cc(Cl)ccc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588639 GF On-Demand Anodyne CCR1 44 39 O[C@H](COc1cc(Cl)ccc1Cl)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588641 GF On-Demand Anodyne CCR1 44 39 O[C@@H](COc1cc(Cl)ccc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588643 GF On-Demand Anodyne CCR1 44 39 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)NCCCc1ccccc1 ZINC000880588645 ED On-Demand Anodyne CRTM 33 40 O[C@@H]1CN(C[C@@H](O)COc2cc(Cl)ccc2Cl)CC2(CCOCC2)C1 ZINC000880588646 GF On-Demand Anodyne CCR1 44 39 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)NCCCc1ccccc1 ZINC000880588647 ED On-Demand Anodyne CRTM 33 40 Cc1ccccc1CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588649 DD On-Demand Anodyne ANPEP 21 50 Cc1ccccc1CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588649 DD On-Demand Anodyne NPR 41 39 Cc1ccccc1CNC(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880588649 DD On-Demand Anodyne AMP1_PLAFQ 23 40 COC(=O)c1sccc1NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588709 FD On-Demand Anodyne FAS 45 46 COC(=O)c1sccc1NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588711 FD On-Demand Anodyne FAS 45 46 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne OPRM1 29 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne OPRD1 21 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne TIMP3 47 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne CAPN1 46 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne ACE2 45 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588782 FD On-Demand Anodyne PSMB8 58 45 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne OPRM1 29 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne OPRD1 21 40 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne TIMP3 47 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne CAPN1 46 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne ACE2 45 33 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588784 FD On-Demand Anodyne PSMB8 58 45 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne OPRM1 29 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne OPRD1 21 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne TIMP3 47 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne CAPN1 46 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne ACE2 45 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588785 FD On-Demand Anodyne PSMB8 58 45 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne OPRM1 29 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne OPRD1 21 40 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne TIMP3 47 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne CAPN1 46 35 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne ACE2 45 33 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588786 FD On-Demand Anodyne PSMB8 58 45 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588800 GD On-Demand Anodyne ADRB1 18 44 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588801 GD On-Demand Anodyne ADRB1 18 44 CC(=O)Nc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588802 GD On-Demand Anodyne ADRB1 18 44 CC(=O)Nc1ccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880588803 GD On-Demand Anodyne ADRB1 18 44 COc1ccc([C@H](NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)C(C)C)cc1 ZINC000880588820 GE On-Demand Anodyne EDNRB 17 41 COc1ccc([C@@H](NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)C(C)C)cc1 ZINC000880588821 GE On-Demand Anodyne EDNRB 17 41 COc1ccc([C@@H](NC(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)C(C)C)cc1 ZINC000880588822 GE On-Demand Anodyne EDNRB 17 41 COc1ccc([C@H](NC(=O)CN2C[C@H](O)CC3(CCOCC3)C2)C(C)C)cc1 ZINC000880588823 GE On-Demand Anodyne EDNRB 17 41 CC(C)c1cccc(C(C)C)c1NC(=O)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588851 GH On-Demand Anodyne SOAT1 52 40 CC(C)c1cccc(C(C)C)c1NC(=O)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588852 GH On-Demand Anodyne SOAT1 52 40 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588894 GF On-Demand Anodyne ACOX1 68 37 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588897 GF On-Demand Anodyne ACOX1 68 37 O[C@@H]1CN(C[C@@H](O)COc2ccc(Cl)c(Cl)c2)CC2(CCOCC2)C1 ZINC000880588899 GF On-Demand Anodyne ACOX1 68 37 O[C@@H](COc1ccc(Cl)c(Cl)c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588901 GF On-Demand Anodyne ACOX1 68 37 O[C@@H]1CN(CCOc2ccc(Br)cc2)CC2(CCOCC2)C1 ZINC000880588919 FF On-Demand Anodyne LTA4H 28 42 O[C@H]1CN(CCOc2ccc(Br)cc2)CC2(CCOCC2)C1 ZINC000880588921 FF On-Demand Anodyne LTA4H 28 42 O[C@@H]1CN(C(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588924 EH On-Demand Anodyne OPRL1 17 40 O[C@H]1CN(C(c2ccccc2)c2ccccc2)CC2(CCOCC2)C1 ZINC000880588925 EH On-Demand Anodyne OPRL1 17 40 O=[N+]([O-])c1cccc(CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880588939 DD On-Demand Bother CACNA1D 51 33 O=[N+]([O-])c1cccc(CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880588941 DD On-Demand Bother CACNA1D 51 33 O[C@H](COc1ccccc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588952 DD On-Demand Anodyne ABCB1 45 39 O[C@H](COc1ccccc1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588955 DD On-Demand Anodyne ABCB1 45 39 O[C@@H](COc1ccccc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588956 DD On-Demand Anodyne ABCB1 45 39 O[C@@H]1CN(C[C@@H](O)COc2ccccc2)CC2(CCOCC2)C1 ZINC000880588958 DD On-Demand Anodyne ABCB1 45 39 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588974 GF On-Demand Anodyne CCR2 26 41 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880588974 GF On-Demand Anodyne EPHX2 18 44 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588976 GF On-Demand Anodyne CCR2 26 41 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880588976 GF On-Demand Anodyne EPHX2 18 44 Cc1ccccc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880589001 BE On-Demand Anodyne ANPEP 20 42 CCOC(=O)[C@@H]1CCCCN1C(=O)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880589005 EC On-Demand Anodyne LGMN 41 36 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880589061 FD On-Demand Anodyne ACOX1 53 33 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880589061 FD On-Demand Anodyne ABCB1 38 51 CC(=O)c1cccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880589062 FD On-Demand Anodyne ACOX1 53 33 CC(=O)c1cccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)c1 ZINC000880589062 FD On-Demand Anodyne ABCB1 38 51 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880589063 FD On-Demand Anodyne ACOX1 53 33 CC(=O)c1cccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880589063 FD On-Demand Anodyne ABCB1 38 51 CC(=O)c1cccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880589064 FD On-Demand Anodyne ACOX1 53 33 CC(=O)c1cccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)c1 ZINC000880589064 FD On-Demand Anodyne ABCB1 38 51 COc1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880589111 EE On-Demand Anodyne HRH3 46 45 COc1ccc(OCCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880589111 EE On-Demand Anodyne MMP13 15 43 COc1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880589112 EE On-Demand Anodyne HRH3 46 45 COc1ccc(OCCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880589112 EE On-Demand Anodyne MMP13 15 43 O[C@H](COc1ccccc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589151 FD On-Demand Anodyne ABCB1 47 37 O[C@H](COc1ccccc1Cl)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589152 FD On-Demand Anodyne ABCB1 47 37 O[C@@H](COc1ccccc1Cl)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589153 FD On-Demand Anodyne ABCB1 47 37 O[C@@H]1CN(C[C@@H](O)COc2ccccc2Cl)CC2(CCOCC2)C1 ZINC000880589154 FD On-Demand Anodyne ABCB1 47 37 O[C@H](COc1ccc2ccccc2c1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589155 FE On-Demand Anodyne ACOX1 78 36 O[C@H](COc1ccc2ccccc2c1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589155 FE On-Demand Anodyne ABCB1 32 42 O[C@H](COc1ccc2ccccc2c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589156 FE On-Demand Anodyne ACOX1 78 36 O[C@H](COc1ccc2ccccc2c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589156 FE On-Demand Anodyne ABCB1 32 42 O[C@@H]1CN(C[C@@H](O)COc2ccc3ccccc3c2)CC2(CCOCC2)C1 ZINC000880589157 FE On-Demand Anodyne ACOX1 78 36 O[C@@H]1CN(C[C@@H](O)COc2ccc3ccccc3c2)CC2(CCOCC2)C1 ZINC000880589157 FE On-Demand Anodyne ABCB1 32 42 O[C@@H](COc1ccc2ccccc2c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589158 FE On-Demand Anodyne ACOX1 78 36 O[C@@H](COc1ccc2ccccc2c1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589158 FE On-Demand Anodyne ABCB1 32 42 O[C@@H]1CN(CCOc2cccc(F)c2)CC2(CCOCC2)C1 ZINC000880589201 DE On-Demand Anodyne EPHX2 15 40 O[C@H]1CN(CCOc2cccc(F)c2)CC2(CCOCC2)C1 ZINC000880589202 DE On-Demand Anodyne EPHX2 15 40 O[C@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589222 FE On-Demand Anodyne ADRB2 17 46 O[C@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589222 FE On-Demand Anodyne ADRB1 15 43 O[C@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589222 FE On-Demand Anodyne ABCB1 49 45 O[C@H](COc1cccc2ccccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589223 FE On-Demand Anodyne ADRB2 17 46 O[C@H](COc1cccc2ccccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589223 FE On-Demand Anodyne ADRB1 15 43 O[C@H](COc1cccc2ccccc12)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880589223 FE On-Demand Anodyne ABCB1 49 45 O[C@@H]1CN(C[C@@H](O)COc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880589224 FE On-Demand Anodyne ADRB2 17 46 O[C@@H]1CN(C[C@@H](O)COc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880589224 FE On-Demand Anodyne ADRB1 15 43 O[C@@H]1CN(C[C@@H](O)COc2cccc3ccccc23)CC2(CCOCC2)C1 ZINC000880589224 FE On-Demand Anodyne ABCB1 49 45 O[C@@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589225 FE On-Demand Anodyne ADRB2 17 46 O[C@@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589225 FE On-Demand Anodyne ADRB1 15 43 O[C@@H](COc1cccc2ccccc12)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880589225 FE On-Demand Anodyne ABCB1 49 45 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880589227 IJ On-Demand Mild HDAC1 22 42 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880589227 IJ On-Demand Mild DDR1 51 37 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880589227 IJ On-Demand Mild KCNK3 87 40 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000880589227 IJ On-Demand Mild KCNK9 52 33 O[C@@H]1CN(CCCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880589238 DE On-Demand Anodyne HRH3 37 45 O[C@@H]1CN(CCCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880589238 DE On-Demand Anodyne EPHX2 18 42 O[C@H]1CN(CCCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880589239 DE On-Demand Anodyne HRH3 37 45 O[C@H]1CN(CCCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880589239 DE On-Demand Anodyne EPHX2 18 42 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880589268 FF On-Demand Anodyne CCR2 51 39 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880589268 FF On-Demand Anodyne EPHX2 28 44 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880589269 FF On-Demand Anodyne CCR2 51 39 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(C(F)(F)F)c1 ZINC000880589269 FF On-Demand Anodyne EPHX2 28 44 O[C@@H]1CN(CCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880589324 CE On-Demand Anodyne SIGMAR1 33 43 O[C@H]1CN(CCCc2ccccc2)CC2(CCOCC2)C1 ZINC000880589325 CE On-Demand Anodyne SIGMAR1 33 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880589384 EE On-Demand Anodyne EPHX2 20 43 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880589384 EE On-Demand Anodyne MCHR1 23 45 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880589385 EE On-Demand Anodyne EPHX2 20 43 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)Nc1cccc(Cl)c1 ZINC000880589385 EE On-Demand Anodyne MCHR1 23 45 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)N2CCN(c3cc(C#N)ccn3)CC2)c1 ZINC000880589394 JG On-Demand Mild SLC6A9 24 43 N#CCCn1cc(C(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c2ccccc21 ZINC000880589424 GF On-Demand Mild CNR1 15 46 N#CCCn1cc(C(=O)CN2C[C@@H](O)CC3(CCOCC3)C2)c2ccccc21 ZINC000880589424 GF On-Demand Mild CNR2 22 46 N#CCCn1cc(C(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c2ccccc21 ZINC000880589425 GF On-Demand Mild CNR1 15 46 N#CCCn1cc(C(=O)CN2C[C@H](O)CC3(CCOCC3)C2)c2ccccc21 ZINC000880589425 GF On-Demand Mild CNR2 22 46 O[C@@H]1CN(CCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589440 EF On-Demand Anodyne LTA4H 28 42 O[C@H]1CN(CCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589441 EF On-Demand Anodyne LTA4H 28 42 O[C@@H]1CN(CCCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589541 EF On-Demand Anodyne HRH3 34 45 O[C@@H]1CN(CCCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589541 EF On-Demand Anodyne EPHX2 16 50 O[C@H]1CN(CCCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589542 EF On-Demand Anodyne HRH3 34 45 O[C@H]1CN(CCCOc2ccc(Cl)cc2)CC2(CCOCC2)C1 ZINC000880589542 EF On-Demand Anodyne EPHX2 16 50 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589593 FE On-Demand Anodyne BDKRB1 47 42 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589593 FE On-Demand Anodyne XIAP 20 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589593 FE On-Demand Anodyne BIRC3 44 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589595 FE On-Demand Anodyne BDKRB1 47 42 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589595 FE On-Demand Anodyne XIAP 20 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589595 FE On-Demand Anodyne BIRC3 44 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589597 FE On-Demand Anodyne BDKRB1 47 42 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589597 FE On-Demand Anodyne XIAP 20 40 O=C(CN1C[C@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880589597 FE On-Demand Anodyne BIRC3 44 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589599 FE On-Demand Anodyne BDKRB1 47 42 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589599 FE On-Demand Anodyne XIAP 20 40 O=C(CN1C[C@@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880589599 FE On-Demand Anodyne BIRC3 44 40 CC(=O)Oc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880589676 CD On-Demand Anodyne CACNA1B 38 44 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1Cl ZINC000880589707 CF On-Demand Anodyne PDE6A 42 33 CS(=O)(=O)c1ccnc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880589718 GE On-Demand Anodyne SLC6A9 39 48 CS(=O)(=O)c1ccnc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880589718 GE On-Demand Anodyne FAAH 22 44 CCN(C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1nc2ccccc2s1 ZINC000880589791 FE On-Demand Anodyne TMPRSS6 41 35 CS(=O)(=O)c1ccnc(NC(=O)NCCCCC2CC2)c1 ZINC000880589795 DE On-Demand Anodyne CCR3 17 41 O[C@@H]1CN(CCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880589840 CD On-Demand Anodyne LTA4H 42 45 O[C@H]1CN(CCOc2ccccc2)CC2(CCOCC2)C1 ZINC000880589846 CD On-Demand Anodyne LTA4H 42 45 CC[C@@](C)(NC(=O)Nc1ccc(C(=O)OC)nc1)c1ccccc1 ZINC000880589849 EG On-Demand Anodyne IMDH_CRYPV 42 34 O=C(COC1CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880589852 DF On-Demand Anodyne TBXAS1 40 43 O=C(COC1CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880589852 DF On-Demand Anodyne CHRNA7 46 41 O=C(COC1CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880589852 DF On-Demand Anodyne CES1 40 37 O=C(COC1CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880589852 DF On-Demand Anodyne ACHP_LYMST 29 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(F)(F)CC2)c1 ZINC000880589937 DD On-Demand Anodyne NPY5R 30 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)c1 ZINC000880589952 GE On-Demand Anodyne EPHX2 19 48 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)c1 ZINC000880589954 GE On-Demand Anodyne EPHX2 19 48 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)c1 ZINC000880589990 GE On-Demand Anodyne EPHX2 15 42 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)c1 ZINC000880589992 GE On-Demand Anodyne EPHX2 15 42 CS(=O)(=O)c1ccnc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)c1 ZINC000880590009 FF On-Demand Anodyne EPHX2 15 40 CS(=O)(=O)c1ccnc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)c1 ZINC000880590009 FF On-Demand Anodyne SMO 24 40 O=C([C@H]1CCc2nncn2CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880590076 GF On-Demand Anodyne CHRNA7 40 38 O=C([C@@H]1CCc2nncn2CC1)N(CCc1ccccc1)Cc1cccnc1 ZINC000880590077 GF On-Demand Anodyne CHRNA7 40 38 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)c1 ZINC000880590090 GF On-Demand Anodyne CASR 23 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)c1 ZINC000880590091 GF On-Demand Anodyne CASR 23 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)c1 ZINC000880590092 GF On-Demand Anodyne CASR 23 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)c1 ZINC000880590093 GF On-Demand Anodyne CASR 23 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(OC[C@@H]3CCCO3)CC2)c1 ZINC000880590105 GD On-Demand Anodyne GPR119 45 37 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(OC[C@H]3CCCO3)CC2)c1 ZINC000880590108 GD On-Demand Anodyne GPR119 45 37 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)c1 ZINC000880590136 FF On-Demand Anodyne OXTR 45 34 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)c1 ZINC000880590136 FF On-Demand Anodyne NPY5R 40 49 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)c1 ZINC000880590139 FF On-Demand Anodyne OXTR 45 34 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)c1 ZINC000880590139 FF On-Demand Anodyne NPY5R 40 49 CCOc1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590218 EE On-Demand Anodyne LTA4H 32 41 CCOc1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590220 EE On-Demand Anodyne LTA4H 32 41 CCOc1ccccc1NC(=O)[C@@H](C)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880590221 FE On-Demand Anodyne HCN1 49 41 CCOc1ccccc1NC(=O)[C@@H](C)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880590221 FE On-Demand Anodyne HCN4 40 33 CCOc1ccccc1NC(=O)[C@H](C)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880590222 FE On-Demand Anodyne HCN1 49 41 CCOc1ccccc1NC(=O)[C@H](C)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880590222 FE On-Demand Anodyne HCN4 40 33 CCOc1ccccc1NC(=O)[C@@H](C)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590225 FE On-Demand Anodyne HCN1 49 41 CCOc1ccccc1NC(=O)[C@@H](C)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590225 FE On-Demand Anodyne HCN4 40 33 CCOc1ccccc1NC(=O)[C@H](C)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590227 FE On-Demand Anodyne HCN1 49 41 CCOc1ccccc1NC(=O)[C@H](C)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590227 FE On-Demand Anodyne HCN4 40 33 O[C@@H]1CN(C[C@@H](O)COc2ccc(-c3ccccc3)cc2)CC2(CCOCC2)C1 ZINC000880590247 GF On-Demand Anodyne ACOX1 52 36 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590249 GF On-Demand Anodyne ACOX1 52 36 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880590250 GF On-Demand Anodyne ACOX1 52 36 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1C[C@H](O)CC2(CCOCC2)C1 ZINC000880590251 GF On-Demand Anodyne ACOX1 52 36 COc1ccc(OCCN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590253 DD On-Demand Anodyne LTA4H 32 41 COc1ccc(OCCN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590254 DD On-Demand Anodyne LTA4H 32 41 COc1ccc2c(CN(C)[C@@H](CC(C)C)C(N)=O)cc(=O)oc2c1 ZINC000880590256 EE On-Demand Anodyne MAOA 48 38 COc1ccc2c(CN(C)[C@@H](CC(C)C)C(N)=O)cc(=O)oc2c1 ZINC000880590256 EE On-Demand Anodyne MAOB 39 44 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(F)CC2)c1 ZINC000880590258 DD On-Demand Anodyne TYK2 41 31 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(F)CC2)c1 ZINC000880590258 DD On-Demand Anodyne GPR119 57 38 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880590299 FE On-Demand Anodyne HTR7 15 51 O=C(CCN1C[C@@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880590300 FE On-Demand Anodyne HTR7 15 51 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)N[C@H]1CCCc2ccccc21 ZINC000880590301 FE On-Demand Anodyne HTR7 15 51 O=C(CCN1C[C@H](O)CC2(CCOCC2)C1)N[C@@H]1CCCc2ccccc21 ZINC000880590302 FE On-Demand Anodyne HTR7 15 51 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C1 ZINC000880590327 ED On-Demand Anodyne HCRTR1 17 50 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C1 ZINC000880590327 ED On-Demand Anodyne HCRTR2 31 50 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne BMP1 57 39 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne CACNA1B 39 48 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne MMP3 18 46 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne MMP8 17 46 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne MMP9 18 46 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne MMP12 19 46 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne MMP1 27 46 COc1ccc(CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590341 CE On-Demand Anodyne AOC3 17 45 COc1cccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880590434 CD On-Demand Anodyne MTNR1A 27 45 COc1cccc(OCCN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880590434 CD On-Demand Anodyne MTNR1B 29 45 O[C@@H]1CN(CCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880590467 DE On-Demand Anodyne LTA4H 32 42 O[C@H]1CN(CCOc2ccc(F)cc2)CC2(CCOCC2)C1 ZINC000880590468 DE On-Demand Anodyne LTA4H 32 42 Cc1ccc(OC[C@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590487 ED On-Demand Anodyne ACOX1 68 32 Cc1ccc(OC[C@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590488 ED On-Demand Anodyne ACOX1 68 32 Cc1ccc(OC[C@@H](O)CN2C[C@@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590489 ED On-Demand Anodyne ACOX1 68 32 Cc1ccc(OC[C@@H](O)CN2C[C@H](O)CC3(CCOCC3)C2)cc1 ZINC000880590490 ED On-Demand Anodyne ACOX1 68 32 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@](F)(c3ccccc3)C2)c1 ZINC000880590592 GF On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@](F)(c3ccccc3)C2)c1 ZINC000880590593 GF On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)c1ccnc(NC(=O)NCCC2CCC2)c1 ZINC000880590598 CD On-Demand Anodyne PRMT3 17 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(C3CCCCC3)CC2)c1 ZINC000880590645 FG On-Demand Anodyne EPHX2 22 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(C3CCCCC3)CC2)c1 ZINC000880590645 FG On-Demand Anodyne GPR119 38 40 O=C(CN1CCCCS1(=O)=O)N(CCc1ccccc1)Cc1ccncc1 ZINC000880590654 GE On-Demand Anodyne MRGPRX1 31 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880590671 GD On-Demand Anodyne FAAH 24 44 O=C(COC1CC1)N(CCc1ccccc1)Cc1ccncc1 ZINC000880590672 DF On-Demand Anodyne CES1 43 36 CO[C@@H](CN(C)[C@@H](CC(C)C)C(N)=O)c1ccccc1 ZINC000880590681 CE On-Demand Anodyne NPR 64 34 COc1ncccc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880590699 CD On-Demand Anodyne PLM1_PLAFA 42 31 COc1ncccc1CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880590699 CD On-Demand Anodyne NPR 48 32 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)c1 ZINC000880590716 FE On-Demand Anodyne EPHX2 16 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)c1 ZINC000880590716 FE On-Demand Anodyne GPR119 65 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)c1 ZINC000880590717 FE On-Demand Anodyne EPHX2 16 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)c1 ZINC000880590717 FE On-Demand Anodyne GPR119 65 41 CC(=O)c1cccc(NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880590758 DD On-Demand Anodyne KCNK3 41 34 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA2 23 50 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA6 19 43 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA1 18 50 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA7 21 43 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA13 38 43 CCC(CC)[C@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590771 HD On-Demand Anodyne CA4 18 50 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA2 23 50 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA6 19 43 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA1 18 50 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA7 21 43 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA13 38 43 CCC(CC)[C@@H](CNC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)N1CCOCC1 ZINC000880590772 HD On-Demand Anodyne CA4 18 50 CCOc1ccc([C@@H]2CCCN2C(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880590903 GF On-Demand Anodyne CPT1A 45 34 CN1CCN(C2CCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)CC1 ZINC000880590938 GC On-Demand Anodyne HTR1F 51 31 CN1CCN(C2CCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)CC1 ZINC000880590938 GC On-Demand Anodyne L3MBTL3 62 42 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne PRSS2 55 31 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne MAPK14 22 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne CCR3 20 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne MLNR 38 44 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne MAPK10 18 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne EPHX2 28 44 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880590952 GE On-Demand Anodyne GPR119 74 43 C#CCC1(O)CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)CC1 ZINC000880591014 EC On-Demand Mild S1PR2 25 40 C[C@@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@@H]1c1ccccc1 ZINC000880591015 FG On-Demand Anodyne EPHX2 22 42 C[C@@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@@H]1c1ccccc1 ZINC000880591015 FG On-Demand Anodyne SMO 27 42 C[C@@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@H]1c1ccccc1 ZINC000880591016 FG On-Demand Anodyne EPHX2 22 42 C[C@@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@H]1c1ccccc1 ZINC000880591016 FG On-Demand Anodyne SMO 27 42 C[C@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@H]1c1ccccc1 ZINC000880591017 FG On-Demand Anodyne EPHX2 22 42 C[C@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@H]1c1ccccc1 ZINC000880591017 FG On-Demand Anodyne SMO 27 42 C[C@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@@H]1c1ccccc1 ZINC000880591018 FG On-Demand Anodyne EPHX2 22 42 C[C@H]1CCN(C(=O)Nc2cc(S(C)(=O)=O)ccn2)C[C@@H]1c1ccccc1 ZINC000880591018 FG On-Demand Anodyne SMO 27 42 COc1ccccc1N1CC[C@@H](N(C)[C@@H](CC(C)C)C(N)=O)C1=O ZINC000880591041 ED On-Demand Anodyne HTR1A 45 38 COc1ccccc1N1CC[C@H](N(C)[C@@H](CC(C)C)C(N)=O)C1=O ZINC000880591042 ED On-Demand Anodyne HTR1A 45 38 CC(=O)c1ccc(NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880591088 DD On-Demand Anodyne F3 81 36 CC(=O)c1ccc(NC(=O)CN(C)[C@@H](CC(C)C)C(N)=O)cc1 ZINC000880591088 DD On-Demand Anodyne ACR 48 35 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880591134 GG On-Demand Anodyne EPHX2 15 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880591149 GG On-Demand Anodyne HTR1F 47 34 CCCCNC(=O)CCN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591152 CD On-Demand Anodyne NOD1 52 37 CC(C)(C)OC(=O)N1CC2(CCC2)[C@H]1C1CCN(Cc2ncccn2)CC1 ZINC000880591196 FG On-Demand Anodyne GPR119 15 43 CC(C)(C)OC(=O)N1CC2(CCC2)[C@@H]1C1CCN(Cc2ncccn2)CC1 ZINC000880591197 FG On-Demand Anodyne GPR119 15 43 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)c1 ZINC000880591209 GE On-Demand Anodyne EPHX2 18 50 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)c1 ZINC000880591209 GE On-Demand Anodyne TRPM8 18 46 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)c1 ZINC000880591210 GE On-Demand Anodyne EPHX2 18 50 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)c1 ZINC000880591210 GE On-Demand Anodyne TRPM8 18 46 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne MME 40 42 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne FCER2 55 38 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne RNPEP 29 43 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne CACNA1B 42 40 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne CAPNS1 65 38 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne HLA-DRB1 59 36 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne CAPN1 62 38 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne CAPN2 70 40 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne MMP1 20 45 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne FPR1 58 41 CO[C@@H](Cc1ccccc1)CN(C)[C@@H](CC(C)C)C(N)=O ZINC000880591234 CE On-Demand Anodyne NPR 83 39 O=C(CCc1cn[nH]c1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591304 FG On-Demand Anodyne SIGMAR1 57 40 O=C(CCc1cn[nH]c1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591304 FG On-Demand Anodyne CCR8 48 46 CS(=O)(=O)c1ccnc(NC(=O)N2CCC3(CCCC3)CC2)c1 ZINC000880591322 EF On-Demand Anodyne NPY5R 27 40 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCCCC2)C1 ZINC000880591369 EE On-Demand Bother SLC6A9 24 56 COCC1CN(C(=O)c2cc3ccccc3oc2=O)C1 ZINC000880591371 CD On-Demand Anodyne MAOB 16 49 COCC1CN(C(=O)COc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880591372 DD On-Demand Anodyne MAOA 77 56 COCC1CN(C(=O)COc2ccc3c(C)cc(=O)oc3c2)C1 ZINC000880591372 DD On-Demand Anodyne MAOB 53 56 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880591407 FG On-Demand Anodyne CPT1A 77 42 CS(=O)(=O)c1ccnc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880591409 FG On-Demand Anodyne CPT1A 77 42 COCC1CN(C(=O)Cc2csc(-c3ccccn3)n2)C1 ZINC000880591410 DD On-Demand Anodyne CPT1A 18 46 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCCCC3)ccc2Cl)C1 ZINC000880591433 GE On-Demand Anodyne CASP7 44 36 COCC1CN(C(=O)COc2cccc(Br)c2)C1 ZINC000880591462 DD On-Demand Anodyne CPT1A 56 36 CS(=O)(=O)c1ccnc(NC(=O)N2CCN(c3cccc(F)n3)CC2)c1 ZINC000880591489 GD On-Demand Anodyne FAAH 23 42 COCC1CN(C(=O)c2cc(-c3ccccn3)nc3ccccc23)C1 ZINC000880591582 EG On-Demand Anodyne METAP1 50 44 CCCCCCCCNC(=O)Nc1cc(S(C)(=O)=O)ccn1 ZINC000880591583 EF On-Demand Mild ASAH1 65 33 COCC1CN(C(=O)c2oc3ccc(OC)cc3c2C)C1 ZINC000880591584 CE On-Demand Anodyne MTNR1A 46 40 COCC1CN(C(=O)c2oc3ccc(OC)cc3c2C)C1 ZINC000880591584 CE On-Demand Anodyne MTNR1B 35 40 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)c1 ZINC000880591591 GD On-Demand Anodyne S1PR2 24 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)c1 ZINC000880591592 GD On-Demand Anodyne S1PR2 24 41 COCC1CN(C(=O)[C@@H]2Cc3ccccc3CN2C(=O)c2ccccc2)C1 ZINC000880591608 FE On-Demand Anodyne PREP 52 48 COCC1CN(C(=O)[C@@H]2Cc3ccccc3CN2C(=O)c2ccccc2)C1 ZINC000880591608 FE On-Demand Anodyne CFTR 75 42 COCC1CN(C(=O)[C@@H]2Cc3ccccc3CN2C(=O)c2ccccc2)C1 ZINC000880591608 FE On-Demand Anodyne ADAM9 62 37 NC(=O)C[C@H](NC(=O)c1ccccc1Cl)C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880591622 IF On-Demand Mild GRM4 45 38 NC(=O)C[C@H](NC(=O)c1ccccc1Cl)C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880591622 IF On-Demand Mild NR2E3 53 36 NC(=O)C[C@@H](NC(=O)c1ccccc1Cl)C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880591623 IF On-Demand Mild GRM4 45 38 NC(=O)C[C@@H](NC(=O)c1ccccc1Cl)C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880591623 IF On-Demand Mild NR2E3 53 36 COCC1CN(C(=O)[C@H](CCSC)NC(=O)COc2ccccc2)C1 ZINC000880591633 FD On-Demand Anodyne P2RY12 150 40 COCC1CN(C(=O)[C@@H](CCSC)NC(=O)COc2ccccc2)C1 ZINC000880591635 FD On-Demand Anodyne P2RY12 150 40 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne CCKAR 49 35 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne PRS 59 46 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne ACACB 15 45 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne TACR3 24 47 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne MT-CO2 53 46 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3ccccc23)C1 ZINC000880591643 EH On-Demand Anodyne VCP 35 41 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)c3cnc4cc[nH]c4c3)CC2)C1 ZINC000880591656 FG On-Demand Anodyne ACACA 46 40 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)c3cnc4cc[nH]c4c3)CC2)C1 ZINC000880591656 FG On-Demand Anodyne ACACB 42 40 N#Cc1ccnc(N2CCN(C(=O)c3cc(Cl)ccc3[N+](=O)[O-])CC2)c1 ZINC000880591680 FE On-Demand Mild SLC6A9 20 43 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)C1 ZINC000880591683 GD On-Demand Anodyne CASP3 28 41 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1CC(=O)NCc1cccnc1 ZINC000880591685 EG On-Demand Anodyne CHRNA7 40 37 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1CC(=O)NCc1cccnc1 ZINC000880591685 EG On-Demand Anodyne NAMPT 82 46 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne CHRM2 20 73 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne DRD2 17 44 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne DRD4 36 42 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne OPRD1 15 41 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne CHRM3 18 73 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne SIGMAR1 83 48 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne CCR5 22 49 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne NPFFR2 35 40 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne FAAH 22 41 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne CCR8 62 56 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne NPFFR1 46 40 O=C(c1c(O)cccc1O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591695 GH On-Demand Anodyne PA 17 40 N#Cc1ccccc1/C=C\C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880591879 EI On-Demand Mild GRM5 16 40 COCC1CN(C(=O)c2cc(-c3ccc(OC)cc3)nc3ccccc23)C1 ZINC000880591894 FH On-Demand Anodyne PRS 48 45 COCC1CN(C(=O)c2cc(-c3ccc(OC)cc3)nc3ccccc23)C1 ZINC000880591894 FH On-Demand Anodyne TACR3 27 48 COCC1CN(C(=O)c2cc(-c3ccc(OC)cc3)nc3ccccc23)C1 ZINC000880591894 FH On-Demand Anodyne LUCI_PHOPY 18 53 COCC1CN(C(=O)c2cc(-c3ccc(OC)cc3)nc3ccccc23)C1 ZINC000880591894 FH On-Demand Anodyne MT-CO2 52 44 COCC1CN(C(=O)c2cc(-c3ccc(OC)cc3)nc3ccccc23)C1 ZINC000880591894 FH On-Demand Anodyne VCP 27 42 COCC1CN(C(=O)c2cc(S(=O)(=O)N(C)C)ccc2N2CCCCC2)C1 ZINC000880591897 GD On-Demand Anodyne SLC6A9 30 48 COCC1CN(C(=O)c2ccc(COc3ccc4c(C)cc(=O)oc4c3)cc2)C1 ZINC000880591898 GG On-Demand Anodyne CYP11B1 16 41 COCC1CN(C(=O)c2ccc(COc3ccc4c(C)cc(=O)oc4c3)cc2)C1 ZINC000880591898 GG On-Demand Anodyne MAOA 64 46 COCC1CN(C(=O)c2ccc(COc3ccc4c(C)cc(=O)oc4c3)cc2)C1 ZINC000880591898 GG On-Demand Anodyne MAOB 65 56 COCC1CN(C(=O)c2cccc(-n3cnnn3)c2)C1 ZINC000880591901 CC On-Demand Anodyne KCNJ1 47 35 CCCOc1ccc(OCC(=O)N2CC(COC)C2)cc1 ZINC000880591907 CD On-Demand Anodyne PLA2G4B 86 37 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)c1 ZINC000880591916 GD On-Demand Anodyne SFRP1 45 32 CS(=O)(=O)c1ccnc(NC(=O)NCCCCCCCN2CCCC2)c1 ZINC000880591924 GF On-Demand Anodyne DRD3 54 37 CS(=O)(=O)c1ccnc(NC(=O)NCCCCCCCN2CCCC2)c1 ZINC000880591924 GF On-Demand Anodyne FGFR1 23 41 CS(=O)(=O)c1ccnc(NC(=O)NCCCCCCCN2CCCC2)c1 ZINC000880591924 GF On-Demand Anodyne CCR3 27 46 CS(=O)(=O)c1ccnc(NC(=O)NCCCCCCCN2CCCC2)c1 ZINC000880591924 GF On-Demand Anodyne CHRNA7 22 48 CS(=O)(=O)c1ccnc(NC(=O)NCCCCCCCN2CCCC2)c1 ZINC000880591924 GF On-Demand Anodyne HNMT 67 38 COCC1CN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880591925 CF On-Demand Anodyne EBP 15 42 COCC1CN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880591926 CF On-Demand Anodyne EBP 15 42 CNc1ncc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)s1 ZINC000880591927 GH On-Demand Anodyne ACHE 19 40 CNc1ncc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)s1 ZINC000880591927 GH On-Demand Anodyne SIGMAR1 51 39 CNc1ncc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)s1 ZINC000880591927 GH On-Demand Anodyne CCR8 52 46 CNc1ncc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)s1 ZINC000880591927 GH On-Demand Anodyne MGEA5 34 43 CNc1ncc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)s1 ZINC000880591927 GH On-Demand Anodyne NPFFR1 41 36 COCC1CN(C(=O)C(O)(c2ccccc2)c2ccccc2)C1 ZINC000880591932 DE On-Demand Anodyne AMY2 54 31 COCC1CN(C(=O)c2cc(=O)c3ccccc3o2)C1 ZINC000880591935 CD On-Demand Anodyne TNKS 27 42 COCC1CN(C(=O)c2csc(NC3CCCCC3)n2)C1 ZINC000880591949 DF On-Demand Anodyne TRPC6 56 42 COCC1CN(C(=O)c2csc(NC3CCCCC3)n2)C1 ZINC000880591949 DF On-Demand Anodyne TRPC3 49 42 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne CHRM2 23 60 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne DRD2 21 40 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne DRD4 51 41 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne ACHE 42 41 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne DRD3 15 40 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne CHRM3 23 60 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne SIGMAR1 92 50 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne TIMP3 74 34 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne MCHR2 65 35 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne CCR8 57 50 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne NPFFR1 42 37 O=C(COC1CC1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880591950 EG On-Demand Anodyne PA 21 40 COCC1CN(C(=O)COc2ccc(Cl)cc2Cl)C1 ZINC000880591952 DE On-Demand Anodyne CCR1 19 41 COCC1CN(C(=O)COc2ccc(Cl)cc2Cl)C1 ZINC000880591952 DE On-Demand Anodyne ALPL 43 36 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccsc1 ZINC000880591955 HK On-Demand Mild GRM4 58 41 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccsc1 ZINC000880591955 HK On-Demand Mild NR1H4 15 48 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccsc1 ZINC000880591955 HK On-Demand Mild KCNK3 88 50 O=C(Nc1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1)c1ccsc1 ZINC000880591955 HK On-Demand Mild KCNK9 63 34 COCC1CN(C(=O)c2ccc(Cl)c(S(=O)(=O)N3CCCC3)c2)C1 ZINC000880591961 FD On-Demand Anodyne CNR2 15 63 COCC1CN(C(=O)c2ccc(Cl)c(S(=O)(=O)N3CCCC3)c2)C1 ZINC000880591961 FD On-Demand Anodyne CACNA1I 42 34 COCC1CN(C(=O)c2ccc(Cl)c(S(=O)(=O)N3CCCC3)c2)C1 ZINC000880591961 FD On-Demand Anodyne L3MBTL3 52 38 COCC1CN(C(=O)COc2ccc3ccc(=O)oc3c2)C1 ZINC000880591968 DD On-Demand Anodyne MAOA 33 42 COCC1CN(C(=O)COc2ccc3ccc(=O)oc3c2)C1 ZINC000880591968 DD On-Demand Anodyne MAOB 22 44 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild DRD4 18 41 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild ACHE 20 41 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild SIGMAR1 62 44 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild MCHR2 43 31 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild CCR8 45 45 C#CCC(CC#C)C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592036 FH On-Demand Mild NPFFR1 42 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880592101 DD On-Demand Anodyne CTSK 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880592103 DD On-Demand Anodyne CTSK 15 48 COCC1CN(C(=O)COc2ccccc2-c2ccccc2)C1 ZINC000880592124 DF On-Demand Anodyne PTGIR 45 35 COCC1CN(C(=O)COc2ccccc2-c2ccccc2)C1 ZINC000880592124 DF On-Demand Anodyne PLA2G1B 60 38 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne ACE 43 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CELA1 32 43 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne ELANE 58 53 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne MME 32 40 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CMA1 24 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTRA_BOVIN 56 34 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CASP3 28 48 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne BMP1 23 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne KLK3 81 38 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTSB 76 59 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne PAPA1_CARPA 83 43 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CYSP_TRYCR 56 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTSG 41 32 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTSK 59 59 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTSL 51 50 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CCR1 37 56 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne PGA 24 46 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne PREP 17 45 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CAPNS1 69 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CELA2A 41 32 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne MMP11 52 32 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTSS 28 50 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CAPN1 92 55 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CASP1 35 48 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CTRC 20 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CAPN2 142 49 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CASP6 16 48 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CASP9 42 48 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne TGM2 33 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne NPR 74 39 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne CASP10 38 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne PSMB5 47 40 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C1 ZINC000880592127 EE On-Demand Anodyne Q6PRC7_IXORI 41 33 COCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880592131 FD On-Demand Anodyne CELA1 19 43 COCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880592131 FD On-Demand Anodyne PREP 47 47 COCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880592131 FD On-Demand Anodyne SLC12A5 54 35 COCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880592131 FD On-Demand Anodyne Q9NAW4_PLAFA 25 40 COCC1CN(C(=O)[C@@H]2CC(=O)N(C3CCCC3)C2)C1 ZINC000880592135 CC On-Demand Anodyne INHA 19 44 COCC1CN(C(=O)[C@H]2CC(=O)N(C3CCCC3)C2)C1 ZINC000880592137 CC On-Demand Anodyne INHA 19 44 O=C1NCC[C@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592158 FE On-Demand Anodyne CHRM2 16 54 O=C1NCC[C@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592158 FE On-Demand Anodyne ACHE 35 42 O=C1NCC[C@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592158 FE On-Demand Anodyne CHRM3 15 54 O=C1NCC[C@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592158 FE On-Demand Anodyne SIGMAR1 65 40 O=C1NCC[C@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592158 FE On-Demand Anodyne CCR8 42 42 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592160 FE On-Demand Anodyne CHRM2 16 54 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592160 FE On-Demand Anodyne ACHE 35 42 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592160 FE On-Demand Anodyne CHRM3 15 54 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592160 FE On-Demand Anodyne SIGMAR1 65 40 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592160 FE On-Demand Anodyne CCR8 42 42 COCC1CN(C(=O)c2cc(-c3ccncc3)nc3ccccc23)C1 ZINC000880592178 EG On-Demand Anodyne PRS 31 42 COCC1CN(C(=O)c2cc(-c3ccncc3)nc3ccccc23)C1 ZINC000880592178 EG On-Demand Anodyne TACR3 22 45 COCC1CN(C(=O)c2cc(-c3ccncc3)nc3ccccc23)C1 ZINC000880592178 EG On-Demand Anodyne MT-CO2 49 42 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1Cc1cc(=O)c(O)co1 ZINC000880592181 DH On-Demand Anodyne DAO 21 44 CS(=O)(=O)c1ccnc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)c1 ZINC000880592185 GF On-Demand Anodyne GCK 17 40 CS(=O)(=O)c1ccnc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)c1 ZINC000880592187 GF On-Demand Anodyne GCK 17 40 COCC1CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880592189 CD On-Demand Anodyne MTNR1A 22 46 COCC1CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880592189 CD On-Demand Anodyne MTNR1B 21 46 COCC1CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880592190 CD On-Demand Anodyne MTNR1A 22 46 COCC1CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880592190 CD On-Demand Anodyne MTNR1B 21 46 COCC1CN(C(=O)COc2cccc(C(C)=O)c2)C1 ZINC000880592204 CD On-Demand Anodyne CPT1A 65 40 COCC1CN(C(=O)c2cc(-c3ccc(OC)c(OC)c3)nc3ccccc23)C1 ZINC000880592221 GH On-Demand Anodyne PRS 20 40 COCC1CN(C(=O)c2cc(-c3ccc(OC)c(OC)c3)nc3ccccc23)C1 ZINC000880592221 GH On-Demand Anodyne TACR3 24 41 COCC1CN(C(=O)c2cc(-c3ccc(OC)c(OC)c3)nc3ccccc23)C1 ZINC000880592221 GH On-Demand Anodyne MT-CO2 30 40 CO[C@@H](CN(C)[C@@H](CC(C)C)C(N)=O)c1ccc(F)cc1 ZINC000880592245 CE On-Demand Anodyne AOC3 16 56 CO[C@@H](CN(C)[C@@H](CC(C)C)C(N)=O)c1ccc(F)cc1 ZINC000880592245 CE On-Demand Anodyne LEF 37 45 COc1ccc(N2CCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)cc1 ZINC000880592284 GD On-Demand Clean PDGFRB 47 40 COc1ccc(N2CCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)cc1 ZINC000880592284 GD On-Demand Clean MMP13 28 40 COc1ccc(N2CCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)cc1 ZINC000880592284 GD On-Demand Clean MMP3 24 40 COCC1CN(C(=O)c2ccc(C)c(S(=O)(=O)N3CCOCC3)c2)C1 ZINC000880592289 FC On-Demand Anodyne CNR2 22 64 COCC1CN(C(=O)c2ccc(C)c(S(=O)(=O)N3CCOCC3)c2)C1 ZINC000880592289 FC On-Demand Anodyne NR1H4 18 43 COCC1CN(C(=O)c2ccc(Cl)c(S(=O)(=O)N3CCCCC3)c2)C1 ZINC000880592299 GE On-Demand Anodyne CNR2 15 62 COCC1CN(C(=O)c2ccc(Cl)c(S(=O)(=O)N3CCCCC3)c2)C1 ZINC000880592299 GE On-Demand Anodyne L3MBTL3 48 38 CS(=O)(=O)c1ccnc(NC(=O)NC23CCC(CC2)C3)c1 ZINC000880592336 DD On-Demand Anodyne EPHX2 37 43 CS(=O)(=O)c1ccnc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880592344 GE On-Demand Anodyne EPHX2 40 38 CS(=O)(=O)c1ccnc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880592344 GE On-Demand Anodyne L3MBTL3 53 33 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCCO)CC2)c1 ZINC000880592354 ED On-Demand Anodyne GPR119 40 39 Cc1nn(CC(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)c(=O)o1 ZINC000880592364 GE On-Demand Anodyne SIGMAR1 62 40 Cc1nn(CC(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)c(=O)o1 ZINC000880592364 GE On-Demand Anodyne CCR8 46 42 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCC(C)CC2)C1 ZINC000880592386 EF On-Demand Bother SLC6A9 21 46 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne CHRM2 15 67 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne DRD4 22 40 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne SIGMAR1 62 42 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne FAAH 21 41 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne MCHR2 44 32 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne CCR8 49 48 O=C(c1n[nH]c(O)n1)N1CCC2(CCN(Cc3ccccc3)CC2)CC1 ZINC000880592389 FE On-Demand Anodyne NPFFR1 40 35 CCOc1ccccc1OCC(=O)N1CC(COC)C1 ZINC000880592411 CD On-Demand Anodyne HCN1 50 33 CCOc1ccccc1OCC(=O)N1CC(COC)C1 ZINC000880592411 CD On-Demand Anodyne HCN4 43 33 COCC1CN(C(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880592422 DF On-Demand Anodyne PDE4D 25 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCN3CCOCC3)CC2)c1 ZINC000880592459 GD On-Demand Anodyne CASR 31 43 COCC1CN(C(=O)c2cc(S(C)(=O)=O)ccc2Cl)C1 ZINC000880592465 DD On-Demand Anodyne SLC6A9 40 43 CS(=O)(=O)c1ccnc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880592498 GD On-Demand Anodyne TRPV1 15 43 CS(=O)(=O)c1ccnc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880592498 GD On-Demand Anodyne SLC6A9 29 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880592498 GD On-Demand Anodyne FAAH 22 40 CS(=O)(=O)c1ccnc(NC(=O)N2CCCN(c3ncccc3F)CC2)c1 ZINC000880592498 GD On-Demand Anodyne RBP4 16 45 COCC1CN(C(=O)c2cc(-c3ccccc3)nc3ccc(C)cc23)C1 ZINC000880592516 EH On-Demand Anodyne P2RY12 51 39 COCC1CN(C(=O)c2cc(-c3ccccc3)nc3ccc(C)cc23)C1 ZINC000880592516 EH On-Demand Anodyne PRS 47 36 COCC1CN(C(=O)c2cc(-c3ccccc3)nc3ccc(C)cc23)C1 ZINC000880592516 EH On-Demand Anodyne MT-CO2 50 36 COCC1CN(C(=O)c2cc(-c3ccccc3)nc3ccc(C)cc23)C1 ZINC000880592516 EH On-Demand Anodyne VCP 34 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne ACE 42 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CELA1 25 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne ELANE 38 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne MME 30 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CMA1 15 47 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTRA_BOVIN 56 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CASP3 16 49 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne BMP1 24 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne KLK3 80 37 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTSB 73 51 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne PAPA1_CARPA 83 42 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CYSP_TRYCR 55 42 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTSG 41 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTSK 58 52 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTSL 53 51 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne PGA 22 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CAPNS1 67 39 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CELA2A 45 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTSS 29 52 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CAPN1 90 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CASP1 26 42 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CTRC 15 47 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CAPN2 144 44 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne ACE2 43 35 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CASP9 33 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne NPR 70 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne GAG-PRO 45 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne CASP10 37 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne PSMB5 52 43 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880592519 EE On-Demand Anodyne F2RL1 19 40 CS(=O)(=O)c1ccnc(NC(=O)N[C@@H]2Cc3ccc(Cl)cc3C2)c1 ZINC000880592521 FE On-Demand Anodyne CA7 17 44 CS(=O)(=O)c1ccnc(NC(=O)N[C@H]2Cc3ccc(Cl)cc3C2)c1 ZINC000880592522 FE On-Demand Anodyne CA7 17 44 COCC1CN(C(=O)[C@H]2CC(=O)N(Cc3ccccc3Cl)C2)C1 ZINC000880592529 ED On-Demand Anodyne P2RX7 18 43 COCC1CN(C(=O)[C@@H]2CC(=O)N(Cc3ccccc3Cl)C2)C1 ZINC000880592530 ED On-Demand Anodyne P2RX7 18 43 COCC1CN(C(=O)Cc2cccs2)C1 ZINC000880592550 BD On-Demand Anodyne ETHR 17 43 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne GHRHR 57 33 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne SIGMAR1 67 43 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne CCKBR 20 40 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne MCHR2 64 34 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne CCR8 49 44 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592606 FG On-Demand Anodyne NPFFR1 42 39 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne GHRHR 57 33 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne SIGMAR1 67 43 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne CCKBR 20 40 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne MCHR2 64 34 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne CCR8 49 44 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@H](C)O ZINC000880592607 FG On-Demand Anodyne NPFFR1 42 39 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne GHRHR 57 33 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne SIGMAR1 67 43 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne CCKBR 20 40 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne MCHR2 64 34 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne CCR8 49 44 CC[C@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592608 FG On-Demand Anodyne NPFFR1 42 39 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne GHRHR 57 33 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne SIGMAR1 67 43 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne CCKBR 20 40 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne MCHR2 64 34 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne CCR8 49 44 CC[C@@H](C(=O)N1CCC2(CCN(Cc3ccccc3)CC2)CC1)[C@@H](C)O ZINC000880592609 FG On-Demand Anodyne NPFFR1 42 39 COc1cccc(SCCN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880592637 DF On-Demand Anodyne MTNR1A 20 49 COc1cccc(SCCN(C)[C@@H](CC(C)C)C(N)=O)c1 ZINC000880592637 DF On-Demand Anodyne MTNR1B 22 49 C#CC(C)(C)NC(=O)Nc1cc(S(C)(=O)=O)ccn1 ZINC000880592667 CD On-Demand Mild TYK2 49 33 COCC1CN(C(=O)c2ccnc(N3CCN(C(=O)OC(C)(C)C)CC3)c2)C1 ZINC000880592672 GD On-Demand Anodyne GPR119 52 47 COCC1CN(C(=O)c2ccc(OCc3ccccc3)c(OC)c2)C1 ZINC000880592673 EF On-Demand Anodyne PDGFRB 16 42 COCC1CN(C(=O)c2ccc(OCc3ccccc3)c(OC)c2)C1 ZINC000880592673 EF On-Demand Anodyne PTGER1 58 37 Cc1cccc2c1CCN(C(=O)Nc1cc(S(C)(=O)=O)ccn1)C2 ZINC000880592676 EE On-Demand Anodyne P2RY14 47 33 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne CHRM2 16 69 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne CHRM3 15 64 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne SIGMAR1 67 42 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne FAAH 24 48 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne MCHR2 48 33 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne CCR8 60 49 Cn1nnc(C(=O)N2CCC3(CCN(Cc4ccccc4)CC3)CC2)n1 ZINC000880592687 FD On-Demand Anodyne NPFFR1 43 38 COCC1CN(C(=O)c2cc(-c3cccs3)nc3ccccc23)C1 ZINC000880592696 EH On-Demand Anodyne TACR3 18 52 COCC1CN(C(=O)COc2ccc3c(c2)CCC3)C1 ZINC000880592699 CD On-Demand Anodyne CPT1A 38 43 COCC1CN(C(=O)COc2ccc3c(c2)CCC3)C1 ZINC000880592699 CD On-Demand Anodyne CPT2 45 43 COCC1CN(C(=O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880592703 DE On-Demand Anodyne CPT1A 37 46 COCC1CN(C(=O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880592703 DE On-Demand Anodyne CHRNA10 20 46 COCC1CN(C(=O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880592703 DE On-Demand Anodyne GALR3 44 30 COCC1CN(C(=O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880592703 DE On-Demand Anodyne LIPG 44 35 COCC1CN(C(=O)COc2cccc(C(F)(F)F)c2)C1 ZINC000880592703 DE On-Demand Anodyne PDS 49 39 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c1 ZINC000880592714 GE On-Demand Anodyne NPY5R 38 44 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c1 ZINC000880592714 GE On-Demand Anodyne EPHX2 17 42 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)c3ccc4c(O)ncnc4c3)CC2)C1 ZINC000880592715 GF On-Demand Anodyne ACACA 48 36 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)c1 ZINC000880592727 FG On-Demand Anodyne EPHX2 27 46 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)c1 ZINC000880592727 FG On-Demand Anodyne MAP3K12 41 42 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)c1 ZINC000880592728 FG On-Demand Anodyne EPHX2 27 46 CS(=O)(=O)c1ccnc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)c1 ZINC000880592728 FG On-Demand Anodyne MAP3K12 41 42 COCC1CN(C(=O)c2cc(-c3cccnc3)nc3ccccc23)C1 ZINC000880592731 EG On-Demand Anodyne TACR3 28 44 COCC1CN(C(=O)c2cc(-c3cccnc3)nc3ccccc23)C1 ZINC000880592731 EG On-Demand Anodyne MT-CO2 45 38 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@@H](c3ccccn3)C2)c1 ZINC000880592739 ED On-Demand Anodyne MAP3K12 43 41 CS(=O)(=O)c1ccnc(NC(=O)N2CC[C@H](c3ccccn3)C2)c1 ZINC000880592740 ED On-Demand Anodyne MAP3K12 43 41 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2Cl)C1 ZINC000880592742 CD On-Demand Bother CACNA1C 40 36 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2Cl)C1 ZINC000880592742 CD On-Demand Bother CACNA1D 65 36 C[C@@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880592743 CD On-Demand Anodyne CPT1A 68 36 C[C@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880592744 CD On-Demand Anodyne CPT1A 68 36 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)C1 ZINC000880592751 FC On-Demand Anodyne CASP3 26 40 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)C1 ZINC000880592751 FC On-Demand Anodyne PKM 41 37 c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592757 CD On-Demand Anodyne LTA4H 66 47 c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592757 CD On-Demand Anodyne HRH3 33 49 c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592757 CD On-Demand Anodyne HTR5A 28 47 c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592757 CD On-Demand Anodyne PSMB2 40 39 c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592757 CD On-Demand Anodyne PSMB1 43 40 c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880592765 CE On-Demand Anodyne LTA4H 44 40 c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880592765 CE On-Demand Anodyne HRH3 68 50 c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880592765 CE On-Demand Anodyne SIGMAR1 21 45 c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880592765 CE On-Demand Anodyne HTR5A 37 53 Fc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880592774 BE On-Demand Anodyne GABRA1 19 41 Fc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880592774 BE On-Demand Anodyne GABRA2 23 41 COCC1CN(C(=O)CSc2ccc([N+](=O)[O-])cc2)C1 ZINC000880592779 CD On-Demand Bother FAS 17 41 COCC1CN(C(=O)c2ccc(Cl)c([N+](=O)[O-])c2)C1 ZINC000880592819 CD On-Demand Bother TAAR1 17 43 O=C(CN1CCc2ncncc2C1)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000880592835 GD On-Demand Anodyne CPT1A 49 37 O=C(CN1CCc2ncncc2C1)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000880592836 GD On-Demand Anodyne CPT1A 49 37 Cc1cccc(NC(=O)[C@@H](C)N2CCc3ncncc3C2)c1 ZINC000880592837 CE On-Demand Anodyne P2RY14 43 35 Cc1cccc(NC(=O)[C@@H](C)N2CCc3ncncc3C2)c1 ZINC000880592837 CE On-Demand Anodyne KCNK3 43 34 Cc1cccc(NC(=O)[C@H](C)N2CCc3ncncc3C2)c1 ZINC000880592838 CE On-Demand Anodyne P2RY14 43 35 Cc1cccc(NC(=O)[C@H](C)N2CCc3ncncc3C2)c1 ZINC000880592838 CE On-Demand Anodyne KCNK3 43 34 NS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592850 EC On-Demand Anodyne LTA4H 44 36 NS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592850 EC On-Demand Anodyne CA7 23 42 NS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592850 EC On-Demand Anodyne HRH3 20 53 NS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592850 EC On-Demand Anodyne HTR5A 20 40 NS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880592850 EC On-Demand Anodyne CA9 15 54 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592851 CD On-Demand Anodyne PREP 57 67 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592851 CD On-Demand Anodyne SFRP1 17 40 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592851 CD On-Demand Anodyne WNT3 32 40 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592852 CD On-Demand Anodyne PREP 57 67 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592852 CD On-Demand Anodyne SFRP1 17 40 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880592852 CD On-Demand Anodyne WNT3 32 40 O=C(CN1CCc2ncncc2C1)NCCCN1CCCC1=O ZINC000880592863 DB On-Demand Anodyne TYRO3 19 42 O[C@H](COc1ccc(Cl)cc1)CN1CCc2ncncc2C1 ZINC000880592864 DD On-Demand Anodyne ACOX1 60 33 O[C@@H](COc1ccc(Cl)cc1)CN1CCc2ncncc2C1 ZINC000880592865 DD On-Demand Anodyne ACOX1 60 33 CCOc1ccccc1NC(=O)[C@@H](c1ccccc1)N1CCc2ncncc2C1 ZINC000880592902 GH On-Demand Anodyne KCNQ2 42 34 CCOc1ccccc1NC(=O)[C@H](c1ccccc1)N1CCc2ncncc2C1 ZINC000880592903 GH On-Demand Anodyne KCNQ2 42 34 COc1ccccc1-c1nc(CN2CCc3ncncc3C2)cs1 ZINC000880592921 EG On-Demand Anodyne ABCB1 18 48 COC(=O)c1sccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880592948 ED On-Demand Anodyne FAS 53 48 CS(=O)(=O)c1ccnc(NC(=O)NCc2ccc(N3CCCC3)cc2)c1 ZINC000880592965 FE On-Demand Clean NAMPT 104 42 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)cc1 ZINC000880592980 EE On-Demand Anodyne PRCP 29 44 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)cc1 ZINC000880592980 EE On-Demand Anodyne MAPK1 44 36 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)cc1 ZINC000880592981 EE On-Demand Anodyne PRCP 29 44 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)cc1 ZINC000880592981 EE On-Demand Anodyne MAPK1 44 36 COc1ccccc1COC[C@@H](O)CN1CCc2ncncc2C1 ZINC000880592982 ED On-Demand Anodyne ABCB1 44 35 COc1ccccc1COC[C@H](O)CN1CCc2ncncc2C1 ZINC000880592983 ED On-Demand Anodyne ABCB1 44 35 c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880592987 BE On-Demand Anodyne SIGMAR1 43 59 c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880592987 BE On-Demand Anodyne HTR5A 20 40 c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880592987 BE On-Demand Anodyne ABCB1 21 43 O=[N+]([O-])c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880592992 CD On-Demand Bother KCNJ1 29 47 O[C@@H](COc1ccc(Oc2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880592999 GG On-Demand Anodyne ACOX1 47 39 O[C@@H](COc1ccc(Oc2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880592999 GG On-Demand Anodyne ABCB1 54 40 O[C@H](COc1ccc(Oc2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593000 GG On-Demand Anodyne ACOX1 47 39 O[C@H](COc1ccc(Oc2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593000 GG On-Demand Anodyne ABCB1 54 40 COCC1CN(C(=O)[C@@H](CCSC)NC(=O)OC(C)(C)C)C1 ZINC000880593008 ED On-Demand Anodyne PAPA1_CARPA 33 53 COCC1CN(C(=O)[C@H](CCSC)NC(=O)OC(C)(C)C)C1 ZINC000880593009 ED On-Demand Anodyne PAPA1_CARPA 33 53 O=C1c2ccccc2C(=O)N1CCCN1CCc2ncncc2C1 ZINC000880593031 DD On-Demand Anodyne HTR1A 15 62 CCCCCCCCCC(=O)N1CC(COC)C1 ZINC000880593032 CG On-Demand Mild CQSS 55 35 O[C@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593035 EE On-Demand Anodyne ADRB2 17 53 O[C@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593035 EE On-Demand Anodyne ADRB1 15 44 O[C@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593035 EE On-Demand Anodyne ABCB1 68 43 O[C@@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593036 EE On-Demand Anodyne ADRB2 17 53 O[C@@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593036 EE On-Demand Anodyne ADRB1 15 44 O[C@@H](COc1cccc2ccccc12)CN1CCc2ncncc2C1 ZINC000880593036 EE On-Demand Anodyne ABCB1 68 43 COCC1CN(C(=O)c2cccnc2Cl)C1 ZINC000880593047 BD On-Demand Anodyne G2YM83_BOTF4 73 39 N#Cc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593055 CD On-Demand Mild LTA4H 49 38 N#Cc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593055 CD On-Demand Mild HRH3 22 49 N#Cc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593055 CD On-Demand Mild HTR5A 22 43 N#Cc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593055 CD On-Demand Mild PSMB1 40 35 N#Cc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593055 CD On-Demand Mild MEN1 42 39 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne DRD2 19 50 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne HTR2A 17 52 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne LTA4H 31 43 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne HRH3 70 43 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne SIGMAR1 15 52 Fc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593071 CE On-Demand Anodyne HTR5A 36 67 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593073 DE On-Demand Anodyne PAPA1_CARPA 33 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593073 DE On-Demand Anodyne CTSK 22 49 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593073 DE On-Demand Anodyne REN 26 44 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593073 DE On-Demand Anodyne POLG_HCV1 27 47 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593073 DE On-Demand Anodyne FPR1 51 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593074 DE On-Demand Anodyne PAPA1_CARPA 33 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593074 DE On-Demand Anodyne CTSK 22 49 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593074 DE On-Demand Anodyne REN 26 44 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593074 DE On-Demand Anodyne POLG_HCV1 27 47 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880593074 DE On-Demand Anodyne FPR1 51 40 CC(=O)c1cccc(OC[C@@H](O)CN2CCc3ncncc3C2)c1 ZINC000880593094 ED On-Demand Anodyne ACOX1 61 39 CC(=O)c1cccc(OC[C@@H](O)CN2CCc3ncncc3C2)c1 ZINC000880593094 ED On-Demand Anodyne ABCB1 70 57 CC(=O)c1cccc(OC[C@H](O)CN2CCc3ncncc3C2)c1 ZINC000880593095 ED On-Demand Anodyne ACOX1 61 39 CC(=O)c1cccc(OC[C@H](O)CN2CCc3ncncc3C2)c1 ZINC000880593095 ED On-Demand Anodyne ABCB1 70 57 c1ccc2c(c1)OC[C@@H](CN1CCc3ncncc3C1)O2 ZINC000880593096 CD On-Demand Anodyne ADRA2B 20 45 c1ccc2c(c1)OC[C@H](CN1CCc3ncncc3C1)O2 ZINC000880593097 CD On-Demand Anodyne ADRA2B 20 45 O[C@@H](CN1CCc2ncncc2C1)c1ccc(F)cc1 ZINC000880593102 CD On-Demand Anodyne SLC6A3 18 45 O[C@H](CN1CCc2ncncc2C1)c1ccc(F)cc1 ZINC000880593103 CD On-Demand Anodyne SLC6A3 18 45 COC(=O)c1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880593104 FD On-Demand Anodyne ABCB1 76 38 COC(=O)c1ccc(OC[C@H](O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880593105 FD On-Demand Anodyne ABCB1 76 38 O[C@H](COC(c1ccccc1)c1ccccc1)CN1CCc2ncncc2C1 ZINC000880593106 GG On-Demand Anodyne SLC6A3 39 44 O[C@@H](COC(c1ccccc1)c1ccccc1)CN1CCc2ncncc2C1 ZINC000880593107 GG On-Demand Anodyne SLC6A3 39 44 COCC1CN(C(=O)c2c(-c3c(Cl)cccc3Cl)noc2C)C1 ZINC000880593113 FH On-Demand Anodyne NR1H4 48 36 COCC1CN(C(=O)c2c(-c3c(Cl)cccc3Cl)noc2C)C1 ZINC000880593113 FH On-Demand Anodyne GPBAR1 30 46 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C1 ZINC000880593117 ED On-Demand Bother SLC6A9 26 60 COc1ccc(CNC(=O)[C@H](C)N2CCc3ncncc3C2)cc1OC ZINC000880593130 FD On-Demand Anodyne HCRTR1 15 41 COc1ccc(CNC(=O)[C@H](C)N2CCc3ncncc3C2)cc1OC ZINC000880593130 FD On-Demand Anodyne DRTS_TRYCR 47 33 COCC1CN(C(=O)c2ccc(S(=O)(=O)N3CCCC3)o2)C1 ZINC000880593140 EC On-Demand Anodyne LPL 40 36 COc1ccc(OC)c([C@H]2CCCN2C(=O)CN2CCc3ncncc3C2)c1 ZINC000880593152 GE On-Demand Anodyne CPT1A 88 38 COCC1CN(C(=O)c2cc(-c3ccc4c(c3)OCCO4)nc3ccccc23)C1 ZINC000880593153 GG On-Demand Anodyne TACR3 16 41 O[C@@H](COc1ccc(Cl)c(Cl)c1)CN1CCc2ncncc2C1 ZINC000880593154 FF On-Demand Anodyne ACOX1 81 38 O[C@H](COc1ccc(Cl)c(Cl)c1)CN1CCc2ncncc2C1 ZINC000880593155 FF On-Demand Anodyne ACOX1 81 38 CC(C)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880593164 DF On-Demand Anodyne ACOX1 42 34 CC(C)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880593164 DF On-Demand Anodyne P2RY14 43 36 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne CHRM2 38 41 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP13 72 42 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP2 47 38 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP3 68 39 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne PRTN3 70 44 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP9 64 42 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP7 47 39 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(OC)cc2)C1 ZINC000880593178 GE On-Demand Anodyne MMP1 67 42 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCc3ccccc3)CC2)c1 ZINC000880593188 GG On-Demand Anodyne GRIN2B 44 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCc3ccccc3)CC2)c1 ZINC000880593188 GG On-Demand Anodyne FAAH 16 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCc3ccccc3)CC2)c1 ZINC000880593188 GG On-Demand Anodyne EPHX2 18 41 CS(=O)(=O)c1ccnc(NC(=O)N2CCC(CCc3ccccc3)CC2)c1 ZINC000880593188 GG On-Demand Anodyne ST14 56 34 COCC1CN(C(=O)CSc2nnc(-c3ccc(OC)cc3)o2)C1 ZINC000880593199 ED On-Demand Anodyne GSK3B 15 47 COCC1CN(C(=O)CSc2nnc(-c3ccc(OC)cc3)o2)C1 ZINC000880593199 ED On-Demand Anodyne GSK3A 30 43 O[C@@H](COc1ccccc1Cl)CN1CCc2ncncc2C1 ZINC000880593214 DD On-Demand Anodyne ABCB1 59 40 O[C@H](COc1ccccc1Cl)CN1CCc2ncncc2C1 ZINC000880593215 DD On-Demand Anodyne ABCB1 59 40 O[C@@H](COc1cc(Cl)ccc1Cl)CN1CCc2ncncc2C1 ZINC000880593217 FF On-Demand Anodyne GPBAR1 18 42 O[C@H](COc1cc(Cl)ccc1Cl)CN1CCc2ncncc2C1 ZINC000880593218 FF On-Demand Anodyne GPBAR1 18 42 N#Cc1c(NC(=O)CCN2CCc3ncncc3C2)sc2c1CCCCC2 ZINC000880593219 GG On-Demand Mild VIPR1 31 52 CC[C@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880593229 CD On-Demand Anodyne CPT1A 48 35 CC[C@@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880593230 CD On-Demand Anodyne CPT1A 48 35 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2cc(C)ccc2C)C1 ZINC000880593240 GF On-Demand Anodyne PRTN3 47 33 COCC1CN(C(=O)c2ccccc2NS(=O)(=O)c2cc(C)ccc2C)C1 ZINC000880593240 GF On-Demand Anodyne CCR8 51 31 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593249 FF On-Demand Anodyne ACOX1 73 39 O[C@H](COc1ccc(-c2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593249 FF On-Demand Anodyne ABCB1 57 40 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593250 FF On-Demand Anodyne ACOX1 73 39 O[C@@H](COc1ccc(-c2ccccc2)cc1)CN1CCc2ncncc2C1 ZINC000880593250 FF On-Demand Anodyne ABCB1 57 40 CCCCSCC(=O)N1CC(COC)C1 ZINC000880593251 BD On-Demand Anodyne CES1 16 40 CCCCSCC(=O)N1CC(COC)C1 ZINC000880593251 BD On-Demand Anodyne EST1_PIG 46 40 COCC1CN(C(=O)c2ccccc2NS(C)(=O)=O)C1 ZINC000880593260 CC On-Demand Anodyne PRTN3 45 32 CCCCCCCC(=O)N1CC(COC)C1 ZINC000880593266 BE On-Demand Mild CQSS 55 35 O=C(CN1CCc2ncncc2C1)NC[C@H]1COc2ccccc2O1 ZINC000880593275 EC On-Demand Anodyne ADRA2B 16 43 O=C(CN1CCc2ncncc2C1)NC[C@@H]1COc2ccccc2O1 ZINC000880593276 EC On-Demand Anodyne ADRA2B 16 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne F2 34 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PLG 31 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne ACE 87 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TYR 33 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne OPRM1 53 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne OPRD1 51 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne GHRHR 58 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne P2RY12 100 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne ELANE 29 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne MME 103 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne ANPEP 49 33 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TACR1 24 56 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PGC 50 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne MC4R 56 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CMA1 30 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTRA_BOVIN 76 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne FCER2 42 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CASP3 17 47 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne BMP1 20 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne KLK3 87 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTSB 93 53 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TRY2_BOVIN 61 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PAPA1_CARPA 101 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TRY1_BOVIN 46 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CYSP_TRYCR 77 50 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CCKAR 17 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTSG 50 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTSK 64 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTSL 71 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CACNA1B 39 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne NPFFR2 60 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TIMP3 62 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PREP 19 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CAPNS1 88 48 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne ECE1 24 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne HLA-DRB1 43 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CELA2A 68 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne REN 85 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne MMP11 72 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTSS 45 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CAPN1 136 48 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CASP1 26 44 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTRC 19 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CAPN2 160 53 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne ACE2 85 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PLAU 20 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TGM2 36 47 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne TPSAB1 44 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne KLK1 24 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne FPR1 65 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne CTRB_BOVIN 46 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne NPR 79 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne PSMB5 50 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne BLA1_STEMA 44 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593287 GF On-Demand Anodyne NPFFR1 49 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne F2 34 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PLG 31 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne ACE 87 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TYR 33 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne OPRM1 53 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne OPRD1 51 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne GHRHR 58 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne P2RY12 100 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne ELANE 29 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne MME 103 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne ANPEP 49 33 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TACR1 24 56 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PGC 50 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne MC4R 56 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CMA1 30 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTRA_BOVIN 76 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne FCER2 42 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CASP3 17 47 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne BMP1 20 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne KLK3 87 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTSB 93 53 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TRY2_BOVIN 61 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PAPA1_CARPA 101 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TRY1_BOVIN 46 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CYSP_TRYCR 77 50 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CCKAR 17 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTSG 50 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTSK 64 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTSL 71 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CACNA1B 39 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne NPFFR2 60 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TIMP3 62 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PREP 19 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CAPNS1 88 48 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne ECE1 24 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne HLA-DRB1 43 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CELA2A 68 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne REN 85 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne MMP11 72 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTSS 45 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CAPN1 136 48 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CASP1 26 44 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTRC 19 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CAPN2 160 53 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne ACE2 85 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PLAU 20 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TGM2 36 47 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne TPSAB1 44 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne KLK1 24 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne FPR1 65 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne CTRB_BOVIN 46 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne NPR 79 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne PSMB5 50 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne BLA1_STEMA 44 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C1 ZINC000880593288 GF On-Demand Anodyne NPFFR1 49 32 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593292 DD On-Demand Anodyne CTSK 15 53 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593292 DD On-Demand Anodyne PGA5 24 43 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593292 DD On-Demand Anodyne POLG_HCV1 23 41 COCC1CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593293 DD On-Demand Anodyne CTSK 15 53 COCC1CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593293 DD On-Demand Anodyne PGA5 24 43 COCC1CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880593293 DD On-Demand Anodyne POLG_HCV1 23 41 CCCCCCC(=O)N1CC(COC)C1 ZINC000880593294 BE On-Demand Anodyne CQSS 55 35 COCC1CN(C(=O)[C@@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880593301 CD On-Demand Anodyne CTSK 18 43 COCC1CN(C(=O)[C@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880593302 CD On-Demand Anodyne CTSK 18 43 O[C@@H](COc1c(Cl)cccc1Cl)CN1CCc2ncncc2C1 ZINC000880593304 FF On-Demand Anodyne ABCB1 44 35 O[C@H](COc1c(Cl)cccc1Cl)CN1CCc2ncncc2C1 ZINC000880593305 FF On-Demand Anodyne ABCB1 44 35 Cc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)c(C)c1 ZINC000880593318 DD On-Demand Anodyne ABCB1 59 43 Cc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)c(C)c1 ZINC000880593319 DD On-Demand Anodyne ABCB1 59 43 CSc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880593321 CF On-Demand Anodyne NOD2 34 47 O=C(CN1CCc2ncncc2C1)Nc1ccc(CN2CCOCC2)cc1 ZINC000880593331 FD On-Demand Anodyne EPHX2 16 43 O=C(CN1CCc2ncncc2C1)Nc1ccc(CN2CCOCC2)cc1 ZINC000880593331 FD On-Demand Anodyne AURKA 17 40 O=C(CN1CCc2ncncc2C1)Nc1ccc(CN2CCOCC2)cc1 ZINC000880593331 FD On-Demand Anodyne NOD2 45 39 O[C@H](COc1cccc(Br)c1)CN1CCc2ncncc2C1 ZINC000880593340 FE On-Demand Anodyne ACOX1 66 36 O[C@@H](COc1cccc(Br)c1)CN1CCc2ncncc2C1 ZINC000880593341 FE On-Demand Anodyne ACOX1 66 36 O=C(c1ccc(CN2CCc3ncncc3C2)cc1)N1CCCC1 ZINC000880593342 DE On-Demand Anodyne FABI 42 35 O=C(c1ccc(CN2CCc3ncncc3C2)cc1)N1CCCC1 ZINC000880593342 DE On-Demand Anodyne HRH3 17 45 O=C(c1ccc(CN2CCc3ncncc3C2)cc1)N1CCCC1 ZINC000880593342 DE On-Demand Anodyne L3MBTL3 55 45 O=C(c1ccc(CN2CCc3ncncc3C2)cc1)N1CCCC1 ZINC000880593342 DE On-Demand Anodyne NOD2 45 38 Fc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593353 CE On-Demand Anodyne LTA4H 55 49 Fc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593353 CE On-Demand Anodyne HRH3 31 40 Fc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593353 CE On-Demand Anodyne HTR5A 31 60 Fc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593353 CE On-Demand Anodyne PSMB1 41 36 COCC1CN(C(=O)/C=C/c2ccc(OC)cc2)C1 ZINC000880593356 CD On-Demand Anodyne MMP2 17 41 COCC1CN(C(=O)/C=C/c2ccc(OC)cc2)C1 ZINC000880593356 CD On-Demand Anodyne MMP3 43 38 COCC1CN(C(=O)/C=C/c2ccc(OC)cc2)C1 ZINC000880593356 CD On-Demand Anodyne MMP9 30 41 COCC1CN(C(=O)/C=C\c2ccc(OC)cc2)C1 ZINC000880593357 CD On-Demand Anodyne MMP2 17 41 COCC1CN(C(=O)/C=C\c2ccc(OC)cc2)C1 ZINC000880593357 CD On-Demand Anodyne MMP3 43 38 COCC1CN(C(=O)/C=C\c2ccc(OC)cc2)C1 ZINC000880593357 CD On-Demand Anodyne MMP9 30 41 Brc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880593359 EF On-Demand Anodyne LTA4H 27 41 Brc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880593359 EF On-Demand Anodyne HMOX2 21 44 N#Cc1c(NC(=O)CCN2CCc3ncncc3C2)sc2c1CCCC2 ZINC000880593364 FF On-Demand Mild VIPR1 32 53 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA2 35 41 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA1 28 40 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA7 40 37 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA4 26 41 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA12 27 40 COCC1CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C1 ZINC000880593371 DC On-Demand Anodyne CA9 24 41 COCC1CN(C(=O)/C=C\c2ccc(OC)c(OC)c2)C1 ZINC000880593374 CD On-Demand Anodyne CYP1A1 15 43 COCC1CN(C(=O)/C=C\c2ccc(OC)c(OC)c2)C1 ZINC000880593374 CD On-Demand Anodyne ABCG2 15 45 COCC1CN(C(=O)/C=C/c2ccc(OC)c(OC)c2)C1 ZINC000880593375 CD On-Demand Anodyne CYP1A1 15 43 COCC1CN(C(=O)/C=C/c2ccc(OC)c(OC)c2)C1 ZINC000880593375 CD On-Demand Anodyne ABCG2 15 45 O=C(CN1CCc2ncncc2C1)NC[C@H]1CCCO1 ZINC000880593376 CC On-Demand Anodyne TNK2 45 34 O=C(CN1CCc2ncncc2C1)NC[C@@H]1CCCO1 ZINC000880593377 CC On-Demand Anodyne TNK2 45 34 Cc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593380 CD On-Demand Anodyne ACOX1 84 38 Cc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593380 CD On-Demand Anodyne ABCB1 50 39 Cc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593381 CD On-Demand Anodyne ACOX1 84 38 Cc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593381 CD On-Demand Anodyne ABCB1 50 39 COCC1CN(C(=O)[C@@H]2CSCN2C(=O)c2ccccc2)C1 ZINC000880593386 DD On-Demand Anodyne PREP 42 46 COCC1CN(C(=O)[C@H]2CSCN2C(=O)c2ccccc2)C1 ZINC000880593387 DD On-Demand Anodyne PREP 42 46 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne ESR1 18 41 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne LTA4H 57 47 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne HRH3 45 38 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne HTR5A 25 47 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne ABCB1 18 57 COc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593391 CD On-Demand Anodyne PSMB1 42 37 O[C@H](COCc1ccccc1)CN1CCc2ncncc2C1 ZINC000880593396 CD On-Demand Anodyne ABCB1 42 35 O[C@@H](COCc1ccccc1)CN1CCc2ncncc2C1 ZINC000880593397 CD On-Demand Anodyne ABCB1 42 35 COCC1CN(C(=O)C2CCN(C(=O)/C=C/c3ccccc3)CC2)C1 ZINC000880593399 EE On-Demand Anodyne ITGAL 35 40 COCC1CN(C(=O)C2CCN(C(=O)/C=C\c3ccccc3)CC2)C1 ZINC000880593400 EE On-Demand Anodyne ITGAL 35 40 NC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593401 CD On-Demand Anodyne TRY2_BOVIN 54 32 NC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593401 CD On-Demand Anodyne NOD2 40 34 O[C@@H](COc1ccccc1F)CN1CCc2ncncc2C1 ZINC000880593403 DD On-Demand Anodyne ABCB1 59 40 O[C@H](COc1ccccc1F)CN1CCc2ncncc2C1 ZINC000880593404 DD On-Demand Anodyne ABCB1 59 40 COC(=O)c1ccc(CN2CCc3ncncc3C2)o1 ZINC000880593413 CD On-Demand Anodyne NOD2 41 35 CN(Cc1ccc(F)cc1)C(=O)CN1CCc2ncncc2C1 ZINC000880593421 DD On-Demand Anodyne PLA2G7 46 41 COc1cc(CN2CCc3ncncc3C2)ccc1OC(F)F ZINC000880593428 DF On-Demand Anodyne ABCB1 22 43 COCC1CN(C(=O)c2ccc(NC(=O)OC)cc2)C1 ZINC000880593431 CD On-Demand Anodyne ACR 41 34 O[C@@H](COc1ccc2ccccc2c1)CN1CCc2ncncc2C1 ZINC000880593432 EE On-Demand Anodyne ACOX1 82 40 O[C@@H](COc1ccc2ccccc2c1)CN1CCc2ncncc2C1 ZINC000880593432 EE On-Demand Anodyne ABCB1 50 38 O[C@H](COc1ccc2ccccc2c1)CN1CCc2ncncc2C1 ZINC000880593433 EE On-Demand Anodyne ACOX1 82 40 O[C@H](COc1ccc2ccccc2c1)CN1CCc2ncncc2C1 ZINC000880593433 EE On-Demand Anodyne ABCB1 50 38 CCCCCCCCC(=O)N1CC(COC)C1 ZINC000880593435 BF On-Demand Mild CQSS 55 35 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne DRD2 15 40 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne LTA4H 32 41 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne HTR7 16 43 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne HRH3 82 43 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne SIGMAR1 26 41 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne HTR5A 29 53 COc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593453 CE On-Demand Anodyne ABCB1 19 55 C=CCc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880593454 FE On-Demand Mild ABCB1 50 37 C=CCc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880593455 FE On-Demand Mild ABCB1 50 37 O=C1c2ccccc2C(=O)N1CCCCN1CCc2ncncc2C1 ZINC000880593459 ED On-Demand Anodyne HTR1A 19 66 O=C1c2ccccc2C(=O)N1CCCCN1CCc2ncncc2C1 ZINC000880593459 ED On-Demand Anodyne HTR7 17 43 Cc1oc(-c2ccccc2)nc1CN1CCc2ncncc2C1 ZINC000880593462 DF On-Demand Anodyne PPARG 62 38 Cc1oc(-c2ccccc2)nc1CN1CCc2ncncc2C1 ZINC000880593462 DF On-Demand Anodyne PPARA 63 38 Cc1oc(-c2ccccc2)nc1CN1CCc2ncncc2C1 ZINC000880593462 DF On-Demand Anodyne PDE8B 68 41 COCC1CN(C(=O)CNC(=O)c2ccc(-c3ccccc3)cc2)C1 ZINC000880593469 EE On-Demand Anodyne DRD3 15 41 COCC1CN(C(=O)CNC(=O)c2ccc(-c3ccccc3)cc2)C1 ZINC000880593469 EE On-Demand Anodyne P2RY12 56 40 COCC1CN(C(=O)CNC(=O)c2ccc(-c3ccccc3)cc2)C1 ZINC000880593469 EE On-Demand Anodyne CACNA1I 41 33 COCC1CN(C(=O)CNC(=O)c2ccc(-c3ccccc3)cc2)C1 ZINC000880593469 EE On-Demand Anodyne UTS2 46 37 c1ccc(C(OCCN2CCc3ncncc3C2)c2ccccc2)cc1 ZINC000880593472 EH On-Demand Anodyne SLC6A4 26 52 c1ccc(C(OCCN2CCc3ncncc3C2)c2ccccc2)cc1 ZINC000880593472 EH On-Demand Anodyne SLC6A3 68 59 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc2ccccc2c1 ZINC000880593474 EF On-Demand Anodyne ACOX1 47 49 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc2ccccc2c1 ZINC000880593475 EF On-Demand Anodyne ACOX1 47 49 CC(=O)c1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593498 ED On-Demand Anodyne ACOX1 56 36 CC(=O)c1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593498 ED On-Demand Anodyne ABCB1 56 43 CC(=O)c1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593499 ED On-Demand Anodyne ACOX1 56 36 CC(=O)c1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880593499 ED On-Demand Anodyne ABCB1 56 43 O=C(CN1CCc2ncncc2C1)N1CCC[C@H]1c1ccc2c(c1)OCCCO2 ZINC000880593505 GE On-Demand Anodyne CPT1A 43 37 O=C(CN1CCc2ncncc2C1)N1CCC[C@@H]1c1ccc2c(c1)OCCCO2 ZINC000880593506 GE On-Demand Anodyne CPT1A 43 37 CCOc1ccc(-c2nc(CN3CCc4ncncc4C3)cs2)cc1OC ZINC000880593523 GH On-Demand Anodyne PPARD 17 41 CCOc1ccc(-c2nc(CN3CCc4ncncc4C3)cs2)cc1OC ZINC000880593523 GH On-Demand Anodyne ABCB1 16 57 O=C(CN1CCc2ncncc2C1)NCC1(N2CCOCC2)CCCCC1 ZINC000880593524 FC On-Demand Anodyne HCN1 56 35 O=C(CN1CCc2ncncc2C1)NCC1(N2CCOCC2)CCCCC1 ZINC000880593524 FC On-Demand Anodyne HCN4 51 35 c1coc(-c2noc(CN3CCc4ncncc4C3)n2)c1 ZINC000880593535 CD On-Demand Anodyne ADORA2A 19 53 CCCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593537 DF On-Demand Anodyne LTA4H 55 43 CCCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593537 DF On-Demand Anodyne HRH3 33 40 CCCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593537 DF On-Demand Anodyne HTR5A 25 44 CCCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593537 DF On-Demand Anodyne PSMB2 40 37 CCCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593537 DF On-Demand Anodyne PSMB1 43 37 COCC1CN(C(=O)COc2ccc(N3CCCC3=O)cc2)C1 ZINC000880593540 DD On-Demand Anodyne CPT1A 30 40 COCC1CN(C(=O)c2cccc(S(=O)(=O)N(C)OC)c2)C1 ZINC000880593562 EC On-Demand Anodyne CACNA1B 24 41 O=C(CN1CCc2ncncc2C1)N1CCc2ccccc2C1 ZINC000880593587 DD On-Demand Anodyne HTR7 17 41 COCC1CN(C(=O)c2cc(S(=O)(=O)NC3CC3)c(Cl)cc2Cl)C1 ZINC000880593596 GE On-Demand Anodyne CCR8 49 33 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne ACE 61 46 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne GHRHR 44 31 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CELA1 27 48 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne ELANE 38 44 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne MME 38 42 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTRA_BOVIN 55 33 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CASP3 18 46 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne KLK3 86 39 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTSB 72 48 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne PAPA1_CARPA 80 40 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CYSP_TRYCR 60 42 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTSG 41 31 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTSK 57 51 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTSL 54 51 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne PREP 20 53 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CAPNS1 70 40 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CELA2A 41 33 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne MMP11 46 32 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTSS 32 51 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CAPN1 94 47 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CASP1 27 42 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CTRC 15 47 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CAPN2 146 42 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne PLAU 20 41 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne CASP9 30 40 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne TGM2 36 43 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne TPSAB1 27 40 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne NPR 82 37 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne PSMB5 47 42 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne BIRC2 24 40 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne Q6PRC7_IXORI 44 38 COCC1CN(C(=O)[C@H](C)NC(=O)OCc2ccccc2)C1 ZINC000880593605 DD On-Demand Anodyne SLC12A5 45 35 O=C(CN1CCc2ncncc2C1)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000880593611 GD On-Demand Anodyne DRD4 36 48 O=C(CN1CCc2ncncc2C1)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000880593611 GD On-Demand Anodyne SIGMAR1 18 48 O=C(CN1CCc2ncncc2C1)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000880593611 GD On-Demand Anodyne FAAH 32 49 CCOC(=O)C1=C(CN2CCc3ncncc3C2)NC(=O)N[C@H]1c1ccccc1 ZINC000880593623 GD On-Demand Anodyne SLC27A4 44 32 CCOC(=O)C1=C(CN2CCc3ncncc3C2)NC(=O)N[C@@H]1c1ccccc1 ZINC000880593624 GD On-Demand Anodyne SLC27A4 44 32 CS(=O)(=O)c1ccnc(NC(=O)NC2CCN(CC3CCCCC3)CC2)c1 ZINC000880593628 GF On-Demand Anodyne SSTR5 44 40 CS(=O)(=O)c1ccnc(NC(=O)NC2CCN(CC3CCCCC3)CC2)c1 ZINC000880593628 GF On-Demand Anodyne EPHX2 44 39 CS(=O)(=O)c1ccnc(NC(=O)NC2CCN(CC3CCCCC3)CC2)c1 ZINC000880593628 GF On-Demand Anodyne CXCR3 17 42 Fc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593629 BE On-Demand Anodyne GABRA1 20 44 Fc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593629 BE On-Demand Anodyne SIGMAR1 15 49 Fc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593629 BE On-Demand Anodyne GABRA2 24 44 Fc1ccccc1OCCN1CCc2ncncc2C1 ZINC000880593630 CE On-Demand Anodyne HTR5A 21 43 O=C(CN1CCc2ncncc2C1)NCCc1ccc(F)cc1 ZINC000880593636 DD On-Demand Anodyne SLC27A1 43 36 CCOC(=O)Nc1ccc(C(=O)N2CC(COC)C2)cc1 ZINC000880593637 CD On-Demand Anodyne ACR 45 34 COCC1CN(C(=O)c2ccc(NC(N)=O)cc2)C1 ZINC000880593643 CC On-Demand Anodyne ACR 62 38 COC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593649 CD On-Demand Anodyne FAAH 25 43 COC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593649 CD On-Demand Anodyne P2RY14 43 37 COC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593649 CD On-Demand Anodyne ABCG2 33 43 COC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593649 CD On-Demand Anodyne NOD2 46 39 COCC1CN(C(=O)c2cc3ccc(C(C)C)cc3[nH]2)C1 ZINC000880593676 CG On-Demand Anodyne GRIN2B 25 45 COCC1CN(C(=O)c2cc3ccc(C(C)C)cc3[nH]2)C1 ZINC000880593676 CG On-Demand Anodyne HRH4 25 42 COCC1CN(C(=O)c2cc3ccc(C(C)C)cc3[nH]2)C1 ZINC000880593676 CG On-Demand Anodyne AKR1C3 18 40 c1ccc(CCOCCCN2CCc3ncncc3C2)cc1 ZINC000880593683 CE On-Demand Anodyne HRH3 17 60 c1ccc(CCOCCCN2CCc3ncncc3C2)cc1 ZINC000880593683 CE On-Demand Anodyne SIGMAR1 35 48 c1ccc(CCOCCCN2CCc3ncncc3C2)cc1 ZINC000880593683 CE On-Demand Anodyne HTR5A 29 41 Cc1ccccc1CN1CCC(NC(=O)CN2CCc3ncncc3C2)CC1 ZINC000880593701 GD On-Demand Anodyne DRD4 23 52 Cc1ccccc1CN1CCC(NC(=O)CN2CCc3ncncc3C2)CC1 ZINC000880593701 GD On-Demand Anodyne SIGMAR1 17 45 Cc1ccccc1CN1CCC(NC(=O)CN2CCc3ncncc3C2)CC1 ZINC000880593701 GD On-Demand Anodyne SSTR5 45 38 C[C@H](C(=O)Nc1cccc(Br)c1)N1CCc2ncncc2C1 ZINC000880593704 FF On-Demand Anodyne EGFR 76 41 O=[N+]([O-])c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593707 DE On-Demand Bother HRH3 50 54 O=[N+]([O-])c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593707 DE On-Demand Bother HTR5A 24 56 O=C(CCN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880593709 ED On-Demand Anodyne NOS2 59 33 O=C(CCN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880593709 ED On-Demand Anodyne DYRK2 42 33 O=C(CCN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880593709 ED On-Demand Anodyne TRPC6 27 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880593709 ED On-Demand Anodyne TRPC3 29 40 COc1ccc(CN(C)C(=O)CN2CCc3ncncc3C2)cc1OC ZINC000880593724 FD On-Demand Anodyne ABCB1B 42 37 CC(C)c1cccc(C(C)C)c1NC(=O)CN1CCc2ncncc2C1 ZINC000880593747 FH On-Demand Anodyne SOAT1 57 40 COCC1CN(C(=O)c2cc(C)n(Cc3ccccc3)c2C)C1 ZINC000880593770 DF On-Demand Anodyne PLA2G2A 59 36 O=C(CCN1CCc2ncncc2C1)Nc1cccc(Cl)c1 ZINC000880593775 DF On-Demand Anodyne HTR7 17 40 N#Cc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593779 CE On-Demand Mild HRH3 58 55 N#Cc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593779 CE On-Demand Mild HTR5A 25 48 N#Cc1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880593779 CE On-Demand Mild MEN1 50 44 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne MME 44 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne CMA1 50 36 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne CTRA_BOVIN 40 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne TRY2_BOVIN 41 31 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne ACE2 54 34 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne PLM2_PLAFA 40 31 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne PSMB8 48 38 CC(=O)[C@@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593790 ED On-Demand Anodyne GPR142 51 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne MME 44 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne CMA1 50 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne CTRA_BOVIN 40 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne TRY2_BOVIN 41 31 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne ACE2 54 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne PLM2_PLAFA 40 31 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne BLA1_STEMA 40 32 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne PSMB8 48 38 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN1CCc2ncncc2C1 ZINC000880593792 ED On-Demand Anodyne GPR142 51 35 COc1ccc(C)cc1NC(=O)CN1CCc2ncncc2C1 ZINC000880593795 DD On-Demand Anodyne ABCG2 32 41 Brc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593798 EF On-Demand Anodyne LTA4H 53 49 Brc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593798 EF On-Demand Anodyne HTR5A 22 44 Brc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593798 EF On-Demand Anodyne PSMB1 41 36 O=C(CCN1CCc2ncncc2C1)Nc1ccc(F)cc1 ZINC000880593801 DE On-Demand Anodyne CHRNA7 17 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(F)cc1 ZINC000880593801 DE On-Demand Anodyne ABCB1B 30 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(F)cc1 ZINC000880593801 DE On-Demand Anodyne ABCG2 23 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(F)cc1 ZINC000880593801 DE On-Demand Anodyne NOD2 40 35 COCC1CN(C(=O)COc2cccc(C#N)c2)C1 ZINC000880593806 CD On-Demand Mild CPT1A 70 44 COCC1CN(C(=O)COc2cccc(C#N)c2)C1 ZINC000880593806 CD On-Demand Mild CPT2 42 37 COCC1CN(C(=O)COc2cccc(C#N)c2)C1 ZINC000880593806 CD On-Demand Mild CHRNA10 20 45 O=C(CN1CCc2ncncc2C1)N1CCc2ccccc21 ZINC000880593809 CD On-Demand Anodyne EIF2AK3 44 33 COc1cc2c(cc1OC)CN(C(=O)CN1CCc3ncncc3C1)CC2 ZINC000880593819 FD On-Demand Anodyne ABCB1B 65 43 COc1cc2c(cc1OC)CN(C(=O)CN1CCc3ncncc3C1)CC2 ZINC000880593819 FD On-Demand Anodyne ABCB1 28 47 COc1cc2c(cc1OC)CN(C(=O)CN1CCc3ncncc3C1)CC2 ZINC000880593819 FD On-Demand Anodyne ABCG2 37 43 COCC1CN(C(=O)COCc2ccc(OC)cc2)C1 ZINC000880593829 CD On-Demand Anodyne UGCG 20 43 COCC1CN(C(=O)COCc2ccc(OC)cc2)C1 ZINC000880593829 CD On-Demand Anodyne GBA2 29 43 Fc1ccc(CN2CCc3ncncc3C2)cc1F ZINC000880593836 CE On-Demand Anodyne ABCC1 42 34 O=C(NCc1ccco1)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880593866 EF On-Demand Anodyne CHRM3 15 41 COCC1CN(C(=O)CCc2c(C)c3ccc(OC)cc3oc2=O)C1 ZINC000880593893 EE On-Demand Anodyne MAOB 35 48 COCC1CN(C(=O)CCc2c(C)c3ccc(OC)cc3oc2=O)C1 ZINC000880593893 EE On-Demand Anodyne NQO1 37 47 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1CCc2ncncc2C1 ZINC000880593894 FF On-Demand Anodyne KIT 15 41 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1CCc2ncncc2C1 ZINC000880593894 FF On-Demand Anodyne TRPV1 15 43 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1CCc2ncncc2C1 ZINC000880593894 FF On-Demand Anodyne KDR 18 41 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)N1CCc2ncncc2C1 ZINC000880593894 FF On-Demand Anodyne RIPK1 41 33 COCC1CN(C(=O)CCCNS(=O)(=O)c2ccc(F)cc2)C1 ZINC000880593895 EC On-Demand Anodyne HTR7 15 44 COCC1CN(C(=O)CCCNS(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000880593896 GD On-Demand Anodyne CACNA1B 58 38 COCC1CN(C(=O)CCCNS(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000880593896 GD On-Demand Anodyne CCR2 41 35 COCC1CN(C(=O)CCCNS(=O)(=O)c2cccc(C(F)(F)F)c2)C1 ZINC000880593896 GD On-Demand Anodyne SFRP1 48 37 CC(C)(C)N1CCC(NC(=O)Nc2cc(S(C)(=O)=O)ccn2)CC1 ZINC000880593898 FD On-Demand Anodyne EPHX2 41 41 O=C(CN1CCc2ncncc2C1)NCC1(c2ccccc2)CCCC1 ZINC000880593903 FE On-Demand Anodyne NPFFR1 22 40 O[C@@H]1CCCC[C@H]1N1CCc2ncncc2C1 ZINC000880593914 BD On-Demand Anodyne SLC18A3 34 41 O=C(c1cccc(CN2CCc3ncncc3C2)c1)N1CCCCC1 ZINC000880593924 EF On-Demand Anodyne PARP1 17 42 COCC1CN(C(=O)C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880593927 DD On-Demand Anodyne GPR119 40 40 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCCC3)ccc2Cl)C1 ZINC000880593950 FD On-Demand Anodyne CASP7 48 36 CN(C)S(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880593951 FD On-Demand Anodyne HRH3 22 43 COCC1CN(C(=O)c2cc(S(C)(=O)=O)ccc2Br)C1 ZINC000880593967 FD On-Demand Anodyne SLC6A9 40 42 CCOC(=O)N[C@H](CNC(=O)Nc1cc(CN(C)C)ccn1)CC(C)C ZINC000880593988 FE On-Demand Anodyne CAPN2 43 32 CCOC(=O)N[C@@H](CNC(=O)Nc1cc(CN(C)C)ccn1)CC(C)C ZINC000880593989 FE On-Demand Anodyne CAPN2 43 32 COc1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594003 CD On-Demand Anodyne DRD4 26 41 COc1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594003 CD On-Demand Anodyne ABCB1B 52 40 COc1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594003 CD On-Demand Anodyne ABCB1 26 40 COc1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594003 CD On-Demand Anodyne ABCG2 36 40 N#Cc1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594008 CD On-Demand Mild CCR3 15 43 N#Cc1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594008 CD On-Demand Mild MCHR1 35 41 COCC1CN(C(=O)c2cc3c(Br)cccc3[nH]2)C1 ZINC000880594009 DF On-Demand Anodyne GRIN2B 24 44 COCC1CN(C(=O)c2cc3c(Br)cccc3[nH]2)C1 ZINC000880594009 DF On-Demand Anodyne HRH4 23 61 CSc1ccc(NC(=O)CN2CCc3ncncc3C2)cc1 ZINC000880594010 DE On-Demand Anodyne NOD1 15 46 CSc1ccc(NC(=O)CN2CCc3ncncc3C2)cc1 ZINC000880594010 DE On-Demand Anodyne NOD2 41 46 O=C(CN1CCc2ncncc2C1)NCc1ccc(F)cc1 ZINC000880594022 DD On-Demand Anodyne PLA2G7 17 41 O=C(CN1CCc2ncncc2C1)NCc1ccc(F)cc1 ZINC000880594022 DD On-Demand Anodyne SLC27A1 52 37 CCCOc1cccc(CNC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594025 ED On-Demand Anodyne HRH2 35 42 CCCOc1cccc(CNC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594025 ED On-Demand Anodyne PDS 42 32 O=C(CN1CCc2ncncc2C1)N1CCc2cc([N+](=O)[O-])ccc21 ZINC000880594036 ED On-Demand Bother EIF2AK3 56 33 N#Cc1c(NC(=O)CN2CCc3ncncc3C2)sc2c1CCCCC2 ZINC000880594044 FF On-Demand Mild VIPR1 31 51 COC(=O)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594052 ED On-Demand Anodyne FLT4 22 42 COC(=O)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594052 ED On-Demand Anodyne P2RY14 49 38 O=C(CN1CCc2ncncc2C1)NCCOc1cccc(C(F)(F)F)c1 ZINC000880594058 GE On-Demand Anodyne HRH2 28 44 O=C(CN1CCc2ncncc2C1)NCCOc1cccc(C(F)(F)F)c1 ZINC000880594058 GE On-Demand Anodyne GALR3 52 37 O=C(CN1CCc2ncncc2C1)NCCOc1cccc(C(F)(F)F)c1 ZINC000880594058 GE On-Demand Anodyne PDS 42 41 O=C(CN1CCc2ncncc2C1)Nc1ccccc1Cl ZINC000880594059 DE On-Demand Anodyne EPHB3 58 37 COCC1CN(C(=O)CC[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880594060 FG On-Demand Anodyne CTSK 16 44 COCC1CN(C(=O)CC[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880594060 FG On-Demand Anodyne FPR1 44 35 Fc1ccc(CN2CCc3ncncc3C2)c(Cl)c1 ZINC000880594066 CF On-Demand Anodyne P2RX7 48 42 COCC1CN(C(=O)c2cn(C)c3ccccc23)C1 ZINC000880594068 CD On-Demand Anodyne CNR1 21 45 COCC1CN(C(=O)c2cn(C)c3ccccc23)C1 ZINC000880594068 CD On-Demand Anodyne HTR4 25 46 COCC1CN(C(=O)c2cn(C)c3ccccc23)C1 ZINC000880594068 CD On-Demand Anodyne CNR2 21 41 COCC1CN(C(=O)c2cn(C)c3ccccc23)C1 ZINC000880594068 CD On-Demand Anodyne TPSAB1 20 48 O=C(CN1CCc2ncncc2C1)N1CCC(Cc2ccccc2)CC1 ZINC000880594077 FE On-Demand Anodyne GRIN2B 82 44 O=C(CN1CCc2ncncc2C1)N1CCC(Cc2ccccc2)CC1 ZINC000880594077 FE On-Demand Anodyne SIGMAR1 17 42 O=C(CN1CCc2ncncc2C1)N1CCC(Cc2ccccc2)CC1 ZINC000880594077 FE On-Demand Anodyne CCR3 25 40 CC(=O)Nc1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880594093 ED On-Demand Anodyne P2RY14 47 37 C[C@H](C(=O)Nc1ccccc1Cl)N1CCc2ncncc2C1 ZINC000880594099 DF On-Demand Anodyne EPHB3 56 35 O=C(CN1CCc2ncncc2C1)Nc1ccc2c(c1)OCCO2 ZINC000880594103 ED On-Demand Anodyne IMDH_CRYPV 19 47 CCOC(=O)N1CCC(NC(=O)CN2CCc3ncncc3C2)CC1 ZINC000880594105 EC On-Demand Anodyne CCR8 29 42 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)c(Cl)c1 ZINC000880594108 FG On-Demand Anodyne MAPK1 50 47 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(Cl)c(Cl)c1 ZINC000880594110 FG On-Demand Anodyne MAPK1 50 47 COCC1CN(C(=O)[C@@H]2CC(c3ccccc3)=NO2)C1 ZINC000880594122 CD On-Demand Anodyne LUCI_PHOPY 68 38 COCC1CN(C(=O)[C@H]2CC(c3ccccc3)=NO2)C1 ZINC000880594123 CD On-Demand Anodyne LUCI_PHOPY 68 38 O=C(CCN1CCc2ncncc2C1)N1CCc2ccccc21 ZINC000880594126 DD On-Demand Anodyne HTR7 17 42 O=C(CCN1CCc2ncncc2C1)N1CCc2ccccc21 ZINC000880594126 DD On-Demand Anodyne EIF2AK3 48 32 COCC1CN(C(=O)c2c(C)oc3ccc(OC)cc23)C1 ZINC000880594129 CE On-Demand Anodyne SLC22A12 39 43 O[C@H](COc1ccccc1)CN1CCc2ncncc2C1 ZINC000880594134 CD On-Demand Anodyne ACOX1 46 34 O[C@H](COc1ccccc1)CN1CCc2ncncc2C1 ZINC000880594134 CD On-Demand Anodyne ABCB1 62 40 O[C@@H](COc1ccccc1)CN1CCc2ncncc2C1 ZINC000880594135 CD On-Demand Anodyne ACOX1 46 34 O[C@@H](COc1ccccc1)CN1CCc2ncncc2C1 ZINC000880594135 CD On-Demand Anodyne ABCB1 62 40 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880594153 EE On-Demand Anodyne KIT 17 41 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880594153 EE On-Demand Anodyne KDR 19 46 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880594153 EE On-Demand Anodyne EPHX2 16 42 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880594153 EE On-Demand Anodyne RIPK1 46 40 N#Cc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880594155 CD On-Demand Mild HRH3 17 43 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1 ZINC000880594157 FF On-Demand Clean PDGFRB 49 39 O[C@H](COc1ccc(F)cc1)CN1CCc2ncncc2C1 ZINC000880594164 DD On-Demand Anodyne ACOX1 49 36 O[C@H](COc1ccc(F)cc1)CN1CCc2ncncc2C1 ZINC000880594164 DD On-Demand Anodyne ABCB1 42 46 O[C@@H](COc1ccc(F)cc1)CN1CCc2ncncc2C1 ZINC000880594166 DD On-Demand Anodyne ACOX1 49 36 O[C@@H](COc1ccc(F)cc1)CN1CCc2ncncc2C1 ZINC000880594166 DD On-Demand Anodyne ABCB1 42 46 CN(C)Cc1ccnc(NC(=O)N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)c1 ZINC000880594169 GE On-Demand Bother SSTR1 43 44 CCOC(=O)N1CCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880594202 ED On-Demand Anodyne P2RY12 49 37 Cc1ccc(N2CCCN(C(=O)Nc3cc(S(C)(=O)=O)ccn3)CC2)cc1 ZINC000880594206 GF On-Demand Anodyne SLC6A9 19 40 CN(C)C(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594209 CD On-Demand Anodyne NOD2 40 35 O=C(CCN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880594225 FD On-Demand Anodyne HTR7 21 41 O=C(CCN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880594225 FD On-Demand Anodyne SSTR1 34 43 O=C(CCN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880594225 FD On-Demand Anodyne SLC27A1 41 35 CS(=O)(=O)c1ccnc(NC(=O)NC2CCCCCCC2)c1 ZINC000880594227 EF On-Demand Anodyne EPHX2 48 46 NC(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594243 CD On-Demand Anodyne NOD1 18 41 NC(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594243 CD On-Demand Anodyne NOD2 47 40 CN(C)Cc1ccnc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)c1 ZINC000880594267 GF On-Demand Anodyne L3MBTL3 56 35 CN(C)Cc1ccnc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)c1 ZINC000880594267 GF On-Demand Anodyne NAMPT 24 48 CS(=O)(=O)c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880594286 ED On-Demand Anodyne HTR7 16 42 CS(=O)(=O)c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880594286 ED On-Demand Anodyne HRH3 64 43 CS(=O)(=O)c1ccc(OCCCN2CCc3ncncc3C2)cc1 ZINC000880594286 ED On-Demand Anodyne HTR5A 26 45 c1ncc2c(n1)CCN(Cc1csc(-c3ccc4c(c3)OCO4)n1)C2 ZINC000880594289 FF On-Demand Anodyne CLK2 44 38 c1ncc2c(n1)CCN(Cc1csc(-c3ccc4c(c3)OCO4)n1)C2 ZINC000880594289 FF On-Demand Anodyne CLK4 70 38 COCC1CN(C(=O)CC[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880594295 FG On-Demand Anodyne CTSK 16 44 COCC1CN(C(=O)CC[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880594295 FG On-Demand Anodyne FPR1 44 35 COCC1CN(C(=O)[C@@H]2C[C@@H](O)CN2C(=O)OCc2ccccc2)C1 ZINC000880594302 EC On-Demand Anodyne PREP 52 48 COCC1CN(C(=O)[C@@H]2C[C@@H](O)CN2C(=O)OCc2ccccc2)C1 ZINC000880594302 EC On-Demand Anodyne SLC12A5 46 35 COCC1CN(C(=O)[C@@H]2C[C@@H](O)CN2C(=O)OCc2ccccc2)C1 ZINC000880594302 EC On-Demand Anodyne Q9NAW4_PLAFA 33 52 COc1ccc(NC(=O)[C@H](C)N2CCc3ncncc3C2)cc1OC ZINC000880594304 ED On-Demand Anodyne ENPP1 74 42 COCC1CN(C(=O)Cc2c[nH]c3cc(F)ccc23)C1 ZINC000880594309 CD On-Demand Anodyne MPO 77 36 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594312 DE On-Demand Anodyne CTSD 16 42 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594312 DE On-Demand Anodyne CTSK 15 43 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594312 DE On-Demand Anodyne ECE1 37 42 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594312 DE On-Demand Anodyne POLG_HCV1 23 43 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594314 DE On-Demand Anodyne CTSD 16 42 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594314 DE On-Demand Anodyne CTSK 15 43 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594314 DE On-Demand Anodyne ECE1 37 42 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594314 DE On-Demand Anodyne POLG_HCV1 23 43 CS(=O)(=O)c1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880594330 ED On-Demand Anodyne NR1H3 42 34 N#Cc1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880594341 CE On-Demand Mild HRH3 42 44 N#Cc1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880594341 CE On-Demand Mild HTR5A 25 44 N#Cc1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880594341 CE On-Demand Mild MEN1 41 36 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880594366 FD On-Demand Anodyne PIK3CA 42 38 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880594366 FD On-Demand Anodyne MAPKAPK5 40 34 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880594366 FD On-Demand Anodyne MTOR 84 38 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880594366 FD On-Demand Anodyne STAT6 66 36 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880594366 FD On-Demand Anodyne SLC27A1 41 39 CS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880594380 ED On-Demand Anodyne LTA4H 44 37 CS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880594380 ED On-Demand Anodyne HRH3 25 40 CS(=O)(=O)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880594380 ED On-Demand Anodyne HTR5A 22 40 O=C(CN1CCc2ncncc2C1)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880594392 FD On-Demand Anodyne DRD4 28 42 O=C(CN1CCc2ncncc2C1)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880594392 FD On-Demand Anodyne SSTR5 41 35 O=C(CN1CCc2ncncc2C1)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880594392 FD On-Demand Anodyne MCHR1 16 42 O=C(CN1CCc2ncncc2C1)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880594392 FD On-Demand Anodyne HPGDS 45 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCC(F)(F)F)C1 ZINC000880594395 DD On-Demand Anodyne PREP 46 44 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCC(F)(F)F)C1 ZINC000880594395 DD On-Demand Anodyne WNT3 40 33 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCC(F)(F)F)C1 ZINC000880594396 DD On-Demand Anodyne PREP 46 44 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCC(F)(F)F)C1 ZINC000880594396 DD On-Demand Anodyne WNT3 40 33 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne HTR1D 22 44 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne HTR1B 16 41 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne CCR3 16 40 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne MCHR1 32 41 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne P2RY14 54 43 CC(=O)Nc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880594405 CD On-Demand Anodyne NOD2 45 39 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccccc2F)CC1 ZINC000880594410 FD On-Demand Anodyne HTR1A 16 40 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccccc2F)CC1 ZINC000880594410 FD On-Demand Anodyne HTR7 15 40 COCC1CN(C(=O)c2cc3c(Cl)c(Cl)ccc3[nH]2)C1 ZINC000880594431 DG On-Demand Anodyne HRH4 25 61 CN(C)Cc1ccnc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)c1 ZINC000880594433 FG On-Demand Anodyne TYK2 22 41 CN(C)Cc1ccnc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)c1 ZINC000880594434 FG On-Demand Anodyne TYK2 22 41 COc1ccc(-c2cnc(CN3CCc4ncncc4C3)o2)cc1 ZINC000880594436 DF On-Demand Anodyne ABCB1 15 41 c1ccc2c(CCCN3CCc4ncncc4C3)cccc2c1 ZINC000880594446 DH On-Demand Anodyne SIGMAR1 16 47 c1ccc2c(CCCN3CCc4ncncc4C3)cccc2c1 ZINC000880594446 DH On-Demand Anodyne EBP 41 40 COCC1CN(C(=O)Cc2csc(-c3ccc(Cl)cc3Cl)n2)C1 ZINC000880594448 FH On-Demand Anodyne ALPL 45 38 COCC1CN(C(=O)Cc2csc(-c3ccc(Cl)cc3Cl)n2)C1 ZINC000880594448 FH On-Demand Anodyne DPP8 68 36 COCC1CN(C(=O)Cc2csc(-c3ccc(Cl)cc3Cl)n2)C1 ZINC000880594448 FH On-Demand Anodyne DPP9 66 36 O[C@H](COc1ccc(Br)cc1)CN1CCc2ncncc2C1 ZINC000880594461 FE On-Demand Anodyne ACOX1 55 33 O[C@@H](COc1ccc(Br)cc1)CN1CCc2ncncc2C1 ZINC000880594462 FE On-Demand Anodyne ACOX1 55 33 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne LTA4H 53 38 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne HRH3 31 40 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne SIGMAR1 15 40 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne BCHE 17 41 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne HTR5A 25 50 c1ccc2cc(OCCN3CCc4ncncc4C3)ccc2c1 ZINC000880594463 DG On-Demand Anodyne ABCB1 15 45 COCC1CN(C(=O)c2cc(-c3ccc(C)cc3)nc3c2cnn3C(C)C)C1 ZINC000880594467 GH On-Demand Anodyne EZH2 16 43 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594476 CD On-Demand Anodyne ABCG2 37 45 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594476 CD On-Demand Anodyne NOD1 20 46 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594476 CD On-Demand Anodyne NOD2 54 46 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCc2ncncc2C1 ZINC000880594489 DD On-Demand Anodyne DRD4 31 53 C[C@@H]1Cc2ccccc2N1C(=O)CN1CCc2ncncc2C1 ZINC000880594489 DD On-Demand Anodyne TPP2 58 35 O=C(CN1CCc2ncncc2C1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880594493 FD On-Demand Anodyne HTR1A 30 45 O=C(CN1CCc2ncncc2C1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880594493 FD On-Demand Anodyne HTR2A 24 45 O=C(CN1CCc2ncncc2C1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880594493 FD On-Demand Anodyne DRD3 18 45 O=C(CN1CCc2ncncc2C1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880594493 FD On-Demand Anodyne HTR7 32 45 O=C(CN1CCc2ncncc2C1)N1CCN(c2cccc(Cl)c2)CC1 ZINC000880594493 FD On-Demand Anodyne MAPK1 22 46 C[C@H](Cc1ccccc1Cl)NC(=O)Nc1cc(S(C)(=O)=O)ccn1 ZINC000880594498 FF On-Demand Anodyne TYK2 42 38 C[C@@H](Cc1ccccc1Cl)NC(=O)Nc1cc(S(C)(=O)=O)ccn1 ZINC000880594499 FF On-Demand Anodyne TYK2 42 38 CC(=O)c1ccc(N2CCN(C(=O)CN3CCc4ncncc4C3)CC2)c(F)c1 ZINC000880594510 GD On-Demand Anodyne SLC6A9 16 42 O=C(Nc1ccccc1)C1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880594511 GD On-Demand Anodyne MAPK1 21 40 COCC1CN(C(=O)CNC(=O)c2ccc(Cl)c(Cl)c2)C1 ZINC000880594526 ED On-Demand Anodyne UTS2R 23 41 COCC1CN(C(=O)CNC(=O)c2ccc(Cl)c(Cl)c2)C1 ZINC000880594526 ED On-Demand Anodyne CACNA1I 64 49 CCOc1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594559 DD On-Demand Anodyne HCN1 47 32 COCC1CN(C(=O)C[C@H]2c3ccccc3CCN2C(C)=O)C1 ZINC000880594588 DD On-Demand Anodyne MTNR1B 15 56 COCC1CN(C(=O)C[C@@H]2c3ccccc3CCN2C(C)=O)C1 ZINC000880594590 DD On-Demand Anodyne MTNR1B 15 56 O=C(CN1CCc2ncncc2C1)NCCc1ccc(Cl)cc1 ZINC000880594592 ED On-Demand Anodyne SCN10A 22 40 O=C(CN1CCc2ncncc2C1)NCCc1ccc(Cl)cc1 ZINC000880594592 ED On-Demand Anodyne MRGPRX1 40 35 O=C(CCN1CCc2ncncc2C1)N[C@H]1CCCc2ccccc21 ZINC000880594601 EE On-Demand Anodyne HTR7 23 56 O=C(CCN1CCc2ncncc2C1)N[C@H]1CCCc2ccccc21 ZINC000880594601 EE On-Demand Anodyne BDKRB1 56 41 O=C(CCN1CCc2ncncc2C1)N[C@@H]1CCCc2ccccc21 ZINC000880594603 EE On-Demand Anodyne HTR7 23 56 O=C(CCN1CCc2ncncc2C1)N[C@@H]1CCCc2ccccc21 ZINC000880594603 EE On-Demand Anodyne BDKRB1 56 41 O=C(CN1CCc2ncncc2C1)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880594609 GD On-Demand Anodyne NAMPT 35 41 COc1cc(CNC(=O)CN2CCc3ncncc3C2)cc(OC)c1OC ZINC000880594613 FD On-Demand Anodyne ABCB1B 47 35 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1Cl ZINC000880594633 DF On-Demand Anodyne EPHB3 56 36 O=C(CN1CCc2ncncc2C1)Nc1ccc2c(c1)CCC2 ZINC000880594634 DD On-Demand Anodyne ACOX1 22 43 O=C(CN1CCc2ncncc2C1)Nc1ccc2c(c1)CCC2 ZINC000880594634 DD On-Demand Anodyne NOD1 18 40 C[C@H](C(=O)Nc1cccc(Cl)c1)N1CCc2ncncc2C1 ZINC000880594638 DF On-Demand Anodyne P2RY14 34 40 COc1ccc(-c2noc(CN3CCc4ncncc4C3)n2)c(OC)c1 ZINC000880594659 FE On-Demand Anodyne ABCB1 17 41 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880594662 FE On-Demand Anodyne PDGFRB 24 42 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880594662 FE On-Demand Anodyne MTNR1A 15 41 CC(=O)c1cccc(NC(=O)[C@@H](C)N2CCc3ncncc3C2)c1 ZINC000880594664 DE On-Demand Anodyne P2RY14 40 35 CC(=O)c1cccc(NC(=O)[C@H](C)N2CCc3ncncc3C2)c1 ZINC000880594665 DE On-Demand Anodyne P2RY14 40 35 O=C(CN1CCc2ncncc2C1)NC(=O)NC12CC3CC(CC(C3)C1)C2 ZINC000880594672 FD On-Demand Anodyne EPHX2 79 45 COCC1CN(C(=O)CNc2cccc(C(F)(F)F)c2)C1 ZINC000880594693 DE On-Demand Anodyne CACNA1B 47 34 COCC1CN(C(=O)CNc2cccc(C(F)(F)F)c2)C1 ZINC000880594693 DE On-Demand Anodyne CCR2 78 40 COCC1CN(C(=O)CNc2cccc(C(F)(F)F)c2)C1 ZINC000880594693 DE On-Demand Anodyne EPHX2 15 47 COCC1CN(C(=O)CNc2cccc(C(F)(F)F)c2)C1 ZINC000880594693 DE On-Demand Anodyne PDS 41 36 O=C(CN1CCc2ncncc2C1)NNC(=O)c1ccc(F)cc1 ZINC000880594695 EC On-Demand Reactive SLC27A1 42 34 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594697 DD On-Demand Anodyne PAPA1_CARPA 34 50 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880594697 DD On-Demand Anodyne CTSK 20 44 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880594727 FG On-Demand Anodyne ABL1 41 38 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880594727 FG On-Demand Anodyne RAF1 28 40 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880594727 FG On-Demand Anodyne MCHR1 16 42 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880594727 FG On-Demand Anodyne BRAF 16 42 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880594727 FG On-Demand Anodyne IMDH_CRYPV 32 43 O=C(CN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880594734 DD On-Demand Anodyne NOS2 69 33 O=C(CN1CCc2ncncc2C1)Nc1ccc2c(c1)OCO2 ZINC000880594734 DD On-Demand Anodyne IMDH_CRYPV 17 41 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(OC(F)(F)F)cc1 ZINC000880594736 GF On-Demand Anodyne PTGER4 15 43 C[C@@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(OC(F)(F)F)cc1 ZINC000880594736 GF On-Demand Anodyne P2RY1 20 41 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(OC(F)(F)F)cc1 ZINC000880594737 GF On-Demand Anodyne PTGER4 15 43 C[C@H](NC(=O)CN1CCc2ncncc2C1)c1ccc(OC(F)(F)F)cc1 ZINC000880594737 GF On-Demand Anodyne P2RY1 20 41 N#Cc1ccsc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594743 CD On-Demand Mild MAPK9 16 40 N#Cc1ccsc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594743 CD On-Demand Mild MAPK10 20 40 N#Cc1ccsc1NC(=O)CN1CCc2ncncc2C1 ZINC000880594743 CD On-Demand Mild MAPK8 23 40 CCC(=O)N1CSC[C@H]1C(=O)N1CC(COC)C1 ZINC000880594751 CC On-Demand Anodyne PREP 18 41 CCC(=O)N1CSC[C@@H]1C(=O)N1CC(COC)C1 ZINC000880594752 CC On-Demand Anodyne PREP 18 41 COCC1CN(C(=O)COc2cccnc2)C1 ZINC000880594756 BC On-Demand Anodyne CHRNA7 29 41 COCC1CN(C(=O)COc2cccnc2)C1 ZINC000880594756 BC On-Demand Anodyne CPT1A 74 40 O=C(CN1CCc2ncncc2C1)Nc1ccc(I)cc1 ZINC000880594758 GE On-Demand Anodyne NOD2 40 34 COCCCS(=O)(=O)NCCN1CCc2ncncc2C1 ZINC000880594760 DB On-Demand Anodyne HTR7 15 42 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne ACE 24 41 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne KLK3 70 34 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CTSB 59 45 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne PAPA1_CARPA 47 38 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CYSP_TRYCR 50 38 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CTSK 41 45 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CTSL 45 43 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne PREP 23 53 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CAPNS1 62 35 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CAPN1 76 40 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne CAPN2 124 40 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne TGM2 38 40 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne NPR 75 39 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne F13A1 24 40 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne NAAA 22 40 COCC1CN(C(=O)CNC(=O)OCc2ccccc2)C1 ZINC000880594781 CD On-Demand Anodyne SLC12A5 52 36 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne DRD2 15 45 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne LTA4H 45 40 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne HRH3 48 51 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne SIGMAR1 26 41 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne HTR5A 37 49 c1ccc(OCCCCN2CCc3ncncc3C2)cc1 ZINC000880594793 CF On-Demand Anodyne ABCB1 19 45 CN(C(=O)c1cccs1)c1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880594812 IK On-Demand Mild KCNK3 52 38 CN(C(=O)c1cccs1)c1ccccc1C(=O)Nc1cccc(C#Cc2ccccn2)c1 ZINC000880594812 IK On-Demand Mild KCNK9 46 38 COCC1CN(C(=O)c2cccnc2Nc2ccc(Cl)c(Cl)c2)C1 ZINC000880594814 FH On-Demand Anodyne PTK6 48 36 CN(C)Cc1ccnc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)c1 ZINC000880594831 GF On-Demand Clean EPHB4 81 36 COCC1CN(C(=O)c2cc3ccc(OCc4ccccc4)cc3[nH]2)C1 ZINC000880594836 FG On-Demand Anodyne GRIN2B 41 52 COCC1CN(C(=O)c2cc3ccc(OCc4ccccc4)cc3[nH]2)C1 ZINC000880594836 FG On-Demand Anodyne HRH4 18 41 COCC1CN(C(=O)c2cc3ccc(OCc4ccccc4)cc3[nH]2)C1 ZINC000880594836 FG On-Demand Anodyne AKR1C3 17 40 COc1cccc(OC)c1OC[C@@H](O)CN1CCc2ncncc2C1 ZINC000880594855 ED On-Demand Anodyne ABCB1 77 38 COc1cccc(OC)c1OC[C@H](O)CN1CCc2ncncc2C1 ZINC000880594856 ED On-Demand Anodyne ABCB1 77 38 O=C(CN1CCc2ncncc2C1)NCCOc1cccc(Cl)c1 ZINC000880594857 ED On-Demand Anodyne HRH2 34 41 O=C(CN1CCc2ncncc2C1)NCCOc1cccc(Cl)c1 ZINC000880594857 ED On-Demand Anodyne AVPR1B 41 39 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)c1 ZINC000880594860 EF On-Demand Anodyne ADRB1 32 41 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)c1 ZINC000880594860 EF On-Demand Anodyne ADRB3 46 41 O=C(CN1CCc2ncncc2C1)NC1C2CC3CC(C2)CC1C3 ZINC000880594861 ED On-Demand Anodyne HSD11B1 40 30 CCOc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594870 ED On-Demand Anodyne ACOX1 65 34 CCOc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594870 ED On-Demand Anodyne ABCB1 41 39 CCOc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594871 ED On-Demand Anodyne ACOX1 65 34 CCOc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594871 ED On-Demand Anodyne ABCB1 41 39 CCCCCNC(=O)CN1CCc2ncncc2C1 ZINC000880594878 CD On-Demand Anodyne ASAH1 58 30 COC(=O)C1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880594894 DC On-Demand Anodyne PTR1 46 33 O=C(CN1CCc2ncncc2C1)N(Cc1ccccc1)Cc1ccco1 ZINC000880594896 FF On-Demand Anodyne MRGPRX1 30 45 Cc1ccc(OC[C@@H](C)NC(=O)Nc2cc(S(C)(=O)=O)ccn2)cc1 ZINC000880594898 FE On-Demand Anodyne GCK 19 40 Cc1ccc(OC[C@H](C)NC(=O)Nc2cc(S(C)(=O)=O)ccn2)cc1 ZINC000880594899 FE On-Demand Anodyne GCK 19 40 FC(F)(F)Oc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594923 DF On-Demand Anodyne NOD1 15 49 FC(F)(F)Oc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880594923 DF On-Demand Anodyne NOD2 43 49 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1CC(=O)NC1CCN(C)CC1 ZINC000880594928 EF On-Demand Anodyne SIGMAR1 20 44 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1CC(=O)NC1CCN(C)CC1 ZINC000880594928 EF On-Demand Anodyne EPHX2 18 41 COCC1CN(C(=O)c2ccc(Oc3ccc(C(F)(F)F)cn3)cc2)C1 ZINC000880594930 FH On-Demand Anodyne LIPE 28 55 CCOC(=O)[C@@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880594931 EC On-Demand Anodyne FKBP1A 43 37 CCOC(=O)[C@@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880594931 EC On-Demand Anodyne CPT1A 63 40 CCOC(=O)[C@@H]1CCCCN1C(=O)CN1CCc2ncncc2C1 ZINC000880594931 EC On-Demand Anodyne CPT2 47 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne F2 53 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne PLG 51 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne ACE 102 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne OPRM1 51 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne OPRD1 44 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne GHRHR 58 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne P2RY12 121 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne MME 115 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne ANPEP 45 33 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne TACR1 22 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne MC4R 72 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne FCER2 72 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CTSB 48 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne TRY2_BOVIN 99 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne PAPA1_CARPA 61 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne TRY1_BOVIN 48 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CYSP_TRYCR 58 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CTSK 28 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CTSL 60 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne NPFFR2 72 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne TIMP3 73 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CAPNS1 77 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne MMP3 24 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne HLA-DRB1 60 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CELA2A 41 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne REN 47 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CTSS 26 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CAPN1 83 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CAPN2 51 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne ACE2 84 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne ST14 105 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne MMP1 29 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne FPR1 58 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne CTRB_BOVIN 56 33 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne GAG-PRO 49 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne BLA1_STEMA 55 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne BRCA1 43 30 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594934 CC On-Demand Anodyne NPFFR1 71 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne F2 53 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne PLG 51 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne ACE 102 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne OPRM1 51 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne OPRD1 44 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne GHRHR 58 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne P2RY12 121 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne MME 115 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne ANPEP 45 33 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne TACR1 22 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne MC4R 72 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne FCER2 72 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CTSB 48 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne TRY2_BOVIN 99 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne PAPA1_CARPA 61 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne TRY1_BOVIN 48 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CYSP_TRYCR 58 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CTSK 28 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CTSL 60 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne NPFFR2 72 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne TIMP3 73 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CAPNS1 77 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne MMP3 24 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne HLA-DRB1 60 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CELA2A 41 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne REN 47 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CTSS 26 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CAPN1 83 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CAPN2 51 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne ACE2 84 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne ST14 105 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne MMP1 29 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne FPR1 58 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne CTRB_BOVIN 56 33 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne GAG-PRO 49 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne BLA1_STEMA 55 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne BRCA1 43 30 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C1 ZINC000880594937 CC On-Demand Anodyne NPFFR1 71 35 O=C(CN1CCc2ncncc2C1)N[C@@H]1CCCc2ccccc21 ZINC000880594953 DE On-Demand Anodyne HTR7 16 51 O=C(CN1CCc2ncncc2C1)N[C@@H]1CCCc2ccccc21 ZINC000880594953 DE On-Demand Anodyne BDKRB1 63 40 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)C1 ZINC000880594954 DD On-Demand Anodyne PREP 18 47 O=C(CN1CCc2ncncc2C1)N[C@H]1CCCc2ccccc21 ZINC000880594955 DE On-Demand Anodyne HTR7 16 51 O=C(CN1CCc2ncncc2C1)N[C@H]1CCCc2ccccc21 ZINC000880594955 DE On-Demand Anodyne BDKRB1 63 40 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OC(C)(C)C)C2)C1 ZINC000880594956 DD On-Demand Anodyne PREP 18 47 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne ADRB2 15 46 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne ADRB1 35 46 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne ADRB3 25 40 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne ACOX1 62 41 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne ABCB1 51 38 CC(=O)Nc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594957 ED On-Demand Anodyne NOD2 40 38 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne ADRB2 15 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne ADRB1 35 46 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne ADRB3 25 40 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne ACOX1 62 41 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne ABCB1 51 38 CC(=O)Nc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880594959 ED On-Demand Anodyne NOD2 40 38 C[C@H]1CCc2ccccc2N1C(=O)CN1CCc2ncncc2C1 ZINC000880594960 DE On-Demand Anodyne DRD4 26 43 COCC1CN(C(=O)c2cc([N+](=O)[O-])ccc2I)C1 ZINC000880594969 GD On-Demand Bother CACNA1D 44 35 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(Cl)c1 ZINC000880594974 EF On-Demand Anodyne IMDH_CRYPV 37 42 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)c1 ZINC000880594977 EF On-Demand Anodyne ADRB1 32 41 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)c1 ZINC000880594977 EF On-Demand Anodyne ADRB3 46 41 c1ncc2c(n1)CCN(CCCOc1ccc3c(c1)OCO3)C2 ZINC000880594981 DE On-Demand Anodyne HRH3 36 49 c1ncc2c(n1)CCN(CCCOc1ccc3c(c1)OCO3)C2 ZINC000880594981 DE On-Demand Anodyne HTR5A 23 42 CC(=O)c1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(F)c1 ZINC000880594984 GF On-Demand Anodyne NPY2R 71 38 CC(=O)c1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(F)c1 ZINC000880594984 GF On-Demand Anodyne SLC6A9 15 41 O=C(CN1CCc2ncncc2C1)OCc1ccccc1 ZINC000880595004 CD On-Demand Anodyne CHRM5 15 40 c1ncc2c(n1)CCN(CCN1CCCCC1)C2 ZINC000880595023 BD On-Demand Anodyne HRH3 25 43 c1ncc2c(n1)CCN(CCN1CCCCC1)C2 ZINC000880595023 BD On-Demand Anodyne HNMT 54 32 C[C@H](C(=O)Nc1ccccc1C(F)(F)F)N1CCc2ncncc2C1 ZINC000880595048 FF On-Demand Anodyne RBP4 43 31 O=C(CN1CCc2ncncc2C1)Nc1cc(F)ccc1F ZINC000880595052 DD On-Demand Anodyne SLC27A1 55 40 FC(F)(F)COc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880595058 DF On-Demand Anodyne NOD2 40 37 COCC1CN(C(=O)C[C@H](NC(N)=O)c2ccccc2C)C1 ZINC000880595062 DD On-Demand Anodyne CTSA 61 39 COCC1CN(C(=O)C[C@@H](NC(N)=O)c2ccccc2C)C1 ZINC000880595075 DD On-Demand Anodyne CTSA 61 39 c1ncc2c(n1)CCN(Cc1nc(-c3ccc4c(c3)OCO4)no1)C2 ZINC000880595089 ED On-Demand Anodyne CLK4 60 37 CC(=O)c1ccc(NC(=O)CN2CCc3ncncc3C2)cc1 ZINC000880595103 DD On-Demand Anodyne PRNP 46 36 CC(=O)c1ccc(NC(=O)CN2CCc3ncncc3C2)cc1 ZINC000880595103 DD On-Demand Anodyne NOD2 43 37 O=C(CN1CCc2ncncc2C1)Nc1cccc(Cl)c1 ZINC000880595104 DE On-Demand Anodyne IMDH_CRYPV 31 41 COCC1CN(C(=O)c2ccc(CN3CCN(C)CC3)cc2)C1 ZINC000880595122 DD On-Demand Anodyne HRH3 15 44 COCC1CN(C(=O)c2ccc(CN3CCN(C)CC3)cc2)C1 ZINC000880595122 DD On-Demand Anodyne SIGMAR1 25 42 COCC1CN(C(=O)c2ccc(CN3CCN(C)CC3)cc2)C1 ZINC000880595122 DD On-Demand Anodyne LSS 15 46 COCC1CN(C(=O)c2ccc(CN3CCN(C)CC3)cc2)C1 ZINC000880595122 DD On-Demand Anodyne L3MBTL3 36 45 Cc1c(NC(=O)[C@H](C)N2CCc3ncncc3C2)c(=O)n(-c2ccccc2)n1C ZINC000880595127 GD On-Demand Anodyne FPR2 59 43 Cc1c(NC(=O)[C@@H](C)N2CCc3ncncc3C2)c(=O)n(-c2ccccc2)n1C ZINC000880595130 GD On-Demand Anodyne FPR2 59 43 CCOC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880595144 ED On-Demand Anodyne GRIN2B 22 42 CCOC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880595144 ED On-Demand Anodyne SSTR5 54 38 CCOC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880595144 ED On-Demand Anodyne EPHX2 41 42 CCOC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880595144 ED On-Demand Anodyne CCR8 23 41 CC(C)(C)OC(=O)N1CC[C@H](CN2CCc3ncncc3C2)C1 ZINC000880595145 DE On-Demand Anodyne GPR119 46 42 CC(C)(C)OC(=O)N1CC[C@@H](CN2CCc3ncncc3C2)C1 ZINC000880595148 DE On-Demand Anodyne GPR119 46 42 Fc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880595158 CE On-Demand Anodyne LTA4H 28 41 Fc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880595158 CE On-Demand Anodyne HTR5A 23 46 CC(C)(C)OC(=O)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880595164 EE On-Demand Anodyne GPR119 50 45 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCCC2)cc1 ZINC000880595184 EE On-Demand Anodyne SLC27A1 43 40 O=C(CN1CCc2ncncc2C1)NNC(=O)c1cccc(Cl)c1 ZINC000880595186 EC On-Demand Reactive LUCI_LUCLA 16 41 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCCCCC2)cc1 ZINC000880595197 FF On-Demand Anodyne SLC27A1 43 39 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880595200 GD On-Demand Bother SSTR1 46 45 Fc1ccc(CCN2CCc3ncncc3C2)cc1F ZINC000880595213 CE On-Demand Anodyne ABCC1 106 42 Fc1ccc(CCN2CCc3ncncc3C2)cc1F ZINC000880595213 CE On-Demand Anodyne ABCB1A 51 36 COCC1CN(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 ZINC000880595223 DG On-Demand Anodyne OPRK1 22 42 COC(=O)c1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880595228 ED On-Demand Anodyne ACOX1 57 37 COC(=O)c1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880595228 ED On-Demand Anodyne ABCB1 53 42 COC(=O)c1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880595229 ED On-Demand Anodyne ACOX1 57 37 COC(=O)c1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880595229 ED On-Demand Anodyne ABCB1 53 42 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne LTA4H 57 40 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne HRH3 37 40 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne HTR5A 25 44 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne CACNA2D2 40 31 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne PSMB2 40 36 CCOc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595233 CE On-Demand Anodyne PSMB1 43 37 COCC1CN(C(=O)/C=C(/C)c2ccccc2OC)C1 ZINC000880595238 CE On-Demand Anodyne KCNA3 43 39 COCC1CN(C(=O)/C=C(\C)c2ccccc2OC)C1 ZINC000880595239 CE On-Demand Anodyne KCNA3 43 39 CCN1CC[C@H](CNC(=O)Nc2cc(CN(C)C)ccn2)C1 ZINC000880595256 DD On-Demand Anodyne CACNA1I 56 34 N#Cc1ccc(NC(=O)CN2CCc3ncncc3C2)cc1Cl ZINC000880595258 ED On-Demand Mild IMDH_CRYPV 21 43 c1ncc2c(n1)CCN(CCc1ccc3c(c1)CCO3)C2 ZINC000880595286 CE On-Demand Anodyne KCNJ1 49 39 CSc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595289 DF On-Demand Anodyne LTA4H 50 39 CSc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595289 DF On-Demand Anodyne HTR5A 23 45 CSc1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595289 DF On-Demand Anodyne PSMB1 41 35 COc1cc(CN2CCc3ncncc3C2)ccc1SC ZINC000880595303 DF On-Demand Anodyne ABCB1 19 42 Ic1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880595308 FF On-Demand Anodyne NOD2 40 34 O=S(=O)(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880595313 DD On-Demand Anodyne HTR7 15 46 c1ccc2c(OCCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595324 DG On-Demand Anodyne HTR5A 39 57 c1ccc2c(OCCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595324 DG On-Demand Anodyne ABCB1B 40 32 c1ccc2c(OCCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595324 DG On-Demand Anodyne ABCB1 19 41 c1ccc2c(OCCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595324 DG On-Demand Anodyne MCL1 38 42 O=S(=O)(NCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880595327 DC On-Demand Anodyne HTR7 44 64 O=S(=O)(NCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880595327 DC On-Demand Anodyne HTR6 20 51 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCc2ncncc2C1 ZINC000880595342 FE On-Demand Anodyne ACOX1 66 35 O[C@H](COc1cccc(C(F)(F)F)c1)CN1CCc2ncncc2C1 ZINC000880595342 FE On-Demand Anodyne PDS 41 36 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCc2ncncc2C1 ZINC000880595343 FE On-Demand Anodyne ACOX1 66 35 O[C@@H](COc1cccc(C(F)(F)F)c1)CN1CCc2ncncc2C1 ZINC000880595343 FE On-Demand Anodyne PDS 41 36 COCC1CN(C(=O)Cn2nc(C)c(Cl)c2C)C1 ZINC000880595350 CD On-Demand Anodyne CCR1 23 49 O=C(CN1CCc2ncncc2C1)NCc1cccnc1 ZINC000880595353 CC On-Demand Anodyne SCD 15 41 O=C(CN1CCc2ncncc2C1)NCc1cccnc1 ZINC000880595353 CC On-Demand Anodyne NAMPT 74 40 COc1ccc(OCCN2CCc3ncncc3C2)c([N+](=O)[O-])c1 ZINC000880595359 ED On-Demand Bother ABCB1 17 43 O=C(CN1CCc2ncncc2C1)N1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880595369 GD On-Demand Anodyne P2RY14 47 37 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne CTSD 38 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne PGC 56 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne REN 74 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne REN1 18 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne BACE1 28 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne FPR1 46 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN1CCc2ncncc2C1 ZINC000880595371 GE On-Demand Anodyne PLM2_PLAFA 52 32 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne FKBP1A 32 46 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne CELA1 19 43 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne GRIN2B 46 51 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne CCR5 22 44 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne PREP 52 48 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne TGM2 39 45 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne F13A1 43 45 COCC1CN(C(=O)C2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880595381 EE On-Demand Anodyne SLC12A5 63 40 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1 ZINC000880595404 CD On-Demand Anodyne ABCB1B 30 40 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1 ZINC000880595404 CD On-Demand Anodyne ABCG2 23 40 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1 ZINC000880595404 CD On-Demand Anodyne NOD2 40 35 O=C(CN1CCc2ncncc2C1)NCc1ccc(F)cc1C(F)(F)F ZINC000880595408 FE On-Demand Anodyne P2RX7 40 47 c1ccc2c(OCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595420 DG On-Demand Anodyne HTR1A 16 41 c1ccc2c(OCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595420 DG On-Demand Anodyne HTR1D 18 40 c1ccc2c(OCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595420 DG On-Demand Anodyne HTR1B 18 41 c1ccc2c(OCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595420 DG On-Demand Anodyne HTR5A 28 52 c1ccc2c(OCCN3CCc4ncncc4C3)cccc2c1 ZINC000880595420 DG On-Demand Anodyne ABCB1B 40 32 O=C(CN1CCc2ncncc2C1)NCCc1nc2ccccc2s1 ZINC000880595426 FD On-Demand Anodyne ACOX1 49 34 COCC1CN(C(=O)CC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880595427 EE On-Demand Anodyne GPR119 37 42 O=C(CN1CCc2ncncc2C1)N1CCC[C@@H]1c1ccc(Cl)c(Cl)c1 ZINC000880595432 GH On-Demand Anodyne CPT1A 69 34 O=C(CN1CCc2ncncc2C1)N1CCC[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000880595433 GH On-Demand Anodyne CPT1A 69 34 O=C(CN1CCc2ncncc2C1)Nc1cccnc1Cl ZINC000880595435 DD On-Demand Anodyne G2YM83_BOTF4 61 34 CN1CCCC[C@H]1CCN1CCc2ncncc2C1 ZINC000880595441 CD On-Demand Anodyne CHRNA10 43 35 CN1CCCC[C@@H]1CCN1CCc2ncncc2C1 ZINC000880595442 CD On-Demand Anodyne CHRNA10 43 35 O=C(CN1CCc2ncncc2C1)Nc1ccccc1C(F)(F)F ZINC000880595453 EE On-Demand Anodyne RBP4 53 33 COCC1CN(C(=O)C(=O)NCCCc2ccccc2)C1 ZINC000880595454 CC On-Demand Anodyne FKBP1A 29 41 COCC1CN(C(=O)C(=O)NCCCc2ccccc2)C1 ZINC000880595454 CC On-Demand Anodyne AMP1_PLAFQ 27 41 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1F ZINC000880595456 DD On-Demand Anodyne ABCG2 35 44 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1F ZINC000880595456 DD On-Demand Anodyne NOD2 43 36 COCC1CN(C(=O)c2c[nH]c3ccc([N+](=O)[O-])cc23)C1 ZINC000880595461 CD On-Demand Bother GABRA1 17 49 COCC1CN(C(=O)c2c[nH]c3ccc([N+](=O)[O-])cc23)C1 ZINC000880595461 CD On-Demand Bother CACNA1D 50 35 COCC1CN(C(=O)c2c[nH]c3ccc([N+](=O)[O-])cc23)C1 ZINC000880595461 CD On-Demand Bother GABRA2 17 46 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne KLK3 49 33 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CTSB 41 39 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CTSK 30 40 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne PREP 35 51 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CAPNS1 53 32 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CTSS 16 40 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CAPN1 58 42 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne CAPN2 98 42 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne TGM2 33 42 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne KLK5 21 41 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne NPR 64 38 COCC1CN(C(=O)CCCNC(=O)OCc2ccccc2)C1 ZINC000880595467 DD On-Demand Anodyne SLC12A5 42 34 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880595487 FD On-Demand Anodyne DRD4 29 40 O=C(CN1CCc2ncncc2C1)Nc1cccc(C(=O)NC2CC2)c1 ZINC000880595487 FD On-Demand Anodyne MCHR1 18 41 O=C(CN1CCc2ncncc2C1)N1CCN(Cc2ccccc2)CC1 ZINC000880595496 FD On-Demand Anodyne SIGMAR1 41 42 O=C(CN1CCc2ncncc2C1)N1CCN(Cc2ccccc2)CC1 ZINC000880595496 FD On-Demand Anodyne FAAH 27 43 COc1ccc2c(CN3CCc4ncncc4C3)cc(=O)oc2c1 ZINC000880595505 DE On-Demand Anodyne CYP19A1 16 52 COc1ccc2c(CN3CCc4ncncc4C3)cc(=O)oc2c1 ZINC000880595505 DE On-Demand Anodyne CYP11B1 20 46 Fc1ccc(SCCN2CCc3ncncc3C2)cc1 ZINC000880595523 CF On-Demand Anodyne HTR5A 16 43 c1ncc2c(n1)CCN(Cc1ccc(CN3CCc4ncncc4C3)cc1)C2 ZINC000880595532 FE On-Demand Anodyne NOD2 40 35 O=C(CN1CCc2ncncc2C1)NCc1ccc2c(c1)OCO2 ZINC000880595534 EC On-Demand Anodyne NOS2 111 44 O=C(CN1CCc2ncncc2C1)NCc1ccc2c(c1)OCO2 ZINC000880595534 EC On-Demand Anodyne MCHR1 22 42 O=C(CN1CCc2ncncc2C1)NCc1ccc2c(c1)OCO2 ZINC000880595534 EC On-Demand Anodyne CLK1 21 40 O=C(CN1CCc2ncncc2C1)NCc1ccc2c(c1)OCO2 ZINC000880595534 EC On-Demand Anodyne CLK4 45 37 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCCCC2)cc1 ZINC000880595540 FE On-Demand Anodyne SLC27A1 43 39 CN(C)S(=O)(=O)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880595547 GC On-Demand Anodyne P2RY14 43 35 O=[N+]([O-])c1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880595556 DD On-Demand Bother HTR5A 18 41 O=[N+]([O-])c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595585 DD On-Demand Bother LTA4H 44 54 O=[N+]([O-])c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595585 DD On-Demand Bother HTR5A 20 51 CCOC(=O)N1CCN(C(=O)[C@@H](C)N2CCc3ncncc3C2)CC1 ZINC000880595587 EC On-Demand Anodyne P2RY12 49 35 CCOC(=O)N1CCN(C(=O)[C@H](C)N2CCc3ncncc3C2)CC1 ZINC000880595588 EC On-Demand Anodyne P2RY12 49 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)/C=C/c2ccc(C(N)=O)cc2)C1 ZINC000880595599 FC On-Demand Anodyne PREP 64 39 COCC1CN(C(=O)[C@H]2CCCN2C(=O)/C=C/c2ccc(C(N)=O)cc2)C1 ZINC000880595600 FC On-Demand Anodyne PREP 64 39 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)/C=C\c2ccc(C(N)=O)cc2)C1 ZINC000880595601 FC On-Demand Anodyne PREP 64 39 COCC1CN(C(=O)[C@H]2CCCN2C(=O)/C=C\c2ccc(C(N)=O)cc2)C1 ZINC000880595602 FC On-Demand Anodyne PREP 64 39 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne HTR1A 15 40 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne DRD2 17 40 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne ACHE 17 45 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne HTR2A 15 55 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne HRH3 70 45 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne BCHE 23 45 c1ccc2cc(OCCCN3CCc4ncncc4C3)ccc2c1 ZINC000880595615 DG On-Demand Anodyne HTR5A 29 55 CN(C)Cc1ccnc(NC(=O)NCCc2cccnc2)c1 ZINC000880595616 CD On-Demand Anodyne PTAFR 21 40 CN(C)Cc1ccnc(NC(=O)NCCc2cccnc2)c1 ZINC000880595616 CD On-Demand Anodyne NAMPT 50 44 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne ACE 35 44 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne P2RY12 97 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne MME 47 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne PTAFR 30 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne MC4R 30 51 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CTRA_BOVIN 31 47 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne TRY2_BOVIN 54 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne PAPA1_CARPA 25 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CYSP_TRYCR 51 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CTSL 38 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne TIMP3 41 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CTRB1 40 35 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CTSS 26 46 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne ACE2 67 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne CTRB_BOVIN 55 33 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne PSMB5 42 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595635 FD On-Demand Anodyne BLA1_STEMA 46 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne ACE 35 44 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne P2RY12 97 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne MME 47 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne PTAFR 30 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne MC4R 30 51 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CTRA_BOVIN 31 47 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne TRY2_BOVIN 54 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne PAPA1_CARPA 25 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CYSP_TRYCR 51 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CTSL 38 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne TIMP3 41 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CTRB1 40 35 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CTSS 26 46 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne ACE2 67 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne CTRB_BOVIN 55 33 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne PSMB5 42 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccnc2)C1 ZINC000880595636 FD On-Demand Anodyne BLA1_STEMA 46 36 COc1ccc([C@@H]2CCCN2C(=O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880595637 GE On-Demand Anodyne CPT1A 103 40 COc1ccc([C@@H]2CCCN2C(=O)CN2CCc3ncncc3C2)c(OC)c1 ZINC000880595637 GE On-Demand Anodyne CPT2 37 40 COc1cccc(S(=O)(=O)CCN2CCc3ncncc3C2)c1 ZINC000880595649 ED On-Demand Anodyne HTR7 19 47 COc1cccc(S(=O)(=O)CCN2CCc3ncncc3C2)c1 ZINC000880595649 ED On-Demand Anodyne CYP11B2 17 41 COc1cccc(S(=O)(=O)CCN2CCc3ncncc3C2)c1 ZINC000880595649 ED On-Demand Anodyne ABCB1B 47 34 O=[N+]([O-])c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880595656 CD On-Demand Bother ABCC1 18 41 O=[N+]([O-])c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880595656 CD On-Demand Bother ABCG2 18 41 O=[N+]([O-])c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880595656 CD On-Demand Bother KCNJ1 43 56 O=C(CN1CCc2ncncc2C1)NCC1(c2ccccc2)CC1 ZINC000880595770 DD On-Demand Anodyne NPFFR1 27 42 O=C(CN1CCc2ncncc2C1)NCc1ccc(CN2CCCC2)cc1 ZINC000880595777 FD On-Demand Anodyne BDKRB1 30 41 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CC2(Cl)Cl)c1 ZINC000880595788 DE On-Demand Anodyne TYK2 30 44 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CC2(Cl)Cl)c1 ZINC000880595789 DE On-Demand Anodyne TYK2 30 44 c1ccc(OCCOCCN2CCc3ncncc3C2)cc1 ZINC000880595795 CD On-Demand Anodyne LTA4H 47 41 c1ccc(OCCOCCN2CCc3ncncc3C2)cc1 ZINC000880595795 CD On-Demand Anodyne HRH3 23 43 c1ccc(OCCOCCN2CCc3ncncc3C2)cc1 ZINC000880595795 CD On-Demand Anodyne HTR5A 25 45 COCC1CN(C(=O)[C@@H]2CC(c3cccc(F)c3)=NO2)C1 ZINC000880595796 CD On-Demand Anodyne LUCI_PHOPY 29 43 COCC1CN(C(=O)[C@H]2CC(c3cccc(F)c3)=NO2)C1 ZINC000880595798 CD On-Demand Anodyne LUCI_PHOPY 29 43 O=C(CN1CCc2ncncc2C1)Nc1ccc(F)c(Cl)c1 ZINC000880595805 DE On-Demand Anodyne ERBB4 55 38 O=C(CN1CCc2ncncc2C1)Nc1ccc(F)c(Cl)c1 ZINC000880595805 DE On-Demand Anodyne MCHR1 30 42 O=C(CN1CCc2ncncc2C1)NCc1cccc(OCC(F)(F)F)c1 ZINC000880595818 GE On-Demand Anodyne PDS 41 36 O=C(CN1CCc2ncncc2C1)N(Cc1ccc(C(F)(F)F)cc1)C1CC1 ZINC000880595819 GG On-Demand Anodyne TRPM8 43 36 COc1ccc(-c2csc(NC(=O)CN3CCc4ncncc4C3)n2)cc1 ZINC000880595822 GF On-Demand Anodyne ACOX1 49 33 COc1ccc(-c2csc(NC(=O)CN3CCc4ncncc4C3)n2)cc1 ZINC000880595822 GF On-Demand Anodyne ROCK1 20 41 COc1ccc(-c2csc(NC(=O)CN3CCc4ncncc4C3)n2)cc1 ZINC000880595822 GF On-Demand Anodyne ROCK2 15 41 COCC1CN(C(=O)c2cccc(NC(=O)OC)c2)C1 ZINC000880595829 CD On-Demand Anodyne KCNK3 76 35 COCC1CN(C(=O)c2cccc(NC(=O)OC)c2)C1 ZINC000880595829 CD On-Demand Anodyne KCNK9 43 33 c1ccc(CCCN2CCc3ncncc3C2)cc1 ZINC000880595844 CE On-Demand Anodyne SLC6A3 18 40 c1ccc(CCCN2CCc3ncncc3C2)cc1 ZINC000880595844 CE On-Demand Anodyne SIGMAR1 48 63 c1ccc(CCCN2CCc3ncncc3C2)cc1 ZINC000880595844 CE On-Demand Anodyne HTR5A 30 47 CC(=O)c1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880595858 DD On-Demand Anodyne ABCB1B 30 40 CC(=O)c1ccccc1NC(=O)CN1CCc2ncncc2C1 ZINC000880595858 DD On-Demand Anodyne ABCG2 25 40 COCC1CN(C(=O)c2cccc(OCC(=O)OC)c2)C1 ZINC000880595859 CC On-Demand Anodyne DRD4 40 30 COCC1CN(C(=O)CNc2cc(Cl)ccc2OC)C1 ZINC000880595867 CD On-Demand Anodyne CPT1A 44 38 COCC1CN(C(=O)CNc2cc(Cl)ccc2OC)C1 ZINC000880595867 CD On-Demand Anodyne CPT2 40 35 COCC1CN(C(=O)CNc2cc(Cl)ccc2OC)C1 ZINC000880595867 CD On-Demand Anodyne RBP4 20 42 O=C(CCN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880595870 FF On-Demand Anodyne KIT 18 41 O=C(CCN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880595870 FF On-Demand Anodyne KDR 20 47 O=C(CCN1CCc2ncncc2C1)Nc1cccc(C(F)(F)F)c1 ZINC000880595870 FF On-Demand Anodyne EPHX2 18 43 COCC1CN(C(=O)c2cn(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)C1 ZINC000880595887 GD On-Demand Anodyne GPR119 47 39 O[C@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595895 DD On-Demand Anodyne ADRB1 21 46 O[C@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595895 DD On-Demand Anodyne HTR1A 17 54 O[C@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595895 DD On-Demand Anodyne SLC6A4 20 45 O[C@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595895 DD On-Demand Anodyne ABCB1 48 37 O[C@@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595896 DD On-Demand Anodyne ADRB1 21 46 O[C@@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595896 DD On-Demand Anodyne HTR1A 17 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595896 DD On-Demand Anodyne SLC6A4 20 45 O[C@@H](COc1cccc2[nH]ccc12)CN1CCc2ncncc2C1 ZINC000880595896 DD On-Demand Anodyne ABCB1 48 37 O=C(CN1CCc2ncncc2C1)NCc1ccc(-c2ccc(Cl)cc2)o1 ZINC000880595906 GG On-Demand Anodyne SCN10A 24 40 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880595916 FD On-Demand Anodyne PLA2G7 28 43 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880595916 FD On-Demand Anodyne SSTR1 20 40 O=C(CN1CCc2ncncc2C1)N1CCN(c2ccc(F)cc2)CC1 ZINC000880595916 FD On-Demand Anodyne SLC27A1 59 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne F2 21 49 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne PLG 26 49 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne ACE 66 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne GHRHR 59 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne P2RY12 54 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CELA1 20 49 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne MME 80 37 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne TACR1 16 50 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSD 20 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne PGC 64 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne MC4R 56 41 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CMA1 45 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTRA_BOVIN 42 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne FCER2 42 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSB 44 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne PAPA1_CARPA 79 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne TRY1_BOVIN 27 49 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CYSP_TRYCR 63 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CCKAR 66 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSG 43 33 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSK 45 52 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSL 57 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CACNA1B 51 39 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne PGA 33 43 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne TIMP3 54 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTRB1 40 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne TACR3 18 47 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CAPNS1 60 34 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne HLA-DRB1 34 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CELA2A 49 32 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne REN 107 48 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne REN1 27 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CCKBR 32 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSS 29 55 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CAPN1 73 47 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CAPN2 50 38 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTSE 15 40 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne ACE2 71 36 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne KLK5 33 42 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne FPR1 81 49 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne CTRB_BOVIN 60 45 COCC1CN(C(=O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595918 EE On-Demand Anodyne BLA1_STEMA 40 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne F2 21 49 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne PLG 26 49 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne ACE 66 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne GHRHR 59 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne P2RY12 54 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CELA1 20 49 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne MME 80 37 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne TACR1 16 50 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSD 20 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne PGC 64 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne MC4R 56 41 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CMA1 45 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTRA_BOVIN 42 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne FCER2 42 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSB 44 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne PAPA1_CARPA 79 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne TRY1_BOVIN 27 49 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CYSP_TRYCR 63 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CCKAR 66 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSG 43 33 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSK 45 52 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSL 57 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CACNA1B 51 39 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne PGA 33 43 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne TIMP3 54 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTRB1 40 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne TACR3 18 47 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CAPNS1 60 34 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne HLA-DRB1 34 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CELA2A 49 32 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne REN 107 48 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne REN1 27 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CCKBR 32 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSS 29 55 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CAPN1 73 47 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CAPN2 50 38 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTSE 15 40 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne ACE2 71 36 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne KLK5 33 42 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne FPR1 81 49 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne CTRB_BOVIN 60 45 COCC1CN(C(=O)[C@@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880595919 EE On-Demand Anodyne BLA1_STEMA 40 34 C[C@H](C(=O)Nc1cccnc1Cl)N1CCc2ncncc2C1 ZINC000880595923 DD On-Demand Anodyne G2YM83_BOTF4 54 34 O=C(CN1CCc2ncncc2C1)NCCc1ccc(OC(F)(F)F)cc1 ZINC000880595927 GE On-Demand Anodyne NOD2 24 41 O=C(CCN1CCc2ncncc2C1)N1CCN(c2ccccn2)CC1 ZINC000880595937 FC On-Demand Anodyne DRD4 27 42 O=C(CCN1CCc2ncncc2C1)N1CCN(c2ccccn2)CC1 ZINC000880595937 FC On-Demand Anodyne SSTR1 21 40 NC(=O)COc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880595956 CC On-Demand Anodyne NOD2 45 41 FC(F)(F)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595957 DF On-Demand Anodyne LTA4H 47 52 FC(F)(F)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595957 DF On-Demand Anodyne HTR5A 21 44 FC(F)(F)c1ccc(OCCN2CCc3ncncc3C2)cc1 ZINC000880595957 DF On-Demand Anodyne PSMB1 40 40 O=C(CN1CCc2ncncc2C1)NCCOc1ccc2c(c1)OCO2 ZINC000880595958 FC On-Demand Anodyne HRH2 15 40 O=C(CN1CCc2ncncc2C1)NCCOc1ccc2c(c1)OCO2 ZINC000880595958 FC On-Demand Anodyne EDNRA 27 40 O=C(CN1CCc2ncncc2C1)NCCOc1ccc2c(c1)OCO2 ZINC000880595958 FC On-Demand Anodyne NOS2 63 33 CC(=O)c1cccc(NC(=O)CN2CCc3ncncc3C2)c1 ZINC000880595962 DD On-Demand Anodyne P2RY14 48 38 C[C@H](C(=O)Nc1sc2c(c1C#N)CCCCC2)N1CCc2ncncc2C1 ZINC000880595964 GG On-Demand Mild VIPR1 26 42 C[C@@H](C(=O)Nc1sc2c(c1C#N)CCCCC2)N1CCc2ncncc2C1 ZINC000880595969 GG On-Demand Mild VIPR1 26 42 O=C(CN1CCc2ncncc2C1)Nc1ccc(C(F)(F)F)cc1 ZINC000880595982 EE On-Demand Anodyne EPHX2 25 41 O=C(CN1CCc2ncncc2C1)Nc1ccc(C(F)(F)F)cc1 ZINC000880595982 EE On-Demand Anodyne TRPM8 51 47 O=C(CN1CCc2ncncc2C1)NCC1(c2ccc(F)cc2)CCCC1 ZINC000880596006 FF On-Demand Anodyne SLC27A1 53 37 COCC1CN(C(=O)c2ccc(N3CCN(C(C)C)CC3)cc2)C1 ZINC000880596012 ED On-Demand Anodyne HRH3 16 44 COCC1CN(C(=O)c2ccc(N3CCN(C(C)C)CC3)cc2)C1 ZINC000880596012 ED On-Demand Anodyne PRNP 53 43 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)cc1 ZINC000880596042 DE On-Demand Anodyne IMDH_CRYPV 28 42 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)cc1 ZINC000880596042 DE On-Demand Anodyne NOD1 16 43 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)cc1 ZINC000880596042 DE On-Demand Anodyne NOD2 40 34 CN(C)Cc1ccnc(NC(=O)N(C)Cc2ccc(Cl)nc2)c1 ZINC000880596044 EF On-Demand Anodyne NACHRBETA2 24 43 COCC1CN(C(=O)[C@@H]2CCCN2C)C1 ZINC000880596050 BC On-Demand Anodyne PREP 24 40 COCC1CN(C(=O)[C@H]2CCCN2C)C1 ZINC000880596051 BC On-Demand Anodyne PREP 24 40 CN(C)Cc1ccnc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880596052 FE On-Demand Anodyne GPR119 47 44 c1ccc2cc(CCN3CCc4ncncc4C3)ccc2c1 ZINC000880596053 CG On-Demand Anodyne SIGMAR1 20 44 c1ccc2cc(CCN3CCc4ncncc4C3)ccc2c1 ZINC000880596053 CG On-Demand Anodyne ABCB1 18 44 FC(F)(F)c1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880596056 EG On-Demand Anodyne HRH3 32 45 FC(F)(F)c1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880596056 EG On-Demand Anodyne HTR5A 24 44 FC(F)(F)c1cccc(OCCCN2CCc3ncncc3C2)c1 ZINC000880596056 EG On-Demand Anodyne GALR3 72 46 CC(=O)c1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880596092 DE On-Demand Anodyne PRNP 45 35 CC(=O)c1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880596092 DE On-Demand Anodyne ABCB1B 31 40 CC(=O)c1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880596092 DE On-Demand Anodyne ABCG2 25 40 CC(=O)c1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880596092 DE On-Demand Anodyne NOD2 44 38 COCC1CN(C(=O)c2ccc(NC(=O)OC(C)(C)C)cc2Cl)C1 ZINC000880596094 FG On-Demand Anodyne NPY2R 40 40 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCc3ncncc3C2)cc1 ZINC000880596095 FF On-Demand Anodyne CPT1A 110 41 CCOc1ccc([C@@H]2CCCN2C(=O)CN2CCc3ncncc3C2)cc1 ZINC000880596095 FF On-Demand Anodyne CPT2 39 41 COc1ccc(-c2csc(NC(=O)[C@@H](C)N3CCc4ncncc4C3)n2)cc1 ZINC000880596112 GF On-Demand Anodyne ROCK1 19 40 COc1ccc(-c2csc(NC(=O)[C@H](C)N3CCc4ncncc4C3)n2)cc1 ZINC000880596113 GF On-Demand Anodyne ROCK1 19 40 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1C(=O)NC1CC1 ZINC000880596122 FD On-Demand Anodyne ABCB1B 32 44 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1C(=O)NC1CC1 ZINC000880596122 FD On-Demand Anodyne ABCG2 24 44 O=C(CN1CCc2ncncc2C1)NCc1ccc(OC(F)(F)F)cc1 ZINC000880596148 FE On-Demand Anodyne NOD2 25 42 O=C(NC1CCN(C(=O)CN2CCc3ncncc3C2)CC1)c1ccccc1 ZINC000880596151 GD On-Demand Anodyne DRD4 21 41 O=C(NC1CCN(C(=O)CN2CCc3ncncc3C2)CC1)c1ccccc1 ZINC000880596151 GD On-Demand Anodyne SSTR5 42 37 O=C(NC1CCN(C(=O)CN2CCc3ncncc3C2)CC1)c1ccccc1 ZINC000880596151 GD On-Demand Anodyne CCR8 51 37 O=C(NC1CCN(C(=O)CN2CCc3ncncc3C2)CC1)c1ccccc1 ZINC000880596151 GD On-Demand Anodyne HPGDS 39 42 COCC1CN(C(=O)Cc2ccc([N+](=O)[O-])cc2Br)C1 ZINC000880596152 EE On-Demand Bother CACNA1D 40 35 C[C@H](C(=O)Nc1nc2ccccc2s1)N1CCc2ncncc2C1 ZINC000880596153 EE On-Demand Anodyne BCL2L1 52 33 C[C@@H](C(=O)Nc1nc2ccccc2s1)N1CCc2ncncc2C1 ZINC000880596154 EE On-Demand Anodyne BCL2L1 52 33 COc1ccc([C@@H]2CCCCCN2C(=O)CN2CCc3ncncc3C2)cc1 ZINC000880596157 GF On-Demand Anodyne CPT1A 124 43 COc1ccc([C@@H]2CCCCCN2C(=O)CN2CCc3ncncc3C2)cc1 ZINC000880596157 GF On-Demand Anodyne CPT2 45 39 O=S(=O)(CCCN1CCc2ncncc2C1)c1ccc(F)cc1 ZINC000880596169 ED On-Demand Anodyne HTR5A 15 41 COc1ccc(N2CCC(NC(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1 ZINC000880596170 GF On-Demand Clean F10 15 46 COc1ccc(N2CCC(NC(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1 ZINC000880596170 GF On-Demand Clean PDK1 49 36 COc1ccc(N2CCC(NC(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1 ZINC000880596170 GF On-Demand Clean MCHR1 19 41 COCC1CN(C(=O)c2cc(Cl)c(NC(=O)OC(C)(C)C)cc2OC)C1 ZINC000880596180 GG On-Demand Anodyne HTR4 58 35 O=C(CN1CCc2ncncc2C1)N1CCc2sccc2[C@H]1c1ccccc1 ZINC000880596181 GG On-Demand Anodyne TRPM8 20 43 O=C(CN1CCc2ncncc2C1)N1CCc2sccc2[C@@H]1c1ccccc1 ZINC000880596182 GG On-Demand Anodyne TRPM8 20 43 COc1ccc([C@@H]2CCCN2C(=O)CN2CCc3ncncc3C2)cc1OC ZINC000880596192 GE On-Demand Anodyne CPT1A 81 37 O=C(CCN1CCc2ncncc2C1)NC(c1ccccc1)c1ccccc1 ZINC000880596221 FG On-Demand Anodyne PRCP 27 45 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne F2 47 41 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne ACE 46 45 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne FKBP1A 82 50 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CELA1 29 65 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne GRIN2B 23 42 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne ELANE 29 44 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CTRA_BOVIN 64 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne TRY1_BOVIN 62 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CTSG 43 33 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CPT1A 40 41 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CPT2 48 41 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne PREP 150 72 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne CELA2A 52 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne LGMN 85 49 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne ACE2 20 44 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne KLK5 28 50 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne WNT3 44 35 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne SLC12A5 70 40 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880596226 ED On-Demand Anodyne TMPRSS11D 55 37 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880596258 GF On-Demand Anodyne CACNA1I 41 32 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CCCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880596259 GF On-Demand Anodyne CACNA1I 41 32 COCC1CN(C(=O)c2cc3cc(OC)c(OC)cc3[nH]2)C1 ZINC000880596269 DD On-Demand Anodyne GRIN2B 23 46 COCC1CN(C(=O)c2cc3cc(OC)c(OC)cc3[nH]2)C1 ZINC000880596269 DD On-Demand Anodyne HRH4 25 43 COCC1CN(C(=O)c2ccc(NC=O)cc2)C1 ZINC000880596272 BC On-Demand Anodyne L3MBTL3 35 40 O=C(CN1CCc2ncncc2C1)N1CC=C(c2c[nH]c3ccccc23)CC1 ZINC000880596281 FF On-Demand Anodyne SLC6A4 16 49 CN(C)Cc1ccnc(NC(=O)NCc2ccc(Cl)nc2)c1 ZINC000880596287 DF On-Demand Anodyne NAMPT 20 47 CN(C)Cc1ccnc(NC(=O)NCc2ccc(Cl)nc2)c1 ZINC000880596287 DF On-Demand Anodyne NACHRBETA2 18 40 COCC1CN(C(=O)c2cc(S(=O)(=O)N3CCC3)ccc2Cl)C1 ZINC000880596288 FD On-Demand Anodyne CASP7 47 37 CCOC(=O)N1CCCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880596291 ED On-Demand Anodyne P2RY12 40 36 COCC1CN(C(=O)/C=C(\C)c2cccc(C(F)(F)F)c2)C1 ZINC000880596299 DG On-Demand Anodyne CACNA1B 54 35 COCC1CN(C(=O)/C=C(\C)c2cccc(C(F)(F)F)c2)C1 ZINC000880596299 DG On-Demand Anodyne CCR2 73 39 COCC1CN(C(=O)/C=C(/C)c2cccc(C(F)(F)F)c2)C1 ZINC000880596300 DG On-Demand Anodyne CACNA1B 54 35 COCC1CN(C(=O)/C=C(/C)c2cccc(C(F)(F)F)c2)C1 ZINC000880596300 DG On-Demand Anodyne CCR2 73 39 c1cncc(CCN2CCc3ncncc3C2)c1 ZINC000880596301 BD On-Demand Anodyne SIGMAR1 15 47 COCC1CN(C(=O)c2ccccc2OCC(C)C)C1 ZINC000880596302 CE On-Demand Anodyne HCN1 64 32 COCC1CN(C(=O)c2ccccc2OCC(C)C)C1 ZINC000880596302 CE On-Demand Anodyne HCN4 48 32 O=C(CCN1CCc2ncncc2C1)N[C@@H](c1ccccc1)c1cccs1 ZINC000880596311 GG On-Demand Anodyne PRCP 23 43 O=C(CCN1CCc2ncncc2C1)N[C@H](c1ccccc1)c1cccs1 ZINC000880596312 GG On-Demand Anodyne PRCP 23 43 COCC1CN(C(=O)CN2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880596335 FD On-Demand Anodyne GRIN2B 33 45 COCC1CN(C(=O)CN2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880596335 FD On-Demand Anodyne PREP 27 40 COCC1CN(C(=O)CN2CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000880596335 FD On-Demand Anodyne SLC12A5 53 37 COCC1CN(C(=O)c2cccc(OC)n2)C1 ZINC000880596341 BC On-Demand Anodyne ALS 46 30 CN(C)Cc1ccnc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880596345 FE On-Demand Clean EPHB4 81 36 CN(C)Cc1ccnc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000880596345 FE On-Demand Clean STAT6 56 34 O=C(CN1CCc2ncncc2C1)Nc1nc2ccc(F)cc2s1 ZINC000880596350 EE On-Demand Anodyne CSNK1D 45 41 O=C(CN1CCc2ncncc2C1)Nc1nc2ccc(F)cc2s1 ZINC000880596350 EE On-Demand Anodyne PIK3CA 19 44 O=C(CN1CCc2ncncc2C1)Nc1nc2ccc(F)cc2s1 ZINC000880596350 EE On-Demand Anodyne SLC27A1 51 43 CNc1nc(C(=O)N2CC(COC)C2)cs1 ZINC000880596354 BC On-Demand Anodyne TRPC6 61 44 CNc1nc(C(=O)N2CC(COC)C2)cs1 ZINC000880596354 BC On-Demand Anodyne TRPC3 54 44 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880596367 FD On-Demand Anodyne ADRB1 52 37 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)COc2cccc(F)c2)c1 ZINC000880596367 FD On-Demand Anodyne PDS 52 40 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880596368 FD On-Demand Anodyne ADRB1 52 37 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)c1 ZINC000880596368 FD On-Demand Anodyne PDS 52 40 c1cc(CN2CCc3ncncc3C2)cc(CN2CCc3ncncc3C2)c1 ZINC000880596369 FE On-Demand Anodyne SIGMAR1 17 40 COCC1CN(C(=O)/C=C(\C)c2cccc(Cl)c2)C1 ZINC000880596373 CF On-Demand Anodyne CACNA1I 47 40 COCC1CN(C(=O)/C=C(/C)c2cccc(Cl)c2)C1 ZINC000880596374 CF On-Demand Anodyne CACNA1I 47 40 Cc1ccc(-c2csc(NC(=O)CN3CCc4ncncc4C3)n2)cc1C ZINC000880596375 GG On-Demand Anodyne MPL 17 47 COCC1CN(C(=O)/C=C(/C)c2cccc(OC)c2)C1 ZINC000880596378 CE On-Demand Anodyne DRD4 46 35 COCC1CN(C(=O)/C=C(/C)c2cccc(OC)c2)C1 ZINC000880596378 CE On-Demand Anodyne MTNR1A 26 41 COCC1CN(C(=O)/C=C(/C)c2cccc(OC)c2)C1 ZINC000880596378 CE On-Demand Anodyne MTNR1B 32 41 COCC1CN(C(=O)/C=C(\C)c2cccc(OC)c2)C1 ZINC000880596379 CE On-Demand Anodyne DRD4 46 35 COCC1CN(C(=O)/C=C(\C)c2cccc(OC)c2)C1 ZINC000880596379 CE On-Demand Anodyne MTNR1A 26 41 COCC1CN(C(=O)/C=C(\C)c2cccc(OC)c2)C1 ZINC000880596379 CE On-Demand Anodyne MTNR1B 32 41 COCC1CN(C(=O)C[C@H](C)C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880596384 FF On-Demand Anodyne GPR119 29 44 COCC1CN(C(=O)C[C@@H](C)C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880596385 FF On-Demand Anodyne GPR119 29 44 COCC1CN(C(=O)/C=C(/C)c2ccccc2C(F)(F)F)C1 ZINC000880596389 DG On-Demand Anodyne RBP4 84 38 COCC1CN(C(=O)/C=C(\C)c2ccccc2C(F)(F)F)C1 ZINC000880596390 DG On-Demand Anodyne RBP4 84 38 CN(C)Cc1ccnc(NC(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880596394 GF On-Demand Anodyne GRIN2B 21 41 CN(C)Cc1ccnc(NC(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880596394 GF On-Demand Anodyne CACNA1I 58 37 CN(C)Cc1ccnc(NC(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880596394 GF On-Demand Anodyne GPR119 53 42 COCC1CN(C(=O)c2cccn2C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880596398 GF On-Demand Anodyne GPR119 45 40 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCCCC2)nc1 ZINC000880596403 FD On-Demand Anodyne SLC27A1 60 46 N#Cc1c(NC(=O)CCN2CCc3ncncc3C2)sc2c1CCC2 ZINC000880596404 FE On-Demand Mild VIPR1 30 51 CN(C)Cc1ccnc(NC(=O)Nc2cnn(C(C)(C)C)c2)c1 ZINC000880596409 DF On-Demand Anodyne TYK2 19 42 COCC1CN(C(=O)C[C@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880596426 CD On-Demand Anodyne CTSK 15 40 COCC1CN(C(=O)C[C@@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880596427 CD On-Demand Anodyne CTSK 15 40 C[C@H](C(=O)Nc1sc2c(c1C#N)CCC2)N1CCc2ncncc2C1 ZINC000880596428 FE On-Demand Mild VIPR1 25 41 C[C@@H](C(=O)Nc1sc2c(c1C#N)CCC2)N1CCc2ncncc2C1 ZINC000880596429 FE On-Demand Mild VIPR1 25 41 COCC1CN(C(=O)c2ccc(NC(=O)OCC(F)(F)F)cc2)C1 ZINC000880596443 EF On-Demand Anodyne EPHX2 23 41 COCC1CN(C(=O)c2ccc(NC(=O)OCC(F)(F)F)cc2)C1 ZINC000880596443 EF On-Demand Anodyne ACR 41 35 O=C(CN1CCc2ncncc2C1)Nc1ccc2nc(C(F)(F)F)[nH]c2c1 ZINC000880596450 GE On-Demand Anodyne MCHR1 16 42 N#Cc1cccc(NC(=O)CCN2CCc3ncncc3C2)c1 ZINC000880596452 DD On-Demand Mild CCR3 15 43 COCC1CN(C(=O)c2cc(C(F)(F)F)ccc2F)C1 ZINC000880596457 CF On-Demand Anodyne LIPG 56 41 COC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880596458 ED On-Demand Anodyne SSTR5 44 34 COC(=O)N1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880596458 ED On-Demand Anodyne EPHX2 42 41 COCC1CN(C(=O)c2cc(C)ccc2N2CCCC2)C1 ZINC000880596459 CE On-Demand Anodyne HCRTR1 53 37 O=C(CN1CCc2ncncc2C1)Nc1ncc(Cc2ccc(F)cc2)s1 ZINC000880596466 GF On-Demand Anodyne SLC27A1 50 41 O=C(CN1CCc2ncncc2C1)Nc1ccc(N2CCc3ccccc32)cc1 ZINC000880596473 GG On-Demand Anodyne NOD2 40 34 COCC1CN(C(=O)C[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596483 EF On-Demand Anodyne CTSK 20 46 COCC1CN(C(=O)C[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596483 EF On-Demand Anodyne FPR1 44 35 COCC1CN(C(=O)C[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596484 EF On-Demand Anodyne CTSK 20 46 COCC1CN(C(=O)C[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596484 EF On-Demand Anodyne FPR1 44 35 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880596493 GF On-Demand Anodyne ACACB 15 44 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880596493 GF On-Demand Anodyne CACNA1I 53 33 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880596494 GF On-Demand Anodyne ACACB 15 44 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880596494 GF On-Demand Anodyne CACNA1I 53 33 N#Cc1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1Cl ZINC000880596495 EE On-Demand Mild IMDH_CRYPV 18 46 O=C(CN1CCc2ncncc2C1)Nc1nc2c(s1)CCC2 ZINC000880596506 DD On-Demand Anodyne SLC27A1 62 56 CN(C)Cc1ccnc(NC(=O)NCc2ccccc2N2CCOCC2)c1 ZINC000880596514 FE On-Demand Anodyne SCN10A 18 44 O=C(CCN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880596523 FD On-Demand Anodyne MTOR 55 36 O=C(CCN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880596523 FD On-Demand Anodyne EPHX2 17 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880596523 FD On-Demand Anodyne STAT6 60 35 O=C(CCN1CCc2ncncc2C1)Nc1ccc(N2CCOCC2)cc1 ZINC000880596523 FD On-Demand Anodyne DGAT1 15 40 COCC1CN(C(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596530 FF On-Demand Anodyne CTSK 21 44 COCC1CN(C(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596530 FF On-Demand Anodyne FPR1 46 37 COCC1CN(C(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596531 FF On-Demand Anodyne CTSK 21 44 COCC1CN(C(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596531 FF On-Demand Anodyne FPR1 46 37 COCC1CN(C(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596532 FF On-Demand Anodyne CTSK 21 44 COCC1CN(C(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596532 FF On-Demand Anodyne FPR1 46 37 COCC1CN(C(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596533 FF On-Demand Anodyne CTSK 21 44 COCC1CN(C(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596533 FF On-Demand Anodyne FPR1 46 37 O=C(CN1CCc2ncncc2C1)Nc1cccc(CN2CCSCC2)c1 ZINC000880596534 GE On-Demand Anodyne P2RY14 45 37 O=C(CN1CCc2ncncc2C1)Nc1nc2c(s1)CCCC2 ZINC000880596545 ED On-Demand Anodyne SLC27A1 64 58 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne PGC 56 38 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne PAPA1_CARPA 44 46 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne CCKAR 52 38 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne CTSK 21 47 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne CTSL 26 46 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne TACR3 15 40 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne REN 78 41 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne FPR1 53 42 COCC1CN(C(=O)C[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880596594 FF On-Demand Anodyne CTRB_BOVIN 29 40 CN(C)Cc1ccnc(NC(=O)NC2CCN(CC3CCCCC3)CC2)c1 ZINC000880596614 FG On-Demand Anodyne SSTR5 50 36 CN(C)Cc1ccnc(NC(=O)NC2CCN(CC3CCCCC3)CC2)c1 ZINC000880596614 FG On-Demand Anodyne CXCR3 16 43 O=C(CN1CCc2ncncc2C1)Nc1nccs1 ZINC000880596620 CC On-Demand Anodyne MAP1 96 47 O=C(CN1CCc2ncncc2C1)Nc1nccs1 ZINC000880596620 CC On-Demand Anodyne SLC27A1 36 42 C[C@H](C(=O)Nc1nccs1)N1CCc2ncncc2C1 ZINC000880596641 CD On-Demand Anodyne MAP1 87 35 C[C@@H](C(=O)Nc1nccs1)N1CCc2ncncc2C1 ZINC000880596642 CD On-Demand Anodyne MAP1 87 35 COCC1CN(C(=O)[C@H](Cc2c[nH]c3cc(F)ccc23)NC(C)=O)C1 ZINC000880596680 ED On-Demand Anodyne TACR1 16 41 COCC1CN(C(=O)[C@H](Cc2c[nH]c3cc(F)ccc23)NC(C)=O)C1 ZINC000880596680 ED On-Demand Anodyne GRPR 51 33 COCC1CN(C(=O)[C@@H](Cc2c[nH]c3cc(F)ccc23)NC(C)=O)C1 ZINC000880596681 ED On-Demand Anodyne TACR1 16 41 COCC1CN(C(=O)[C@@H](Cc2c[nH]c3cc(F)ccc23)NC(C)=O)C1 ZINC000880596681 ED On-Demand Anodyne GRPR 51 33 COCC1CN(C(=O)[C@@H](CNC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596684 EE On-Demand Anodyne CTSK 15 41 COCC1CN(C(=O)[C@@H](CNC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596684 EE On-Demand Anodyne FPR1 44 35 COCC1CN(C(=O)[C@H](CNC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596685 EE On-Demand Anodyne CTSK 15 41 COCC1CN(C(=O)[C@H](CNC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880596685 EE On-Demand Anodyne FPR1 44 35 O=C(CCN1CCc2ncncc2C1)Nc1cccc2ccccc12 ZINC000880596691 EG On-Demand Anodyne HTR7 19 40 O=C(CCN1CCc2ncncc2C1)Nc1cccc2ccccc12 ZINC000880596691 EG On-Demand Anodyne ABCB1B 49 41 O=C(CCN1CCc2ncncc2C1)Nc1cccc2ccccc12 ZINC000880596691 EG On-Demand Anodyne ABCG2 26 41 COc1ccc(N2CCCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1 ZINC000880596708 GF On-Demand Clean PDGFRB 46 37 CN(C)Cc1ccnc(NC(=O)N2CCC(CNC(=O)OC(C)(C)C)CC2)c1 ZINC000880596713 GF On-Demand Anodyne ACACB 15 43 CN(C)Cc1ccnc(NC(=O)N2CCC(CNC(=O)OC(C)(C)C)CC2)c1 ZINC000880596713 GF On-Demand Anodyne CACNA1I 52 33 O=C(CN1CCc2ncncc2C1)Nc1nc2ccccc2s1 ZINC000880596715 EE On-Demand Anodyne CSNK1D 39 48 O=C(CN1CCc2ncncc2C1)Nc1nc2ccccc2s1 ZINC000880596715 EE On-Demand Anodyne ACOX1 47 35 O=C(CN1CCc2ncncc2C1)Nc1nc2ccccc2s1 ZINC000880596715 EE On-Demand Anodyne BCL2L1 52 33 O=C(CN1CCc2ncncc2C1)Nc1nc2ccccc2s1 ZINC000880596715 EE On-Demand Anodyne SLC27A1 45 54 O=C(CCN1CCc2ncncc2C1)Nc1ccc(Cl)cc1 ZINC000880596736 DF On-Demand Anodyne NOD1 16 44 O=C(CCN1CCc2ncncc2C1)Nc1ccc(Cl)cc1 ZINC000880596736 DF On-Demand Anodyne NOD2 41 35 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne KLK3 46 32 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne CTSB 43 39 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne CYSP_TRYCR 45 37 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne PREP 33 55 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne CAPNS1 48 32 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne CAPN1 55 39 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne CAPN2 92 39 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne TGM2 32 43 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne KLK5 21 43 COCC1CN(C(=O)CCCCNC(=O)OCc2ccccc2)C1 ZINC000880596738 EE On-Demand Anodyne NPR 63 39 CN(C)Cc1ccnc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880596774 GF On-Demand Anodyne GPR119 44 42 CC(C)(C)OC(=O)N1CCC(CCN2CCc3ncncc3C2)CC1 ZINC000880596775 EF On-Demand Anodyne GPR119 51 47 O=C(CCN1CCc2ncncc2C1)Nc1ccccc1C(F)(F)F ZINC000880596787 FF On-Demand Anodyne RBP4 44 31 C=CCN1CCC(NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880596789 DD On-Demand Mild SSTR5 46 36 O=C(CCN1CCc2ncncc2C1)c1ccc(F)cc1 ZINC000880596799 CE On-Demand Anodyne HTR2A 20 48 O=C(CCN1CCc2ncncc2C1)c1ccc(F)cc1 ZINC000880596799 CE On-Demand Anodyne HTR5A 17 48 COCC1CN(C(=O)CCC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880596811 EF On-Demand Anodyne GPR119 32 41 COCC1CN(C(=O)CNC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880596825 FC On-Demand Anodyne PGA5 29 44 COCC1CN(C(=O)CNC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C1 ZINC000880596825 FC On-Demand Anodyne POLG_HCV1 23 42 Cc1ccc(NC(=O)c2nnc(CN3CCc4ncncc4C3)s2)cc1 ZINC000880596840 FE On-Demand Anodyne NOD2 43 37 CCOc1ccccc1C(F)(F)C(=O)N1CC(COC)C1 ZINC000880596855 CE On-Demand Anodyne HCN1 41 31 CCOc1ccccc1C(F)(F)C(=O)N1CC(COC)C1 ZINC000880596855 CE On-Demand Anodyne HCN4 41 31 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne LTA4H 56 52 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne ABCB1B 31 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne ABCB1 19 42 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne MCHR1 15 49 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne ABCG2 24 40 O=C(CCN1CCc2ncncc2C1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880596870 GG On-Demand Anodyne NOD2 44 40 COCC1CN(C(=O)[C@H](CC(F)F)NC(=O)OC(C)(C)C)C1 ZINC000880596923 DD On-Demand Anodyne POLG_HCV1 27 49 COCC1CN(C(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C)C1 ZINC000880596924 DD On-Demand Anodyne POLG_HCV1 27 49 CN(C)Cc1ccnc(NC(=O)NC(C)(C)c2ccc(F)cc2)c1 ZINC000880596926 EG On-Demand Anodyne MAPK14 16 40 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne DRD4 40 31 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne LTA4H 28 43 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne HRH3 26 47 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne SIGMAR1 21 40 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne HTR5A 24 40 COc1cccc(OCCN2CCc3ncncc3C2)c1 ZINC000880596927 CD On-Demand Anodyne ABCB1 22 47 Cc1cccc2c1CCN(C(=O)Nc1cc(CN(C)C)ccn1)C2 ZINC000880596950 DG On-Demand Anodyne P2RY14 51 36 N#C[C@@H](c1ccc(F)cc1)N1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880596952 GD On-Demand Mild PTAFR 40 45 N#C[C@H](c1ccc(F)cc1)N1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880596953 GD On-Demand Mild PTAFR 40 45 c1cc(CCCN2CCc3ncncc3C2)ccn1 ZINC000880596959 CD On-Demand Anodyne SIGMAR1 21 40 COC(=O)[C@@H](c1ccccc1)N1CCc2ncncc2C1 ZINC000880596974 CD On-Demand Anodyne NPY2R 15 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PLG 18 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne ACE 54 44 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne GHRHR 56 33 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne P2RY12 90 39 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CELA1 30 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne ELANE 36 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne MME 42 38 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne ANPEP 35 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne TACR1 17 46 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSD 32 46 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTRA_BOVIN 55 34 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne FCER2 49 36 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CASP3 31 51 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne BMP1 18 43 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne KLK3 109 49 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSB 90 59 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PAPA1_CARPA 91 51 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CYSP_TRYCR 68 51 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSG 42 33 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSK 86 68 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSL 69 68 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CACNA1B 49 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PGA 40 42 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PREP 20 43 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CAPNS1 92 51 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne MMP3 40 44 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne HLA-DRB1 83 39 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CELA2A 50 34 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne REN 80 44 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne REN1 45 42 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne MMP11 61 37 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne TGM1 24 42 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CTSS 44 68 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CAPN1 127 57 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CASP1 35 49 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne CAPN2 190 53 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PLAU 18 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne TGM2 41 46 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne POLG_HCV1 17 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne KLK5 42 40 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne MMP1 26 42 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne FPR1 79 42 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne NPR 98 44 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne AMP1_PLAFQ 25 41 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne PSMB5 61 53 COCC1CN(C(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596978 EE On-Demand Anodyne Q6PRC7_IXORI 40 31 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PLG 18 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne ACE 54 44 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne GHRHR 56 33 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne P2RY12 90 39 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CELA1 30 40 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne ELANE 36 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne MME 42 38 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne ANPEP 35 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne TACR1 17 46 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSD 32 46 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTRA_BOVIN 55 34 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne FCER2 49 36 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CASP3 31 51 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne BMP1 18 43 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne KLK3 109 49 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSB 90 59 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PAPA1_CARPA 91 51 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CYSP_TRYCR 68 51 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSG 42 33 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSK 86 68 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSL 69 68 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CACNA1B 49 40 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PGA 40 42 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PREP 20 43 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CAPNS1 92 51 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne MMP3 40 44 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne HLA-DRB1 83 39 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CELA2A 50 34 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne REN 80 44 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne REN1 45 42 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne MMP11 61 37 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne TGM1 24 42 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CTSS 44 68 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CAPN1 127 57 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CASP1 35 49 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne CAPN2 190 53 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PLAU 18 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne TGM2 41 46 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne POLG_HCV1 17 40 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne KLK5 42 40 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne MMP1 26 42 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne FPR1 79 42 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne NPR 98 44 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne AMP1_PLAFQ 25 41 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne PSMB5 61 53 COCC1CN(C(=O)[C@@H](CC(C)C)NC(=O)OCc2ccccc2)C1 ZINC000880596979 EE On-Demand Anodyne Q6PRC7_IXORI 40 31 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne ACE 20 45 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne SSTR2 82 46 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne GHRHR 32 49 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MME 26 42 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne EDNRB 24 42 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne EDNRA 33 53 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne TACR1 40 59 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne PGC 50 35 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MC4R 46 40 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne CCKAR 151 61 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne CTSL 24 61 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne PGA 23 49 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne BRS3 26 41 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne NMBR 45 45 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MC3R 60 36 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MC5R 65 33 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MMP2 28 45 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MMP8 35 45 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne GRPR 68 34 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne ECE1 66 47 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne REN 56 49 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne REN1 31 49 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne SSTR3 22 51 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MMP11 100 37 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne CCKBR 121 58 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne GHSR 69 49 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MMP9 26 45 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MC1R 86 36 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne MMP1 19 41 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne FPR1 51 54 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne NPR 27 40 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne KISS1R 65 33 COCC1CN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)OC(C)(C)C)C1 ZINC000880596981 GF On-Demand Anodyne ERAP2 42 36 c1cn(CCCN2CCc3ncncc3C2)cn1 ZINC000880596993 BD On-Demand Anodyne TBXAS1 32 41 c1cn(CCCN2CCc3ncncc3C2)cn1 ZINC000880596993 BD On-Demand Anodyne QPCT 23 42 COCC1CN(C(=O)c2cnc3ccccn23)C1 ZINC000880596995 BD On-Demand Anodyne EPHB3 19 43 CN(C)Cc1ccnc(NC(=O)N2CCC[C@@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880597007 GF On-Demand Anodyne ACACB 15 41 CN(C)Cc1ccnc(NC(=O)N2CCC[C@H](CNC(=O)OC(C)(C)C)C2)c1 ZINC000880597008 GF On-Demand Anodyne ACACB 15 41 FC(F)(F)Oc1cccc(CCN2CCc3ncncc3C2)c1 ZINC000880597028 DF On-Demand Anodyne ABCB1 17 41 COC(=O)c1ccc(CN2CCc3ncncc3C2)c(F)c1 ZINC000880597031 DD On-Demand Anodyne BDKRB1 19 40 COC(=O)c1ccc(CN2CCc3ncncc3C2)c(F)c1 ZINC000880597031 DD On-Demand Anodyne NOD2 40 33 O=C(CCN1CCc2ncncc2C1)c1ccccc1 ZINC000880597033 CE On-Demand Anodyne SLC6A1 26 40 O=C(CCN1CCc2ncncc2C1)c1ccccc1 ZINC000880597033 CE On-Demand Anodyne HTR5A 19 46 O=C(CCN1CCc2ncncc2C1)c1ccccc1 ZINC000880597033 CE On-Demand Anodyne CYP2J2 47 33 CN(C)Cc1ccnc(NC(=O)N2CCCN(C(=O)Oc3ccccc3)CC2)c1 ZINC000880597036 GF On-Demand Anodyne FAAH 25 40 O=C(CCN1CCc2ncncc2C1)Nc1cccc(Br)c1 ZINC000880597042 FF On-Demand Anodyne EGFR 51 54 Cc1ccc(C(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880597063 CE On-Demand Anodyne CYP2J2 40 40 CN(C)Cc1ccnc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880597075 GF On-Demand Anodyne EPHX2 42 38 CN(C)Cc1ccnc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880597075 GF On-Demand Anodyne GPR119 53 41 O[C@@H](COc1ccccc1C(F)(F)F)CN1CCc2ncncc2C1 ZINC000880597086 FE On-Demand Anodyne ABCB1 54 39 O[C@H](COc1ccccc1C(F)(F)F)CN1CCc2ncncc2C1 ZINC000880597087 FE On-Demand Anodyne ABCB1 54 39 O=C(CCN1CCc2ncncc2C1)N1CCc2ccccc2C1 ZINC000880597094 DD On-Demand Anodyne HTR7 20 47 NS(=O)(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597102 DC On-Demand Anodyne CA2 39 43 NS(=O)(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597102 DC On-Demand Anodyne CA1 41 43 NS(=O)(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597102 DC On-Demand Anodyne CA12 26 43 NS(=O)(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597102 DC On-Demand Anodyne CA9 36 43 CC(=O)Oc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880597110 CD On-Demand Anodyne NOD1 17 41 CC(=O)Oc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880597110 CD On-Demand Anodyne NOD2 47 42 Fc1cccc(CCCN2CCc3ncncc3C2)c1 ZINC000880597111 CF On-Demand Anodyne SIGMAR1 27 54 c1ccc2c(c1)CC[C@H](CN1CCc3ncncc3C1)C2 ZINC000880597124 CF On-Demand Anodyne PTGIR 41 35 c1ccc2c(c1)CC[C@@H](CN1CCc3ncncc3C1)C2 ZINC000880597125 CF On-Demand Anodyne PTGIR 41 35 OCc1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880597155 CD On-Demand Anodyne NOD2 40 34 CN(C)Cc1ccnc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)c1 ZINC000880597217 FG On-Demand Anodyne TYK2 18 42 CN(C)Cc1ccnc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)c1 ZINC000880597218 FG On-Demand Anodyne TYK2 18 42 N#Cc1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597229 CD On-Demand Mild KCNJ1 38 44 c1ccc(CCCCN2CCc3ncncc3C2)cc1 ZINC000880597263 CF On-Demand Anodyne SIGMAR1 47 57 c1ccc(CCCCN2CCc3ncncc3C2)cc1 ZINC000880597263 CF On-Demand Anodyne HTR5A 31 48 c1ccc(CCCCN2CCc3ncncc3C2)cc1 ZINC000880597263 CF On-Demand Anodyne FAAH 45 40 c1ccc(CCCCN2CCc3ncncc3C2)cc1 ZINC000880597263 CF On-Demand Anodyne ABCB1 20 40 c1ccc(CCCCN2CCc3ncncc3C2)cc1 ZINC000880597263 CF On-Demand Anodyne CES1 45 36 O=c1c2ccccc2ncn1CCN1CCc2ncncc2C1 ZINC000880597264 DD On-Demand Anodyne HTR1B 18 42 O=c1c2ccccc2ncn1CCN1CCc2ncncc2C1 ZINC000880597264 DD On-Demand Anodyne ABCB1B 48 37 O=c1c2ccccc2ncn1CCN1CCc2ncncc2C1 ZINC000880597264 DD On-Demand Anodyne HNMT 48 32 COCC1CN(C(=O)c2ccc(-n3cnc4ccccc43)nc2)C1 ZINC000880597267 DE On-Demand Anodyne HPGD 47 39 Cc1cccc(C(=O)NNC(=O)CN2CCc3ncncc3C2)c1 ZINC000880597273 EC On-Demand Reactive KCNK3 48 35 Cc1cccc(C(=O)NNC(=O)CN2CCc3ncncc3C2)c1 ZINC000880597273 EC On-Demand Reactive KCNK9 41 35 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCc2ncncc2C1 ZINC000880597313 FF On-Demand Anodyne PPARG 43 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCc2ncncc2C1 ZINC000880597313 FF On-Demand Anodyne PPARA 40 38 CCOC(=O)c1nc(-c2ccccc2)oc1CN1CCc2ncncc2C1 ZINC000880597313 FF On-Demand Anodyne PDE8B 53 32 COc1cc(Br)ccc1CCCN1CCc2ncncc2C1 ZINC000880597343 FG On-Demand Anodyne ABCB1 21 41 c1ccc(COCCCN2CCc3ncncc3C2)cc1 ZINC000880597383 CE On-Demand Anodyne HRH3 18 52 c1ccc(COCCCN2CCc3ncncc3C2)cc1 ZINC000880597383 CE On-Demand Anodyne SIGMAR1 23 43 c1ccc(COCCCN2CCc3ncncc3C2)cc1 ZINC000880597383 CE On-Demand Anodyne HTR5A 25 52 c1ncc2c(n1)CCN(CCCN1CCCCC1)C2 ZINC000880597387 CD On-Demand Anodyne HRH3 39 48 c1ncc2c(n1)CCN(CCCN1CCCCC1)C2 ZINC000880597387 CD On-Demand Anodyne SIGMAR1 15 42 c1ncc2c(n1)CCN(CCCN1CCCCC1)C2 ZINC000880597387 CD On-Demand Anodyne HNMT 81 35 COCC1CN(C(=O)[C@@H]2C[C@H]2C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880597390 FE On-Demand Anodyne GPR119 33 43 COCC1CN(C(=O)c2cc(F)c(C(F)(F)F)cc2F)C1 ZINC000880597396 DF On-Demand Anodyne LRRK2 21 40 Fc1ccccc1-c1noc(CN2CCc3ncncc3C2)n1 ZINC000880597418 DE On-Demand Anodyne GABRA3 44 39 COCC1CN(C(=O)[C@@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597421 ED On-Demand Anodyne FKBP1A 15 41 COCC1CN(C(=O)[C@@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597421 ED On-Demand Anodyne PREP 49 52 COCC1CN(C(=O)[C@@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597421 ED On-Demand Anodyne LGMN 45 38 COCC1CN(C(=O)[C@@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597421 ED On-Demand Anodyne KLK5 42 42 COCC1CN(C(=O)[C@@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597421 ED On-Demand Anodyne SLC12A5 58 36 COCC1CN(C(=O)[C@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597423 ED On-Demand Anodyne FKBP1A 15 41 COCC1CN(C(=O)[C@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597423 ED On-Demand Anodyne PREP 49 52 COCC1CN(C(=O)[C@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597423 ED On-Demand Anodyne LGMN 45 38 COCC1CN(C(=O)[C@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597423 ED On-Demand Anodyne KLK5 42 42 COCC1CN(C(=O)[C@H]2COCCN2C(=O)OCc2ccccc2)C1 ZINC000880597423 ED On-Demand Anodyne SLC12A5 58 36 COCC1CN(C(=O)/C(C)=C/c2ccc(OC)c(F)c2)C1 ZINC000880597427 CE On-Demand Anodyne TUBB1 46 51 COCC1CN(C(=O)/C(C)=C\c2ccc(OC)c(F)c2)C1 ZINC000880597429 CE On-Demand Anodyne TUBB1 46 51 COCC1CN(C(=O)CCN(C)C(=O)OCc2ccccc2)C1 ZINC000880597471 DD On-Demand Anodyne SLC12A5 44 32 O=C(OCc1ccccc1)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880597492 FF On-Demand Anodyne GRIN2B 46 56 O=C(OCc1ccccc1)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880597492 FF On-Demand Anodyne PREP 28 41 O=C(OCc1ccccc1)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880597492 FF On-Demand Anodyne TGM2 30 44 O=C(OCc1ccccc1)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880597492 FF On-Demand Anodyne F13A1 38 44 O=C(OCc1ccccc1)N1CCC(CN2CCc3ncncc3C2)CC1 ZINC000880597492 FF On-Demand Anodyne CCR8 20 41 COCC1CN(C(=O)Cc2ccc3c(c2)N(C(=O)OC(C)(C)C)CC3)C1 ZINC000880597501 FF On-Demand Anodyne GPR119 27 42 COC(=O)[C@@H](c1ccc(Cl)cc1Cl)N1CCc2ncncc2C1 ZINC000880597551 FG On-Demand Anodyne CNR1 47 29 N#C[C@@H](c1cccs1)N1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880597575 GD On-Demand Mild PTAFR 39 48 N#C[C@H](c1cccs1)N1CCN(C(=O)CN2CCc3ncncc3C2)CC1 ZINC000880597576 GD On-Demand Mild PTAFR 39 48 CC(C)(C)OC(=O)NCCCCCCCN1CCc2ncncc2C1 ZINC000880597612 EG On-Demand Anodyne DRD2 21 49 CC(C)(C)OC(=O)NCCCCCCCN1CCc2ncncc2C1 ZINC000880597612 EG On-Demand Anodyne DRD3 46 40 CC(C)(C)OC(=O)NCCCCCCN1CCc2ncncc2C1 ZINC000880597623 EF On-Demand Anodyne DRD2 21 49 CC(C)(C)OC(=O)NCCCCCCN1CCc2ncncc2C1 ZINC000880597623 EF On-Demand Anodyne DRD3 46 40 COCC1CN(C(=O)CNC(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597627 FC On-Demand Anodyne F2 21 42 COCC1CN(C(=O)CNC(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597627 FC On-Demand Anodyne CELA1 44 34 COCC1CN(C(=O)CNC(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597627 FC On-Demand Anodyne PREP 22 49 COCC1CN(C(=O)CNC(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597629 FC On-Demand Anodyne F2 21 42 COCC1CN(C(=O)CNC(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597629 FC On-Demand Anodyne CELA1 44 34 COCC1CN(C(=O)CNC(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880597629 FC On-Demand Anodyne PREP 22 49 NC(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597680 CD On-Demand Anodyne ABCB1B 31 42 NC(=O)c1ccc(CCN2CCc3ncncc3C2)cc1 ZINC000880597680 CD On-Demand Anodyne ABCG2 28 42 COCC1CN(C(=O)CC[C@@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880597704 DD On-Demand Anodyne CTSK 15 40 COCC1CN(C(=O)CC[C@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880597705 DD On-Demand Anodyne CTSK 15 40 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2ccccc2Cl)c1 ZINC000880597712 EF On-Demand Anodyne TYK2 41 43 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2ccccc2Cl)c1 ZINC000880597713 EF On-Demand Anodyne TYK2 41 43 CN(C)Cc1ccnc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)c1 ZINC000880597731 GE On-Demand Anodyne EPHX2 16 44 CN(C)Cc1ccnc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)c1 ZINC000880597731 GE On-Demand Anodyne CACNA1I 56 34 C[C@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1cc(CN(C)C)ccn1 ZINC000880597733 GF On-Demand Anodyne GPR119 38 42 C[C@@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1cc(CN(C)C)ccn1 ZINC000880597734 GF On-Demand Anodyne GPR119 38 42 CN(C)Cc1ccnc(NC(=O)NCc2ccon2)c1 ZINC000880597740 CD On-Demand Anodyne KIT 18 42 CN(C)Cc1ccnc(NC(=O)NCc2ccon2)c1 ZINC000880597740 CD On-Demand Anodyne BRAF 16 42 N#CCCNC(=O)CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597770 ED On-Demand Mild CTSF 43 34 N#CCCNC(=O)CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597771 ED On-Demand Mild CTSF 43 34 N#CCCNC(=O)CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597772 ED On-Demand Mild CTSF 43 34 N#CCCNC(=O)CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597773 ED On-Demand Mild CTSF 43 34 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne F2 47 41 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne ACE 46 45 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne FKBP1A 82 50 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CELA1 29 65 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne GRIN2B 23 42 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne ELANE 29 44 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CTRA_BOVIN 64 35 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne TRY1_BOVIN 62 35 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CTSG 43 33 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CPT1A 40 41 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CPT2 48 41 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne PREP 150 72 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne CELA2A 52 35 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne LGMN 85 49 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne ACE2 20 44 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne KLK5 28 50 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne WNT3 44 35 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne SLC12A5 70 40 COCC1CN(C(=O)[C@H]2CCCN2C(=O)OCc2ccccc2)C1 ZINC000880597783 ED On-Demand Anodyne TMPRSS11D 55 37 CNS(=O)(=O)c1ccc(CN2CCc3ncncc3C2)cc1 ZINC000880597794 DC On-Demand Anodyne NOD2 40 35 COCC1CN(C(=O)c2ccc3c(c2)CCN3C(=O)OC(C)(C)C)C1 ZINC000880597796 EF On-Demand Anodyne GPR119 24 48 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(F)c1 ZINC000880597831 DE On-Demand Anodyne IKBKB 50 30 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(F)c1 ZINC000880597831 DE On-Demand Anodyne ENV 40 35 O=C(CN1CCc2ncncc2C1)Nc1ccc(Cl)c(F)c1 ZINC000880597831 DE On-Demand Anodyne IMDH_CRYPV 33 41 COC(=O)NCc1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880597855 FF On-Demand Anodyne ROCK2 16 44 COC(=O)NCc1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880597855 FF On-Demand Anodyne PDGFRA 40 35 FC(F)(F)OCCCN1CCc2ncncc2C1 ZINC000880597859 CD On-Demand Anodyne HTR5A 19 40 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2c(F)cccc2Cl)c1 ZINC000880597864 FF On-Demand Anodyne TYK2 37 42 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2c(F)cccc2Cl)c1 ZINC000880597865 FF On-Demand Anodyne TYK2 37 42 COC(=O)N(C)Cc1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880597883 FF On-Demand Anodyne RAF1 18 40 COC(=O)N(C)Cc1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880597883 FF On-Demand Anodyne PDGFRA 44 36 CN(C)Cc1ccnc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880597884 FH On-Demand Anodyne HTR1F 43 33 CN(C)Cc1ccnc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)c1 ZINC000880597884 FH On-Demand Anodyne CCR1 31 42 COCC1CN(C(=O)/C(=C\c2ccccc2)OC)C1 ZINC000880597885 CD On-Demand Anodyne TLR4 25 42 COCC1CN(C(=O)/C(=C/c2ccccc2)OC)C1 ZINC000880597886 CD On-Demand Anodyne TLR4 25 42 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne FKBP1A 33 43 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne CELA1 19 43 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne GRIN2B 44 48 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne CCR5 19 43 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne PREP 50 48 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne TGM2 31 42 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne F13A1 30 42 COCC1CN(C(=O)[C@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597887 ED On-Demand Anodyne SLC12A5 63 39 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne FKBP1A 33 43 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne CELA1 19 43 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne GRIN2B 44 48 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne CCR5 19 43 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne PREP 50 48 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne TGM2 31 42 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne F13A1 30 42 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880597888 ED On-Demand Anodyne SLC12A5 63 39 COCC1CN(C(=O)[C@@H](COC)NC(=O)OC(C)(C)C)C1 ZINC000880597902 DC On-Demand Anodyne PAPA1_CARPA 36 42 COCC1CN(C(=O)[C@@H](COC)NC(=O)OC(C)(C)C)C1 ZINC000880597902 DC On-Demand Anodyne CTSK 16 43 COCC1CN(C(=O)[C@@H](COC)NC(=O)OC(C)(C)C)C1 ZINC000880597902 DC On-Demand Anodyne POLG_HCV1 23 42 CC(C)(C)C(=O)NNC(=O)CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597906 GD On-Demand Reactive MME 66 38 CC(C)(C)C(=O)NNC(=O)CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597907 GD On-Demand Reactive MME 66 38 CC(C)(C)C(=O)NNC(=O)CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597908 GD On-Demand Reactive MME 66 38 CC(C)(C)C(=O)NNC(=O)CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597909 GD On-Demand Reactive MME 66 38 CN(C)Cc1ccnc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)c1 ZINC000880597914 EH On-Demand Anodyne CCR1 38 40 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)c1 ZINC000880597915 EH On-Demand Anodyne CCR1 38 40 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive ACE 39 41 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive MME 106 41 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive ANPEP 44 39 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CTSB 41 37 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive PAPA1_CARPA 45 35 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CYSP_TRYCR 49 34 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CTSF 42 34 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CAPNS1 57 32 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive HLA-DRB1 44 32 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CAPN1 55 36 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive CAPN2 60 35 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive ACE2 58 36 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive FPR1 42 33 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597917 FD On-Demand Reactive Q82323_9DELA 54 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive ACE 39 41 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive MME 106 41 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive ANPEP 44 39 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CTSB 41 37 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive PAPA1_CARPA 45 35 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CYSP_TRYCR 49 34 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CTSF 42 34 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CAPNS1 57 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive HLA-DRB1 44 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CAPN1 55 36 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive CAPN2 60 35 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive ACE2 58 36 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive FPR1 42 33 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880597918 FD On-Demand Reactive Q82323_9DELA 54 32 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive ACE 39 41 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive MME 106 41 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive ANPEP 44 39 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CTSB 41 37 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive PAPA1_CARPA 45 35 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CYSP_TRYCR 49 34 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CTSF 42 34 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CAPNS1 57 32 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive HLA-DRB1 44 32 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CAPN1 55 36 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive CAPN2 60 35 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive ACE2 58 36 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive FPR1 42 33 CCC(=O)NNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597919 FD On-Demand Reactive Q82323_9DELA 54 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive ACE 39 41 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive MME 106 41 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive ANPEP 44 39 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CTSB 41 37 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive PAPA1_CARPA 45 35 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CYSP_TRYCR 49 34 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CTSF 42 34 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CAPNS1 57 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive HLA-DRB1 44 32 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CAPN1 55 36 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive CAPN2 60 35 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive ACE2 58 36 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive FPR1 42 33 CCC(=O)NNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880597920 FD On-Demand Reactive Q82323_9DELA 54 32 COCC1CN(C(=O)c2cnc(C3CCN(C(=O)OC(C)(C)C)CC3)o2)C1 ZINC000880597925 GF On-Demand Anodyne GPR119 47 42 COCC1CN(C(=O)c2ncccc2Oc2ccccc2)C1 ZINC000880597926 CF On-Demand Anodyne TSPO 47 30 COCC1CN(C(=O)c2cc(-c3ccccc3C(F)(F)F)on2)C1 ZINC000880597944 EG On-Demand Anodyne RBP4 47 36 COCC1CN(C(=O)c2cc3c(Br)c(F)ccc3[nH]2)C1 ZINC000880597946 EF On-Demand Anodyne HRH4 25 47 COCC1CN(C(=O)Cc2ccc(Cl)c(F)c2)C1 ZINC000880597950 CE On-Demand Anodyne OPRK1 18 41 O=C(CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NNC(=O)c1ccccc1 ZINC000880597953 GD On-Demand Reactive CTRB1 35 41 O=C(CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NNC(=O)c1ccccc1 ZINC000880597954 GD On-Demand Reactive CTRB1 35 41 O=C(CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NNC(=O)c1ccccc1 ZINC000880597955 GD On-Demand Reactive CTRB1 35 41 O=C(CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NNC(=O)c1ccccc1 ZINC000880597956 GD On-Demand Reactive CTRB1 35 41 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CTSB 28 49 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CYSP_TRYCR 41 35 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CTSK 29 49 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CTSL 39 49 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne PREP 27 40 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CAPNS1 52 31 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CAPN1 41 35 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne CAPN2 65 35 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne NPR 48 31 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne NAAA 54 37 COCC1CN(C(=O)[C@H]2C[C@@H](NC(=O)OCc3ccccc3)C2)C1 ZINC000880597964 ED On-Demand Anodyne SLC12A5 65 34 O=C(CN1CCc2ncncc2C1)Nc1ccccn1 ZINC000880597984 CC On-Demand Anodyne SLC27A1 32 40 c1ccc2c(c1)CC[C@H]2CCN1CCc2ncncc2C1 ZINC000880598005 CF On-Demand Anodyne EBP 17 46 c1ccc2c(c1)CC[C@@H]2CCN1CCc2ncncc2C1 ZINC000880598007 CF On-Demand Anodyne EBP 17 46 COC(=O)c1ccc2nc(CN3CCc4ncncc4C3)[nH]c2c1 ZINC000880598012 DD On-Demand Anodyne ABCG2 30 40 N#C[C@@H](c1ccccc1)N1CCc2ncncc2C1 ZINC000880598024 CE On-Demand Mild PTAFR 27 44 N#C[C@H](c1ccccc1)N1CCc2ncncc2C1 ZINC000880598025 CE On-Demand Mild PTAFR 27 44 COCC1CN(C(=O)COC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880598033 ED On-Demand Anodyne GPR119 34 44 CC(=O)c1ccccc1NC(=O)CCCN1CCc2ncncc2C1 ZINC000880598067 EE On-Demand Anodyne HTR7 15 41 CC(=O)c1ccccc1NC(=O)CCCN1CCc2ncncc2C1 ZINC000880598067 EE On-Demand Anodyne ABCB1B 32 42 CC(=O)c1ccccc1NC(=O)CCCN1CCc2ncncc2C1 ZINC000880598067 EE On-Demand Anodyne ABCB1 15 42 CC(=O)c1ccccc1NC(=O)CCCN1CCc2ncncc2C1 ZINC000880598067 EE On-Demand Anodyne ABCG2 28 42 COCC1CN(C(=O)c2cccc([C@H]3CCCN(C)C3)c2)C1 ZINC000880598106 DE On-Demand Anodyne L3MBTL3 49 40 COCC1CN(C(=O)c2cccc([C@@H]3CCCN(C)C3)c2)C1 ZINC000880598108 DE On-Demand Anodyne L3MBTL3 49 40 COCC1CN(C(=O)CN(C)C(=O)OCc2ccccc2)C1 ZINC000880598114 DD On-Demand Anodyne FKBP1A 15 40 COCC1CN(C(=O)CN(C)C(=O)OCc2ccccc2)C1 ZINC000880598114 DD On-Demand Anodyne SLC12A5 67 35 COCC1CN(C(=O)[C@@H]2CSCN2C(=O)OC(C)(C)C)C1 ZINC000880598119 DD On-Demand Anodyne PREP 19 40 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598145 DD On-Demand Anodyne LUXR 75 44 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598145 DD On-Demand Anodyne TRAR 85 46 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598145 DD On-Demand Anodyne LASR 51 46 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598147 DD On-Demand Anodyne LUXR 75 44 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598147 DD On-Demand Anodyne TRAR 85 46 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598147 DD On-Demand Anodyne LASR 51 46 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598148 DD On-Demand Anodyne LUXR 75 44 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598148 DD On-Demand Anodyne TRAR 85 46 O=C1OCC[C@@H]1N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598148 DD On-Demand Anodyne LASR 51 46 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598150 DD On-Demand Anodyne LUXR 75 44 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598150 DD On-Demand Anodyne TRAR 85 46 O=C1OCC[C@@H]1N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598150 DD On-Demand Anodyne LASR 51 46 COCC1CN(C(=O)C(F)(F)c2ccccc2NC(C)=O)C1 ZINC000880598152 DD On-Demand Anodyne RBP4 65 35 COCC1CN(C(=O)c2ccc3c(c2)CCCN3C(=O)OC(C)(C)C)C1 ZINC000880598153 FG On-Demand Anodyne GPR119 23 43 COCC1CN(C(=O)[C@H]2CCC[C@@H]2c2ccccc2)C1 ZINC000880598154 CF On-Demand Anodyne SLC6A3 16 47 COCC1CN(C(=O)[C@H]2CCC[C@@H]2c2ccccc2)C1 ZINC000880598154 CF On-Demand Anodyne CCR5 17 42 COCC1CN(C(=O)[C@H]2CCC[C@H]2c2ccccc2)C1 ZINC000880598156 CF On-Demand Anodyne SLC6A3 16 47 COCC1CN(C(=O)[C@H]2CCC[C@H]2c2ccccc2)C1 ZINC000880598156 CF On-Demand Anodyne CCR5 17 42 COCC1CN(C(=O)[C@@H]2CCC[C@@H]2c2ccccc2)C1 ZINC000880598158 CF On-Demand Anodyne SLC6A3 16 47 COCC1CN(C(=O)[C@@H]2CCC[C@@H]2c2ccccc2)C1 ZINC000880598158 CF On-Demand Anodyne CCR5 17 42 COCC1CN(C(=O)[C@@H]2CCC[C@H]2c2ccccc2)C1 ZINC000880598161 CF On-Demand Anodyne SLC6A3 16 47 COCC1CN(C(=O)[C@@H]2CCC[C@H]2c2ccccc2)C1 ZINC000880598161 CF On-Demand Anodyne CCR5 17 42 COCC1CN(C(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598163 GG On-Demand Anodyne PGC 46 34 COCC1CN(C(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598163 GG On-Demand Anodyne PAPA1_CARPA 35 40 COCC1CN(C(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598163 GG On-Demand Anodyne CTSK 15 44 COCC1CN(C(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598163 GG On-Demand Anodyne REN 42 36 COCC1CN(C(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598163 GG On-Demand Anodyne FPR1 46 37 COCC1CN(C(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598165 GG On-Demand Anodyne PGC 46 34 COCC1CN(C(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598165 GG On-Demand Anodyne PAPA1_CARPA 35 40 COCC1CN(C(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598165 GG On-Demand Anodyne CTSK 15 44 COCC1CN(C(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598165 GG On-Demand Anodyne REN 42 36 COCC1CN(C(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880598165 GG On-Demand Anodyne FPR1 46 37 COCC1CN(C(=O)[C@H]2CCN(C(=O)OC(C)(C)C)CC2(F)F)C1 ZINC000880598171 ED On-Demand Anodyne GPR119 31 40 COCC1CN(C(=O)[C@@H]2CCN(C(=O)OC(C)(C)C)CC2(F)F)C1 ZINC000880598173 ED On-Demand Anodyne GPR119 31 40 CN(C)Cc1ccnc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880598180 FG On-Demand Anodyne TYK2 22 42 CN(C)Cc1ccnc(NC(=O)NC2CCC(N3CCCCC3)CC2)c1 ZINC000880598180 FG On-Demand Anodyne L3MBTL3 72 36 CN(C)Cc1ccnc(NC(=O)N2CCc3c(F)cccc3C2)c1 ZINC000880598203 EF On-Demand Anodyne P2RY14 42 32 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598207 ED On-Demand Mild MME 83 39 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598207 ED On-Demand Mild CTSD 16 40 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598207 ED On-Demand Mild PAPA1_CARPA 46 39 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598207 ED On-Demand Mild CTSF 46 35 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598207 ED On-Demand Mild AMP1_PLAFQ 41 36 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598209 ED On-Demand Mild MME 83 39 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598209 ED On-Demand Mild CTSD 16 40 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598209 ED On-Demand Mild PAPA1_CARPA 46 39 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598209 ED On-Demand Mild CTSF 46 35 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598209 ED On-Demand Mild AMP1_PLAFQ 41 36 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598210 ED On-Demand Mild MME 83 39 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598210 ED On-Demand Mild CTSD 16 40 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598210 ED On-Demand Mild PAPA1_CARPA 46 39 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598210 ED On-Demand Mild CTSF 46 35 C#CCNC(=O)[C@H](C)N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598210 ED On-Demand Mild AMP1_PLAFQ 41 36 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598212 ED On-Demand Mild MME 83 39 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598212 ED On-Demand Mild CTSD 16 40 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598212 ED On-Demand Mild PAPA1_CARPA 46 39 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598212 ED On-Demand Mild CTSF 46 35 C#CCNC(=O)[C@H](C)N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598212 ED On-Demand Mild AMP1_PLAFQ 41 36 COCC1CN(C(=O)[C@@H](CCC(=O)OC)NC(=O)OC(C)(C)C)C1 ZINC000880598222 EC On-Demand Anodyne POLG_HCV1 22 41 COCC1CN(C(=O)[C@H](CCC(=O)OC)NC(=O)OC(C)(C)C)C1 ZINC000880598224 EC On-Demand Anodyne POLG_HCV1 22 41 CN(C)Cc1ccnc(NC(=O)NCCNc2ccccc2)c1 ZINC000880598236 DE On-Demand Anodyne ADRB1 40 31 CN(C)Cc1ccnc(NC(=O)NCCNc2ccccc2)c1 ZINC000880598236 DE On-Demand Anodyne KIT 17 43 CN(C)Cc1ccnc(NC(=O)NCCNc2ccccc2)c1 ZINC000880598236 DE On-Demand Anodyne BRAF 22 43 CN(C)Cc1ccnc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880598251 GE On-Demand Anodyne NPY1R 25 41 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c1 ZINC000880598252 GE On-Demand Anodyne NPY1R 25 41 c1ncc2c(n1)CCN(Cc1ccc(CN3CCCCC3)cc1)C2 ZINC000880598258 DG On-Demand Anodyne HRH3 32 49 COCC1CN(C(=O)c2ccc3c(c2)CCN3C)C1 ZINC000880598263 CD On-Demand Anodyne SRD5A1 19 40 CN(C)Cc1ccnc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c1 ZINC000880598264 GF On-Demand Anodyne FAAH 26 45 CN(C)Cc1ccnc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c1 ZINC000880598264 GF On-Demand Anodyne NACHRBETA2 49 35 COCC1CN(C(=O)c2ccc(C(=O)c3cccc(O)c3)cc2)C1 ZINC000880598266 EE On-Demand Anodyne HSD17B1 24 42 COCC1CN(C(=O)c2ccc(C(=O)c3cccc(O)c3)cc2)C1 ZINC000880598266 EE On-Demand Anodyne HSD17B2 28 42 CN(C)Cc1ccnc(NC(=O)NCC2Cc3ccccc3C2)c1 ZINC000880598269 DF On-Demand Anodyne TYK2 15 41 COc1cccc(SCCN2CCc3ncncc3C2)c1 ZINC000880598276 DF On-Demand Anodyne ABCB1 20 43 COC(=O)c1ccc(OC)c(CN2CCc3ncncc3C2)c1 ZINC000880598283 DD On-Demand Anodyne SLC9A1 44 31 COC(=O)c1ccc(OC)c(CN2CCc3ncncc3C2)c1 ZINC000880598283 DD On-Demand Anodyne NOD2 40 35 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880598286 FC On-Demand Anodyne ACOX1 48 31 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880598286 FC On-Demand Anodyne ABCB1 43 40 COc1ccc(O)c(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598289 EE On-Demand Clean PDGFRB 27 43 COc1ccc(O)c(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598289 EE On-Demand Clean MTNR1A 16 40 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598291 DC On-Demand Mild MME 52 38 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598291 DC On-Demand Mild PAPA1_CARPA 39 40 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598291 DC On-Demand Mild CTSL 19 40 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598292 DC On-Demand Mild MME 52 38 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598292 DC On-Demand Mild PAPA1_CARPA 39 40 C#CCNC(=O)CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598292 DC On-Demand Mild CTSL 19 40 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598293 DC On-Demand Mild MME 52 38 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598293 DC On-Demand Mild PAPA1_CARPA 39 40 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880598293 DC On-Demand Mild CTSL 19 40 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598294 DC On-Demand Mild MME 52 38 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598294 DC On-Demand Mild PAPA1_CARPA 39 40 C#CCNC(=O)CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880598294 DC On-Demand Mild CTSL 19 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598296 FG On-Demand Mild ROCK2 31 42 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598296 FG On-Demand Mild PDS 54 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598297 FG On-Demand Mild ROCK2 31 42 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880598297 FG On-Demand Mild PDS 54 36 CC(C)(C)OC(=O)N1CCC(CCCN2CCc3ncncc3C2)CC1 ZINC000880598301 FG On-Demand Anodyne GPR119 51 49 CN(C)Cc1ccnc(NC(=O)N2CCOC[C@H]2C[C@H](O)c2ccccc2)c1 ZINC000880598334 GE On-Demand Anodyne CASR 41 35 CN(C)Cc1ccnc(NC(=O)N2CCOC[C@@H]2C[C@H](O)c2ccccc2)c1 ZINC000880598335 GE On-Demand Anodyne CASR 41 35 CN(C)Cc1ccnc(NC(=O)N2CCOC[C@@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880598337 GE On-Demand Anodyne CASR 41 35 CN(C)Cc1ccnc(NC(=O)N2CCOC[C@H]2C[C@@H](O)c2ccccc2)c1 ZINC000880598338 GE On-Demand Anodyne CASR 41 35 CC(C)(C)OC(=O)N1CCC([C@@H](O)CN2CCc3ncncc3C2)CC1 ZINC000880598360 FD On-Demand Anodyne GPR119 53 43 CC(C)(C)OC(=O)N1CCC([C@H](O)CN2CCc3ncncc3C2)CC1 ZINC000880598361 FD On-Demand Anodyne GPR119 53 43 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880598365 CD On-Demand Anodyne PAPA1_CARPA 34 42 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880598365 CD On-Demand Anodyne CTSK 17 40 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(COC)C1 ZINC000880598365 CD On-Demand Anodyne POLG_HCV1 22 40 COc1ccccc1-c1nc(CN2CCc3ncncc3C2)co1 ZINC000880598370 DF On-Demand Anodyne ABCB1 15 49 COCC1CN(C(=O)CN2CCCC[C@@H](OCc3ccccc3)C2=O)C1 ZINC000880598384 FD On-Demand Anodyne ACE 21 43 COCC1CN(C(=O)CN2CCCC[C@@H](OCc3ccccc3)C2=O)C1 ZINC000880598384 FD On-Demand Anodyne FKBP1A 39 41 COCC1CN(C(=O)CN2CCCC[C@@H](OCc3ccccc3)C2=O)C1 ZINC000880598384 FD On-Demand Anodyne F10 15 40 COCC1CN(C(=O)CN2CCCC[C@@H](OCc3ccccc3)C2=O)C1 ZINC000880598384 FD On-Demand Anodyne PREP 45 38 COCC1CN(C(=O)CN2CCCC[C@H](OCc3ccccc3)C2=O)C1 ZINC000880598390 FD On-Demand Anodyne ACE 21 43 COCC1CN(C(=O)CN2CCCC[C@H](OCc3ccccc3)C2=O)C1 ZINC000880598390 FD On-Demand Anodyne FKBP1A 39 41 COCC1CN(C(=O)CN2CCCC[C@H](OCc3ccccc3)C2=O)C1 ZINC000880598390 FD On-Demand Anodyne F10 15 40 COCC1CN(C(=O)CN2CCCC[C@H](OCc3ccccc3)C2=O)C1 ZINC000880598390 FD On-Demand Anodyne PREP 45 38 COc1cc(CN2CCc3ncncc3C2)ccc1Cl ZINC000880598395 CF On-Demand Anodyne DRD4 21 44 COc1cc(CN2CCc3ncncc3C2)ccc1Cl ZINC000880598395 CF On-Demand Anodyne SSTR5 40 39 COc1cc(CN2CCc3ncncc3C2)ccc1Cl ZINC000880598395 CF On-Demand Anodyne ABCB1 21 46 CN(C)Cc1ccnc(NC(=O)Nc2ccc(CN3CCOC3=O)cc2)c1 ZINC000880598421 FF On-Demand Anodyne MTOR 18 40 COCC1CN(C(=O)[C@@]2(C)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880598431 EE On-Demand Anodyne GRIN2B 19 41 COCC1CN(C(=O)[C@@]2(C)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880598431 EE On-Demand Anodyne SLC12A5 69 39 COCC1CN(C(=O)[C@]2(C)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880598433 EE On-Demand Anodyne GRIN2B 19 41 COCC1CN(C(=O)[C@]2(C)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880598433 EE On-Demand Anodyne SLC12A5 69 39 COCC1CN(C(=O)CSC2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880598457 FE On-Demand Anodyne GPR119 32 40 CN(C)Cc1ccnc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880598462 FH On-Demand Anodyne CACNA1H 41 33 CN(C)Cc1ccnc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880598462 FH On-Demand Anodyne CCR1 18 42 CN(C)Cc1ccnc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880598462 FH On-Demand Anodyne CCR5 73 33 CN(C)Cc1ccnc(NC(=O)N2CCC(c3cccc(F)c3)CC2)c1 ZINC000880598462 FH On-Demand Anodyne LIPE 15 42 COCC1CN(C(=O)[C@@H](CCN(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880598487 EC On-Demand Anodyne POLG_HCV1 22 40 COCC1CN(C(=O)[C@H](CCN(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880598489 EC On-Demand Anodyne POLG_HCV1 22 40 O=C(CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)Nc1ccc(O)cc1 ZINC000880598491 FE On-Demand Anodyne MME 35 40 O=C(CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)Nc1ccc(O)cc1 ZINC000880598493 FE On-Demand Anodyne MME 35 40 O=C(CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)Nc1ccc(O)cc1 ZINC000880598495 FE On-Demand Anodyne MME 35 40 O=C(CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)Nc1ccc(O)cc1 ZINC000880598497 FE On-Demand Anodyne MME 35 40 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1F ZINC000880598534 GF On-Demand Clean PDGFRB 43 37 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1F ZINC000880598534 GF On-Demand Clean CCR1 23 40 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)cc1F ZINC000880598534 GF On-Demand Clean RBP4 17 40 COCC1CN(C(=O)c2ccc3c(c2)CCN(C(=O)OC(C)(C)C)CC3)C1 ZINC000880598588 FF On-Demand Anodyne GPR119 39 40 N#Cc1ccccc1OC[C@@H](O)CN1CCc2ncncc2C1 ZINC000880598594 DD On-Demand Mild ADRB1 55 37 N#Cc1ccccc1OC[C@@H](O)CN1CCc2ncncc2C1 ZINC000880598594 DD On-Demand Mild ABCB1 56 40 N#Cc1ccccc1OC[C@H](O)CN1CCc2ncncc2C1 ZINC000880598595 DD On-Demand Mild ADRB1 55 37 N#Cc1ccccc1OC[C@H](O)CN1CCc2ncncc2C1 ZINC000880598595 DD On-Demand Mild ABCB1 56 40 FC(F)(F)Oc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880598606 DF On-Demand Anodyne NOD2 24 40 O=C(CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NCc1ccccn1 ZINC000880598643 FD On-Demand Anodyne GPR142 48 38 O=C(CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NCc1ccccn1 ZINC000880598644 FD On-Demand Anodyne GPR142 48 38 O=C(CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NCc1ccccn1 ZINC000880598645 FD On-Demand Anodyne GPR142 48 38 O=C(CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NCc1ccccn1 ZINC000880598646 FD On-Demand Anodyne GPR142 48 38 COCC1CN(C(=O)[C@H](C)[C@@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880598660 DD On-Demand Anodyne CTSK 15 40 COCC1CN(C(=O)[C@H](C)[C@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880598661 DD On-Demand Anodyne CTSK 15 40 COCC1CN(C(=O)[C@@H](C)[C@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880598662 DD On-Demand Anodyne CTSK 15 40 COCC1CN(C(=O)[C@@H](C)[C@@H](C)NC(=O)OC(C)(C)C)C1 ZINC000880598663 DD On-Demand Anodyne CTSK 15 40 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2c(Cl)cccc2Cl)c1 ZINC000880598691 GG On-Demand Anodyne TYK2 51 46 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2c(Cl)cccc2Cl)c1 ZINC000880598693 GG On-Demand Anodyne TYK2 51 46 COCC1CN(C(=O)CN2C(=O)C(F)(F)c3cc([N+](=O)[O-])ccc32)C1 ZINC000880598695 FD On-Demand Bother CACNA1D 50 34 COCC1CN(C(=O)[C@@H]2CC(c3cccc(OC)c3)=NO2)C1 ZINC000880598719 DD On-Demand Anodyne LUCI_PHOPY 41 48 COCC1CN(C(=O)[C@H]2CC(c3cccc(OC)c3)=NO2)C1 ZINC000880598720 DD On-Demand Anodyne LUCI_PHOPY 41 48 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne CTSK 25 53 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne CACNA1B 22 46 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne ECE1 23 40 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne REN 64 46 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne CTSS 24 57 COCC1CN(C(=O)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598724 FF On-Demand Anodyne FPR1 15 45 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne CTSK 25 53 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne CACNA1B 22 46 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne ECE1 23 40 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne REN 64 46 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne CTSS 24 57 COCC1CN(C(=O)[C@@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C1 ZINC000880598725 FF On-Demand Anodyne FPR1 15 45 COCC1CN(C(=O)c2ccc(C(=O)OCc3ccccc3)[nH]2)C1 ZINC000880598726 EE On-Demand Anodyne CACNA1C 19 40 COCC1CN(C(=O)c2ccc(C(=O)OCc3ccccc3)[nH]2)C1 ZINC000880598726 EE On-Demand Anodyne SLC12A5 45 33 COCC1CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)c2c(F)cccc2F)C1 ZINC000880598758 FF On-Demand Anodyne PAPA1_CARPA 31 40 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2c(F)cccc2F)C1 ZINC000880598759 FF On-Demand Anodyne PAPA1_CARPA 31 40 COCC1CN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880598773 CC On-Demand Anodyne PREP 44 43 COCC1CN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880598774 CC On-Demand Anodyne PREP 44 43 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne CTSK 28 45 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne PREP 15 42 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne CAPN2 49 37 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne NPR 57 35 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne SLC12A5 67 38 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne HCN1 49 31 COCC1CN(C(=O)CC2(CNC(=O)OCc3ccccc3)CCCCC2)C1 ZINC000880598779 GG On-Demand Anodyne HCN4 47 31 c1cc(CN2CCCCC2)cc(CN2CCc3ncncc3C2)c1 ZINC000880598780 DG On-Demand Anodyne HRH3 25 44 CSc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880598781 ED On-Demand Anodyne ACOX1 53 33 CSc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880598782 ED On-Demand Anodyne ACOX1 53 33 CCOC(=O)Nc1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880598794 FG On-Demand Anodyne PDGFRA 41 35 O=C1CCc2cc(OC[C@@H](O)CN3CCc4ncncc4C3)ccc2N1 ZINC000880598798 FD On-Demand Anodyne ACOX1 71 35 O=C1CCc2cc(OC[C@H](O)CN3CCc4ncncc4C3)ccc2N1 ZINC000880598799 FD On-Demand Anodyne ACOX1 71 35 CC(C)(C)OC(=O)N1CC[C@H](CCN2CCc3ncncc3C2)C1 ZINC000880598823 EE On-Demand Anodyne GPR119 44 42 CC(C)(C)OC(=O)N1CC[C@@H](CCN2CCc3ncncc3C2)C1 ZINC000880598824 EE On-Demand Anodyne GPR119 44 42 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880598835 GF On-Demand Anodyne GPR119 44 37 CN(C)Cc1ccnc(NC(=O)N[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880598836 GF On-Demand Anodyne GPR119 44 37 c1ccc(COCCN2CCc3ncncc3C2)cc1 ZINC000880598859 CE On-Demand Anodyne LTA4H 21 40 c1ccc(COCCN2CCc3ncncc3C2)cc1 ZINC000880598859 CE On-Demand Anodyne HTR5A 22 46 CC(C)(C)OC(=O)N1CC(CCN2CCc3ncncc3C2)C1 ZINC000880598862 DE On-Demand Anodyne GPR119 36 40 COCC1CN(C(=O)c2cc(=O)c3cc(Br)ccc3o2)C1 ZINC000880598904 FE On-Demand Anodyne GPR35 46 33 O=C(CCCN1CCc2ncncc2C1)c1ccc(Br)cc1 ZINC000880598931 FG On-Demand Anodyne CYP2J2 50 35 Fc1cc(OCCN2CCc3ncncc3C2)ccc1Cl ZINC000880598934 DF On-Demand Anodyne HRH3 15 41 Fc1cc(OCCN2CCc3ncncc3C2)ccc1Cl ZINC000880598934 DF On-Demand Anodyne HTR5A 21 42 COCC1CN(C(=O)Cc2cc3cc(Cl)ccc3[nH]2)C1 ZINC000880598938 CE On-Demand Anodyne PYGL 67 39 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)C2CCC2)C1 ZINC000880599017 DD On-Demand Anodyne POLG_HCV1 18 44 COCC1CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)C2CCC2)C1 ZINC000880599022 DD On-Demand Anodyne POLG_HCV1 18 44 O=C(CN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NNC(=O)C1CC1 ZINC000880599055 FC On-Demand Reactive F11 44 38 O=C(CN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NNC(=O)C1CC1 ZINC000880599056 FC On-Demand Reactive F11 44 38 O=C(CN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)NNC(=O)C1CC1 ZINC000880599057 FC On-Demand Reactive F11 44 38 O=C(CN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)NNC(=O)C1CC1 ZINC000880599058 FC On-Demand Reactive F11 44 38 C#CC(C)(C)NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880599059 CD On-Demand Mild TYK2 48 32 COCC1CN(C(=O)[C@@H](CCCC#N)NC(=O)OC(C)(C)C)C1 ZINC000880599072 ED On-Demand Mild PAPA1_CARPA 36 45 COCC1CN(C(=O)[C@H](CCCC#N)NC(=O)OC(C)(C)C)C1 ZINC000880599073 ED On-Demand Mild PAPA1_CARPA 36 45 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CTRA_BOVIN 41 31 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne KLK3 73 36 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CTSB 50 39 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CYSP_TRYCR 53 39 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CTSK 39 45 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CTSL 44 38 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CAPNS1 60 34 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CTSS 24 45 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CAPN1 69 38 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne CAPN2 108 37 COCC1CN(C(=O)CC[C@H](NC(=O)OCc2ccccc2)C(F)(F)F)C1 ZINC000880599086 GF On-Demand Anodyne NPR 60 33 COCC1CN(C(=O)C2=NOC3(CCN(C(=O)OC(C)(C)C)CC3)C2)C1 ZINC000880599103 FD On-Demand Anodyne GPR119 20 49 COCC1CN(C(=O)CCNC(=O)[C@@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880599118 FC On-Demand Anodyne PREP 16 47 COCC1CN(C(=O)CCNC(=O)[C@H]2CCCN2C(=O)OC(C)(C)C)C1 ZINC000880599119 FC On-Demand Anodyne PREP 16 47 COCC1CN(C(=O)C(=O)c2ccccc2OC)C1 ZINC000880599140 CC On-Demand Anodyne KCNA3 40 37 COCC1CN(C(=O)[C@@]2(F)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880599148 FD On-Demand Anodyne GRIN2B 19 40 COCC1CN(C(=O)[C@@]2(F)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880599148 FD On-Demand Anodyne SLC12A5 68 38 COCC1CN(C(=O)[C@]2(F)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880599149 FD On-Demand Anodyne GRIN2B 19 40 COCC1CN(C(=O)[C@]2(F)CCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880599149 FD On-Demand Anodyne SLC12A5 68 38 CN(C)Cc1ccnc(NC(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)c1 ZINC000880599165 FH On-Demand Anodyne CCR1 19 41 CN(C)Cc1ccnc(NC(=O)N2CCC[C@@H]2c2ccc(F)c(F)c2)c1 ZINC000880599166 FH On-Demand Anodyne CCR1 19 41 CN(C)Cc1ccnc(NC(=O)N(C)[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599217 GF On-Demand Anodyne GPR119 46 39 CN(C)Cc1ccnc(NC(=O)N(C)[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599218 GF On-Demand Anodyne GPR119 46 39 O=C(NCCCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(F)(F)F ZINC000880599220 FE On-Demand Anodyne AMP1_PLAFQ 34 40 O=C(NCCCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(F)(F)F ZINC000880599220 FE On-Demand Anodyne NPFFR1 41 31 O=C(NCCCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(F)(F)F ZINC000880599221 FE On-Demand Anodyne AMP1_PLAFQ 34 40 O=C(NCCCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(F)(F)F ZINC000880599221 FE On-Demand Anodyne NPFFR1 41 31 O=C(NCCCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(F)(F)F ZINC000880599222 FE On-Demand Anodyne AMP1_PLAFQ 34 40 O=C(NCCCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(F)(F)F ZINC000880599222 FE On-Demand Anodyne NPFFR1 41 31 O=C(NCCCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(F)(F)F ZINC000880599223 FE On-Demand Anodyne AMP1_PLAFQ 34 40 O=C(NCCCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(F)(F)F ZINC000880599223 FE On-Demand Anodyne NPFFR1 41 31 COCC1CN(C(=O)[C@@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599226 EF On-Demand Anodyne ALPL 45 38 COCC1CN(C(=O)[C@@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599226 EF On-Demand Anodyne DPP8 41 35 COCC1CN(C(=O)[C@@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599226 EF On-Demand Anodyne DPP9 41 35 COCC1CN(C(=O)[C@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599227 EF On-Demand Anodyne ALPL 45 38 COCC1CN(C(=O)[C@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599227 EF On-Demand Anodyne DPP8 41 35 COCC1CN(C(=O)[C@H]2CC(c3ccc(Cl)cc3Cl)=NO2)C1 ZINC000880599227 EF On-Demand Anodyne DPP9 41 35 COCC1CN(C(=O)[C@@H]2C[C@H]2c2ccccc2)C1 ZINC000880599242 BD On-Demand Anodyne SLC6A3 17 44 C[C@H]1CN(C(=O)Nc2cc(CN(C)C)ccn2)CCN1C(=O)OC(C)(C)C ZINC000880599243 GF On-Demand Anodyne GPR119 32 40 C[C@@H]1CN(C(=O)Nc2cc(CN(C)C)ccn2)CCN1C(=O)OC(C)(C)C ZINC000880599244 GF On-Demand Anodyne GPR119 32 40 COCC1CN(C(=O)c2cc(=O)c3ccc(F)cc3o2)C1 ZINC000880599270 CD On-Demand Anodyne KCNH2 15 49 COCC1CN(C(=O)CCc2cc(C(F)(F)F)ccc2Br)C1 ZINC000880599276 GH On-Demand Anodyne LIPG 46 36 COCC1CN(C(=O)[C@H](CCCCC#N)NC(=O)OC(C)(C)C)C1 ZINC000880599290 EE On-Demand Mild PAPA1_CARPA 36 45 COCC1CN(C(=O)[C@@H](CCCCC#N)NC(=O)OC(C)(C)C)C1 ZINC000880599291 EE On-Demand Mild PAPA1_CARPA 36 45 CN(C)Cc1ccnc(NC(=O)NCC[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599306 GF On-Demand Anodyne GPR119 42 42 CN(C)Cc1ccnc(NC(=O)NCC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599307 GF On-Demand Anodyne GPR119 42 42 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne HTR1A 76 54 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne DRD2 48 54 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne DRD4 42 50 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne HTR2A 49 54 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne DRD3 50 50 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne DRD5 17 45 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne HTR7 81 44 c1ccc(N2CCN(CCCN3CCc4ncncc4C3)CC2)cc1 ZINC000880599308 EE On-Demand Anodyne SIGMAR1 24 49 CN(C)c1ccc(NC(=O)CCN2CCc3ncncc3C2)cc1 ZINC000880599389 ED On-Demand Anodyne ABCB1B 49 39 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880599512 EE On-Demand Anodyne PGC 45 34 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880599512 EE On-Demand Anodyne PAPA1_CARPA 34 40 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880599512 EE On-Demand Anodyne CTSK 22 46 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880599512 EE On-Demand Anodyne REN 41 36 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)C1 ZINC000880599512 EE On-Demand Anodyne FPR1 46 37 c1ccc(CN2CC[C@H](N3CCc4ncncc4C3)C2)cc1 ZINC000880599570 CE On-Demand Anodyne DRD4 29 40 c1ccc(CN2CC[C@H](N3CCc4ncncc4C3)C2)cc1 ZINC000880599570 CE On-Demand Anodyne SIGMAR1 43 41 c1ccc(CN2CC[C@@H](N3CCc4ncncc4C3)C2)cc1 ZINC000880599572 CE On-Demand Anodyne DRD4 29 40 c1ccc(CN2CC[C@@H](N3CCc4ncncc4C3)C2)cc1 ZINC000880599572 CE On-Demand Anodyne SIGMAR1 43 41 COCCc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599583 ED On-Demand Anodyne ADRB1 19 46 COCCc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599583 ED On-Demand Anodyne ACOX1 40 32 COCCc1ccc(OC[C@@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599583 ED On-Demand Anodyne ABCB1 58 40 COCCc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599585 ED On-Demand Anodyne ADRB1 19 46 COCCc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599585 ED On-Demand Anodyne ACOX1 40 32 COCCc1ccc(OC[C@H](O)CN2CCc3ncncc3C2)cc1 ZINC000880599585 ED On-Demand Anodyne ABCB1 58 40 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1Cl ZINC000880599607 DE On-Demand Anodyne ABCG2 36 45 COC(=O)c1ccc(CN2CCc3ncncc3C2)cc1Cl ZINC000880599607 DE On-Demand Anodyne NOD2 44 38 O=C(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880599683 CE On-Demand Anodyne HTR2A 18 53 O=C(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880599683 CE On-Demand Anodyne HTR7 20 41 O=C(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880599683 CE On-Demand Anodyne HTR5A 30 53 O=C(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880599683 CE On-Demand Anodyne FAAH 42 38 O=C(CCCN1CCc2ncncc2C1)c1ccccc1 ZINC000880599683 CE On-Demand Anodyne CYP2J2 56 39 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild MME 85 38 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild ANPEP 50 35 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild PGC 41 32 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild CYSP_TRYCR 41 34 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild CTSF 45 34 C=CC[C@H](N[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599689 EE On-Demand Mild ACE2 47 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild MME 85 38 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild ANPEP 50 35 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild PGC 41 32 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild CYSP_TRYCR 41 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild CTSF 45 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599691 EE On-Demand Mild ACE2 47 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild MME 85 38 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild ANPEP 50 35 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild PGC 41 32 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild CYSP_TRYCR 41 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild CTSF 45 34 C=CC[C@H](N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)C(=O)OC ZINC000880599693 EE On-Demand Mild ACE2 47 34 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild MME 85 38 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild ANPEP 50 35 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild PGC 41 32 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild CYSP_TRYCR 41 34 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild CTSF 45 34 C=CC[C@H](N[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)C(=O)OC ZINC000880599696 EE On-Demand Mild ACE2 47 34 COCC1CN(C(=O)c2cc(C3CCN(C(=O)OC(C)(C)C)CC3)no2)C1 ZINC000880599700 GF On-Demand Anodyne GPR119 44 41 COCC1CN(C(=O)CN2CCCC[C@H](NC(=O)OC(C)(C)C)C2=O)C1 ZINC000880599742 FC On-Demand Anodyne F10 20 44 COCC1CN(C(=O)CN2CCCC[C@@H](NC(=O)OC(C)(C)C)C2=O)C1 ZINC000880599743 FC On-Demand Anodyne F10 20 44 c1ccc(Cn2cncc2CN2CCc3ncncc3C2)cc1 ZINC000880599778 DE On-Demand Anodyne CYP11B1 15 45 c1ccc(CN2CCCO[C@H](CN3CCc4ncncc4C3)C2)cc1 ZINC000880599780 EE On-Demand Anodyne DRD4 17 45 c1ccc(CN2CCCO[C@@H](CN3CCc4ncncc4C3)C2)cc1 ZINC000880599783 EE On-Demand Anodyne DRD4 17 45 CCOc1cc(CN2CCc3ncncc3C2)ccc1[N+](=O)[O-] ZINC000880599788 DE On-Demand Bother SSTR5 66 38 COCC1CN(C(=O)C(F)(F)c2ccc([N+](=O)[O-])cc2)C1 ZINC000880599810 DD On-Demand Bother SLC27A4 43 32 O=C(CCN1CCc2ncncc2C1)Nc1cccnc1 ZINC000880599820 CD On-Demand Anodyne CHRNA7 20 44 CC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880599825 CE On-Demand Anodyne P2RY14 40 36 CC(=O)c1cccc(CN2CCc3ncncc3C2)c1 ZINC000880599825 CE On-Demand Anodyne NOD2 42 36 CCCOc1cccc(CN2CCc3ncncc3C2)c1 ZINC000880599832 CF On-Demand Anodyne HRH2 28 42 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne HTR1A 56 40 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne DRD2 47 40 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne ADRA1D 24 42 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne HTR2A 23 44 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne ADRA1A 27 42 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne DRD3 47 40 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne HTR7 40 45 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne SIGMAR1 22 43 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne HTR5A 35 42 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne ABCB1B 54 36 COc1cccc(OC)c1OCCCCN1CCc2ncncc2C1 ZINC000880599846 EF On-Demand Anodyne ABCB1 29 46 CC(C)(C)OC(=O)N1CC(N2CCc3ncncc3C2)C1 ZINC000880599875 CD On-Demand Anodyne GPR119 37 40 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599895 FE On-Demand Anodyne GPR119 47 38 CN(C)Cc1ccnc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880599897 FE On-Demand Anodyne GPR119 47 38 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne ACE 41 45 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne GHRHR 59 33 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne P2RY12 180 41 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne ELANE 26 40 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTRA_BOVIN 57 38 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CASP3 15 41 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne KLK3 85 39 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTSB 70 46 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne PAPA1_CARPA 78 41 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CYSP_TRYCR 61 42 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTSG 42 33 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTSK 57 53 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTSL 55 53 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne PREP 18 42 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CAPNS1 70 40 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CELA2A 52 38 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne MMP11 66 32 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CTSS 35 53 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CAPN1 94 47 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CASP1 25 43 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne CAPN2 144 44 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne TGM2 38 48 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne TPSAB1 47 36 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne NPR 76 36 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599901 FD On-Demand Anodyne PSMB5 45 42 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne ACE 41 45 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne GHRHR 59 33 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne P2RY12 180 41 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne ELANE 26 40 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTRA_BOVIN 57 38 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CASP3 15 41 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne KLK3 85 39 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTSB 70 46 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne PAPA1_CARPA 78 41 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CYSP_TRYCR 61 42 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTSG 42 33 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTSK 57 53 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTSL 55 53 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne PREP 18 42 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CAPNS1 70 40 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CELA2A 52 38 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne MMP11 66 32 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CTSS 35 53 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CAPN1 94 47 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CASP1 25 43 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne CAPN2 144 44 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne TGM2 38 48 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne TPSAB1 47 36 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne NPR 76 36 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)N1CC(COC)C1 ZINC000880599903 FD On-Demand Anodyne PSMB5 45 42 CC(C)(C)OC(=O)N1CCN(CCN2CCc3ncncc3C2)CC1 ZINC000880599909 ED On-Demand Anodyne GPR119 40 41 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne PLG 25 40 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne PGC 53 36 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne TRY2_BOVIN 67 33 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne PAPA1_CARPA 39 47 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne TRY1_BOVIN 15 40 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne CTSK 15 42 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne CTSL 35 47 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne CACNA1B 29 41 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne REN 60 39 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne CTSS 25 47 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne ST14 42 38 COCC1CN(C(=O)[C@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599919 GE On-Demand Anodyne FPR1 53 40 CN(CCN1CCc2ncncc2C1)Cc1ccccc1 ZINC000880599922 CD On-Demand Anodyne SIGMAR1 24 49 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne PLG 25 40 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne PGC 53 36 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne TRY2_BOVIN 67 33 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne PAPA1_CARPA 39 47 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne TRY1_BOVIN 15 40 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne CTSK 15 42 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne CTSL 35 47 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne CACNA1B 29 41 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne REN 60 39 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne CTSS 25 47 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne ST14 42 38 COCC1CN(C(=O)[C@@H](Cc2cccc(OC)c2)NC(=O)OC(C)(C)C)C1 ZINC000880599923 GE On-Demand Anodyne FPR1 53 40 C[C@H](C#N)OCCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880599930 DE On-Demand Mild CTSF 40 35 C[C@H](C#N)OCCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880599931 DE On-Demand Mild CTSF 40 35 C[C@H](C#N)OCCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F ZINC000880599932 DE On-Demand Mild CTSF 40 35 C[C@H](C#N)OCCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F ZINC000880599933 DE On-Demand Mild CTSF 40 35 O=C(CCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599936 EE On-Demand Anodyne ACE 15 42 O=C(CCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599936 EE On-Demand Anodyne MME 34 42 O=C(CCN[C@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599936 EE On-Demand Anodyne PREP 32 40 O=C(CCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599937 EE On-Demand Anodyne ACE 15 42 O=C(CCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599937 EE On-Demand Anodyne MME 34 42 O=C(CCN[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)F)N1CCCC1 ZINC000880599937 EE On-Demand Anodyne PREP 32 40 O=C(CCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599938 EE On-Demand Anodyne ACE 15 42 O=C(CCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599938 EE On-Demand Anodyne MME 34 42 O=C(CCN[C@@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599938 EE On-Demand Anodyne PREP 32 40 O=C(CCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599939 EE On-Demand Anodyne ACE 15 42 O=C(CCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599939 EE On-Demand Anodyne MME 34 42 O=C(CCN[C@H](Cc1ccccc1)[C@H](O)C(F)(F)F)N1CCCC1 ZINC000880599939 EE On-Demand Anodyne PREP 32 40 COCC1CN(C(=O)c2csc(C3CCN(C(=O)OC(C)(C)C)CC3)n2)C1 ZINC000880599954 GF On-Demand Anodyne GPR119 40 41 CN(C)Cc1ccnc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880599985 EH On-Demand Anodyne CPT1A 90 42 CN(C)Cc1ccnc(NC(=O)N2CCCC[C@@H]2c2ccccc2)c1 ZINC000880599985 EH On-Demand Anodyne TYK2 17 41 CN(C)Cc1ccnc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880599986 EH On-Demand Anodyne CPT1A 90 42 CN(C)Cc1ccnc(NC(=O)N2CCCC[C@H]2c2ccccc2)c1 ZINC000880599986 EH On-Demand Anodyne TYK2 17 41 CN(C)Cc1ccnc(NC(=O)NNC(=O)C2CCC2)c1 ZINC000880599993 CD On-Demand Reactive TYK2 55 38 CN(C)Cc1ccnc(NC(=O)NC[C@@](C)(O)c2ccccc2Cl)c1 ZINC000880600009 FF On-Demand Anodyne TYK2 53 33 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne FKBP1A 44 44 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne SLC6A1 55 36 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne CELA1 20 47 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne GRIN2B 27 44 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne CCR5 23 46 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne PREP 86 55 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne DPP7 50 38 COCC1CN(C(=O)[C@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600049 EE On-Demand Anodyne SLC12A5 68 40 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne FKBP1A 44 44 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne SLC6A1 55 36 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne CELA1 20 47 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne GRIN2B 27 44 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne CCR5 23 46 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne PREP 86 55 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne DPP7 50 38 COCC1CN(C(=O)[C@@H]2CCCN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600050 EE On-Demand Anodyne SLC12A5 68 40 COc1cc(CN2CCc3ncncc3C2)ccc1C ZINC000880600084 CE On-Demand Anodyne SSTR5 42 38 COc1cc(CN2CCc3ncncc3C2)ccc1C ZINC000880600084 CE On-Demand Anodyne ABCB1B 41 35 COc1cc(CN2CCc3ncncc3C2)ccc1C ZINC000880600084 CE On-Demand Anodyne ABCB1 24 45 COCC1CN(C(=O)c2ccc(C(F)(F)F)cc2O)C1 ZINC000880600094 CE On-Demand Anodyne CACNA1B 45 37 COCC1CN(C(=O)c2ccc(C(F)(F)F)cc2O)C1 ZINC000880600094 CE On-Demand Anodyne LIPG 51 39 CN(C)Cc1ccnc(NC(=O)NC[C@](C)(O)c2ccccc2Cl)c1 ZINC000880600109 FF On-Demand Anodyne TYK2 53 33 COCC1CN(C(=O)c2cccc(S(=O)(=O)C(F)(F)F)c2)C1 ZINC000880600117 ED On-Demand Anodyne AKR1C3 44 35 COCC1CN(C(=O)c2cccc(S(=O)(=O)C(F)(F)F)c2)C1 ZINC000880600117 ED On-Demand Anodyne SFRP1 41 35 COCC1CN(C(=O)[C@H](F)Cc2ccccc2)C1 ZINC000880600119 CD On-Demand Anodyne ACE 51 36 COCC1CN(C(=O)[C@H](F)Cc2ccccc2)C1 ZINC000880600119 CD On-Demand Anodyne MME 52 36 COCC1CN(C(=O)[C@@H](F)Cc2ccccc2)C1 ZINC000880600122 CD On-Demand Anodyne ACE 51 36 COCC1CN(C(=O)[C@@H](F)Cc2ccccc2)C1 ZINC000880600122 CD On-Demand Anodyne MME 52 36 CC(C)(C)OC(=O)NCCCN1CCc2ncncc2C1 ZINC000880600149 CD On-Demand Anodyne ADRA1D 16 44 CC(C)(C)OC(=O)NCCCN1CCc2ncncc2C1 ZINC000880600149 CD On-Demand Anodyne ADRA1A 18 44 COCC1CN(C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)C)C1 ZINC000880600166 CC On-Demand Anodyne ELANE 29 44 NC(=O)c1ccc(CCN[C@@H](Cc2ccccc2)[C@@H](O)C(F)(F)F)cc1 ZINC000880600218 FE On-Demand Anodyne ANPEP 43 32 NC(=O)c1ccc(CCN[C@@H](Cc2ccccc2)[C@@H](O)C(F)(F)F)cc1 ZINC000880600218 FE On-Demand Anodyne LAP3 42 33 NC(=O)c1ccc(CCN[C@H](Cc2ccccc2)[C@@H](O)C(F)(F)F)cc1 ZINC000880600220 FE On-Demand Anodyne ANPEP 43 32 NC(=O)c1ccc(CCN[C@H](Cc2ccccc2)[C@@H](O)C(F)(F)F)cc1 ZINC000880600220 FE On-Demand Anodyne LAP3 42 33 NC(=O)c1ccc(CCN[C@@H](Cc2ccccc2)[C@H](O)C(F)(F)F)cc1 ZINC000880600221 FE On-Demand Anodyne ANPEP 43 32 NC(=O)c1ccc(CCN[C@@H](Cc2ccccc2)[C@H](O)C(F)(F)F)cc1 ZINC000880600221 FE On-Demand Anodyne LAP3 42 33 NC(=O)c1ccc(CCN[C@H](Cc2ccccc2)[C@H](O)C(F)(F)F)cc1 ZINC000880600223 FE On-Demand Anodyne ANPEP 43 32 NC(=O)c1ccc(CCN[C@H](Cc2ccccc2)[C@H](O)C(F)(F)F)cc1 ZINC000880600223 FE On-Demand Anodyne LAP3 42 33 CN(C)Cc1ccnc(NC(=O)NNc2ccc(OC(F)(F)F)cc2)c1 ZINC000880600242 FG On-Demand Reactive P2RY1 64 38 CN(C)Cc1ccnc(NC(=O)NNc2ccc(OC(F)(F)F)cc2)c1 ZINC000880600242 FG On-Demand Reactive RAF1 22 42 CN(C)Cc1ccnc(NC(=O)NNc2ccc(OC(F)(F)F)cc2)c1 ZINC000880600242 FG On-Demand Reactive EPHX2 38 42 CN(C)Cc1ccnc(NC(=O)NNc2ccc(OC(F)(F)F)cc2)c1 ZINC000880600242 FG On-Demand Reactive MCHR2 23 42 CN(C)Cc1ccnc(NC(=O)NNc2ccc(OC(F)(F)F)cc2)c1 ZINC000880600242 FG On-Demand Reactive SHH 44 42 COCC1CN(C(=O)[C@H]2C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600243 FD On-Demand Anodyne PREP 44 47 COCC1CN(C(=O)[C@H]2C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600243 FD On-Demand Anodyne Q9NAW4_PLAFA 26 40 COCC1CN(C(=O)[C@@H]2C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600244 FD On-Demand Anodyne PREP 44 47 COCC1CN(C(=O)[C@@H]2C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600244 FD On-Demand Anodyne Q9NAW4_PLAFA 26 40 CN(C)Cc1ccnc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c1 ZINC000880600260 FD On-Demand Anodyne HTR2A 24 42 CN(C)Cc1ccnc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c1 ZINC000880600260 FD On-Demand Anodyne EPHX2 22 42 N#Cc1ccc(CN2CCc3ncncc3C2)cc1F ZINC000880600280 CE On-Demand Mild KCNJ1 21 41 CN(C)Cc1ccnc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)c1 ZINC000880600284 GC On-Demand Anodyne SSTR5 44 35 COCC1CN(C(=O)C(=O)c2cc(Cl)cc(Cl)c2)C1 ZINC000880600310 DE On-Demand Anodyne CACNA1I 61 36 COCC1CN(C(=O)c2cccc(Oc3ccccn3)c2)C1 ZINC000880600315 CF On-Demand Anodyne CFTR 41 46 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne CELA1 24 40 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne PGC 54 36 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne CMA1 32 40 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne CTRA_BOVIN 20 40 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne PAPA1_CARPA 40 39 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne CTSK 30 42 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne REN 68 44 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne CAPN2 42 39 COCC1CN(C(=O)[C@H](NC(=O)OC(C)(C)C)[C@H](C)OCc2ccccc2)C1 ZINC000880600329 GF On-Demand Anodyne FPR1 49 40 CCCCCCCC[C@H](C)C(=O)N1CC(COC)C1 ZINC000880600366 CG On-Demand Mild NOD1 56 36 CCCCCCCC[C@@H](C)C(=O)N1CC(COC)C1 ZINC000880600367 CG On-Demand Mild NOD1 56 36 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne ACE 23 41 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne GHRHR 57 33 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne ELANE 35 42 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTRA_BOVIN 60 32 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CASP3 15 42 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne KLK3 74 36 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTSB 66 45 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne PAPA1_CARPA 74 39 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CYSP_TRYCR 57 42 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTSG 46 33 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTSK 47 46 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTSL 50 46 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne PREP 15 42 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne AMY2 42 29 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CAPNS1 64 36 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CELA2A 52 33 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CTSS 28 46 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CAPN1 79 51 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CAPN2 126 39 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne TGM2 34 41 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne NPR 58 39 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne CASP10 35 42 COCC1CN(C(=O)[C@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600371 EE On-Demand Anodyne PSMB5 40 38 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne ACE 23 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne GHRHR 57 33 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne ELANE 35 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTRA_BOVIN 60 32 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CASP3 15 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne KLK3 74 36 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTSB 66 45 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne PAPA1_CARPA 74 39 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CYSP_TRYCR 57 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTSG 46 33 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTSK 47 46 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTSL 50 46 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne PREP 15 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne AMY2 42 29 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CAPNS1 64 36 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CELA2A 52 33 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CTSS 28 46 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CAPN1 79 51 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CAPN2 126 39 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne TGM2 34 41 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne NPR 58 39 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne CASP10 35 42 COCC1CN(C(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)(C)C)C1 ZINC000880600372 EE On-Demand Anodyne PSMB5 40 38 CC(=O)N1CCC[C@@H]1C(=O)NNc1ccc(-c2ccc(Cl)s2)nn1 ZINC000880600409 FE On-Demand Reactive TRY1_BOVIN 56 39 CC(=O)N1CCC[C@@H]1C(=O)NNc1ccc(-c2ccc(Cl)s2)nn1 ZINC000880600409 FE On-Demand Reactive LGMN 67 33 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne FKBP1A 15 43 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne CTSK 29 44 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne PREP 23 41 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne CAPNS1 58 34 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne CAPN1 57 37 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne CAPN2 99 36 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne NPR 61 34 COCC1CN(C(=O)C2(CNC(=O)OCc3ccccc3)CCCC2)C1 ZINC000880600420 FF On-Demand Anodyne SLC12A5 69 39 COCC1CN(C(=O)C2(O)CN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600473 EC On-Demand Anodyne GRIN2B 19 41 COCC1CN(C(=O)C2(O)CN(C(=O)OCc3ccccc3)C2)C1 ZINC000880600473 EC On-Demand Anodyne SLC12A5 62 37 COCC1CN(C(=O)c2ccc(Nc3ccc(OC)cc3OC)cc2)C1 ZINC000880600485 FG On-Demand Anodyne AKR1C3 35 43 COCC1CN(C(=O)c2ccc(Nc3ccc(OC)cc3OC)cc2)C1 ZINC000880600485 FG On-Demand Anodyne AKR1C2 48 43 COCC1CN(C(=O)[C@@]2(C)C[C@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600512 GD On-Demand Anodyne SLC12A5 52 36 COCC1CN(C(=O)[C@]2(C)C[C@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600513 GD On-Demand Anodyne SLC12A5 52 36 COCC1CN(C(=O)[C@]2(C)C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600514 GD On-Demand Anodyne SLC12A5 52 36 COCC1CN(C(=O)[C@@]2(C)C[C@@H](OC)CN2C(=O)OCc2ccccc2)C1 ZINC000880600515 GD On-Demand Anodyne SLC12A5 52 36 COCC1CN(C(=O)c2cc(-c3cccc(C(F)(F)F)c3)ccn2)C1 ZINC000880600516 FG On-Demand Anodyne CACNA1B 41 33 COCC1CN(C(=O)[C@@H]2CCCC[C@H]2c2cccc(Cl)c2)C1 ZINC000880600523 DH On-Demand Anodyne MDM2 69 33 O=C(NCCCOc1ncccn1)c1ccccc1OC1CC1 ZINC000880600536 DE On-Demand Anodyne KCNA3 45 44 O=C(NCCCOc1ncccn1)c1ccccc1OC1CC1 ZINC000880600536 DE On-Demand Anodyne SCD 23 42 O=C(NCCCOc1ncccn1)c1ccccc1OC1CC1 ZINC000880600536 DE On-Demand Anodyne HCN1 69 36 O=C(NCCCOc1ncccn1)c1ccccc1OC1CC1 ZINC000880600536 DE On-Demand Anodyne HCN4 53 36 CN(C)Cc1ccnc(NC(=O)NNc2ccccc2C(F)(F)F)c1 ZINC000880600540 FG On-Demand Reactive P2RY1 33 47 CN(C)Cc1ccnc(NC(=O)NNc2ccccc2C(F)(F)F)c1 ZINC000880600540 FG On-Demand Reactive RBP4 24 41 COCC1CN(C(=O)c2cc3c(C)ccc(F)c3[nH]2)C1 ZINC000880600542 CE On-Demand Anodyne HRH4 31 54 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)CC1 ZINC000880600552 GE On-Demand Anodyne TBK1 80 35 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)CC1 ZINC000880600552 GE On-Demand Anodyne GPR119 46 48 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)CC1 ZINC000880600554 GE On-Demand Anodyne TBK1 80 35 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)CC1 ZINC000880600554 GE On-Demand Anodyne GPR119 46 48 COCC1CN(C(=O)[C@@H]2C[C@@]23CCN(C(=O)OCc2ccccc2)C3)C1 ZINC000880600555 FE On-Demand Anodyne SLC12A5 66 39 COCC1CN(C(=O)[C@@H]2C[C@]23CCN(C(=O)OCc2ccccc2)C3)C1 ZINC000880600557 FE On-Demand Anodyne SLC12A5 66 39 COCC1CN(C(=O)[C@H]2C[C@]23CCN(C(=O)OCc2ccccc2)C3)C1 ZINC000880600559 FE On-Demand Anodyne SLC12A5 66 39 COCC1CN(C(=O)[C@H]2C[C@@]23CCN(C(=O)OCc2ccccc2)C3)C1 ZINC000880600560 FE On-Demand Anodyne SLC12A5 66 39 CN(C)Cc1ccnc(NC(=O)NNC(=O)CCCc2ccccc2)c1 ZINC000880600567 FE On-Demand Reactive FAAH 52 36 CN(C)Cc1ccnc(NC(=O)NNC(=O)CCCc2ccccc2)c1 ZINC000880600567 FE On-Demand Reactive CES1 61 34 CN(C)Cc1ccnc(NC(=O)NNC(=O)CCCc2ccccc2)c1 ZINC000880600567 FE On-Demand Reactive CES1D 43 31 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(CN(C)C)ccn2)C1 ZINC000880600571 ED On-Demand Anodyne SSTR5 51 37 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(CN(C)C)ccn2)C1 ZINC000880600571 ED On-Demand Anodyne CCR8 22 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(CN(C)C)ccn2)C1 ZINC000880600573 ED On-Demand Anodyne SSTR5 51 37 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(CN(C)C)ccn2)C1 ZINC000880600573 ED On-Demand Anodyne CCR8 22 40 CN(C)Cc1ccnc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)c1 ZINC000880600580 FF On-Demand Anodyne PRSS2 56 32 CN(C)Cc1ccnc(NC(=O)NC23CCC(CC2)C3)c1 ZINC000880600593 CF On-Demand Anodyne EPHX2 42 41 CN(C)Cc1ccnc(NC(=O)N2CCC(c3ccc(N(C)C)cc3)CC2)c1 ZINC000880600597 GH On-Demand Anodyne CCR1 30 41 O=C(NCCCOc1ncccn1)c1ccc(CF)cc1 ZINC000880600600 CE On-Demand Anodyne DRD3 18 41 O=C(Cn1ccc(Br)cc1=O)NCCCOc1ncccn1 ZINC000880600605 FC On-Demand Anodyne PSMB5 15 44 COCC1CN(C(=O)c2cn([C@H]3CCCN(C(=O)OC(C)(C)C)CC3)nn2)C1 ZINC000880600610 GD On-Demand Anodyne GPR119 41 37 COCC1CN(C(=O)c2cn([C@@H]3CCCN(C(=O)OC(C)(C)C)CC3)nn2)C1 ZINC000880600611 GD On-Demand Anodyne GPR119 41 37 COCC1CN(C(=O)C(C)(C)[C@@H](O)c2cc(Cl)cc(Cl)c2)C1 ZINC000880600614 EG On-Demand Anodyne CACNA1I 44 35 COCC1CN(C(=O)C(C)(C)[C@H](O)c2cc(Cl)cc(Cl)c2)C1 ZINC000880600615 EG On-Demand Anodyne CACNA1I 44 35 COCC1CN(C(=O)c2cccc(Oc3ccc(Cl)cn3)c2)C1 ZINC000880600616 EG On-Demand Anodyne CFTR 31 40 COc1ccc(CN(CCc2ccccn2)C(=O)COC2CC2)cc1 ZINC000880600627 EF On-Demand Anodyne MMP9 16 40 COc1ccc(CN(CCc2ccccn2)C(=O)COC2CC2)cc1 ZINC000880600627 EF On-Demand Anodyne ADAM9 15 40 CC[C@@H](Nc1cccnc1Cl)C(=O)NCCCOc1ncccn1 ZINC000880600634 EE On-Demand Anodyne G2YM83_BOTF4 64 33 CC[C@H](Nc1cccnc1Cl)C(=O)NCCCOc1ncccn1 ZINC000880600635 EE On-Demand Anodyne G2YM83_BOTF4 64 33 CC(C)(C)OC(=O)N1C[C@H]2[C@@H](C1)[C@@H]2C(=O)NCCCOc1ncccn1 ZINC000880600671 FD On-Demand Anodyne GPR119 29 43 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880600688 GG On-Demand Anodyne GPR119 47 39 CN(C)Cc1ccnc(NC(=O)N[C@@H]2CCCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880600689 GG On-Demand Anodyne GPR119 47 39 COC[C@@H](O)CNC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880600690 CC On-Demand Anodyne ADRB1 41 30 O=C(NCCCOc1ncccn1)c1ccnc(C(F)(F)F)c1 ZINC000880600694 EE On-Demand Anodyne KDM4E 25 43 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880600705 FF On-Demand Anodyne CAPNS1 47 34 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880600705 FF On-Demand Anodyne CAPN1 43 36 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880600705 FF On-Demand Anodyne CAPN2 53 33 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880600705 FF On-Demand Anodyne NPR 62 32 CN(C)Cc1ccnc(NC(=O)N2Cc3ccc(Br)cc3C2)c1 ZINC000880600723 GG On-Demand Anodyne QRFPR 17 40 CC[C@@H](Nc1cccnc1Cl)C(=O)N1CC(COC)C1 ZINC000880600725 CE On-Demand Anodyne G2YM83_BOTF4 66 35 CC[C@H](Nc1cccnc1Cl)C(=O)N1CC(COC)C1 ZINC000880600726 CE On-Demand Anodyne G2YM83_BOTF4 66 35 CN(C)Cc1ccnc(NC(=O)NNC(=O)C2CCCC2)c1 ZINC000880600733 DD On-Demand Reactive TYK2 55 38 COCC1CN(C(=O)CCc2cnc(NC(=O)OC(C)(C)C)s2)C1 ZINC000880600749 FF On-Demand Anodyne MGEA5 30 40 COCC1CN(C(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880600750 CD On-Demand Anodyne MPO 52 33 COCC1CN(C(=O)c2cc(-c3ccc(Cl)cc3Cl)on2)C1 ZINC000880600779 EG On-Demand Anodyne ALPL 48 42 COCC1CN(C(=O)c2cc(-c3ccc(Cl)cc3Cl)on2)C1 ZINC000880600779 EG On-Demand Anodyne DPP8 60 37 COCC1CN(C(=O)c2cc(-c3ccc(Cl)cc3Cl)on2)C1 ZINC000880600779 EG On-Demand Anodyne DPP9 60 37 COc1cnc(C(=O)NCCCOc2ncccn2)c(F)c1 ZINC000880600834 DD On-Demand Anodyne DRD4 40 31 COc1cnc(C(=O)NCCCOc2ncccn2)c(F)c1 ZINC000880600834 DD On-Demand Anodyne MTNR1A 23 40 COc1cnc(C(=O)NCCCOc2ncccn2)c(F)c1 ZINC000880600834 DD On-Demand Anodyne MTNR1B 20 40 CN(C)Cc1ccnc(NC(=O)N[C@H]2Cc3ccc(Cl)cc3C2)c1 ZINC000880600847 EG On-Demand Anodyne TYK2 27 45 CN(C)Cc1ccnc(NC(=O)N[C@@H]2Cc3ccc(Cl)cc3C2)c1 ZINC000880600848 EG On-Demand Anodyne TYK2 27 45 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne DRD4 40 30 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne PPARG 41 39 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne PPARA 27 41 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne NQO2 35 45 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne PPARD 55 46 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne MTNR1A 82 41 COc1ccc2c(c1)CC[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880600853 EE On-Demand Anodyne MTNR1B 76 40 C[C@@H](CCc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880600859 EF On-Demand Anodyne LEF 61 37 C[C@H](CCc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880600860 EF On-Demand Anodyne LEF 61 37 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive PPIA 17 45 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive KIT 18 41 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive RAF1 21 43 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive KDR 22 41 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive TEK 35 41 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive BRAF 39 45 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive EPHB4 17 45 CN(C)Cc1ccnc(NC(=O)NNc2cccc(C(F)(F)F)c2)c1 ZINC000880600861 FG On-Demand Reactive RIPK1 41 40 CC(C)(C)OC(=O)N1CCC[C@@H](CCC(=O)NCCCOc2ncccn2)C1 ZINC000880600865 GF On-Demand Anodyne GPR119 34 41 CC(C)(C)OC(=O)N1CCC[C@H](CCC(=O)NCCCOc2ncccn2)C1 ZINC000880600866 GF On-Demand Anodyne GPR119 34 41 CC(C)(C)OC(=O)N1CCC(C#CC(=O)NCCCOc2ncccn2)CC1 ZINC000880600882 GE On-Demand Mild GPR119 46 47 O=C(O)c1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)s1 ZINC000880600903 EG On-Demand Mild GRM4 43 41 O=C(O)c1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)s1 ZINC000880600903 EG On-Demand Mild GRM5 21 43 O=C(O)c1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)s1 ZINC000880600903 EG On-Demand Mild KCNK3 60 43 CN(C)Cc1ccnc(NC(=O)NNC(=O)C2CC2)c1 ZINC000880600908 CC On-Demand Reactive TYK2 61 41 COCC1CN(C(=O)[C@H]2CCc3cc(OC)ccc32)C1 ZINC000880600910 CD On-Demand Anodyne PPARD 38 42 COCC1CN(C(=O)[C@H]2CCc3cc(OC)ccc32)C1 ZINC000880600910 CD On-Demand Anodyne MTNR1A 15 42 COCC1CN(C(=O)[C@H]2CCc3cc(OC)ccc32)C1 ZINC000880600910 CD On-Demand Anodyne MTNR1B 19 42 COCC1CN(C(=O)[C@@H]2CCc3cc(OC)ccc32)C1 ZINC000880600911 CD On-Demand Anodyne PPARD 38 42 COCC1CN(C(=O)[C@@H]2CCc3cc(OC)ccc32)C1 ZINC000880600911 CD On-Demand Anodyne MTNR1A 15 42 COCC1CN(C(=O)[C@@H]2CCc3cc(OC)ccc32)C1 ZINC000880600911 CD On-Demand Anodyne MTNR1B 19 42 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880600927 GF On-Demand Anodyne CACNA1I 58 35 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880600927 GF On-Demand Anodyne GPR119 45 38 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880600928 GF On-Demand Anodyne CACNA1I 58 35 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)c1 ZINC000880600928 GF On-Demand Anodyne GPR119 45 38 COCC1CN(C(=O)CN2c3ccccc3Sc3ccccc32)C1 ZINC000880600938 EG On-Demand Anodyne BCHE 15 40 COCC1CN(C(=O)[C@H](CCC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880600941 EE On-Demand Anodyne CTSK 15 41 COCC1CN(C(=O)[C@H](CCC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880600941 EE On-Demand Anodyne POLG_HCV1 23 40 COCC1CN(C(=O)[C@@H](CCC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880600942 EE On-Demand Anodyne CTSK 15 41 COCC1CN(C(=O)[C@@H](CCC(C)C)NC(=O)OC(C)(C)C)C1 ZINC000880600942 EE On-Demand Anodyne POLG_HCV1 23 40 COCC1CN(C(=O)c2cc3c(C4CC4)cccc3[nH]2)C1 ZINC000880600958 CF On-Demand Anodyne GRIN2B 26 45 COCC1CN(C(=O)c2cc3c(C4CC4)cccc3[nH]2)C1 ZINC000880600958 CF On-Demand Anodyne HRH4 20 46 COCC1CN(C(=O)[C@@H]2N(C(=O)OCc3ccccc3)CC2(C)C)C1 ZINC000880600960 EE On-Demand Anodyne PREP 31 41 COCC1CN(C(=O)[C@@H]2N(C(=O)OCc3ccccc3)CC2(C)C)C1 ZINC000880600960 EE On-Demand Anodyne SLC12A5 46 35 COCC1CN(C(=O)[C@H]2N(C(=O)OCc3ccccc3)CC2(C)C)C1 ZINC000880600961 EE On-Demand Anodyne PREP 31 41 COCC1CN(C(=O)[C@H]2N(C(=O)OCc3ccccc3)CC2(C)C)C1 ZINC000880600961 EE On-Demand Anodyne SLC12A5 46 35 COCC1CN(C(=O)c2ccc3c(c2)[C@@H](CNC(=O)OC(C)(C)C)CCC3)C1 ZINC000880600963 GG On-Demand Anodyne NQO2 18 40 COCC1CN(C(=O)c2ccc3c(c2)[C@H](CNC(=O)OC(C)(C)C)CCC3)C1 ZINC000880600964 GG On-Demand Anodyne NQO2 18 40 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880600977 GF On-Demand Anodyne P2RY12 41 33 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880600977 GF On-Demand Anodyne GRIN2B 20 41 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880600979 GF On-Demand Anodyne P2RY12 41 33 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880600979 GF On-Demand Anodyne GRIN2B 20 41 COCC1CN(C(=O)c2cnnn2C2CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880600991 GD On-Demand Anodyne GPR119 47 40 C[C@@H](Oc1cccc(Cl)c1)C(=O)NNC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880601009 GE On-Demand Reactive PTGER1 19 41 C[C@@H](Oc1cccc(Cl)c1)C(=O)NNC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880601009 GE On-Demand Reactive IMDH_CRYPV 24 41 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne GHRHR 51 33 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne PGC 54 36 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne PAPA1_CARPA 47 43 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne CCKAR 25 40 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne CTSK 20 41 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne CTSL 20 43 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne REN 58 40 COCC1CN(C(=O)[C@@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601010 GE On-Demand Anodyne FPR1 50 39 COc1cccc(C(C)(C)C(=O)NCCCOc2ncccn2)c1 ZINC000880601023 EE On-Demand Anodyne DRD4 41 31 COc1cccc(C(C)(C)C(=O)NCCCOc2ncccn2)c1 ZINC000880601023 EE On-Demand Anodyne MTNR1A 61 47 COc1cccc(C(C)(C)C(=O)NCCCOc2ncccn2)c1 ZINC000880601023 EE On-Demand Anodyne MTNR1B 62 47 COC(=O)c1cc(C(=O)NCCCOc2ncccn2)ccc1C ZINC000880601028 ED On-Demand Anodyne DRD4 41 33 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](c3ccccn3)C2)c1 ZINC000880601038 EF On-Demand Anodyne MAP3K12 42 43 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H](c3ccccn3)C2)c1 ZINC000880601039 EF On-Demand Anodyne MAP3K12 42 43 O=C(CC[C@@H]1CCc2ccccc21)NCCCOc1ncccn1 ZINC000880601045 EF On-Demand Anodyne NQO2 22 46 O=C(CC[C@H]1CCc2ccccc21)NCCCOc1ncccn1 ZINC000880601046 EF On-Demand Anodyne NQO2 22 46 O=C1CC[C@@H](c2ccc(C(=O)NCCCOc3ncccn3)cc2)N1 ZINC000880601048 ED On-Demand Anodyne PLD2 44 36 O=C1CC[C@H](c2ccc(C(=O)NCCCOc3ncccn3)cc2)N1 ZINC000880601049 ED On-Demand Anodyne PLD2 44 36 CN1C[C@H](C(=O)NCCCOc2ncccn2)CCC1=O ZINC000880601050 CC On-Demand Anodyne TBK1 54 34 CN1C[C@@H](C(=O)NCCCOc2ncccn2)CCC1=O ZINC000880601051 CC On-Demand Anodyne TBK1 54 34 O=C(CCc1cccc2ccccc12)NCCCOc1ncccn1 ZINC000880601063 EG On-Demand Anodyne NQO2 30 40 O=C(CCc1cccc2ccccc12)NCCCOc1ncccn1 ZINC000880601063 EG On-Demand Anodyne MTNR1A 74 47 O=C(CCc1cccc2ccccc12)NCCCOc1ncccn1 ZINC000880601063 EG On-Demand Anodyne MTNR1B 60 43 O=C(CCc1cccc2ccccc12)NCCCOc1ncccn1 ZINC000880601063 EG On-Demand Anodyne SUCNR1 51 39 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne GHRHR 51 33 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne PGC 54 36 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne PAPA1_CARPA 47 43 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne CCKAR 25 40 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne CTSK 20 41 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne CTSL 20 43 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne REN 58 40 COCC1CN(C(=O)[C@H](CN(C)Cc2ccccc2)NC(=O)OC(C)(C)C)C1 ZINC000880601076 GE On-Demand Anodyne FPR1 50 39 CCC(=O)Nc1ccccc1C(=O)NCCCOc1ncccn1 ZINC000880601100 EE On-Demand Anodyne MAP1 25 44 CCC(=O)Nc1ccccc1C(=O)NCCCOc1ncccn1 ZINC000880601100 EE On-Demand Anodyne G2YM83_BOTF4 43 32 COCC1CN(C(=O)[C@@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880601103 DF On-Demand Anodyne C3AR1 43 44 COCC1CN(C(=O)[C@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880601105 DF On-Demand Anodyne C3AR1 43 44 COCC1CN(C(=O)Cc2csc(COc3ccccc3)n2)C1 ZINC000880601113 EE On-Demand Anodyne CPT1A 47 36 COC(=O)Nc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880601126 FF On-Demand Anodyne KIT 15 43 COC(=O)Nc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880601126 FF On-Demand Anodyne ROCK2 35 47 COC(=O)Nc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880601126 FF On-Demand Anodyne TYK2 15 40 COC(=O)Nc1cccc(CNC(=O)Nc2cc(CN(C)C)ccn2)c1 ZINC000880601126 FF On-Demand Anodyne BRAF 19 43 CN(C)Cc1ccnc(NC(=O)N2CCN(c3nc(F)c(F)cc3F)CC2)c1 ZINC000880601128 GE On-Demand Anodyne FAAH 22 40 CS(=O)(=O)C1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880601152 EC On-Demand Anodyne MTNR1A 20 42 CS(=O)(=O)C1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880601152 EC On-Demand Anodyne MTNR1B 16 42 CS(=O)(=O)C1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880601152 EC On-Demand Anodyne TBK1 64 34 CC(C)(C)OC(=O)N1CC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880601153 ED On-Demand Anodyne GPR119 22 41 CC(C)(C)OC(=O)N1CC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880601154 ED On-Demand Anodyne GPR119 22 41 CN(C)Cc1ccnc(NC(=O)NNC(=O)[C@@H]2CCOC2)c1 ZINC000880601155 DC On-Demand Reactive MAPK10 15 50 CN(C)Cc1ccnc(NC(=O)NNC(=O)[C@H]2CCOC2)c1 ZINC000880601156 DC On-Demand Reactive MAPK10 15 50 O=C(NCCCOc1ncccn1)c1ncsc1C1CC1 ZINC000880601167 DE On-Demand Anodyne MAP1 78 36 O=C(NCCCOc1ncccn1)[C@H](O)c1cccnc1 ZINC000880601168 CC On-Demand Anodyne ADRB3 35 41 O=C(NCCCOc1ncccn1)[C@@H](O)c1cccnc1 ZINC000880601169 CC On-Demand Anodyne ADRB3 35 41 O=C(NCCCOc1ncccn1)c1csc(Br)n1 ZINC000880601187 ED On-Demand Anodyne HDAC3 17 45 O=C(NCCCOc1ncccn1)[C@@H]1CCc2nncn2CC1 ZINC000880601195 DC On-Demand Anodyne TBK1 61 32 O=C(NCCCOc1ncccn1)[C@H]1CCc2nncn2CC1 ZINC000880601196 DC On-Demand Anodyne TBK1 61 32 O=C(NCCCOc1ncccn1)c1sccc1F ZINC000880601201 CD On-Demand Anodyne MAP1 65 35 C[C@]1(C(=O)NCCCOc2ncccn2)CC(c2ccccc2)=NO1 ZINC000880601212 ED On-Demand Anodyne NPPA 43 34 C[C@@]1(C(=O)NCCCOc2ncccn2)CC(c2ccccc2)=NO1 ZINC000880601213 ED On-Demand Anodyne NPPA 43 34 CC(C)(C)OC(=O)N1CCC[C@@H](CC(=O)NCCCOc2ncccn2)C1 ZINC000880601235 GE On-Demand Anodyne GPR119 37 42 CC(C)(C)OC(=O)N1CCC[C@H](CC(=O)NCCCOc2ncccn2)C1 ZINC000880601236 GE On-Demand Anodyne GPR119 37 42 CC(C)(C(=O)NCCCOc1ncccn1)c1ccc(C#N)cc1 ZINC000880601238 DE On-Demand Mild CTRB_BOVIN 47 33 CN(C)Cc1ccnc(NC(=O)N2Cc3cccc(Cl)c3C2)c1 ZINC000880601243 EG On-Demand Anodyne TYK2 57 36 COc1cccc([C@H](O)CN(Cc2ccccc2)C(=O)COC2CC2)c1 ZINC000880601245 FF On-Demand Anodyne TIMP3 50 34 COc1cccc([C@H](O)CN(Cc2ccccc2)C(=O)COC2CC2)c1 ZINC000880601245 FF On-Demand Anodyne PTGES 20 44 O=C(NCCCOc1ncccn1)c1sccc1C(F)F ZINC000880601258 DF On-Demand Anodyne MAP1 49 33 CN(C)Cc1ccnc(NC(=O)NCc2cc(Cl)cc(Cl)c2O)c1 ZINC000880601272 FG On-Demand Clean TYK2 17 41 COc1cccc([C@H](O)CN(Cc2ccccc2)C(=O)c2cnc(C3CC3)o2)c1 ZINC000880601274 GH On-Demand Anodyne PTGES 19 41 CN(C)Cc1ccnc(NC(=O)NNc2ccc(C(F)(F)F)cc2)c1 ZINC000880601280 FG On-Demand Reactive RAF1 20 40 CC(C)(C)OC(=O)N1CSC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880601288 FD On-Demand Anodyne CACNA1B 16 43 CN(C)Cc1ccnc(NC(=O)N2CCC(CNC(=O)C(F)(F)F)CC2)c1 ZINC000880601290 GE On-Demand Anodyne CACNA1I 52 33 CC(C)(C)OC(=O)N1CC(CCC(=O)NCCCOc2ncccn2)C1 ZINC000880601292 FE On-Demand Anodyne GPR119 33 40 O=C(NCCCOc1ncccn1)c1cc(CN2CCCC2)on1 ZINC000880601294 ED On-Demand Anodyne HRH2 34 40 O=C(NCCCOc1ncccn1)c1cnc(CC2CC2)s1 ZINC000880601301 DE On-Demand Anodyne SIRT3 40 32 O=C(NCCCOc1ncccn1)c1cnc(CC2CC2)s1 ZINC000880601301 DE On-Demand Anodyne SIRT1 40 32 CN(C)Cc1ccnc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c1 ZINC000880601341 GG On-Demand Anodyne TYK2 38 42 CN(C)C(=O)C1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880601364 ED On-Demand Anodyne TBK1 58 34 O=C(NCCCOc1ncccn1)c1cccn(C2CC2)c1=O ZINC000880601380 DD On-Demand Anodyne POLR1A 59 33 CC(C)(C)OC(=O)N1CC[C@H](CC(=O)NCCCOc2ncccn2)C1 ZINC000880601397 FE On-Demand Anodyne GPR119 47 46 CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C(=O)NCCCOc2ncccn2)C1 ZINC000880601406 GD On-Demand Anodyne GPR119 45 46 CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C(=O)NCCCOc2ncccn2)C1 ZINC000880601407 GD On-Demand Anodyne GPR119 45 46 CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C(=O)NCCCOc2ncccn2)C1 ZINC000880601408 GD On-Demand Anodyne GPR119 45 46 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C(=O)NCCCOc2ncccn2)C1 ZINC000880601409 GD On-Demand Anodyne GPR119 45 46 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CC(c3ccc4c(c3)CCO4)=NO2)c1 ZINC000880601428 GE On-Demand Anodyne LUCI_PHOPY 42 31 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CC(c3ccc4c(c3)CCO4)=NO2)c1 ZINC000880601429 GE On-Demand Anodyne LUCI_PHOPY 42 31 O=C(NCCCOc1ncccn1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880601446 FF On-Demand Anodyne FKBP1A 17 41 O=C(NCCCOc1ncccn1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880601446 FF On-Demand Anodyne C3AR1 44 43 O=C(NCCCOc1ncccn1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880601447 FF On-Demand Anodyne FKBP1A 17 41 O=C(NCCCOc1ncccn1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880601447 FF On-Demand Anodyne C3AR1 44 43 O=C(COCc1cccnc1)NCCCOc1ncccn1 ZINC000880601448 DC On-Demand Anodyne PTAFR 24 44 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne PPIA 34 43 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne KIT 19 41 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne RAF1 22 43 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne TYK2 32 41 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne BRAF 25 41 CN(C)Cc1ccnc(NC(=O)Nc2cccc(C(C)(C)O)c2)c1 ZINC000880601456 EG On-Demand Anodyne EPHB4 25 41 CN(C)Cc1ccnc(NC(=O)NNc2ccccc2OC(F)(F)F)c1 ZINC000880601472 FG On-Demand Reactive P2RY1 48 44 CN(C)Cc1ccnc(NC(=O)NC[C@@]2(C)CCN(Cc3ccccc3)C2)c1 ZINC000880601478 GG On-Demand Anodyne NPFFR1 41 36 CN(C)Cc1ccnc(NC(=O)NC[C@]2(C)CCN(Cc3ccccc3)C2)c1 ZINC000880601479 GG On-Demand Anodyne NPFFR1 41 36 C[C@H]1CN(C(=O)OC(C)(C)C)CC[C@H]1NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880601498 GF On-Demand Anodyne GPR119 43 37 C[C@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880601499 GF On-Demand Anodyne GPR119 43 37 CCCC[C@](C)(F)C(=O)NCCCOc1ncccn1 ZINC000880601503 CE On-Demand Anodyne ASAH1 40 31 CCCC[C@@](C)(F)C(=O)NCCCOc1ncccn1 ZINC000880601504 CE On-Demand Anodyne ASAH1 40 31 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild KIT 16 41 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild GRM4 54 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild GRM5 33 46 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild DDR1 58 41 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild KCNK3 85 49 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(C(=O)O)nc1 ZINC000880601511 EF On-Demand Mild KCNK9 44 35 CN(C)Cc1ccnc(NC(=O)N2CCN(c3cccc(F)n3)CC2)c1 ZINC000880601551 FE On-Demand Anodyne FAAH 22 41 CC(C)(C)OC(=O)N1CCN(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880601614 GD On-Demand Anodyne DRD2 28 41 CC(C)(C)OC(=O)N1CCN(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880601614 GD On-Demand Anodyne DRD3 43 38 CC(C)(C)OC(=O)N1CCN(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880601614 GD On-Demand Anodyne HRP1_PLAFA 26 41 CC(C)(C)OC(=O)N1CCN(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880601614 GD On-Demand Anodyne GPR119 35 43 CN(C)Cc1ccnc(NC(=O)N2CCc3cc(Cl)nnc3C2)c1 ZINC000880601626 EE On-Demand Anodyne MAPK1 42 35 CN(C)Cc1ccnc(NC(=O)N2CCc3cc(Cl)nnc3C2)c1 ZINC000880601626 EE On-Demand Anodyne QRFPR 21 40 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880601628 FE On-Demand Anodyne SSTR2 44 39 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880601628 FE On-Demand Anodyne TBK1 79 35 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880601628 FE On-Demand Anodyne GPBAR1 20 41 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880601628 FE On-Demand Anodyne GPR119 37 43 O=C(NCCCOc1ncccn1)c1cccc(C2OCCO2)c1 ZINC000880601636 ED On-Demand Anodyne DRD4 41 31 NC(=O)COc1cccc(NC(=O)COc2ccccc2C=O)c1 ZINC000880601658 ED On-Demand Anodyne KCNK3 46 33 NC(=O)COc1cccc(NC(=O)COc2ccccc2C=O)c1 ZINC000880601658 ED On-Demand Anodyne KCNK9 43 33 O=C(NCCCOc1ncccn1)C1CCC(O)CC1 ZINC000880601700 CC On-Demand Anodyne MTNR1A 22 41 O=C(NCCCOc1ncccn1)C1CCC(O)CC1 ZINC000880601700 CC On-Demand Anodyne MTNR1B 19 41 O=C(NCCCOc1ncccn1)C1CCC(O)CC1 ZINC000880601700 CC On-Demand Anodyne TBK1 70 33 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne HTR1A 32 43 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne DRD2 40 41 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne DRD4 24 43 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne HTR2A 29 40 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne DRD3 71 45 O=C(NCCCOc1ncccn1)c1ccccc1N1CCOCC1 ZINC000880601706 ED On-Demand Anodyne HPGDS 20 41 CN(C)Cc1ccnc(NC(=O)N[C@@H]2C[C@H](O)c3ccccc32)c1 ZINC000880601730 EE On-Demand Anodyne TYK2 19 40 CN(C)Cc1ccnc(NC(=O)N[C@H]2C[C@H](O)c3ccccc32)c1 ZINC000880601731 EE On-Demand Anodyne TYK2 19 40 CN(C)Cc1ccnc(NC(=O)N[C@@H]2C[C@@H](O)c3ccccc32)c1 ZINC000880601732 EE On-Demand Anodyne TYK2 19 40 CN(C)Cc1ccnc(NC(=O)N[C@H]2C[C@@H](O)c3ccccc32)c1 ZINC000880601733 EE On-Demand Anodyne TYK2 19 40 COc1ccc(N2CC[C@H](NC(=O)Nc3cc(CN(C)C)ccn3)C2)cc1 ZINC000880601750 FF On-Demand Clean EPHX2 18 43 COc1ccc(N2CC[C@H](NC(=O)Nc3cc(CN(C)C)ccn3)C2)cc1 ZINC000880601750 FF On-Demand Clean MCHR1 17 43 CN(C)Cc1ccnc(NC(=O)N2CCC[C@@](O)(c3ccc(Cl)cc3)C2)c1 ZINC000880601776 GG On-Demand Anodyne CCR1 57 36 CN(C)Cc1ccnc(NC(=O)N2CCC[C@](O)(c3ccc(Cl)cc3)C2)c1 ZINC000880601777 GG On-Demand Anodyne CCR1 57 36 CN(C)Cc1ccnc(NC(=O)N2CCC[C@H](OC(=O)N(C)C)C2)c1 ZINC000880601780 ED On-Demand Anodyne MAP3K12 26 40 CN(C)Cc1ccnc(NC(=O)N2CCC[C@@H](OC(=O)N(C)C)C2)c1 ZINC000880601781 ED On-Demand Anodyne MAP3K12 26 40 O=C(Cc1ccc(Cl)c(F)c1)NCCCOc1ncccn1 ZINC000880601788 DE On-Demand Anodyne NCE103 15 43 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c1 ZINC000880601802 EE On-Demand Anodyne CACNA1I 41 33 CN(C)Cc1ccnc(NC(=O)NC[C@H]2CCN(C(C)(C)C)C2)c1 ZINC000880601803 EE On-Demand Anodyne CACNA1I 41 33 CN(C)Cc1ccnc(NC(=O)NCc2cc(Cl)ccc2O)c1 ZINC000880601819 EF On-Demand Clean TYK2 15 40 CN1CC[C@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601820 ED On-Demand Anodyne HTR1A 19 45 CN1CC[C@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601820 ED On-Demand Anodyne DRD2 18 45 CN1CC[C@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601820 ED On-Demand Anodyne TBK1 58 34 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601821 ED On-Demand Anodyne HTR1A 19 45 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601821 ED On-Demand Anodyne DRD2 18 45 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)c2ccccc21 ZINC000880601821 ED On-Demand Anodyne TBK1 58 34 CC(C)(C)OC(=O)N1CC[C@H](CCC(=O)NCCCOc2ncccn2)C1 ZINC000880601824 GE On-Demand Anodyne GPR119 43 44 CC(C)(C)OC(=O)N1CC[C@@H](CCC(=O)NCCCOc2ncccn2)C1 ZINC000880601825 GE On-Demand Anodyne GPR119 43 44 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne MME 81 43 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne PAPA1_CARPA 40 35 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne NPFFR2 44 34 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne MMP8 15 43 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne CAPN1 44 34 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne CAPN2 51 34 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne AMP1_PLAFQ 49 43 O=C(NCCCOc1ncccn1)[C@@H](F)Cc1ccccc1 ZINC000880601943 DD On-Demand Anodyne NPFFR1 59 34 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne MME 81 43 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne PAPA1_CARPA 40 35 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne NPFFR2 44 34 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne MMP8 15 43 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne CAPN1 44 34 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne CAPN2 51 34 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne AMP1_PLAFQ 49 43 O=C(NCCCOc1ncccn1)[C@H](F)Cc1ccccc1 ZINC000880601944 DD On-Demand Anodyne NPFFR1 59 34 Cc1sc(Br)nc1C(=O)NCCCOc1ncccn1 ZINC000880601949 FE On-Demand Anodyne HDAC3 15 47 CC(C)[C@H](O)CC(=O)NCCCOc1ncccn1 ZINC000880601953 CC On-Demand Anodyne PLM2_PLAFA 33 42 CN(C)Cc1ccnc(NC(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)c1 ZINC000880601986 GH On-Demand Anodyne KIT 15 43 CN(C)Cc1ccnc(NC(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)c1 ZINC000880601986 GH On-Demand Anodyne ROCK2 24 44 CN(C)Cc1ccnc(NC(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)c1 ZINC000880601986 GH On-Demand Anodyne BRAF 21 43 CC(C)(C(=O)NCCCOc1ncccn1)C1CCCCC1 ZINC000880601992 DF On-Demand Anodyne AMY2 51 35 O=C(NCCCOc1ncccn1)C1CCN(C2CC2)CC1 ZINC000880601993 DD On-Demand Anodyne TBK1 77 38 O=C(NCCCOc1ncccn1)c1cncc(Cl)n1 ZINC000880602005 CD On-Demand Anodyne SCN2A 18 40 O=C(NCCCOc1ncccn1)c1cncc(Cl)n1 ZINC000880602005 CD On-Demand Anodyne SCN10A 42 40 CN(C)Cc1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)c1 ZINC000880602008 FG On-Demand Anodyne EPHX2 17 41 CN(C)Cc1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)c1 ZINC000880602009 FG On-Demand Anodyne EPHX2 17 41 CN(C)Cc1ccnc(NC(=O)N2CCC=C(Cl)C2)c1 ZINC000880602018 CF On-Demand Anodyne TYK2 17 42 CN(C)Cc1ccnc(NC(=O)N2C[C@H]3CC[C@H]2CN3C(=O)OC(C)(C)C)c1 ZINC000880602040 GF On-Demand Anodyne GPR119 19 41 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H]3CN(C(=O)OC(C)(C)C)C[C@@H]32)c1 ZINC000880602055 GF On-Demand Anodyne GPR119 36 41 CC(C)(C)OC(=O)N1CCC(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880602071 GF On-Demand Anodyne GRIN2B 21 40 CC(C)(C)OC(=O)N1CCC(CCC(=O)NCCCOc2ncccn2)CC1 ZINC000880602071 GF On-Demand Anodyne GPR119 53 49 O=C(NCCCOc1ncccn1)c1coc(C2CCOCC2)n1 ZINC000880602074 ED On-Demand Anodyne TBXA2R 34 41 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880602075 CC On-Demand Anodyne LUXR 79 42 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880602075 CC On-Demand Anodyne TRAR 91 42 CN(C)Cc1ccnc(NC(=O)N[C@H]2CCOC2=O)c1 ZINC000880602075 CC On-Demand Anodyne LASR 62 40 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne F2 42 41 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne FKBP1A 27 43 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne CELA1 45 34 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne ELANE 44 36 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne TRY1_BOVIN 46 35 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880602115 EC On-Demand Anodyne TPP2 27 40 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne F2 42 41 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne FKBP1A 27 43 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne CELA1 45 34 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne ELANE 44 36 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne TRY1_BOVIN 46 35 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880602116 EC On-Demand Anodyne TPP2 27 40 CC(C)(C)OC(=O)N1CC(CC(=O)NCCCOc2ncccn2)C1 ZINC000880602158 FD On-Demand Anodyne GPR119 35 41 O=C(NCCCOc1ncccn1)c1ccnc(N2CCCC2)n1 ZINC000880602160 ED On-Demand Anodyne HTR1A 20 47 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne HRH2 33 41 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne SCNN1A 58 40 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne SCN2A 19 40 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne MTNR1A 27 41 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne MTNR1B 32 45 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne FAAH 69 40 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne CES1 79 37 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne AMP1_PLAFQ 27 47 O=C(NCCCOc1ncccn1)C(=O)NCCCc1ccccc1 ZINC000880602245 ED On-Demand Anodyne CRTM 41 40 O=C(NCCCOc1ncccn1)[C@H]1CCN(C2CCCCC2)C1 ZINC000880602273 EE On-Demand Anodyne TBK1 61 34 O=C(NCCCOc1ncccn1)[C@@H]1CCN(C2CCCCC2)C1 ZINC000880602274 EE On-Demand Anodyne TBK1 61 34 COc1ccccc1/C(C)=C/C(=O)NCCCOc1ncccn1 ZINC000880602275 EE On-Demand Anodyne ADRA1D 19 40 COc1ccccc1/C(C)=C/C(=O)NCCCOc1ncccn1 ZINC000880602275 EE On-Demand Anodyne ADRA1A 15 40 COc1ccccc1/C(C)=C/C(=O)NCCCOc1ncccn1 ZINC000880602275 EE On-Demand Anodyne KCNA3 42 39 COc1ccccc1/C(C)=C\C(=O)NCCCOc1ncccn1 ZINC000880602276 EE On-Demand Anodyne ADRA1D 19 40 COc1ccccc1/C(C)=C\C(=O)NCCCOc1ncccn1 ZINC000880602276 EE On-Demand Anodyne ADRA1A 15 40 COc1ccccc1/C(C)=C\C(=O)NCCCOc1ncccn1 ZINC000880602276 EE On-Demand Anodyne KCNA3 42 39 CN(C)Cc1ccnc(NC(=O)NC2CCN(CC(=O)OC(C)(C)C)CC2)c1 ZINC000880602291 GE On-Demand Anodyne SSTR5 49 35 C[C@@H](Oc1cccc(CO)c1)C(=O)NCCCOc1ncccn1 ZINC000880602308 ED On-Demand Anodyne HRH2 29 42 C[C@@H](Oc1cccc(CO)c1)C(=O)NCCCOc1ncccn1 ZINC000880602308 ED On-Demand Anodyne MTNR1A 46 44 C[C@@H](Oc1cccc(CO)c1)C(=O)NCCCOc1ncccn1 ZINC000880602308 ED On-Demand Anodyne MTNR1B 48 44 COc1cccc(C(=O)NCCCOc2ncccn2)n1 ZINC000880602314 CD On-Demand Anodyne DRD3 16 42 COc1cccc(C(=O)NCCCOc2ncccn2)n1 ZINC000880602314 CD On-Demand Anodyne ALS 41 32 CN1CCOc2ccc(C(=O)NCCCOc3ncccn3)cc21 ZINC000880602315 ED On-Demand Anodyne HTR1A 23 40 CN1CCOc2ccc(C(=O)NCCCOc3ncccn3)cc21 ZINC000880602315 ED On-Demand Anodyne DRD2 25 44 CN1CCOc2ccc(C(=O)NCCCOc3ncccn3)cc21 ZINC000880602315 ED On-Demand Anodyne DRD4 45 35 CN1CCOc2ccc(C(=O)NCCCOc3ncccn3)cc21 ZINC000880602315 ED On-Demand Anodyne HTR2A 15 40 CN1CCOc2ccc(C(=O)NCCCOc3ncccn3)cc21 ZINC000880602315 ED On-Demand Anodyne DRD3 46 44 N#CCOc1cccc(CC(=O)NCCCOc2ncccn2)c1 ZINC000880602331 ED On-Demand Mild HRH2 38 40 N#CCOc1cccc(CC(=O)NCCCOc2ncccn2)c1 ZINC000880602331 ED On-Demand Mild MTNR1A 25 42 N#CCOc1cccc(CC(=O)NCCCOc2ncccn2)c1 ZINC000880602331 ED On-Demand Mild MTNR1B 21 42 O=C(NCCCOc1ncccn1)c1csc(Cl)n1 ZINC000880602344 CD On-Demand Anodyne HDAC3 16 41 CC(C)(C)OC(=O)N1Cc2ccc(C(=O)NCCCOc3ncccn3)cc2C1 ZINC000880602348 GF On-Demand Anodyne DRD4 40 31 O=C(NCCCOc1ncccn1)[C@H](F)c1ccccc1 ZINC000880602373 CE On-Demand Anodyne C3AR1 45 33 O=C(NCCCOc1ncccn1)[C@@H](F)c1ccccc1 ZINC000880602374 CE On-Demand Anodyne C3AR1 45 33 CN(C)Cc1ccnc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)c1 ZINC000880602391 GE On-Demand Anodyne RBP4 44 34 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@@H]3C2)c1 ZINC000880602392 GE On-Demand Anodyne RBP4 44 34 CN(C)Cc1ccnc(NC(=O)N2CC[C@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)c1 ZINC000880602393 GE On-Demand Anodyne RBP4 44 34 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H]3CN(C(=O)C(F)(F)F)C[C@H]3C2)c1 ZINC000880602394 GE On-Demand Anodyne RBP4 44 34 CN(C)Cc1ccnc(NC(=O)N2CCC(c3nc(C4CCC4)no3)CC2)c1 ZINC000880602439 GG On-Demand Anodyne ETHR 63 43 CN(C)Cc1ccnc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880602440 FE On-Demand Anodyne FAAH 23 44 CN(C)Cc1ccnc(NC(=O)NC[C@H](O)c2ccc(Cl)c(Cl)c2)c1 ZINC000880602445 GG On-Demand Anodyne TYK2 16 41 CN(C)Cc1ccnc(NC(=O)NC[C@@H](O)c2ccc(Cl)c(Cl)c2)c1 ZINC000880602446 GG On-Demand Anodyne TYK2 16 41 CN(C)Cc1ccnc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)c1 ZINC000880602457 GF On-Demand Mild NPY2R 22 42 CN(C)Cc1ccnc(NC(=O)N2CCC(C(=O)NCCO)CC2)c1 ZINC000880602464 EC On-Demand Anodyne TYK2 46 36 CN(C)Cc1ccnc(NC(=O)N2CCC3(CCNC3=O)CC2)c1 ZINC000880602500 ED On-Demand Anodyne MAPKAPK2 41 33 CC(C)(C)OC(=O)N1CC[C@@H](CC(=O)NCCCOc2ncccn2)C1 ZINC000880602506 FE On-Demand Anodyne GPR119 47 46 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCCCOc3ncccn3)ccc21 ZINC000880602507 GF On-Demand Anodyne DRD2 19 40 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCCCOc3ncccn3)ccc21 ZINC000880602507 GF On-Demand Anodyne DRD4 46 36 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCCCOc3ncccn3)ccc21 ZINC000880602507 GF On-Demand Anodyne DRD3 36 40 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCCCOc3ncccn3)ccc21 ZINC000880602507 GF On-Demand Anodyne GPR119 15 41 CC(C)(C)OC(=O)N1CCC2(CC1)C[C@H]2C(=O)NCCCOc1ncccn1 ZINC000880602508 GE On-Demand Anodyne GPR119 32 42 CC(C)(C)OC(=O)N1CCC2(CC1)C[C@@H]2C(=O)NCCCOc1ncccn1 ZINC000880602509 GE On-Demand Anodyne GPR119 32 42 CC(C)(C)OC(=O)N1CC(C(=O)NCCCOc2ncccn2)C1 ZINC000880602525 ED On-Demand Anodyne TBK1 60 32 CC(C)(C)OC(=O)N1CC(C(=O)NCCCOc2ncccn2)C1 ZINC000880602525 ED On-Demand Anodyne GPR119 30 42 CC(C)(C)OC(=O)N1CCC[C@H](CC(=O)NCCCOc2ncccn2)CC1 ZINC000880602529 GF On-Demand Anodyne GPR119 47 47 CC(C)(C)OC(=O)N1CCC[C@@H](CC(=O)NCCCOc2ncccn2)CC1 ZINC000880602530 GF On-Demand Anodyne GPR119 47 47 O=C(NCCCOc1ncccn1)[C@@H](F)CC1CCCCC1 ZINC000880602537 DF On-Demand Anodyne DPEP1 40 32 O=C(NCCCOc1ncccn1)[C@H](F)CC1CCCCC1 ZINC000880602538 DF On-Demand Anodyne DPEP1 40 32 COc1cccc(C2=NO[C@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602558 FD On-Demand Anodyne MTNR1A 44 42 COc1cccc(C2=NO[C@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602558 FD On-Demand Anodyne MTNR1B 44 42 COc1cccc(C2=NO[C@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602558 FD On-Demand Anodyne LUCI_PHOPY 37 46 COc1cccc(C2=NO[C@@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602559 FD On-Demand Anodyne MTNR1A 44 42 COc1cccc(C2=NO[C@@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602559 FD On-Demand Anodyne MTNR1B 44 42 COc1cccc(C2=NO[C@@H](C(=O)NCCCOc3ncccn3)C2)c1 ZINC000880602559 FD On-Demand Anodyne LUCI_PHOPY 37 46 CN(C)Cc1ccnc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)c1 ZINC000880602569 FE On-Demand Anodyne NAMPT 47 35 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602580 FD On-Demand Anodyne EPHX2 20 41 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602580 FD On-Demand Anodyne TBK1 66 32 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602580 FD On-Demand Anodyne GPR119 46 47 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602581 FD On-Demand Anodyne EPHX2 20 41 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602581 FD On-Demand Anodyne TBK1 66 32 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602581 FD On-Demand Anodyne GPR119 46 47 O=C(NCCCOc1ncccn1)[C@@H]1C[C@H]1c1ccccc1 ZINC000880602605 CE On-Demand Anodyne NAMPT 19 53 C[C@H]1c2ccccc2C[C@H]1NC(=O)Nc1cc(CN(C)C)ccn1 ZINC000880602632 DF On-Demand Anodyne TYK2 16 40 CN1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602643 CC On-Demand Anodyne TBK1 82 41 O=C1CCCc2cc(C(=O)NCCCOc3ncccn3)ccc2N1 ZINC000880602661 ED On-Demand Anodyne DRD4 40 30 O=C1CCCc2cc(C(=O)NCCCOc3ncccn3)ccc2N1 ZINC000880602661 ED On-Demand Anodyne HDAC9 26 55 Cc1oc(-c2cccs2)nc1C(=O)NCCCOc1ncccn1 ZINC000880602683 EF On-Demand Anodyne PPARA 27 41 O=C(Cc1cccs1)NCCCOc1ncccn1 ZINC000880602687 CD On-Demand Anodyne CA5B 38 47 O=C(Cc1cccs1)NCCCOc1ncccn1 ZINC000880602687 CD On-Demand Anodyne CA5A 37 43 CN(C)C(=O)c1ccc(NC(=O)NCCc2cccnc2)nc1 ZINC000880602707 DD On-Demand Anodyne PTAFR 29 43 CN(C)C(=O)c1ccc(NC(=O)NCCc2cccnc2)nc1 ZINC000880602707 DD On-Demand Anodyne NAMPT 59 45 CN(C)Cc1ccnc(NC(=O)NCc2cc(O)ccc2Cl)c1 ZINC000880602712 EF On-Demand Anodyne TYK2 20 42 O=C(CSc1nc2ccccc2s1)NCCCOc1ncccn1 ZINC000880602718 FF On-Demand Anodyne ST14 48 35 O=C(CSc1nc2ccccc2s1)NCCCOc1ncccn1 ZINC000880602718 FF On-Demand Anodyne HMOX2 33 43 O=C(CSc1nc2ccccc2s1)NCCCOc1ncccn1 ZINC000880602718 FF On-Demand Anodyne TMPRSS6 71 35 C[C@@H](NC(=O)CCc1ccc2ccccc2n1)c1nnc(O)n1C ZINC000880602724 ED On-Demand Anodyne CYSLTR1 40 39 CCOc1ccccc1C(F)(F)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880602727 ED On-Demand Anodyne PLK1 46 36 CCOc1ccccc1C(F)(F)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880602729 ED On-Demand Anodyne PLK1 46 36 C[C@H](NC(=O)CCc1ccc2ccccc2n1)c1nnc(O)n1C ZINC000880602730 ED On-Demand Anodyne CYSLTR1 40 39 CN(C)Cc1ccnc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)c1 ZINC000880602746 FG On-Demand Anodyne NPY5R 34 42 CN(C)Cc1ccnc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)c1 ZINC000880602751 FG On-Demand Anodyne NPY5R 34 42 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne PRSS2 58 33 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne MAPK14 23 40 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne CCR3 30 40 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne MLNR 48 43 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne MAPK10 17 40 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)c1 ZINC000880602764 FF On-Demand Anodyne EPHX2 21 43 CNC(=O)N(C)c1ccc(NC(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880602785 FF On-Demand Anodyne SMG1 47 31 CCOC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602801 ED On-Demand Anodyne P2RY12 44 36 CCOC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602801 ED On-Demand Anodyne GRIN2B 21 41 CCOC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602801 ED On-Demand Anodyne TBK1 77 35 N#CCOc1ccccc1C(=O)NCCCOc1ncccn1 ZINC000880602814 DD On-Demand Mild FOLH1 19 40 N#CCOc1ccccc1C(=O)NCCCOc1ncccn1 ZINC000880602814 DD On-Demand Mild HCN1 51 31 CC(C)(C)OC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602826 FE On-Demand Anodyne EPHX2 18 42 CC(C)(C)OC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602826 FE On-Demand Anodyne TBK1 78 33 CC(C)(C)OC(=O)N1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880602826 FE On-Demand Anodyne GPR119 53 52 CC(C)c1ccc(OCC(=O)NCCCOc2ncccn2)cc1 ZINC000880602837 EF On-Demand Anodyne PLA2G4B 43 31 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602845 FE On-Demand Anodyne SSTR2 44 39 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602845 FE On-Demand Anodyne TBK1 79 35 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602845 FE On-Demand Anodyne GPBAR1 20 41 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880602845 FE On-Demand Anodyne GPR119 37 43 CN(C)C(=O)c1ccc(NC(=O)NCCCOc2ccccc2F)nc1 ZINC000880602868 FF On-Demand Anodyne ADRB1 41 33 C[C@@H](NC(=O)c1c(F)cccc1Br)c1nnc(O)n1C ZINC000880602876 ED On-Demand Anodyne DAC 23 41 O=C(NCCCOc1ncccn1)C1CCCCCCC1 ZINC000880602959 CF On-Demand Anodyne HRH2 30 42 O=C(NCCCOc1ncccn1)C1CCCCCCC1 ZINC000880602959 CF On-Demand Anodyne IKBKE 43 39 O=C(NCCCOc1ncccn1)C1CCCCCCC1 ZINC000880602959 CF On-Demand Anodyne TBK1 88 40 O=C(CCN1CCOCC1)NCCCOc1ncccn1 ZINC000880602960 CC On-Demand Anodyne EPHX2 23 42 C[C@@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603018 GE On-Demand Anodyne GPR119 29 41 C[C@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603019 GE On-Demand Anodyne GPR119 29 41 CCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603040 CE On-Demand Mild ASAH1 20 41 CCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603040 CE On-Demand Mild LASR 47 37 CCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603040 CE On-Demand Mild NOD1 93 46 CCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603040 CE On-Demand Mild CQSS 54 35 CCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603042 CE On-Demand Mild ASAH1 20 41 CCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603042 CE On-Demand Mild LASR 47 37 CCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603042 CE On-Demand Mild NOD1 93 46 CCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603042 CE On-Demand Mild CQSS 54 35 CN(C)C(=O)c1ccc(NC(=O)NCc2ccn(C)n2)nc1 ZINC000880603062 DC On-Demand Anodyne GCK 15 41 C[C@@H](NC(=O)Cc1cccs1)c1nnc(O)n1C ZINC000880603070 CD On-Demand Anodyne CA5B 31 40 C[C@@H](NC(=O)Cc1cccs1)c1nnc(O)n1C ZINC000880603070 CD On-Demand Anodyne CA5A 31 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCOCC3)cc2)nc1 ZINC000880603098 GD On-Demand Clean F10 17 44 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCOCC3)cc2)nc1 ZINC000880603098 GD On-Demand Clean PIK3CA 37 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCOCC3)cc2)nc1 ZINC000880603098 GD On-Demand Clean MTOR 65 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCOCC3)cc2)nc1 ZINC000880603098 GD On-Demand Clean EPHB4 50 32 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCOCC3)cc2)nc1 ZINC000880603098 GD On-Demand Clean STAT6 68 39 CN(C)Cc1ccnc(NC(=O)NNC(=O)C2CCOCC2)c1 ZINC000880603100 DC On-Demand Reactive MAPK10 15 49 CN(C)Cc1ccnc(NC(=O)NNC(=O)C2CCOCC2)c1 ZINC000880603100 DC On-Demand Reactive TYK2 53 38 CCCOc1ccc(OCC(=O)N[C@H](C)c2nnc(O)n2C)cc1 ZINC000880603127 ED On-Demand Anodyne ACACA 15 49 CCCOc1ccc(OCC(=O)N[C@H](C)c2nnc(O)n2C)cc1 ZINC000880603127 ED On-Demand Anodyne ACACB 17 49 CCCOc1ccc(OCC(=O)N[C@H](C)c2nnc(O)n2C)cc1 ZINC000880603127 ED On-Demand Anodyne PLA2G4B 64 33 CCCOc1ccc(OCC(=O)N[C@@H](C)c2nnc(O)n2C)cc1 ZINC000880603128 ED On-Demand Anodyne ACACA 15 49 CCCOc1ccc(OCC(=O)N[C@@H](C)c2nnc(O)n2C)cc1 ZINC000880603128 ED On-Demand Anodyne ACACB 17 49 CCCOc1ccc(OCC(=O)N[C@@H](C)c2nnc(O)n2C)cc1 ZINC000880603128 ED On-Demand Anodyne PLA2G4B 64 33 Cc1ccc(N2CCCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880603144 GF On-Demand Anodyne PRNP 41 38 CCCCSCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603147 CD On-Demand Anodyne EST1_PIG 41 36 CCCCSCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603148 CD On-Demand Anodyne EST1_PIG 41 36 C/C=C\c1ccc(OCC(=O)NCCCOc2ncccn2)c(OC)c1 ZINC000880603156 FE On-Demand Anodyne MTNR1B 23 43 C/C=C/c1ccc(OCC(=O)NCCCOc2ncccn2)c(OC)c1 ZINC000880603157 FE On-Demand Anodyne MTNR1B 23 43 CN(C)Cc1ccnc(NC(=O)N2CCO[C@H](c3noc(C4CC4)n3)C2)c1 ZINC000880603193 FE On-Demand Anodyne ETHR 59 34 CN(C)Cc1ccnc(NC(=O)N2CCO[C@@H](c3noc(C4CC4)n3)C2)c1 ZINC000880603194 FE On-Demand Anodyne ETHR 59 34 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCCOc1ncccn1 ZINC000880603195 GD On-Demand Anodyne CA5B 38 41 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCCOc1ncccn1 ZINC000880603195 GD On-Demand Anodyne CA5A 38 41 C[C@H]1CN(C(=O)Nc2cc(CN(C)C)ccn2)Cc2ccccc21 ZINC000880603213 DG On-Demand Anodyne QRFPR 18 43 C[C@@H]1CN(C(=O)Nc2cc(CN(C)C)ccn2)Cc2ccccc21 ZINC000880603214 DG On-Demand Anodyne QRFPR 18 43 CN(C)Cc1ccnc(NC(=O)N2C[C@@H](CO)[C@@H](CO)C2)c1 ZINC000880603235 DC On-Demand Anodyne TYK2 15 42 CC(C)c1cc([C@@H]2CCCN(C(=O)Nc3cc(CN(C)C)ccn3)C2)n[nH]1 ZINC000880603241 FG On-Demand Anodyne MAP3K12 32 41 CN(C)Cc1ccnc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)c1 ZINC000880603247 GE On-Demand Clean FLT3 21 47 CN(C)Cc1ccnc(NC(=O)N2[C@H]3CC[C@H]2CN(C(=O)OC(C)(C)C)C3)c1 ZINC000880603253 GF On-Demand Anodyne GPR119 48 41 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(OC)c1 ZINC000880603259 GF On-Demand Clean HTR1A 24 43 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(OC)c1 ZINC000880603259 GF On-Demand Clean HTR1B 16 43 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(OC)c1 ZINC000880603259 GF On-Demand Clean PDGFRB 71 46 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(OC)c1 ZINC000880603259 GF On-Demand Clean LCK 19 41 COc1ccc(N2CCN(C(=O)Nc3cc(CN(C)C)ccn3)CC2)c(OC)c1 ZINC000880603259 GF On-Demand Clean TNIK 40 39 CN(C)Cc1ccnc(NC(=O)N2C[C@@H]3CC[C@H](C2)N3C(=O)OC(C)(C)C)c1 ZINC000880603262 GF On-Demand Anodyne GPR119 34 41 CONC(=O)C1CCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880603266 ED On-Demand Anodyne TYK2 47 36 CCOC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603355 ED On-Demand Anodyne TBK1 77 35 CCOC(=O)N1CCC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603355 ED On-Demand Anodyne GPBAR1 19 42 CCOC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603357 ED On-Demand Anodyne TBK1 77 35 CCOC(=O)N1CCC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603357 ED On-Demand Anodyne GPBAR1 19 42 O=C(NCCCOc1ncccn1)c1cccc(N2CCOC2=O)c1 ZINC000880603365 ED On-Demand Anodyne DRD4 44 35 O=C(NCCCOc1ncccn1)c1cccc(N2CCOC2=O)c1 ZINC000880603365 ED On-Demand Anodyne DRD3 23 41 CCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603367 CD On-Demand Anodyne ASAH1 20 41 CCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603367 CD On-Demand Anodyne LASR 47 37 CCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603367 CD On-Demand Anodyne NOD1 93 46 CCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603367 CD On-Demand Anodyne CQSS 54 35 CCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603369 CD On-Demand Anodyne ASAH1 20 41 CCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603369 CD On-Demand Anodyne LASR 47 37 CCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603369 CD On-Demand Anodyne NOD1 93 46 CCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603369 CD On-Demand Anodyne CQSS 54 35 COc1ccc(CN(C)C(=O)Nc2ccc(C(=O)N(C)C)cn2)cc1F ZINC000880603370 FF On-Demand Anodyne F10 27 40 COc1ccc(CN(C)C(=O)Nc2ccc(C(=O)N(C)C)cn2)cc1F ZINC000880603370 FF On-Demand Anodyne MT-ND1 17 41 Cc1nnc(SCC(=O)NCCCOc2ncccn2)n1Cc1ccccc1 ZINC000880603373 GE On-Demand Anodyne PLA2G2A 42 33 CCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603414 CE On-Demand Mild ASAH1 20 41 CCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603414 CE On-Demand Mild LASR 47 37 CCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603414 CE On-Demand Mild NOD1 93 46 CCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603414 CE On-Demand Mild CQSS 54 35 CCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603415 CE On-Demand Mild ASAH1 20 41 CCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603415 CE On-Demand Mild LASR 47 37 CCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603415 CE On-Demand Mild NOD1 93 46 CCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603415 CE On-Demand Mild CQSS 54 35 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603424 DD On-Demand Anodyne ACE 28 46 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603424 DD On-Demand Anodyne MME 48 46 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603424 DD On-Demand Anodyne ACE2 67 43 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603425 DD On-Demand Anodyne ACE 28 46 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603425 DD On-Demand Anodyne MME 48 46 C[C@@H](Cc1ccc(F)cc1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603425 DD On-Demand Anodyne ACE2 67 43 CCN(Cc1ccc(C(F)(F)F)cc1)C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603427 GH On-Demand Anodyne F10 17 43 CCN(Cc1ccc(C(F)(F)F)cc1)C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603427 GH On-Demand Anodyne MTTP 25 43 C[C@H](NC(=O)c1cccnc1Cl)c1nnc(O)n1C ZINC000880603430 CD On-Demand Anodyne G2YM83_BOTF4 77 39 C[C@@H](NC(=O)c1cccnc1Cl)c1nnc(O)n1C ZINC000880603431 CD On-Demand Anodyne G2YM83_BOTF4 77 39 CC(C)c1ccc(OCC(=O)N[C@H](C)c2nnc(O)n2C)cc1 ZINC000880603433 DD On-Demand Anodyne ACACA 16 40 CC(C)c1ccc(OCC(=O)N[C@H](C)c2nnc(O)n2C)cc1 ZINC000880603433 DD On-Demand Anodyne ACACB 17 40 CC(C)c1ccc(OCC(=O)N[C@@H](C)c2nnc(O)n2C)cc1 ZINC000880603434 DD On-Demand Anodyne ACACA 16 40 CC(C)c1ccc(OCC(=O)N[C@@H](C)c2nnc(O)n2C)cc1 ZINC000880603434 DD On-Demand Anodyne ACACB 17 40 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880603442 IF On-Demand Anodyne KDR 41 36 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880603442 IF On-Demand Anodyne GRM4 19 52 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880603442 IF On-Demand Anodyne ENPP1 50 32 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880603442 IF On-Demand Anodyne KCNK3 55 42 COc1cc(NC(=O)c2ccco2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880603442 IF On-Demand Anodyne KCNK9 51 42 O=C(CCCn1cncn1)NCCCOc1ncccn1 ZINC000880603452 CC On-Demand Anodyne HIS3 50 34 O=C(NCCCOc1ncccn1)c1cc(C2CC2)[nH]n1 ZINC000880603453 CD On-Demand Anodyne PKNB 67 38 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)CC1=O ZINC000880603455 CC On-Demand Anodyne TBK1 76 36 CN1CC[C@H](C(=O)NCCCOc2ncccn2)CC1=O ZINC000880603456 CC On-Demand Anodyne TBK1 76 36 NC(=O)COc1cccc(NC(=O)CSc2nc3cc(Cl)ccc3n2Cc2ccccc2)c1 ZINC000880603461 JI On-Demand Anodyne CYSLTR1 26 41 NC(=O)COc1cccc(NC(=O)CSc2nc3cc(Cl)ccc3n2Cc2ccccc2)c1 ZINC000880603461 JI On-Demand Anodyne ALOX5AP 48 42 NC(=O)COc1cccc(NC(=O)CSc2nc3cc(Cl)ccc3n2Cc2ccccc2)c1 ZINC000880603461 JI On-Demand Anodyne PLA2G2A 78 37 NC(=O)COc1cccc(NC(=O)CSc2nc3cc(Cl)ccc3n2Cc2ccccc2)c1 ZINC000880603461 JI On-Demand Anodyne ENPP1 68 35 NC(=O)COc1cccc(NC(=O)CSc2nc3cc(Cl)ccc3n2Cc2ccccc2)c1 ZINC000880603461 JI On-Demand Anodyne IMDH_CRYPV 26 41 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603484 GD On-Demand Anodyne FKBP1A 24 41 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603484 GD On-Demand Anodyne CELA1 45 35 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603484 GD On-Demand Anodyne TRY1_BOVIN 40 34 O=C(NCCCOc1ncccn1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603484 GD On-Demand Anodyne LGMN 70 37 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603485 GD On-Demand Anodyne FKBP1A 24 41 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603485 GD On-Demand Anodyne CELA1 45 35 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603485 GD On-Demand Anodyne TRY1_BOVIN 40 34 O=C(NCCCOc1ncccn1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880603485 GD On-Demand Anodyne LGMN 70 37 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cc(CN(C)C)ccn1)CC2 ZINC000880603488 FF On-Demand Anodyne P2RY14 43 32 CN(C)Cc1ccnc(NC(=O)NCc2ncc(Cl)s2)c1 ZINC000880603510 EF On-Demand Anodyne TYK2 15 42 O=C(CCCn1ccnc1)NCCCOc1ncccn1 ZINC000880603522 CD On-Demand Anodyne TBXAS1 61 46 O=C(CCCn1ccnc1)NCCCOc1ncccn1 ZINC000880603522 CD On-Demand Anodyne HMOX1 19 42 O=C(CCCn1ccnc1)NCCCOc1ncccn1 ZINC000880603522 CD On-Demand Anodyne HMOX2 35 42 O=C(CCCn1ccnc1)NCCCOc1ncccn1 ZINC000880603522 CD On-Demand Anodyne QPCT 40 43 CN(C)Cc1ccnc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)c1 ZINC000880603538 FD On-Demand Anodyne HTR1F 48 34 CN(C)Cc1ccnc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)c1 ZINC000880603538 FD On-Demand Anodyne L3MBTL3 67 42 CCNc1nc(C)c(C(=O)NCCCOc2ncccn2)s1 ZINC000880603556 DD On-Demand Anodyne SCD1 21 40 C[C@@H](NC(=O)CCCn1ccnc1)c1nnc(O)n1C ZINC000880603585 CC On-Demand Anodyne TBXAS1 48 43 CN(C)C(=O)c1ccc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603595 GE On-Demand Anodyne ACE 22 40 CN(C)C(=O)c1ccc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603595 GE On-Demand Anodyne F10 29 40 CN(C)C(=O)c1ccc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603595 GE On-Demand Anodyne MME 15 40 CN(C)C(=O)c1ccc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603596 GE On-Demand Anodyne ACE 22 40 CN(C)C(=O)c1ccc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603596 GE On-Demand Anodyne F10 29 40 CN(C)C(=O)c1ccc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)nc1 ZINC000880603596 GE On-Demand Anodyne MME 15 40 C[C@@H](NC(=O)Cc1c[nH]c2cc(F)ccc12)c1nnc(O)n1C ZINC000880603634 DD On-Demand Anodyne MPO 69 38 C[C@H](NC(=O)Cc1c[nH]c2cc(F)ccc12)c1nnc(O)n1C ZINC000880603635 DD On-Demand Anodyne MPO 69 38 C[C@@H](NC(=O)Cc1ccc(Cl)c(F)c1)c1nnc(O)n1C ZINC000880603637 DD On-Demand Anodyne AVPR1A 15 43 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne DRD2 28 41 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne ADRA1D 20 53 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne ADRA1A 21 53 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne DRD3 53 41 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne CHRNA7 21 48 CN(C)C(=O)c1ccc(NC(=O)NCCCCCCCN2CCCC2)nc1 ZINC000880603641 GF On-Demand Anodyne HNMT 65 39 CN(C)C(=O)c1ccc(NC(=O)NNc2ccc(C(C)(C)C)cc2)nc1 ZINC000880603646 FG On-Demand Reactive MAP3K5 43 32 C[C@@H](NC(=O)c1ccccc1OC1CC1)c1nnc(O)n1C ZINC000880603673 DD On-Demand Anodyne HCN1 56 32 C[C@@H](NC(=O)c1ccccc1OC1CC1)c1nnc(O)n1C ZINC000880603673 DD On-Demand Anodyne HCN4 40 32 C[C@H](NC(=O)c1ccccc1OC1CC1)c1nnc(O)n1C ZINC000880603674 DD On-Demand Anodyne HCN1 56 32 C[C@H](NC(=O)c1ccccc1OC1CC1)c1nnc(O)n1C ZINC000880603674 DD On-Demand Anodyne HCN4 40 32 CC(C)(C)OC(=O)N1CCC(CC(=O)NCCCOc2ncccn2)CC1 ZINC000880603676 GE On-Demand Anodyne GRIN2B 21 41 CC(C)(C)OC(=O)N1CCC(CC(=O)NCCCOc2ncccn2)CC1 ZINC000880603676 GE On-Demand Anodyne GPR119 53 50 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCCCC3=O)cc2)nc1 ZINC000880603684 GF On-Demand Anodyne F10 17 49 C[C@@H](NC(=O)CCCOc1cccc(Br)c1)c1nnc(O)n1C ZINC000880603688 GE On-Demand Anodyne HMOX2 19 40 C[C@@H](Cc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880603699 DE On-Demand Anodyne MME 61 40 C[C@@H](Cc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880603699 DE On-Demand Anodyne GRIA1 46 37 C[C@@H](Cc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880603699 DE On-Demand Anodyne ACE2 56 40 C[C@@H](Cc1ccc(F)cc1)C(=O)NCCCOc1ncccn1 ZINC000880603699 DE On-Demand Anodyne LEF 65 35 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne GRIN2B 30 57 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne PREP 38 42 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne TGM2 43 40 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne KLK5 40 36 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne F13A1 35 40 O=C(NCCCOc1ncccn1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880603712 GE On-Demand Anodyne TBK1 74 33 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne CNR1 20 51 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne LPAR1 25 45 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne LPAR2 18 45 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne PLA2G4B 61 33 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne FAAH 47 40 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne EPHX2 15 47 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne ASAH1 84 37 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne NOD1 58 39 CCCCCCC(=O)NCCCOc1ncccn1 ZINC000880603715 CE On-Demand Anodyne CQSS 49 30 COc1cc(C(=O)N[C@@H](C)c2nnc(O)n2C)ccc1OCc1ccccc1 ZINC000880603774 GF On-Demand Anodyne TSHR 44 36 COc1cc(C(=O)N[C@@H](C)c2nnc(O)n2C)ccc1OCc1ccccc1 ZINC000880603774 GF On-Demand Anodyne PTGER1 52 40 COc1cc(C(=O)N[C@@H](C)c2nnc(O)n2C)ccc1OCc1ccccc1 ZINC000880603774 GF On-Demand Anodyne CTSK 19 42 COc1cc(C(=O)N[C@@H](C)c2nnc(O)n2C)ccc1OCc1ccccc1 ZINC000880603774 GF On-Demand Anodyne HCRTR2 17 40 COc1cc(C(=O)N[C@@H](C)c2nnc(O)n2C)ccc1OCc1ccccc1 ZINC000880603774 GF On-Demand Anodyne ABCG2 27 40 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603781 CC On-Demand Anodyne TBK1 61 36 CN1CC[C@@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603781 CC On-Demand Anodyne GPBAR1 16 40 CN1CC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603782 CC On-Demand Anodyne TBK1 61 36 CN1CC[C@H](C(=O)NCCCOc2ncccn2)C1 ZINC000880603782 CC On-Demand Anodyne GPBAR1 16 40 Cc1ccc(CN2CCO[C@H](CNC(=O)Nc3cc(CN(C)C)ccn3)C2)cc1 ZINC000880603825 GE On-Demand Anodyne DRD4 15 41 O=C(Cc1ccncc1)NCCCOc1ncccn1 ZINC000880603830 CC On-Demand Anodyne CA5B 22 46 O=C(Cc1ccncc1)NCCCOc1ncccn1 ZINC000880603830 CC On-Demand Anodyne CA5A 20 46 COc1csc(C(=O)NCCCOc2ncccn2)c1 ZINC000880603834 CD On-Demand Anodyne MTNR1A 20 40 COc1csc(C(=O)NCCCOc2ncccn2)c1 ZINC000880603834 CD On-Demand Anodyne MTNR1B 19 40 COc1csc(C(=O)NCCCOc2ncccn2)c1 ZINC000880603834 CD On-Demand Anodyne IKBKE 19 42 COc1csc(C(=O)NCCCOc2ncccn2)c1 ZINC000880603834 CD On-Demand Anodyne TBK1 24 42 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880603863 GH On-Demand Anodyne RBP4 40 42 COc1ccccc1[C@H]1CCCN(C(=O)Nc2cc(CN(C)C)ccn2)CC1 ZINC000880603865 GH On-Demand Anodyne RBP4 40 42 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cc(CN(C)C)ccn1)CC2 ZINC000880603874 GG On-Demand Anodyne QRFPR 15 42 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cc(CN(C)C)ccn1)CC2 ZINC000880603875 GG On-Demand Anodyne QRFPR 15 42 CN(C)Cc1ccnc(NC(=O)N2CCc3c(CC(N)=O)cccc3C2)c1 ZINC000880603880 FD On-Demand Anodyne P2RY14 42 31 C[C@@H](NC(=O)Cc1cc2cc(Cl)ccc2[nH]1)c1nnc(O)n1C ZINC000880603924 EE On-Demand Anodyne PYGL 53 39 C[C@H](NC(=O)Cc1cc2cc(Cl)ccc2[nH]1)c1nnc(O)n1C ZINC000880603925 EE On-Demand Anodyne PYGL 53 39 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N(C)C)c(F)c2)nc1 ZINC000880603943 FE On-Demand Clean F10 24 42 C[C@@H]1CCOCCN1C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603966 DD On-Demand Anodyne MTOR 34 41 C[C@H]1CCOCCN1C(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880603967 DD On-Demand Anodyne MTOR 34 41 CCCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603975 CF On-Demand Mild ASAH1 20 41 CCCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603975 CF On-Demand Mild LASR 47 37 CCCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603975 CF On-Demand Mild NOD1 93 46 CCCCCCCCCC(=O)N[C@H](C)c1nnc(O)n1C ZINC000880603975 CF On-Demand Mild CQSS 54 35 CCCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603976 CF On-Demand Mild ASAH1 20 41 CCCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603976 CF On-Demand Mild LASR 47 37 CCCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603976 CF On-Demand Mild NOD1 93 46 CCCCCCCCCC(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880603976 CF On-Demand Mild CQSS 54 35 CCOC(=O)N1CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880603988 ED On-Demand Anodyne P2RY12 51 42 O=C(NCCCOc1ncccn1)c1ccc(F)c(C(F)(F)F)c1 ZINC000880603990 EF On-Demand Anodyne TAAR1 24 47 O=C(NCCCOc1ncccn1)c1ccc(F)c(C(F)(F)F)c1 ZINC000880603990 EF On-Demand Anodyne SUCNR1 48 39 O=C(CSc1ccc(Cl)cc1)NCCCOc1ncccn1 ZINC000880603996 EF On-Demand Anodyne FAS 43 36 O=C(NCCCOc1ncccn1)C1CCN(C(=O)/C=C/c2ccccc2)CC1 ZINC000880604006 GE On-Demand Anodyne TBK1 43 31 O=C(NCCCOc1ncccn1)C1CCN(C(=O)/C=C\c2ccccc2)CC1 ZINC000880604007 GE On-Demand Anodyne TBK1 43 31 O=C(NCCCOc1ncccn1)[C@@H]1CC(c2cccc(F)c2)=NO1 ZINC000880604009 ED On-Demand Anodyne LUCI_PHOPY 22 42 O=C(NCCCOc1ncccn1)[C@H]1CC(c2cccc(F)c2)=NO1 ZINC000880604010 ED On-Demand Anodyne LUCI_PHOPY 22 42 C[C@@H](NC(=O)CCc1ccc(-c2ccccc2)[nH]1)c1nnc(O)n1C ZINC000880604017 EE On-Demand Anodyne PARP3 21 40 COCCCONC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880604045 CC On-Demand Anodyne F10 25 40 O=C(NCc1nnc(O)n1C1CC1)C(=O)c1cc(Cl)cc(Cl)c1 ZINC000880604060 FE On-Demand Anodyne CACNA1I 46 33 O=C(CCc1ccc2ccccc2n1)NCCCOc1ncccn1 ZINC000880604158 EF On-Demand Anodyne CYSLTR1 58 42 O=C(CCc1ccc2ccccc2n1)NCCCOc1ncccn1 ZINC000880604158 EF On-Demand Anodyne PDE10A 15 41 O=C(CCc1ccc2ccccc2n1)NCCCOc1ncccn1 ZINC000880604158 EF On-Demand Anodyne SUCNR1 66 41 CN(C)Cc1ccnc(NC(=O)N2CCc3ncncc3C2)c1 ZINC000880604166 DD On-Demand Anodyne P2RY14 47 36 CCOC(=O)N1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880604291 FD On-Demand Anodyne P2RY12 42 40 CCONC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880604316 CC On-Demand Anodyne F10 22 40 C#CC[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880604333 FF On-Demand Mild GCK 18 42 C#CC[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880604334 FF On-Demand Mild GCK 18 42 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne DRD2 35 48 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne DRD4 43 34 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne ADRA1D 23 43 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne HTR2A 32 41 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne HTR2C 33 41 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne SLC6A4 15 41 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne ADRA1A 25 43 Cc1ccc(N2CCCC2)c(C(=O)NCCCOc2ncccn2)c1 ZINC000880604343 EF On-Demand Anodyne DRD3 62 48 O=C(NCCCOc1ncccn1)c1sccc1SC(F)F ZINC000880604403 EG On-Demand Anodyne MAP1 52 34 CN(C)Cc1ccnc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880604447 GF On-Demand Anodyne NPY2R 65 40 CN(C)Cc1ccnc(NC(=O)N2CCN(c3ccc(F)cc3F)CC2)c1 ZINC000880604447 GF On-Demand Anodyne FAAH 21 42 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1cc(CN(C)C)ccn1)C2 ZINC000880604454 FF On-Demand Anodyne QRFPR 25 42 CN(C)C(=O)c1ccc(NC(=O)NC[C@H](O)c2cccc(C(F)(F)F)c2)nc1 ZINC000880604474 GF On-Demand Anodyne MTTP 26 41 CN(C)C(=O)c1ccc(NC(=O)NC[C@@H](O)c2cccc(C(F)(F)F)c2)nc1 ZINC000880604475 GF On-Demand Anodyne MTTP 26 41 N#Cc1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880604482 DD On-Demand Mild MTNR1A 24 40 N#Cc1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880604482 DD On-Demand Mild MTNR1B 18 40 O=C(NCCCOc1ncccn1)[C@@H]1CC(c2ccccc2)=NO1 ZINC000880604488 ED On-Demand Anodyne LUCI_PHOPY 54 37 O=C(NCCCOc1ncccn1)[C@H]1CC(c2ccccc2)=NO1 ZINC000880604490 ED On-Demand Anodyne LUCI_PHOPY 54 37 O=C(NCCCOc1ncccn1)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880604525 FD On-Demand Anodyne CA2 19 42 O=C(NCCCOc1ncccn1)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880604542 FD On-Demand Anodyne TBK1 74 40 CCn1c(S)nc2cc(C(=O)NCCCOc3ncccn3)ccc2c1=O ZINC000880604545 GD On-Demand Anodyne POLR1A 51 33 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA2 74 50 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA1 57 50 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA7 44 38 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA5B 55 38 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA4 74 50 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA5A 59 38 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA12 33 40 CN(CC(=O)NC(C)(C)C)C(=O)c1cc(S(N)(=O)=O)ccc1F ZINC000880604546 EC On-Demand Anodyne CA9 34 40 O=C(NCCCOc1ncccn1)c1ccc(S(=O)(=O)C(F)(F)F)cc1 ZINC000880604547 GD On-Demand Anodyne CA2 15 42 O=C(NCCCOc1ncccn1)c1ccc(N2CCOCC2)nc1 ZINC000880604550 EC On-Demand Anodyne DRD3 30 41 O=C(NCCCOc1ncccn1)c1ccc(N2CCOCC2)nc1 ZINC000880604550 EC On-Demand Anodyne HDAC1 19 40 O=C(NCCCOc1ncccn1)c1ccc(N2CCOCC2)nc1 ZINC000880604550 EC On-Demand Anodyne SCN10A 15 40 O=C(NCCCOc1ncccn1)c1ccc(N2CCOCC2)nc1 ZINC000880604550 EC On-Demand Anodyne DGAT1 28 41 O=C(NCCCOc1ncccn1)c1ccc(N2CCOCC2)nc1 ZINC000880604550 EC On-Demand Anodyne HPGDS 42 50 CCCCCCCCNC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880604561 DG On-Demand Mild ASAH1 72 34 CC[C@@H](NC(=O)Nc1ccc(C(=O)N(C)C)cn1)c1ccccc1OC ZINC000880604574 FG On-Demand Anodyne GCK 21 41 COc1ccc(N2CCC(NC(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880604603 GF On-Demand Clean F10 20 42 COc1ccc(N2CCC(NC(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880604603 GF On-Demand Clean MCHR1 16 47 C[C@H](NC(=O)c1ccc(F)c(C(F)(F)F)c1)c1nnc(O)n1C ZINC000880604606 EE On-Demand Anodyne TAAR1 20 43 C[C@@H](NC(=O)c1ccc(F)c(C(F)(F)F)c1)c1nnc(O)n1C ZINC000880604609 EE On-Demand Anodyne TAAR1 20 43 C[C@H](NC(=O)/C=C/c1ccsc1)c1nnc(O)n1C ZINC000880604614 CD On-Demand Anodyne UL26 71 48 C[C@H](NC(=O)/C=C/c1ccsc1)c1nnc(O)n1C ZINC000880604614 CD On-Demand Anodyne SCAF_EBVB9 61 34 C[C@H](NC(=O)/C=C\c1ccsc1)c1nnc(O)n1C ZINC000880604619 CD On-Demand Anodyne UL26 71 48 C[C@H](NC(=O)/C=C\c1ccsc1)c1nnc(O)n1C ZINC000880604619 CD On-Demand Anodyne SCAF_EBVB9 61 34 O=C(NCc1nnc(O)n1C1CC1)c1cccc(SC(F)(F)F)c1 ZINC000880604627 FF On-Demand Anodyne CCR2 44 41 CCCCCCCC[C@@H](C)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880604641 DG On-Demand Mild NOD1 76 39 CCCCCCCC[C@@H](C)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880604643 DG On-Demand Mild NOD1 76 39 CCCCCCCC[C@H](C)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880604645 DG On-Demand Mild NOD1 76 39 CCCCCCCC[C@H](C)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880604648 DG On-Demand Mild NOD1 76 39 O=C(NCc1nnc(O)n1C1CC1)[C@H](F)CC1CCCCC1 ZINC000880604720 DE On-Demand Anodyne PROC 40 32 O=C(NCc1nnc(O)n1C1CC1)[C@@H](F)CC1CCCCC1 ZINC000880604721 DE On-Demand Anodyne PROC 40 32 O=C(NCc1nnc(O)n1C1CC1)c1cc2c(Br)c(F)ccc2[nH]1 ZINC000880604724 GF On-Demand Anodyne PLD1 60 35 O=C(NCc1nnc(O)n1C1CC1)c1cc2c(Br)c(F)ccc2[nH]1 ZINC000880604724 GF On-Demand Anodyne PLD2 42 35 O=C(NCc1nnc(O)n1C1CC1)c1ccccc1OC1CC1 ZINC000880604726 DD On-Demand Anodyne SCD 24 41 O=C(NCc1nnc(O)n1C1CC1)c1ccccc1OC1CC1 ZINC000880604726 DD On-Demand Anodyne HCN1 76 39 O=C(NCc1nnc(O)n1C1CC1)c1ccccc1OC1CC1 ZINC000880604726 DD On-Demand Anodyne HCN4 57 39 CN(C)Cc1ccnc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)c1 ZINC000880604735 FE On-Demand Mild PDGFRB 16 41 CN(C)Cc1ccnc(NC(=O)N2CC[C@H](c3cc(O)nc(N(C)C)n3)C2)c1 ZINC000880604749 GD On-Demand Anodyne MAP3K12 37 42 CN(C)Cc1ccnc(NC(=O)N2CC[C@@H](c3cc(O)nc(N(C)C)n3)C2)c1 ZINC000880604751 GD On-Demand Anodyne MAP3K12 37 42 O=C(NCCCOc1ncccn1)c1cc(Cl)nc(N2CCCC2)c1 ZINC000880604756 FE On-Demand Anodyne HTR1A 15 40 O=C(NCCCOc1ncccn1)c1cc(Cl)nc(N2CCCC2)c1 ZINC000880604756 FE On-Demand Anodyne DRD4 44 35 O=C(NCCCOc1ncccn1)c1cc(Cl)nc(N2CCCC2)c1 ZINC000880604756 FE On-Demand Anodyne DRD3 43 38 O=C(Cc1ccc(Cl)c(F)c1)NCc1nnc(O)n1C1CC1 ZINC000880604762 DD On-Demand Anodyne AVPR1A 15 43 O=C(Cc1ccc(Cl)c(F)c1)NCc1nnc(O)n1C1CC1 ZINC000880604762 DD On-Demand Anodyne P2RX7 68 38 CN(C)Cc1ccnc(NC(=O)N2C[C@@H](CN(C)C)[C@H](CN(C)C)C2)c1 ZINC000880604774 FD On-Demand Anodyne TYK2 15 42 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne F2 43 41 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne FKBP1A 41 46 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne CELA1 50 37 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne TRY1_BOVIN 52 39 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne PREP 41 45 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne LGMN 59 33 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne TPP2 30 40 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCCOc1ncccn1 ZINC000880604816 FD On-Demand Anodyne TBK1 48 30 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne F2 43 41 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne FKBP1A 41 46 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne CELA1 50 37 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne TRY1_BOVIN 52 39 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne PREP 41 45 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne LGMN 59 33 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne TPP2 30 40 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCCOc1ncccn1 ZINC000880604817 FD On-Demand Anodyne TBK1 48 30 CN(C)Cc1ccnc(NC(=O)N2CCc3cc(F)c(F)cc3C2)c1 ZINC000880604837 EG On-Demand Anodyne QRFPR 25 41 COc1ccc(CN(CCO)C(=O)Nc2cc(CN(C)C)ccn2)cc1 ZINC000880604838 FE On-Demand Anodyne ROCK2 22 44 C[C@@H](NC(=O)c1ccc(CN2CCN(C)CC2)cc1)c1nnc(O)n1C ZINC000880604848 FC On-Demand Anodyne HSP90AA1 19 42 C[C@@H](NC(=O)c1ccc(CN2CCN(C)CC2)cc1)c1nnc(O)n1C ZINC000880604848 FC On-Demand Anodyne NOD2 41 35 C[C@H](NC(=O)c1ccc(CN2CCN(C)CC2)cc1)c1nnc(O)n1C ZINC000880604850 FC On-Demand Anodyne HSP90AA1 19 42 C[C@H](NC(=O)c1ccc(CN2CCN(C)CC2)cc1)c1nnc(O)n1C ZINC000880604850 FC On-Demand Anodyne NOD2 41 35 COc1ccc(CC(=O)NCCCOc2ncccn2)cc1F ZINC000880604851 DD On-Demand Anodyne DRD3 15 40 COc1ccc(CC(=O)NCCCOc2ncccn2)cc1F ZINC000880604851 DD On-Demand Anodyne MTNR1A 26 41 COc1ccc(CC(=O)NCCCOc2ncccn2)cc1F ZINC000880604851 DD On-Demand Anodyne MTNR1B 24 42 COc1ccc(CC(=O)NCCCOc2ncccn2)cc1F ZINC000880604851 DD On-Demand Anodyne MET 41 39 COc1ccc(N2CCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880604862 GE On-Demand Clean PDGFRB 48 39 O=C(NCCCOc1ncccn1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880604870 ED On-Demand Anodyne INHA 22 46 O=C(NCCCOc1ncccn1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880604872 ED On-Demand Anodyne INHA 22 46 C[C@H](NC(=O)c1cccn1[C@@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604877 FF On-Demand Anodyne MME 66 36 C[C@H](NC(=O)c1cccn1[C@@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604877 FF On-Demand Anodyne ACE2 41 35 C[C@H](NC(=O)c1cccn1[C@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604879 FF On-Demand Anodyne MME 66 36 C[C@H](NC(=O)c1cccn1[C@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604879 FF On-Demand Anodyne ACE2 41 35 C[C@@H](Cc1ccccc1)n1cccc1C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880604880 FF On-Demand Anodyne MME 66 36 C[C@@H](Cc1ccccc1)n1cccc1C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880604880 FF On-Demand Anodyne ACE2 41 35 C[C@@H](NC(=O)c1cccn1[C@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604881 FF On-Demand Anodyne MME 66 36 C[C@@H](NC(=O)c1cccn1[C@H](C)Cc1ccccc1)c1nnc(O)n1C ZINC000880604881 FF On-Demand Anodyne ACE2 41 35 C[C@H](NC(=O)/C=C\c1csc(C(F)(F)F)c1)c1nnc(O)n1C ZINC000880604899 EE On-Demand Anodyne UL26 44 34 C[C@H](NC(=O)/C=C/c1csc(C(F)(F)F)c1)c1nnc(O)n1C ZINC000880604904 EE On-Demand Anodyne UL26 44 34 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880604942 FE On-Demand Anodyne FPR1 20 40 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880604945 FE On-Demand Anodyne FPR1 20 40 CN(C)C(=O)c1ccc(NC(=O)NC[C@@]2(C)CCN(Cc3ccccc3)C2)nc1 ZINC000880604956 GF On-Demand Anodyne NPFFR1 43 37 CN(C)C(=O)c1ccc(NC(=O)NC[C@]2(C)CCN(Cc3ccccc3)C2)nc1 ZINC000880604960 GF On-Demand Anodyne NPFFR1 43 37 C[C@@H](NC(=O)CCSc1ccc(Cl)cc1)c1nnc(O)n1C ZINC000880604988 EF On-Demand Anodyne PRCP 18 41 CCc1ccc(C(=O)N[C@H](C)c2nnc(O)n2C)s1 ZINC000880605004 CD On-Demand Anodyne FOLR1 44 34 CCc1ccc(C(=O)N[C@H](C)c2nnc(O)n2C)s1 ZINC000880605004 CD On-Demand Anodyne SLC46A1 40 30 CCc1ccc(C(=O)N[C@@H](C)c2nnc(O)n2C)s1 ZINC000880605006 CD On-Demand Anodyne FOLR1 44 34 CCc1ccc(C(=O)N[C@@H](C)c2nnc(O)n2C)s1 ZINC000880605006 CD On-Demand Anodyne SLC46A1 40 30 C[C@@H](NC(=O)CCCc1ccc(C(C)(C)C)cc1)c1nnc(O)n1C ZINC000880605008 EG On-Demand Anodyne LHCGR 31 41 CCOc1ccccc1OCC(=O)NCCCOc1ncccn1 ZINC000880605082 ED On-Demand Anodyne HCN1 46 31 O=C(COc1cccc(Br)c1)NCCCOc1ncccn1 ZINC000880605083 FE On-Demand Anodyne HRH2 27 41 O=C(COc1cccc(Br)c1)NCCCOc1ncccn1 ZINC000880605083 FE On-Demand Anodyne MTNR1A 32 43 O=C(COc1cccc(Br)c1)NCCCOc1ncccn1 ZINC000880605083 FE On-Demand Anodyne MTNR1B 29 43 O=C(COc1cccc(Br)c1)NCCCOc1ncccn1 ZINC000880605083 FE On-Demand Anodyne HMOX2 19 41 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne HTR1A 25 40 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne DRD2 29 42 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne DRD4 42 32 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne ADRA1A 20 40 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne DRD3 43 42 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne MTNR1A 30 42 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne MTNR1B 34 42 COc1cccc(OC)c1C(=O)NCCCOc1ncccn1 ZINC000880605088 DD On-Demand Anodyne ALS 47 36 O=C(Cc1ccc(Br)cc1Cl)NCc1nnc(O)n1C1CC1 ZINC000880605098 GF On-Demand Anodyne P2RX7 47 39 CN(C)C(=O)c1ccc(NC(=O)NCc2ccccc2N2CCOCC2)nc1 ZINC000880605120 GD On-Demand Anodyne F10 19 49 CN(C)C(=O)c1ccc(NC(=O)NCc2ccccc2N2CCOCC2)nc1 ZINC000880605120 GD On-Demand Anodyne PIK3CA 36 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccccc2N2CCOCC2)nc1 ZINC000880605120 GD On-Demand Anodyne MTOR 58 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccccc2N2CCOCC2)nc1 ZINC000880605120 GD On-Demand Anodyne SCN10A 21 48 C[C@H](Sc1nc2ccccc2s1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880605129 FE On-Demand Anodyne ST14 40 34 C[C@H](Sc1nc2ccccc2s1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880605129 FE On-Demand Anodyne TMPRSS6 56 34 C[C@H](NC(=O)[C@@H](C)Sc1nc2ccccc2s1)c1nnc(O)n1C ZINC000880605130 FE On-Demand Anodyne ST14 40 34 C[C@H](NC(=O)[C@@H](C)Sc1nc2ccccc2s1)c1nnc(O)n1C ZINC000880605130 FE On-Demand Anodyne TMPRSS6 56 34 C[C@H](Sc1nc2ccccc2s1)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880605131 FE On-Demand Anodyne ST14 40 34 C[C@H](Sc1nc2ccccc2s1)C(=O)N[C@@H](C)c1nnc(O)n1C ZINC000880605131 FE On-Demand Anodyne TMPRSS6 56 34 C[C@@H](Sc1nc2ccccc2s1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880605132 FE On-Demand Anodyne ST14 40 34 C[C@@H](Sc1nc2ccccc2s1)C(=O)N[C@H](C)c1nnc(O)n1C ZINC000880605132 FE On-Demand Anodyne TMPRSS6 56 34 Cc1cccc2c1CCN(C(=O)Nc1ccc(C(=O)N(C)C)cn1)C2 ZINC000880605136 EF On-Demand Anodyne P2RY14 44 33 CCCCSCC(=O)NCCCOc1ncccn1 ZINC000880605171 CD On-Demand Anodyne EST1_PIG 45 39 C[C@H](NC(=O)CSc1nc2ccccc2s1)c1nnc(O)n1C ZINC000880605175 EE On-Demand Anodyne ST14 41 35 C[C@H](NC(=O)CSc1nc2ccccc2s1)c1nnc(O)n1C ZINC000880605175 EE On-Demand Anodyne TMPRSS6 59 35 CC(=O)N1CCc2ccccc2[C@@H]1CC(=O)NCCCOc1ncccn1 ZINC000880605184 FD On-Demand Anodyne MTNR1A 15 41 CC(=O)N1CCc2ccccc2[C@@H]1CC(=O)NCCCOc1ncccn1 ZINC000880605184 FD On-Demand Anodyne MTNR1B 24 48 COc1ccc(N2CCCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880605192 GF On-Demand Clean F10 16 49 COc1ccc(N2CCCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880605192 GF On-Demand Clean PDGFRB 43 37 C#CCN1CCC(C(=O)NCCCOc2ncccn2)CC1 ZINC000880605220 DC On-Demand Mild TBK1 66 34 CC(=O)c1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880605247 ED On-Demand Anodyne DRD4 40 30 CC(=O)c1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880605247 ED On-Demand Anodyne HRH2 27 44 CC(=O)c1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880605247 ED On-Demand Anodyne MTNR1A 55 44 CC(=O)c1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880605247 ED On-Demand Anodyne MTNR1B 50 44 CC(=O)c1cccc(OCC(=O)NCCCOc2ncccn2)c1 ZINC000880605247 ED On-Demand Anodyne PLA2G4B 26 40 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCCC3)cc2)nc1 ZINC000880605254 FF On-Demand Clean F10 24 41 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCCC3)cc2)nc1 ZINC000880605254 FF On-Demand Clean FLT3 15 42 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCCC3)cc2)nc1 ZINC000880605254 FF On-Demand Clean NAMPT 41 38 CC(C)c1cc(NC(=O)Nc2cc(CN(C)C)ccn2)ccc1O ZINC000880605258 EH On-Demand Anodyne THRA 60 35 CC(C)c1cc(NC(=O)Nc2cc(CN(C)C)ccn2)ccc1O ZINC000880605258 EH On-Demand Anodyne THRB 60 38 CN(C)C(=O)c1ccc(NC(=O)NCCc2ccc(N3CCCCC3)cc2)nc1 ZINC000880605307 GG On-Demand Anodyne F10 17 41 CN(C)C(=O)c1ccc(NC(=O)NCCc2ccc(N3CCCCC3)cc2)nc1 ZINC000880605307 GG On-Demand Anodyne CTSK 24 40 C[C@H](Cc1ccccc1Cl)NC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880605335 FG On-Demand Anodyne GCK 19 41 C[C@@H](Cc1ccccc1Cl)NC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880605336 FG On-Demand Anodyne GCK 19 41 O=C(NCc1nnc(O)n1C1CC1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880605379 FE On-Demand Anodyne C3AR1 45 46 O=C(CCn1ccnc1)NCCCOc1ncccn1 ZINC000880605380 CC On-Demand Anodyne TBXAS1 58 45 O=C(CCn1ccnc1)NCCCOc1ncccn1 ZINC000880605380 CC On-Demand Anodyne HMOX1 19 40 O=C(CCn1ccnc1)NCCCOc1ncccn1 ZINC000880605380 CC On-Demand Anodyne HMOX2 27 40 O=C(CCn1ccnc1)NCCCOc1ncccn1 ZINC000880605380 CC On-Demand Anodyne QPCT 36 42 O=C(NCc1nnc(O)n1C1CC1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880605381 FE On-Demand Anodyne C3AR1 45 46 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C1 ZINC000880605392 GE On-Demand Anodyne NPY5R 27 42 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(N3CCCC3=O)cc2)nc1 ZINC000880605414 GE On-Demand Anodyne F10 16 48 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)nc1 ZINC000880605417 GE On-Demand Anodyne L3MBTL3 49 36 CN(C)C(=O)c1ccc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)nc1 ZINC000880605417 GE On-Demand Anodyne NAMPT 45 52 C[C@@H](NC(=O)c1ccc(CCN(C)C)cc1)c1nnc(O)n1C ZINC000880605481 DD On-Demand Anodyne UTS2 44 34 C[C@H](NC(=O)c1ccc(CCN(C)C)cc1)c1nnc(O)n1C ZINC000880605482 DD On-Demand Anodyne UTS2 44 34 CCc1ccc(N2CCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)cc1 ZINC000880605528 GF On-Demand Anodyne PRNP 42 36 CN(C)C(=O)c1ccc(NC(=O)NOCCC2CC2)nc1 ZINC000880605536 CD On-Demand Anodyne GCK 22 42 CN(C)C(=O)c1ccc(NC(=O)Nc2cccc(C(C)(C)O)c2)nc1 ZINC000880605560 EF On-Demand Anodyne KIT 20 42 CN(C)C(=O)c1ccc(NC(=O)Nc2cccc(C(C)(C)O)c2)nc1 ZINC000880605560 EF On-Demand Anodyne IMDH_CRYPV 52 40 C[C@@H](NC(=O)CCc1cccc2ccccc12)c1nnc(O)n1C ZINC000880605590 DE On-Demand Anodyne MTNR1A 25 40 C[C@@H](NC(=O)CCc1cccc2ccccc12)c1nnc(O)n1C ZINC000880605590 DE On-Demand Anodyne PARP3 22 43 C[C@H](NC(=O)CCc1cccc2ccccc12)c1nnc(O)n1C ZINC000880605591 DE On-Demand Anodyne MTNR1A 25 40 C[C@H](NC(=O)CCc1cccc2ccccc12)c1nnc(O)n1C ZINC000880605591 DE On-Demand Anodyne PARP3 22 43 CN(C)C(=O)c1ccc(NC(=O)NC[C@@](C)(O)c2ccc(F)cc2F)nc1 ZINC000880605703 GE On-Demand Anodyne F10 15 43 CN(C)C(=O)c1ccc(NC(=O)NC[C@](C)(O)c2ccc(F)cc2F)nc1 ZINC000880605704 GE On-Demand Anodyne F10 15 43 CN(C)C(=O)c1ccc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)nc1 ZINC000880605819 GF On-Demand Anodyne MTTP 28 43 CN(C)C(=O)c1ccc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)nc1 ZINC000880605820 GF On-Demand Anodyne MTTP 28 43 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C1CC1 ZINC000880605826 ED On-Demand Anodyne NQO2 29 40 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C1CC1 ZINC000880605826 ED On-Demand Anodyne MTNR1A 28 41 O=C(Cc1cc2cc(Cl)ccc2[nH]1)NCc1nnc(O)n1C1CC1 ZINC000880605834 EE On-Demand Anodyne PYGL 74 39 O=C(Cc1cc2cc(Cl)ccc2[nH]1)NCc1nnc(O)n1C1CC1 ZINC000880605834 EE On-Demand Anodyne PLD1 51 33 Cc1ccc(F)c2[nH]c(C(=O)NCc3nnc(O)n3C3CC3)cc12 ZINC000880605898 EE On-Demand Anodyne PLD1 41 34 O=C(NCc1nnc(O)n1C1CC1)[C@@H]1C[C@H]1c1ccccc1 ZINC000880605992 CD On-Demand Anodyne PLD1 16 45 CN(C)C(=O)c1ccc(NC(=O)NC[C@@](C)(O)c2ccccc2Cl)nc1 ZINC000880606029 GE On-Demand Anodyne ECR 47 34 CN(C)C(=O)c1ccc(NC(=O)NC[C@](C)(O)c2ccccc2Cl)nc1 ZINC000880606030 GE On-Demand Anodyne ECR 47 34 O=C(NCc1nnc(O)n1C1CC1)c1ccnc(C(F)(F)F)c1 ZINC000880606032 ED On-Demand Anodyne CCR2 41 37 COCCONC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880606048 CC On-Demand Anodyne F10 30 42 COCCONC(=O)Nc1ccc(C(=O)N(C)C)cn1 ZINC000880606048 CC On-Demand Anodyne GCK 34 40 CN(C)C(=O)c1ccc(NC(=O)N[C@H]2Cc3ccc(Cl)cc3C2)nc1 ZINC000880606051 FF On-Demand Anodyne F10 39 40 CN(C)C(=O)c1ccc(NC(=O)N[C@@H]2Cc3ccc(Cl)cc3C2)nc1 ZINC000880606052 FF On-Demand Anodyne F10 39 40 CN(C)C(=O)c1ccc(NC(=O)N[C@@H](CCO)Cc2ccccc2)nc1 ZINC000880606155 FD On-Demand Anodyne GCK 16 43 CN(C)C(=O)c1ccc(NC(=O)N[C@H](CCO)Cc2ccccc2)nc1 ZINC000880606156 FD On-Demand Anodyne GCK 16 43 O=C(Cc1ccc2cnccc2c1)NCc1nnc(O)n1C1CC1 ZINC000880606175 DD On-Demand Anodyne NAMPT 40 37 CN1CCC(CNC(=O)Nc2ccc(C(=O)N(C)C)cn2)(c2ccccc2)CC1 ZINC000880606293 GF On-Demand Anodyne KCNA3 48 39 CN1CCC(CNC(=O)Nc2ccc(C(=O)N(C)C)cn2)(c2ccccc2)CC1 ZINC000880606293 GF On-Demand Anodyne SOAT1 17 44 O=C(CNc1cccc(C(F)(F)F)c1)NCc1nnc(O)n1C1CC1 ZINC000880606359 FE On-Demand Anodyne CCR2 107 39 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C1 ZINC000880606362 DD On-Demand Anodyne HCRTR1 17 41 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C1 ZINC000880606362 DD On-Demand Anodyne HCRTR2 30 41 O=C(NCc1nnc(O)n1C1CC1)[C@H](F)Cc1ccccc1 ZINC000880606385 DD On-Demand Anodyne ACE 44 35 O=C(NCc1nnc(O)n1C1CC1)[C@H](F)Cc1ccccc1 ZINC000880606385 DD On-Demand Anodyne MME 62 36 O=C(NCc1nnc(O)n1C1CC1)[C@H](F)Cc1ccccc1 ZINC000880606385 DD On-Demand Anodyne AMP1_PLAFQ 44 38 O=C(NCc1nnc(O)n1C1CC1)[C@@H](F)Cc1ccccc1 ZINC000880606386 DD On-Demand Anodyne ACE 44 35 O=C(NCc1nnc(O)n1C1CC1)[C@@H](F)Cc1ccccc1 ZINC000880606386 DD On-Demand Anodyne MME 62 36 O=C(NCc1nnc(O)n1C1CC1)[C@@H](F)Cc1ccccc1 ZINC000880606386 DD On-Demand Anodyne AMP1_PLAFQ 44 38 CN(C)C(=O)c1ccc(NC(=O)N[C@](C)(CO)Cc2ccc(Cl)cc2)nc1 ZINC000880606414 GF On-Demand Anodyne KLKB1 17 41 CN(C)C(=O)c1ccc(NC(=O)N[C@](C)(CO)Cc2ccc(Cl)cc2)nc1 ZINC000880606414 GF On-Demand Anodyne F10 36 41 CN(C)C(=O)c1ccc(NC(=O)N[C@@](C)(CO)Cc2ccc(Cl)cc2)nc1 ZINC000880606415 GF On-Demand Anodyne KLKB1 17 41 CN(C)C(=O)c1ccc(NC(=O)N[C@@](C)(CO)Cc2ccc(Cl)cc2)nc1 ZINC000880606415 GF On-Demand Anodyne F10 36 41 CN1CCN(C2CCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)CC1 ZINC000880606422 FD On-Demand Anodyne HTR1F 54 32 CN1CCN(C2CCN(C(=O)Nc3ccc(C(=O)N(C)C)cn3)CC2)CC1 ZINC000880606422 FD On-Demand Anodyne L3MBTL3 82 45 O=C(NCc1nnc(O)n1C1CC1)c1ccc(F)c(C(F)(F)F)c1 ZINC000880606451 EE On-Demand Anodyne PLD1 48 34 O=C(NCc1nnc(O)n1C1CC1)[C@@H]1C[C@@H]1Cc1ccccc1 ZINC000880606465 DD On-Demand Anodyne TMPRSS11D 58 34 O=C(NCc1nnc(O)n1C1CC1)[C@H]1C[C@@H]1Cc1ccccc1 ZINC000880606466 DD On-Demand Anodyne TMPRSS11D 58 34 O=C(NCc1nnc(O)n1C1CC1)[C@H]1C[C@H]1Cc1ccccc1 ZINC000880606467 DD On-Demand Anodyne TMPRSS11D 58 34 O=C(NCc1nnc(O)n1C1CC1)[C@@H]1C[C@H]1Cc1ccccc1 ZINC000880606468 DD On-Demand Anodyne TMPRSS11D 58 34 O=C(NCc1nnc(O)n1C1CC1)c1ccc2[nH]ccc2c1 ZINC000880606482 CD On-Demand Anodyne PLD1 48 36 CN(C)C(=O)c1ccc(NC(=O)NN2CCCCC2)nc1 ZINC000880606487 CD On-Demand Anodyne F10 19 40 CN(C)C(=O)c1ccc(NC(=O)NOCC2CC2)nc1 ZINC000880606540 CD On-Demand Anodyne GCK 18 40 CCOc1ccccc1C(F)(F)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606566 FE On-Demand Anodyne HCN1 49 36 CCOc1ccccc1C(F)(F)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606566 FE On-Demand Anodyne HCN4 44 36 COc1ccccc1/C(C)=C\C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606601 EE On-Demand Anodyne KCNA3 44 39 COc1ccccc1/C(C)=C/C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606602 EE On-Demand Anodyne KCNA3 44 39 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606612 GH On-Demand Anodyne AVPR2 17 42 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606612 GH On-Demand Anodyne RBP4 44 40 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606612 GH On-Demand Anodyne SMO 18 41 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606613 GH On-Demand Anodyne AVPR2 17 42 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606613 GH On-Demand Anodyne RBP4 44 40 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606613 GH On-Demand Anodyne SMO 18 41 CN(C)C(=O)c1ccc(NC(=O)NCc2cccc(OC(C)(C)C)c2)nc1 ZINC000880606629 FG On-Demand Anodyne ROCK2 40 42 CN(C)C(=O)c1ccc(NC(=O)NCc2cccc(OC(C)(C)C)c2)nc1 ZINC000880606629 FG On-Demand Anodyne GCK 27 41 COc1ccc(N2CC[C@H](CNC(=O)Nc3ccc(C(=O)N(C)C)cn3)C2)cc1 ZINC000880606655 GE On-Demand Clean F10 41 32 O=C(CCCn1ccnc1)NCc1nnc(O)n1C1CC1 ZINC000880606735 CC On-Demand Anodyne TBXAS1 43 40 O=C(NCc1nnc(O)n1C1CC1)c1ccc(C(F)(F)F)nc1Cl ZINC000880606760 FE On-Demand Anodyne TRPV1 49 35 O=C(NCc1nnc(O)n1C1CC1)c1cc(C(F)(F)F)ccc1F ZINC000880606765 EE On-Demand Anodyne CCR2 63 37 O=C(NCc1nnc(O)n1C1CC1)c1cc(C(F)(F)F)ccc1F ZINC000880606765 EE On-Demand Anodyne LIPG 48 35 CCC1(N2CCCCC2)CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606777 GG On-Demand Anodyne HCN1 40 31 CCC1(N2CCCCC2)CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880606777 GG On-Demand Anodyne HCN4 40 31 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606845 GF On-Demand Anodyne ST14 47 33 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606845 GF On-Demand Anodyne TMPRSS6 64 33 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606846 GF On-Demand Anodyne ST14 47 33 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C1CC1 ZINC000880606846 GF On-Demand Anodyne TMPRSS6 64 33 O=C(NCc1nnc(O)n1C1CC1)c1cnc2ccccn12 ZINC000880606926 CC On-Demand Anodyne EPHB3 21 44 CCC(=O)c1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1F ZINC000880606928 ED On-Demand Anodyne PLD1 53 34 C[C@@H]1CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C[C@H]1c1ccccc1 ZINC000880606935 FG On-Demand Anodyne SMO 30 43 C[C@H]1CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C[C@H]1c1ccccc1 ZINC000880606936 FG On-Demand Anodyne SMO 30 43 C[C@@H]1CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C[C@@H]1c1ccccc1 ZINC000880606937 FG On-Demand Anodyne SMO 30 43 C[C@H]1CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C[C@@H]1c1ccccc1 ZINC000880606938 FG On-Demand Anodyne SMO 30 43 CN(C)C(=O)c1ccc(NC(=O)NOCC2CCC2)nc1 ZINC000880606954 CD On-Demand Anodyne GCK 21 43 O=C(NCc1nnc(O)n1C1CC1)c1[nH]c2ccccc2c1Cl ZINC000880607036 EE On-Demand Anodyne PLD1 40 34 O=C(CSc1nc2ccccc2s1)NCc1nnc(O)n1C1CC1 ZINC000880607050 FE On-Demand Anodyne TMPRSS6 54 33 CCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607058 CD On-Demand Anodyne LASR 62 37 CCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607058 CD On-Demand Anodyne NOD1 52 36 CCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607058 CD On-Demand Anodyne CQSS 50 31 CONC(=O)C1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880607131 DD On-Demand Anodyne TYK2 52 37 Cc1nonc1CNC(=O)Nc1ccnc(N(C)C)c1 ZINC000880607196 CD On-Demand Anodyne CASP7 40 33 COc1ccc(CN(CCO)C(=O)Nc2ccnc(N(C)C)c2)cc1 ZINC000880607202 EE On-Demand Anodyne BMP1 30 41 COc1ccc(CN(CCO)C(=O)Nc2ccnc(N(C)C)c2)cc1 ZINC000880607202 EE On-Demand Anodyne ROCK2 18 46 O=C(NCc1nnc(O)n1C1CC1)c1cccnc1Cl ZINC000880607242 CD On-Demand Anodyne G2YM83_BOTF4 76 39 C[C@@H]1[C@H](C(=O)NNC(=O)Nc2ccnc(N(C)C)c2)CCCN1C ZINC000880607259 ED On-Demand Reactive TYK2 48 32 C#CCC1(O)CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880607271 DD On-Demand Mild S1PR2 27 40 C#CC1(F)CN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)C1 ZINC000880607303 CC On-Demand Mild NPY5R 15 40 Cc1cccc2c1OCC[C@@H]2NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880607361 EG On-Demand Anodyne TRPV1 15 43 C#CCC1(O)CCN(C(=O)Nc2ccc(C(=O)N(C)C)cn2)CC1 ZINC000880607418 ED On-Demand Mild S1PR2 23 41 CN1CCN(C2CCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)CC1 ZINC000880607426 ED On-Demand Anodyne L3MBTL3 67 40 CCCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607435 CF On-Demand Mild LASR 62 37 CCCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607435 CF On-Demand Mild NOD1 52 36 CCCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607435 CF On-Demand Mild CQSS 50 31 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1ccnc(N(C)C)c1)C2 ZINC000880607464 FF On-Demand Anodyne P2RY14 45 31 COC(=O)c1ccc(OC)c2c1CCN(C(=O)Nc1ccnc(N(C)C)c1)C2 ZINC000880607468 GF On-Demand Anodyne P2RY14 46 32 O=C(NCc1nnc(O)n1C1CC1)c1cc(Cl)nc(Cl)c1 ZINC000880607496 ED On-Demand Anodyne CACNA1I 41 32 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccnc(N(C)C)c1)CC2 ZINC000880607565 FF On-Demand Anodyne P2RY14 50 35 CC(=O)C1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880607600 CD On-Demand Anodyne TYK2 43 35 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880607640 CE On-Demand Mild EPHX2 35 40 COc1ccc(CN(CCO)C(=O)Nc2ccc(C(=O)N(C)C)cn2)cc1 ZINC000880607680 FD On-Demand Anodyne ROCK2 17 42 CCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607735 CE On-Demand Mild LASR 62 37 CCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607735 CE On-Demand Mild NOD1 52 36 CCCCCCCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607735 CE On-Demand Mild CQSS 50 31 C[C@H]1c2sccc2CCN1C(=O)Nc1ccnc(N(C)C)c1 ZINC000880607741 DG On-Demand Anodyne TRPM8 22 41 CCc1nc2ccccc2n1CC(=O)NCc1nnc(O)n1C1CC1 ZINC000880607797 ED On-Demand Anodyne FPR2 22 40 COC[C@@H](O)CNC(=O)Nc1ccnc(N(C)C)c1 ZINC000880607831 CC On-Demand Anodyne ADRB1 42 33 O=C(Cc1cccs1)NCc1nnc(O)n1C1CC1 ZINC000880607869 CD On-Demand Anodyne CA5B 32 44 O=C(Cc1cccs1)NCc1nnc(O)n1C1CC1 ZINC000880607869 CD On-Demand Anodyne CA5A 31 44 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)NCc1nnc(O)n1C1CC1 ZINC000880607882 FE On-Demand Anodyne FPR1 25 40 O=C(NCc1nnc(O)n1C1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880607898 FF On-Demand Anodyne PDE4D 19 43 CCCOc1ccc(OCC(=O)NCc2nnc(O)n2C2CC2)cc1 ZINC000880607910 ED On-Demand Anodyne PLA2G4B 59 33 COC(=O)N1CCC(NC(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880607919 DD On-Demand Anodyne EPHX2 54 47 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880608013 FE On-Demand Anodyne MTNR1A 16 41 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880608013 FE On-Demand Anodyne PDGFRA 41 39 CCOC(=O)N1CCCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880608033 ED On-Demand Anodyne P2RY12 43 41 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608034 EE On-Demand Anodyne ADRB1 41 31 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608034 EE On-Demand Anodyne KCNK3 43 38 CC[C@H](C#N)Oc1cc(CNC(=O)Nc2ccnc(N(C)C)c2)ccc1OC ZINC000880608038 GG On-Demand Mild ROCK2 15 42 CCN1[C@@H](C)CN(C(=O)Cc2ccccc2[N+](=O)[O-])C[C@H]1C ZINC000880608061 DE On-Demand Bother COLA 115 36 COc1ccc(CN(C)C(=O)Nc2ccnc(N(C)C)c2)cc1F ZINC000880608070 EF On-Demand Anodyne MET 58 39 COc1ccc(CN(C)C(=O)Nc2ccnc(N(C)C)c2)cc1F ZINC000880608070 EF On-Demand Anodyne PDGFRA 41 37 CCOC(=O)N1CCC(NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880608084 ED On-Demand Anodyne EPHX2 53 48 CCOC(=O)N1CCC(NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880608084 ED On-Demand Anodyne CCR8 23 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nnc(O)n1C1CC1)C2 ZINC000880608172 ED On-Demand Anodyne MTNR1A 34 41 O=C(NCc1nnc(O)n1C1CC1)c1cc(Cl)nc2ccccc12 ZINC000880608173 EE On-Demand Anodyne TACR3 17 44 CNc1nc(C(=O)N2CCN(CC(F)(F)CO)CC2)cs1 ZINC000880608213 DC On-Demand Anodyne TRPC6 55 40 CNc1nc(C(=O)N2CCN(CC(F)(F)CO)CC2)cs1 ZINC000880608213 DC On-Demand Anodyne TRPC3 47 40 CN(C)C(=O)OC1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880608230 ED On-Demand Anodyne LIMK2 15 43 O=C(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCN(CC(F)(F)CO)CC1 ZINC000880608233 FD On-Demand Bother L3MBTL3 17 41 CCOc1ccccc1OCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880608282 ED On-Demand Anodyne HCN1 52 38 CCOc1ccccc1OCC(=O)NCc1nnc(O)n1C1CC1 ZINC000880608282 ED On-Demand Anodyne HCN4 47 38 CCN1[C@@H](C)CN(C(=O)COc2ccc3ccc(=O)oc3c2)C[C@H]1C ZINC000880608300 EE On-Demand Anodyne MAOA 32 41 CCN1[C@@H](C)CN(C(=O)COc2ccc3ccc(=O)oc3c2)C[C@H]1C ZINC000880608300 EE On-Demand Anodyne MAOB 18 43 C[C@@H]1CCNC(=O)[C@@H]1NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608305 CC On-Demand Anodyne TYK2 46 34 C[C@H]1CCNC(=O)[C@H]1NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608307 CC On-Demand Anodyne TYK2 46 34 C[C@H]1CCNC(=O)[C@@H]1NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608309 CC On-Demand Anodyne TYK2 46 34 C[C@@H]1CCNC(=O)[C@H]1NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880608311 CC On-Demand Anodyne TYK2 46 34 CCOC(=O)N1CCC(NC(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880608335 ED On-Demand Anodyne EPHX2 57 49 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608345 FD On-Demand Anodyne PAPA1_CARPA 32 40 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608345 FD On-Demand Anodyne CTSK 15 46 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608347 FD On-Demand Anodyne PAPA1_CARPA 32 40 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608347 FD On-Demand Anodyne CTSK 15 46 CC(=O)N1CCC[C@@H]1C(=O)NNc1c(Cl)cccc1Br ZINC000880608358 FF On-Demand Reactive CELA1 28 41 CC(=O)N1CCC[C@@H]1C(=O)NNc1c(Cl)cccc1Br ZINC000880608358 FF On-Demand Reactive LGMN 68 38 CC(=O)N1CCC[C@@H]1C(=O)NNc1c(Cl)cccc1Br ZINC000880608358 FF On-Demand Reactive XIAP 44 40 Cc1nnc(CCNC(=O)Nc2ccnc(N(C)C)c2)s1 ZINC000880608368 DD On-Demand Anodyne PRMT3 43 32 O=C(NCc1nnc(O)n1C1CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880608372 EE On-Demand Anodyne OPRL1 17 44 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880608376 GG On-Demand Anodyne PDGFRB 41 36 CCN1[C@@H](C)CN(C(=O)[C@H](O)c2cccnc2)C[C@H]1C ZINC000880608399 CD On-Demand Anodyne PTAFR 15 40 CCN1[C@@H](C)CN(C(=O)[C@@H](O)c2cccnc2)C[C@H]1C ZINC000880608400 CD On-Demand Anodyne PTAFR 15 40 CC[C@@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1ccccc1OC ZINC000880608407 EG On-Demand Anodyne KCNK3 51 40 CC[C@@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1ccccc1OC ZINC000880608407 EG On-Demand Anodyne KCNK9 43 40 CCN1[C@@H](C)CN(C(=O)c2cn(CCOC)c3ccccc23)C[C@H]1C ZINC000880608424 EF On-Demand Anodyne CNR1 30 56 CCN1[C@@H](C)CN(C(=O)c2cn(CCOC)c3ccccc23)C[C@H]1C ZINC000880608424 EF On-Demand Anodyne CNR2 37 56 CCN1[C@@H](C)CN(C(=O)c2cn(CCOC)c3ccccc23)C[C@H]1C ZINC000880608424 EF On-Demand Anodyne TPSAB1 22 54 CCN1[C@@H](C)CN(C(=O)CSc2nnc(-c3ccc(OC)cc3)o2)C[C@H]1C ZINC000880608425 GF On-Demand Anodyne GSK3A 18 42 COC(=O)N1CCC(NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880608448 ED On-Demand Anodyne EPHX2 55 48 CCN1[C@@H](C)CN(C(=O)c2cccc(NC(=O)OC)c2)C[C@H]1C ZINC000880608457 DE On-Demand Anodyne KCNK3 60 34 C[C@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880608473 GF On-Demand Clean MTOR 45 38 C[C@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880608473 GF On-Demand Clean EPHB4 75 37 C[C@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880608473 GF On-Demand Clean STAT6 52 31 CCN1[C@@H](C)CN(C(=O)c2ccnc(N3CCCC3)n2)C[C@H]1C ZINC000880608481 DD On-Demand Anodyne SORD 42 35 O=C(COc1cccc(C(F)(F)F)c1)NCc1nnc(O)n1C1CC1 ZINC000880608506 FE On-Demand Anodyne CCR2 81 39 O=C(COc1cccc(C(F)(F)F)c1)NCc1nnc(O)n1C1CC1 ZINC000880608506 FE On-Demand Anodyne PDS 48 43 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne TSHR 49 33 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne PPARG 15 45 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne PTGER1 44 33 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne MTNR1B 15 43 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne SLC6A5 27 40 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne SLC5A7 35 40 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne F7 15 49 COc1cc(C(=O)NCc2nnc(O)n2C2CC2)ccc1OCc1ccccc1 ZINC000880608507 GF On-Demand Anodyne ACKR3 41 35 O=C1CC[C@@H](c2ccc(C(=O)N3CCN(CC(F)(F)CO)CC3)cc2)N1 ZINC000880608515 FD On-Demand Anodyne L3MBTL3 41 33 O=C1CC[C@H](c2ccc(C(=O)N3CCN(CC(F)(F)CO)CC3)cc2)N1 ZINC000880608516 FD On-Demand Anodyne L3MBTL3 41 33 O=C(NCc1nnc(O)n1C1CC1)c1cc2c(F)cccc2s1 ZINC000880608559 EF On-Demand Anodyne F9 50 35 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne F2 47 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne PLG 41 38 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne ACE 100 39 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne OPRM1 53 42 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne OPRD1 46 39 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne GHRHR 59 32 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne P2RY12 87 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne MME 115 39 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne ANPEP 55 37 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne TACR1 21 42 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne MC4R 75 37 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne FCER2 69 34 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CTSB 46 38 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne TRY2_BOVIN 100 38 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne PAPA1_CARPA 54 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne TRY1_BOVIN 48 38 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CYSP_TRYCR 59 38 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CTSL 51 39 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne NPFFR2 72 35 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne TIMP3 72 33 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne MC3R 44 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CAPNS1 77 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne MMP3 18 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne HLA-DRB1 62 37 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CELA2A 48 32 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CAPN1 91 40 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CAPN2 61 37 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne ACE2 86 39 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne MC1R 48 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne ST14 83 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne FPR1 56 45 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne CTRB_BOVIN 48 35 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne GAG-PRO 49 34 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne BLA1_STEMA 56 37 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne BRCA1 58 30 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608624 ED On-Demand Anodyne NPFFR1 72 35 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne F2 47 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne PLG 41 38 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne ACE 100 39 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne OPRM1 53 42 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne OPRD1 46 39 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne GHRHR 59 32 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne P2RY12 87 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne MME 115 39 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne ANPEP 55 37 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne TACR1 21 42 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne MC4R 75 37 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne FCER2 69 34 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CTSB 46 38 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne TRY2_BOVIN 100 38 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne PAPA1_CARPA 54 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne TRY1_BOVIN 48 38 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CYSP_TRYCR 59 38 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CTSL 51 39 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne NPFFR2 72 35 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne TIMP3 72 33 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne MC3R 44 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CAPNS1 77 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne MMP3 18 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne HLA-DRB1 62 37 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CELA2A 48 32 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CAPN1 91 40 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CAPN2 61 37 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne ACE2 86 39 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne MC1R 48 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne ST14 83 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne FPR1 56 45 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne CTRB_BOVIN 48 35 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne GAG-PRO 49 34 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne BLA1_STEMA 56 37 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne BRCA1 58 30 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C ZINC000880608625 ED On-Demand Anodyne NPFFR1 72 35 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA2 96 44 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA1 82 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA7 72 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CCR5 16 44 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA5B 51 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA4 61 42 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA5A 54 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA14 47 39 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA12 64 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CA9 71 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne CYNT 29 40 CCN1[C@@H](C)CN(C(=O)Cc2ccc(S(N)(=O)=O)cc2)C[C@H]1C ZINC000880608636 EC On-Demand Anodyne NCE103 20 40 CCN1[C@@H](C)CN(C(=O)[C@@H](CC(C)C)NC(=O)OC)C[C@H]1C ZINC000880608661 DD On-Demand Anodyne CAPN1 16 42 CCN1[C@@H](C)CN(C(=O)[C@H](CC(C)C)NC(=O)OC)C[C@H]1C ZINC000880608662 DD On-Demand Anodyne CAPN1 16 42 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880608670 FE On-Demand Anodyne LIMK2 21 41 CCN1[C@@H](C)CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@H]1C ZINC000880608674 FD On-Demand Anodyne CA2 31 42 CCN1[C@@H](C)CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@H]1C ZINC000880608674 FD On-Demand Anodyne CA1 25 42 CCN1[C@@H](C)CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@H]1C ZINC000880608674 FD On-Demand Anodyne CA4 26 42 CCN1[C@@H](C)CN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@H]1C ZINC000880608674 FD On-Demand Anodyne CA9 16 41 CCN1[C@@H](C)CN(C(=O)c2ccnc(-n3ccnc3)c2)C[C@H]1C ZINC000880608683 DD On-Demand Anodyne NOS2 57 33 CCN1[C@@H](C)CN(C(=O)c2ccc3cc[nH]c3c2)C[C@H]1C ZINC000880608686 CF On-Demand Anodyne GHSR 16 58 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccnc(N(C)C)c2)C1 ZINC000880608708 DD On-Demand Anodyne EPHX2 43 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccnc(N(C)C)c2)C1 ZINC000880608709 DD On-Demand Anodyne EPHX2 43 45 COc1ccc(CC(=O)NCc2nnc(O)n2C2CC2)cc1F ZINC000880608718 DD On-Demand Anodyne TRPV1 17 40 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccnc(N(C)C)c2)C1 ZINC000880608733 FE On-Demand Anodyne EPHX2 32 41 CCN1[C@@H](C)CN(C(=O)COCc2ccc(OC)cc2)C[C@H]1C ZINC000880608805 DE On-Demand Anodyne UGCG 17 42 CCN1[C@@H](C)CN(C(=O)COCc2ccc(OC)cc2)C[C@H]1C ZINC000880608805 DE On-Demand Anodyne GBA2 23 42 CCN1[C@@H](C)CN(C(=O)[C@@H](C)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608824 DD On-Demand Anodyne CTSK 19 41 CCN1[C@@H](C)CN(C(=O)[C@H](C)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880608825 DD On-Demand Anodyne CTSK 19 41 CCN1[C@@H](C)CN(C(=O)COc2cccc(C#N)c2)C[C@H]1C ZINC000880608834 DD On-Demand Mild CPT1A 27 42 CCN1[C@@H](C)CN(C(=O)c2ccc(NC(=O)OC)cc2)C[C@H]1C ZINC000880608856 DE On-Demand Anodyne ACR 41 33 CCN1[C@@H](C)CN(C(=O)CN2CCN(c3ccccn3)CC2)C[C@H]1C ZINC000880608886 ED On-Demand Anodyne HTR1A 15 48 CCN1[C@@H](C)CN(C(=O)CN2CCN(c3ccccn3)CC2)C[C@H]1C ZINC000880608886 ED On-Demand Anodyne DRD2 15 48 CCN1[C@@H](C)CN(C(=O)CN2CCN(c3ccccn3)CC2)C[C@H]1C ZINC000880608886 ED On-Demand Anodyne DRD4 47 43 CCN1[C@@H](C)CN(C(=O)CN2CCN(c3ccccn3)CC2)C[C@H]1C ZINC000880608886 ED On-Demand Anodyne SLC27A1 33 42 CCN1[C@@H](C)CN(C(=O)c2ccccc2NS(C)(=O)=O)C[C@H]1C ZINC000880608902 ED On-Demand Anodyne PRTN3 45 32 CCN1[C@@H](C)CN(C(=O)CCn2ccnc2)C[C@H]1C ZINC000880608904 CD On-Demand Anodyne TBXAS1 37 41 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609031 FE On-Demand Anodyne PDGFRB 32 43 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609031 FE On-Demand Anodyne PDGFRA 40 38 CCN1[C@@H](C)CN(C(=O)CCCn2ccnc2)C[C@H]1C ZINC000880609038 CD On-Demand Anodyne TBXAS1 44 46 COc1ccc(N2CCC(NC(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609055 GF On-Demand Clean EPHX2 49 41 COc1ccc(N2CCC(NC(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609055 GF On-Demand Clean PDK1 46 33 COc1ccc(N2CCC(NC(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609055 GF On-Demand Clean MCHR1 26 43 CCN1[C@@H](C)CN(C(=O)Cn2nc(C)c(Cl)c2C)C[C@H]1C ZINC000880609057 DE On-Demand Anodyne CCR1 19 44 CCN1[C@@H](C)CN(C(=O)c2ccc(NC(N)=O)cc2)C[C@H]1C ZINC000880609070 DD On-Demand Anodyne ACR 46 33 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne ACE 28 41 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CELA1 18 40 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne KLK3 71 34 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CTSB 64 45 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne PAPA1_CARPA 52 38 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CYSP_TRYCR 53 40 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CTSK 44 45 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CTSL 47 41 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne PREP 23 53 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CAPNS1 63 37 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CAPN1 80 40 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne CAPN2 124 40 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne NPR 75 41 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne NAAA 53 37 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne SLC12A5 49 34 CCN1[C@@H](C)CN(C(=O)CNC(=O)OCc2ccccc2)C[C@H]1C ZINC000880609093 ED On-Demand Anodyne PDS 42 34 COc1ccc(N2CCCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609094 GF On-Demand Clean PDGFRB 55 40 COc1ccc(N2CCCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609094 GF On-Demand Clean EPHB4 44 35 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880609104 FG On-Demand Mild ROCK2 28 46 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880609104 FG On-Demand Mild PDS 43 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880609109 FG On-Demand Mild ROCK2 28 46 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880609109 FG On-Demand Mild PDS 43 36 CCN1[C@@H](C)CN(C(=O)c2ccc(N3CCOCC3)nc2)C[C@H]1C ZINC000880609118 ED On-Demand Anodyne HPGDS 15 45 C[C@H](O)c1ccc(CNC(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880609127 EF On-Demand Anodyne ROCK2 15 40 CN(Cc1ccc(Cl)nc1)C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609135 DF On-Demand Anodyne Q8WSF8_APLCA 20 43 CN(Cc1ccc(Cl)nc1)C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609135 DF On-Demand Anodyne NACHRBETA2 25 43 COc1ccc(O)c(CNC(=O)Nc2ccnc(N(C)C)c2)c1 ZINC000880609147 DE On-Demand Clean MTNR1A 23 41 CCOC(=O)N1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880609172 ED On-Demand Anodyne P2RY12 53 41 CCN1[C@@H](C)CN(C(=O)Cc2cccs2)C[C@H]1C ZINC000880609179 CE On-Demand Anodyne ETHR 24 46 CCOC(=O)Nc1ccc(C(=O)N2C[C@H](C)N(CC)[C@H](C)C2)cc1 ZINC000880609180 EF On-Demand Anodyne ACR 45 35 NC(=O)COc1cccc(NC(=O)c2ccccc2CSC2=NCCS2)c1 ZINC000880609185 HG On-Demand Anodyne KCNK3 49 35 NC(=O)COc1cccc(NC(=O)c2ccccc2CSC2=NCCS2)c1 ZINC000880609185 HG On-Demand Anodyne KCNK9 50 35 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc(OC)cc(OC)c2)C[C@H]1C ZINC000880609206 FD On-Demand Anodyne DRD4 41 31 CCN1[C@@H](C)CN(C(=O)Cn2cnc3c(N)ncnc32)C[C@H]1C ZINC000880609225 DC On-Demand Anodyne AHCY 86 45 CCN1[C@@H](C)CN(C(=O)Cn2cnc3c(N)ncnc32)C[C@H]1C ZINC000880609225 DC On-Demand Anodyne OXGR1 110 38 CCN1[C@@H](C)CN(C(=O)c2cnn3ccccc23)C[C@H]1C ZINC000880609226 CD On-Demand Anodyne EPHB3 27 41 CCN1CC[C@H](CNC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880609236 DD On-Demand Anodyne CCR3 47 38 CCN1CC[C@H](CNC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880609236 DD On-Demand Anodyne CACNA1I 49 33 CCN1[C@@H](C)CN(C(=O)c2c[nH]c3ccc([N+](=O)[O-])cc23)C[C@H]1C ZINC000880609240 EF On-Demand Bother GABRA1 15 48 CCN1[C@@H](C)CN(C(=O)c2c[nH]c3ccc([N+](=O)[O-])cc23)C[C@H]1C ZINC000880609240 EF On-Demand Bother GABRA2 15 45 CCN1[C@@H](C)CN(C(=O)c2cccc(CS(N)(=O)=O)c2)C[C@H]1C ZINC000880609259 ED On-Demand Anodyne TRY2_BOVIN 67 34 CCN1[C@@H](C)CN(C(=O)c2cccnc2Cl)C[C@H]1C ZINC000880609260 CE On-Demand Anodyne G2YM83_BOTF4 77 44 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2ccccn2)C[C@H]1C ZINC000880609263 DC On-Demand Anodyne GRM4 49 38 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)/C=C/c3ccccc3)CC2)C[C@H]1C ZINC000880609278 GF On-Demand Anodyne CCR2 17 40 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)/C=C\c3ccccc3)CC2)C[C@H]1C ZINC000880609279 GF On-Demand Anodyne CCR2 17 40 CCN1[C@@H](C)CN(C(=O)c2cccc(NS(C)(=O)=O)c2)C[C@H]1C ZINC000880609286 ED On-Demand Anodyne NR3C2 18 41 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880609287 ED On-Demand Anodyne EPHX2 35 40 COC(=O)N1CCC[C@H](NC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880609288 ED On-Demand Anodyne EPHX2 35 40 CCN1[C@@H](C)CN(C(=O)c2cc3cc(OC)c(OC)cc3[nH]2)C[C@H]1C ZINC000880609293 EF On-Demand Anodyne GRIN2B 17 43 CCN1[C@@H](C)CN(C(=O)c2cc3cc(OC)c(OC)cc3[nH]2)C[C@H]1C ZINC000880609293 EF On-Demand Anodyne HRH4 27 44 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)c3cccnc3)CC2)C[C@H]1C ZINC000880609295 FD On-Demand Anodyne SLC18A3 15 46 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)c3cccnc3)CC2)C[C@H]1C ZINC000880609295 FD On-Demand Anodyne SMO 34 40 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)c3cccnc3)CC2)C[C@H]1C ZINC000880609295 FD On-Demand Anodyne L3MBTL3 64 36 CCN1[C@@H](C)CN(C(=O)CCNS(=O)(=O)c2cccnc2)C[C@H]1C ZINC000880609296 FC On-Demand Anodyne TBXAS1 46 39 CCN1[C@@H](C)CN(C(=O)C[C@@H](NC(N)=O)c2ccccc2C)C[C@H]1C ZINC000880609304 EE On-Demand Anodyne CTSA 58 36 CCN1[C@@H](C)CN(C(=O)C[C@H](NC(N)=O)c2ccccc2C)C[C@H]1C ZINC000880609305 EE On-Demand Anodyne CTSA 58 36 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2ccc(C#N)cc2)C[C@H]1C ZINC000880609317 ED On-Demand Mild CTRB_BOVIN 49 38 C[C@@H]1CCOCCN1C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609405 CD On-Demand Anodyne EPHB4 46 30 C[C@H]1CCOCCN1C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609406 CD On-Demand Anodyne EPHB4 46 30 Cc1cccc2c1CCN(C(=O)Nc1ccnc(N(C)C)c1)C2 ZINC000880609416 DG On-Demand Anodyne P2RY14 55 39 C#CC(C)(C)NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880609417 BD On-Demand Mild TYK2 52 33 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(F)c1 ZINC000880609428 GF On-Demand Anodyne NPY2R 94 38 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(F)c1 ZINC000880609428 GF On-Demand Anodyne PRNP 16 41 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(F)c1 ZINC000880609428 GF On-Demand Anodyne SLC6A9 19 43 CCN1CC[C@H](CNC(=O)Nc2ccnc(N(C)C)c2)C1 ZINC000880609452 CD On-Demand Anodyne CCR3 62 41 CCN1CC[C@H](CNC(=O)Nc2ccnc(N(C)C)c2)C1 ZINC000880609452 CD On-Demand Anodyne CACNA1I 57 35 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne CCKAR 15 51 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne CYP51A1 23 44 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne PYGL 81 44 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne PLD1 18 45 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne PYGM 31 44 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne PLD2 18 42 CCN1[C@@H](C)CN(C(=O)CNC(=O)c2cc3ccccc3[nH]2)C[C@H]1C ZINC000880609467 ED On-Demand Anodyne AKR1C3 17 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne ACE 23 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne GHRHR 42 29 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne P2RY12 126 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne PTAFR 32 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne MC4R 36 45 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CTSB 17 40 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne TRY2_BOVIN 82 35 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CYSP_TRYCR 38 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CTSL 20 40 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CCR1 17 42 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CHRNA7 33 41 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne ACE2 59 34 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne CTRB_BOVIN 55 33 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne PSMB5 46 36 CCN1[C@@H](C)CN(C(=O)[C@@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609497 GE On-Demand Anodyne ACHP_LYMST 17 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne ACE 23 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne GHRHR 42 29 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne P2RY12 126 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne PTAFR 32 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne MC4R 36 45 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CTSB 17 40 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne TRY2_BOVIN 82 35 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CYSP_TRYCR 38 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CTSL 20 40 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CCR1 17 42 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CHRNA7 33 41 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne ACE2 59 34 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne CTRB_BOVIN 55 33 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne PSMB5 46 36 CCN1[C@@H](C)CN(C(=O)[C@H](Cc2cccnc2)NC(=O)c2ccccc2)C[C@H]1C ZINC000880609498 GE On-Demand Anodyne ACHP_LYMST 17 41 C[C@H](NC(=O)Nc1ccnc(N(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880609507 FF On-Demand Clean MAPKAPK5 41 35 C[C@H](NC(=O)Nc1ccnc(N(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880609507 FF On-Demand Clean MTOR 42 38 C[C@H](NC(=O)Nc1ccnc(N(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880609507 FF On-Demand Clean PIK3CB 41 37 C[C@H](NC(=O)Nc1ccnc(N(C)C)c1)c1ccc(N2CCOCC2)cc1 ZINC000880609507 FF On-Demand Clean EPHB4 88 38 CCN1[C@@H](C)CN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C[C@H]1C ZINC000880609521 GD On-Demand Bother SLC6A9 19 60 CCN1[C@@H](C)CN(C(=O)c2ccc(N3CCNC3=O)cc2)C[C@H]1C ZINC000880609526 ED On-Demand Anodyne L3MBTL3 40 35 CCN1[C@@H](C)CN(C(=O)c2cccc(-n3cnnn3)c2)C[C@H]1C ZINC000880609533 DD On-Demand Anodyne KCNJ1 45 34 CCN1[C@@H](C)CN(C(=O)c2ccccc2OCC(N)=O)C[C@H]1C ZINC000880609539 DD On-Demand Anodyne HCN1 42 31 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880609548 EE On-Demand Anodyne KCNK3 49 39 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880609548 EE On-Demand Anodyne KCNK9 42 39 CCOC(=O)N1CCCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880609566 ED On-Demand Anodyne P2RY12 40 40 CCN1[C@@H](C)CN(C(=O)Cc2csc(NC(=O)c3ccoc3C)n2)C[C@H]1C ZINC000880609569 GF On-Demand Anodyne CPT1A 26 40 CCN1[C@@H](C)CN(C(=O)Cc2csc(NC(=O)c3ccoc3C)n2)C[C@H]1C ZINC000880609569 GF On-Demand Anodyne CPT1B 36 40 CCN1[C@@H](C)CN(C(=O)CN2C(=O)CCc3ccccc32)C[C@H]1C ZINC000880609575 ED On-Demand Anodyne ACE 17 41 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609582 FF On-Demand Clean EPHB4 92 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccnc(N(C)C)c1 ZINC000880609582 FF On-Demand Clean STAT6 52 33 CCN1[C@@H](C)CN(C(=O)c2cc3ccccc3oc2=O)C[C@H]1C ZINC000880609652 DE On-Demand Anodyne MAOB 16 50 CCOC(=O)N1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880609661 DD On-Demand Anodyne P2RY12 54 43 CCOC(=O)N1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880609661 DD On-Demand Anodyne PDGFRB 42 41 C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880609697 EF On-Demand Anodyne CCR3 44 38 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1ccnc(N(C)C)c1 ZINC000880609698 EF On-Demand Anodyne CCR3 44 38 CCN1[C@@H](C)CN(C(=O)c2cc(=O)c3ccccc3o2)C[C@H]1C ZINC000880609707 DE On-Demand Anodyne TNKS 26 42 COc1ccc(CN(C)C(=O)Nc2ccnc(CN(C)C)c2)cc1F ZINC000880609720 EF On-Demand Anodyne MET 59 39 COc1ccc(CN(C)C(=O)Nc2ccnc(CN(C)C)c2)cc1F ZINC000880609720 EF On-Demand Anodyne PDGFRA 41 37 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)c(F)c1 ZINC000880609824 GF On-Demand Anodyne NPY2R 91 40 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)c(F)c1 ZINC000880609824 GF On-Demand Anodyne SLC6A9 17 43 COc1ccc(N2CCCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880609847 FF On-Demand Clean PDGFRB 55 42 COc1ccc(N2CCCN(C(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880609847 FF On-Demand Clean EPHB4 60 38 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609860 FF On-Demand Clean HTR1B 15 44 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609860 FF On-Demand Clean PDGFRB 59 42 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880609860 FF On-Demand Clean EPHB4 41 35 C=CCN1CCC(NC(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880609861 DD On-Demand Mild EPHX2 39 42 C=CCN1CCC(NC(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880609861 DD On-Demand Mild CXCR3 21 41 CCN(CCNC(=O)Nc1ccnc(N(C)C)c1)C(C)C ZINC000880609867 CD On-Demand Anodyne DOT1L 40 31 CCN1[C@@H](C)CN(C(=O)C2CCN(C(=O)OC(C)(C)C)CC2)C[C@H]1C ZINC000880609896 FF On-Demand Anodyne GPR119 41 39 CCN1[C@@H](C)CN(C(=O)c2cccc3oc(O)nc23)C[C@H]1C ZINC000880609917 DE On-Demand Anodyne HTR3A 23 40 CCN1[C@@H](C)CN(C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)C)C[C@H]1C ZINC000880609936 ED On-Demand Anodyne ELANE 24 44 CC[C@H](C#N)Oc1cc(CNC(=O)Nc2ccnc(CN(C)C)c2)ccc1OC ZINC000880609948 GG On-Demand Mild ROCK2 15 41 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609979 FG On-Demand Mild ROCK2 31 45 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609979 FG On-Demand Mild PDS 42 35 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609980 FG On-Demand Mild ROCK2 31 45 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609980 FG On-Demand Mild PDS 42 35 CCN1[C@@H](C)CN(C(=O)c2cnc3ccccn23)C[C@H]1C ZINC000880609984 CD On-Demand Anodyne EPHB3 19 43 COc1ccc(O)c(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609989 EE On-Demand Clean PDGFRB 31 41 COc1ccc(O)c(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609989 EE On-Demand Clean MTNR1A 22 40 COc1ccc(O)c(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880609989 EE On-Demand Clean MTNR1B 20 40 COc1ccc(N2CCC(NC(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880610031 FF On-Demand Clean EPHX2 48 40 COc1ccc(N2CCC(NC(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880610031 FF On-Demand Clean PDGFRA 27 42 COc1ccc(N2CCC(NC(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880610031 FF On-Demand Clean MCHR1 23 42 COc1ccc(N2CCC(NC(=O)Nc3ccnc(N(C)C)c3)CC2)cc1 ZINC000880610031 FF On-Demand Clean EPHB4 43 37 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880610054 FC On-Demand Anodyne ACOX1 51 35 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccnc(N(C)C)c2)CC1 ZINC000880610054 FC On-Demand Anodyne ABCB1 32 43 CCN1[C@@H](C)CN(C(=O)CCCCCCC(C)=O)C[C@H]1C ZINC000880610139 CF On-Demand Anodyne PAOX 40 38 Cc1cccc2c1CCN(C(=O)Nc1ccnc(CN(C)C)c1)C2 ZINC000880610163 DG On-Demand Anodyne P2RY14 56 39 COC(=O)NCc1ccc(NC(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880610189 FF On-Demand Anodyne ROCK2 19 41 CCN1[C@@H](C)CN(C(=O)c2cc(=O)c3ccc(F)cc3o2)C[C@H]1C ZINC000880610192 EE On-Demand Anodyne KCNH2 15 46 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880610211 FC On-Demand Anodyne ACOX1 50 34 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880610211 FC On-Demand Anodyne ABCB1 34 44 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne ACE 36 43 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne GHRHR 60 34 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne P2RY12 189 39 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CELA1 23 40 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTRA_BOVIN 63 37 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CASP3 15 42 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne BMP1 16 40 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne KLK3 83 38 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTSB 73 45 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne PAPA1_CARPA 78 40 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CYSP_TRYCR 62 43 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTSG 41 33 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTSK 62 49 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTSL 54 49 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne PREP 16 41 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne AMY2 43 30 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CAPNS1 70 41 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CELA2A 52 37 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne MMP11 63 33 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CTSS 35 49 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CAPN1 97 43 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CASP1 27 41 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne CAPN2 143 43 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne TGM2 33 47 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne TPSAB1 42 35 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne NPR 72 37 CCN1[C@@H](C)CN(C(=O)[C@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610248 GE On-Demand Anodyne PSMB5 44 41 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne ACE 36 43 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne GHRHR 60 34 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne P2RY12 189 39 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CELA1 23 40 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTRA_BOVIN 63 37 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CASP3 15 42 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne BMP1 16 40 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne KLK3 83 38 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTSB 73 45 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne PAPA1_CARPA 78 40 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CYSP_TRYCR 62 43 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTSG 41 33 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTSK 62 49 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTSL 54 49 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne PREP 16 41 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne AMY2 43 30 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CAPNS1 70 41 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CELA2A 52 37 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne MMP11 63 33 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CTSS 35 49 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CAPN1 97 43 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CASP1 27 41 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne CAPN2 143 43 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne TGM2 33 47 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne TPSAB1 42 35 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne NPR 72 37 CCN1[C@@H](C)CN(C(=O)[C@@H](CCOC)NC(=O)OCc2ccccc2)C[C@H]1C ZINC000880610249 GE On-Demand Anodyne PSMB5 44 41 CCN1[C@@H](C)CN(C(=O)[C@@H](CCC(=O)OC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610255 GD On-Demand Anodyne PAPA1_CARPA 33 40 CCN1[C@@H](C)CN(C(=O)[C@H](CCC(=O)OC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610256 GD On-Demand Anodyne PAPA1_CARPA 33 40 CCN1[C@@H](C)CN(C(=O)COCc2cccnc2)C[C@H]1C ZINC000880610272 CD On-Demand Anodyne CHRNA7 41 36 CCN1[C@@H](C)CN(C(=O)c2cc3occc3[nH]2)C[C@H]1C ZINC000880610306 CE On-Demand Anodyne HRH4 21 42 CCN1[C@@H](C)CN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C ZINC000880610310 ED On-Demand Anodyne PREP 34 42 CCN1[C@@H](C)CN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C ZINC000880610349 ED On-Demand Anodyne PREP 34 42 CCN1[C@@H](C)CN(C(=O)C(F)(F)c2ccccc2NC(C)=O)C[C@H]1C ZINC000880610350 FF On-Demand Anodyne RBP4 70 35 CCN(CCNC(=O)Nc1ccnc(CN(C)C)c1)C(C)C ZINC000880610357 DD On-Demand Anodyne DOT1L 40 30 CCN1[C@@H](C)CN(C(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610368 FE On-Demand Anodyne POLG_HCV1 27 48 CCN1[C@@H](C)CN(C(=O)[C@H](CC(F)F)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610369 FE On-Demand Anodyne POLG_HCV1 27 48 CCN1[C@@H](C)CN(C(=O)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)C[C@H]1C ZINC000880610391 FF On-Demand Anodyne GPR119 32 42 CCN1[C@@H](C)CN(C(=O)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)C[C@H]1C ZINC000880610392 FF On-Demand Anodyne GPR119 32 42 C[C@H]1CN(C(=O)Nc2ccnc(CN(C)C)c2)CCN1C(=O)OC(C)(C)C ZINC000880610402 GF On-Demand Anodyne GPR119 33 40 C[C@@H]1CN(C(=O)Nc2ccnc(CN(C)C)c2)CCN1C(=O)OC(C)(C)C ZINC000880610403 GF On-Demand Anodyne GPR119 33 40 CCN1[C@@H](C)CN(C(=O)[C@@H](COC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610431 ED On-Demand Anodyne PAPA1_CARPA 36 44 CCN1[C@@H](C)CN(C(=O)[C@@H](COC)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880610431 ED On-Demand Anodyne CTSK 17 42 Cc1ccc(N2CC[C@H](NC(=O)Nc3ccnc(CN(C)C)c3)C2=O)cc1 ZINC000880610452 FE On-Demand Anodyne CCKBR 46 33 CCN1[C@@H](C)CN(C(=O)c2cccc(Cl)c2O)C[C@H]1C ZINC000880610469 CF On-Demand Anodyne P2RX7 17 43 CC[C@@](C)(NC(=O)Nc1ccnc(CN(C)C)c1)c1ccccc1 ZINC000880610472 EH On-Demand Anodyne IMDH_CRYPV 50 36 C=CCN1CCC(NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880610510 DD On-Demand Mild EPHX2 38 43 CCN1[C@@H](C)CN(C(=O)Cc2cncn2Cc2ccccc2)C[C@H]1C ZINC000880610524 EE On-Demand Anodyne CYP11B1 17 47 CCN1[C@@H](C)CN(C(=O)C(=O)c2c[nH]c3cc(F)ccc23)C[C@H]1C ZINC000880610659 EE On-Demand Anodyne MPO 59 34 COC(=O)N(C)Cc1ccc(NC(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880610676 FF On-Demand Anodyne PDGFRA 40 34 CCN1[C@@H](C)CN(C(=O)c2ccccc2N2CCOCC2)C[C@H]1C ZINC000880610731 EE On-Demand Anodyne PIK3CB 19 41 CCN1[C@@H](C)CN(C(=O)c2csc(NC)n2)C[C@H]1C ZINC000880610793 CD On-Demand Anodyne TRPC6 63 43 CCN1[C@@H](C)CN(C(=O)c2csc(NC)n2)C[C@H]1C ZINC000880610793 CD On-Demand Anodyne TRPC3 57 43 CCN1[C@@H](C)CN(C(=O)c2nccc(C)n2)C[C@H]1C ZINC000880610847 CD On-Demand Anodyne SORD 41 35 CCN1[C@@H](C)CN(C(=O)c2coc(=O)c3ccccc23)C[C@H]1C ZINC000880610903 DE On-Demand Anodyne INHA 62 34 CCN1[C@@H](C)CN(C(=O)c2csc(Br)n2)C[C@H]1C ZINC000880610913 EE On-Demand Anodyne TRPC6 41 36 CCN1[C@@H](C)CN(C(=O)[C@@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880611119 FF On-Demand Mild PAPA1_CARPA 36 45 CCN1[C@@H](C)CN(C(=O)[C@@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880611119 FF On-Demand Mild CTSK 15 41 CCN1[C@@H](C)CN(C(=O)[C@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880611120 FF On-Demand Mild PAPA1_CARPA 36 45 CCN1[C@@H](C)CN(C(=O)[C@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C ZINC000880611120 FF On-Demand Mild CTSK 15 41 C[C@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccnc(CN(C)C)c1 ZINC000880611129 GF On-Demand Anodyne GPR119 39 42 C[C@@H]1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1ccnc(CN(C)C)c1 ZINC000880611130 GF On-Demand Anodyne GPR119 39 42 Cc1ccc2nc(C(=O)N3CCN(C)[C@H](C(C)(C)C)C3)cn2c1 ZINC000880611157 DE On-Demand Anodyne MAP3K5 35 40 Cc1ccc2nc(C(=O)N3CCN(C)[C@@H](C(C)(C)C)C3)cn2c1 ZINC000880611158 DE On-Demand Anodyne MAP3K5 35 40 CCN1[C@@H](C)CN(C(=O)c2c(C)cccc2O)C[C@H]1C ZINC000880611186 CE On-Demand Anodyne CCR5 25 43 CN1CCN(C(=O)c2coc(=O)c3ccccc23)C[C@H]1C(C)(C)C ZINC000880611268 EF On-Demand Anodyne INHA 43 33 CN1CCN(C(=O)c2coc(=O)c3ccccc23)C[C@@H]1C(C)(C)C ZINC000880611269 EF On-Demand Anodyne INHA 43 33 CN1CCN(C(=O)[C@@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C(C)(C)C ZINC000880611273 GF On-Demand Mild PAPA1_CARPA 32 44 CN1CCN(C(=O)[C@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@H]1C(C)(C)C ZINC000880611274 GF On-Demand Mild PAPA1_CARPA 32 44 CN1CCN(C(=O)[C@@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@@H]1C(C)(C)C ZINC000880611275 GF On-Demand Mild PAPA1_CARPA 32 44 CN1CCN(C(=O)[C@H](CCCC#N)NC(=O)OC(C)(C)C)C[C@@H]1C(C)(C)C ZINC000880611276 GF On-Demand Mild PAPA1_CARPA 32 44 C#CC(C)(C)NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880611369 CD On-Demand Mild TYK2 43 31 CCN1[C@@H](C)CN(C(=O)[C@@H]2CCc3nc[nH]c3C2)C[C@H]1C ZINC000880611417 CD On-Demand Anodyne HTR3A 15 47 CCN1[C@@H](C)CN(C(=O)[C@H]2CCc3nc[nH]c3C2)C[C@H]1C ZINC000880611425 CD On-Demand Anodyne HTR3A 15 47 CN1CCN(C(=O)[C@@H](O)c2cccnc2)C[C@H]1C(C)(C)C ZINC000880611467 CD On-Demand Anodyne PTAFR 15 42 CN1CCN(C(=O)[C@@H](O)c2cccnc2)C[C@@H]1C(C)(C)C ZINC000880611468 CD On-Demand Anodyne PTAFR 15 42 CN1CCN(C(=O)[C@H](O)c2cccnc2)C[C@H]1C(C)(C)C ZINC000880611469 CD On-Demand Anodyne PTAFR 15 42 CN1CCN(C(=O)[C@H](O)c2cccnc2)C[C@@H]1C(C)(C)C ZINC000880611470 CD On-Demand Anodyne PTAFR 15 42 CCN1[C@@H](C)CN(C(=O)c2cc3c([nH]2)CCCC3)C[C@H]1C ZINC000880611479 CE On-Demand Anodyne HRH4 18 59 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611528 IE On-Demand Anodyne ENPP1 48 30 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611528 IE On-Demand Anodyne KCNK3 55 42 COc1cc(NC(=O)[C@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611528 IE On-Demand Anodyne KCNK9 51 42 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611529 IE On-Demand Anodyne ENPP1 48 30 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611529 IE On-Demand Anodyne KCNK3 55 42 COc1cc(NC(=O)[C@@H]2C[C@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611529 IE On-Demand Anodyne KCNK9 51 42 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611530 IE On-Demand Anodyne ENPP1 48 30 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611530 IE On-Demand Anodyne KCNK3 55 42 COc1cc(NC(=O)[C@@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611530 IE On-Demand Anodyne KCNK9 51 42 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611531 IE On-Demand Anodyne ENPP1 48 30 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611531 IE On-Demand Anodyne KCNK3 55 42 COc1cc(NC(=O)[C@H]2C[C@@H]2C)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880611531 IE On-Demand Anodyne KCNK9 51 42 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1F ZINC000880611577 GF On-Demand Clean PDGFRB 60 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1F ZINC000880611577 GF On-Demand Clean CCR1 20 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1F ZINC000880611577 GF On-Demand Clean MET 64 39 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1F ZINC000880611577 GF On-Demand Clean RBP4 17 40 CCN1[C@@H](C)CN(C(=O)c2ccc(N=S(C)(C)=O)cc2)C[C@H]1C ZINC000880611582 EF On-Demand Anodyne L3MBTL3 40 35 CCN1[C@@H](C)CN(C(=O)c2ccc(C(N)=S)cc2)C[C@H]1C ZINC000880611614 DD On-Demand Anodyne L3MBTL3 43 35 CNc1nc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)cs1 ZINC000880611769 CD On-Demand Anodyne TRPC6 61 41 CNc1nc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)cs1 ZINC000880611769 CD On-Demand Anodyne TRPC3 54 41 CNc1nc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)cs1 ZINC000880611770 CD On-Demand Anodyne TRPC6 61 41 CNc1nc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)cs1 ZINC000880611770 CD On-Demand Anodyne TRPC3 54 41 CN1CCN(C(=O)c2cnc3ccccn23)C[C@H]1C(C)(C)C ZINC000880611778 DE On-Demand Anodyne EPHB3 20 42 CN1CCN(C(=O)c2cnc3ccccn23)C[C@@H]1C(C)(C)C ZINC000880611779 DE On-Demand Anodyne EPHB3 20 42 CN1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C(C)(C)C ZINC000880611810 ED On-Demand Anodyne PREP 31 44 CN1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C(C)(C)C ZINC000880611810 ED On-Demand Anodyne WNT3 45 36 CN1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C[C@@H]1C(C)(C)C ZINC000880611811 ED On-Demand Anodyne PREP 31 44 CN1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C[C@@H]1C(C)(C)C ZINC000880611811 ED On-Demand Anodyne WNT3 45 36 CN1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C(C)(C)C ZINC000880611812 ED On-Demand Anodyne PREP 31 44 CN1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C[C@H]1C(C)(C)C ZINC000880611812 ED On-Demand Anodyne WNT3 45 36 CN1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C[C@@H]1C(C)(C)C ZINC000880611813 ED On-Demand Anodyne PREP 31 44 CN1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C[C@@H]1C(C)(C)C ZINC000880611813 ED On-Demand Anodyne WNT3 45 36 COC(=O)Nc1cccc(CNC(=O)Nc2ccnc(CN(C)C)c2)c1 ZINC000880611932 FF On-Demand Anodyne ROCK2 36 48 CN1CCN(C(=O)c2ccccc2NS(C)(=O)=O)C[C@H]1C(C)(C)C ZINC000880611946 FD On-Demand Anodyne PRTN3 45 32 CN1CCN(C(=O)c2ccccc2NS(C)(=O)=O)C[C@H]1C(C)(C)C ZINC000880611946 FD On-Demand Anodyne CCR8 47 32 CN1CCN(C(=O)c2ccccc2NS(C)(=O)=O)C[C@@H]1C(C)(C)C ZINC000880611947 FD On-Demand Anodyne PRTN3 45 32 CN1CCN(C(=O)c2ccccc2NS(C)(=O)=O)C[C@@H]1C(C)(C)C ZINC000880611947 FD On-Demand Anodyne CCR8 47 32 COC[C@@H](O)CNC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880611962 CC On-Demand Anodyne ADRB1 41 32 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@@H]1C(C)(C)C ZINC000880611974 EC On-Demand Anodyne AHCY 83 45 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@@H]1C(C)(C)C ZINC000880611974 EC On-Demand Anodyne OXGR1 109 36 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@@H]1C(C)(C)C ZINC000880611974 EC On-Demand Anodyne DOT1L 53 35 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@H]1C(C)(C)C ZINC000880611975 EC On-Demand Anodyne AHCY 83 45 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@H]1C(C)(C)C ZINC000880611975 EC On-Demand Anodyne OXGR1 109 36 CN1CCN(C(=O)Cn2cnc3c(N)ncnc32)C[C@H]1C(C)(C)C ZINC000880611975 EC On-Demand Anodyne DOT1L 53 35 Cc1ccccc1[C@@H](O)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880611988 GG On-Demand Anodyne P2RY14 43 32 Cc1ccccc1[C@H](O)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880611989 GG On-Demand Anodyne P2RY14 43 32 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880612019 GF On-Demand Anodyne P2RY12 42 33 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880612020 GF On-Demand Anodyne P2RY12 42 33 CN1CCN(C(=O)Cn2cc([N+](=O)[O-])ccc2=O)C[C@@H]1C(C)(C)C ZINC000880612108 EC On-Demand Bother SSTR1 41 36 CN1CCN(C(=O)Cn2cc([N+](=O)[O-])ccc2=O)C[C@H]1C(C)(C)C ZINC000880612109 EC On-Demand Bother SSTR1 41 36 CN1CCN(C(=O)c2cccc(CS(N)(=O)=O)c2)C[C@H]1C(C)(C)C ZINC000880612128 FD On-Demand Anodyne TRY2_BOVIN 92 36 CN1CCN(C(=O)c2cccc(CS(N)(=O)=O)c2)C[C@H]1C(C)(C)C ZINC000880612128 FD On-Demand Anodyne ST14 73 34 CN1CCN(C(=O)c2cccc(CS(N)(=O)=O)c2)C[C@@H]1C(C)(C)C ZINC000880612129 FD On-Demand Anodyne TRY2_BOVIN 92 36 CN1CCN(C(=O)c2cccc(CS(N)(=O)=O)c2)C[C@@H]1C(C)(C)C ZINC000880612129 FD On-Demand Anodyne ST14 73 34 CN1CCN(C(=O)c2ccccc2OCC(N)=O)C[C@H]1C(C)(C)C ZINC000880612143 ED On-Demand Anodyne HCN1 42 31 CN1CCN(C(=O)c2ccccc2OCC(N)=O)C[C@@H]1C(C)(C)C ZINC000880612144 ED On-Demand Anodyne HCN1 42 31 COc1cccc(C(C)(C)C(=O)NCc2cc3n(n2)CCCC3)c1 ZINC000880612254 EF On-Demand Anodyne DRD4 44 34 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880612260 GF On-Demand Mild REN 47 36 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880612261 GF On-Demand Mild REN 47 36 CC(=O)N(C)c1ccc(CNC(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880612278 FE On-Demand Anodyne ROCK2 15 40 O=C(NCc1cc2n(n1)CCCC2)c1cnn2c(-c3cccnc3)ccnc12 ZINC000880612285 FE On-Demand Anodyne BRAF 16 40 N#CCSc1ccccc1C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000880612290 EE On-Demand Mild KCNK3 65 39 N#CCSc1ccccc1C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000880612290 EE On-Demand Mild KCNK9 57 39 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612313 FF On-Demand Anodyne CAPNS1 47 35 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612313 FF On-Demand Anodyne CAPN1 41 36 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612313 FF On-Demand Anodyne CAPN2 47 35 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612313 FF On-Demand Anodyne NPR 50 32 CN1CCN(C(=O)c2ccccc2N2CCOCC2)C[C@@H]1C(C)(C)C ZINC000880612336 EE On-Demand Anodyne AKR1C3 15 43 CN1CCN(C(=O)c2ccccc2N2CCOCC2)C[C@H]1C(C)(C)C ZINC000880612337 EE On-Demand Anodyne AKR1C3 15 43 C[C@H]1CN(C(=O)OC(C)(C)C)CC[C@H]1NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612357 GF On-Demand Anodyne GPR119 40 40 C[C@H]1CN(C(=O)OC(C)(C)C)CC[C@@H]1NC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880612358 GF On-Demand Anodyne GPR119 40 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880612391 ED On-Demand Anodyne EPHX2 40 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880612392 ED On-Demand Anodyne EPHX2 40 45 O=C(Cc1ccc(F)cn1)NCc1cc2n(n1)CCCC2 ZINC000880612501 CD On-Demand Anodyne SLC27A1 42 34 O=C(NCc1cc2n(n1)CCCC2)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880612595 FG On-Demand Anodyne C3AR1 43 42 O=C(NCc1cc2n(n1)CCCC2)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880612596 FG On-Demand Anodyne C3AR1 43 42 CN1CCN(C(=O)[C@@H]2CCc3nc[nH]c3C2)C[C@H]1C(C)(C)C ZINC000880612688 DD On-Demand Anodyne HTR3A 15 47 CN1CCN(C(=O)[C@@H]2CCc3nc[nH]c3C2)C[C@@H]1C(C)(C)C ZINC000880612689 DD On-Demand Anodyne HTR3A 15 47 CN1CCN(C(=O)[C@H]2CCc3nc[nH]c3C2)C[C@@H]1C(C)(C)C ZINC000880612690 DD On-Demand Anodyne HTR3A 15 47 CN1CCN(C(=O)[C@H]2CCc3nc[nH]c3C2)C[C@H]1C(C)(C)C ZINC000880612691 DD On-Demand Anodyne HTR3A 15 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880612762 FD On-Demand Anodyne CACNA1B 15 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880612764 FD On-Demand Anodyne CACNA1B 15 43 O=C(Cc1cccc2ncccc12)NCc1cc2n(n1)CCCC2 ZINC000880612770 DF On-Demand Anodyne HNMT 40 34 CN1CCN(C(=O)Cc2ccccc2[N+](=O)[O-])C[C@H]1C(C)(C)C ZINC000880612822 DE On-Demand Bother COLA 107 35 CN1CCN(C(=O)Cc2ccccc2[N+](=O)[O-])C[C@@H]1C(C)(C)C ZINC000880612823 DE On-Demand Bother COLA 107 35 O=C(OCc1ccccc1)N1CC(O)(C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880612824 GD On-Demand Anodyne SLC12A5 59 34 CN1CCN(C(=O)c2cc(S(C)(=O)=O)ccc2Cl)C[C@H]1C(C)(C)C ZINC000880612868 FF On-Demand Anodyne CACNA1B 43 35 CN1CCN(C(=O)c2cc(S(C)(=O)=O)ccc2Cl)C[C@H]1C(C)(C)C ZINC000880612868 FF On-Demand Anodyne SLC6A9 41 42 CN1CCN(C(=O)c2cc(S(C)(=O)=O)ccc2Cl)C[C@@H]1C(C)(C)C ZINC000880612870 FF On-Demand Anodyne CACNA1B 43 35 CN1CCN(C(=O)c2cc(S(C)(=O)=O)ccc2Cl)C[C@@H]1C(C)(C)C ZINC000880612870 FF On-Demand Anodyne SLC6A9 41 42 CN1CCN(C(=O)c2ccccc2-n2cnnn2)C[C@H]1C(C)(C)C ZINC000880612899 ED On-Demand Anodyne KCNJ1 54 33 CN1CCN(C(=O)c2ccccc2-n2cnnn2)C[C@@H]1C(C)(C)C ZINC000880612900 ED On-Demand Anodyne KCNJ1 54 33 O=C(NCc1cc2n(n1)CCCC2)c1cc2c(Cl)nccc2o1 ZINC000880612907 EF On-Demand Anodyne NAMPT 25 41 CN1CCN(C(=O)c2cccc3oc(O)nc23)C[C@@H]1C(C)(C)C ZINC000880612945 DE On-Demand Anodyne HTR3A 24 43 CN1CCN(C(=O)c2cccc3oc(O)nc23)C[C@H]1C(C)(C)C ZINC000880612946 DE On-Demand Anodyne HTR3A 24 43 CCC(=O)N1CSC[C@@H]1C(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880613002 ED On-Demand Anodyne PREP 18 41 CCC(=O)N1CSC[C@@H]1C(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880613003 ED On-Demand Anodyne PREP 18 41 CCC(=O)N1CSC[C@H]1C(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880613004 ED On-Demand Anodyne PREP 18 41 CCC(=O)N1CSC[C@H]1C(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880613005 ED On-Demand Anodyne PREP 18 41 COc1ccc(N2CC[C@H](NC(=O)Nc3ccnc(CN(C)C)c3)C2)cc1 ZINC000880613043 FF On-Demand Clean MCHR1 22 45 COC(=O)c1cc(C(=O)NCc2cc3n(n2)CCCC3)ccc1C ZINC000880613098 EE On-Demand Anodyne DRD4 40 31 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)N1Cc1ccccc1 ZINC000880613151 GD On-Demand Anodyne F2 40 37 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)N1Cc1ccccc1 ZINC000880613151 GD On-Demand Anodyne TMPRSS11D 59 35 CN1CCN(C(=O)c2ccc(NC(N)=O)cc2)C[C@H]1C(C)(C)C ZINC000880613184 DD On-Demand Anodyne ACR 48 35 CN1CCN(C(=O)c2ccc(NC(N)=O)cc2)C[C@@H]1C(C)(C)C ZINC000880613186 DD On-Demand Anodyne ACR 48 35 COC(=O)Nc1ccc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)cc1 ZINC000880613188 EF On-Demand Anodyne EPHX2 15 43 COC(=O)Nc1ccc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)cc1 ZINC000880613190 EF On-Demand Anodyne EPHX2 15 43 O=C(Cc1ccc2cccnc2c1)NCc1cc2n(n1)CCCC2 ZINC000880613207 DF On-Demand Anodyne SUCNR1 49 35 O=C(Cc1csc(COc2ccccc2)n1)NCc1cc2n(n1)CCCC2 ZINC000880613209 GG On-Demand Anodyne ADAM17 44 35 CC(=O)Nc1ccccc1C(F)(F)C(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880613250 FF On-Demand Anodyne RBP4 66 36 CC(=O)Nc1ccccc1C(F)(F)C(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880613251 FF On-Demand Anodyne RBP4 66 36 CN1CCN(C(=O)c2cccc(CS(C)(=O)=O)c2)C[C@H]1C(C)(C)C ZINC000880613444 FE On-Demand Anodyne TRY2_BOVIN 83 36 CN1CCN(C(=O)c2cccc(CS(C)(=O)=O)c2)C[C@@H]1C(C)(C)C ZINC000880613446 FE On-Demand Anodyne TRY2_BOVIN 83 36 CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880613556 GE On-Demand Anodyne GPR119 31 43 CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880613558 GE On-Demand Anodyne GPR119 31 43 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880613560 GE On-Demand Anodyne GPR119 31 43 CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880613562 GE On-Demand Anodyne GPR119 31 43 CCOC(=O)Nc1ccc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)cc1 ZINC000880613597 EG On-Demand Anodyne EPHX2 15 40 CCOC(=O)Nc1ccc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)cc1 ZINC000880613597 EG On-Demand Anodyne ACR 44 34 CCOC(=O)Nc1ccc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)cc1 ZINC000880613599 EG On-Demand Anodyne EPHX2 15 40 CCOC(=O)Nc1ccc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)cc1 ZINC000880613599 EG On-Demand Anodyne ACR 44 34 O=C(Cc1ccc2cnccc2c1)NCc1cc2n(n1)CCCC2 ZINC000880613634 DF On-Demand Anodyne NAMPT 50 42 C[C@@H](Oc1cccc(Cl)c1)C(=O)NNC(=O)Nc1ccnc(CN(C)C)c1 ZINC000880613650 GE On-Demand Reactive IMDH_CRYPV 26 43 O=C(NCc1cc2n(n1)CCCC2)c1cccc(Oc2ccccn2)c1 ZINC000880613667 EG On-Demand Anodyne DRD4 44 36 CN1CCN(C(=O)c2cc(=O)c3ccccc3o2)C[C@H]1C(C)(C)C ZINC000880613680 EF On-Demand Anodyne TNKS 27 47 CN1CCN(C(=O)c2cc(=O)c3ccccc3o2)C[C@@H]1C(C)(C)C ZINC000880613681 EF On-Demand Anodyne TNKS 27 47 O=C(NCc1cc2n(n1)CCCC2)c1ccc(C(F)(F)Br)nc1 ZINC000880613685 GF On-Demand Anodyne NAMPT 32 40 O=C(NCc1cc2n(n1)CCCC2)c1cnc2nccn2c1 ZINC000880613744 CD On-Demand Anodyne NAMPT 19 58 O=C(NCc1cc2n(n1)CCCC2)C1(c2ccnc3ccccc23)CC1 ZINC000880613758 EG On-Demand Anodyne HNMT 47 35 CN1CCN(C(=O)c2cc(=O)c3ccc(F)cc3o2)C[C@H]1C(C)(C)C ZINC000880613763 EF On-Demand Anodyne KCNH2 16 46 CN1CCN(C(=O)c2cc(=O)c3ccc(F)cc3o2)C[C@@H]1C(C)(C)C ZINC000880613765 EF On-Demand Anodyne KCNH2 16 46 CC(=O)CCCCCCC(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880613821 DG On-Demand Anodyne PAOX 25 41 CC(=O)CCCCCCC(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880613823 DG On-Demand Anodyne PAOX 25 41 CN1CCN(C(=O)Cc2cccs2)C[C@@H]1C(C)(C)C ZINC000880613844 CE On-Demand Anodyne ETHR 33 43 CN1CCN(C(=O)Cc2cccs2)C[C@H]1C(C)(C)C ZINC000880613845 CE On-Demand Anodyne ETHR 33 43 C[C@H]1CC(=O)N[C@@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880613853 CC On-Demand Anodyne TRHR 50 34 O=C(NNc1ccccc1C(F)(F)F)c1ccc(C(=O)O)nc1 ZINC000880613863 EF On-Demand Reactive RBP4 55 35 CN1CCN(C(=O)c2ccc(C#N)o2)C[C@@H]1C(C)(C)C ZINC000880613940 CD On-Demand Mild CSF1R 22 40 CN1CCN(C(=O)c2ccc(C#N)o2)C[C@H]1C(C)(C)C ZINC000880613941 CD On-Demand Mild CSF1R 22 40 C#CCN1CCC[C@H]1C(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880613987 CD On-Demand Mild PREP 19 40 O=C(NCc1cc2n(n1)CCCC2)c1cnc2cc[nH]c2c1 ZINC000880613990 CE On-Demand Anodyne NAMPT 26 41 C#CCN1CCC[C@H]1C(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880613992 CD On-Demand Mild PREP 19 40 CN1CCN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@H]1C(C)(C)C ZINC000880614038 FD On-Demand Anodyne CA2 21 40 CN1CCN(C(=O)c2cc(S(N)(=O)=O)ccc2Cl)C[C@@H]1C(C)(C)C ZINC000880614039 FD On-Demand Anodyne CA2 21 40 COc1cccc(OC)c1C(=O)N1CCN(C)[C@H](C(C)(C)C)C1 ZINC000880614040 DF On-Demand Anodyne SSTR1 64 38 COc1cccc(OC)c1C(=O)N1CCN(C)[C@@H](C(C)(C)C)C1 ZINC000880614041 DF On-Demand Anodyne SSTR1 64 38 CN(C)C(=O)Nc1cccc(C(=O)N2CCN(C)[C@H](C(C)(C)C)C2)c1 ZINC000880614043 EF On-Demand Anodyne KCNK3 55 34 CN(C)C(=O)Nc1cccc(C(=O)N2CCN(C)[C@@H](C(C)(C)C)C2)c1 ZINC000880614044 EF On-Demand Anodyne KCNK3 55 34 CN1CCN(C(=O)c2ccc3cc[nH]c3c2)C[C@H]1C(C)(C)C ZINC000880614062 CF On-Demand Anodyne GHSR 15 55 CN1CCN(C(=O)c2ccc3cc[nH]c3c2)C[C@@H]1C(C)(C)C ZINC000880614063 CF On-Demand Anodyne GHSR 15 55 CN1CCN(C(=O)c2cccc(-n3cnnn3)c2)C[C@H]1C(C)(C)C ZINC000880614096 ED On-Demand Anodyne KCNJ1 53 38 CN1CCN(C(=O)c2cccc(-n3cnnn3)c2)C[C@@H]1C(C)(C)C ZINC000880614097 ED On-Demand Anodyne KCNJ1 53 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne F2 57 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne PLG 53 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne ACE 78 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne OPRM1 52 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne OPRD1 44 39 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne GHRHR 81 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne P2RY12 191 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MME 100 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne ANPEP 54 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne TACR1 25 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne UGCG 38 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MC4R 101 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CMA1 41 39 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CTRA_BOVIN 44 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne FCER2 46 33 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CTSB 42 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne TRY2_BOVIN 107 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne PAPA1_CARPA 44 37 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne TRY1_BOVIN 53 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CYSP_TRYCR 68 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CTSL 59 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne NPFFR2 76 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CYP51A1 22 44 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MC3R 43 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MC5R 59 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CAPNS1 74 32 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MMP3 23 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne HLA-DRB1 52 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CELA2A 51 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne PLAT 15 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne GHSR 34 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CAPN1 73 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CAPN2 42 35 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne ACE2 72 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne MC1R 42 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CTSV 40 30 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne ST14 109 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne FPR1 61 43 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne CTRB_BOVIN 50 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne GAG-PRO 40 31 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne BLA1_STEMA 69 42 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne QRFPR 42 33 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne BRCA1 44 31 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614188 ED On-Demand Anodyne NPFFR1 75 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne F2 57 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne PLG 53 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne ACE 78 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne OPRM1 52 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne OPRD1 44 39 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne GHRHR 81 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne P2RY12 191 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MME 100 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne ANPEP 54 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne TACR1 25 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne UGCG 38 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MC4R 101 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CMA1 41 39 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CTRA_BOVIN 44 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne FCER2 46 33 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CTSB 42 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne TRY2_BOVIN 107 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne PAPA1_CARPA 44 37 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne TRY1_BOVIN 53 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CYSP_TRYCR 68 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CTSL 59 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne NPFFR2 76 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CYP51A1 22 44 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MC3R 43 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MC5R 59 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CAPNS1 74 32 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MMP3 23 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne HLA-DRB1 52 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CELA2A 51 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne PLAT 15 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne GHSR 34 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CAPN1 73 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CAPN2 42 35 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne ACE2 72 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne MC1R 42 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CTSV 40 30 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne ST14 109 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne FPR1 61 43 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne CTRB_BOVIN 50 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne GAG-PRO 40 31 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne BLA1_STEMA 69 42 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne QRFPR 42 33 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne BRCA1 44 31 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@H]1C(C)(C)C ZINC000880614189 ED On-Demand Anodyne NPFFR1 75 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne F2 57 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne PLG 53 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne ACE 78 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne OPRM1 52 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne OPRD1 44 39 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne GHRHR 81 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne P2RY12 191 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MME 100 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne ANPEP 54 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne TACR1 25 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne UGCG 38 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MC4R 101 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CMA1 41 39 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CTRA_BOVIN 44 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne FCER2 46 33 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CTSB 42 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne TRY2_BOVIN 107 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne PAPA1_CARPA 44 37 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne TRY1_BOVIN 53 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CYSP_TRYCR 68 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CTSL 59 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne NPFFR2 76 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CYP51A1 22 44 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MC3R 43 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MC5R 59 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CAPNS1 74 32 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MMP3 23 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne HLA-DRB1 52 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CELA2A 51 34 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne PLAT 15 40 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne GHSR 34 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CAPN1 73 41 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CAPN2 42 35 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne ACE2 72 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne MC1R 42 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CTSV 40 30 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne ST14 109 38 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne FPR1 61 43 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne CTRB_BOVIN 50 36 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne GAG-PRO 40 31 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne BLA1_STEMA 69 42 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne QRFPR 42 33 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne BRCA1 44 31 CN1CCN(C(=O)[C@@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614190 ED On-Demand Anodyne NPFFR1 75 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne F2 57 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne PLG 53 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne ACE 78 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne OPRM1 52 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne OPRD1 44 39 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne GHRHR 81 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne P2RY12 191 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MME 100 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne ANPEP 54 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne TACR1 25 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne UGCG 38 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MC4R 101 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CMA1 41 39 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CTRA_BOVIN 44 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne FCER2 46 33 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CTSB 42 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne TRY2_BOVIN 107 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne PAPA1_CARPA 44 37 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne TRY1_BOVIN 53 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CYSP_TRYCR 68 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CTSL 59 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne NPFFR2 76 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CYP51A1 22 44 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MC3R 43 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MC5R 59 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CAPNS1 74 32 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MMP3 23 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne HLA-DRB1 52 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CELA2A 51 34 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne PLAT 15 40 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne GHSR 34 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CAPN1 73 41 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CAPN2 42 35 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne ACE2 72 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne MC1R 42 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CTSV 40 30 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne ST14 109 38 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne FPR1 61 43 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne CTRB_BOVIN 50 36 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne GAG-PRO 40 31 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne BLA1_STEMA 69 42 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne QRFPR 42 33 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne BRCA1 44 31 CN1CCN(C(=O)[C@H](Cc2ccccc2)NC(N)=O)C[C@@H]1C(C)(C)C ZINC000880614191 ED On-Demand Anodyne NPFFR1 75 38 CN1CCN(C(=O)[C@H]2CCCN2C)C[C@@H]1C(C)(C)C ZINC000880614194 CD On-Demand Anodyne PREP 22 41 COC(=O)c1ccc(OC)c2c1CCN(C(=O)Nc1ccnc(CN(C)C)c1)C2 ZINC000880614233 GF On-Demand Anodyne P2RY14 47 33 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccnc(CN(C)C)c1)CC2 ZINC000880614302 FF On-Demand Anodyne P2RY14 50 35 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean HTR1A 25 48 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean ADRA1D 20 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean HTR1D 17 48 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean HTR1B 20 48 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean ADRA1A 18 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean PDGFRB 85 51 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean HTR7 19 43 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean LCK 20 40 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean KDR 41 38 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean PDGFRA 42 43 COc1ccc(N2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c(OC)c1 ZINC000880614314 GF On-Demand Clean FLT3 16 43 C[C@H]1c2sccc2CCN1C(=O)Nc1ccnc(CN(C)C)c1 ZINC000880614324 EG On-Demand Anodyne TRPM8 17 42 CN1CCN(C(=O)c2cccnc2Cl)C[C@@H]1C(C)(C)C ZINC000880614344 CF On-Demand Anodyne G2YM83_BOTF4 73 39 CN1CCN(C(=O)c2cccnc2Cl)C[C@H]1C(C)(C)C ZINC000880614345 CF On-Demand Anodyne G2YM83_BOTF4 73 39 CN1CCN(C(=O)c2cnn3ccccc23)C[C@H]1C(C)(C)C ZINC000880614394 DE On-Demand Anodyne EPHB3 32 41 CN1CCN(C(=O)c2cnn3ccccc23)C[C@@H]1C(C)(C)C ZINC000880614395 DE On-Demand Anodyne EPHB3 32 41 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)cc1 ZINC000880614402 GG On-Demand Anodyne PDGFRB 42 37 COc1cc(C(=O)NCc2cc3n(n2)CCCC3)ccc1C#N ZINC000880614452 DE On-Demand Mild DRD4 41 32 Cc1ccc(CN2CCO[C@H](CNC(=O)Nc3ccnc(CN(C)C)c3)C2)cc1 ZINC000880614465 GE On-Demand Anodyne CCR3 15 47 O=C(NCc1cc2n(n1)CCCC2)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880614468 GE On-Demand Anodyne CCR2 41 35 O=C(NCc1cc2n(n1)CCCC2)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880614468 GE On-Demand Anodyne AKR1C3 46 36 O=C(NCc1cc2n(n1)CCCC2)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880614468 GE On-Demand Anodyne SFRP1 60 34 O=C(NCc1cc2n(n1)CCCC2)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880614468 GE On-Demand Anodyne NAMPT 40 40 CN1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C[C@H]1C(C)(C)C ZINC000880614538 ED On-Demand Anodyne HPGDS 18 45 CN1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C[C@@H]1C(C)(C)C ZINC000880614539 ED On-Demand Anodyne HPGDS 18 45 CN1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCC3)o2)C[C@H]1C(C)(C)C ZINC000880614578 GD On-Demand Anodyne LPL 43 34 CN1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCC3)o2)C[C@@H]1C(C)(C)C ZINC000880614579 GD On-Demand Anodyne LPL 43 34 CN1CCN(C(=O)c2ccnc(-n3ccnc3)c2)C[C@H]1C(C)(C)C ZINC000880614616 EE On-Demand Anodyne NOS2 42 35 CN1CCN(C(=O)c2ccnc(-n3ccnc3)c2)C[C@@H]1C(C)(C)C ZINC000880614617 EE On-Demand Anodyne NOS2 42 35 O=C(Cc1cc2cc(Cl)ccc2[nH]1)NCc1cc2n(n1)CCCC2 ZINC000880614686 EG On-Demand Anodyne PYGL 68 38 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880614720 DD On-Demand Anodyne CAPN1 44 38 COC(=O)N[C@@H](CC(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880614720 DD On-Demand Anodyne CAPN2 77 33 CN1CCN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C[C@@H]1C(C)(C)C ZINC000880614783 GE On-Demand Bother SLC6A9 20 62 CN1CCN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C[C@@H]1C(C)(C)C ZINC000880614783 GE On-Demand Bother SSTR1 44 38 CN1CCN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C[C@H]1C(C)(C)C ZINC000880614785 GE On-Demand Bother SLC6A9 20 62 CN1CCN(C(=O)c2cc([N+](=O)[O-])ccc2N2CCOCC2)C[C@H]1C(C)(C)C ZINC000880614785 GE On-Demand Bother SSTR1 44 38 CC(C)c1cc(NC(=O)Nc2ccnc(CN(C)C)c2)ccc1O ZINC000880614790 EH On-Demand Anodyne THRA 51 34 CC(C)c1cc(NC(=O)Nc2ccnc(CN(C)C)c2)ccc1O ZINC000880614790 EH On-Demand Anodyne THRB 54 38 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccnc(CN(C)C)c2)C1 ZINC000880614812 GE On-Demand Anodyne EPHX2 30 41 CN(C)CC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880614849 GD On-Demand Anodyne CACNA1B 17 42 CN(C)CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880614850 GD On-Demand Anodyne CACNA1B 17 42 CC(=O)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880614891 DD On-Demand Anodyne TYK2 34 42 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c1 ZINC000880614893 GG On-Demand Anodyne PDGFRB 40 36 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccnc(CN(C)C)c3)CC2)c1 ZINC000880614893 GG On-Demand Anodyne LIMK2 17 40 O=C(NCc1cc2n(n1)CCCC2)c1coc(=O)c2ccccc12 ZINC000880614933 DE On-Demand Anodyne INHA 67 34 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1ccnc(CN(C)C)c1)C2 ZINC000880614936 FF On-Demand Anodyne P2RY14 43 32 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880614962 GH On-Demand Anodyne RBP4 45 42 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880614963 GH On-Demand Anodyne RBP4 45 42 O=C(NCc1cc2n(n1)CCCC2)c1cc(=O)c2ccc(Cl)cc2o1 ZINC000880614970 FF On-Demand Anodyne BCHE 37 43 O=C(CCc1cccnc1Cl)NCc1cc2n(n1)CCCC2 ZINC000880615009 DF On-Demand Anodyne SUCNR1 43 35 O=C(NCc1cc2n(n1)CCCC2)c1cc(Cl)nc(C2CC2)c1 ZINC000880615061 EG On-Demand Anodyne CACNA1I 41 32 COc1ccc(CN(CCO)C(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880615098 FE On-Demand Anodyne BMP1 21 40 COc1ccc(CN(CCO)C(=O)Nc2ccnc(CN(C)C)c2)cc1 ZINC000880615098 FE On-Demand Anodyne ROCK2 24 46 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615112 GF On-Demand Anodyne GPR119 39 41 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615113 GF On-Demand Anodyne GPR119 39 41 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615145 GD On-Demand Anodyne PREP 34 43 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615145 GD On-Demand Anodyne LGMN 70 38 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615145 GD On-Demand Anodyne SLC12A5 40 32 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615145 GD On-Demand Anodyne TMPRSS11D 54 35 O=C(NCc1cc2n(n1)CCCC2)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615146 GD On-Demand Anodyne PREP 34 43 O=C(NCc1cc2n(n1)CCCC2)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615146 GD On-Demand Anodyne LGMN 70 38 O=C(NCc1cc2n(n1)CCCC2)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615146 GD On-Demand Anodyne SLC12A5 40 32 O=C(NCc1cc2n(n1)CCCC2)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880615146 GD On-Demand Anodyne TMPRSS11D 54 35 CC[C@@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1cccc(OC)c1OC ZINC000880615189 FG On-Demand Anodyne PDGFRA 42 38 CC[C@@H](NC(=O)Nc1ccnc(CN(C)C)c1)c1cccc(OC)c1OC ZINC000880615189 FG On-Demand Anodyne KCNK3 43 38 CONC(=O)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880615234 ED On-Demand Anodyne TYK2 47 36 CONC(=O)C1CCN(C(=O)Nc2ccnc(CN(C)C)c2)CC1 ZINC000880615234 ED On-Demand Anodyne PTR1 45 33 O=C(NCc1cc2n(n1)CCCC2)[C@@H](F)c1ccccc1 ZINC000880615236 CF On-Demand Anodyne KCNQ2 32 42 O=C(NCc1cc2n(n1)CCCC2)[C@H](F)c1ccccc1 ZINC000880615237 CF On-Demand Anodyne KCNQ2 32 42 O=C(NCc1cc2n(n1)CCCC2)[C@@H](F)c1ccc(C(F)(F)F)cc1 ZINC000880615257 FH On-Demand Anodyne TRPV1 42 34 O=C(NCc1cc2n(n1)CCCC2)[C@H](F)c1ccc(C(F)(F)F)cc1 ZINC000880615258 FH On-Demand Anodyne TRPV1 42 34 N#Cc1ccc(C(=O)NCc2cc3n(n2)CCCC3)o1 ZINC000880615273 CD On-Demand Mild CSF1R 23 47 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@H]1c1ccccc1 ZINC000880615284 CF On-Demand Anodyne NAMPT 17 41 Cc1oc(-c2ccccc2)c(C(=O)NCc2cc3n(n2)CCCC3)c1C ZINC000880615285 EI On-Demand Anodyne PDE8B 56 33 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne PPIA 23 40 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne F10 56 54 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne KIT 17 44 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne ROCK1 43 33 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne PRNP 45 44 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne KDR 19 44 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne GRM4 42 39 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne NR1H4 20 57 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne HDAC1 44 46 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne PLAU 24 46 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne TAAR1 42 45 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne SIRT2 32 52 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne SMO 42 38 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne Q25615_ONCVO 40 37 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne KCNK3 117 46 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccc(Cl)cc2)c1 ZINC000880615290 HH On-Demand Anodyne KCNK9 81 41 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne GRM4 29 41 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne NR1H4 15 49 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne PLAU 15 41 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne SIRT2 23 45 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne KCNK3 82 42 NC(=O)COc1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2Br)c1 ZINC000880615293 JH On-Demand Anodyne KCNK9 66 42 CC(C)(C)OC(=O)N1CCC(OCC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615295 GE On-Demand Anodyne GPR119 39 40 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615297 GE On-Demand Anodyne GRIN2B 39 47 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615297 GE On-Demand Anodyne PREP 35 40 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615297 GE On-Demand Anodyne DPP7 41 37 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615297 GE On-Demand Anodyne TMPRSS11D 44 37 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615298 GE On-Demand Anodyne GRIN2B 39 47 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615298 GE On-Demand Anodyne PREP 35 40 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615298 GE On-Demand Anodyne DPP7 41 37 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880615298 GE On-Demand Anodyne TMPRSS11D 44 37 O=C(NCc1cc2n(n1)CCCC2)c1cnc2ccccn12 ZINC000880615303 CD On-Demand Anodyne EPHB3 22 45 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C2CC2)CC1 ZINC000880615318 DD On-Demand Anodyne L3MBTL3 60 33 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615343 GG On-Demand Anodyne PGC 42 33 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615343 GG On-Demand Anodyne REN 50 35 CC(C)(C)OC(=O)N[C@H](CC(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615344 GG On-Demand Anodyne PGC 42 33 CC(C)(C)OC(=O)N[C@H](CC(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615344 GG On-Demand Anodyne REN 50 35 CC(C)(C)OC(=O)N1CCC[C@H](CC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615359 GG On-Demand Anodyne GPR119 40 41 CC(C)(C)OC(=O)N1CCC[C@@H](CC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615360 GG On-Demand Anodyne GPR119 40 41 O=C(NCc1cc2n(n1)CCCC2)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880615368 FE On-Demand Anodyne CCR2 51 41 O=C(NCc1cc2n(n1)CCCC2)[C@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880615369 FE On-Demand Anodyne CCR2 51 41 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880615381 ED On-Demand Anodyne F2 39 42 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880615382 ED On-Demand Anodyne F2 39 42 CN1C[C@H](C(=O)NCc2cc3n(n2)CCCC3)c2ccccc2C1=O ZINC000880615401 ED On-Demand Anodyne P2RX7 47 35 CN1C[C@@H](C(=O)NCc2cc3n(n2)CCCC3)c2ccccc2C1=O ZINC000880615402 ED On-Demand Anodyne P2RX7 47 35 CC(C)(C)OC(=O)NC1CCN(CC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615410 GD On-Demand Anodyne CACNA1I 42 36 O=C(NCc1cc2n(n1)CCCC2)c1cc2occc2[nH]1 ZINC000880615435 CE On-Demand Anodyne NAMPT 17 40 O=C(CCCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880615437 GF On-Demand Anodyne PREP 22 46 O=C(CCCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880615437 GF On-Demand Anodyne TGM2 31 41 COc1cccc(C2=NO[C@@H](C(=O)NCc3cc4n(n3)CCCC4)C2)c1 ZINC000880615446 FE On-Demand Anodyne DRD4 41 32 COc1cccc(C2=NO[C@@H](C(=O)NCc3cc4n(n3)CCCC4)C2)c1 ZINC000880615446 FE On-Demand Anodyne LUCI_PHOPY 22 41 COc1cccc(C2=NO[C@H](C(=O)NCc3cc4n(n3)CCCC4)C2)c1 ZINC000880615447 FE On-Demand Anodyne DRD4 41 32 COc1cccc(C2=NO[C@H](C(=O)NCc3cc4n(n3)CCCC4)C2)c1 ZINC000880615447 FE On-Demand Anodyne LUCI_PHOPY 22 41 O=C(COCc1cccnc1)NCc1cc2n(n1)CCCC2 ZINC000880615507 DD On-Demand Anodyne CHRNA7 43 34 O=C(COCc1cccnc1)NCc1cc2n(n1)CCCC2 ZINC000880615507 DD On-Demand Anodyne NAMPT 41 41 CC(C)(C)OC(=O)NCc1cccc(C(=O)NCc2cc3n(n2)CCCC3)c1 ZINC000880615524 GG On-Demand Anodyne DRD4 43 34 O=C(NCc1cc2n(n1)CCCC2)c1ccccc1OC1CC1 ZINC000880615615 DF On-Demand Anodyne SCD 23 41 O=C(NCc1cc2n(n1)CCCC2)c1ccccc1OC1CC1 ZINC000880615615 DF On-Demand Anodyne HCN1 69 36 O=C(NCc1cc2n(n1)CCCC2)c1ccccc1OC1CC1 ZINC000880615615 DF On-Demand Anodyne HCN4 53 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne OPRM1 35 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne OPRD1 28 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CELA1 18 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne MME 47 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne TACR1 17 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSD 33 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne PGC 69 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CMA1 36 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTRA_BOVIN 23 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne FCER2 52 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSB 41 38 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne PAPA1_CARPA 75 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne TRY1_BOVIN 23 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CYSP_TRYCR 56 38 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CCKAR 58 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSK 26 53 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSL 64 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CACNA1B 61 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne PGA 43 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne TIMP3 76 37 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne TACR3 24 48 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CAPNS1 60 32 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne HLA-DRB1 33 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne REN 140 50 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne REN1 71 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSS 31 54 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CAPN1 50 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CAPN2 51 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSE 27 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne ACE2 45 33 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne SCN10A 26 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne CTSV 49 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne FPR1 71 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615628 GF On-Demand Anodyne BRCA1 49 29 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615650 EE On-Demand Anodyne CACNA1B 17 44 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615650 EE On-Demand Anodyne REN 54 35 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615686 GE On-Demand Anodyne PAPA1_CARPA 33 49 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615686 GE On-Demand Anodyne CACNA1B 18 42 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615686 GE On-Demand Anodyne FPR1 26 41 COC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615693 FD On-Demand Anodyne CACNA1B 20 46 COC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615693 FD On-Demand Anodyne REN 43 35 CN(CCC(=O)NCc1cc2n(n1)CCCC2)C(=O)OCc1ccccc1 ZINC000880615700 FE On-Demand Anodyne SLC12A5 47 33 COc1ccc(O)cc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615703 DD On-Demand Anodyne HCRTR2 18 40 CC(C)(C)OC(=O)N1CCC(CCC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880615706 GG On-Demand Anodyne GPR119 46 44 CC(C)(C)OC(=O)N1CC[C@H](CCC(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615713 GF On-Demand Anodyne GPR119 33 40 CC(C)(C)OC(=O)N1CC[C@@H](CCC(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615714 GF On-Demand Anodyne GPR119 33 40 CC(C)(C(=O)NCc1cc2n(n1)CCCC2)c1ccc2c(c1)OCO2 ZINC000880615719 EF On-Demand Anodyne NOS2 70 33 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615759 EE On-Demand Anodyne CACNA1I 40 31 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615759 EE On-Demand Anodyne GPR119 36 42 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615760 EE On-Demand Anodyne CACNA1I 40 31 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615760 EE On-Demand Anodyne GPR119 36 42 COc1cc(C(=O)NCc2cc3n(n2)CCCC3)cnc1Br ZINC000880615765 FE On-Demand Anodyne DRD4 41 32 O=C(NCc1cc2n(n1)CCCC2)c1cc(=O)c2ccc(F)cc2o1 ZINC000880615779 EE On-Demand Anodyne KCNH2 15 46 CCOc1ccccc1C(F)(F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615869 EG On-Demand Anodyne HCN1 48 32 CCOc1ccccc1C(F)(F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615869 EG On-Demand Anodyne HCN4 40 31 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615878 GG On-Demand Anodyne REN 62 35 CC(C)(C)OC(=O)N[C@@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880615878 GG On-Demand Anodyne Q82323_9DELA 67 31 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615909 FE On-Demand Anodyne PGC 44 34 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615909 FE On-Demand Anodyne CACNA1B 23 44 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615909 FE On-Demand Anodyne REN 60 38 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615909 FE On-Demand Anodyne POLG_HCV1 32 42 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615909 FE On-Demand Anodyne FPR1 43 34 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615910 FE On-Demand Anodyne PGC 44 34 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615910 FE On-Demand Anodyne CACNA1B 23 44 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615910 FE On-Demand Anodyne REN 60 38 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615910 FE On-Demand Anodyne POLG_HCV1 32 42 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880615910 FE On-Demand Anodyne FPR1 43 34 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615936 FE On-Demand Anodyne CACNA1I 40 31 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880615936 FE On-Demand Anodyne GPR119 29 40 O=C(Cc1ccc(Cl)c(F)c1)NCc1cc2n(n1)CCCC2 ZINC000880615956 DF On-Demand Anodyne P2RX7 71 38 O=C(CCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616012 FF On-Demand Anodyne PREP 23 43 O=C(CCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616012 FF On-Demand Anodyne CAPN1 16 41 O=C(CCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616012 FF On-Demand Anodyne CAPN2 34 41 O=C(CCCNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616012 FF On-Demand Anodyne TGM2 31 40 O=C(CNC(=O)c1ccccn1)NCc1cc2n(n1)CCCC2 ZINC000880616046 DC On-Demand Anodyne GRM4 50 35 O=C(CCCn1ccnc1)NCc1cc2n(n1)CCCC2 ZINC000880616051 CD On-Demand Anodyne TBXAS1 54 39 Cc1oc(-c2cccs2)nc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616071 EG On-Demand Anodyne PDE8B 42 34 O=C1CCCc2cc(C(=O)NCc3cc4n(n3)CCCC4)ccc2N1 ZINC000880616072 EE On-Demand Anodyne HDAC9 18 43 CS(=O)(=O)Nc1cc(C(=O)NCc2cc3n(n2)CCCC3)ccc1F ZINC000880616088 FD On-Demand Anodyne TRPV1 74 36 COc1cccc(OC)c1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616172 DE On-Demand Anodyne DRD2 29 44 COc1cccc(OC)c1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616172 DE On-Demand Anodyne DRD4 43 33 O=C(NCc1cc2n(n1)CCCC2)c1ccc(N2CCOCC2)nc1 ZINC000880616174 ED On-Demand Anodyne HPGDS 29 44 O=C(NCc1cc2n(n1)CCCC2)c1ccc(N2CCOCC2)nc1 ZINC000880616174 ED On-Demand Anodyne NAMPT 21 49 COC(=O)[C@@H]1CN(C(=O)c2nnn(C)n2)C[C@H]1c1ccc(Cl)cc1 ZINC000880616187 EC On-Demand Anodyne SLC6A4 34 54 COC(=O)[C@@H]1CN(C(=O)c2nnn(C)n2)C[C@H]1c1ccc(Cl)cc1 ZINC000880616187 EC On-Demand Anodyne SLC6A3 57 54 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880616223 FD On-Demand Anodyne EPHX2 18 48 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880616223 FD On-Demand Anodyne L3MBTL3 58 36 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880616223 FD On-Demand Anodyne NAMPT 34 43 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne KLK3 67 34 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne CYSP_TRYCR 40 33 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne CAPNS1 56 31 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne CAPN1 49 35 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne CAPN2 72 33 C[C@@H](NC(=O)c1c2c(nn1C)CCSC2)C(=O)OCc1ccccc1 ZINC000880616224 FE On-Demand Anodyne NPR 55 33 Cn1nc2c(c1NC(=O)NCCCOc1ccccc1F)CCCC2 ZINC000880616228 EG On-Demand Anodyne BCHE 61 36 O=C(CCc1ccc2ccccc2n1)NCc1cc2n(n1)CCCC2 ZINC000880616229 EG On-Demand Anodyne SUCNR1 51 35 Cn1nc2c(c1NC(=O)N1CCN(c3ccc([N+](=O)[O-])cc3)CC1)CCCC2 ZINC000880616231 GF On-Demand Bother SSTR1 42 38 COc1ccc(-c2nnc(S)n2CC(=O)NCc2cc3n(n2)CCCC3)cc1 ZINC000880616241 GE On-Demand Anodyne AVPR1B 55 39 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CELA1 25 41 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne ELANE 28 41 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne MME 35 46 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne KLK3 70 37 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CTSB 55 41 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne PAPA1_CARPA 50 34 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CTSK 37 40 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CTSL 40 39 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne PREP 17 40 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CAPNS1 81 37 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CAPN1 97 42 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne CAPN2 128 39 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne NPR 77 35 C[C@@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616243 DF On-Demand Anodyne Q6PRC7_IXORI 41 33 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CELA1 25 41 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne ELANE 28 41 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne MME 35 46 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne KLK3 70 37 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CTSB 55 41 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne PAPA1_CARPA 50 34 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CTSK 37 40 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CTSL 40 39 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne PREP 17 40 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CAPNS1 81 37 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CAPN1 97 42 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne CAPN2 128 39 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne NPR 77 35 C[C@H](NC(=O)C[C@@H]1C[C@H]1C1CC1)C(=O)OCc1ccccc1 ZINC000880616244 DF On-Demand Anodyne Q6PRC7_IXORI 41 33 O=C(Cc1csc(-c2ccc3c(c2)OCO3)n1)NCc1cc2n(n1)CCCC2 ZINC000880616298 GF On-Demand Anodyne NOS2 90 35 O=C(Cc1csc(-c2ccc3c(c2)OCO3)n1)NCc1cc2n(n1)CCCC2 ZINC000880616298 GF On-Demand Anodyne CLK4 57 38 O=C(Cc1ccccc1[N+](=O)[O-])NCc1cc2n(n1)CCCC2 ZINC000880616323 DD On-Demand Bother COLA 81 32 O=C(CNc1cccc(C(F)(F)F)c1)NCc1cc2n(n1)CCCC2 ZINC000880616328 FF On-Demand Anodyne CCR2 57 36 O=C(NCc1cc2n(n1)CCCC2)c1cc(C2CC2)nc2ccccc12 ZINC000880616348 EH On-Demand Anodyne TACR3 15 43 COC(=O)[C@@H]1CN(C(=O)c2nccnc2SC)C[C@H]1c1ccc(Cl)cc1 ZINC000880616349 GF On-Demand Anodyne SLC6A4 21 48 COC(=O)[C@@H]1CN(C(=O)c2nccnc2SC)C[C@H]1c1ccc(Cl)cc1 ZINC000880616349 GF On-Demand Anodyne SLC6A3 37 48 Cn1nc2c(c1NC(=O)NCc1ccc(-n3ccnc3)nc1)CCCC2 ZINC000880616355 FE On-Demand Anodyne NOS2 69 34 Cn1nc2c(c1NC(=O)NCc1ccc(-n3ccnc3)nc1)CCCC2 ZINC000880616355 FE On-Demand Anodyne NAMPT 33 54 O=C(NCc1cc2n(n1)CCCC2)c1ccc(-n2ccnc2)nc1 ZINC000880616370 DD On-Demand Anodyne NOS2 60 33 O=C(NCc1cc2n(n1)CCCC2)c1ccc(-n2ccnc2)nc1 ZINC000880616370 DD On-Demand Anodyne NAMPT 22 41 CC[C@@H](NC(=O)c1nccnc1SC)c1ccccc1F ZINC000880616385 DG On-Demand Anodyne CTSA 54 38 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616398 DD On-Demand Anodyne CAPN1 44 38 COC(=O)N[C@H](CC(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616398 DD On-Demand Anodyne CAPN2 77 33 O=C(NCc1cc2n(n1)CCCC2)c1ccc(S(=O)(=O)N2CCCC2)o1 ZINC000880616404 GD On-Demand Anodyne NAMPT 52 46 O=C(NCc1cc2n(n1)CCCC2)c1nc(Cl)ccc1Cl ZINC000880616414 EF On-Demand Anodyne CNR1 49 31 CC(C)(C)OC(=O)NC[C@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880616415 GG On-Demand Anodyne KCNQ2 40 34 CC(C)(C)OC(=O)NC[C@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880616415 GG On-Demand Anodyne REN 45 33 CC(C)(C)OC(=O)NC[C@@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880616417 GG On-Demand Anodyne KCNQ2 40 34 CC(C)(C)OC(=O)NC[C@@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1 ZINC000880616417 GG On-Demand Anodyne REN 45 33 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne MME 36 41 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne KLK3 70 35 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne CTSB 52 40 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne PAPA1_CARPA 55 34 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne CYSP_TRYCR 56 43 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne CAPNS1 62 35 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne CAPN1 76 40 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne CAPN2 112 37 CSc1nccnc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880616426 EE On-Demand Anodyne NPR 79 36 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne MME 36 41 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne KLK3 70 35 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne CTSB 52 40 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne PAPA1_CARPA 55 34 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne CYSP_TRYCR 56 43 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne CAPNS1 62 35 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne CAPN1 76 40 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne CAPN2 112 37 CSc1nccnc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880616428 EE On-Demand Anodyne NPR 79 36 O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)NCc1cc2n(n1)CCCC2 ZINC000880616430 GF On-Demand Anodyne CACNA1I 18 41 Cn1cc(-c2cccc(C(=O)NCc3cc4n(n3)CCCC4)c2)cn1 ZINC000880616434 EF On-Demand Anodyne DRD4 41 33 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne MME 26 40 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne KLK3 69 36 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne CTSB 48 38 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne PAPA1_CARPA 55 33 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne CAPNS1 56 34 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne CAPN1 77 39 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne CAPN2 113 36 C[C@@H](NC(=O)c1cc(C(F)F)[nH]n1)C(=O)OCc1ccccc1 ZINC000880616443 DE On-Demand Anodyne NPR 77 38 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616469 GE On-Demand Anodyne GRPR 59 35 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616469 GE On-Demand Anodyne GHSR 15 40 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616469 GE On-Demand Anodyne MC1R 43 38 Cn1nc2c(c1NC(=O)NCc1ccc(C(=O)N3CCCC3)cc1)CCCC2 ZINC000880616471 GF On-Demand Anodyne AVPR2 17 43 O=C(COc1ccccc1-c1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616478 FH On-Demand Anodyne PTGIR 48 34 O=C(CNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616479 ED On-Demand Anodyne PREP 26 42 O=C(CNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616479 ED On-Demand Anodyne NPR 43 31 O=C(CNC(=O)OCc1ccccc1)NCc1cc2n(n1)CCCC2 ZINC000880616479 ED On-Demand Anodyne SLC12A5 53 34 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616493 FF On-Demand Anodyne PAPA1_CARPA 36 47 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616493 FF On-Demand Anodyne REN 47 34 CN1CC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)CC1=O ZINC000880616497 CC On-Demand Anodyne P2RX7 21 40 CN1CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)CC1=O ZINC000880616499 CC On-Demand Anodyne P2RX7 21 40 O=C(Cc1cccs1)NCc1cc2n(n1)CCCC2 ZINC000880616500 CE On-Demand Anodyne CA5B 32 46 O=C(Cc1cccs1)NCc1cc2n(n1)CCCC2 ZINC000880616500 CE On-Demand Anodyne CA5A 31 46 O=C(NCCCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616507 ED On-Demand Anodyne FKBP1A 15 42 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne MME 30 42 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne GALR1 46 33 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne KLK3 83 38 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CTSB 54 39 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne PAPA1_CARPA 46 35 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CYSP_TRYCR 50 37 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CTSK 36 41 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CTSL 40 39 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CAPNS1 74 34 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne LGMN 50 38 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CAPN1 89 40 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne CAPN2 123 36 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne NPR 79 34 C[C@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616514 DC On-Demand Anodyne R1A_CVHSA 25 50 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne MME 30 42 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne GALR1 46 33 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne KLK3 83 38 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CTSB 54 39 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne PAPA1_CARPA 46 35 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CYSP_TRYCR 50 37 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CTSK 36 41 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CTSL 40 39 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CAPNS1 74 34 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne LGMN 50 38 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CAPN1 89 40 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne CAPN2 123 36 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne NPR 79 34 C[C@@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616516 DC On-Demand Anodyne R1A_CVHSA 25 50 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne MME 30 42 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne GALR1 46 33 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne KLK3 83 38 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CTSB 54 39 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne PAPA1_CARPA 46 35 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CYSP_TRYCR 50 37 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CTSK 36 41 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CTSL 40 39 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CAPNS1 74 34 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne LGMN 50 38 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CAPN1 89 40 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne CAPN2 123 36 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne NPR 79 34 C[C@H](NC(=O)C[C@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616517 DC On-Demand Anodyne R1A_CVHSA 25 50 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne MME 30 42 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne GALR1 46 33 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne KLK3 83 38 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CTSB 54 39 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne PAPA1_CARPA 46 35 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CYSP_TRYCR 50 37 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CTSK 36 41 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CTSL 40 39 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CAPNS1 74 34 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne LGMN 50 38 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CAPN1 89 40 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne CAPN2 123 36 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne NPR 79 34 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)C(=O)OCc1ccccc1 ZINC000880616518 DC On-Demand Anodyne R1A_CVHSA 25 50 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CSCN1C(=O)c1ccccc1 ZINC000880616529 FE On-Demand Anodyne PREP 28 41 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CSCN1C(=O)c1ccccc1 ZINC000880616530 FE On-Demand Anodyne PREP 28 41 COCCn1cc(C(=O)NCc2cc3n(n2)CCCC3)c2ccccc21 ZINC000880616531 FF On-Demand Anodyne CNR1 21 46 COCCn1cc(C(=O)NCc2cc3n(n2)CCCC3)c2ccccc21 ZINC000880616531 FF On-Demand Anodyne CNR2 31 49 CC(C)(C)OC(=O)N1CCC(CC(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880616537 GF On-Demand Anodyne GPR119 44 42 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne MME 18 42 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne KLK3 56 34 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne CTSB 53 37 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne CTSL 40 38 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne CAPNS1 60 34 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne CAPN1 71 39 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne CAPN2 109 35 C[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616555 FE On-Demand Anodyne NPR 74 34 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne MME 18 42 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne KLK3 56 34 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne CTSB 53 37 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne CTSL 40 38 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne CAPNS1 60 34 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne CAPN1 71 39 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne CAPN2 109 35 C[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616556 FE On-Demand Anodyne NPR 74 34 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne MME 18 42 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne KLK3 56 34 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne CTSB 53 37 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne CTSL 40 38 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne CAPNS1 60 34 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne CAPN1 71 39 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne CAPN2 109 35 C[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616557 FE On-Demand Anodyne NPR 74 34 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne MME 18 42 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne KLK3 56 34 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne CTSB 53 37 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne CTSL 40 38 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne CAPNS1 60 34 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne CAPN1 71 39 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne CAPN2 109 35 C[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C(=O)OCc1ccccc1 ZINC000880616558 FE On-Demand Anodyne NPR 74 34 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne CTSB 41 36 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne CCR5 19 43 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne CAPNS1 77 34 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne LGMN 47 36 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne CAPN1 77 39 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne CAPN2 99 36 C[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)C(=O)OCc1ccccc1 ZINC000880616560 ED On-Demand Anodyne NPR 49 32 Cn1nc2c(c1NC(=O)NC[C@H](O)c1cccc(Cl)c1)CCCC2 ZINC000880616565 EF On-Demand Anodyne ADRB1 28 41 Cn1nc2c(c1NC(=O)NC[C@H](O)c1cccc(Cl)c1)CCCC2 ZINC000880616565 EF On-Demand Anodyne ADRB3 43 41 Cn1nc2c(c1NC(=O)NC[C@@H](O)c1cccc(Cl)c1)CCCC2 ZINC000880616566 EF On-Demand Anodyne ADRB1 28 41 Cn1nc2c(c1NC(=O)NC[C@@H](O)c1cccc(Cl)c1)CCCC2 ZINC000880616566 EF On-Demand Anodyne ADRB3 43 41 CCCOc1ccc(OCC(=O)NCc2cc3n(n2)CCCC3)cc1 ZINC000880616575 EF On-Demand Anodyne PLA2G4B 71 32 CC[C@@H](NC(=O)COC1CC1)c1ccccc1F ZINC000880616578 CF On-Demand Anodyne TIMP3 73 34 C#CCNS(=O)(=O)c1ccc(C(=O)NCc2cc3n(n2)CCCC3)cc1 ZINC000880616581 FD On-Demand Mild NAMPT 30 41 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne KLK3 74 36 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne CTSB 46 38 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne PAPA1_CARPA 60 35 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne CYSP_TRYCR 49 36 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne CAPNS1 56 33 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne CAPN1 71 38 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne CAPN2 107 35 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne NPR 66 34 C[C@@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616631 GD On-Demand Anodyne Q6PRC7_IXORI 41 31 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne KLK3 74 36 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne CTSB 46 38 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne PAPA1_CARPA 60 35 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne CYSP_TRYCR 49 36 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne CAPNS1 56 33 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne CAPN1 71 38 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne CAPN2 107 35 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne NPR 66 34 C[C@H](NC(=O)Cc1c(Br)cnn1C)C(=O)OCc1ccccc1 ZINC000880616633 GD On-Demand Anodyne Q6PRC7_IXORI 41 31 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne ACE 40 41 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne MME 39 42 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne KLK3 55 33 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CTSB 52 42 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne PAPA1_CARPA 45 34 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CYSP_TRYCR 41 37 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CTSK 36 42 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne PREP 26 40 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CAPNS1 69 35 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne LGMN 53 37 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CAPN1 77 41 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne CAPN2 106 37 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne ACE2 46 33 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne NPR 70 36 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne BIRC2 22 41 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne Q6PRC7_IXORI 42 33 C[C@@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616638 FC On-Demand Anodyne SLC12A5 70 40 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne ACE 40 41 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne MME 39 42 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne KLK3 55 33 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CTSB 52 42 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne PAPA1_CARPA 45 34 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CYSP_TRYCR 41 37 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CTSK 36 42 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne PREP 26 40 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CAPNS1 69 35 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne LGMN 53 37 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CAPN1 77 41 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne CAPN2 106 37 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne ACE2 46 33 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne NPR 70 36 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne BIRC2 22 41 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne Q6PRC7_IXORI 42 33 C[C@H](NC(=O)CN1CCCCS1(=O)=O)C(=O)OCc1ccccc1 ZINC000880616639 FC On-Demand Anodyne SLC12A5 70 40 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880616644 FD On-Demand Anodyne F2 40 38 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880616644 FD On-Demand Anodyne LGMN 73 37 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880616647 FD On-Demand Anodyne F2 40 38 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880616647 FD On-Demand Anodyne LGMN 73 37 NC(=O)COc1ccccc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616659 ED On-Demand Anodyne HCN1 69 35 NC(=O)COc1ccccc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616659 ED On-Demand Anodyne HCN4 52 34 CC[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1ccccc1F ZINC000880616665 EH On-Demand Anodyne PLD1 56 37 CC[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1ccccc1F ZINC000880616665 EH On-Demand Anodyne CTSA 43 36 CC[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1ccccc1F ZINC000880616666 EH On-Demand Anodyne PLD1 56 37 CC[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1ccccc1F ZINC000880616666 EH On-Demand Anodyne CTSA 43 36 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne CTSB 41 38 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne PAPA1_CARPA 40 33 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne CAPNS1 59 33 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne CAPN1 67 39 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne CAPN2 101 36 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne NPR 61 35 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne PSMB8 58 33 C[C@@H](NC(=O)CC[C@@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616685 EF On-Demand Anodyne SLC12A5 48 37 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne CTSB 41 38 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne PAPA1_CARPA 40 33 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne CAPNS1 59 33 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne CAPN1 67 39 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne CAPN2 101 36 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne NPR 61 35 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne PSMB8 58 33 C[C@@H](NC(=O)CC[C@H]1CC(C)(C)CO1)C(=O)OCc1ccccc1 ZINC000880616689 EF On-Demand Anodyne SLC12A5 48 37 O=C(NCc1cc2n(n1)CCCC2)c1cccnc1Cl ZINC000880616693 CE On-Demand Anodyne G2YM83_BOTF4 71 36 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne ELANE 21 48 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne MME 48 42 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne ANPEP 40 34 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CASP3 17 42 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne KLK3 88 40 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CTSB 62 41 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne PAPA1_CARPA 74 37 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CYSP_TRYCR 53 39 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CTSK 39 41 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CTSL 43 38 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CAPNS1 67 38 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne HLA-DRB1 59 34 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne MMP11 71 35 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CTSS 18 40 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne GHSR 41 37 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CAPN1 94 44 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne CAPN2 130 42 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne NPR 87 39 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne PSMB5 48 41 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne Q6PRC7_IXORI 41 32 C[C@@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616697 CC On-Demand Anodyne SLC12A5 45 34 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne ELANE 21 48 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne MME 48 42 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne ANPEP 40 34 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CASP3 17 42 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne KLK3 88 40 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CTSB 62 41 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne PAPA1_CARPA 74 37 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CYSP_TRYCR 53 39 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CTSK 39 41 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CTSL 43 38 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CAPNS1 67 38 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne HLA-DRB1 59 34 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne MMP11 71 35 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CTSS 18 40 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne GHSR 41 37 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CAPN1 94 44 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne CAPN2 130 42 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne NPR 87 39 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne PSMB5 48 41 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne Q6PRC7_IXORI 41 32 C[C@H](NC(=O)c1nnn(C)n1)C(=O)OCc1ccccc1 ZINC000880616699 CC On-Demand Anodyne SLC12A5 45 34 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc2n(n1)CCCC2 ZINC000880616704 FD On-Demand Anodyne DRD4 28 42 O=C(CN1CCN(c2ccccn2)CC1)NCc1cc2n(n1)CCCC2 ZINC000880616704 FD On-Demand Anodyne SLC27A1 63 53 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne PREP 35 43 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne LGMN 65 37 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne SLC12A5 40 32 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne Q9NAW4_PLAFA 42 50 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne TMPRSS11D 52 36 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880616711 GD On-Demand Anodyne VHL 68 41 O=C(NCc1cc2n(n1)CCCC2)c1cnn2ccccc12 ZINC000880616808 CD On-Demand Anodyne EPHB3 37 45 O=C(NCc1cc2n(n1)CCCC2)c1ccnc(-n2ccnc2)c1 ZINC000880616826 DD On-Demand Anodyne NOS2 87 35 Cc1nnc(-c2cccc(C(=O)NCc3cc4n(n3)CCCC4)c2)o1 ZINC000880616835 EF On-Demand Anodyne DRD4 40 31 Cc1oc(-c2ccccc2F)nc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616836 FG On-Demand Anodyne PDE8B 46 33 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616851 GE On-Demand Anodyne PAPA1_CARPA 33 49 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616851 GE On-Demand Anodyne CACNA1B 18 42 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880616851 GE On-Demand Anodyne FPR1 26 41 COC(=O)c1cc(C(=O)NCc2cc3n(n2)CCCC3)ccn1 ZINC000880616852 DD On-Demand Anodyne DRD4 40 31 O=C(Cn1nc(-c2ccccc2)oc1=O)NCc1cc2n(n1)CCCC2 ZINC000880616858 FD On-Demand Anodyne PDE8B 48 33 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CELA1 17 41 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne MME 29 41 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CASP3 21 43 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne KLK3 58 34 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CTSB 47 40 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne PAPA1_CARPA 61 34 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CYSP_TRYCR 52 38 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CTSK 26 40 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CAPNS1 57 34 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CAPN1 74 40 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CASP1 27 41 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne CAPN2 108 37 Cc1ncc(CC(=O)N[C@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616895 DD On-Demand Anodyne NPR 76 35 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CELA1 17 41 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne MME 29 41 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CASP3 21 43 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne KLK3 58 34 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CTSB 47 40 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne PAPA1_CARPA 61 34 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CYSP_TRYCR 52 38 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CTSK 26 40 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CAPNS1 57 34 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CAPN1 74 40 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CASP1 27 41 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne CAPN2 108 37 Cc1ncc(CC(=O)N[C@@H](C)C(=O)OCc2ccccc2)o1 ZINC000880616896 DD On-Demand Anodyne NPR 76 35 CS(=O)(=O)C1CCC(C(=O)Nc2cc3cc[nH]c3cn2)CC1 ZINC000880616904 DE On-Demand Anodyne GSK3A 29 44 Cn1nc2c(c1NC(=O)NCC(=O)NCc1ccccc1)CCCC2 ZINC000880616907 ED On-Demand Anodyne ACHE 41 38 Cn1nc2c(c1NC(=O)NCC(=O)NCc1ccccc1)CCCC2 ZINC000880616907 ED On-Demand Anodyne FABP4 42 39 Cn1nc2c(c1NC(=O)NCC(=O)NCc1ccccc1)CCCC2 ZINC000880616907 ED On-Demand Anodyne BCHE 65 36 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne ACE 27 42 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne OPRM1 19 40 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CELA1 18 41 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne ELANE 28 42 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne MME 45 46 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CASP3 16 41 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne KLK3 78 37 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CTSB 56 43 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne PAPA1_CARPA 63 38 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CYSP_TRYCR 41 38 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CTSK 34 43 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CTSL 33 43 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CAPNS1 68 39 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CTSS 15 43 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CAPN1 84 43 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CASP1 27 40 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne CAPN2 118 39 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne NPR 85 44 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne PSMB5 32 40 CC(=O)N(CC(=O)N[C@@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616923 FE On-Demand Anodyne Q6PRC7_IXORI 45 36 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne ACE 27 42 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne OPRM1 19 40 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CELA1 18 41 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne ELANE 28 42 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne MME 45 46 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CASP3 16 41 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne KLK3 78 37 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CTSB 56 43 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne PAPA1_CARPA 63 38 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CYSP_TRYCR 41 38 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CTSK 34 43 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CTSL 33 43 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CAPNS1 68 39 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CTSS 15 43 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CAPN1 84 43 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CASP1 27 40 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne CAPN2 118 39 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne NPR 85 44 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne PSMB5 32 40 CC(=O)N(CC(=O)N[C@H](C)C(=O)OCc1ccccc1)c1ccccc1 ZINC000880616924 FE On-Demand Anodyne Q6PRC7_IXORI 45 36 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne ACE 58 40 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CELA1 18 41 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne MME 71 41 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne ANPEP 51 35 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne KLK3 80 37 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CTSB 67 42 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne PAPA1_CARPA 67 36 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CYSP_TRYCR 51 36 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CTSK 42 42 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CTSL 48 38 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CAPNS1 71 40 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne HLA-DRB1 50 32 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne REN 45 37 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CAPN1 96 45 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CASP1 26 40 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne CAPN2 145 42 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne ACE2 56 36 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne FPR1 51 37 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne NPR 89 40 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne PSMB5 57 41 C[C@@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616925 EF On-Demand Anodyne PSMB8 15 41 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne ACE 58 40 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CELA1 18 41 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne MME 71 41 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne ANPEP 51 35 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne KLK3 80 37 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CTSB 67 42 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne PAPA1_CARPA 67 36 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CYSP_TRYCR 51 36 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CTSK 42 42 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CTSL 48 38 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CAPNS1 71 40 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne HLA-DRB1 50 32 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne REN 45 37 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CAPN1 96 45 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CASP1 26 40 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne CAPN2 145 42 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne ACE2 56 36 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne FPR1 51 37 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne NPR 89 40 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne PSMB5 57 41 C[C@H](NC(=O)c1cnc(CC2CC2)s1)C(=O)OCc1ccccc1 ZINC000880616926 EF On-Demand Anodyne PSMB8 15 41 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616927 FG On-Demand Anodyne PAPA1_CARPA 40 48 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616927 FG On-Demand Anodyne CTSK 22 41 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616927 FG On-Demand Anodyne TACR3 16 40 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616927 FG On-Demand Anodyne FPR1 50 41 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616928 FG On-Demand Anodyne PAPA1_CARPA 40 48 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616928 FG On-Demand Anodyne CTSK 22 41 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616928 FG On-Demand Anodyne TACR3 16 40 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)c1ccccc1F ZINC000880616928 FG On-Demand Anodyne FPR1 50 41 O=C(NCc1cc2n(n1)CCCC2)c1ccc(CS(=O)(=O)c2ccccc2)o1 ZINC000880616933 GF On-Demand Anodyne NAMPT 53 39 O=C(CCC(=O)c1ccc2c(c1)OCCO2)NCc1cc2n(n1)CCCC2 ZINC000880616939 FE On-Demand Anodyne NOS2 41 31 CCOc1ccccc1OCC(=O)NCc1cc2n(n1)CCCC2 ZINC000880616943 EE On-Demand Anodyne HCN1 50 34 CCOc1ccccc1OCC(=O)NCc1cc2n(n1)CCCC2 ZINC000880616943 EE On-Demand Anodyne HCN4 42 33 COC(=O)[C@@H]1CN(C(=O)c2cccn3nccc23)C[C@H]1c1ccc(Cl)cc1 ZINC000880616947 GG On-Demand Anodyne SLC6A4 18 47 COC(=O)[C@@H]1CN(C(=O)c2cccn3nccc23)C[C@H]1c1ccc(Cl)cc1 ZINC000880616947 GG On-Demand Anodyne SLC6A3 33 47 O=C(CNC(=O)c1cc2ccccc2[nH]1)NCc1cc2n(n1)CCCC2 ZINC000880617017 FD On-Demand Anodyne PYGL 48 36 O=C(CNC(=O)c1cc2ccccc2[nH]1)NCc1cc2n(n1)CCCC2 ZINC000880617017 FD On-Demand Anodyne PLD2 31 42 O=C(CNC(=O)c1cc2ccccc2[nH]1)NCc1cc2n(n1)CCCC2 ZINC000880617017 FD On-Demand Anodyne NAMPT 16 40 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc2n(n1)CCCC2 ZINC000880617031 FD On-Demand Anodyne ACHE 38 42 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc2n(n1)CCCC2 ZINC000880617031 FD On-Demand Anodyne AVPR1B 16 42 O=C(CN1CCN(Cc2ccccc2)CC1)NCc1cc2n(n1)CCCC2 ZINC000880617031 FD On-Demand Anodyne SIGMAR1 37 44 O=C(NCc1cc2n(n1)CCCC2)c1ccc2[nH]ccc2c1 ZINC000880617033 CF On-Demand Anodyne NAMPT 15 41 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CC(=O)N(c2ccc(F)cc2)C1 ZINC000880617039 FE On-Demand Anodyne P2RX7 15 42 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CC(=O)N(c2ccc(F)cc2)C1 ZINC000880617040 FE On-Demand Anodyne P2RX7 15 42 O=C(NCc1cc2n(n1)CCCC2)c1cc2cccc(Cl)c2o1 ZINC000880617064 EH On-Demand Anodyne NAMPT 27 40 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617109 FF On-Demand Anodyne SLC6A1 78 38 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617109 FF On-Demand Anodyne CCR3 71 39 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617109 FF On-Demand Anodyne CACNA1G 28 43 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617110 FF On-Demand Anodyne SLC6A1 78 38 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617110 FF On-Demand Anodyne CCR3 71 39 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880617110 FF On-Demand Anodyne CACNA1G 28 43 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880617120 ED On-Demand Anodyne INHA 22 47 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880617121 ED On-Demand Anodyne INHA 22 47 O=C(CCn1c(S)nc2ccccc2c1=O)NCc1cc2n(n1)CCCC2 ZINC000880617123 GD On-Demand Anodyne HTR7 16 41 O=C(NCc1cc2n(n1)CCCC2)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880617124 GF On-Demand Anodyne P2RX7 57 55 O=C(NCc1cc2n(n1)CCCC2)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880617125 GF On-Demand Anodyne P2RX7 57 55 Cn1nc2c(c1NC(=O)NCCc1cccnc1)CCCC2 ZINC000880617132 CE On-Demand Anodyne PTAFR 22 40 Cn1nc2c(c1NC(=O)NCCc1cccnc1)CCCC2 ZINC000880617132 CE On-Demand Anodyne NAMPT 49 48 CC(C)(C)OC(=O)N1CCC(C(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880617146 FE On-Demand Anodyne EPHX2 19 41 CC(C)(C)OC(=O)N1CCC(C(=O)NCc2cc3n(n2)CCCC3)CC1 ZINC000880617146 FE On-Demand Anodyne GPR119 45 42 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne MME 39 44 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne KLK3 52 33 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CTSB 52 38 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CYSP_TRYCR 46 37 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CTSK 40 41 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CTSL 47 34 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne TIMP3 41 33 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CAPNS1 60 33 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CAPN1 75 38 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CASP1 28 42 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne CAPN2 117 38 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne NPR 78 38 C[C@@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617151 DE On-Demand Anodyne PSMB5 46 36 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne MME 39 44 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne KLK3 52 33 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CTSB 52 38 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne PAPA1_CARPA 54 33 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CYSP_TRYCR 46 37 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CTSK 40 41 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CTSL 47 34 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne TIMP3 41 33 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CAPNS1 60 33 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CAPN1 75 38 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CASP1 28 42 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne CAPN2 117 38 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne NPR 78 38 C[C@H](NC(=O)c1cnc(C2CC2)o1)C(=O)OCc1ccccc1 ZINC000880617152 DE On-Demand Anodyne PSMB5 46 36 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne ACE 45 41 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CELA1 30 41 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne ELANE 21 40 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne MME 41 46 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne KLK3 67 35 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CTSB 60 41 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne PAPA1_CARPA 61 36 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CYSP_TRYCR 41 38 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CTSK 39 41 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CTSL 43 40 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne PREP 22 42 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CAPNS1 76 37 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CTSS 29 41 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CAPN1 102 40 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne CAPN2 126 39 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne NPR 77 34 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne XIAP 42 35 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne PSMB5 42 38 C[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)C(=O)OCc1ccccc1 ZINC000880617161 FD On-Demand Anodyne SLC12A5 43 34 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne MME 20 41 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne KLK3 73 35 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CTSB 46 38 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne PAPA1_CARPA 48 32 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CYSP_TRYCR 42 34 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CTSK 31 40 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne MAP1 52 38 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CAPNS1 59 33 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CAPN1 69 38 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne CAPN2 111 35 C[C@@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617163 EF On-Demand Anodyne NPR 75 34 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne MME 20 41 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne KLK3 73 35 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CTSB 46 38 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne PAPA1_CARPA 48 32 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CYSP_TRYCR 42 34 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CTSK 31 40 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne MAP1 52 38 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CAPNS1 59 33 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CAPN1 69 38 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne CAPN2 111 35 C[C@H](NC(=O)c1ncsc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617164 EF On-Demand Anodyne NPR 75 34 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne MME 24 42 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne KLK3 58 34 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne CTSB 48 39 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne PAPA1_CARPA 60 33 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne CYSP_TRYCR 46 38 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne CAPNS1 57 35 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne CAPN1 78 41 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne CAPN2 106 36 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617165 EF On-Demand Anodyne NPR 77 37 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne MME 24 42 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne KLK3 58 34 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne CTSB 48 39 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne PAPA1_CARPA 60 33 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne CYSP_TRYCR 46 38 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne CAPNS1 57 35 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne CAPN1 78 41 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne CAPN2 106 36 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617166 EF On-Demand Anodyne NPR 77 37 O=C(NCc1cc2n(n1)CCCC2)c1cc(=O)c2ccccc2o1 ZINC000880617169 DE On-Demand Anodyne BCHE 39 46 O=C(NCc1cc2n(n1)CCCC2)c1cc(=O)c2ccccc2o1 ZINC000880617169 DE On-Demand Anodyne NAMPT 26 40 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CELA1 19 44 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild MME 49 43 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CASP3 17 44 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild KLK3 84 39 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CTSB 64 45 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild PAPA1_CARPA 74 37 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CYSP_TRYCR 45 39 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CTSK 37 40 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CTSL 37 40 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CAPNS1 65 37 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild HLA-DRB1 53 34 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild REN 22 41 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CTSS 18 40 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CAPN1 97 45 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CASP1 29 42 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild CAPN2 129 42 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild FPR1 43 37 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild NPR 85 39 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild PSMB5 60 40 C=CC(C)(C)CC(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880617176 CF On-Demand Mild Q6PRC7_IXORI 45 36 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CELA1 19 44 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild MME 49 43 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CASP3 17 44 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild KLK3 84 39 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CTSB 64 45 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild PAPA1_CARPA 74 37 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CYSP_TRYCR 45 39 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CTSK 37 40 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CTSL 37 40 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CAPNS1 65 37 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild HLA-DRB1 53 34 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild REN 22 41 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CTSS 18 40 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CAPN1 97 45 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CASP1 29 42 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild CAPN2 129 42 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild FPR1 43 37 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild NPR 85 39 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild PSMB5 60 40 C=CC(C)(C)CC(=O)N[C@@H](C)C(=O)OCc1ccccc1 ZINC000880617177 CF On-Demand Mild Q6PRC7_IXORI 45 36 COC(=O)[C@@H]1CN(C(=O)c2cc(C)co2)C[C@H]1c1ccc(Cl)cc1 ZINC000880617182 EG On-Demand Anodyne SLC6A4 30 51 COC(=O)[C@@H]1CN(C(=O)c2cc(C)co2)C[C@H]1c1ccc(Cl)cc1 ZINC000880617182 EG On-Demand Anodyne SLC6A3 52 51 CC[C@@H](NC(=O)CN1CCCCS1(=O)=O)c1ccccc1F ZINC000880617186 ED On-Demand Anodyne KCNQ2 29 41 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617220 EE On-Demand Anodyne F2 42 40 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617220 EE On-Demand Anodyne CACNA1B 15 43 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617220 EE On-Demand Anodyne PREP 20 46 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617220 EE On-Demand Anodyne LGMN 65 33 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617221 EE On-Demand Anodyne F2 42 40 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617221 EE On-Demand Anodyne CACNA1B 15 43 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617221 EE On-Demand Anodyne PREP 20 46 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617221 EE On-Demand Anodyne LGMN 65 33 O=C(CCn1ccnc1)NCc1cc2n(n1)CCCC2 ZINC000880617230 CD On-Demand Anodyne TBXAS1 48 37 O=C(N[C@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1)c1ccccc1 ZINC000880617237 GG On-Demand Anodyne MTTP 71 41 O=C(N[C@@H](C(=O)NCc1cc2n(n1)CCCC2)c1ccccc1)c1ccccc1 ZINC000880617238 GG On-Demand Anodyne MTTP 71 41 O=C(NCc1cc2n(n1)CCCC2)c1c(F)cccc1Cl ZINC000880617240 DF On-Demand Anodyne TYK2 18 40 CN1C(=O)CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)[C@H]1c1ccccc1 ZINC000880617259 FE On-Demand Anodyne P2RX7 31 40 CN1C(=O)CC[C@H](C(=O)NCc2cc3n(n2)CCCC3)[C@@H]1c1ccccc1 ZINC000880617260 FE On-Demand Anodyne P2RX7 31 40 CN1C(=O)CC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)[C@@H]1c1ccccc1 ZINC000880617261 FE On-Demand Anodyne P2RX7 31 40 CN1C(=O)CC[C@@H](C(=O)NCc2cc3n(n2)CCCC3)[C@H]1c1ccccc1 ZINC000880617262 FE On-Demand Anodyne P2RX7 31 40 O=C(NCc1cc2n(n1)CCCC2)c1cc(Cl)nc(Cl)c1 ZINC000880617280 EF On-Demand Anodyne CACNA1I 41 32 CS(=O)(=O)Nc1cccc(C(=O)NCc2cc3n(n2)CCCC3)c1 ZINC000880617288 ED On-Demand Anodyne DRD4 40 32 O=C(COc1cccnc1)NCc1cc2n(n1)CCCC2 ZINC000880617293 CD On-Demand Anodyne NAMPT 20 41 N#CCOc1ccccc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617304 DE On-Demand Mild HCN1 68 34 N#CCOc1ccccc1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617304 DE On-Demand Mild HCN4 51 33 CO[C@@](C)(CO)CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880617327 DE On-Demand Anodyne ADCYAP1R1 55 35 COc1ccc(O)c(C(=O)NCc2cc3n(n2)CCCC3)c1 ZINC000880617330 DD On-Demand Anodyne DRD4 40 31 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne GRIN2B 36 48 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne PREP 37 42 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne LGMN 49 36 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne EPHX2 21 40 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne SLC12A5 44 33 O=C(NCc1cc2n(n1)CCCC2)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880617342 GF On-Demand Anodyne TMPRSS11D 51 38 CO[C@@](C)(CO)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880617349 DD On-Demand Anodyne GABRA1 15 49 CO[C@@](C)(CO)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880617349 DD On-Demand Anodyne MPO 50 36 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne ACE 23 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CELA1 15 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne ELANE 29 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne KLK3 75 35 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CTSB 65 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne PAPA1_CARPA 70 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CYSP_TRYCR 54 38 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CTSK 37 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CTSL 47 39 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne PREP 17 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CAPNS1 69 36 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne REN 42 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CTSS 26 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CAPN1 83 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CASP1 25 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne CAPN2 130 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne PLAU 15 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne TPSAB1 19 53 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne NPR 73 36 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne PSMB5 53 39 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne Q6PRC7_IXORI 48 39 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617364 FE On-Demand Anodyne SLC12A5 56 32 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne MME 36 43 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne KLK3 59 34 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne CTSB 52 39 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne PAPA1_CARPA 50 34 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne CTSK 34 42 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne CAPNS1 62 34 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne CAPN1 83 40 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne CAPN2 121 37 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne NPR 80 36 C[C@@H](NC(=O)c1c[nH]cc1C1CC1)C(=O)OCc1ccccc1 ZINC000880617366 DF On-Demand Anodyne Q6PRC7_IXORI 47 35 CC(=O)c1cccc(OCC(=O)NCc2cc3n(n2)CCCC3)c1 ZINC000880617378 EE On-Demand Anodyne DRD4 41 32 COc1ccc(-c2nnc(SCC(=O)NCc3cc4n(n3)CCCC4)o2)cc1 ZINC000880617388 GF On-Demand Anodyne GSK3A 15 41 O=C(COc1cccc(C(F)(F)F)c1)NCc1cc2n(n1)CCCC2 ZINC000880617407 FF On-Demand Anodyne PDS 45 42 O=C(NCc1cc2n(n1)CCCC2)c1cnc(-c2ncccn2)s1 ZINC000880617423 EE On-Demand Anodyne NAMPT 20 43 CN(C)[C@@H](Cc1ccccc1)C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617426 EE On-Demand Anodyne GPR142 52 33 O=C(NCc1cc2n(n1)CCCC2)c1ccc(S(=O)(=O)C(F)(F)F)cc1 ZINC000880617435 GE On-Demand Anodyne SFRP1 53 33 O=C(NCc1cc2n(n1)CCCC2)c1ccc(S(=O)(=O)C(F)(F)F)cc1 ZINC000880617435 GE On-Demand Anodyne NAMPT 47 42 CN(C)[C@@H]1C[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880617455 DF On-Demand Anodyne MTNR1A 24 46 CN(C)[C@@H]1C[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880617455 DF On-Demand Anodyne MTNR1B 26 46 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](N(C)C)C1)C2 ZINC000880617485 DE On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](N(C)C)C1)C2 ZINC000880617485 DE On-Demand Anodyne MTNR1A 41 44 CS(=O)(=O)C1CCC(C(=O)NCCCc2c(Cl)cccc2Cl)CC1 ZINC000880617527 GH On-Demand Anodyne MTNR1A 30 47 CS(=O)(=O)C1CCC(C(=O)NCCCc2c(Cl)cccc2Cl)CC1 ZINC000880617527 GH On-Demand Anodyne MTNR1B 25 47 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne ACE 31 43 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne MME 63 44 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne ANPEP 56 34 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CASP3 18 45 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne KLK3 79 37 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CTSB 72 44 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne PAPA1_CARPA 75 37 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CYSP_TRYCR 48 38 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CTSK 36 44 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CTSL 40 44 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CAPNS1 74 37 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne HLA-DRB1 52 34 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CTSS 26 44 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CAPN1 96 43 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CASP1 26 41 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne CAPN2 131 40 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne NPR 86 40 Cc1coc(C(=O)N[C@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617543 CE On-Demand Anodyne PSMB5 52 40 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne ACE 31 43 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne MME 63 44 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne ANPEP 56 34 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CASP3 18 45 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne KLK3 79 37 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CTSB 72 44 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne PAPA1_CARPA 75 37 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CYSP_TRYCR 48 38 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CTSK 36 44 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CTSL 40 44 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CAPNS1 74 37 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne HLA-DRB1 52 34 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CTSS 26 44 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CAPN1 96 43 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CASP1 26 41 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne CAPN2 131 40 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne NPR 86 40 Cc1coc(C(=O)N[C@@H](C)C(=O)OCc2ccccc2)c1 ZINC000880617546 CE On-Demand Anodyne PSMB5 52 40 O=C(COc1ccc2ccc(=O)oc2c1)NCc1cc2n(n1)CCCC2 ZINC000880617561 FE On-Demand Anodyne BCHE 16 42 Cc1cnc(Cl)c(C(=O)NC[C@@H]2C[C@H](N(C)C)C2)c1 ZINC000880617570 CE On-Demand Anodyne CACNA1I 50 35 O=C(NCc1cc2n(n1)CCCC2)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880617576 FE On-Demand Anodyne NAMPT 41 41 COc1ccc2c(C)c(CCC(=O)NCc3cc4n(n3)CCCC4)c(=O)oc2c1 ZINC000880617583 GF On-Demand Anodyne MAOB 27 41 Cc1cnc(CCNC(=O)CC[C@H]2CCc3ccccc32)c(C)c1 ZINC000880617594 DH On-Demand Anodyne NQO2 20 42 Cc1cnc(CCNC(=O)CC[C@@H]2CCc3ccccc32)c(C)c1 ZINC000880617597 DH On-Demand Anodyne NQO2 20 42 CC[C@@H](NC(=O)c1cn(C[C@@H]2CNC(=O)O2)nn1)c1ccccc1F ZINC000880617600 ED On-Demand Anodyne CTSA 44 34 CC[C@@H](NC(=O)c1cn(C[C@H]2CNC(=O)O2)nn1)c1ccccc1F ZINC000880617601 ED On-Demand Anodyne CTSA 44 34 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880617606 FE On-Demand Anodyne CACNA1I 40 31 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCc2cc3n(n2)CCCC3)C1 ZINC000880617606 FE On-Demand Anodyne GPR119 29 40 CC(=O)c1ccc(N2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c(F)c1 ZINC000880617617 GF On-Demand Anodyne NPY2R 55 37 O=C(Nc1cc2cc[nH]c2cn1)c1ccc(CN2CCOCC2)o1 ZINC000880617632 EE On-Demand Anodyne PRKCQ 15 42 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)NCc1cc2n(n1)CCCC2 ZINC000880617638 FG On-Demand Anodyne P2RX7 17 42 COC(=O)[C@@H]1CN(C(=O)c2cnc3cc[nH]c3c2)C[C@H]1c1ccc(Cl)cc1 ZINC000880617644 GG On-Demand Anodyne SLC6A4 19 48 COC(=O)[C@@H]1CN(C(=O)c2cnc3cc[nH]c3c2)C[C@H]1c1ccc(Cl)cc1 ZINC000880617644 GG On-Demand Anodyne SLC6A3 31 48 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne MME 23 42 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne KLK3 55 34 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne CYSP_TRYCR 47 35 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne CAPNS1 58 32 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne CAPN1 64 45 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne CAPN2 95 45 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne NPR 80 37 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne PSMB8 55 41 C[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617645 FD On-Demand Anodyne SLC12A5 42 32 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne MME 23 42 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne KLK3 55 34 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne CYSP_TRYCR 47 35 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne CAPNS1 58 32 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne CAPN1 64 45 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne CAPN2 95 45 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne NPR 80 37 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne PSMB8 55 41 C[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)C(=O)OCc1ccccc1 ZINC000880617646 FD On-Demand Anodyne SLC12A5 42 32 COC(=O)[C@@H]1CN(C(=O)c2cncc3[nH]ccc23)C[C@H]1c1ccc(Cl)cc1 ZINC000880617651 GG On-Demand Anodyne SLC6A3 23 45 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne ACE 42 41 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne MME 40 42 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CASP3 23 40 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne KLK3 83 35 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CTSB 62 38 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne PAPA1_CARPA 66 35 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CYSP_TRYCR 56 38 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CTSL 52 39 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CAPNS1 69 35 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne REN 16 40 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne LGMN 43 36 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne FURIN 55 36 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CAPN1 86 39 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne CAPN2 125 38 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne KLK5 40 35 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne NPR 76 34 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne XIAP 40 37 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne PSMB5 49 38 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne POLG_WNV 41 30 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne BIRC2 36 41 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne Q6PRC7_IXORI 54 40 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OCc1ccccc1 ZINC000880617668 GF On-Demand Anodyne SLC12A5 65 36 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@](C)(CO)OC)C2 ZINC000880617680 DD On-Demand Anodyne NQO2 31 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@](C)(CO)OC)C2 ZINC000880617680 DD On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@](C)(CO)OC)C2 ZINC000880617680 DD On-Demand Anodyne MTNR1B 37 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@](C)(CO)OC)C2 ZINC000880617681 DD On-Demand Anodyne NQO2 31 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@](C)(CO)OC)C2 ZINC000880617681 DD On-Demand Anodyne MTNR1A 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@](C)(CO)OC)C2 ZINC000880617681 DD On-Demand Anodyne MTNR1B 37 43 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617682 DH On-Demand Mild HRH3 16 46 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617682 DH On-Demand Mild PREP 23 40 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617682 DH On-Demand Mild L3MBTL3 40 36 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617682 DH On-Demand Mild MAP3K12 29 43 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617683 DH On-Demand Mild HRH3 16 46 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617683 DH On-Demand Mild PREP 23 40 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617683 DH On-Demand Mild L3MBTL3 40 36 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3ccc(C)cn3)cc2)C1 ZINC000880617683 DH On-Demand Mild MAP3K12 29 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000880617684 GD On-Demand Anodyne PAPA1_CARPA 36 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000880617685 GD On-Demand Anodyne PAPA1_CARPA 36 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000880617686 GD On-Demand Anodyne PAPA1_CARPA 36 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000880617687 GD On-Demand Anodyne PAPA1_CARPA 36 43 COc1ccc(N2CCC(NC(=O)Nc3c4c(nn3C)CCCC4)CC2)cc1 ZINC000880617706 GG On-Demand Clean EPHX2 25 43 C#C[C@@H]1CCCN(C(=O)c2ccc3c(O)ncnc3c2)C1 ZINC000880617720 CD On-Demand Mild L3MBTL3 53 36 C#C[C@@H]1CCCN(C(=O)c2ccc3c(O)ncnc3c2)C1 ZINC000880617720 CD On-Demand Mild HPGD 48 39 C#C[C@H]1CCCN(C(=O)c2ccc3c(O)ncnc3c2)C1 ZINC000880617721 CD On-Demand Mild L3MBTL3 53 36 C#C[C@H]1CCCN(C(=O)c2ccc3c(O)ncnc3c2)C1 ZINC000880617721 CD On-Demand Mild HPGD 48 39 Cn1nnc(C(=O)NCCCc2c(Cl)cccc2Cl)n1 ZINC000880617745 DD On-Demand Anodyne HTR2A 25 40 Cn1nnc(C(=O)NCCCc2c(Cl)cccc2Cl)n1 ZINC000880617745 DD On-Demand Anodyne HTR2C 28 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617758 FF On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617758 FF On-Demand Anodyne CCKAR 53 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617758 FF On-Demand Anodyne CTSL 24 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617758 FF On-Demand Anodyne CTSS 16 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617758 FF On-Demand Anodyne FPR1 44 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617764 FF On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617764 FF On-Demand Anodyne CCKAR 53 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617764 FF On-Demand Anodyne CTSL 24 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617764 FF On-Demand Anodyne CTSS 16 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(C)c1OC ZINC000880617764 FF On-Demand Anodyne FPR1 44 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ncc(C)cc1C ZINC000880617772 FE On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ncc(C)cc1C ZINC000880617773 FE On-Demand Anodyne PAPA1_CARPA 39 42 C#C[C@H]1CCCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880617798 DG On-Demand Mild L3MBTL3 48 34 C#C[C@@H]1CCCN(C(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880617800 DG On-Demand Mild L3MBTL3 48 34 CN(C)[C@@H]1C[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880617828 DD On-Demand Anodyne GABRA1 18 47 CN(C)[C@@H]1C[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880617828 DD On-Demand Anodyne MPO 49 35 CN(C)[C@@H]1C[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880617828 DD On-Demand Anodyne GABRA2 15 47 C=CC(C)(C)CC(=O)N1CCC(c2ccc3cccnc3n2)CC1 ZINC000880617864 DH On-Demand Mild ETHR 44 31 COC(=O)Nc1cccc(NC(=O)Nc2c3c(nn2C)CCCC3)c1 ZINC000880617867 EG On-Demand Anodyne KCNK3 46 33 C=CCCCCCNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880617927 DG On-Demand Mild PLD1 43 38 C=CCCCCCNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880617927 DG On-Demand Mild HDAC9 23 44 C=CCCCCCNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880617928 DG On-Demand Mild PLD1 43 38 C=CCCCCCNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880617928 DG On-Demand Mild HDAC9 23 44 O=C1NCC[C@H]1CC(=O)N1CCC(c2ccc3cccnc3n2)CC1 ZINC000880617929 ED On-Demand Anodyne ETHR 44 31 O=C1NCC[C@@H]1CC(=O)N1CCC(c2ccc3cccnc3n2)CC1 ZINC000880617931 ED On-Demand Anodyne ETHR 44 31 C=CCCCCCNC(=O)[C@H]1CC[C@@H](C(N)=O)N1Cc1ccccc1 ZINC000880617938 EE On-Demand Mild F2 19 40 Cn1nc2c(c1NC(=O)NCC[C@H]1CCN(C(=O)OC(C)(C)C)C1)CCCC2 ZINC000880617975 GG On-Demand Anodyne GPR119 22 40 Cn1nc2c(c1NC(=O)NCC[C@@H]1CCN(C(=O)OC(C)(C)C)C1)CCCC2 ZINC000880617977 GG On-Demand Anodyne GPR119 22 40 C=CCCCCCNC(=O)c1coc(-c2ccccn2)n1 ZINC000880617995 CG On-Demand Mild TBXA2R 26 46 O=C1NCC[C@H]1CC(=O)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618047 FF On-Demand Anodyne HTR2A 18 56 O=C1NCC[C@@H]1CC(=O)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618048 FF On-Demand Anodyne HTR2A 18 56 C#C[C@@H]1CCCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880618053 EG On-Demand Mild SFRP1 57 32 C#C[C@@H]1CCCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880618053 EG On-Demand Mild WNT3 50 30 C#C[C@H]1CCCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880618054 EG On-Demand Mild SFRP1 57 32 C#C[C@H]1CCCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880618054 EG On-Demand Mild WNT3 50 30 C=CCCCCCNC(=O)c1cccn2nccc12 ZINC000880618063 CF On-Demand Mild POLR1A 40 33 CO[C@@](C)(CO)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880618186 CE On-Demand Anodyne NQO2 21 43 CO[C@@](C)(CO)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880618186 CE On-Demand Anodyne MTNR1B 22 40 CO[C@@](C)(CO)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880618189 CE On-Demand Anodyne NQO2 21 43 CO[C@@](C)(CO)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880618189 CE On-Demand Anodyne MTNR1B 22 40 Cc1c(Br)cccc1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880618221 GF On-Demand Anodyne P2RX7 27 42 Cc1c(Br)cccc1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880618221 GF On-Demand Anodyne MTNR1A 18 40 Cc1c(Br)cccc1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880618221 GF On-Demand Anodyne EPHX2 15 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ncc(C)cc1C)C2 ZINC000880618224 EG On-Demand Anodyne NQO2 40 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ncc(C)cc1C)C2 ZINC000880618224 EG On-Demand Anodyne MTNR1A 74 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ncc(C)cc1C)C2 ZINC000880618224 EG On-Demand Anodyne MTNR1B 63 41 Cc1cnc(CCNC(=O)C2CCC(S(C)(=O)=O)CC2)c(C)c1 ZINC000880618254 ED On-Demand Anodyne EPHX2 20 42 C=CCCCCCNC(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880618346 EH On-Demand Mild DRD2 21 41 C=CCCCCCNC(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880618346 EH On-Demand Mild DRD3 42 41 C#CCOc1cc(F)ccc1NC(=O)Nc1c2c(nn1C)CCCC2 ZINC000880618385 EG On-Demand Mild Q9FYV8_MAIZE 23 40 Cn1nnc(C(=O)NCC2(c3cccc(OC(F)(F)F)c3)CCC2)n1 ZINC000880618392 FD On-Demand Anodyne SOAT1 15 42 O=C(NCc1nc([C@H]2CCCO2)n[nH]1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880618394 FF On-Demand Anodyne PDE4D 15 42 O=C(NCc1nc([C@@H]2CCCO2)n[nH]1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880618397 FF On-Demand Anodyne PDE4D 15 42 Cn1nc2c(c1NC(=O)N1CCC[C@@H]1C[C@H](O)c1ccccc1)CCCC2 ZINC000880618420 FG On-Demand Anodyne Q8WSF8_APLCA 17 45 Cn1nc2c(c1NC(=O)N1CCC[C@H]1C[C@H](O)c1ccccc1)CCCC2 ZINC000880618421 FG On-Demand Anodyne Q8WSF8_APLCA 17 45 Cn1nc2c(c1NC(=O)N1CCC[C@H]1C[C@@H](O)c1ccccc1)CCCC2 ZINC000880618422 FG On-Demand Anodyne Q8WSF8_APLCA 17 45 Cn1nc2c(c1NC(=O)N1CCC[C@@H]1C[C@@H](O)c1ccccc1)CCCC2 ZINC000880618424 FG On-Demand Anodyne Q8WSF8_APLCA 17 45 Cc1c(Br)cccc1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880618456 GF On-Demand Anodyne P2RX7 34 46 Cn1nc2c(c1NC(=O)N1CC[C@H](CNC(=O)OC(C)(C)C)C1)CCCC2 ZINC000880618475 GF On-Demand Anodyne CACNA1I 50 35 Cn1nc2c(c1NC(=O)N1CC[C@@H](CNC(=O)OC(C)(C)C)C1)CCCC2 ZINC000880618476 GF On-Demand Anodyne CACNA1I 50 35 Cn1nc2c(c1NC(=O)N1CCN(Cc3ccc(Cl)nc3)CC1)CCCC2 ZINC000880618602 GF On-Demand Anodyne FAAH 17 42 Cn1nc2c(c1NC(=O)N1CCN(Cc3ccc(Cl)nc3)CC1)CCCC2 ZINC000880618602 GF On-Demand Anodyne NACHRBETA2 40 33 Cc1c(Br)cccc1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880618618 FF On-Demand Anodyne P2RX7 37 42 Cc1c(Br)cccc1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880618618 FF On-Demand Anodyne EPHX2 17 43 Cc1c(Br)cccc1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880618622 FF On-Demand Anodyne P2RX7 37 42 Cc1c(Br)cccc1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880618622 FF On-Demand Anodyne EPHX2 17 43 C#C[C@H]1CCCN(C(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880618685 EG On-Demand Mild FKBP1A 56 42 C#C[C@H]1CCCN(C(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880618685 EG On-Demand Mild PREP 51 42 C#C[C@@H]1CCCN(C(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880618686 EG On-Demand Mild FKBP1A 56 42 C#C[C@@H]1CCCN(C(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880618686 EG On-Demand Mild PREP 51 42 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618691 EE On-Demand Anodyne PAPA1_CARPA 43 32 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618691 EE On-Demand Anodyne CAPNS1 57 32 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618691 EE On-Demand Anodyne CAPN1 60 36 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618691 EE On-Demand Anodyne CAPN2 84 33 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618692 EE On-Demand Anodyne PAPA1_CARPA 43 32 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618692 EE On-Demand Anodyne CAPNS1 57 32 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618692 EE On-Demand Anodyne CAPN1 60 36 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](C)C(=O)OCc1ccccc1 ZINC000880618692 EE On-Demand Anodyne CAPN2 84 33 C[C@@H](NC(=O)[C@H]1c2c[nH]nc2CC[C@H]1C)C(=O)OCc1ccccc1 ZINC000880618693 EE On-Demand Anodyne PAPA1_CARPA 43 32 C[C@@H](NC(=O)[C@H]1c2c[nH]nc2CC[C@H]1C)C(=O)OCc1ccccc1 ZINC000880618693 EE On-Demand Anodyne CAPNS1 57 32 C[C@@H](NC(=O)[C@H]1c2c[nH]nc2CC[C@H]1C)C(=O)OCc1ccccc1 ZINC000880618693 EE On-Demand Anodyne CAPN1 60 36 C[C@@H](NC(=O)[C@H]1c2c[nH]nc2CC[C@H]1C)C(=O)OCc1ccccc1 ZINC000880618693 EE On-Demand Anodyne CAPN2 84 33 O=C([C@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618740 GG On-Demand Anodyne HTR2A 22 53 O=C([C@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618740 GG On-Demand Anodyne PRCP 44 32 O=C([C@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618740 GG On-Demand Anodyne ADAMTS4 49 33 O=C([C@@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618741 GG On-Demand Anodyne HTR2A 22 53 O=C([C@@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618741 GG On-Demand Anodyne PRCP 44 32 O=C([C@@H]1CCc2nncn2CC1)N1CCC(CCc2ccc(F)cc2F)CC1 ZINC000880618741 GG On-Demand Anodyne ADAMTS4 49 33 Cn1nnc(C(=O)N2CCC(CCc3ccc(F)cc3F)CC2)n1 ZINC000880618770 ED On-Demand Anodyne HTR2A 28 63 Cn1nnc(C(=O)N2CCC(CCc3ccc(F)cc3F)CC2)n1 ZINC000880618770 ED On-Demand Anodyne PRCP 41 32 Cn1nnc(C(=O)N2CCC(CCc3ccc(F)cc3F)CC2)n1 ZINC000880618770 ED On-Demand Anodyne ADAMTS4 44 38 Cn1nc2c(c1NC(=O)N(CCc1ccccc1)C1CC1)CCCC2 ZINC000880618772 EH On-Demand Anodyne MBTPS1 41 29 C=CCCCCCNC(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880618784 CG On-Demand Mild HDAC3 16 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C1CC1)[C@H]1CCCCO1 ZINC000880618832 FE On-Demand Anodyne REN 43 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C1CC1)[C@@H]1CCCCO1 ZINC000880618833 FE On-Demand Anodyne REN 43 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C1CC1)[C@@H]1CCCCO1 ZINC000880618834 FE On-Demand Anodyne REN 43 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C1CC1)[C@H]1CCCCO1 ZINC000880618835 FE On-Demand Anodyne REN 43 39 C#C[C@H]1CCCN(C(=O)c2cc(C(F)(F)F)ccn2)C1 ZINC000880618845 CF On-Demand Mild MAP3K12 47 47 C#C[C@@H]1CCCN(C(=O)c2cc(C(F)(F)F)ccn2)C1 ZINC000880618846 CF On-Demand Mild MAP3K12 47 47 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3CCc4ccccc4NC3=O)cc2)N1 ZINC000880618854 FE On-Demand Anodyne PYGM 21 51 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCc4ccccc4NC3=O)cc2)N1 ZINC000880618855 FE On-Demand Anodyne PYGM 21 51 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3CCc4ccccc4NC3=O)cc2)N1 ZINC000880618856 FE On-Demand Anodyne PYGM 21 51 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCc4ccccc4NC3=O)cc2)N1 ZINC000880618857 FE On-Demand Anodyne PYGM 21 51 Cn1nc2c(c1NC(=O)NCC1CCN(C(=O)OC(C)(C)C)CC1)CCCC2 ZINC000880618894 GG On-Demand Anodyne CACNA1I 44 35 Cc1c(Br)cccc1CNC(=O)CN1CCCCS1(=O)=O ZINC000880618899 GD On-Demand Anodyne P2RX7 18 42 CSc1nccnc1C(=O)Nc1ccccc1OCCC(C)C ZINC000880618973 EH On-Demand Anodyne MAP1 49 39 Cn1nc2c(c1NC(=O)NC[C@@H](O)COc1cccc(F)c1)CCCC2 ZINC000880618978 FD On-Demand Anodyne ADRB1 45 36 Cn1nc2c(c1NC(=O)NC[C@@H](O)COc1cccc(F)c1)CCCC2 ZINC000880618978 FD On-Demand Anodyne ACOX1 45 33 Cn1nc2c(c1NC(=O)NC[C@H](O)COc1cccc(F)c1)CCCC2 ZINC000880618979 FD On-Demand Anodyne ADRB1 45 36 Cn1nc2c(c1NC(=O)NC[C@H](O)COc1cccc(F)c1)CCCC2 ZINC000880618979 FD On-Demand Anodyne ACOX1 45 33 C#C[C@@H]1CCCN(C(=O)c2coc(-c3ccccn3)n2)C1 ZINC000880618984 CE On-Demand Mild MAP3K12 29 40 C#C[C@H]1CCCN(C(=O)c2coc(-c3ccccn3)n2)C1 ZINC000880618985 CE On-Demand Mild MAP3K12 29 40 Cn1nc2c(c1C(=O)N[C@H]1CCc3ccccc3NC1=O)CSCC2 ZINC000880619025 FD On-Demand Anodyne PYGM 29 44 Cn1nc2c(c1C(=O)N[C@@H]1CCc3ccccc3NC1=O)CSCC2 ZINC000880619026 FD On-Demand Anodyne PYGM 29 44 C#C[C@H]1CCCN(C(=O)CN(C(C)=O)c2ccccc2)C1 ZINC000880619027 CD On-Demand Mild PREP 43 35 C#C[C@@H]1CCCN(C(=O)CN(C(C)=O)c2ccccc2)C1 ZINC000880619028 CD On-Demand Mild PREP 43 35 C#C[C@@H]1CCCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880619031 CF On-Demand Mild MTNR1B 15 46 C#C[C@@H]1CCCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880619032 CF On-Demand Mild MTNR1B 15 46 C#C[C@H]1CCCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880619033 CF On-Demand Mild MTNR1B 15 46 C#C[C@H]1CCCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880619034 CF On-Demand Mild MTNR1B 15 46 C#C[C@@H]1CCCN(C(=O)[C@H](CNC(=O)OC(C)(C)C)OC)C1 ZINC000880619039 DD On-Demand Mild SSTR2 42 35 C#C[C@H]1CCCN(C(=O)[C@H](CNC(=O)OC(C)(C)C)OC)C1 ZINC000880619040 DD On-Demand Mild SSTR2 42 35 C#C[C@H]1CCCN(C(=O)[C@@H]2C[C@]2(C)c2ccccc2)C1 ZINC000880619132 CF On-Demand Mild PREP 43 38 C#C[C@@H]1CCCN(C(=O)[C@@H]2C[C@]2(C)c2ccccc2)C1 ZINC000880619133 CF On-Demand Mild PREP 43 38 Cn1nc2c(c1NC(=O)NCc1ccccc1N1CCOCC1)CCCC2 ZINC000880619159 FE On-Demand Anodyne AVPR2 22 42 Cn1nc2c(c1NC(=O)NCc1ccccc1N1CCOCC1)CCCC2 ZINC000880619159 FE On-Demand Anodyne SCN10A 15 44 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)C1 ZINC000880619162 DH On-Demand Mild L3MBTL3 43 35 C#C[C@H]1CCCN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)C1 ZINC000880619162 DH On-Demand Mild MAP3K12 32 44 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)C1 ZINC000880619163 DH On-Demand Mild L3MBTL3 43 35 C#C[C@@H]1CCCN(C(=O)c2ccc(Oc3cc(C)ccn3)cc2)C1 ZINC000880619163 DH On-Demand Mild MAP3K12 32 44 Cn1nc2c(c1NC(=O)N1CCC(CNC(=O)OC(C)(C)C)CC1)CCCC2 ZINC000880619178 GG On-Demand Anodyne CACNA1I 41 32 Cc1ccc(N2CCCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)cc1 ZINC000880619214 FG On-Demand Anodyne SLC27A1 22 42 Cn1nc2c(c1NC(=O)N1CCC[C@@H](CNC(=O)OC(C)(C)C)C1)CCCC2 ZINC000880619322 GG On-Demand Anodyne CACNA1I 41 32 Cn1nc2c(c1NC(=O)N1CCC[C@H](CNC(=O)OC(C)(C)C)C1)CCCC2 ZINC000880619323 GG On-Demand Anodyne CACNA1I 41 32 Cc1coc(C(=O)N[C@@H]2CCc3ccccc3NC2=O)c1 ZINC000880619333 CE On-Demand Anodyne PYGM 22 53 Cc1coc(C(=O)N[C@H]2CCc3ccccc3NC2=O)c1 ZINC000880619334 CE On-Demand Anodyne PYGM 22 53 C#C[C@H]1CCCN(C(=O)c2ccnc(N3CCN(C(=O)OC(C)(C)C)CC3)c2)C1 ZINC000880619335 GF On-Demand Mild GPR119 41 46 C#C[C@@H]1CCCN(C(=O)c2ccnc(N3CCN(C(=O)OC(C)(C)C)CC3)c2)C1 ZINC000880619336 GF On-Demand Mild GPR119 41 46 COC[C@@H](CC(C)(C)C)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880619362 EF On-Demand Anodyne KCNQ2 41 33 Cn1nc2c(c1NC(=O)NCc1ccc(N3CCOCC3)cc1)CCCC2 ZINC000880619363 FE On-Demand Clean MTOR 49 41 C#C[C@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880619370 CF On-Demand Mild MAP3K12 29 41 C#C[C@@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880619372 CF On-Demand Mild MAP3K12 29 41 Cc1c(Br)cccc1CNC(=O)c1nnn(C)n1 ZINC000880619373 DD On-Demand Anodyne P2RX7 16 40 C#C[C@@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880619376 ED On-Demand Mild PREP 109 44 C#C[C@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880619380 ED On-Demand Mild PREP 109 44 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCN2C[C@H](O)C[C@H]2C1 ZINC000880619385 GD On-Demand Anodyne PREP 51 48 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCN2C[C@H](O)C[C@H]2C1 ZINC000880619385 GD On-Demand Anodyne SLC12A5 45 34 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCN2C[C@H](O)C[C@H]2C1 ZINC000880619385 GD On-Demand Anodyne Q9NAW4_PLAFA 28 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](N(C)C)C1 ZINC000880619386 ED On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](N(C)C)C1 ZINC000880619390 ED On-Demand Anodyne PAPA1_CARPA 37 45 Cn1nc2c(c1NC(=O)NCc1ccc(Cl)nc1)CCCC2 ZINC000880619412 DF On-Demand Anodyne NAMPT 22 45 C#C[C@H]1CCCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880619565 CG On-Demand Mild PREP 52 40 C#C[C@@H]1CCCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880619566 CG On-Demand Mild PREP 52 40 C#C[C@H]1CCCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880619567 CG On-Demand Mild PREP 52 40 C#C[C@@H]1CCCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880619568 CG On-Demand Mild PREP 52 40 C#C[C@H]1CCCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880619602 CE On-Demand Mild L3MBTL3 56 40 C#C[C@@H]1CCCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880619603 CE On-Demand Mild L3MBTL3 56 40 C#C[C@@H]1CCCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880619604 CE On-Demand Mild L3MBTL3 56 40 C#C[C@H]1CCCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880619605 CE On-Demand Mild L3MBTL3 56 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1C[C@H]2C=C[C@H]1C2 ZINC000880619609 FF On-Demand Anodyne PAPA1_CARPA 37 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1C[C@H]2C=C[C@H]1C2 ZINC000880619610 FF On-Demand Anodyne PAPA1_CARPA 37 42 Cc1c(Br)cccc1CNC(=O)COC1CC1 ZINC000880619652 CF On-Demand Anodyne P2RX7 24 42 C[C@@H](CNC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OC(C)(C)C ZINC000880619703 FE On-Demand Anodyne SSTR2 43 31 C[C@@H](CNC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OC(C)(C)C ZINC000880619703 FE On-Demand Anodyne KCNQ2 61 35 C[C@H](CNC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OC(C)(C)C ZINC000880619704 FE On-Demand Anodyne SSTR2 43 31 C[C@H](CNC(=O)Cc1ccccc1N1CCCC1=O)C(=O)OC(C)(C)C ZINC000880619704 FE On-Demand Anodyne KCNQ2 61 35 C[C@@H](CNC(=O)c1cccn2nccc12)C(=O)OC(C)(C)C ZINC000880619802 DE On-Demand Anodyne TYK2 17 41 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H](OC4CCC4)C3)cc2)N1 ZINC000880619872 EF On-Demand Anodyne L3MBTL3 42 37 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H](OC4CCC4)C3)cc2)N1 ZINC000880619873 EF On-Demand Anodyne L3MBTL3 42 37 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@H](OC4CCC4)C3)cc2)N1 ZINC000880619874 EF On-Demand Anodyne L3MBTL3 42 37 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@H](OC4CCC4)C3)cc2)N1 ZINC000880619875 EF On-Demand Anodyne L3MBTL3 42 37 Cn1nc2c(c1NC(=O)NCc1cc(Cl)ccn1)CCCC2 ZINC000880619912 DF On-Demand Anodyne HRP1_PLAFA 53 32 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@H](OC2CCC2)C1 ZINC000880619915 GI On-Demand Anodyne RBP4 52 34 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@@H](OC2CCC2)C1 ZINC000880619916 GI On-Demand Anodyne RBP4 52 34 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H](OC3CCC3)C2)N1Cc1ccccc1 ZINC000880619949 GE On-Demand Anodyne PREP 85 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H](OC3CCC3)C2)N1Cc1ccccc1 ZINC000880619950 GE On-Demand Anodyne PREP 85 43 C[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C(=O)OC(C)(C)C ZINC000880620051 EF On-Demand Anodyne MPO 47 34 Cn1nnc2c1CC[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C2 ZINC000880620077 FE On-Demand Anodyne UTS2R 22 41 Cn1nnc2c1CC[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C2 ZINC000880620077 FE On-Demand Anodyne EZH2 40 36 Cn1nnc2c1CC[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C2 ZINC000880620078 FE On-Demand Anodyne UTS2R 22 41 Cn1nnc2c1CC[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C2 ZINC000880620078 FE On-Demand Anodyne EZH2 40 36 Cn1nc2c(c1NC(=O)NC[C@H]1CCN(C(=O)OC(C)(C)C)C1)CCCC2 ZINC000880620079 GF On-Demand Anodyne CACNA1I 47 35 Cn1nc2c(c1NC(=O)NC[C@@H]1CCN(C(=O)OC(C)(C)C)C1)CCCC2 ZINC000880620080 GF On-Demand Anodyne CACNA1I 47 35 C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)Nc1c2c(nn1C)CCCC2 ZINC000880620180 FG On-Demand Anodyne CCR3 56 38 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1c2c(nn1C)CCCC2 ZINC000880620181 FG On-Demand Anodyne CCR3 56 38 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620239 EF On-Demand Anodyne NQO2 28 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620239 EF On-Demand Anodyne MTNR1A 41 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620239 EF On-Demand Anodyne MTNR1B 36 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620240 EF On-Demand Anodyne NQO2 28 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620240 EF On-Demand Anodyne MTNR1A 41 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)C(=O)OC(C)(C)C)C2 ZINC000880620240 EF On-Demand Anodyne MTNR1B 36 47 Cn1nnc2c1CC[C@@H](NC(=O)c1cc3cc(F)ccc3[nH]c1=O)C2 ZINC000880620253 ED On-Demand Anodyne PLD2 45 38 Cn1nnc2c1CC[C@H](NC(=O)c1cc3cc(F)ccc3[nH]c1=O)C2 ZINC000880620254 ED On-Demand Anodyne PLD2 45 38 Cn1cnnc1N1CCN(C(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1 ZINC000880620312 FC On-Demand Anodyne HRH4 18 49 Cn1nc2c(c1NC(=O)NCCNc1ccccc1)CCCC2 ZINC000880620336 DF On-Demand Anodyne ACHE 37 42 Cn1nc2c(c1NC(=O)NCCNc1ccccc1)CCCC2 ZINC000880620336 DF On-Demand Anodyne BCHE 59 42 Cn1cnnc1N1CCN(C(=O)CC[C@@H]2CCc3ccccc32)CC1 ZINC000880620461 ED On-Demand Anodyne SSTR1 45 42 Cn1cnnc1N1CCN(C(=O)CC[C@H]2CCc3ccccc32)CC1 ZINC000880620462 ED On-Demand Anodyne SSTR1 45 42 Cn1nc2c(c1NC(=O)Nc1cccc(C(C)(C)O)c1)CCCC2 ZINC000880620472 EG On-Demand Anodyne IMDH_CRYPV 40 32 Cc1cnc(Cl)c(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880620478 GF On-Demand Anodyne CNR2 30 41 Cc1cnc(Cl)c(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880620478 GF On-Demand Anodyne SSTR5 42 39 Cc1cnc(Cl)c(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880620478 GF On-Demand Anodyne EPHX2 41 50 Cc1cnc(Cl)c(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880620478 GF On-Demand Anodyne TGM2 52 44 Cc1cnc(Cl)c(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880620478 GF On-Demand Anodyne SFRP1 63 39 O=C(N[C@H]1c2ccccc2C[C@@H]1O)[C@H]1CCc2nncn2CC1 ZINC000880620480 DD On-Demand Anodyne PLM2_PLAFA 52 35 O=C(N[C@H]1c2ccccc2C[C@@H]1O)[C@@H]1CCc2nncn2CC1 ZINC000880620481 DD On-Demand Anodyne PLM2_PLAFA 52 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cc(F)c(F)cc2C1 ZINC000880620493 FF On-Demand Anodyne CTSK 15 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cc(F)c(F)cc2C1 ZINC000880620494 FF On-Demand Anodyne CTSK 15 43 Cn1nc2c(c1NC(=O)NNC(=O)c1ccc(Cl)cc1F)CCCC2 ZINC000880620501 FF On-Demand Reactive CNR1 51 31 O=C(C[C@H]1CCNC1=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620502 CC On-Demand Anodyne PLM1_PLAFA 46 41 O=C(C[C@H]1CCNC1=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620502 CC On-Demand Anodyne PLM2_PLAFA 36 41 Cn1nc2c(c1NC(=O)NNC(=O)Cc1cccc3ccccc13)CCCC2 ZINC000880620507 GF On-Demand Reactive BCHE 44 33 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(=O)Nc3ccccc3C2)N1Cc1ccccc1 ZINC000880620519 GD On-Demand Anodyne CALCRL 49 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](OC(C)(C)C)C1 ZINC000880620528 FE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](OC(C)(C)C)C1 ZINC000880620529 FE On-Demand Anodyne PAPA1_CARPA 35 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2Cc3cc(F)c(F)cc3C2)N1Cc1ccccc1 ZINC000880620547 GE On-Demand Anodyne SIGMAR1 16 41 CC1(C)CC[C@@H](CC(=O)N2CC(=O)Nc3ccccc3C2)OC1 ZINC000880620554 DF On-Demand Anodyne CALCRL 46 37 O=C(C[C@@H]1C[C@H]1C1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620559 FE On-Demand Anodyne SIGMAR1 15 46 O=C(C[C@@H]1C[C@H]1C1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620559 FE On-Demand Anodyne EPHX2 29 53 O=C(C[C@@H]1C[C@H]1C1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620559 FE On-Demand Anodyne TGM2 84 45 O=C(C[C@@H]1C[C@H]1C1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620559 FE On-Demand Anodyne F13A1 80 43 O=C(C[C@@H]1C[C@H]1C1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620559 FE On-Demand Anodyne SFRP1 41 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CTSD 17 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne PGC 54 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne PAPA1_CARPA 46 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CYSP_TRYCR 34 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CTSK 24 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CTSL 20 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CAPNS1 51 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne REN 73 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CAPN1 34 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne CAPN2 47 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620563 FE On-Demand Anodyne FPR1 56 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CTSD 17 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne PGC 54 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne PAPA1_CARPA 46 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CYSP_TRYCR 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CTSL 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CAPNS1 51 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne REN 73 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CAPN1 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne CAPN2 47 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620564 FE On-Demand Anodyne FPR1 56 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CTSD 17 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne PGC 54 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne PAPA1_CARPA 46 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CYSP_TRYCR 34 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CTSK 24 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CTSL 20 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CAPNS1 51 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne REN 73 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CAPN1 34 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne CAPN2 47 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880620565 FE On-Demand Anodyne FPR1 56 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CTSD 17 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne PGC 54 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne PAPA1_CARPA 46 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CYSP_TRYCR 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CTSL 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CAPNS1 51 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne REN 73 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CAPN1 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne CAPN2 47 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880620566 FE On-Demand Anodyne FPR1 56 43 C[C@@H](Cc1ccccn1)NC(=O)c1ncsc1C1CC1 ZINC000880620582 CF On-Demand Anodyne MAP1 104 38 C[C@H](Cc1ccccn1)NC(=O)c1ncsc1C1CC1 ZINC000880620583 CF On-Demand Anodyne MAP1 104 38 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ncsc1C1CC1 ZINC000880620598 GF On-Demand Anodyne EPHX2 20 52 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ncsc1C1CC1 ZINC000880620598 GF On-Demand Anodyne TGM2 54 44 CC1(C)CC[C@@H](CC(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)OC1 ZINC000880620603 GF On-Demand Anodyne EPHX2 34 47 CC1(C)CC[C@@H](CC(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)OC1 ZINC000880620603 GF On-Demand Anodyne TGM2 72 43 CC1(C)CC[C@@H](CC(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)OC1 ZINC000880620603 GF On-Demand Anodyne F13A1 64 41 CC1(C)CC[C@@H](CC(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)OC1 ZINC000880620603 GF On-Demand Anodyne SFRP1 45 39 C[C@@H](Cc1ccccn1)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880620638 EH On-Demand Anodyne PDE4D 20 40 C[C@H](Cc1ccccn1)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880620639 EH On-Demand Anodyne PDE4D 20 40 COc1ccc2c(c1)CN(C(=O)Cc1ccccc1N1CCCC1=O)C2 ZINC000880620703 FF On-Demand Anodyne DRD5 17 41 COc1ccc2c(c1)CN(C(=O)Cc1ccccc1N1CCCC1=O)C2 ZINC000880620703 FF On-Demand Anodyne HTR7 16 43 COc1ccc2c(c1)CN(C(=O)Cc1ccccc1N1CCCC1=O)C2 ZINC000880620703 FF On-Demand Anodyne MTNR1A 21 40 COc1ccc2c(c1)CN(C(=O)Cc1ccccc1N1CCCC1=O)C2 ZINC000880620703 FF On-Demand Anodyne EBP 41 34 COc1ccc2c(c1)CN(C(=O)Cc1ccccc1N1CCCC1=O)C2 ZINC000880620703 FF On-Demand Anodyne AKR1C3 20 43 C[C@@H](Cc1ccccn1)NC(=O)COC1CC1 ZINC000880620722 BD On-Demand Anodyne TIMP3 70 38 C[C@H](Cc1ccccn1)NC(=O)COC1CC1 ZINC000880620723 BD On-Demand Anodyne TIMP3 70 38 O=C(C[C@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620729 FC On-Demand Anodyne BDKRB1 54 41 O=C(C[C@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620729 FC On-Demand Anodyne EPHX2 24 50 O=C(C[C@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620729 FC On-Demand Anodyne TGM2 65 43 O=C(C[C@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620729 FC On-Demand Anodyne F13A1 53 41 O=C(C[C@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620729 FC On-Demand Anodyne SFRP1 50 39 O=C(C[C@@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620730 FC On-Demand Anodyne BDKRB1 54 41 O=C(C[C@@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620730 FC On-Demand Anodyne EPHX2 24 50 O=C(C[C@@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620730 FC On-Demand Anodyne TGM2 65 43 O=C(C[C@@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620730 FC On-Demand Anodyne F13A1 53 41 O=C(C[C@@H]1CCNC1=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620730 FC On-Demand Anodyne SFRP1 50 39 Cn1nc2c(c1NC(=O)NNC(=O)c1cccc(C(F)(F)F)c1)CCCC2 ZINC000880620747 GF On-Demand Reactive CCR2 65 37 COc1ccc2c(c1)CN(C(=O)c1cnc(CC3CC3)s1)C2 ZINC000880620751 DG On-Demand Anodyne CPT2 29 40 COc1ccc2c(c1)CN(C(=O)C[C@@H]1C[C@H]1C1CC1)C2 ZINC000880620756 CF On-Demand Anodyne MTNR1B 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620757 GD On-Demand Anodyne CCKAR 16 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620757 GD On-Demand Anodyne FPR1 41 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620757 GD On-Demand Anodyne CALCRL 18 50 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620758 GD On-Demand Anodyne CCKAR 16 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620758 GD On-Demand Anodyne FPR1 41 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)Nc2ccccc2C1 ZINC000880620758 GD On-Demand Anodyne CALCRL 18 50 COc1ccc2c(c1)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880620776 DI On-Demand Anodyne NQO2 28 50 COc1ccc2c(c1)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880620776 DI On-Demand Anodyne PPARD 34 42 COc1ccc2c(c1)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880620776 DI On-Demand Anodyne MTNR1A 31 47 COc1ccc2c(c1)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880620776 DI On-Demand Anodyne MTNR1B 41 49 COc1ccc2c(c1)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880620776 DI On-Demand Anodyne EBP 28 42 COc1ccc2c(c1)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880620777 DI On-Demand Anodyne NQO2 28 50 COc1ccc2c(c1)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880620777 DI On-Demand Anodyne PPARD 34 42 COc1ccc2c(c1)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880620777 DI On-Demand Anodyne MTNR1A 31 47 COc1ccc2c(c1)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880620777 DI On-Demand Anodyne MTNR1B 41 49 COc1ccc2c(c1)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880620777 DI On-Demand Anodyne EBP 28 42 COc1ccc2c(c1)CN(C(=O)COC1CC1)C2 ZINC000880620793 BD On-Demand Anodyne CPT2 32 42 COc1ccc2c(c1)CN(C(=O)COC1CC1)C2 ZINC000880620793 BD On-Demand Anodyne MTNR1A 37 41 COc1ccc2c(c1)CN(C(=O)COC1CC1)C2 ZINC000880620793 BD On-Demand Anodyne MTNR1B 38 42 Cn1nc2c(c1NC(=O)NNC(=O)CCc1ccccc1)CCCC2 ZINC000880620828 EE On-Demand Reactive VIPR1 23 41 COc1ccccc1-c1ccc(C(=O)N[C@@H]2C[C@@H](OC(C)(C)C)C2)c(O)n1 ZINC000880620832 FH On-Demand Anodyne HTR3A 15 45 COc1ccc2c(c1)CN(C(=O)c1ccc(CN3CCOCC3)o1)C2 ZINC000880620847 EE On-Demand Anodyne MMP13 16 40 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccn2nccc12 ZINC000880620864 GD On-Demand Anodyne EPHX2 18 49 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccn2nccc12 ZINC000880620864 GD On-Demand Anodyne TGM2 51 44 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3c4ccccc4C[C@@H]3O)cc2)N1 ZINC000880620867 EE On-Demand Anodyne PLM1_PLAFA 43 40 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3c4ccccc4C[C@@H]3O)cc2)N1 ZINC000880620867 EE On-Demand Anodyne PLM2_PLAFA 35 40 Cn1nc2c(c1NC(=O)N1CCCC[C@@H]1c1ccccc1)CCCC2 ZINC000880620897 EI On-Demand Anodyne CPT1A 54 39 Cn1nc2c(c1NC(=O)N1CCCC[C@H]1c1ccccc1)CCCC2 ZINC000880620898 EI On-Demand Anodyne CPT1A 54 39 COc1ccc2c(c1)CN(C(=O)C1CCC(S(C)(=O)=O)CC1)C2 ZINC000880620899 EE On-Demand Anodyne MTNR1A 29 49 COc1ccc2c(c1)CN(C(=O)C1CCC(S(C)(=O)=O)CC1)C2 ZINC000880620899 EE On-Demand Anodyne MTNR1B 25 49 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cncc2[nH]ccc12 ZINC000880620904 GE On-Demand Anodyne EPHX2 18 49 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cncc2[nH]ccc12 ZINC000880620904 GE On-Demand Anodyne TGM2 55 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccc(OC)cc2C1 ZINC000880620916 FE On-Demand Anodyne HDAC8 15 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccc(OC)cc2C1 ZINC000880620917 FE On-Demand Anodyne HDAC8 15 44 COc1ccc2c(c1)CN(C(=O)CCCCc1ccc(OC)c(OC)c1)C2 ZINC000880620923 FH On-Demand Anodyne INHA 41 38 COc1ccc2c(c1)CN(C(=O)CCCCc1ccc(OC)c(OC)c1)C2 ZINC000880620923 FH On-Demand Anodyne MTNR1B 38 42 COc1ccc2c(c1)CN(C(=O)CCCCc1ccc(OC)c(OC)c1)C2 ZINC000880620923 FH On-Demand Anodyne EBP 19 40 COc1ccc2c(c1)CN(C(=O)CCCCc1ccc(OC)c(OC)c1)C2 ZINC000880620923 FH On-Demand Anodyne ABCB1 24 47 COc1ccc2c(c1)CN(C(=O)CCCCc1ccc(OC)c(OC)c1)C2 ZINC000880620923 FH On-Demand Anodyne HCRTR2 15 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620932 DD On-Demand Anodyne PLM1_PLAFA 49 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620932 DD On-Demand Anodyne PLM2_PLAFA 88 41 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620933 DD On-Demand Anodyne PLM1_PLAFA 49 40 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620933 DD On-Demand Anodyne PLM2_PLAFA 88 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620934 DD On-Demand Anodyne PLM1_PLAFA 49 40 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880620934 DD On-Demand Anodyne PLM2_PLAFA 88 41 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild HSD11B1 15 41 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild TGM1 26 48 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild EPHX2 38 54 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild TGM2 108 51 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild F13A1 105 48 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild SFRP1 113 44 C=CC(C)(C)CC(=O)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620977 FF On-Demand Mild WNT3 68 34 COc1ccc2c(c1)CN(C(=O)[C@H](CNC(=O)OC(C)(C)C)OC)C2 ZINC000880620980 FE On-Demand Anodyne MTNR1A 50 36 COc1ccc2c(c1)CN(C(=O)[C@H](CNC(=O)OC(C)(C)C)OC)C2 ZINC000880620980 FE On-Demand Anodyne MTNR1B 45 34 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne PTPN2 41 32 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne SIGMAR1 18 43 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne TGM1 15 47 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne EPHX2 40 55 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne TGM2 84 47 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne F13A1 81 47 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne SFRP1 106 44 O=C(COC1CC1)NC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880620985 ED On-Demand Anodyne WNT3 58 32 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C)Cc1ccccn1)C2 ZINC000880621004 DF On-Demand Anodyne MMP3 15 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C)Cc1ccccn1)C2 ZINC000880621004 DF On-Demand Anodyne FAAH 17 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C)Cc1ccccn1)C2 ZINC000880621004 DF On-Demand Anodyne ADAM9 27 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C)Cc1ccccn1)C2 ZINC000880621007 DF On-Demand Anodyne MMP3 15 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C)Cc1ccccn1)C2 ZINC000880621007 DF On-Demand Anodyne FAAH 17 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C)Cc1ccccn1)C2 ZINC000880621007 DF On-Demand Anodyne ADAM9 27 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccn(-c2ccc(C)cc2)n1 ZINC000880621022 GG On-Demand Anodyne AMP1_PLAFQ 19 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccn(-c2ccc(C)cc2)n1 ZINC000880621023 GG On-Demand Anodyne AMP1_PLAFQ 19 41 O=C(CC[C@H]1CCc2ccccc21)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621026 DG On-Demand Anodyne PLM1_PLAFA 48 42 O=C(CC[C@H]1CCc2ccccc21)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621026 DG On-Demand Anodyne PLM2_PLAFA 45 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne CCKAR 41 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne CTSK 20 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne CTSL 22 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne FPR1 48 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne PLM1_PLAFA 53 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880621036 FD On-Demand Anodyne PLM2_PLAFA 87 46 Cn1nc2c(c1NC(=O)NNC(=O)c1cccc(OC(F)F)c1)CCCC2 ZINC000880621047 GE On-Demand Reactive DRD4 40 30 COc1ccc2c(c1)CN(C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)C2 ZINC000880621052 GE On-Demand Anodyne SIGMAR1 17 40 COc1ccc2c(c1)CN(C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)C2 ZINC000880621052 GE On-Demand Anodyne PLA2G2A 45 42 COc1ccc2c(c1)CN(C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)C2 ZINC000880621052 GE On-Demand Anodyne CPT2 41 44 COc1ccc2c(c1)CN(C(=O)C[C@@H]1CCNC1=O)C2 ZINC000880621054 CD On-Demand Anodyne MTNR1B 20 40 COc1ccc2c(c1)CN(C(=O)C[C@H]1CCNC1=O)C2 ZINC000880621055 CD On-Demand Anodyne MTNR1B 20 40 O=C(CC[C@@H]1CCc2ccccc21)N1Cc2cc(F)c(F)cc2C1 ZINC000880621062 EI On-Demand Anodyne SSTR1 29 40 O=C(CC[C@H]1CCc2ccccc21)N1Cc2cc(F)c(F)cc2C1 ZINC000880621063 EI On-Demand Anodyne SSTR1 29 40 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne F2 44 40 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne ELANE 28 40 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne CTRA_BOVIN 41 32 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne TRY1_BOVIN 71 37 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne CELA2A 48 32 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne XIAP 76 39 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne BIRC8 44 34 C[C@@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621072 FD On-Demand Anodyne BRCA1 63 34 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne F2 44 40 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne ELANE 28 40 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne CTRA_BOVIN 41 32 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne TRY1_BOVIN 71 37 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne CELA2A 48 32 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne XIAP 76 39 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne BIRC8 44 34 C[C@H](Cc1ccccn1)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880621073 FD On-Demand Anodyne BRCA1 63 34 CC[C@@H]1CCC[C@@]1(C)C(=O)N[C@H](C)Cc1ccccn1 ZINC000880621079 CG On-Demand Anodyne TIMP3 72 35 CC[C@@H]1CCC[C@@]1(C)C(=O)N[C@@H](C)Cc1ccccn1 ZINC000880621081 CG On-Demand Anodyne TIMP3 72 35 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880621095 GD On-Demand Anodyne EPHX2 27 58 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880621095 GD On-Demand Anodyne TGM2 49 41 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880621095 GD On-Demand Anodyne F13A1 32 41 CC1(C)CC[C@@H](CC(=O)N[C@H]2c3ccccc3C[C@@H]2O)OC1 ZINC000880621102 DE On-Demand Anodyne PLM1_PLAFA 45 38 CC1(C)CC[C@@H](CC(=O)N[C@H]2c3ccccc3C[C@@H]2O)OC1 ZINC000880621102 DE On-Demand Anodyne PLM2_PLAFA 86 38 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne DRD4 19 42 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne CNR2 16 42 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne SIGMAR1 16 45 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne EPHX2 47 52 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne TGM2 65 48 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne F13A1 48 43 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne AKR1C3 44 37 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne SFRP1 113 44 Cc1coc(C(=O)NC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000880621103 EE On-Demand Anodyne WNT3 72 33 O=C(CN1CCCCS1(=O)=O)Nc1nn(-c2ccc(F)cc2)c2c1CCC2 ZINC000880621112 GD On-Demand Anodyne CDK1 15 40 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621123 GE On-Demand Anodyne PLM1_PLAFA 45 37 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621123 GE On-Demand Anodyne PLM2_PLAFA 79 37 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621124 GE On-Demand Anodyne PLM1_PLAFA 45 37 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621124 GE On-Demand Anodyne PLM2_PLAFA 79 37 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621125 GE On-Demand Anodyne PLM1_PLAFA 45 37 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)N[C@H]2c3ccccc3C[C@@H]2O)CO1 ZINC000880621125 GE On-Demand Anodyne PLM2_PLAFA 79 37 CC[C@@H](C(=O)NNC(=O)Nc1c2c(nn1C)CCCC2)c1ccccc1 ZINC000880621138 FF On-Demand Reactive KCNQ2 48 42 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)[C@@H]1CCCCO1 ZINC000880621193 FE On-Demand Anodyne PAPA1_CARPA 26 40 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)[C@H]1CCCCO1 ZINC000880621194 FE On-Demand Anodyne PAPA1_CARPA 26 40 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)[C@H]1CCCCO1 ZINC000880621195 FE On-Demand Anodyne PAPA1_CARPA 26 40 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)[C@@H]1CCCCO1 ZINC000880621196 FE On-Demand Anodyne PAPA1_CARPA 26 40 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc(C(F)F)[nH]n1 ZINC000880621197 FD On-Demand Anodyne CACNA1I 41 34 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc2ccccc2cc1F ZINC000880621236 GH On-Demand Anodyne CCR3 25 41 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc2ccccc2cc1F ZINC000880621236 GH On-Demand Anodyne CACNA1I 48 34 CC[C@@H](O)CNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880621253 EG On-Demand Anodyne ADRB1 52 38 Cn1nc2c(c1NC(=O)N1CC[C@H](Oc3ccc(F)cc3)C1)CCCC2 ZINC000880621272 FG On-Demand Anodyne EPHX2 19 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880621355 EI On-Demand Anodyne RBP4 41 36 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880621356 EI On-Demand Anodyne RBP4 41 36 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@H]2C[C@H]2C1 ZINC000880621357 EI On-Demand Anodyne RBP4 41 36 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880621358 EI On-Demand Anodyne RBP4 41 36 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CC[C@H](O)CC1 ZINC000880621363 FH On-Demand Anodyne EPHX2 52 45 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1c[nH]cc1C1CC1 ZINC000880621383 EE On-Demand Anodyne CACNA1I 44 32 Cn1nc2c(c1NC(=O)N1CCC[C@@](O)(c3ccc(Cl)cc3)C1)CCCC2 ZINC000880621427 GG On-Demand Anodyne CCR1 47 37 Cn1nc2c(c1NC(=O)N1CCC[C@](O)(c3ccc(Cl)cc3)C1)CCCC2 ZINC000880621428 GG On-Demand Anodyne CCR1 47 37 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880621474 FG On-Demand Anodyne S1PR2 29 43 O=C(N[C@H]1CCCN2CCCC[C@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621556 EF On-Demand Anodyne GABRA1 17 44 O=C(N[C@H]1CCCN2CCCC[C@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621556 EF On-Demand Anodyne GABRA2 16 44 O=C(N[C@@H]1CCCN2CCCC[C@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621557 EF On-Demand Anodyne GABRA1 17 44 O=C(N[C@@H]1CCCN2CCCC[C@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621557 EF On-Demand Anodyne GABRA2 16 44 O=C(N[C@H]1CCCN2CCCC[C@@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621558 EF On-Demand Anodyne GABRA1 17 44 O=C(N[C@H]1CCCN2CCCC[C@@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621558 EF On-Demand Anodyne GABRA2 16 44 O=C(N[C@@H]1CCCN2CCCC[C@@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621559 EF On-Demand Anodyne GABRA1 17 44 O=C(N[C@@H]1CCCN2CCCC[C@@H]12)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880621559 EF On-Demand Anodyne GABRA2 16 44 CC(=O)c1cc(NC(=O)Cc2ccccc2N2CCCC2=O)ccc1C ZINC000880621585 FH On-Demand Anodyne AVPR2 58 39 CC(=O)c1cc(NC(=O)Cc2ccccc2N2CCCC2=O)ccc1C ZINC000880621585 FH On-Demand Anodyne KCNQ2 49 37 CC(C)(C)OC(=O)CN(C(=O)c1cnc2cc[nH]c2c1)C1CCC1 ZINC000880621672 EF On-Demand Anodyne ACE 48 35 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cnc2cc[nH]c2c1 ZINC000880621697 FE On-Demand Anodyne CACNA1I 62 37 C[C@@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621743 DG On-Demand Anodyne JAK3 24 40 C[C@@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621743 DG On-Demand Anodyne JAK1 18 40 C[C@@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621743 DG On-Demand Anodyne TYK2 22 40 C[C@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621746 DG On-Demand Anodyne JAK3 24 40 C[C@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621746 DG On-Demand Anodyne JAK1 18 40 C[C@H](NC(=O)c1cccn2nccc12)C1CCC(F)(F)CC1 ZINC000880621746 DG On-Demand Anodyne TYK2 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne FKBP1A 43 37 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MMP13 17 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MTNR1A 29 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MMP3 27 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MMP7 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621761 EF On-Demand Anodyne MMP1 22 40 CC(=O)c1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1C ZINC000880621763 DH On-Demand Anodyne JUN 19 44 CC(=O)c1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1C ZINC000880621763 DH On-Demand Anodyne CSF1R 18 42 CC(=O)c1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1C ZINC000880621763 DH On-Demand Anodyne BTK 24 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne FKBP1A 43 37 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MMP13 17 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MTNR1A 29 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MMP3 27 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MMP7 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621764 EF On-Demand Anodyne MMP1 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne FKBP1A 43 37 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MMP13 17 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MTNR1A 29 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MMP3 27 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MMP7 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCN3CCCC[C@@H]13)C2 ZINC000880621768 EF On-Demand Anodyne MMP1 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne FKBP1A 43 37 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MMP13 17 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MTNR1A 29 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MMP3 27 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MMP7 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCN3CCCC[C@H]13)C2 ZINC000880621771 EF On-Demand Anodyne MMP1 22 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)(CO)CC1 ZINC000880621793 GF On-Demand Anodyne CACNA1H 40 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)(CO)CC1 ZINC000880621793 GF On-Demand Anodyne PDGFRB 38 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)(CO)CC1 ZINC000880621793 GF On-Demand Anodyne S1PR2 32 47 CS(=O)(=O)C1CCC(C(=O)N2Cc3ccccc3-c3ccccc32)CC1 ZINC000880621826 FH On-Demand Anodyne HSD17B3 17 46 O=C(N[C@@H]1CCCN2CCCC[C@H]12)c1cccn2nccc12 ZINC000880621835 CE On-Demand Anodyne JAK3 16 40 O=C(N[C@@H]1CCCN2CCCC[C@H]12)c1cccn2nccc12 ZINC000880621835 CE On-Demand Anodyne TYK2 19 40 O=C(N[C@H]1CCCN2CCCC[C@H]12)c1cccn2nccc12 ZINC000880621836 CE On-Demand Anodyne JAK3 16 40 O=C(N[C@H]1CCCN2CCCC[C@H]12)c1cccn2nccc12 ZINC000880621836 CE On-Demand Anodyne TYK2 19 40 O=C(N[C@H]1CCCN2CCCC[C@@H]12)c1cccn2nccc12 ZINC000880621837 CE On-Demand Anodyne JAK3 16 40 O=C(N[C@H]1CCCN2CCCC[C@@H]12)c1cccn2nccc12 ZINC000880621837 CE On-Demand Anodyne TYK2 19 40 O=C(N[C@@H]1CCCN2CCCC[C@@H]12)c1cccn2nccc12 ZINC000880621838 CE On-Demand Anodyne JAK3 16 40 O=C(N[C@@H]1CCCN2CCCC[C@@H]12)c1cccn2nccc12 ZINC000880621838 CE On-Demand Anodyne TYK2 19 40 CCOC(=O)Cn1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)n1 ZINC000880621944 FE On-Demand Anodyne MTNR1B 20 41 CCOC(=O)Cn1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)n1 ZINC000880621946 FE On-Demand Anodyne MTNR1B 20 41 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCCN(C(=O)C(F)(F)F)C3)cc2)N1 ZINC000880621971 GE On-Demand Anodyne CACNA1I 55 32 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCCN(C(=O)C(F)(F)F)C3)cc2)N1 ZINC000880621973 GE On-Demand Anodyne CACNA1I 55 32 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCCN(C(=O)C(F)(F)F)C3)cc2)N1 ZINC000880621975 GE On-Demand Anodyne CACNA1I 55 32 C[C@@]1(C#N)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880621977 FH On-Demand Mild CACNA1H 38 40 C[C@@]1(C#N)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880621977 FH On-Demand Mild S1PR2 28 42 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCCN(C(=O)C(F)(F)F)C3)cc2)N1 ZINC000880621978 GE On-Demand Anodyne CACNA1I 55 32 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne CPT1A 44 31 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne ROCK1 44 33 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne PRNP 42 39 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne KDR 42 39 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne ABCB1B 25 41 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne GRM4 27 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne NR1H4 18 50 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne HDAC1 27 45 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne HDAC2 22 45 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne ABCB1 22 43 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne PLAU 24 46 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne TAAR1 42 42 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne ABCG2 41 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne ENPP1 56 32 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne SMO 41 48 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne KCNK3 135 57 COc1cc(NC(=O)c2ccccc2)c(C(=O)Nc2cccc(OCC(N)=O)c2)cc1OC ZINC000880621984 IG On-Demand Anodyne KCNK9 95 48 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC(=O)N[C@H]1c1cncn1C)C2 ZINC000880622064 GD On-Demand Anodyne MTNR1A 20 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC(=O)N[C@H]1c1cncn1C)C2 ZINC000880622064 GD On-Demand Anodyne MTNR1B 22 41 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1c3c(nn1C)CCCC3)CC2 ZINC000880622074 FF On-Demand Anodyne P2RY14 44 32 Cn1nc2c(c1NC(=O)NCc1cc(F)cnc1Cl)CCCC2 ZINC000880622084 EF On-Demand Anodyne P2RX7 41 37 Cc1cnc(Cl)c(C(=O)N(CC(=O)OC(C)(C)C)C2CCC2)c1 ZINC000880622092 EG On-Demand Anodyne ACE 55 42 C#CCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880622093 GH On-Demand Mild PDGFRB 40 38 C#CCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880622093 GH On-Demand Mild S1PR2 34 49 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ncc(Br)cn1)C2 ZINC000880622114 GE On-Demand Reactive FAAH 15 43 Cn1nc2c(c1NC(=O)NCc1cccc3ncccc13)CCCC2 ZINC000880622115 EG On-Demand Anodyne ACHE 45 36 Cn1nc2c(c1NC(=O)NCc1cccc3ncccc13)CCCC2 ZINC000880622115 EG On-Demand Anodyne BCHE 66 36 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880622176 FF On-Demand Anodyne CACNA1I 69 38 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880622177 FF On-Demand Anodyne CACNA1I 69 38 C[C@@H](O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880622244 GH On-Demand Anodyne CACNA1H 32 41 C[C@@H](O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880622244 GH On-Demand Anodyne PDGFRB 42 38 C[C@@H](O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880622244 GH On-Demand Anodyne S1PR2 29 44 Cn1nc2c(c1NC(=O)NC[C@H](O)c1cccc3ccccc13)CCCC2 ZINC000880622260 FG On-Demand Anodyne BCHE 49 35 Cn1nc2c(c1NC(=O)NC[C@@H](O)c1cccc3ccccc13)CCCC2 ZINC000880622263 FG On-Demand Anodyne BCHE 49 35 CC(C)c1cc(NC(=O)Nc2c3c(nn2C)CCCC3)ccc1O ZINC000880622314 EH On-Demand Anodyne THRB 35 40 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3CCCN4CCCC[C@H]34)cc2)N1 ZINC000880622361 EE On-Demand Anodyne SSTR3 29 43 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCCN4CCCC[C@@H]34)cc2)N1 ZINC000880622365 EE On-Demand Anodyne SSTR3 29 43 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCCN4CCCC[C@H]34)cc2)N1 ZINC000880622369 EE On-Demand Anodyne SSTR3 29 43 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3CCCN4CCCC[C@@H]34)cc2)N1 ZINC000880622372 EE On-Demand Anodyne SSTR3 29 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)(CO)C1 ZINC000880622416 GE On-Demand Anodyne S1PR2 29 44 Cn1nc2c(c1NC(=O)N[C@H]1Cc3ccc(Cl)cc3C1)CCCC2 ZINC000880622421 EG On-Demand Anodyne CNR1 40 31 Cn1nc2c(c1NC(=O)N[C@@H]1Cc3ccc(Cl)cc3C1)CCCC2 ZINC000880622424 EG On-Demand Anodyne CNR1 40 31 CN1CCN(C2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)CC1 ZINC000880622440 FD On-Demand Anodyne L3MBTL3 67 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCCN2CCCC[C@H]12 ZINC000880622461 FE On-Demand Anodyne CCKAR 19 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCCN2CCCC[C@@H]12 ZINC000880622462 FE On-Demand Anodyne CCKAR 19 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCN2CCCC[C@H]12 ZINC000880622463 FE On-Demand Anodyne CCKAR 19 47 Cn1nc2c(c1NC(=O)N1CCc3c(CC(N)=O)cccc3C1)CCCC2 ZINC000880622465 FD On-Demand Anodyne P2RY14 40 32 Cc1cnc(Cl)c(C(=O)N2CCC[C@@H](NC(=O)C(F)(F)F)[C@H]2C)c1 ZINC000880622466 FF On-Demand Anodyne TRPC6 50 37 Cc1nc(C(C)C)ncc1C(=O)N1CCC[C@@H](NC(=O)C(F)(F)F)[C@H]1C ZINC000880622479 FF On-Demand Anodyne TRPC6 47 34 CC(=O)c1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1C ZINC000880622503 EG On-Demand Anodyne MAPK14 20 40 CC(=O)c1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1C ZINC000880622503 EG On-Demand Anodyne KCNK3 52 38 CC(=O)c1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1C ZINC000880622505 EG On-Demand Anodyne MAPK14 20 40 CC(=O)c1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1C ZINC000880622505 EG On-Demand Anodyne KCNK3 52 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCN2CCCC[C@@H]12 ZINC000880622547 FE On-Demand Anodyne CCKAR 19 47 CC(=O)c1cc(NC(=O)[C@@H]2CCc3nncn3CC2)ccc1C ZINC000880622576 DE On-Demand Anodyne EPHX2 15 42 CC(=O)c1cc(NC(=O)[C@H]2CCc3nncn3CC2)ccc1C ZINC000880622579 DE On-Demand Anodyne EPHX2 15 42 Cn1nc2c(c1NC(=O)N[C@H]1CCOC1=O)CCCC2 ZINC000880622585 CC On-Demand Anodyne LUXR 67 37 Cn1nc2c(c1NC(=O)N[C@H]1CCOC1=O)CCCC2 ZINC000880622585 CC On-Demand Anodyne TRAR 79 37 Cn1nc2c(c1NC(=O)N[C@H]1CCOC1=O)CCCC2 ZINC000880622585 CC On-Demand Anodyne LASR 58 37 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@H]1C[C@H](O)C1 ZINC000880622597 EF On-Demand Anodyne EPHX2 43 40 Cn1nc2c(c1NC(=O)N1CCC(c3nc(C4CCC4)no3)CC1)CCCC2 ZINC000880622626 GG On-Demand Anodyne ETHR 52 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccc(C)o1)C(F)(F)F ZINC000880622786 GG On-Demand Anodyne FPR1 43 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccc(C)o1)C(F)(F)F ZINC000880622787 GG On-Demand Anodyne FPR1 43 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccc(C)o1)C(F)(F)F ZINC000880622788 GG On-Demand Anodyne FPR1 43 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccc(C)o1)C(F)(F)F ZINC000880622789 GG On-Demand Anodyne FPR1 43 37 CN1C[C@@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1=O ZINC000880622814 GF On-Demand Anodyne CCR3 47 39 CC(=O)c1cc(NC(=O)Cc2c(Br)cnn2C)ccc1C ZINC000880622816 FF On-Demand Anodyne IMDH_CRYPV 25 43 CN1C[C@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1=O ZINC000880622818 GF On-Demand Anodyne CCR3 47 39 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CCC(F)(F)CC1 ZINC000880622840 FH On-Demand Anodyne KCNQ2 41 32 CC(=O)c1cc(NC(=O)CC(C)(C)CC(F)F)ccc1C ZINC000880622874 CI On-Demand Anodyne SLC1A2 41 33 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCC1=O ZINC000880622885 GF On-Demand Anodyne PDGFRB 52 44 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCC1=O ZINC000880622885 GF On-Demand Anodyne S1PR2 27 42 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622890 GE On-Demand Anodyne CCR3 71 47 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622890 GE On-Demand Anodyne MLNR 21 40 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622890 GE On-Demand Anodyne MCHR1 18 42 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622892 GE On-Demand Anodyne CCR3 71 47 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622892 GE On-Demand Anodyne MLNR 21 40 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880622892 GE On-Demand Anodyne MCHR1 18 42 COc1cccc([C@H](O)C2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c1 ZINC000880622928 GG On-Demand Anodyne DRD4 40 31 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880622946 GE On-Demand Anodyne GABRA1 15 44 CS(=O)(=O)C1CCC(C(=O)N[C@H]2CCCN3CCCC[C@@H]23)CC1 ZINC000880623047 ED On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)C1CCC(C(=O)N[C@@H]2CCCN3CCCC[C@@H]23)CC1 ZINC000880623049 ED On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)C1CCC(C(=O)N[C@@H]2CCCN3CCCC[C@H]23)CC1 ZINC000880623051 ED On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)C1CCC(C(=O)N[C@H]2CCCN3CCCC[C@H]23)CC1 ZINC000880623053 ED On-Demand Anodyne EPHX2 16 42 CC(C)(C)OC(=O)CN(C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)C1CCC1 ZINC000880623067 FF On-Demand Anodyne ACE 45 41 CC(C)(C)OC(=O)CN(C(=O)c1ccc([C@H]2CCC(=O)N2)cc1)C1CCC1 ZINC000880623068 FF On-Demand Anodyne ACE 45 41 CC(=O)Nc1cccc2c1CN(C(=O)Nc1c3c(nn1C)CCCC3)CC2 ZINC000880623071 FF On-Demand Anodyne P2RY14 44 32 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(CO)CC1 ZINC000880623091 GF On-Demand Anodyne CACNA1H 40 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(CO)CC1 ZINC000880623091 GF On-Demand Anodyne PDGFRB 45 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(CO)CC1 ZINC000880623091 GF On-Demand Anodyne S1PR2 36 52 CC(C)(C)OC(=O)CN(C(=O)c1cncc2[nH]ccc12)C1CCC1 ZINC000880623103 EF On-Demand Anodyne ACE 41 34 CC(=O)c1cc(NC(=O)c2c[nH]cc2C2CC2)ccc1C ZINC000880623106 CH On-Demand Anodyne HTR1F 67 40 COc1ccc(N2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c(OC)c1 ZINC000880623135 GF On-Demand Clean HTR1A 28 46 COc1ccc(N2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c(OC)c1 ZINC000880623135 GF On-Demand Clean DRD4 42 33 COc1ccc(N2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c(OC)c1 ZINC000880623135 GF On-Demand Clean HTR1B 16 46 COc1ccc(N2CCN(C(=O)Nc3c4c(nn3C)CCCC4)CC2)c(OC)c1 ZINC000880623135 GF On-Demand Clean PDGFRB 53 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)(F)CC1 ZINC000880623150 GG On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)(F)CC1 ZINC000880623150 GG On-Demand Anodyne FPR1 43 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)(F)CC1 ZINC000880623153 GG On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)(F)CC1 ZINC000880623153 GG On-Demand Anodyne FPR1 43 37 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC2(CCCO2)C1 ZINC000880623154 FH On-Demand Anodyne EPHX2 27 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)(F)CC1 ZINC000880623156 GG On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)(F)CC1 ZINC000880623156 GG On-Demand Anodyne FPR1 43 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)(F)CC1 ZINC000880623158 GG On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)(F)CC1 ZINC000880623158 GG On-Demand Anodyne FPR1 43 37 CC(C)(C)OC(=O)CN(C(=O)c1cccn2nccc12)C1CCC1 ZINC000880623186 EF On-Demand Anodyne ACE 54 39 C[C@@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCS1(=O)=O ZINC000880623188 GF On-Demand Anodyne S1PR2 26 40 C[C@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCS1(=O)=O ZINC000880623192 GF On-Demand Anodyne S1PR2 26 40 Cc1coc(C(=O)NC[C@@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880623218 DE On-Demand Anodyne CACNA1I 63 36 Cc1coc(C(=O)NC[C@H]2CCCN(C(=O)C(F)(F)F)C2)c1 ZINC000880623219 DE On-Demand Anodyne CACNA1I 63 36 CC(=O)c1cc(NC(=O)c2ncsc2C2CC2)ccc1C ZINC000880623225 DH On-Demand Anodyne MAP1 57 35 CCN(C(=O)[C@H]1CCc2cc(OC)ccc2C1)c1cnn(C)c1 ZINC000880623226 DF On-Demand Anodyne MTNR1B 17 40 Cn1nc2c(c1NC(=O)NN1CCc3ccccc3C1)CCCC2 ZINC000880623235 EE On-Demand Anodyne NOD2 40 33 Cn1nc2c(c1NC(=O)NCc1nc(-c3ccncc3)cs1)CCCC2 ZINC000880623246 FG On-Demand Anodyne ROCK1 23 45 Cn1nc2c(c1NC(=O)NCc1nc(-c3ccncc3)cs1)CCCC2 ZINC000880623246 FG On-Demand Anodyne ROCK2 16 45 Cn1nc2c(c1NC(=O)N1CC[C@@]3(CCc4ccccc4O3)C1)CCCC2 ZINC000880623338 FG On-Demand Anodyne EPHX2 16 42 Cn1nc2c(c1NC(=O)N1CC[C@@]3(CCc4ccccc4O3)C1)CCCC2 ZINC000880623338 FG On-Demand Anodyne TRPM8 19 46 Cn1nc2c(c1NC(=O)N1CC[C@]3(CCc4ccccc4O3)C1)CCCC2 ZINC000880623339 FG On-Demand Anodyne EPHX2 16 42 Cn1nc2c(c1NC(=O)N1CC[C@]3(CCc4ccccc4O3)C1)CCCC2 ZINC000880623339 FG On-Demand Anodyne TRPM8 19 46 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)CC1 ZINC000880623377 EG On-Demand Anodyne PDGFRB 35 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)CC1 ZINC000880623377 EG On-Demand Anodyne S1PR2 27 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(COC2)C1 ZINC000880623396 FG On-Demand Anodyne S1PR2 27 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(COC2)C1 ZINC000880623396 FG On-Demand Anodyne EPHX2 37 44 N#CCCN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623407 GG On-Demand Mild PDGFRB 47 39 N#CCCN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623407 GG On-Demand Mild S1PR2 28 41 CC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623408 GH On-Demand Anodyne CACNA1H 34 41 CC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623408 GH On-Demand Anodyne PDGFRB 42 39 CC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623408 GH On-Demand Anodyne S1PR2 27 41 CC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880623408 GH On-Demand Anodyne EPHX2 17 40 COC[C@H](C)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880623409 EG On-Demand Anodyne GCK 17 42 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc(C(F)(F)F)ccn1 ZINC000880623438 GF On-Demand Anodyne CCR2 53 36 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc(C(F)(F)F)ccn1 ZINC000880623438 GF On-Demand Anodyne CACNA1I 49 39 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1cc(C(F)(F)F)ccn1 ZINC000880623438 GF On-Demand Anodyne MAP3K12 27 40 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)c1ccc2c(O)ncnc2c1 ZINC000880623528 GD On-Demand Anodyne CACNA1I 63 38 Cc1ncc(CC(=O)N2CCC[C@@H](NC(=O)C(F)(F)F)[C@H]2C)o1 ZINC000880623539 ED On-Demand Anodyne TRPC6 44 33 CC(=O)c1cc(NC(=O)C2CCC(S(C)(=O)=O)CC2)ccc1C ZINC000880623556 EF On-Demand Anodyne EPHX2 18 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCN(C(=O)C(F)(F)F)C1)C2 ZINC000880623559 GF On-Demand Anodyne NQO2 23 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)C2 ZINC000880623561 GF On-Demand Anodyne NQO2 23 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C[C@@H]1CCCO1)C(F)(F)F)C2 ZINC000880623640 FG On-Demand Anodyne NQO2 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C[C@H]1CCCO1)C(F)(F)F)C2 ZINC000880623641 FG On-Demand Anodyne NQO2 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](C[C@H]1CCCO1)C(F)(F)F)C2 ZINC000880623642 FG On-Demand Anodyne NQO2 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](C[C@@H]1CCCO1)C(F)(F)F)C2 ZINC000880623643 FG On-Demand Anodyne NQO2 23 41 CC(=O)c1cc(NC(=O)CC[C@H]2CC(C)(C)CO2)ccc1C ZINC000880623673 DH On-Demand Anodyne PTPRF 45 37 CC(=O)c1cc(NC(=O)CC[C@@H]2CC(C)(C)CO2)ccc1C ZINC000880623675 DH On-Demand Anodyne PTPRF 45 37 CC(=O)c1cc(NC(=O)c2ccc(CN3CCOCC3)o2)ccc1C ZINC000880623705 EF On-Demand Anodyne MAPK14 17 41 CC(=O)c1cc(NC(=O)c2ccc(CN3CCOCC3)o2)ccc1C ZINC000880623705 EF On-Demand Anodyne EPHX2 22 40 Cn1nc2c(c1NC(=O)NCc1cc(Cl)ccc1O)CCCC2 ZINC000880623706 EF On-Demand Clean P2RX7 27 42 CC[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)[C@@H]1CCCCO1 ZINC000880623758 EF On-Demand Anodyne KCNQ2 41 32 CC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)[C@H]1CCCCO1 ZINC000880623760 EF On-Demand Anodyne KCNQ2 41 32 CC[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)[C@H]1CCCCO1 ZINC000880623762 EF On-Demand Anodyne KCNQ2 41 32 CC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)[C@@H]1CCCCO1 ZINC000880623764 EF On-Demand Anodyne KCNQ2 41 32 COC(=O)Nc1cccc(CNC(=O)Nc2c3c(nn2C)CCCC3)c1 ZINC000880623778 FF On-Demand Anodyne ROCK2 23 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC2(CC2)C1 ZINC000880623845 EH On-Demand Anodyne S1PR2 28 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CC1)OCCO2 ZINC000880623884 GH On-Demand Anodyne CACNA1H 38 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CC1)OCCO2 ZINC000880623884 GH On-Demand Anodyne PDGFRB 38 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CC1)OCCO2 ZINC000880623884 GH On-Demand Anodyne S1PR2 30 44 O=C(NC[C@H]1CCC2(CCCC2)O1)c1cccn2nccc12 ZINC000880623890 CF On-Demand Anodyne HCN4 40 31 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CCOC1 ZINC000880623894 EG On-Demand Anodyne CCR3 15 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CCOC1 ZINC000880623894 EG On-Demand Anodyne EPHX2 46 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CC[C@@H](O)CC1 ZINC000880623916 FH On-Demand Anodyne EPHX2 52 45 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(C2(O)CC2)CC1 ZINC000880623921 GH On-Demand Anodyne PDGFRB 33 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(C2(O)CC2)CC1 ZINC000880623921 GH On-Demand Anodyne S1PR2 29 44 CC1(C)CC[C@@H](CC(=O)N[C@H](Cc2ccccc2)c2ncco2)OC1 ZINC000880623975 EH On-Demand Anodyne TIMP3 41 32 CC1(C)CC[C@@H](CC(=O)N[C@@H](Cc2ccccc2)c2ncco2)OC1 ZINC000880623977 EH On-Demand Anodyne TIMP3 41 32 O=C(NC[C@H]1CN(C2CC2)C(=O)O1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880624008 FF On-Demand Anodyne PDE4D 15 42 O=C(NC[C@H]1CN(C2CC2)C(=O)O1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880624008 FF On-Demand Anodyne CACNA1I 57 36 O=C(NC[C@@H]1CN(C2CC2)C(=O)O1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880624009 FF On-Demand Anodyne PDE4D 15 42 O=C(NC[C@@H]1CN(C2CC2)C(=O)O1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880624009 FF On-Demand Anodyne CACNA1I 57 36 COC1(C)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624013 GI On-Demand Anodyne CACNA1H 40 42 COC1(C)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624013 GI On-Demand Anodyne PDGFRB 45 38 COC1(C)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624013 GI On-Demand Anodyne S1PR2 31 46 C[C@H](CCO)N(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624017 FG On-Demand Anodyne NPY5R 34 46 C[C@@H](CCO)N(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624018 FG On-Demand Anodyne NPY5R 34 46 COC[C@@]1(C)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624040 GI On-Demand Anodyne S1PR2 29 43 COC[C@]1(C)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624041 GI On-Demand Anodyne S1PR2 29 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@]2(C1)CC2(F)F ZINC000880624044 GI On-Demand Anodyne S1PR2 28 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@]2(C1)CC2(F)F ZINC000880624045 GI On-Demand Anodyne S1PR2 28 42 O=C(N[C@@H](Cc1ccccc1)c1ncco1)c1cnc(CC2CC2)s1 ZINC000880624063 FH On-Demand Anodyne ANPEP 41 32 O=C(N[C@@H](Cc1ccccc1)c1ncco1)c1cnc(CC2CC2)s1 ZINC000880624063 FH On-Demand Anodyne F11 46 40 O=C(N[C@H](Cc1ccccc1)c1ncco1)c1cnc(CC2CC2)s1 ZINC000880624064 FH On-Demand Anodyne ANPEP 41 32 O=C(N[C@H](Cc1ccccc1)c1ncco1)c1cnc(CC2CC2)s1 ZINC000880624064 FH On-Demand Anodyne F11 46 40 C[C@@H](O)CCCNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624096 FG On-Demand Anodyne ADRB1 44 37 N#CC[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624106 FI On-Demand Mild CCR3 40 44 N#CC[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624107 FI On-Demand Mild CCR3 40 44 NC(=O)C[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624115 GF On-Demand Anodyne CCR3 23 43 NC(=O)C[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624116 GF On-Demand Anodyne CCR3 23 43 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624120 GH On-Demand Anodyne KCNA3 42 36 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624120 GH On-Demand Anodyne HCN1 52 35 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624120 GH On-Demand Anodyne HCN4 49 35 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624121 GH On-Demand Anodyne KCNA3 42 36 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624121 GH On-Demand Anodyne HCN1 52 35 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCC3(CCCC3)O2)c(O)n1 ZINC000880624121 GH On-Demand Anodyne HCN4 49 35 C[C@H](O)CN(C(=O)c1ccc(OC(F)F)c(Cl)c1)C1CC1 ZINC000880624131 DF On-Demand Anodyne PDE4D 18 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCC2(CCCC2)O1 ZINC000880624134 FF On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC2(CCCC2)O1 ZINC000880624135 FF On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCC2(CCCC2)O1 ZINC000880624136 FF On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC2(CCCC2)O1 ZINC000880624137 FF On-Demand Anodyne PAPA1_CARPA 32 42 O=C(N[C@@H](Cc1ccccc1)c1ncco1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880624138 FE On-Demand Anodyne F11 50 43 O=C(N[C@H](Cc1ccccc1)c1ncco1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880624139 FE On-Demand Anodyne F11 50 43 O=C(NCCCCO)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624142 EG On-Demand Anodyne ADRB1 42 37 O=C(NCCCCO)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624142 EG On-Demand Anodyne CCR3 23 40 CC1(CO)CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624178 EF On-Demand Anodyne S1PR2 28 42 COc1cc(NC(=O)c2nnn(C)n2)c(C2CC2)cc1Cl ZINC000880624181 DE On-Demand Anodyne HTR4 48 36 CO[C@@H](C)CNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624230 EG On-Demand Anodyne ADRB1 43 36 C=CCOC(=O)[C@H](CC(=O)N1C[C@@H]2CCCC[C@@H]21)NC(=O)OC(C)(C)C ZINC000880624249 FE On-Demand Mild REN 45 37 COC[C@]1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624254 GG On-Demand Anodyne S1PR2 28 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NN1CCCCC1 ZINC000880624263 EH On-Demand Anodyne HTR2A 16 41 C[C@H]1C[C@H](CO)CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624273 GH On-Demand Anodyne PDGFRB 40 37 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624311 GG On-Demand Anodyne S1PR2 27 40 O=CN1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624322 GF On-Demand Anodyne PDGFRB 41 42 O=CN1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624322 GF On-Demand Anodyne S1PR2 26 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@H](CO)C1 ZINC000880624343 EF On-Demand Anodyne CCR3 27 45 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@H](CO)C1 ZINC000880624344 EF On-Demand Anodyne CCR3 27 45 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](CO)CC1 ZINC000880624352 GH On-Demand Anodyne PDGFRB 48 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](CO)CC1 ZINC000880624352 GH On-Demand Anodyne CCR3 36 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](CO)CC1 ZINC000880624353 GH On-Demand Anodyne PDGFRB 48 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](CO)CC1 ZINC000880624353 GH On-Demand Anodyne CCR3 36 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](Cc1ccccc1)c1ncco1)C2 ZINC000880624355 GH On-Demand Anodyne F11 50 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](Cc1ccccc1)c1ncco1)C2 ZINC000880624355 GH On-Demand Anodyne FAAH 25 54 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](Cc1ccccc1)c1ncco1)C2 ZINC000880624356 GH On-Demand Anodyne F11 50 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](Cc1ccccc1)c1ncco1)C2 ZINC000880624356 GH On-Demand Anodyne FAAH 25 54 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1C[C@H](O)C1 ZINC000880624378 EF On-Demand Anodyne EPHX2 43 40 C[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC[S@]1=O ZINC000880624388 GH On-Demand Anodyne PDGFRB 42 39 C[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC[S@@]1=O ZINC000880624389 GH On-Demand Anodyne PDGFRB 42 39 C[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC[S@]1=O ZINC000880624390 GH On-Demand Anodyne PDGFRB 42 39 C[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC[S@@]1=O ZINC000880624391 GH On-Demand Anodyne PDGFRB 42 39 O=C(N[C@@H](Cc1ccccc1)c1ncco1)[C@@H]1CCc2nncn2CC1 ZINC000880624392 FE On-Demand Anodyne F11 48 41 O=C(N[C@@H](Cc1ccccc1)c1ncco1)[C@H]1CCc2nncn2CC1 ZINC000880624393 FE On-Demand Anodyne F11 48 41 O=C(N[C@H](Cc1ccccc1)c1ncco1)[C@@H]1CCc2nncn2CC1 ZINC000880624394 FE On-Demand Anodyne F11 48 41 O=C(N[C@H](Cc1ccccc1)c1ncco1)[C@H]1CCc2nncn2CC1 ZINC000880624395 FE On-Demand Anodyne F11 48 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@H](CCCO)C1 ZINC000880624420 GH On-Demand Anodyne CCR3 22 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@H](CCCO)C1 ZINC000880624421 GH On-Demand Anodyne CCR3 22 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@](F)(CO)C1 ZINC000880624439 FG On-Demand Anodyne S1PR2 29 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@](F)(CO)C1 ZINC000880624440 FG On-Demand Anodyne S1PR2 29 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2C[C@@H]3CCCC[C@@H]32)N1Cc1ccccc1 ZINC000880624492 ED On-Demand Anodyne ACE 25 42 NC(=O)[C@@H]1CC[C@H](C(=O)N2C[C@@H]3CCCC[C@@H]32)N1Cc1ccccc1 ZINC000880624492 ED On-Demand Anodyne PREP 61 38 CO[C@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCO1 ZINC000880624498 FF On-Demand Anodyne PDGFRB 42 36 CO[C@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCO1 ZINC000880624498 FF On-Demand Anodyne DGAT1 15 41 O=C(COC1CC1)N[C@@H](Cc1ccccc1)c1ncco1 ZINC000880624500 CE On-Demand Anodyne TIMP3 83 37 O=C(COC1CC1)N[C@@H](Cc1ccccc1)c1ncco1 ZINC000880624500 CE On-Demand Anodyne F11 45 39 O=C(COC1CC1)N[C@H](Cc1ccccc1)c1ncco1 ZINC000880624501 CE On-Demand Anodyne TIMP3 83 37 O=C(COC1CC1)N[C@H](Cc1ccccc1)c1ncco1 ZINC000880624501 CE On-Demand Anodyne F11 45 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC(CC(F)F)C1 ZINC000880624522 FI On-Demand Anodyne S1PR2 26 41 C[C@@H](CO)N(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624523 EF On-Demand Anodyne NPY5R 35 48 C[C@H](CO)N(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624524 EF On-Demand Anodyne NPY5R 35 48 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@H]1CCCOC1 ZINC000880624529 EG On-Demand Anodyne CCR3 16 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@H]1CCCOC1 ZINC000880624529 EG On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CCCOC1 ZINC000880624530 EG On-Demand Anodyne CCR3 16 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@@H]1CCCOC1 ZINC000880624530 EG On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](O)C1 ZINC000880624540 EG On-Demand Anodyne HRH3 15 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](O)C1 ZINC000880624540 EG On-Demand Anodyne CCR3 25 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](O)C1 ZINC000880624541 EG On-Demand Anodyne HRH3 15 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](O)C1 ZINC000880624541 EG On-Demand Anodyne CCR3 25 40 O=C(c1cccn2nccc12)N1C[C@@H]2CCCC[C@@H]21 ZINC000880624542 CE On-Demand Anodyne JAK3 16 41 O=C(c1cccn2nccc12)N1C[C@@H]2CCCC[C@@H]21 ZINC000880624542 CE On-Demand Anodyne TYK2 20 41 C[C@H](O)CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624563 GF On-Demand Anodyne PDGFRB 51 40 C[C@H](O)CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624563 GF On-Demand Anodyne S1PR2 29 44 O=C(N[C@@H](Cc1ccccc1)c1ncco1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880624596 EF On-Demand Anodyne F11 42 38 O=C(N[C@H](Cc1ccccc1)c1ncco1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880624597 EF On-Demand Anodyne F11 42 38 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCO2)CC1 ZINC000880624637 GH On-Demand Anodyne CACNA1H 38 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCO2)CC1 ZINC000880624637 GH On-Demand Anodyne S1PR2 30 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCO2)CC1 ZINC000880624637 GH On-Demand Anodyne EPHX2 34 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCO2)CC1 ZINC000880624637 GH On-Demand Anodyne TRPM8 29 42 CS(=O)(=O)C1CCC(C(=O)N[C@@H](Cc2ccccc2)c2ncco2)CC1 ZINC000880624653 GF On-Demand Anodyne KLKB1 25 40 CS(=O)(=O)C1CCC(C(=O)N[C@@H](Cc2ccccc2)c2ncco2)CC1 ZINC000880624653 GF On-Demand Anodyne F11 54 47 CS(=O)(=O)C1CCC(C(=O)N[C@H](Cc2ccccc2)c2ncco2)CC1 ZINC000880624654 GF On-Demand Anodyne KLKB1 25 40 CS(=O)(=O)C1CCC(C(=O)N[C@H](Cc2ccccc2)c2ncco2)CC1 ZINC000880624654 GF On-Demand Anodyne F11 54 47 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@](O)(C(F)F)C1 ZINC000880624659 GG On-Demand Anodyne CACNA1H 35 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@](O)(C(F)F)C1 ZINC000880624659 GG On-Demand Anodyne S1PR2 32 47 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@](O)(C(F)F)C1 ZINC000880624660 GG On-Demand Anodyne CACNA1H 35 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@](O)(C(F)F)C1 ZINC000880624660 GG On-Demand Anodyne S1PR2 32 47 C[C@]1(O)CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624682 GH On-Demand Anodyne CACNA1H 38 41 C[C@]1(O)CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624682 GH On-Demand Anodyne PDGFRB 43 39 C[C@]1(O)CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624682 GH On-Demand Anodyne S1PR2 32 49 C[C@H](O)CN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880624688 DD On-Demand Anodyne SLC6A4 15 46 C[C@H](O)CN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880624688 DD On-Demand Anodyne MPO 66 35 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(Oc4cc(F)cc(F)c4)nc3)C2)CN1 ZINC000880624693 GF On-Demand Anodyne S1PR2 27 42 O=C1C[C@]2(CCN(C(=O)Nc3ccc(Oc4cc(F)cc(F)c4)nc3)C2)CN1 ZINC000880624694 GF On-Demand Anodyne S1PR2 27 42 CC1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624695 DH On-Demand Anodyne MLNR 33 40 CC1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624695 DH On-Demand Anodyne S1PR2 27 41 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)c(C2CC2)cc1Cl ZINC000880624698 GH On-Demand Anodyne DRD4 22 40 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)c(C2CC2)cc1Cl ZINC000880624698 GH On-Demand Anodyne HTR4 54 38 COC[C@@H](O)CNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624727 FE On-Demand Anodyne ADRB1 57 42 C[C@H](O)CN(C(=O)c1cc2cc(F)ccc2[nH]c1=O)C1CC1 ZINC000880624729 DD On-Demand Anodyne PYGL 31 44 COCC1(O)CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624736 FE On-Demand Anodyne PDGFRB 46 36 COCC1(O)CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624736 FE On-Demand Anodyne S1PR2 30 44 O=C(N[C@@H](Cc1ccccc1)c1ncco1)c1ncsc1C1CC1 ZINC000880624739 EH On-Demand Anodyne MAP1 45 37 O=C(N[C@H](Cc1ccccc1)c1ncco1)c1ncsc1C1CC1 ZINC000880624740 EH On-Demand Anodyne MAP1 45 37 CO[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624778 GI On-Demand Anodyne PDGFRB 41 37 CO[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624778 GI On-Demand Anodyne S1PR2 27 41 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H](Cc1ccccc1)c1ncco1 ZINC000880624782 FG On-Demand Anodyne F11 45 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](Cc1ccccc1)c1ncco1 ZINC000880624783 FG On-Demand Anodyne F11 45 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H](Cc1ccccc1)c1ncco1 ZINC000880624784 FG On-Demand Anodyne F11 45 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](Cc1ccccc1)c1ncco1 ZINC000880624785 FG On-Demand Anodyne F11 45 36 COC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624790 GG On-Demand Anodyne CACNA1H 37 40 COC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624790 GG On-Demand Anodyne PDGFRB 49 39 COC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624790 GG On-Demand Anodyne S1PR2 31 46 COC[C@@H](C)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624793 EG On-Demand Anodyne GCK 17 42 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880624812 GG On-Demand Anodyne CPT1A 120 47 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880624812 GG On-Demand Anodyne CPT2 40 35 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne CCR3 66 49 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne SLC6A5 28 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne EPHX2 60 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne MCHR1 25 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCN(CCO)CC1 ZINC000880624814 GF On-Demand Anodyne HPGDS 32 46 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC(F)(F)CC1 ZINC000880624821 FI On-Demand Anodyne NPY5R 16 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCS(=O)(=O)CC1 ZINC000880624832 GF On-Demand Anodyne EPHX2 48 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCOCC1 ZINC000880624835 EG On-Demand Anodyne PDGFRB 37 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCOCC1 ZINC000880624835 EG On-Demand Anodyne LIPE 15 46 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCOCC1 ZINC000880624835 EG On-Demand Anodyne S1PR2 27 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCOCC1 ZINC000880624835 EG On-Demand Anodyne EPHX2 33 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCOCC1 ZINC000880624835 EG On-Demand Anodyne DGAT1 24 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCS(=O)CC1 ZINC000880624837 FF On-Demand Anodyne PDGFRB 33 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCS(=O)CC1 ZINC000880624837 FF On-Demand Anodyne S1PR2 27 41 O=C(NCCOCCO)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624838 FE On-Demand Anodyne ADRB1 42 38 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880624839 GG On-Demand Anodyne HRH3 15 42 C[S@@](=O)CCCNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624845 FG On-Demand Anodyne CCR3 30 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(C(F)F)CC1 ZINC000880624855 GH On-Demand Anodyne CACNA1H 42 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(C(F)F)CC1 ZINC000880624855 GH On-Demand Anodyne PDGFRB 43 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(O)(C(F)F)CC1 ZINC000880624855 GH On-Demand Anodyne S1PR2 33 49 Cc1cncc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)c1 ZINC000880624856 GJ On-Demand Anodyne ADAM17 46 38 Cc1cncc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)c1 ZINC000880624856 GJ On-Demand Anodyne CPT1A 116 42 Cc1cncc([C@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)c1 ZINC000880624857 GJ On-Demand Anodyne ADAM17 46 38 Cc1cncc([C@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)c1 ZINC000880624857 GJ On-Demand Anodyne CPT1A 116 42 CN1C[C@@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCC1=O ZINC000880624858 GF On-Demand Anodyne CCR3 19 40 CN1C[C@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCC1=O ZINC000880624859 GF On-Demand Anodyne CCR3 19 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@H]1CCOC1 ZINC000880624868 EG On-Demand Anodyne CCR3 15 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N[C@H]1CCOC1 ZINC000880624868 EG On-Demand Anodyne EPHX2 46 39 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880624874 GF On-Demand Anodyne NPY5R 15 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624884 GF On-Demand Anodyne UL80 39 40 N#CCC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624887 FI On-Demand Mild PDGFRB 45 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCS(=O)(=O)CC1 ZINC000880624909 GE On-Demand Anodyne PDGFRB 33 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCS(=O)(=O)CC1 ZINC000880624909 GE On-Demand Anodyne S1PR2 28 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCO[C@@]2(CCOC2)C1 ZINC000880624915 GG On-Demand Anodyne EPHX2 33 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCO[C@]2(CCOC2)C1 ZINC000880624916 GG On-Demand Anodyne EPHX2 33 44 COCCCNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624928 EG On-Demand Anodyne ADRB1 41 36 O=C(NCC1(CO)CCOCC1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880624938 GG On-Demand Anodyne EPHX2 18 42 C[C@@H](O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880624947 FG On-Demand Anodyne ALOX5 26 41 N#CCN1CCC(NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624956 GG On-Demand Mild CCR3 39 43 N#CCN1CCC(NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624956 GG On-Demand Mild EPHX2 53 39 N#CCN1CCC(NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624956 GG On-Demand Mild HPGDS 31 42 CCn1ncc(CNC(=O)Nc2nc(COc3ccccc3)cs2)n1 ZINC000880624965 FF On-Demand Anodyne ROCK1 18 42 CCn1ncc(CNC(=O)Nc2nc(COc3ccccc3)cs2)n1 ZINC000880624965 FF On-Demand Anodyne ROCK2 17 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(O)CC1 ZINC000880624966 EF On-Demand Anodyne CPT1A 53 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@H](CCO)C1 ZINC000880624967 FG On-Demand Anodyne CCR3 26 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@H](CCO)C1 ZINC000880624968 FG On-Demand Anodyne CCR3 26 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1Cn1ccnc1 ZINC000880624982 GH On-Demand Anodyne CPT1A 55 39 O=C(CO)N1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624985 GD On-Demand Anodyne PDGFRB 49 42 O=C(CO)N1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880624985 GD On-Demand Anodyne S1PR2 28 42 NC(=O)COc1cccc(NC(=O)[C@H](O)[C@H](O)c2nc3ccccc3s2)c1 ZINC000880624996 GD On-Demand Anodyne F9 27 40 NC(=O)COc1cccc(NC(=O)[C@@H](O)[C@H](O)c2nc3ccccc3s2)c1 ZINC000880624997 GD On-Demand Anodyne F9 27 40 NC(=O)COc1cccc(NC(=O)[C@H](O)[C@@H](O)c2nc3ccccc3s2)c1 ZINC000880624998 GD On-Demand Anodyne F9 27 40 NC(=O)COc1cccc(NC(=O)[C@@H](O)[C@@H](O)c2nc3ccccc3s2)c1 ZINC000880624999 GD On-Demand Anodyne F9 27 40 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625002 EF On-Demand Anodyne CACNA1H 34 41 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625002 EF On-Demand Anodyne HTR1B 15 48 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625002 EF On-Demand Anodyne HTR2C 16 44 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625002 EF On-Demand Anodyne PDGFRB 54 43 CN1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625002 EF On-Demand Anodyne S1PR2 29 43 NC(=O)COc1cccc(NC(=O)CCSc2nc3ccccc3s2)c1 ZINC000880625003 GG On-Demand Anodyne LDHA 33 41 NC(=O)COc1cccc(NC(=O)CCSc2nc3ccccc3s2)c1 ZINC000880625003 GG On-Demand Anodyne ETHR 15 46 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1COCC[C@H]1O ZINC000880625006 ED On-Demand Anodyne ADAM17 20 42 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625010 GF On-Demand Anodyne CCR3 57 37 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625010 GF On-Demand Anodyne MLNR 26 40 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625011 GF On-Demand Anodyne CCR3 57 37 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625011 GF On-Demand Anodyne MLNR 26 40 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCO1 ZINC000880625018 GF On-Demand Anodyne DGAT1 17 40 COC(=O)[C@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCO1 ZINC000880625019 GF On-Demand Anodyne DGAT1 17 40 CC(=O)N1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625020 GF On-Demand Anodyne PDGFRB 52 44 CC(=O)N1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625020 GF On-Demand Anodyne S1PR2 29 44 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(C1)OCCO2 ZINC000880625023 GG On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(C1)OCCO2 ZINC000880625023 GG On-Demand Anodyne EPHX2 36 40 O=C(NCC[C@@H](O)C(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880625024 FF On-Demand Anodyne ADRB1 40 31 O=C(NCC[C@@H](O)C(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880625024 FF On-Demand Anodyne ROCK1 15 40 O=C(NCC[C@H](O)C(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880625025 FF On-Demand Anodyne ADRB1 40 31 O=C(NCC[C@H](O)C(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880625025 FF On-Demand Anodyne ROCK1 15 40 CC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625027 FH On-Demand Anodyne ADAM17 42 35 CC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625027 FH On-Demand Anodyne CPT1A 66 42 CC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625027 FH On-Demand Anodyne SCD1 15 44 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625035 GH On-Demand Anodyne CCR3 31 45 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625035 GH On-Demand Anodyne MLNR 34 40 CONC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625036 GF On-Demand Anodyne CPT1A 52 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCO[C@H]1c1cccnc1 ZINC000880625037 GH On-Demand Anodyne CPT1A 20 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCN(CCO)CC1 ZINC000880625039 GE On-Demand Anodyne PDGFRB 52 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCN(CCO)CC1 ZINC000880625039 GE On-Demand Anodyne FAAH 20 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCN(CCO)CC1 ZINC000880625039 GE On-Demand Anodyne S1PR2 29 43 COC[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625041 GI On-Demand Anodyne PDGFRB 52 38 COC[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625041 GI On-Demand Anodyne CCR3 64 36 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](CO)C1 ZINC000880625043 FG On-Demand Anodyne PDGFRB 42 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](CO)C1 ZINC000880625043 FG On-Demand Anodyne CCR3 52 46 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](CO)C1 ZINC000880625044 FG On-Demand Anodyne PDGFRB 42 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](CO)C1 ZINC000880625044 FG On-Demand Anodyne CCR3 52 46 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCNC2=O)CC1 ZINC000880625061 GF On-Demand Anodyne NPY5R 27 42 CS(=O)(=O)Nc1cc2ccccc2cc1C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000880625066 HE On-Demand Anodyne PLAU 17 44 CS(=O)(=O)Nc1cc2ccccc2cc1C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000880625066 HE On-Demand Anodyne KCNK3 72 39 CS(=O)(=O)Nc1cc2ccccc2cc1C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000880625066 HE On-Demand Anodyne KCNK9 64 39 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(F)F ZINC000880625068 EG On-Demand Anodyne ROCK1 18 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC[C@@H]1O ZINC000880625084 ED On-Demand Anodyne ADAM17 21 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCOC[C@@H]1O ZINC000880625085 ED On-Demand Anodyne ADAM17 21 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC[C@H]1O ZINC000880625086 ED On-Demand Anodyne ADAM17 21 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCOC[C@H]1O ZINC000880625087 ED On-Demand Anodyne ADAM17 21 41 CC(=O)[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625090 FH On-Demand Anodyne CPT1A 75 42 CC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625091 FH On-Demand Anodyne CPT1A 75 42 CC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625097 GG On-Demand Anodyne HRH3 15 47 CC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625097 GG On-Demand Anodyne CCR3 39 40 CC(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625098 GG On-Demand Anodyne HRH3 15 47 CC(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625098 GG On-Demand Anodyne CCR3 39 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625163 GG On-Demand Anodyne CCR3 15 40 COCCO[C@@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625164 GG On-Demand Anodyne CCR3 15 40 COC[C@@H](O)CCNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625177 FF On-Demand Anodyne ADRB1 56 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)(F)CC1 ZINC000880625181 FH On-Demand Anodyne GRM5 15 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)(F)CC1 ZINC000880625181 FH On-Demand Anodyne NPY5R 26 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCOCC2)C1 ZINC000880625189 GI On-Demand Anodyne S1PR2 27 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC2(CCOCC2)C1 ZINC000880625189 GI On-Demand Anodyne EPHX2 42 45 C[C@@H](O)CCN(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625194 FG On-Demand Anodyne NPY5R 27 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCC1 ZINC000880625197 DH On-Demand Anodyne HTR2C 15 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCC1 ZINC000880625197 DH On-Demand Anodyne PDGFRB 45 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCC1 ZINC000880625197 DH On-Demand Anodyne S1PR2 28 43 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCC1 ZINC000880625197 DH On-Demand Anodyne DGAT1 16 41 NC(=O)C[C@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625204 GG On-Demand Anodyne CCR3 50 34 NC(=O)C[C@@H]1CCCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625205 GG On-Demand Anodyne CCR3 50 34 CCOC[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625207 GI On-Demand Anodyne PDGFRB 47 37 CCOC[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625207 GI On-Demand Anodyne CCR3 27 46 CCOC[C@H]1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880625207 GI On-Demand Anodyne S1PR2 26 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CCO)CC1 ZINC000880625226 GH On-Demand Anodyne PDGFRB 46 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CCO)CC1 ZINC000880625226 GH On-Demand Anodyne CCR3 25 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CCO)CC1 ZINC000880625226 GH On-Demand Anodyne S1PR2 26 40 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625230 FH On-Demand Anodyne TIMP3 57 33 O=C(NCCOCCF)Nc1nc(COc2ccccc2)cs1 ZINC000880625231 EF On-Demand Anodyne ROCK1 15 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(OC2CCC2)CC1 ZINC000880625250 GI On-Demand Anodyne ALOX5 22 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(OC2CCC2)CC1 ZINC000880625250 GI On-Demand Anodyne CPT1A 56 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(OC2CCC2)CC1 ZINC000880625250 GI On-Demand Anodyne EPHX2 22 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(OC2CCC2)CC1 ZINC000880625250 GI On-Demand Anodyne SCD1 15 44 COCC(COC)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625257 FF On-Demand Anodyne ROCK1 18 48 CCOC(=O)CCN(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625259 FG On-Demand Anodyne LTA4H 18 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](CO)CC1 ZINC000880625273 FG On-Demand Anodyne CPT1A 45 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](CO)CC1 ZINC000880625275 FG On-Demand Anodyne CPT1A 45 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC(C(F)(F)F)C1 ZINC000880625276 FH On-Demand Anodyne RBP4 58 33 C[C@@H](F)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625296 DH On-Demand Anodyne ROCK1 19 41 CNC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625298 FE On-Demand Anodyne ADAM17 49 37 CNC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625298 FE On-Demand Anodyne CPT1A 54 38 C[C@H](CO)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625303 DF On-Demand Anodyne NPY5R 32 42 C[C@@H](CO)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625304 DF On-Demand Anodyne NPY5R 32 42 CN(C(=O)Nc1nc(COc2ccccc2)cs1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880625312 GH On-Demand Anodyne GLRA1 46 35 C[C@H](CCO)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625317 EF On-Demand Anodyne NPY5R 31 41 C[C@@H](CCO)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625318 EF On-Demand Anodyne NPY5R 31 41 COCC(C)(C)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625322 EH On-Demand Anodyne ROCK1 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCOCC2)CC1 ZINC000880625323 GI On-Demand Anodyne NPY5R 19 43 O=C(NC1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1)C1CC1 ZINC000880625328 FE On-Demand Anodyne ADAM17 42 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]2COC[C@@H]21 ZINC000880625330 FG On-Demand Anodyne CPT1A 93 42 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H](F)C[C@H]1CO ZINC000880625331 FF On-Demand Anodyne ITGA4 43 37 COC(OC)[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625362 FF On-Demand Anodyne ROCK1 16 41 COC(OC)[C@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625363 FF On-Demand Anodyne ROCK1 16 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880625379 ED On-Demand Anodyne CPT1A 44 38 NC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625384 FE On-Demand Anodyne CPT1A 71 41 NC(=O)[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625385 FE On-Demand Anodyne CPT1A 71 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1[C@H]1CCCO1 ZINC000880625391 FH On-Demand Anodyne CPT1A 110 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(CO)(CO)CC1 ZINC000880625392 GE On-Demand Anodyne NPY5R 22 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@H]1CCCO1 ZINC000880625393 FH On-Demand Anodyne CPT1A 110 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1[C@@H]1CCCO1 ZINC000880625394 FH On-Demand Anodyne CPT1A 110 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@@H]1CCCO1 ZINC000880625396 FH On-Demand Anodyne CPT1A 110 42 CO[C@@H](C)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625408 EG On-Demand Anodyne ROCK1 19 40 CC(=O)NCCN(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625409 EE On-Demand Anodyne MTNR1A 25 44 CC(=O)NCCN(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625409 EE On-Demand Anodyne MTNR1B 24 44 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H](CO)[C@H]1CCCOC1 ZINC000880625413 GF On-Demand Anodyne ALOX5 24 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H](CO)[C@@H]1CCCOC1 ZINC000880625415 GF On-Demand Anodyne ALOX5 24 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H](CO)[C@@H]1CCCOC1 ZINC000880625416 GF On-Demand Anodyne ALOX5 24 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H](CO)[C@H]1CCCOC1 ZINC000880625418 GF On-Demand Anodyne ALOX5 24 40 O=C(NCC(=O)N1CCOCC1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625441 GE On-Demand Anodyne EPHX2 29 45 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880625449 FG On-Demand Anodyne RBP4 45 33 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880625450 FG On-Demand Anodyne RBP4 45 33 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880625452 FG On-Demand Anodyne RBP4 45 33 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880625454 FG On-Demand Anodyne RBP4 45 33 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880625455 FG On-Demand Anodyne RBP4 45 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880625457 GH On-Demand Anodyne CPT1A 140 49 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880625457 GH On-Demand Anodyne CPT2 44 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880625458 GH On-Demand Anodyne CPT1A 140 49 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880625458 GH On-Demand Anodyne CPT2 44 42 COC[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625469 EG On-Demand Anodyne CPT1A 115 44 CC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625472 DF On-Demand Anodyne ADRB1 43 33 CC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625472 DF On-Demand Anodyne ROCK1 19 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1nc(COc3ccccc3)cs1)C2 ZINC000880625479 FG On-Demand Anodyne HTR3A 32 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1nc(COc3ccccc3)cs1)C2 ZINC000880625479 FG On-Demand Anodyne SLC6A5 29 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1nc(COc3ccccc3)cs1)C2 ZINC000880625479 FG On-Demand Anodyne GLRA1 47 36 CO[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625495 FH On-Demand Anodyne CPT1A 51 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880625498 GE On-Demand Anodyne FAAH 22 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CC1)OCCCO2 ZINC000880625501 GG On-Demand Anodyne NPY5R 15 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCOCC1 ZINC000880625520 EG On-Demand Anodyne EPHX2 27 40 O=C(NCCCOCCO)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625535 FF On-Demand Anodyne ADRB1 41 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)[C@H]2CCCC[C@@H]21 ZINC000880625538 GH On-Demand Anodyne CPT1A 90 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)[C@H]2CCCC[C@H]21 ZINC000880625539 GH On-Demand Anodyne CPT1A 90 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)[C@@H]2CCCC[C@H]21 ZINC000880625540 GH On-Demand Anodyne CPT1A 90 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)[C@@H]2CCCC[C@@H]21 ZINC000880625541 GH On-Demand Anodyne CPT1A 90 41 CN(C)C[C@@H]1CN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CCO1 ZINC000880625544 GF On-Demand Anodyne MLNR 27 40 COC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625546 GH On-Demand Anodyne PDGFRB 47 38 COC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625546 GH On-Demand Anodyne S1PR2 27 41 COC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625546 GH On-Demand Anodyne DGAT1 22 40 COC(=O)C1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625546 GH On-Demand Anodyne PTR1 46 35 C[C@H](CS(C)(=O)=O)N(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625556 GG On-Demand Anodyne NPY5R 32 45 CON(C)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625565 EE On-Demand Anodyne ROCK1 17 41 COC1(C)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625566 FH On-Demand Anodyne NPY5R 21 42 CN(CC(=O)N1CCCC1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625569 FF On-Demand Anodyne CPT1A 89 41 C#CC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880625582 EH On-Demand Mild CPT1A 53 38 CN1C(=O)N[C@@H]2CN(C(=O)Nc3nc(COc4ccccc4)cs3)CC[C@@H]21 ZINC000880625597 GE On-Demand Anodyne ADAM17 52 37 CS(=O)(=O)C1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880625598 FD On-Demand Anodyne ADAM17 41 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880625602 GI On-Demand Anodyne CPT1A 137 49 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880625602 GI On-Demand Anodyne CPT2 43 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880625603 GI On-Demand Anodyne CPT1A 137 49 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880625603 GI On-Demand Anodyne CPT2 43 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CC1)CC2(F)F ZINC000880625619 GI On-Demand Anodyne NPY5R 17 42 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H](CO)CCF ZINC000880625622 EF On-Demand Anodyne ROCK1 17 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H](CO)CCF ZINC000880625623 EF On-Demand Anodyne ROCK1 17 41 O=C(NCC1=CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880625644 EG On-Demand Anodyne ROCK1 16 42 Cc1nnc([C@@H]2CCCN(C(=O)Nc3nc(COc4ccccc4)cs3)C2)o1 ZINC000880625652 GH On-Demand Anodyne CPT1A 43 37 Cc1nnc(CCNC(=O)Nc2nc(COc3ccccc3)cs2)s1 ZINC000880625654 GG On-Demand Anodyne ROCK1 15 42 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCCN(CCCO)C1 ZINC000880625659 GF On-Demand Anodyne SLC6A1 55 39 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCCN(CCCO)C1 ZINC000880625659 GF On-Demand Anodyne CCR3 27 43 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCCN(CCCO)C1 ZINC000880625659 GF On-Demand Anodyne SLC6A5 34 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCCN(CCCO)C1 ZINC000880625660 GF On-Demand Anodyne SLC6A1 55 39 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCCN(CCCO)C1 ZINC000880625660 GF On-Demand Anodyne CCR3 27 43 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCCN(CCCO)C1 ZINC000880625660 GF On-Demand Anodyne SLC6A5 34 40 O=C(NC[C@H](O)C1CC1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625740 EG On-Demand Anodyne PRMT3 25 43 O=C(NC[C@@H](O)C1CC1)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625741 EG On-Demand Anodyne PRMT3 25 43 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625746 GG On-Demand Anodyne SLC6A3 28 41 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625747 GG On-Demand Anodyne SLC6A3 28 41 C[C@@H](CC[S@@](C)=O)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625751 GG On-Demand Anodyne CCR3 48 33 C[C@@H](CC[S@](C)=O)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625752 GG On-Demand Anodyne CCR3 48 33 C[C@H](CC[S@](C)=O)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625753 GG On-Demand Anodyne CCR3 48 33 C[C@H](CC[S@@](C)=O)NC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880625754 GG On-Demand Anodyne CCR3 48 33 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H]1CO ZINC000880625764 EG On-Demand Anodyne CCR3 18 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H]1CO ZINC000880625765 EG On-Demand Anodyne CCR3 18 42 O=C(Nc1nc(COc2ccccc2)cs1)N1OC2CCC1CC2 ZINC000880625789 EH On-Demand Anodyne CPT1A 41 39 COC[C@@H]1CCCN1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625790 FF On-Demand Anodyne CPT1A 77 40 COC[C@@H]1CCCN1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625790 FF On-Demand Anodyne CHRNA10 41 39 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2COC[C@H]2C1 ZINC000880625806 EF On-Demand Anodyne RBP4 43 32 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)CC1 ZINC000880625807 EH On-Demand Anodyne CPT1A 52 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)CC1 ZINC000880625807 EH On-Demand Anodyne GRM5 15 40 CC(=O)OC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625817 GH On-Demand Anodyne PDGFRB 42 38 CC(=O)OC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880625817 GH On-Demand Anodyne S1PR2 27 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCO[C@H]1c1ccncc1 ZINC000880625823 GH On-Demand Anodyne CPT1A 19 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCO[C@H]1c1ccncc1 ZINC000880625823 GH On-Demand Anodyne ROCK1 20 40 Cc1nn(C)cc1[C@@H]1OCC[C@H]1NC(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880625824 FD On-Demand Anodyne HTR1F 51 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](O)C1 ZINC000880625838 EF On-Demand Anodyne CPT1A 58 39 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1CCCC[C@H]1O ZINC000880625841 EG On-Demand Anodyne CPT1A 62 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@@]2(CCCOC2)C1 ZINC000880625846 GG On-Demand Anodyne EPHX2 16 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@]2(CCCOC2)C1 ZINC000880625847 GG On-Demand Anodyne EPHX2 16 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2ccon2)CC1 ZINC000880625853 GI On-Demand Anodyne CPT1A 61 37 COC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625857 ED On-Demand Anodyne ADRB2 37 41 COC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625857 ED On-Demand Anodyne ADRB1 63 40 COC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625857 ED On-Demand Anodyne ADRB3 37 40 COC[C@@H](O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625857 ED On-Demand Anodyne ROCK1 17 43 CCc1nnc(CNC(=O)Nc2nc(COc3ccccc3)cs2)s1 ZINC000880625865 GG On-Demand Anodyne ROCK1 15 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2ccncn2)CC1 ZINC000880625868 GH On-Demand Anodyne CPT1A 50 41 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)[C@@H](C)O ZINC000880625876 DF On-Demand Anodyne ROCK1 18 42 CN1CC[C@H](N(C)C(=O)Nc2nc(COc3ccccc3)cs2)C1=O ZINC000880625888 FE On-Demand Anodyne CPT1A 47 38 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CC[C@@H](C)O1 ZINC000880625894 FH On-Demand Anodyne CPT1A 43 38 O=C(NCCCCF)Nc1nc(COc2ccccc2)cs1 ZINC000880625897 DH On-Demand Anodyne ROCK1 20 45 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(C2CCC2)CC1 ZINC000880625902 GH On-Demand Anodyne CPT1A 40 37 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(C2CCC2)CC1 ZINC000880625902 GH On-Demand Anodyne SLC6A5 36 45 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(C2CCC2)CC1 ZINC000880625902 GH On-Demand Anodyne EPHX2 28 41 CCNC(=O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625910 ED On-Demand Anodyne ROCK1 20 41 COCC[C@H]1COCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625912 GF On-Demand Anodyne CPT1A 49 38 COCC[C@@H]1COCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625913 GF On-Demand Anodyne CPT1A 49 38 C[C@@H](CF)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880625928 DG On-Demand Anodyne ROCK1 19 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(n2ccnc2)CC1 ZINC000880626014 GI On-Demand Anodyne S1PR2 27 42 CCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626015 GH On-Demand Anodyne CACNA1H 40 41 CCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626015 GH On-Demand Anodyne PDGFRB 50 40 CCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626015 GH On-Demand Anodyne S1PR2 38 56 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]2CC[C@@H](O)[C@@H]21 ZINC000880626016 FG On-Demand Anodyne CPT1A 53 40 COC(=O)C[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626022 EF On-Demand Anodyne ROCK1 15 40 COCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626026 GG On-Demand Anodyne CACNA1H 44 41 COCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626026 GG On-Demand Anodyne PDGFRB 54 39 COCC1(O)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626026 GG On-Demand Anodyne S1PR2 36 53 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(c2ncc[nH]2)CC1 ZINC000880626027 GI On-Demand Anodyne S1PR2 24 40 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626035 GG On-Demand Anodyne CCR3 47 44 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626035 GG On-Demand Anodyne MLNR 40 39 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626035 GG On-Demand Anodyne EPHX2 56 52 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626036 GG On-Demand Anodyne CCR3 47 44 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626036 GG On-Demand Anodyne MLNR 40 39 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)C1 ZINC000880626036 GG On-Demand Anodyne EPHX2 56 52 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)NC1CCOCC1 ZINC000880626045 EG On-Demand Anodyne EPHX2 57 43 CCOCCNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880626051 EG On-Demand Anodyne ADRB1 41 36 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](CF)C1 ZINC000880626062 EH On-Demand Anodyne CPT1A 42 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](CF)C1 ZINC000880626063 EH On-Demand Anodyne CPT1A 42 37 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)CC1 ZINC000880626064 FG On-Demand Anodyne PDGFRB 48 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)CC1 ZINC000880626064 FG On-Demand Anodyne CCR3 27 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)CC1 ZINC000880626064 FG On-Demand Anodyne S1PR2 27 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC(CO)CC1 ZINC000880626064 FG On-Demand Anodyne EPHX2 17 53 COCC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626075 GI On-Demand Anodyne PDGFRB 53 39 COCC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626075 GI On-Demand Anodyne CCR3 27 44 COCC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626075 GI On-Demand Anodyne S1PR2 28 41 COCC1CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626075 GI On-Demand Anodyne EPHX2 15 42 Cn1c(S)nnc1CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626094 GF On-Demand Anodyne ROCK1 15 43 COC[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626097 GI On-Demand Anodyne CPT1A 65 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1Cn1ccnn1 ZINC000880626110 GG On-Demand Anodyne CPT1A 75 41 O=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626119 FG On-Demand Anodyne CPT1A 47 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC1=O ZINC000880626130 EE On-Demand Anodyne NAAA 23 42 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC1=O ZINC000880626130 EE On-Demand Anodyne LUXR 78 47 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC1=O ZINC000880626130 EE On-Demand Anodyne TRAR 95 45 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCOC1=O ZINC000880626130 EE On-Demand Anodyne LASR 60 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]1C(F)(F)F ZINC000880626136 FH On-Demand Anodyne CPT1A 53 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]1C(F)(F)F ZINC000880626138 FH On-Demand Anodyne CPT1A 53 39 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@]2(CCOC2)C1 ZINC000880626156 GH On-Demand Anodyne S1PR2 26 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@]2(CCOC2)C1 ZINC000880626156 GH On-Demand Anodyne EPHX2 38 42 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@]2(CCOC2)C1 ZINC000880626160 GH On-Demand Anodyne S1PR2 26 40 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CC[C@@]2(CCOC2)C1 ZINC000880626160 GH On-Demand Anodyne EPHX2 38 42 C[C@H](O)CN(C)C(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1 ZINC000880626173 EF On-Demand Anodyne NPY5R 27 40 COC[C@@H](CCNC(=O)Nc1nc(COc2ccccc2)cs1)OC ZINC000880626180 FF On-Demand Anodyne ROCK1 17 41 COCC[C@@H](C)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626181 EH On-Demand Anodyne ROCK1 18 42 COCC[C@H](C)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626182 EH On-Demand Anodyne ROCK1 18 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(C(=O)C2CC2)C1 ZINC000880626199 FF On-Demand Anodyne CPT1A 56 39 CC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626248 GH On-Demand Anodyne CACNA1H 40 41 CC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626248 GH On-Demand Anodyne PDGFRB 44 40 CC1(CO)CCN(C(=O)Nc2ccc(Oc3cc(F)cc(F)c3)nc2)CC1 ZINC000880626248 GH On-Demand Anodyne S1PR2 32 47 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCCS(=O)(=O)CC1 ZINC000880626250 GF On-Demand Anodyne S1PR2 27 41 COC[C@@H](CNC(=O)Nc1ccc(Oc2cc(F)cc(F)c2)nc1)OC ZINC000880626259 FF On-Demand Anodyne ADRB1 48 36 CCC1(N(C)C)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626268 GI On-Demand Anodyne NPY5R 17 41 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@H](CCO)C1 ZINC000880626270 GH On-Demand Anodyne CCR3 45 45 O=C(Nc1ccc(Oc2cc(F)cc(F)c2)nc1)N1CCC[C@@H](CCO)C1 ZINC000880626271 GH On-Demand Anodyne CCR3 45 45 C[C@@H]1CC[C@H](O)CN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626291 EG On-Demand Anodyne CPT1A 52 41 Cn1nnnc1C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626293 GF On-Demand Anodyne IL2RA 49 30 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCCC2=O)CC1 ZINC000880626364 GI On-Demand Anodyne NPY5R 30 43 C#C[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626366 EH On-Demand Mild CPT1A 66 38 C#C[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626368 EH On-Demand Mild CPT1A 66 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(O)(CO)CC1 ZINC000880626370 FE On-Demand Anodyne NPY5R 19 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880626372 EH On-Demand Anodyne RBP4 47 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]2C[C@H]2C1 ZINC000880626374 EH On-Demand Anodyne RBP4 47 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]2C[C@@H]2C1 ZINC000880626376 EH On-Demand Anodyne RBP4 47 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]2C[C@H]2C1 ZINC000880626378 EH On-Demand Anodyne RBP4 47 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]1C(F)F ZINC000880626404 EH On-Demand Anodyne ALOX5 20 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]1C(F)F ZINC000880626404 EH On-Demand Anodyne CPT1A 58 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]1C(F)F ZINC000880626405 EH On-Demand Anodyne ALOX5 20 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]1C(F)F ZINC000880626405 EH On-Demand Anodyne CPT1A 58 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CC1)OCCO2 ZINC000880626410 GG On-Demand Anodyne NPY5R 19 44 O=C(NCC1CCC(O)CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626412 FG On-Demand Anodyne GRIN2B 19 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](c2cccnc2)C1 ZINC000880626416 GI On-Demand Anodyne CPT1A 57 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](c2cccnc2)C1 ZINC000880626416 GI On-Demand Anodyne EPHX2 17 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](c2cccnc2)C1 ZINC000880626417 GI On-Demand Anodyne CPT1A 57 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](c2cccnc2)C1 ZINC000880626417 GI On-Demand Anodyne EPHX2 17 41 C[C@H](O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626418 GE On-Demand Anodyne ACOX1 52 36 CCO[C@H]1C[C@@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626423 EG On-Demand Anodyne TIMP3 57 33 CCO[C@@H]1C[C@@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626424 EG On-Demand Anodyne TIMP3 57 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H]1C1CC1 ZINC000880626434 EH On-Demand Anodyne CPT1A 71 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H]1C1CC1 ZINC000880626435 EH On-Demand Anodyne CPT1A 71 39 O=C(NOCCC1CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626436 EH On-Demand Anodyne GRIN2B 18 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](N2CCOCC2)C1 ZINC000880626440 GF On-Demand Anodyne CPT1A 41 36 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](N2CCOCC2)C1 ZINC000880626441 GF On-Demand Anodyne CPT1A 41 36 COCC[C@H](COC)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626446 FF On-Demand Anodyne ROCK1 15 45 COCC[C@@H](COC)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626447 FF On-Demand Anodyne ROCK1 15 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CC(C2CC2)C1 ZINC000880626449 EH On-Demand Anodyne RBP4 44 32 COC1(CO)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626451 GF On-Demand Anodyne NPY5R 24 41 Cn1nccc1[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626452 GH On-Demand Anodyne CPT1A 43 39 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626453 GH On-Demand Anodyne CPT1A 43 39 CC[C@@H](CNC(=O)Nc1nc(COc2ccccc2)cs1)OC ZINC000880626460 EG On-Demand Anodyne ROCK1 17 41 CC[C@@H](CNC(=O)Nc1nc(COc2ccccc2)cs1)OC ZINC000880626460 EG On-Demand Anodyne PDS 56 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOC[C@H]1[C@H]1CCCO1 ZINC000880626506 GG On-Demand Anodyne CPT1A 62 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOC[C@@H]1[C@H]1CCCO1 ZINC000880626507 GG On-Demand Anodyne CPT1A 62 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOC[C@H]1[C@@H]1CCCO1 ZINC000880626508 GG On-Demand Anodyne CPT1A 62 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOC[C@@H]1[C@@H]1CCCO1 ZINC000880626509 GG On-Demand Anodyne CPT1A 62 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](F)C1 ZINC000880626512 EH On-Demand Anodyne CPT1A 53 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](F)C1 ZINC000880626513 EH On-Demand Anodyne CPT1A 53 38 CC[C@@H](NC(=O)Nc1nc(COc2ccccc2)cs1)[C@@H](C)O ZINC000880626514 EG On-Demand Anodyne ROCK1 16 42 CC[C@@H](NC(=O)Nc1nc(COc2ccccc2)cs1)[C@H](C)O ZINC000880626517 EG On-Demand Anodyne ROCK1 16 42 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H]2CCCC[C@@H]21 ZINC000880626518 EI On-Demand Anodyne CPT1A 85 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCO2)CC1 ZINC000880626530 FH On-Demand Anodyne NPY5R 20 46 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCO2)CC1 ZINC000880626530 FH On-Demand Anodyne EPHX2 16 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC2(CCO2)CC1 ZINC000880626530 FH On-Demand Anodyne TRPM8 17 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@@H]1CCCOC1 ZINC000880626539 GI On-Demand Anodyne CPT1A 95 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@H]1CCCOC1 ZINC000880626540 GI On-Demand Anodyne CPT1A 95 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1[C@@H]1CCCOC1 ZINC000880626541 GI On-Demand Anodyne CPT1A 95 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1[C@H]1CCCOC1 ZINC000880626542 GI On-Demand Anodyne CPT1A 95 41 C[C@H]1C[C@H](O)CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626544 EF On-Demand Anodyne ADAM17 51 35 C[C@@H]1C[C@H](O)CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626545 EF On-Demand Anodyne ADAM17 51 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](F)C1 ZINC000880626549 DG On-Demand Anodyne CPT1A 48 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](F)C1 ZINC000880626550 DG On-Demand Anodyne CPT1A 48 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880626560 EF On-Demand Anodyne NPY5R 15 42 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(F)(F)F ZINC000880626564 EH On-Demand Anodyne ROCK1 20 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]2C[C@@H]21 ZINC000880626565 EH On-Demand Anodyne CPT1A 98 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]2C[C@H]21 ZINC000880626566 EH On-Demand Anodyne CPT1A 98 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]2C[C@H]21 ZINC000880626567 EH On-Demand Anodyne CPT1A 98 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]2C[C@@H]21 ZINC000880626568 EH On-Demand Anodyne CPT1A 98 41 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626578 EG On-Demand Anodyne ADAM17 41 38 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626578 EG On-Demand Anodyne CPT1A 112 43 C[C@H]1[C@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626580 EG On-Demand Anodyne ADAM17 41 38 C[C@H]1[C@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626580 EG On-Demand Anodyne CPT1A 112 43 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626581 EG On-Demand Anodyne ADAM17 41 38 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626581 EG On-Demand Anodyne CPT1A 112 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1CCO ZINC000880626582 EG On-Demand Anodyne CPT1A 91 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1CCO ZINC000880626583 EG On-Demand Anodyne CPT1A 91 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1C[C@H]2CCCCN2C1=O ZINC000880626586 GF On-Demand Anodyne CPT1A 76 38 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H]1C[C@@H]2CCCCN2C1=O ZINC000880626587 GF On-Demand Anodyne CPT1A 76 38 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1C[C@@H]2CCCCN2C1=O ZINC000880626588 GF On-Demand Anodyne CPT1A 76 38 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1C[C@H]2CCCCN2C1=O ZINC000880626589 GF On-Demand Anodyne CPT1A 76 38 CC[C@@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(=O)NC ZINC000880626671 EE On-Demand Anodyne ROCK1 15 42 CC[C@@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(=O)NC ZINC000880626671 EE On-Demand Anodyne ACE2 46 35 COCC1(NC(=O)Nc2nc(COc3ccccc3)cs2)CCC1 ZINC000880626683 EG On-Demand Anodyne ROCK1 15 41 C[S@@](=O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626692 EE On-Demand Anodyne ROCK1 16 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@@H]1CCC[C@@H]1O ZINC000880626694 GH On-Demand Anodyne CPT1A 85 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@H]1CCC[C@@H]1O ZINC000880626695 GH On-Demand Anodyne CPT1A 85 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@H]1CCC[C@H]1O ZINC000880626696 GH On-Demand Anodyne CPT1A 85 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1[C@@H]1CCC[C@H]1O ZINC000880626697 GH On-Demand Anodyne CPT1A 85 40 COC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@@H]1C ZINC000880626706 GG On-Demand Anodyne ADAM17 41 38 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCC1 ZINC000880626732 DG On-Demand Anodyne FAAH 23 41 O=C(Nc1nc(COc2ccccc2)cs1)N1[C@H]2CC[C@H]1COC2 ZINC000880626737 EG On-Demand Anodyne CPT1A 40 37 CC(C)[C@H]1CCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626746 EH On-Demand Anodyne ALOX5 29 40 CC(C)[C@H]1CCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626746 EH On-Demand Anodyne ADAM17 48 36 CC(C)[C@H]1CCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626746 EH On-Demand Anodyne CPT1A 69 41 O=C(Nc1nc(COc2ccccc2)cs1)N[C@@H](CO)C1CCC1 ZINC000880626750 EG On-Demand Anodyne ALOX5 24 40 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H](CO)C1CCC1 ZINC000880626751 EG On-Demand Anodyne ALOX5 24 40 C[C@H]1CC[C@@H](O)CN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626759 EG On-Demand Anodyne CPT1A 52 41 C[C@H]1CC[C@H](O)CN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626760 EG On-Demand Anodyne CPT1A 52 41 CC(=O)N[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626762 FE On-Demand Anodyne ADAM17 51 38 CC(=O)N[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626762 FE On-Demand Anodyne CPT1A 36 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626762 FE On-Demand Anodyne SLC6A5 32 43 CC(=O)N[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626763 FE On-Demand Anodyne ADAM17 51 38 CC(=O)N[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626763 FE On-Demand Anodyne CPT1A 36 40 CC(=O)N[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626763 FE On-Demand Anodyne SLC6A5 32 43 COCCCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626776 EH On-Demand Anodyne ROCK1 17 44 O=C(NCCN1CCCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626800 GF On-Demand Anodyne CASR 35 40 O=C(NCCN1CCCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626800 GF On-Demand Anodyne EPHX2 22 43 O=C(NCCN1CCCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626800 GF On-Demand Anodyne HPGDS 23 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880626804 GI On-Demand Anodyne GRIN2B 65 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880626804 GI On-Demand Anodyne CCR3 39 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](Cc2ccncc2)C1 ZINC000880626805 GI On-Demand Anodyne GRIN2B 65 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](Cc2ccncc2)C1 ZINC000880626805 GI On-Demand Anodyne CCR3 39 43 COC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626811 GG On-Demand Anodyne CPT1A 68 39 COC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626811 GG On-Demand Anodyne SCD1 17 46 COC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626811 GG On-Demand Anodyne PTR1 48 35 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C1CCOCC1 ZINC000880626814 FH On-Demand Anodyne GCK 16 42 Cn1cnnc1[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626815 GG On-Demand Anodyne CPT1A 110 43 Cn1cnnc1[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626816 GG On-Demand Anodyne CPT1A 110 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](C2CC2)C1 ZINC000880626827 EH On-Demand Anodyne RBP4 43 31 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](C2CC2)C1 ZINC000880626828 EH On-Demand Anodyne RBP4 43 31 COCC1(O)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880626835 GF On-Demand Anodyne NPY5R 19 41 CCOCCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626838 EH On-Demand Anodyne ROCK1 15 40 CCC(=O)N1CC[C@@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626839 FF On-Demand Anodyne SLC6A5 31 41 CCC(=O)N1CC[C@@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626839 FF On-Demand Anodyne EPHX2 36 52 CCC(=O)N1CC[C@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626841 FF On-Demand Anodyne SLC6A5 31 41 CCC(=O)N1CC[C@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626841 FF On-Demand Anodyne EPHX2 36 52 O=C1NCC2(CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)O1 ZINC000880626843 GF On-Demand Anodyne NPY5R 19 49 O=C1NCC2(CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)O1 ZINC000880626843 GF On-Demand Anodyne TRPM8 21 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](N2CC=CC2)C1 ZINC000880626844 FG On-Demand Anodyne CPT1A 44 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](N2CC=CC2)C1 ZINC000880626846 FG On-Demand Anodyne CPT1A 44 37 COC(=O)C[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626847 GG On-Demand Anodyne CPT1A 84 41 COC(=O)C[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880626848 GG On-Demand Anodyne CPT1A 84 41 O=C(NCC1(CCO)CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880626850 EG On-Demand Anodyne ROCK1 17 41 C[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626857 EH On-Demand Anodyne ADAM17 47 36 C[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626857 EH On-Demand Anodyne CPT1A 77 41 C[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626857 EH On-Demand Anodyne TRPC6 44 36 O=C(NCCCF)Nc1nc(COc2ccccc2)cs1 ZINC000880626863 DG On-Demand Anodyne ROCK1 19 45 CC[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@H]1O ZINC000880626880 EF On-Demand Anodyne ADAM17 52 36 CC[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@@H]1O ZINC000880626881 EF On-Demand Anodyne ADAM17 52 36 CC[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626908 EH On-Demand Anodyne ADAM17 47 36 CC[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626908 EH On-Demand Anodyne CPT1A 45 38 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H](F)C[C@@H]1CO ZINC000880626911 FF On-Demand Anodyne ITGA4 43 37 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H](F)C[C@@H]1CO ZINC000880626912 FF On-Demand Anodyne ITGA4 43 37 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H](F)C[C@H]1CO ZINC000880626913 FF On-Demand Anodyne ITGA4 43 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@]2(O)CCCC[C@@H]2C1 ZINC000880626934 GH On-Demand Anodyne CPT1A 41 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@]2(O)CCCC[C@H]2C1 ZINC000880626935 GH On-Demand Anodyne CPT1A 41 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@]2(O)CCCC[C@@H]2C1 ZINC000880626936 GH On-Demand Anodyne CPT1A 41 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@]2(O)CCCC[C@H]2C1 ZINC000880626937 GH On-Demand Anodyne CPT1A 41 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(CCO)CC1 ZINC000880626955 FD On-Demand Anodyne FAAH 25 41 COCCO[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626967 GF On-Demand Anodyne CPT1A 57 38 COCCO[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626968 GF On-Demand Anodyne CPT1A 57 38 O=C(NCCCCCO)Nc1nc(COc2ccccc2)cs1 ZINC000880626970 EG On-Demand Anodyne ROCK1 16 42 COC[C@@H](CNC(=O)Nc1nc(COc2ccccc2)cs1)OC ZINC000880626976 FF On-Demand Anodyne ROCK1 17 43 CC(=O)N1CCC[C@@H](CNC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626981 GG On-Demand Anodyne ADAM17 42 35 CC(=O)N1CCC[C@H](CNC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880626982 GG On-Demand Anodyne ADAM17 42 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCOCC1 ZINC000880626998 EF On-Demand Anodyne ADAM17 23 40 O=C(NCC1(N2CCOCC2)CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627007 GF On-Demand Anodyne HCN1 73 38 O=C(NCC1(N2CCOCC2)CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627007 GF On-Demand Anodyne HCN4 50 32 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](c2ccccn2)C1 ZINC000880627015 GI On-Demand Anodyne CPT1A 75 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](c2ccccn2)C1 ZINC000880627016 GI On-Demand Anodyne CPT1A 75 42 O=C(NCCCCO)Nc1nc(COc2ccccc2)cs1 ZINC000880627019 DF On-Demand Anodyne ROCK1 16 43 Cc1noc(C2CN(C(=O)Nc3nc(COc4ccccc4)cs3)C2)n1 ZINC000880627021 FG On-Demand Anodyne CPT1A 60 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOC2(CCC2)C1 ZINC000880627025 FH On-Demand Anodyne EPHX2 19 45 C[C@]1(O)CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627042 FG On-Demand Anodyne NPY5R 24 41 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627048 DH On-Demand Anodyne ADAM17 49 37 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627048 DH On-Demand Anodyne CPT1A 56 39 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627048 DH On-Demand Anodyne EPHX2 17 40 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627048 DH On-Demand Anodyne TRPC6 42 41 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627048 DH On-Demand Anodyne TRPC3 35 41 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627049 DH On-Demand Anodyne ADAM17 49 37 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627049 DH On-Demand Anodyne CPT1A 56 39 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627049 DH On-Demand Anodyne EPHX2 17 40 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627049 DH On-Demand Anodyne TRPC6 42 41 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627049 DH On-Demand Anodyne TRPC3 35 41 C=C(C)COCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627057 EG On-Demand Mild ROCK1 17 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCCO1 ZINC000880627079 DG On-Demand Anodyne CPT1A 63 40 C[C@@]1(CO)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627080 EG On-Demand Anodyne SLC12A5 54 33 C[C@]1(CO)CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627081 EG On-Demand Anodyne SLC12A5 54 33 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(=O)N1CCCC1 ZINC000880627082 FF On-Demand Anodyne CPT1A 43 38 O=C(NNC(=O)C1CCCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627090 FG On-Demand Reactive CPT1A 99 42 O=C(NCCC(=O)N1CCCCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627091 GG On-Demand Anodyne CPT1A 52 38 CNC(=O)[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627094 ED On-Demand Anodyne ROCK1 16 40 O=C(NCC1(CO)COC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627101 ED On-Demand Anodyne ROCK1 16 40 COc1cc(Br)ccc1NC(=O)N1CCn2ccnc2C1 ZINC000880627104 FF On-Demand Anodyne PDGFRB 18 41 COc1cc(Br)ccc1NC(=O)N1CCC(C#N)CC1 ZINC000880627108 EG On-Demand Mild RBP4 23 40 COc1cc(Br)ccc1NC(=O)NC1CCN(OC)CC1 ZINC000880627117 FF On-Demand Anodyne EPHX2 39 45 COc1cc(Br)ccc1NC(=O)NCCCN1CCC[C@H]1C(N)=O ZINC000880627134 GD On-Demand Anodyne ACKR3 51 33 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880627140 DG On-Demand Anodyne DPP4 15 44 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880627140 DG On-Demand Anodyne RBP4 41 42 COc1cc(Br)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880627141 DG On-Demand Anodyne DPP4 15 44 COc1cc(Br)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880627141 DG On-Demand Anodyne RBP4 41 42 COC[C@@H]1CCCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880627142 FH On-Demand Anodyne PDGFRB 35 41 COC[C@@H]1CCCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880627142 FH On-Demand Anodyne PTPN2 18 40 COC[C@@H]1CCCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880627142 FH On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H]2C[C@@H]2C1 ZINC000880627146 EG On-Demand Anodyne RBP4 48 35 COc1cc(Br)ccc1NC(=O)N1CC[C@H]2C[C@H]2C1 ZINC000880627147 EG On-Demand Anodyne RBP4 48 35 COc1cc(Br)ccc1NC(=O)N1CC[C@H]2C[C@@H]2C1 ZINC000880627148 EG On-Demand Anodyne RBP4 48 35 COc1cc(Br)ccc1NC(=O)N1CC[C@@H]2C[C@H]2C1 ZINC000880627149 EG On-Demand Anodyne RBP4 48 35 COc1cc(Br)ccc1NC(=O)Nc1cnn(CCN(C)C)c1 ZINC000880627151 GF On-Demand Anodyne HTR2A 25 42 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C2CC2)C1 ZINC000880627154 FF On-Demand Anodyne PDGFRB 20 42 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C2CC2)C1 ZINC000880627154 FF On-Demand Anodyne RBP4 19 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880627163 GF On-Demand Anodyne PDGFRB 28 42 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880627163 GF On-Demand Anodyne RBP4 24 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](Nc2ncccn2)C1 ZINC000880627164 GF On-Demand Anodyne PDGFRB 28 42 COc1cc(Br)ccc1NC(=O)N1CC[C@H](Nc2ncccn2)C1 ZINC000880627164 GF On-Demand Anodyne RBP4 24 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1C ZINC000880627214 EF On-Demand Anodyne DRD2 48 50 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1C ZINC000880627214 EF On-Demand Anodyne DRD4 17 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1C ZINC000880627214 EF On-Demand Anodyne DRD3 21 52 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1C ZINC000880627214 EF On-Demand Anodyne CHRNA10 56 38 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1C ZINC000880627214 EF On-Demand Anodyne ACKR3 78 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1C ZINC000880627216 EF On-Demand Anodyne DRD2 48 50 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1C ZINC000880627216 EF On-Demand Anodyne DRD4 17 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1C ZINC000880627216 EF On-Demand Anodyne DRD3 21 52 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1C ZINC000880627216 EF On-Demand Anodyne CHRNA10 56 38 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1C ZINC000880627216 EF On-Demand Anodyne ACKR3 78 40 C[C@@H](CCCO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627239 EG On-Demand Anodyne ROCK1 16 40 CN(CC1CCOCC1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627242 FH On-Demand Anodyne GCK 15 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](O)C1 ZINC000880627251 EF On-Demand Anodyne CPT1A 58 39 O=C(Nc1nc(COc2ccccc2)cs1)N[C@H]1CCCC[C@@H]1O ZINC000880627254 EG On-Demand Anodyne CPT1A 62 40 O=C(NCCC(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627260 EH On-Demand Anodyne ROCK1 15 42 CC#CCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627263 DG On-Demand Mild ROCK1 16 41 O=C(NNC(=O)C1CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627264 EE On-Demand Reactive CPT1A 53 39 CS(=O)(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627282 GF On-Demand Anodyne ADAM17 43 35 CS(=O)(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627282 GF On-Demand Anodyne CPT1A 47 38 CN(C)C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627285 FG On-Demand Anodyne GRIN2B 42 37 CN(C)C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627285 FG On-Demand Anodyne ADAM17 40 35 N#CCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627298 DG On-Demand Mild ADRB1 44 33 N#CCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627298 DG On-Demand Mild ROCK1 15 41 CN(C[C@@H]1CCn2ccnc2C1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627310 GH On-Demand Anodyne CPT1A 47 36 COC(=O)N1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627314 GG On-Demand Anodyne EPHX2 48 45 Cn1nc2c(cc1=O)CN(C(=O)Nc1nc(COc3ccccc3)cs1)CC2 ZINC000880627318 GE On-Demand Anodyne GRM5 17 40 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2CCC[C@@H]21 ZINC000880627321 EH On-Demand Anodyne CPT1A 60 39 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H]2CCC[C@H]21 ZINC000880627322 EH On-Demand Anodyne CPT1A 60 39 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H]2CCC[C@H]21 ZINC000880627323 EH On-Demand Anodyne CPT1A 60 39 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H]2CCC[C@@H]21 ZINC000880627324 EH On-Demand Anodyne CPT1A 60 39 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CS(C)(=O)=O ZINC000880627332 GE On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CS(C)(=O)=O ZINC000880627332 GE On-Demand Anodyne ACKR3 62 32 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccncn2)CC1 ZINC000880627344 GH On-Demand Anodyne PDGFRB 27 42 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccncn2)CC1 ZINC000880627344 GH On-Demand Anodyne RBP4 26 40 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)N(C)C)CC1 ZINC000880627361 GE On-Demand Anodyne PDGFRB 24 43 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)N(C)C)CC1 ZINC000880627361 GE On-Demand Anodyne RBP4 20 42 COc1cc(Br)ccc1NC(=O)N(C)CCNC(C)=O ZINC000880627365 EE On-Demand Anodyne NQO2 53 32 COc1cc(Br)ccc1NC(=O)N1CCC(=O)N(C)CC1 ZINC000880627371 FE On-Demand Anodyne PDGFRB 33 43 COc1cc(Br)ccc1NC(=O)N1CCC(=O)N(C)CC1 ZINC000880627371 FE On-Demand Anodyne RBP4 21 40 COc1cc(Br)ccc1NC(=O)N1CCC=C(Cl)C1 ZINC000880627374 EH On-Demand Anodyne RBP4 21 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](N2CCOCC2)C1 ZINC000880627376 GE On-Demand Anodyne LRRK2 30 43 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](N2CCOCC2)C1 ZINC000880627376 GE On-Demand Anodyne L3MBTL3 41 35 COc1cc(Br)ccc1NC(=O)N1CC[C@H](N2CCOCC2)C1 ZINC000880627377 GE On-Demand Anodyne LRRK2 30 43 COc1cc(Br)ccc1NC(=O)N1CC[C@H](N2CCOCC2)C1 ZINC000880627377 GE On-Demand Anodyne L3MBTL3 41 35 COc1cc(Br)ccc1NC(=O)N1CCc2nccnc2C1 ZINC000880627378 FF On-Demand Anodyne PDGFRB 26 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CCO)CC1 ZINC000880627414 FG On-Demand Anodyne PDGFRB 31 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CCO)CC1 ZINC000880627414 FG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CCO)CC1 ZINC000880627414 FG On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CCO)CC1 ZINC000880627415 FG On-Demand Anodyne PDGFRB 31 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CCO)CC1 ZINC000880627415 FG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CCO)CC1 ZINC000880627415 FG On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2cccnc2)C1 ZINC000880627426 GH On-Demand Anodyne CHRNA7 27 44 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2cccnc2)C1 ZINC000880627427 GH On-Demand Anodyne CHRNA7 27 44 COCC1(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627436 EG On-Demand Anodyne ROCK1 15 42 C[C@H](C#N)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627453 DG On-Demand Mild ADRB1 41 31 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC([C@H]2CCCO2)CC1 ZINC000880627457 GI On-Demand Anodyne CPT1A 61 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC([C@@H]2CCCO2)CC1 ZINC000880627458 GI On-Demand Anodyne CPT1A 61 39 O=C(NCC[C@@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627461 GG On-Demand Anodyne ADRB1 40 31 O=C(NCC[C@@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627461 GG On-Demand Anodyne ROCK1 17 42 O=C(NCC[C@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627462 GG On-Demand Anodyne ADRB1 40 31 O=C(NCC[C@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627462 GG On-Demand Anodyne ROCK1 17 42 CN1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627471 EF On-Demand Anodyne FAAH 15 40 CC[C@@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627479 EG On-Demand Anodyne ADRB1 43 33 CC[C@@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627479 EG On-Demand Anodyne ROCK1 18 40 CC[C@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627480 EG On-Demand Anodyne ADRB1 43 33 CC[C@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627480 EG On-Demand Anodyne ROCK1 18 40 O=C(NC[C@@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627496 FF On-Demand Anodyne ROCK1 19 40 O=C(NC[C@H](O)C(F)(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627497 FF On-Demand Anodyne ROCK1 19 40 COC[C@@H]1CCCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627501 GI On-Demand Anodyne CPT1A 111 43 COC(=O)[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@@H]1C ZINC000880627504 GG On-Demand Anodyne CPT1A 51 38 COC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@@H]1C ZINC000880627505 GG On-Demand Anodyne CPT1A 51 38 COC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@H]1C ZINC000880627506 GG On-Demand Anodyne CPT1A 51 38 C[C@@H]1CCOCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627508 EG On-Demand Anodyne CPT1A 74 42 C[C@H]1CCOCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627509 EG On-Demand Anodyne CPT1A 74 42 CC(=O)OC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627515 GG On-Demand Anodyne CPT1A 42 39 CC(=O)OC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627515 GG On-Demand Anodyne SCD1 19 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880627516 GH On-Demand Anodyne CPT1A 24 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880627516 GH On-Demand Anodyne EPHX2 21 48 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@H]1CO ZINC000880627517 EF On-Demand Anodyne CPT1A 54 39 C[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@@H]1CO ZINC000880627518 EF On-Demand Anodyne CPT1A 54 39 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@@H]1CO ZINC000880627519 EF On-Demand Anodyne CPT1A 54 39 C[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)[C@H]1CO ZINC000880627520 EF On-Demand Anodyne CPT1A 54 39 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)CC#N)CC1 ZINC000880627541 GE On-Demand Mild PDGFRB 27 40 COc1cc(Br)ccc1NC(=O)N1CCC(Cn2cnnc2)CC1 ZINC000880627559 GF On-Demand Anodyne PDGFRB 31 41 COc1cc(Br)ccc1NC(=O)N1CCCN(C=O)CC1 ZINC000880627576 FE On-Demand Anodyne PDGFRB 22 41 COc1cc(Br)ccc1NC(=O)N1CCCN(C=O)CC1 ZINC000880627576 FE On-Demand Anodyne RBP4 22 42 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCO[C@H]1c1cn[nH]c1 ZINC000880627577 GG On-Demand Anodyne ROCK2 36 45 COc1cc(Br)ccc1NC(=O)N1CCN(c2nncn2C)CC1 ZINC000880627584 GD On-Demand Anodyne PDGFRB 41 44 COc1cc(Br)ccc1NC(=O)N1CCN(c2nncn2C)CC1 ZINC000880627584 GD On-Demand Anodyne RBP4 19 41 COc1cc(Br)ccc1NC(=O)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880627601 FG On-Demand Anodyne RBP4 40 33 COc1cc(Br)ccc1NC(=O)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880627602 FG On-Demand Anodyne RBP4 40 33 COc1cc(Br)ccc1NC(=O)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880627603 FG On-Demand Anodyne RBP4 40 33 COc1cc(Br)ccc1NC(=O)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880627604 FG On-Demand Anodyne RBP4 40 33 COc1cc(Br)ccc1NC(=O)N1CCOCCN1 ZINC000880627613 ED On-Demand Anodyne LRRK2 20 40 COC[C@@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880627616 EG On-Demand Anodyne DRD2 31 42 COC[C@@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880627616 EG On-Demand Anodyne ACKR3 65 33 C#CC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880627627 EG On-Demand Mild RBP4 28 42 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627643 GI On-Demand Anodyne CPT1A 130 49 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627643 GI On-Demand Anodyne CPT2 31 40 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627644 GI On-Demand Anodyne CPT1A 130 49 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627644 GI On-Demand Anodyne CPT2 31 40 O=C(NCCOCC(F)F)Nc1nc(COc2ccccc2)cs1 ZINC000880627645 FG On-Demand Anodyne ADRB1 41 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2ccccn2)CC1 ZINC000880627646 GJ On-Demand Anodyne CPT1A 43 41 CNC(=O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627651 GD On-Demand Anodyne ACOX1 52 36 CNC(=O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627651 GD On-Demand Anodyne FAAH 21 42 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627657 GD On-Demand Anodyne P2RY12 46 35 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627657 GD On-Demand Anodyne FAAH 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](O)C1 ZINC000880627661 DE On-Demand Anodyne ADAM17 43 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](O)C1 ZINC000880627661 DE On-Demand Anodyne CPT1A 42 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)C1 ZINC000880627662 DE On-Demand Anodyne ADAM17 43 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](O)C1 ZINC000880627662 DE On-Demand Anodyne CPT1A 42 38 O=C(NNC(=O)C1CCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627678 EF On-Demand Reactive CPT1A 69 40 Cc1nn(C)cc1[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627689 GI On-Demand Anodyne CPT1A 98 42 Cc1nn(C)cc1[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627690 GI On-Demand Anodyne CPT1A 98 42 CCC1(CO)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627695 GH On-Demand Anodyne NPY5R 18 41 CC1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627702 DG On-Demand Anodyne ADAM17 52 35 CC1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627702 DG On-Demand Anodyne CPT1A 46 38 CCO[C@H]1COCC[C@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627712 GG On-Demand Anodyne ADAM17 18 40 CCO[C@H]1COCC[C@@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627713 GG On-Demand Anodyne ADAM17 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccon2)CC1 ZINC000880627718 GH On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccon2)CC1 ZINC000880627718 GH On-Demand Anodyne SMO 19 49 COc1cc(Br)ccc1NC(=O)N[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880627720 GD On-Demand Anodyne EPHX2 32 45 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880627721 GD On-Demand Anodyne EPHX2 32 45 COC[C@@H](CO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627728 ED On-Demand Anodyne ROCK1 16 46 O=C(NO[C@H]1CCCCO1)Nc1nc(COc2ccccc2)cs1 ZINC000880627732 EG On-Demand Anodyne CPT1A 55 42 COc1cc(Br)ccc1NC(=O)N1CCC(SC)CC1 ZINC000880627735 FH On-Demand Anodyne RBP4 23 40 O=C(NO[C@@H]1CCCCO1)Nc1nc(COc2ccccc2)cs1 ZINC000880627739 EG On-Demand Anodyne CPT1A 55 42 COc1cc(Br)ccc1NC(=O)N1CCN(C)C(=O)C1 ZINC000880627749 ED On-Demand Anodyne PDGFRB 21 42 COC[C@@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627762 FE On-Demand Anodyne ADRB1 43 34 COC[C@@H](O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627762 FE On-Demand Anodyne ROCK1 16 42 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne OPRM1 17 41 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne TRY1_BOVIN 41 33 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne ADAM17 41 37 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne CPT1A 81 40 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne PREP 48 36 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627766 GF On-Demand Anodyne XIAP 43 34 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne OPRM1 17 41 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne TRY1_BOVIN 41 33 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne ADAM17 41 37 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne CPT1A 81 40 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne PREP 48 36 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627768 GF On-Demand Anodyne XIAP 43 34 O=C(CCCNC(=O)Nc1nc(COc2ccccc2)cs1)NC1CC1 ZINC000880627769 FF On-Demand Anodyne TNKS 53 33 COc1cc(Br)ccc1NC(=O)NCCN1CCCC1=O ZINC000880627772 FE On-Demand Anodyne TYRO3 17 40 C#CCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627773 DG On-Demand Mild ROCK1 15 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne F2 48 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne ELANE 45 39 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne HCRTR1 15 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne TRY1_BOVIN 70 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne ADAM17 48 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne CPT1A 102 42 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne CPT2 40 33 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne PREP 50 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne LGMN 66 37 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne XIAP 51 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627777 FE On-Demand Anodyne BRCA1 59 32 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2nc(C)no2)C1 ZINC000880627780 GG On-Demand Anodyne SMO 36 51 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2nc(C)no2)C1 ZINC000880627780 GG On-Demand Anodyne ETHR 49 35 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2nc(C)no2)C1 ZINC000880627781 GG On-Demand Anodyne SMO 36 51 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2nc(C)no2)C1 ZINC000880627781 GG On-Demand Anodyne ETHR 49 35 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCC[C@H](CO)C1 ZINC000880627788 FG On-Demand Anodyne PTGES 15 44 COc1cc(Br)ccc1NC(=O)N[C@H]1CCC[C@H](CO)C1 ZINC000880627789 FG On-Demand Anodyne PTGES 15 44 COc1cc(Br)ccc1NC(=O)N[C@H]1CCC[C@@H](CO)C1 ZINC000880627790 FG On-Demand Anodyne PTGES 15 44 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880627791 FG On-Demand Anodyne PTGES 15 44 COc1cc(Br)ccc1NC(=O)N1CCN(c2nccnn2)CC1 ZINC000880627792 GD On-Demand Anodyne PDGFRB 49 46 COc1cc(Br)ccc1NC(=O)N1CCN(c2nccnn2)CC1 ZINC000880627792 GD On-Demand Anodyne RBP4 20 43 COc1cc(Br)ccc1NC(=O)NC1CCC(OC)CC1 ZINC000880627804 FH On-Demand Anodyne EPHX2 42 45 COc1cc(Br)ccc1NC(=O)NCc1nc(N(C)C)n[nH]1 ZINC000880627810 FD On-Demand Anodyne ROCK2 15 41 O=C(NCCCNC(=O)C1CCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627844 GG On-Demand Anodyne IKBKE 45 38 O=C(NCCCNC(=O)C1CCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880627844 GG On-Demand Anodyne TBK1 88 38 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)[C@H]1CCCOC1 ZINC000880627851 FH On-Demand Anodyne ALOX5 29 44 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)[C@@H]1CCCOC1 ZINC000880627853 FH On-Demand Anodyne ALOX5 29 44 O=C(NCCCCCCO)Nc1nc(COc2ccccc2)cs1 ZINC000880627869 EG On-Demand Anodyne ROCK1 16 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(O)(C(F)F)CC1 ZINC000880627871 GG On-Demand Anodyne NPY5R 17 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(CCCO)CC1 ZINC000880627890 GH On-Demand Anodyne NPY1R 40 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2cccnc2)CC1 ZINC000880627892 GJ On-Demand Anodyne CPT1A 37 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2cccnc2)CC1 ZINC000880627892 GJ On-Demand Anodyne EPHX2 22 44 CC[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880627902 FH On-Demand Anodyne ADAM17 54 36 CC[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880627902 FH On-Demand Anodyne CPT1A 84 38 CC1(CO)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627909 FG On-Demand Anodyne ADAM17 56 36 CC1(CO)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880627909 FG On-Demand Anodyne NPY5R 24 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CC(CC(F)(F)F)C1 ZINC000880627911 FI On-Demand Anodyne RBP4 50 32 C[C@@H](O)CCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627924 EG On-Demand Anodyne ROCK1 18 40 CO[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880627938 EG On-Demand Anodyne CPT1A 56 38 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(=O)N(C)C ZINC000880627942 EE On-Demand Anodyne ROCK1 15 40 C[C@@H]1COCC[C@@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627953 EG On-Demand Anodyne ADAM17 25 42 C[C@@H]1COCC[C@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627955 EG On-Demand Anodyne ADAM17 25 42 C[C@H]1C(=O)N(C)CCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627963 FE On-Demand Anodyne ADAM17 42 36 COCC[C@H](CO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627965 FE On-Demand Anodyne ROCK1 16 43 COCC[C@@H](CO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880627967 FE On-Demand Anodyne ROCK1 16 43 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCO[C@H]1c1cccnc1 ZINC000880627980 GH On-Demand Anodyne CHRNA7 25 47 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1ccnc1 ZINC000880627990 GG On-Demand Anodyne QPCT 19 40 COc1cc(Br)ccc1NC(=O)NCc1c(C2CC2)cnn1C ZINC000880627994 GG On-Demand Anodyne HTR2A 23 40 COc1cc(Br)ccc1NC(=O)NCc1c(C2CC2)cnn1C ZINC000880627994 GG On-Demand Anodyne ROCK2 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1[C@H]2CCC[C@H]1CC2 ZINC000880627995 EI On-Demand Anodyne CPT1A 52 38 COc1cc(Br)ccc1NC(=O)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880627999 GD On-Demand Anodyne PDGFRB 35 41 COc1cc(Br)ccc1NC(=O)N[C@@H]1CC[C@@H](O)CC1 ZINC000880628009 EF On-Demand Anodyne EPHX2 30 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1C1CCOCC1 ZINC000880628066 GI On-Demand Anodyne CPT1A 105 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1C1CCOCC1 ZINC000880628067 GI On-Demand Anodyne CPT1A 105 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@@H]([C@@H]2CCCO2)C1 ZINC000880628069 GG On-Demand Anodyne CPT1A 69 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@@H]([C@H]2CCCO2)C1 ZINC000880628070 GG On-Demand Anodyne CPT1A 69 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@H]([C@@H]2CCCO2)C1 ZINC000880628071 GG On-Demand Anodyne CPT1A 69 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCO[C@H]([C@H]2CCCO2)C1 ZINC000880628072 GG On-Demand Anodyne CPT1A 69 38 O=C(NC[C@H](O)CN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628074 GD On-Demand Anodyne ACOX1 52 36 O=C(NC[C@@H](O)CN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628075 GD On-Demand Anodyne ACOX1 52 36 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)(F)C1 ZINC000880628082 EH On-Demand Anodyne GRM5 15 46 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(F)(F)C1 ZINC000880628082 EH On-Demand Anodyne NPY5R 15 41 O=C(CNC(=O)Nc1nc(COc2ccccc2)cs1)NCC1CC1 ZINC000880628083 FE On-Demand Anodyne GRIN2B 20 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1cn[nH]c1 ZINC000880628084 GI On-Demand Anodyne CPT1A 128 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1cn[nH]c1 ZINC000880628085 GI On-Demand Anodyne CPT1A 128 45 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628090 GH On-Demand Anodyne CPT1A 44 37 CN(C)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628093 FH On-Demand Anodyne CACNA1B 23 40 CN(C)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628093 FH On-Demand Anodyne CPT1A 46 38 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CC[C@@H]1O ZINC000880628111 EF On-Demand Anodyne ADAM17 46 36 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CC[C@H]1O ZINC000880628112 EF On-Demand Anodyne ADAM17 46 36 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CC[C@H]1O ZINC000880628113 EF On-Demand Anodyne ADAM17 46 36 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CC[C@@H]1O ZINC000880628114 EF On-Demand Anodyne ADAM17 46 36 COC(=O)C1(CNC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628130 FF On-Demand Anodyne ROCK1 17 41 C[C@H]1CC[C@@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628138 EI On-Demand Anodyne ADAM17 40 34 C[C@H]1CC[C@@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628138 EI On-Demand Anodyne CPT1A 43 38 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628142 EI On-Demand Anodyne ADAM17 40 34 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628142 EI On-Demand Anodyne CPT1A 43 38 C[C@H]1CC[C@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628147 EI On-Demand Anodyne ADAM17 40 34 C[C@H]1CC[C@H](C)N1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628147 EI On-Demand Anodyne CPT1A 43 38 COc1cc(Br)ccc1NC(=O)N1CCN(CCO)C[C@H]1C ZINC000880628160 FD On-Demand Anodyne CCR1 19 40 COc1cc(Br)ccc1NC(=O)N1CCN(CCO)C[C@@H]1C ZINC000880628161 FD On-Demand Anodyne CCR1 19 40 Cc1n[nH]c(C)c1[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628162 GI On-Demand Anodyne CPT1A 117 43 COc1cc(Br)ccc1NC(=O)NCC1(N(C)C)CC1 ZINC000880628183 EF On-Demand Anodyne SLC6A5 15 42 CNC(=O)[C@@H]1CCC[C@@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628205 FF On-Demand Anodyne ADAM17 37 46 CNC(=O)[C@@H]1CCC[C@H]1NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628210 FF On-Demand Anodyne ADAM17 37 46 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H](O)C[C@H]1CO ZINC000880628217 ED On-Demand Anodyne SPHK2 61 34 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@H](O)C[C@H]1CO ZINC000880628217 ED On-Demand Anodyne SPHK1 47 36 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H](O)C[C@H]1CO ZINC000880628220 ED On-Demand Anodyne SPHK2 61 34 O=C(Nc1nc(COc2ccccc2)cs1)N1C[C@@H](O)C[C@H]1CO ZINC000880628220 ED On-Demand Anodyne SPHK1 47 36 CC[C@@H](C)C(=O)NNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628224 EF On-Demand Reactive MME 15 44 CC[C@@H](C)C(=O)NNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628224 EF On-Demand Reactive ROCK1 15 41 CC[C@@H](C)C(=O)NNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628224 EF On-Demand Reactive CAPN2 40 33 CC[C@@H](C)C(=O)NNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628224 EF On-Demand Reactive ACE2 52 38 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880628243 FE On-Demand Anodyne EPHX2 37 46 COc1cc(Br)ccc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880628246 FG On-Demand Anodyne SLC6A4 16 41 COc1cc(Br)ccc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880628246 FG On-Demand Anodyne HTR3A 26 46 COc1cc(Br)ccc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880628246 FG On-Demand Anodyne SLC6A3 36 41 COc1cc(Br)ccc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880628246 FG On-Demand Anodyne HTR4 17 47 COc1cc(Br)ccc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880628246 FG On-Demand Anodyne GLRA1 44 32 COc1cc(Br)ccc1NC(=O)N[C@H]1CCc2nnnn2CC1 ZINC000880628248 GD On-Demand Anodyne EPHX2 19 40 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCc2nnnn2CC1 ZINC000880628249 GD On-Demand Anodyne EPHX2 19 40 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)no1 ZINC000880628265 GI On-Demand Anodyne ACOX1 41 34 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)no1 ZINC000880628265 GI On-Demand Anodyne ADAM17 57 36 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)no1 ZINC000880628265 GI On-Demand Anodyne CPT1A 134 49 CN(C[C@@H]1CCCO1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628273 EG On-Demand Anodyne CPT1A 64 38 CN(C[C@@H]1CCCO1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628273 EG On-Demand Anodyne TNK2 48 35 O=C(CO)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628282 GD On-Demand Anodyne FAAH 19 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC12CCC2 ZINC000880628285 EI On-Demand Anodyne SLC12A5 42 32 CC1(C)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628315 EH On-Demand Anodyne ADAM17 44 37 CC1(C)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628315 EH On-Demand Anodyne NPY5R 24 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCSCC1 ZINC000880628316 EG On-Demand Anodyne FAAH 15 41 COc1cc(Br)ccc1NC(=O)N1CCC(C(C)=O)CC1 ZINC000880628322 FG On-Demand Anodyne RBP4 24 42 CN(C)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628324 EF On-Demand Anodyne ADAM17 42 43 CN(C)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628324 EF On-Demand Anodyne CPT1A 40 38 COc1cc(Br)ccc1NC(=O)N1CCC(O)CC1 ZINC000880628329 EE On-Demand Anodyne PDGFRB 17 42 COc1cc(Br)ccc1NC(=O)N1CCC(O)CC1 ZINC000880628329 EE On-Demand Anodyne RBP4 29 42 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(C2CC2)CC1 ZINC000880628340 FG On-Demand Anodyne SLC6A5 36 46 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(C2CC2)CC1 ZINC000880628340 FG On-Demand Anodyne EPHX2 29 42 CC(=O)NCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628356 EE On-Demand Anodyne ROCK1 17 42 CC(=O)NCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628356 EE On-Demand Anodyne MTNR1A 33 40 CC(=O)NCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628356 EE On-Demand Anodyne MTNR1B 34 40 C[S@@](=O)CCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628357 FF On-Demand Anodyne ROCK1 15 41 O=C(NCC1(O)CCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628363 EF On-Demand Anodyne ROCK1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC([C@H](C)O)CC1 ZINC000880628364 FG On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)N1CCC([C@@H](C)O)CC1 ZINC000880628365 FG On-Demand Anodyne RBP4 23 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(c2cc[nH]n2)CC1 ZINC000880628366 GH On-Demand Anodyne CPT1A 43 38 Cn1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)cn1 ZINC000880628368 GH On-Demand Anodyne ADAM17 27 40 Cn1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)cn1 ZINC000880628368 GH On-Demand Anodyne CPT1A 107 43 COc1cc(Br)ccc1NC(=O)N1CCC(C2(O)CC2)CC1 ZINC000880628379 FG On-Demand Anodyne PDGFRB 15 41 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CO)C1 ZINC000880628432 EE On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CO)C1 ZINC000880628432 EE On-Demand Anodyne PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CO)C1 ZINC000880628433 EE On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CO)C1 ZINC000880628433 EE On-Demand Anodyne PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CCC(O)(CO)CC1 ZINC000880628470 FD On-Demand Anodyne PDGFRB 25 41 COc1cc(Br)ccc1NC(=O)N1CCC(O)(CO)CC1 ZINC000880628470 FD On-Demand Anodyne RBP4 21 40 Cn1cccc1[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628527 GI On-Demand Anodyne CPT1A 117 45 Cn1cccc1[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628528 GI On-Demand Anodyne CPT1A 117 45 CC[C@H](O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628529 GF On-Demand Anodyne ACOX1 56 39 CC[C@H](O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628529 GF On-Demand Anodyne ABCB1 59 42 CC[C@@H](O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628530 GF On-Demand Anodyne ACOX1 56 39 CC[C@@H](O)CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628530 GF On-Demand Anodyne ABCB1 59 42 O=C(Nc1nc(COc2ccccc2)cs1)N(Cc1ccncc1)C1CC1 ZINC000880628533 GI On-Demand Anodyne CPT1A 27 42 O=C(Nc1nc(COc2ccccc2)cs1)N(Cc1ccncc1)C1CC1 ZINC000880628533 GI On-Demand Anodyne ROCK1 18 46 COc1cc(Br)ccc1NC(=O)N[C@@H](CO)CC(C)C ZINC000880628542 EF On-Demand Anodyne ANPEP 26 52 COc1cc(Br)ccc1NC(=O)N[C@H](CO)CC(C)C ZINC000880628544 EF On-Demand Anodyne ANPEP 26 52 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@@H](O)C1 ZINC000880628569 FD On-Demand Anodyne DRD2 21 41 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@@H](O)C1 ZINC000880628569 FD On-Demand Anodyne DRD4 41 32 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@@H](O)C1 ZINC000880628569 FD On-Demand Anodyne DRD3 25 44 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@H](O)C1 ZINC000880628571 FD On-Demand Anodyne DRD2 21 41 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@H](O)C1 ZINC000880628571 FD On-Demand Anodyne DRD4 41 32 COc1cc(Br)ccc1NC(=O)NCCN1CC[C@H](O)C1 ZINC000880628571 FD On-Demand Anodyne DRD3 25 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](CO)C1 ZINC000880628578 EF On-Demand Anodyne CPT1A 45 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](CO)C1 ZINC000880628582 EF On-Demand Anodyne CPT1A 45 38 COc1cc(Br)ccc1NC(=O)N1CCC(C)(N2CCCC2)CC1 ZINC000880628589 GH On-Demand Anodyne CCR5 25 41 COCC[C@](C)(O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628592 FF On-Demand Anodyne ROCK1 15 42 COCC[C@@](C)(O)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628595 FF On-Demand Anodyne ROCK1 15 42 O=C(Nc1nc(COc2ccccc2)cs1)N1C2CCC1CC2 ZINC000880628611 EH On-Demand Anodyne CPT1A 45 38 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CCO ZINC000880628612 EF On-Demand Anodyne DRD2 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CCO ZINC000880628612 EF On-Demand Anodyne ACKR3 65 33 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CCO ZINC000880628613 EF On-Demand Anodyne DRD2 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CCO ZINC000880628613 EF On-Demand Anodyne ACKR3 65 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1CCCO ZINC000880628616 FG On-Demand Anodyne CPT1A 74 40 COc1cc(Br)ccc1NC(=O)N[C@H]1CCOC1=O ZINC000880628618 ED On-Demand Anodyne LUXR 80 47 COc1cc(Br)ccc1NC(=O)N[C@H]1CCOC1=O ZINC000880628618 ED On-Demand Anodyne TRAR 95 51 COc1cc(Br)ccc1NC(=O)N[C@H]1CCOC1=O ZINC000880628618 ED On-Demand Anodyne LASR 63 47 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1CCCO ZINC000880628620 FG On-Demand Anodyne CPT1A 74 40 COc1cc(Br)ccc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880628622 GI On-Demand Anodyne EPHX2 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880628622 GI On-Demand Anodyne RBP4 24 40 COc1cc(Br)ccc1NC(=O)N1CCCC[C@@H]1CNC(C)=O ZINC000880628658 GF On-Demand Anodyne DRD2 32 43 COc1cc(Br)ccc1NC(=O)N1CCCC[C@@H]1CNC(C)=O ZINC000880628658 GF On-Demand Anodyne ACKR3 65 33 COc1cc(Br)ccc1NC(=O)N1CCCC[C@H]1CNC(C)=O ZINC000880628659 GF On-Demand Anodyne DRD2 32 43 COc1cc(Br)ccc1NC(=O)N1CCCC[C@H]1CNC(C)=O ZINC000880628659 GF On-Demand Anodyne ACKR3 65 33 O=C(NCCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628662 GF On-Demand Anodyne CASR 44 41 O=C(NCCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628662 GF On-Demand Anodyne TACR2 18 51 O=C(NCCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628662 GF On-Demand Anodyne CCR3 20 40 O=C(NCCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628662 GF On-Demand Anodyne EPHX2 30 48 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1CO ZINC000880628663 EF On-Demand Anodyne ADAM17 23 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1CO ZINC000880628663 EF On-Demand Anodyne CPT1A 103 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1CO ZINC000880628663 EF On-Demand Anodyne CPT1B 18 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1CO ZINC000880628664 EF On-Demand Anodyne ADAM17 23 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1CO ZINC000880628664 EF On-Demand Anodyne CPT1A 103 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1CO ZINC000880628664 EF On-Demand Anodyne CPT1B 18 42 COc1cc(Br)ccc1NC(=O)N1CCC(F)CC1 ZINC000880628677 EG On-Demand Anodyne PDGFRB 15 42 COc1cc(Br)ccc1NC(=O)N1CCC(F)CC1 ZINC000880628677 EG On-Demand Anodyne RBP4 42 44 O=C(NCCOCC1CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628679 EG On-Demand Anodyne ADRB1 19 44 O=C(NCCOCC1CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628679 EG On-Demand Anodyne GRIN2B 17 41 COCC[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628683 EG On-Demand Anodyne ROCK1 15 45 COCC[C@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628684 EG On-Demand Anodyne ROCK1 15 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOCC1 ZINC000880628691 DF On-Demand Anodyne CYSLTR1 40 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOCC1 ZINC000880628691 DF On-Demand Anodyne ADAM17 16 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCOCC1 ZINC000880628691 DF On-Demand Anodyne FAAH 17 40 CCOC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628701 GH On-Demand Anodyne PDE6D 53 35 CCOC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628701 GH On-Demand Anodyne ADAM17 43 35 CCOC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628701 GH On-Demand Anodyne CPT1A 56 40 CCOC(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628701 GH On-Demand Anodyne PTR1 46 33 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ccccn2)CC1 ZINC000880628702 GG On-Demand Anodyne PDGFRB 27 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ccccn2)CC1 ZINC000880628702 GG On-Demand Anodyne CPT1A 18 44 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ccccn2)CC1 ZINC000880628702 GG On-Demand Anodyne FAAH 24 43 CCn1ncc(NC(=O)Nc2ccc(Br)cc2OC)c1C ZINC000880628705 FH On-Demand Anodyne HTR2A 17 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](C(C)(C)O)C1 ZINC000880628751 FG On-Demand Anodyne RBP4 33 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](C(C)(C)O)C1 ZINC000880628752 FG On-Demand Anodyne RBP4 33 40 CCOC(=O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628756 EF On-Demand Anodyne ROCK1 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1Cn1cncn1 ZINC000880628765 GG On-Demand Anodyne CPT1A 77 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1Cn1cncn1 ZINC000880628766 GG On-Demand Anodyne CPT1A 77 39 CC(=O)NC[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCO1 ZINC000880628774 GE On-Demand Anodyne ADAM17 46 36 O=C(NCCOC1CCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628777 EG On-Demand Anodyne ADRB1 22 47 Cc1noc(C2CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)n1 ZINC000880628778 GH On-Demand Anodyne CPT1A 70 39 Cc1noc(C2CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)n1 ZINC000880628778 GH On-Demand Anodyne SMO 46 46 Cc1noc(C2CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)n1 ZINC000880628778 GH On-Demand Anodyne ETHR 63 39 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CF)C1 ZINC000880628781 EH On-Demand Anodyne PDGFRB 20 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CF)C1 ZINC000880628782 EH On-Demand Anodyne PDGFRB 20 40 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628788 GG On-Demand Anodyne ADAM17 43 34 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628788 GG On-Demand Anodyne CPT1A 35 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN2CCC[C@H]2C1 ZINC000880628790 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN2CCC[C@H]2C1 ZINC000880628790 FG On-Demand Anodyne CPT1A 47 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN2CCC[C@@H]2C1 ZINC000880628791 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN2CCC[C@@H]2C1 ZINC000880628791 FG On-Demand Anodyne CPT1A 47 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC1 ZINC000880628794 DG On-Demand Anodyne CPT1A 78 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC1 ZINC000880628794 DG On-Demand Anodyne FAAH 18 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1c1ccncc1 ZINC000880628799 GI On-Demand Anodyne ADAM17 26 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1c1ccncc1 ZINC000880628799 GI On-Demand Anodyne CPT1A 114 50 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1c1ccncc1 ZINC000880628800 GI On-Demand Anodyne ADAM17 26 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1c1ccncc1 ZINC000880628800 GI On-Demand Anodyne CPT1A 114 50 O=C(NCCNC(=O)C1CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880628803 FE On-Demand Anodyne ROCK1 15 41 CNC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628810 FF On-Demand Anodyne ADAM17 43 35 CNC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628810 FF On-Demand Anodyne CPT1A 63 39 COC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628813 GG On-Demand Anodyne CPT1A 72 40 COC(=O)[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628813 GG On-Demand Anodyne PTR1 42 30 CNC(=O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628817 ED On-Demand Anodyne ROCK1 17 42 CC(C)(C)NC(=O)CCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628822 GG On-Demand Anodyne ROCK1 17 41 O=C(NCCCN1CCCC1=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628827 FF On-Demand Anodyne TYRO3 20 41 C[C@@H]1CC(=O)NCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628835 FE On-Demand Anodyne CPT1A 43 37 C[C@H]1CC(=O)NCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628836 FE On-Demand Anodyne CPT1A 43 37 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne TBXAS1 43 44 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne ROCK1 15 41 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne HMOX1 15 40 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne HMOX2 41 40 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne QPCT 34 51 O=C(NCCCCn1ccnc1)Nc1nc(COc2ccccc2)cs1 ZINC000880628837 FH On-Demand Anodyne NAMPT 22 44 COCCCN(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628889 EG On-Demand Anodyne LTA4H 19 41 CCC(=O)N1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628900 GG On-Demand Anodyne CPT1A 41 38 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne DRD4 22 40 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne LTA4H 25 45 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne SIGMAR1 15 42 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne CCR3 21 43 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne CPT1A 46 37 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne SLC6A5 35 41 COCCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628903 GF On-Demand Anodyne MCHR1 22 40 CCC1(O)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628905 FG On-Demand Anodyne NPY5R 21 42 CCC1(O)CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628905 FG On-Demand Anodyne S1PR2 26 41 C[C@H](NC(=O)Nc1nc(COc2ccccc2)cs1)C(=O)NC(C)(C)C ZINC000880628910 GG On-Demand Anodyne ROCK1 15 41 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CF)C1 ZINC000880628912 EG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CF)C1 ZINC000880628912 EG On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CF)C1 ZINC000880628913 EG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CF)C1 ZINC000880628913 EG On-Demand Anodyne PTPN1 15 40 CONC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880628917 GE On-Demand Anodyne RBP4 23 40 COCCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628918 EG On-Demand Anodyne ROCK1 17 45 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(CC(F)F)CC1 ZINC000880628919 GH On-Demand Anodyne DRD4 15 41 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(CC(F)F)CC1 ZINC000880628919 GH On-Demand Anodyne SLC6A5 31 41 O=C(Nc1nc(COc2ccccc2)cs1)NC1CCN(CC(F)F)CC1 ZINC000880628919 GH On-Demand Anodyne EPHX2 35 41 CC(=O)NCC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628920 GG On-Demand Anodyne GRIN2B 54 39 CC(=O)NCC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628920 GG On-Demand Anodyne CPT1A 38 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880628921 GH On-Demand Anodyne NPY1R 41 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880628921 GH On-Demand Anodyne CCR3 25 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880628921 GH On-Demand Anodyne CPT1A 74 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](CN2CCCC2)C1 ZINC000880628922 GH On-Demand Anodyne NPY1R 41 34 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](CN2CCCC2)C1 ZINC000880628922 GH On-Demand Anodyne CCR3 25 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](CN2CCCC2)C1 ZINC000880628922 GH On-Demand Anodyne CPT1A 74 39 N#CCCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628929 EH On-Demand Mild ADRB1 43 33 COCC1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628930 FH On-Demand Anodyne CPT1A 65 39 CN1CCC(CNC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628938 FG On-Demand Anodyne CPT1A 45 38 CN1CCC(CNC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880628938 FG On-Demand Anodyne SLC6A5 17 40 COc1cc(Br)ccc1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880628942 GE On-Demand Anodyne DRD4 19 40 COc1cc(Br)ccc1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880628942 GE On-Demand Anodyne HTR4 42 36 COc1cc(Br)ccc1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880628942 GE On-Demand Anodyne CCR3 21 44 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@@H]1C ZINC000880628943 EH On-Demand Anodyne ADAM17 44 35 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@H]1C ZINC000880628944 EH On-Demand Anodyne ADAM17 44 35 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)C[C@@H]1C ZINC000880628945 EH On-Demand Anodyne ADAM17 44 35 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(Br)cc1OC ZINC000880628947 GG On-Demand Anodyne SLC6A4 21 42 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(Br)cc1OC ZINC000880628947 GG On-Demand Anodyne SLC6A3 39 42 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(Br)cc1OC ZINC000880628948 GG On-Demand Anodyne SLC6A4 21 42 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(Br)cc1OC ZINC000880628948 GG On-Demand Anodyne SLC6A3 39 42 CCS(=O)(=O)C[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628951 GF On-Demand Anodyne ROCK1 15 40 CCS(=O)(=O)C[C@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880628952 GF On-Demand Anodyne ROCK1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(C)(N2CCC2)CC1 ZINC000880628959 GH On-Demand Anodyne CCR5 24 40 CC(=O)N[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628969 FF On-Demand Anodyne ADAM17 51 36 CC(=O)N[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628969 FF On-Demand Anodyne CPT1A 50 42 CC(=O)N[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628969 FF On-Demand Anodyne SLC6A5 20 41 CC(=O)N[C@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628969 FF On-Demand Anodyne BIRC2 37 40 CC(=O)N[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628970 FF On-Demand Anodyne ADAM17 51 36 CC(=O)N[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628970 FF On-Demand Anodyne CPT1A 50 42 CC(=O)N[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628970 FF On-Demand Anodyne SLC6A5 20 41 CC(=O)N[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880628970 FF On-Demand Anodyne BIRC2 37 40 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880628972 EG On-Demand Anodyne ADAM17 49 36 C[C@@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880628972 EG On-Demand Anodyne CPT1A 59 38 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880628973 EG On-Demand Anodyne ADAM17 49 36 C[C@H]1CN(C(=O)Nc2nc(COc3ccccc3)cs2)CCCO1 ZINC000880628973 EG On-Demand Anodyne CPT1A 59 38 CC(C)n1ccc(CNC(=O)Nc2nc(COc3ccccc3)cs2)n1 ZINC000880628979 FH On-Demand Anodyne ROCK1 18 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCCCC1 ZINC000880629036 EI On-Demand Anodyne CPT1A 68 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCCCC1 ZINC000880629036 EI On-Demand Anodyne FAAH 18 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1ncc[nH]1 ZINC000880629039 GI On-Demand Anodyne CPT1A 132 47 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@H]1c1ncc[nH]1 ZINC000880629039 GI On-Demand Anodyne CPT2 34 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1ncc[nH]1 ZINC000880629040 GI On-Demand Anodyne CPT1A 132 47 O=C(Nc1nc(COc2ccccc2)cs1)N1CCCC[C@@H]1c1ncc[nH]1 ZINC000880629040 GI On-Demand Anodyne CPT2 34 42 CC(=O)N(C)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629041 GG On-Demand Anodyne CPT1A 33 40 O=C(NCC(=O)N1CCCCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629050 FF On-Demand Anodyne CPT1A 57 39 O=C(NCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629051 FE On-Demand Anodyne CASR 45 42 O=C(NCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629051 FE On-Demand Anodyne EPHX2 24 45 O=C(NCCN1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629051 FE On-Demand Anodyne HPGDS 23 41 C[C@@H](CCN(C)C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629053 EG On-Demand Anodyne UTS2 54 37 CN(CCN1CCOCC1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629061 GF On-Demand Anodyne CASR 61 50 CN(CCN1CCOCC1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629061 GF On-Demand Anodyne EPHX2 15 41 CCc1nc([C@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)no1 ZINC000880629063 GI On-Demand Anodyne CPT1A 116 45 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(C2CC2)CC1 ZINC000880629064 FG On-Demand Anodyne CPT1A 48 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(C2CC2)CC1 ZINC000880629064 FG On-Demand Anodyne FAAH 15 41 COC[C@@H]1CCCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629084 FH On-Demand Anodyne CPT1A 74 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1Cn1cccn1 ZINC000880629085 GH On-Demand Anodyne CPT1A 88 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1Cn1cccn1 ZINC000880629086 GH On-Demand Anodyne CPT1A 88 42 COCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629087 DF On-Demand Anodyne ROCK1 17 45 O=C(NCC1(CO)CC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629091 EF On-Demand Anodyne ROCK1 15 41 O=C(Nc1nc(COc2ccccc2)cs1)N(Cc1cccnc1)C1CC1 ZINC000880629094 GI On-Demand Anodyne CPT1A 26 41 O=C(Nc1nc(COc2ccccc2)cs1)N(Cc1cccnc1)C1CC1 ZINC000880629094 GI On-Demand Anodyne CYP3A4 19 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](c2cc[nH]n2)C1 ZINC000880629107 GH On-Demand Anodyne CPT1A 61 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H](c2cc[nH]n2)C1 ZINC000880629107 GH On-Demand Anodyne MAP3K12 31 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](c2cc[nH]n2)C1 ZINC000880629108 GH On-Demand Anodyne CPT1A 61 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H](c2cc[nH]n2)C1 ZINC000880629108 GH On-Demand Anodyne MAP3K12 31 41 COc1cc(Br)ccc1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880629109 EF On-Demand Anodyne EPHX2 30 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](N2CCCC2)C1 ZINC000880629116 FG On-Demand Anodyne CPT1A 82 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@H](N2CCCC2)C1 ZINC000880629116 FG On-Demand Anodyne L3MBTL3 75 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](N2CCCC2)C1 ZINC000880629117 FG On-Demand Anodyne CPT1A 82 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CC[C@@H](N2CCCC2)C1 ZINC000880629117 FG On-Demand Anodyne L3MBTL3 75 39 CN1C[C@H](NC(=O)Nc2nc(COc3ccccc3)cs2)CCC1=O ZINC000880629121 FE On-Demand Anodyne SLC6A5 26 40 CN1C[C@@H](NC(=O)Nc2nc(COc3ccccc3)cs2)CCC1=O ZINC000880629122 FE On-Demand Anodyne SLC6A5 26 40 CN1CCC[C@H](CNC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629136 FG On-Demand Anodyne ADAM17 41 33 CN1CCC[C@H](CNC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629136 FG On-Demand Anodyne CPT1A 40 38 COc1cc(Br)ccc1NC(=O)N1CCC(c2nnnn2C)CC1 ZINC000880629137 GE On-Demand Anodyne RBP4 22 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ncccn2)CC1 ZINC000880629138 GF On-Demand Anodyne PDGFRB 33 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ncccn2)CC1 ZINC000880629138 GF On-Demand Anodyne CPT1A 19 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ncccn2)CC1 ZINC000880629138 GF On-Demand Anodyne FAAH 24 45 COCCN(Cc1cccnc1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629139 GH On-Demand Anodyne ROCK1 16 40 COCCN(Cc1cccnc1)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629139 GH On-Demand Anodyne ROCK2 17 41 CN1CCC[C@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629142 EF On-Demand Anodyne CPT1A 51 38 CN1CCC[C@H](NC(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629142 EF On-Demand Anodyne SLC6A5 34 45 C[C@H](CCO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629160 DF On-Demand Anodyne ROCK1 18 41 C[C@@H](CCO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629161 DF On-Demand Anodyne ROCK1 18 41 COc1cc(Br)ccc1NC(=O)N1CCO[C@@H](C(F)F)CC1 ZINC000880629162 GG On-Demand Anodyne RBP4 27 40 COc1cc(Br)ccc1NC(=O)N1CCO[C@H](C(F)F)CC1 ZINC000880629163 GG On-Demand Anodyne RBP4 27 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2ccncc2)CC1 ZINC000880629168 GG On-Demand Anodyne FAAH 22 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1C1CC1 ZINC000880629171 EI On-Demand Anodyne CPT1A 112 43 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1C1CC1 ZINC000880629172 EI On-Demand Anodyne CPT1A 112 43 COC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629174 FF On-Demand Anodyne CPT1A 62 39 COC(=O)[C@@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629174 FF On-Demand Anodyne PTR1 45 33 COC(=O)[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629175 FF On-Demand Anodyne CPT1A 62 39 COC(=O)[C@H]1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)C1 ZINC000880629175 FF On-Demand Anodyne PTR1 45 33 COc1cc(Br)ccc1NC(=O)N1CCN(CCC#N)CC1 ZINC000880629180 FF On-Demand Mild DRD3 19 40 COc1cc(Br)ccc1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880629185 FG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880629185 FG On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880629185 FG On-Demand Anodyne RBP4 28 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(CO)CC1 ZINC000880629188 EF On-Demand Anodyne GRIN2B 43 39 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(CO)CC1 ZINC000880629188 EF On-Demand Anodyne CPT1A 40 37 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC(CO)CC1 ZINC000880629188 EF On-Demand Anodyne EPHX2 16 46 COc1cc(Br)ccc1NC(=O)N1CCN([S@@](C)(=N)=O)CC1 ZINC000880629191 GE On-Demand Anodyne PDGFRB 16 41 COc1cc(Br)ccc1NC(=O)N1CCN([S@@](C)(=N)=O)CC1 ZINC000880629191 GE On-Demand Anodyne RBP4 33 42 COc1cc(Br)ccc1NC(=O)N1CCN([S@](C)(=N)=O)CC1 ZINC000880629192 GE On-Demand Anodyne PDGFRB 16 41 COc1cc(Br)ccc1NC(=O)N1CCN([S@](C)(=N)=O)CC1 ZINC000880629192 GE On-Demand Anodyne RBP4 33 42 O=C(Nc1nc(COc2ccccc2)cs1)N(Cc1ccccn1)C1CC1 ZINC000880629194 GI On-Demand Anodyne CPT1A 27 40 CN(C(=O)Nc1nc(COc2ccccc2)cs1)C1CCC1 ZINC000880629205 DH On-Demand Anodyne CPT1A 56 40 COc1cc(Br)ccc1NC(=O)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880629206 GH On-Demand Anodyne RBP4 40 44 COc1cc(Br)ccc1NC(=O)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880629207 GH On-Demand Anodyne RBP4 40 44 COC[C@H](C)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629208 EG On-Demand Anodyne ROCK1 20 45 COC[C@@H](C)CNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629209 EG On-Demand Anodyne ROCK1 20 45 COc1cc(Br)ccc1NC(=O)Nc1cnn(C)c1C1CC1 ZINC000880629223 FH On-Demand Anodyne HTR2A 27 45 CSC[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629224 EH On-Demand Anodyne ROCK1 15 40 O=C(NCC1(O)CCCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629228 EG On-Demand Anodyne ROCK1 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(c2cnccn2)CC1 ZINC000880629231 GF On-Demand Anodyne FAAH 18 44 CCOCCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629252 EG On-Demand Anodyne ROCK1 15 40 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)on1 ZINC000880629264 GI On-Demand Anodyne ADAM17 51 36 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)on1 ZINC000880629264 GI On-Demand Anodyne CPT1A 122 46 Cc1cc([C@@H]2CCCN2C(=O)Nc2nc(COc3ccccc3)cs2)on1 ZINC000880629264 GI On-Demand Anodyne CPT1B 15 40 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1c1ccccn1 ZINC000880629268 GI On-Demand Anodyne CPT1A 124 50 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1c1ccccn1 ZINC000880629269 GI On-Demand Anodyne CPT1A 124 50 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629278 GG On-Demand Anodyne ROCK1 15 41 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629278 GG On-Demand Anodyne ACE2 40 35 CC[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629279 GG On-Demand Anodyne ROCK1 15 41 CC[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629279 GG On-Demand Anodyne ACE2 40 35 O=C(NCCCO)Nc1nc(COc2ccccc2)cs1 ZINC000880629288 DE On-Demand Anodyne ROCK1 17 43 O=C1CC2(CCN(C(=O)Nc3nc(COc4ccccc4)cs3)CC2)CN1 ZINC000880629289 GF On-Demand Anodyne NPY5R 15 43 CCOCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629293 DF On-Demand Anodyne ROCK1 17 41 CN(C)C(=O)C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629305 GG On-Demand Anodyne CPT1A 52 38 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1c1cccnc1 ZINC000880629306 GI On-Demand Anodyne ADAM17 22 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@@H]1c1cccnc1 ZINC000880629306 GI On-Demand Anodyne CPT1A 112 49 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1c1cccnc1 ZINC000880629307 GI On-Demand Anodyne ADAM17 22 42 O=C(Nc1nc(COc2ccccc2)cs1)N1CCC[C@H]1c1cccnc1 ZINC000880629307 GI On-Demand Anodyne CPT1A 112 49 CN1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629318 EF On-Demand Anodyne FAAH 23 42 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629319 GG On-Demand Anodyne NPY5R 27 40 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629320 GG On-Demand Anodyne NPY5R 27 40 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne DRD4 16 42 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne SSTR5 41 35 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne MAPKAPK2 17 40 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne SLC6A5 34 47 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne EPHX2 37 43 CCN1CCC(NC(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629322 FG On-Demand Anodyne MCHR1 18 40 CC[C@H](CCO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629335 EG On-Demand Anodyne ROCK1 16 42 CC[C@@H](CCO)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629336 EG On-Demand Anodyne ROCK1 16 42 C[C@@H](Cn1cncn1)NC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629338 FF On-Demand Anodyne HIS3 73 45 CS(=O)(=O)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629340 GD On-Demand Anodyne FAAH 16 42 CC[C@@H]1COCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629373 EG On-Demand Anodyne CPT1A 40 38 CNC(=O)CCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629381 EE On-Demand Anodyne ROCK1 15 40 CC(C)(C)C(=O)NCCNC(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629383 GG On-Demand Anodyne ROCK1 16 41 COCC(=O)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629393 GE On-Demand Anodyne CPT1A 74 40 COCC(=O)N1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629393 GE On-Demand Anodyne FAAH 16 42 O=C(NCCCOC1CCOCC1)Nc1nc(COc2ccccc2)cs1 ZINC000880629395 GG On-Demand Anodyne ADRB1 15 40 O=C(NCCOCCO)Nc1nc(COc2ccccc2)cs1 ZINC000880629407 ED On-Demand Anodyne ROCK1 15 41 Cn1nccc1C1CCN(C(=O)Nc2nc(COc3ccccc3)cs2)CC1 ZINC000880629408 GH On-Demand Anodyne IL2RA 50 31 O=C(NC[C@H]1CCCCO1)Nc1nc(COc2ccccc2)cs1 ZINC000880629417 EG On-Demand Anodyne CPT1A 73 38 O=C(NC[C@H]1CCCCO1)Nc1nc(COc2ccccc2)cs1 ZINC000880629417 EG On-Demand Anodyne TNK2 51 35 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(C(=O)C2CC2)CC1 ZINC000880629418 GF On-Demand Anodyne CPT1A 72 41 O=C(Nc1nc(COc2ccccc2)cs1)N1CCN(C(=O)C2CC2)CC1 ZINC000880629418 GF On-Demand Anodyne FAAH 21 41 CC[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629419 EI On-Demand Anodyne CPT1A 108 43 CC[C@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629419 EI On-Demand Anodyne CPT1B 16 42 CC[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629420 EI On-Demand Anodyne CPT1A 108 43 CC[C@@H]1CCCN1C(=O)Nc1nc(COc2ccccc2)cs1 ZINC000880629420 EI On-Demand Anodyne CPT1B 16 42 CC[C@H]1CN(C(=O)Nc2ccc(Br)cc2OC)CCCO1 ZINC000880629446 FG On-Demand Anodyne DRD4 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(NC(=O)C2CC2)CC1 ZINC000880629459 GF On-Demand Anodyne EPHX2 37 46 COc1cc(Br)ccc1NC(=O)NOCCOC(C)C ZINC000880629482 EF On-Demand Anodyne XIAP 40 33 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](O)CC1 ZINC000880629483 EF On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](O)CC1 ZINC000880629484 EF On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000880629510 GG On-Demand Anodyne EPHX2 43 53 COc1cc(Br)ccc1NC(=O)N1C[C@H](F)C[C@@H]1CO ZINC000880629558 EE On-Demand Anodyne ITGA4 40 44 COc1cc(Br)ccc1NC(=O)N1C[C@@H](F)C[C@H]1CO ZINC000880629559 EE On-Demand Anodyne ITGA4 40 44 COc1cc(Br)ccc1NC(=O)N1C[C@@H](F)C[C@@H]1CO ZINC000880629560 EE On-Demand Anodyne ITGA4 40 44 COc1cc(Br)ccc1NC(=O)N1C[C@H](F)C[C@H]1CO ZINC000880629561 EE On-Demand Anodyne ITGA4 40 44 COc1cc(Br)ccc1NC(=O)N(C)CCCNC(=O)C1CCC1 ZINC000880629585 GG On-Demand Anodyne TBK1 41 39 COc1cc(Br)ccc1NC(=O)NCc1cnnn1C ZINC000880629587 ED On-Demand Anodyne HTR2A 17 40 COc1cc(Br)ccc1NC(=O)NCCN1CCCOCC1 ZINC000880629594 FE On-Demand Anodyne DRD4 42 33 COc1cc(Br)ccc1NC(=O)NCCN1CCCOCC1 ZINC000880629594 FE On-Demand Anodyne DRD3 31 46 COc1cc(Br)ccc1NC(=O)NCCN1CCCOCC1 ZINC000880629594 FE On-Demand Anodyne EPHX2 22 40 COc1cc(Br)ccc1NC(=O)N(C)Cc1cnc(C(C)C)nc1 ZINC000880629607 GI On-Demand Anodyne ROCK2 16 40 NC(=O)COc1cccc(NC(=O)[C@H](CC(N)=O)NC(=O)c2ccccc2Cl)c1 ZINC000880629615 HC On-Demand Anodyne KCNK3 51 37 NC(=O)COc1cccc(NC(=O)[C@H](CC(N)=O)NC(=O)c2ccccc2Cl)c1 ZINC000880629615 HC On-Demand Anodyne KCNK9 48 37 NC(=O)COc1cccc(NC(=O)[C@@H](CC(N)=O)NC(=O)c2ccccc2Cl)c1 ZINC000880629616 HC On-Demand Anodyne KCNK3 51 37 NC(=O)COc1cccc(NC(=O)[C@@H](CC(N)=O)NC(=O)c2ccccc2Cl)c1 ZINC000880629616 HC On-Demand Anodyne KCNK9 48 37 COc1cc(Br)ccc1NC(=O)N1CC(C2CC2)C1 ZINC000880629646 EG On-Demand Anodyne RBP4 45 32 COc1cc(Br)ccc1NC(=O)N(C)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880629653 GH On-Demand Anodyne SLC6A3 31 40 COc1cc(Br)ccc1NC(=O)N(C)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880629653 GH On-Demand Anodyne GLRA1 43 32 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880629657 GH On-Demand Anodyne DRD4 17 46 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880629657 GH On-Demand Anodyne PDGFRB 27 41 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880629657 GH On-Demand Anodyne RBP4 54 43 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880629657 GH On-Demand Anodyne SMO 21 47 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880629658 GH On-Demand Anodyne DRD4 17 46 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880629658 GH On-Demand Anodyne PDGFRB 27 41 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880629658 GH On-Demand Anodyne RBP4 54 43 COc1cc(Br)ccc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880629658 GH On-Demand Anodyne SMO 21 47 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne DRD2 23 43 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne DRD4 16 43 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne DRD3 20 43 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne HTR4 32 40 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne CCR3 26 45 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne BIRC2 35 42 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880629661 GE On-Demand Anodyne EHMT2 55 30 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne DRD2 23 43 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne DRD4 16 43 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne DRD3 20 43 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne HTR4 32 40 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne CCR3 26 45 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne BIRC2 35 42 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880629662 GE On-Demand Anodyne EHMT2 55 30 COc1cc(Br)ccc1NC(=O)NCCCc1cnn(C)n1 ZINC000880629663 FE On-Demand Anodyne QPCT 15 42 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C(C)=O)C1 ZINC000880629664 GF On-Demand Anodyne DRD2 26 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C(C)=O)C1 ZINC000880629664 GF On-Demand Anodyne CCR3 23 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C(C)=O)C1 ZINC000880629664 GF On-Demand Anodyne CACNA1I 40 30 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C(C)=O)C1 ZINC000880629665 GF On-Demand Anodyne DRD2 26 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C(C)=O)C1 ZINC000880629665 GF On-Demand Anodyne CCR3 23 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C(C)=O)C1 ZINC000880629665 GF On-Demand Anodyne CACNA1I 40 30 COc1cc(Br)ccc1NC(=O)N1CCC2(CC1)OCCO2 ZINC000880629675 FF On-Demand Anodyne PDGFRB 18 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CN1CCOCC1 ZINC000880629684 GF On-Demand Anodyne DRD2 25 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CN1CCOCC1 ZINC000880629684 GF On-Demand Anodyne ACKR3 63 33 COc1cc(Br)ccc1NC(=O)N1CC(C)C1 ZINC000880629689 CF On-Demand Anodyne RBP4 35 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](C)[S@](=O)CC1 ZINC000880629696 GF On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](C)[S@@](=O)CC1 ZINC000880629697 GF On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](C)[S@](=O)CC1 ZINC000880629698 GF On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](C)[S@@](=O)CC1 ZINC000880629699 GF On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CCC(O)(C(F)F)CC1 ZINC000880629720 GG On-Demand Anodyne PDGFRB 17 41 COc1cc(Br)ccc1NC(=O)NCc1nc(C2CC2)n[nH]1 ZINC000880629741 FF On-Demand Anodyne ROCK2 15 40 COc1cc(Br)ccc1NC(=O)N1CCC2(CC1)OCCCO2 ZINC000880629766 GG On-Demand Anodyne PDGFRB 16 40 COc1cc(Br)ccc1NC(=O)N1CCC2(CCC2)C1 ZINC000880629809 EH On-Demand Anodyne EPHX2 25 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1CCCO ZINC000880629820 GE On-Demand Anodyne DRD2 41 52 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN1CCCO ZINC000880629820 GE On-Demand Anodyne ACKR3 65 33 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1CCCO ZINC000880629821 GE On-Demand Anodyne DRD2 41 52 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN1CCCO ZINC000880629821 GE On-Demand Anodyne ACKR3 65 33 COc1cc(Br)ccc1NC(=O)N(C)Cc1nc[nH]n1 ZINC000880629833 EE On-Demand Anodyne ROCK2 20 40 COc1cc(Br)ccc1NC(=O)NOCCO ZINC000880629848 DD On-Demand Anodyne MAP2K1 18 44 COc1cc(Br)ccc1NC(=O)NCCCn1ccnc1C ZINC000880629858 FG On-Demand Anodyne QPCT 26 46 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CC(N)=O)CC1 ZINC000880629873 GF On-Demand Anodyne PDGFRB 24 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CC(N)=O)CC1 ZINC000880629874 GF On-Demand Anodyne PDGFRB 24 40 COc1cc(Br)ccc1NC(=O)N1CCCC[C@@H]1c1nc(C)no1 ZINC000880629883 GH On-Demand Anodyne CPT1A 79 42 COc1cc(Br)ccc1NC(=O)N1CCCC[C@H]1c1nc(C)no1 ZINC000880629884 GH On-Demand Anodyne CPT1A 79 42 COc1cc(Br)ccc1NC(=O)NCc1ccc(C)n(C)c1=O ZINC000880629919 GF On-Demand Anodyne GRIN1 18 41 COc1cc(Br)ccc1NC(=O)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880629923 GG On-Demand Anodyne CPT1A 55 35 COc1cc(Br)ccc1NC(=O)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880629924 GG On-Demand Anodyne CPT1A 55 35 COc1cc(Br)ccc1NC(=O)N1CC2(CCOCC2)C1 ZINC000880629925 FG On-Demand Anodyne LRRK2 20 40 COc1cc(Br)ccc1NC(=O)N1CCC(Cn2cncn2)CC1 ZINC000880629932 GF On-Demand Anodyne PDGFRB 36 40 COc1cc(Br)ccc1NC(=O)Nc1cc(C2CCOCC2)[nH]n1 ZINC000880629934 GH On-Demand Anodyne CDK2 15 51 C=CCN(CCOC)C(=O)Nc1ccc(Br)cc1OC ZINC000880629935 EG On-Demand Mild LSS 48 41 COc1cc(Br)ccc1NC(=O)N1CCN(C[C@H](C)O)CC1 ZINC000880629945 FD On-Demand Anodyne PDGFRB 32 40 COC(=O)Cn1ncc(NC(=O)Nc2ccc(Br)cc2OC)c1C ZINC000880630009 GF On-Demand Anodyne HTR2A 16 40 COc1cc(Br)ccc1NC(=O)N1CCCN(C(=O)C2CC2)CC1 ZINC000880630014 GF On-Demand Anodyne PDGFRB 27 43 COc1cc(Br)ccc1NC(=O)N1CCCN(C(=O)C2CC2)CC1 ZINC000880630014 GF On-Demand Anodyne RBP4 20 42 COc1cc(Br)ccc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880630027 GF On-Demand Anodyne NQO2 17 43 COc1cc(Br)ccc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880630027 GF On-Demand Anodyne MTNR1A 29 41 COc1cc(Br)ccc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880630027 GF On-Demand Anodyne MTNR1B 30 41 COc1cc(Br)ccc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880630027 GF On-Demand Anodyne IKBKE 41 41 COc1cc(Br)ccc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880630027 GF On-Demand Anodyne TBK1 81 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2c[nH]nc2C)CC1 ZINC000880630035 GH On-Demand Anodyne RBP4 35 44 COc1cc(Br)ccc1NC(=O)N1CC(C(F)(F)F)C1 ZINC000880630039 FG On-Demand Anodyne RBP4 52 33 COc1cc(Br)ccc1NC(=O)NCCN1CCN(C)C(C)(C)C1 ZINC000880630047 GF On-Demand Anodyne DRD4 41 31 COc1cc(Br)ccc1NC(=O)NCCN1CCN(C)C(C)(C)C1 ZINC000880630047 GF On-Demand Anodyne DRD3 26 44 COc1cc(Br)ccc1NC(=O)NCC1(N2CCOCC2)CC1 ZINC000880630085 GE On-Demand Anodyne HCN1 66 39 COc1cc(Br)ccc1NC(=O)NCC1(N2CCOCC2)CC1 ZINC000880630085 GE On-Demand Anodyne HCN4 52 37 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880630111 FG On-Demand Anodyne PDGFRB 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880630111 FG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880630111 FG On-Demand Anodyne PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880630112 FG On-Demand Anodyne PDGFRB 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880630112 FG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880630112 FG On-Demand Anodyne PTPN1 16 40 COC(=O)N1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630128 GF On-Demand Anodyne EPHX2 50 50 C=CCN(C)C(=O)Nc1ccc(Br)cc1OC ZINC000880630165 CG On-Demand Mild LSS 41 39 COc1cc(Br)ccc1NC(=O)N1CCC(c2cnn(C)c2)CC1 ZINC000880630171 GH On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)NC1CCC(NC(C)=O)CC1 ZINC000880630180 GG On-Demand Anodyne EPHX2 30 40 COc1cc(Br)ccc1NC(=O)N1CCc2c(ncn2C)C1 ZINC000880630182 FF On-Demand Anodyne PDGFRB 18 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1c1nc(C)no1 ZINC000880630224 GH On-Demand Anodyne CPT1A 50 39 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1c1nc(C)no1 ZINC000880630225 GH On-Demand Anodyne CPT1A 50 39 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](N(C)C)CC1 ZINC000880630234 FG On-Demand Anodyne RBP4 28 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](N(C)C)CC1 ZINC000880630235 FG On-Demand Anodyne RBP4 28 41 COc1cc(Br)ccc1NC(=O)NCC1OCCCO1 ZINC000880630244 EE On-Demand Anodyne GPR35 40 35 COCCCNC(=O)Nc1ccc(Br)cc1OC ZINC000880630339 DF On-Demand Anodyne FOLH1 15 50 COCCCCCNC(=O)Nc1ccc(Br)cc1OC ZINC000880630344 EG On-Demand Anodyne FOLH1 15 48 N#CCCN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630347 FE On-Demand Mild PDGFRB 40 44 N#CCCN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630347 FE On-Demand Mild FAAH 29 48 COc1cc(Br)ccc1NC(=O)N(C)CC(=O)N1CCOCC1 ZINC000880630354 GD On-Demand Anodyne LRRK2 28 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccnn2C)CC1 ZINC000880630360 GH On-Demand Anodyne RBP4 25 40 COc1cc(Br)ccc1NC(=O)N1CCC(NC(=O)C(C)C)CC1 ZINC000880630361 GG On-Demand Anodyne EPHX2 23 40 COc1cc(Br)ccc1NC(=O)N1CCC(NC(=O)C(C)C)CC1 ZINC000880630361 GG On-Demand Anodyne RBP4 26 43 COc1cc(Br)ccc1NC(=O)N(C)[C@H](C)c1cccnc1 ZINC000880630362 FI On-Demand Anodyne KCNA5 21 51 COc1cc(Br)ccc1NC(=O)N(C)[C@@H](C)c1cccnc1 ZINC000880630363 FI On-Demand Anodyne KCNA5 21 51 COC[C@@H]1CCCN(C(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630374 FG On-Demand Anodyne PDGFRB 29 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CCO)C1 ZINC000880630378 FG On-Demand Anodyne PDGFRB 22 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CCO)C1 ZINC000880630379 FG On-Demand Anodyne PDGFRB 22 40 CS[C@@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630392 EG On-Demand Anodyne EPHX2 27 42 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630394 FF On-Demand Anodyne PDGFRB 23 40 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630394 FF On-Demand Anodyne FAAH 16 40 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630394 FF On-Demand Anodyne S1PR2 25 40 COc1cc(Br)ccc1NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000880630399 GD On-Demand Anodyne PDGFRB 19 42 COc1cc(Br)ccc1NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000880630399 GD On-Demand Anodyne RBP4 28 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2nncn2C)CC1 ZINC000880630410 GF On-Demand Anodyne RBP4 23 40 CN1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]21 ZINC000880630416 FF On-Demand Anodyne PDGFRB 27 42 CN1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]21 ZINC000880630416 FF On-Demand Anodyne RBP4 47 35 CN1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]21 ZINC000880630417 FF On-Demand Anodyne PDGFRB 27 42 CN1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]21 ZINC000880630417 FF On-Demand Anodyne RBP4 47 35 COc1cc(Br)ccc1NC(=O)N1CCNC(=O)CC1 ZINC000880630422 ED On-Demand Anodyne RBP4 21 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1cncn1 ZINC000880630558 GF On-Demand Anodyne ACKR3 64 34 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1Cn1cncn1 ZINC000880630560 GF On-Demand Anodyne ACKR3 64 34 COc1cc(Br)ccc1NC(=O)NCCCN1CCCC1=O ZINC000880630561 FF On-Demand Anodyne CCR3 27 40 COc1cc(Br)ccc1NC(=O)NCCCN1CCCC1=O ZINC000880630561 FF On-Demand Anodyne TYRO3 20 46 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CN(C)CCO1 ZINC000880630571 FD On-Demand Anodyne EPHA2 17 45 COc1cc(Br)ccc1NC(=O)N1CCC(c2cnc[nH]2)CC1 ZINC000880630572 GH On-Demand Anodyne RBP4 27 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CN(C)CCO1 ZINC000880630573 FD On-Demand Anodyne EPHA2 17 45 COc1cc(Br)ccc1NC(=O)N1CCC(N(C)C(C)=O)CC1 ZINC000880630576 GF On-Demand Anodyne PDGFRB 15 41 COc1cc(Br)ccc1NC(=O)N1CCC(N(C)C(C)=O)CC1 ZINC000880630576 GF On-Demand Anodyne RBP4 28 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CCCO ZINC000880630578 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CCCO ZINC000880630578 FG On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CCCO ZINC000880630579 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CCCO ZINC000880630579 FG On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)N1CCOCC2(CCOCC2)C1 ZINC000880630591 GG On-Demand Anodyne LRRK2 28 43 COc1cc(Br)ccc1NC(=O)NCCC(=O)N1CCCCC1 ZINC000880630596 GF On-Demand Anodyne HRH2 15 43 COc1cc(Br)ccc1NC(=O)Nc1cnn(CC(=O)N(C)C)c1 ZINC000880630597 GE On-Demand Anodyne HTR2A 18 40 COc1cc(Br)ccc1NC(=O)Nc1cnn(CC(=O)N(C)C)c1 ZINC000880630597 GE On-Demand Anodyne PDGFRB 25 43 COc1cc(Br)ccc1NC(=O)Nc1cnn(CC(=O)N(C)C)c1 ZINC000880630597 GE On-Demand Anodyne FLT4 20 43 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne DRD2 24 48 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne DRD4 24 40 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne DRD3 16 46 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne HTR4 45 48 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne SIGMAR1 17 59 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne SSTR5 49 39 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne CCR3 22 42 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne EPHX2 42 48 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne PDK1 45 32 CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630599 FG On-Demand Anodyne MCHR1 16 41 COc1cc(Br)ccc1NC(=O)NCCCN1CCCCC1=O ZINC000880630602 GF On-Demand Anodyne HRH2 19 42 COc1cc(Br)ccc1NC(=O)NCCCN1CCCCC1=O ZINC000880630602 GF On-Demand Anodyne CCR3 34 40 COc1cc(Br)ccc1NC(=O)NCCCN1CCCCC1=O ZINC000880630602 GF On-Demand Anodyne TYRO3 20 43 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880630604 FG On-Demand Anodyne DRD2 34 43 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880630604 FG On-Demand Anodyne ACKR3 64 33 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CN(C)CCN1C ZINC000880630605 FD On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CN(C)CCN1C ZINC000880630605 FD On-Demand Anodyne ACKR3 60 31 COc1cc(Br)ccc1NC(=O)NC[C@H]1CN(C)CCN1C ZINC000880630606 FD On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CN(C)CCN1C ZINC000880630606 FD On-Demand Anodyne ACKR3 60 31 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880630607 FG On-Demand Anodyne DRD2 34 43 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880630607 FG On-Demand Anodyne ACKR3 64 33 COc1cc(Br)ccc1NC(=O)NCC(=O)NC(C)C ZINC000880630608 EE On-Demand Anodyne F7 22 40 COCCCCNC(=O)Nc1ccc(Br)cc1OC ZINC000880630610 EG On-Demand Anodyne FOLH1 15 49 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)[C@H](C)O)CC1 ZINC000880630617 GD On-Demand Anodyne PDGFRB 27 42 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)[C@H](C)O)CC1 ZINC000880630617 GD On-Demand Anodyne RBP4 19 41 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)[C@@H](C)O)CC1 ZINC000880630619 GD On-Demand Anodyne PDGFRB 27 42 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)[C@@H](C)O)CC1 ZINC000880630619 GD On-Demand Anodyne RBP4 19 41 COc1cc(Br)ccc1NC(=O)N1CCC(CCC(N)=O)CC1 ZINC000880630625 GF On-Demand Anodyne PDGFRB 19 40 COc1cc(Br)ccc1NC(=O)N1CCC(CCC(N)=O)CC1 ZINC000880630625 GF On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(CCC(N)=O)CC1 ZINC000880630625 GF On-Demand Anodyne PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CCC(CCC(N)=O)CC1 ZINC000880630625 GF On-Demand Anodyne RBP4 23 40 C#CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630628 FF On-Demand Mild PDGFRB 31 45 C#CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630628 FF On-Demand Mild FAAH 22 41 C#CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630628 FF On-Demand Mild NPY5R 30 41 C#CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630628 FF On-Demand Mild S1PR2 31 49 COc1cc(Br)ccc1NC(=O)N1CCc2cncnc2C1 ZINC000880630630 FF On-Demand Anodyne MAPK1 45 36 COc1cc(Br)ccc1NC(=O)N[C@@H]1CC[C@H](CO)CC1 ZINC000880630642 FG On-Demand Anodyne EPHX2 28 40 COc1cc(Br)ccc1NC(=O)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880630645 FG On-Demand Anodyne EPHX2 28 40 COc1cc(Br)ccc1NC(=O)NC1CCC(C(N)=O)CC1 ZINC000880630646 FF On-Demand Anodyne EPHX2 22 40 COCC1(O)CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630656 FE On-Demand Anodyne PDGFRB 26 41 COc1cc(Br)ccc1NC(=O)N1CC[C@H](Cc2cnn(C)c2)C1 ZINC000880630658 GG On-Demand Anodyne CCR3 23 41 C[C@@H](O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630660 EF On-Demand Anodyne PDGFRB 40 44 C[C@@H](O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630660 EF On-Demand Anodyne FAAH 19 40 C[C@@H](O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630660 EF On-Demand Anodyne S1PR2 27 42 C[C@@H](O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880630660 EF On-Demand Anodyne EPHX2 24 41 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](Cc2cnn(C)c2)C1 ZINC000880630661 GG On-Demand Anodyne CCR3 23 41 COc1cc(Br)ccc1NC(=O)NCC1CCN(C(C)=O)CC1 ZINC000880630674 GF On-Demand Anodyne CCR3 28 42 COc1cc(Br)ccc1NC(=O)NCC1CCN(C(C)=O)CC1 ZINC000880630674 GF On-Demand Anodyne EPHX2 18 44 COc1cc(Br)ccc1NC(=O)NCC1CCN(C(C)=O)CC1 ZINC000880630674 GF On-Demand Anodyne CACNA1I 58 33 COc1cc(Br)ccc1NC(=O)NCC1CCN(C(C)=O)CC1 ZINC000880630674 GF On-Demand Anodyne ACKR3 59 31 COc1cc(Br)ccc1NC(=O)N1CCN(C)CC1 ZINC000880630676 EE On-Demand Anodyne HTR1B 17 49 COc1cc(Br)ccc1NC(=O)N1CCN(C)CC1 ZINC000880630676 EE On-Demand Anodyne PDGFRB 34 45 COc1cc(Br)ccc1NC(=O)N1CCN(C)CC1 ZINC000880630676 EE On-Demand Anodyne RBP4 25 44 COc1cc(Br)ccc1NC(=O)N1CC[C@H](C2CCN(C)CC2)C1 ZINC000880630678 GH On-Demand Anodyne HTR1B 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](C2CCN(C)CC2)C1 ZINC000880630680 GH On-Demand Anodyne HTR1B 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](N(C)C)C1 ZINC000880630682 EF On-Demand Anodyne RBP4 34 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](N(C)C)C1 ZINC000880630684 EF On-Demand Anodyne RBP4 34 40 COc1cc(Br)ccc1NC(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000880630685 GG On-Demand Anodyne PANC 53 36 COc1cc(Br)ccc1NC(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000880630696 GG On-Demand Anodyne PANC 53 36 COc1cc(Br)ccc1NC(=O)N1CCC(CNC(C)=O)CC1 ZINC000880630701 GF On-Demand Anodyne PDGFRB 20 40 COc1cc(Br)ccc1NC(=O)N1CCC(CNC(C)=O)CC1 ZINC000880630701 GF On-Demand Anodyne PTPN2 19 43 COc1cc(Br)ccc1NC(=O)N1CCC(CNC(C)=O)CC1 ZINC000880630701 GF On-Demand Anodyne PTPN1 17 43 COc1cc(Br)ccc1NC(=O)N1CCC(CNC(C)=O)CC1 ZINC000880630701 GF On-Demand Anodyne CACNA1I 52 31 COCC1CC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630704 EF On-Demand Anodyne EPHX2 29 44 COc1cc(Br)ccc1NC(=O)N1CCC(c2nccs2)CC1 ZINC000880630710 GI On-Demand Anodyne RBP4 28 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](N2CCCC2)C1 ZINC000880630712 FG On-Demand Anodyne L3MBTL3 92 44 COc1cc(Br)ccc1NC(=O)N1CC[C@H](N2CCCC2)C1 ZINC000880630714 FG On-Demand Anodyne L3MBTL3 92 44 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(Br)cc1OC ZINC000880630715 FE On-Demand Anodyne LGMN 64 39 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630716 GG On-Demand Anodyne PDGFRB 24 40 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630716 GG On-Demand Anodyne NPY5R 27 42 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880630716 GG On-Demand Anodyne EPHX2 37 41 COc1cc(Br)ccc1NC(=O)N(C)Cc1cnn(C)c1 ZINC000880630723 FF On-Demand Anodyne ROCK2 17 41 COc1cc(Br)ccc1NC(=O)N1CCC(Cn2cccn2)CC1 ZINC000880630729 GH On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(Cn2cccn2)CC1 ZINC000880630729 GH On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CCN(c2cnccn2)CC1 ZINC000880630756 GF On-Demand Anodyne PDGFRB 53 46 COc1cc(Br)ccc1NC(=O)N1CCN(c2cnccn2)CC1 ZINC000880630756 GF On-Demand Anodyne RBP4 20 42 COc1cc(Br)ccc1NC(=O)N(C)[C@H]1CCN(C)[C@@H](C)C1 ZINC000880630759 FG On-Demand Anodyne ACKR3 59 30 COc1cc(Br)ccc1NC(=O)N(C)[C@@H]1CCN(C)[C@H](C)C1 ZINC000880630760 FG On-Demand Anodyne ACKR3 59 30 COc1cc(Br)ccc1NC(=O)N(C)[C@@H]1CCN(C)[C@@H](C)C1 ZINC000880630761 FG On-Demand Anodyne ACKR3 59 30 COc1cc(Br)ccc1NC(=O)N(C)[C@H]1CCN(C)[C@H](C)C1 ZINC000880630762 FG On-Demand Anodyne ACKR3 59 30 COc1cc(Br)ccc1NC(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000880630767 GF On-Demand Anodyne HTR4 19 40 COc1cc(Br)ccc1NC(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000880630767 GF On-Demand Anodyne EPHX2 49 53 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C)C1 ZINC000880630768 FF On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C)C1 ZINC000880630768 FF On-Demand Anodyne DRD3 18 42 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C)C1 ZINC000880630768 FF On-Demand Anodyne CACNA1I 52 33 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCCN(C)C1 ZINC000880630768 FF On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C)C1 ZINC000880630769 FF On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C)C1 ZINC000880630769 FF On-Demand Anodyne DRD3 18 42 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C)C1 ZINC000880630769 FF On-Demand Anodyne CACNA1I 52 33 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCCN(C)C1 ZINC000880630769 FF On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)NC1CCOCC1 ZINC000880630772 EF On-Demand Anodyne EPHX2 22 40 COc1cc(Br)ccc1NC(=O)N1CCC(C(=O)N(C)C)CC1 ZINC000880630777 GF On-Demand Anodyne RBP4 23 40 CCN1CC[C@H](CNC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630785 FF On-Demand Anodyne DRD2 25 40 CCN1CC[C@H](CNC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630785 FF On-Demand Anodyne DRD4 15 54 CCN1CC[C@H](CNC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630785 FF On-Demand Anodyne HTR4 53 38 CCN1CC[C@H](CNC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630785 FF On-Demand Anodyne CCR3 40 37 CCN1CC[C@H](CNC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630785 FF On-Demand Anodyne CACNA1I 64 35 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne DRD2 31 48 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne DRD4 30 40 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne DRD3 31 46 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne HTR4 68 43 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne SIGMAR1 17 56 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne CCR3 27 46 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne EPHX2 36 43 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne PDK1 45 31 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne MCHR1 21 41 COCCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630789 GF On-Demand Anodyne EHMT2 46 30 COc1cc(Br)ccc1NC(=O)NCCCNC(C)=O ZINC000880630790 EE On-Demand Anodyne FOLH1 32 55 COc1cc(Br)ccc1NC(=O)NCCCNC(C)=O ZINC000880630790 EE On-Demand Anodyne NQO2 55 34 COc1cc(Br)ccc1NC(=O)NCCCNC(C)=O ZINC000880630790 EE On-Demand Anodyne MTNR1A 63 45 COc1cc(Br)ccc1NC(=O)NCCCNC(C)=O ZINC000880630790 EE On-Demand Anodyne MTNR1B 59 45 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)=O)CC1 ZINC000880630793 FE On-Demand Anodyne PDGFRB 32 46 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)=O)CC1 ZINC000880630793 FE On-Demand Anodyne RBP4 25 45 CNC(=O)CN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630794 GD On-Demand Anodyne DRD4 30 43 CNC(=O)CN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630794 GD On-Demand Anodyne SIGMAR1 15 57 CNC(=O)CN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630794 GD On-Demand Anodyne EPHX2 33 43 CNC(=O)CN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630794 GD On-Demand Anodyne PDK1 46 33 CNC(=O)CN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630794 GD On-Demand Anodyne MCHR1 15 41 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630796 FF On-Demand Anodyne SLC6A4 20 45 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630796 FF On-Demand Anodyne SLC6A3 43 45 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630797 FF On-Demand Anodyne SLC6A4 20 45 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630797 FF On-Demand Anodyne SLC6A3 43 45 COc1cc(Br)ccc1NC(=O)N(C)[C@H](C)c1ccccn1 ZINC000880630799 FI On-Demand Anodyne GRM4 16 41 COc1cc(Br)ccc1NC(=O)N(C)[C@@H](C)c1ccccn1 ZINC000880630800 FI On-Demand Anodyne GRM4 16 41 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne EGFR 15 41 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne HTR1A 30 41 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne DRD2 37 43 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne ADRA1D 30 43 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne ADRA1A 35 43 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne ADRA1B 24 43 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne DRD3 57 43 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne CCR3 39 45 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne CHRNA7 16 45 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne MAP2K1 20 41 COc1cc(Br)ccc1NC(=O)NCCCN1CCOCC1 ZINC000880630801 FE On-Demand Anodyne EPHX2 27 43 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1cccn1 ZINC000880630802 GG On-Demand Anodyne DRD2 26 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1cccn1 ZINC000880630802 GG On-Demand Anodyne ACKR3 54 34 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1Cn1cccn1 ZINC000880630803 GG On-Demand Anodyne DRD2 26 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1Cn1cccn1 ZINC000880630803 GG On-Demand Anodyne ACKR3 54 34 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CO ZINC000880630810 EE On-Demand Anodyne DRD2 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1CO ZINC000880630810 EE On-Demand Anodyne ACKR3 65 34 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CO ZINC000880630811 EE On-Demand Anodyne DRD2 31 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CO ZINC000880630811 EE On-Demand Anodyne ACKR3 65 34 COc1cc(Br)ccc1NC(=O)N1CCCN(C(C)=O)CC1 ZINC000880630813 FF On-Demand Anodyne PDGFRB 24 44 COc1cc(Br)ccc1NC(=O)N1CCCN(C(C)=O)CC1 ZINC000880630813 FF On-Demand Anodyne RBP4 24 42 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne CCR1 33 40 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne CCR3 33 43 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne EPHX2 43 47 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne PDK1 44 33 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne CXCR3 20 40 COc1cc(Br)ccc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880630818 GG On-Demand Anodyne MCHR1 17 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](NS(C)(=O)=O)C1 ZINC000880630837 GD On-Demand Anodyne CCR8 72 34 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](NS(C)(=O)=O)C1 ZINC000880630838 GD On-Demand Anodyne CCR8 72 34 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630840 FG On-Demand Anodyne TIMP3 69 35 COc1cc(Br)ccc1NC(=O)NCCCn1ccnc1 ZINC000880630845 FF On-Demand Anodyne TBXAS1 52 48 COc1cc(Br)ccc1NC(=O)NCCCn1ccnc1 ZINC000880630845 FF On-Demand Anodyne HMOX2 40 43 COc1cc(Br)ccc1NC(=O)NCCCn1ccnc1 ZINC000880630845 FF On-Demand Anodyne QPCT 58 68 COc1cc(Br)ccc1NC(=O)N1CCC(CO)CC1 ZINC000880630851 EF On-Demand Anodyne PDGFRB 29 42 COc1cc(Br)ccc1NC(=O)N1CCC(CO)CC1 ZINC000880630851 EF On-Demand Anodyne PTPN2 19 42 COc1cc(Br)ccc1NC(=O)N1CCC(CO)CC1 ZINC000880630851 EF On-Demand Anodyne PTPN1 17 42 COc1cc(Br)ccc1NC(=O)N1CCC(CO)CC1 ZINC000880630851 EF On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)NC1CCN(CC#N)CC1 ZINC000880630853 FF On-Demand Mild EPHX2 31 43 COc1cc(Br)ccc1NC(=O)NC1CCN(CC#N)CC1 ZINC000880630853 FF On-Demand Mild PDK1 43 30 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne DRD2 26 42 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne DRD4 44 35 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne DRD3 38 49 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne CNR2 15 41 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne MAP2K1 15 43 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne EPHX2 25 43 COc1cc(Br)ccc1NC(=O)NCCN1CCOCC1 ZINC000880630861 FD On-Demand Anodyne LRRK2 25 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2CC[C@H](C1)O2 ZINC000880630866 EF On-Demand Anodyne PDGFRB 22 41 COc1cc(Br)ccc1NC(=O)N(C)CCN1CCOCC1 ZINC000880630869 FE On-Demand Anodyne CASR 52 42 COc1cc(Br)ccc1NC(=O)N(C)CCN1CCOCC1 ZINC000880630869 FE On-Demand Anodyne PRKDC 17 42 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1c1ccccn1 ZINC000880630870 GI On-Demand Anodyne DRD4 16 43 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1c1ccccn1 ZINC000880630870 GI On-Demand Anodyne CPT1A 44 35 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1c1ccccn1 ZINC000880630871 GI On-Demand Anodyne DRD4 16 43 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1c1ccccn1 ZINC000880630871 GI On-Demand Anodyne CPT1A 44 35 COc1cc(Br)ccc1NC(=O)N1CCn2cnnc2C1 ZINC000880630873 FE On-Demand Anodyne PDGFRB 16 41 COCC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630880 FG On-Demand Anodyne PDGFRB 31 42 COCC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630880 FG On-Demand Anodyne PTPN2 19 42 COCC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630880 FG On-Demand Anodyne PTPN1 16 42 COCC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630880 FG On-Demand Anodyne RBP4 23 40 NC(=O)COc1cccc(NC(=O)c2ccc3c(c2[N+](=O)[O-])C(=O)c2ccccc2C3=O)c1 ZINC000880630881 IE On-Demand Clean KCNK3 52 34 NC(=O)COc1cccc(NC(=O)c2ccc3c(c2[N+](=O)[O-])C(=O)c2ccccc2C3=O)c1 ZINC000880630881 IE On-Demand Clean KCNK9 50 34 COc1cc(Br)ccc1NC(=O)N1CCN(c2cccnn2)CC1 ZINC000880630889 GF On-Demand Anodyne PDGFRB 41 44 COc1cc(Br)ccc1NC(=O)N1CCN(c2cccnn2)CC1 ZINC000880630889 GF On-Demand Anodyne RBP4 23 44 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C2CC2)CC1 ZINC000880630890 GF On-Demand Anodyne PDGFRB 32 45 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C2CC2)CC1 ZINC000880630890 GF On-Demand Anodyne RBP4 22 44 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](c2nc(C)no2)C1 ZINC000880630894 GH On-Demand Anodyne SMO 22 46 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](c2nc(C)no2)C1 ZINC000880630895 GH On-Demand Anodyne SMO 22 46 COc1cc(Br)ccc1NC(=O)N1CCC(c2cc[nH]n2)CC1 ZINC000880630902 GH On-Demand Anodyne RBP4 28 41 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](NC(=O)C(C)C)C1 ZINC000880630919 GG On-Demand Anodyne BIRC2 34 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](NC(=O)C(C)C)C1 ZINC000880630920 GG On-Demand Anodyne BIRC2 34 40 CCC(=O)N1CCCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630924 GF On-Demand Anodyne PDGFRB 26 41 CCC(=O)N1CCCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880630924 GF On-Demand Anodyne RBP4 19 40 CCN1CC[C@@H]1CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880630931 EE On-Demand Anodyne EPHX2 15 41 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630992 FE On-Demand Anodyne PTR1 45 34 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880630993 FE On-Demand Anodyne PTR1 45 34 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H](C(F)(F)F)O1 ZINC000880630995 GH On-Demand Anodyne RBP4 54 35 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H](C(F)(F)F)O1 ZINC000880630996 GH On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H](C(F)(F)F)O1 ZINC000880630997 GH On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H](C(F)(F)F)O1 ZINC000880630998 GH On-Demand Anodyne RBP4 54 35 COc1cc(Br)ccc1NC(=O)NCC(=O)N1CCCCC1 ZINC000880631000 FF On-Demand Anodyne PRMT3 17 44 COc1cc(Br)ccc1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880631001 GG On-Demand Anodyne RBP4 23 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1OC2CCC1CC2 ZINC000880631005 EG On-Demand Anodyne PDGFRB 20 40 COc1cc(Br)ccc1NC(=O)N1CCS(=O)CC1 ZINC000880631045 EE On-Demand Anodyne RBP4 21 40 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C(C)C)CC1 ZINC000880631051 GF On-Demand Anodyne PDGFRB 29 43 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C(C)C)CC1 ZINC000880631051 GF On-Demand Anodyne RBP4 20 42 CC(=O)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631056 EG On-Demand Anodyne PDGFRB 26 41 CC(=O)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631056 EG On-Demand Anodyne CPT1A 55 37 CC(=O)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631056 EG On-Demand Anodyne EPHX2 18 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631057 EG On-Demand Anodyne PDGFRB 26 41 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631057 EG On-Demand Anodyne CPT1A 55 37 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631057 EG On-Demand Anodyne EPHX2 18 40 CCOC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631063 GG On-Demand Anodyne CCR8 15 41 CCOC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631063 GG On-Demand Anodyne PTR1 48 36 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne HTR1A 55 43 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne DRD2 61 46 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne DRD4 44 44 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne HRH2 15 43 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne ADRA1D 31 44 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne HTR2A 25 44 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne HTR2C 15 41 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne ADRA1A 38 44 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne ADRA1B 24 44 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne DRD3 93 46 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne HTR4 41 40 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne FGFR1 20 40 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne SIGMAR1 15 46 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne SRC 15 40 COc1cc(Br)ccc1NC(=O)NCCCCN1CCN(C)CC1 ZINC000880631079 GF On-Demand Anodyne CCR3 39 44 COc1cc(Br)ccc1NC(=O)N1CCC[C@H](CO)C1 ZINC000880631081 EF On-Demand Anodyne PDGFRB 23 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H](CO)C1 ZINC000880631082 EF On-Demand Anodyne PDGFRB 23 40 COc1cc(Br)ccc1NC(=O)NC[C@H](O)CC(C)C ZINC000880631116 EF On-Demand Anodyne ANPEP 25 46 COc1cc(Br)ccc1NC(=O)NC[C@@H](O)CC(C)C ZINC000880631117 EF On-Demand Anodyne ANPEP 25 46 COc1cc(Br)ccc1NC(=O)N1CCS(=O)(=O)CC1 ZINC000880631119 FD On-Demand Anodyne RBP4 21 40 CN1CCN(C2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CC1 ZINC000880631120 GF On-Demand Anodyne PDGFRB 28 43 CN1CCN(C2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CC1 ZINC000880631120 GF On-Demand Anodyne SLC6A5 15 40 CN1CCN(C2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CC1 ZINC000880631120 GF On-Demand Anodyne SCD1 16 40 CN1CCN(C2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CC1 ZINC000880631120 GF On-Demand Anodyne L3MBTL3 61 42 COc1cc(Br)ccc1NC(=O)N(Cc1cccnc1)C1CC1 ZINC000880631121 GI On-Demand Anodyne CHRNA7 48 48 COc1cc(Br)ccc1NC(=O)N(Cc1cccnc1)C1CC1 ZINC000880631121 GI On-Demand Anodyne ROCK2 29 45 COc1cc(Br)ccc1NC(=O)N(Cc1cccnc1)C1CC1 ZINC000880631121 GI On-Demand Anodyne ACHP_LYMST 22 41 COc1cc(Br)ccc1NC(=O)N1CCN(C[C@@H](C)O)CC1 ZINC000880631122 FD On-Demand Anodyne PDGFRB 32 40 COc1cc(Br)ccc1NC(=O)N1CCN2CCC[C@@H]2C1 ZINC000880631127 FF On-Demand Anodyne L3MBTL3 46 36 COc1cc(Br)ccc1NC(=O)N1CCN2CCC[C@H]2C1 ZINC000880631128 FF On-Demand Anodyne L3MBTL3 46 36 Cc1csc([C@H]2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)n1 ZINC000880631133 GI On-Demand Anodyne CPT1A 36 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880631136 EG On-Demand Anodyne PDGFRB 26 42 COCCN(Cc1cccnc1)C(=O)Nc1ccc(Br)cc1OC ZINC000880631137 GH On-Demand Anodyne CHRNA7 40 45 COCCN(Cc1cccnc1)C(=O)Nc1ccc(Br)cc1OC ZINC000880631137 GH On-Demand Anodyne ROCK2 30 44 COc1cc(Br)ccc1NC(=O)NCCCCn1ccnc1 ZINC000880631144 FG On-Demand Anodyne TBXAS1 52 48 COc1cc(Br)ccc1NC(=O)NCCCCn1ccnc1 ZINC000880631144 FG On-Demand Anodyne HMOX2 40 43 COc1cc(Br)ccc1NC(=O)NCCCCn1ccnc1 ZINC000880631144 FG On-Demand Anodyne QPCT 55 65 O=C1CCCN1C[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631145 GG On-Demand Anodyne CPT1A 107 36 O=C1CCCN1C[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631145 GG On-Demand Anodyne CPT2 43 35 O=C1CCCN1C[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631146 GG On-Demand Anodyne CPT1A 107 36 O=C1CCCN1C[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631146 GG On-Demand Anodyne CPT2 43 35 COc1cc(Br)ccc1NC(=O)N[C@@H](C)Cn1ccnc1 ZINC000880631162 FF On-Demand Anodyne TBXAS1 28 46 COc1cc(Br)ccc1NC(=O)N[C@@H](C)Cn1ccnc1 ZINC000880631162 FF On-Demand Anodyne QPCT 25 45 COc1cc(Br)ccc1NC(=O)N[C@H](C)Cn1ccnc1 ZINC000880631163 FF On-Demand Anodyne TBXAS1 28 46 COc1cc(Br)ccc1NC(=O)N[C@H](C)Cn1ccnc1 ZINC000880631163 FF On-Demand Anodyne QPCT 25 45 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne DRD2 18 44 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne DRD3 19 43 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne HTR4 51 39 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne CCR3 30 45 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne SLC6A5 17 44 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne EPHX2 38 44 COc1cc(Br)ccc1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880631168 GF On-Demand Anodyne MCHR1 17 41 COc1cc(Br)ccc1NC(=O)N1CCC(NC(C)C)CC1 ZINC000880631169 FG On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)NC1CCN(C)CC1 ZINC000880631172 EF On-Demand Anodyne HTR4 29 46 COc1cc(Br)ccc1NC(=O)NC1CCN(C)CC1 ZINC000880631172 EF On-Demand Anodyne EPHX2 43 45 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1c1cccnc1 ZINC000880631179 GI On-Demand Anodyne CHRNA7 30 47 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1c1cccnc1 ZINC000880631179 GI On-Demand Anodyne ACHP_LYMST 19 47 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1c1cccnc1 ZINC000880631180 GI On-Demand Anodyne CHRNA7 30 47 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1c1cccnc1 ZINC000880631180 GI On-Demand Anodyne ACHP_LYMST 19 47 COCC(=O)N1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631187 GD On-Demand Anodyne PDGFRB 29 42 COCC(=O)N1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631187 GD On-Demand Anodyne RBP4 19 41 COc1cc(Br)ccc1NC(=O)N1CCSCC1 ZINC000880631192 EG On-Demand Anodyne PDGFRB 16 42 COc1cc(Br)ccc1NC(=O)N1CCSCC1 ZINC000880631192 EG On-Demand Anodyne RBP4 24 41 COc1cc(Br)ccc1NC(=O)N1CCCN(C(=O)C(C)C)CC1 ZINC000880631204 GG On-Demand Anodyne PDGFRB 26 41 COc1cc(Br)ccc1NC(=O)N1CCCN(C(=O)C(C)C)CC1 ZINC000880631204 GG On-Demand Anodyne RBP4 19 40 COc1cc(Br)ccc1NC(=O)N1CCN(CC(C)(C)O)CC1 ZINC000880631226 GE On-Demand Anodyne PDGFRB 26 40 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCN(C(C)C)C1=O ZINC000880631235 FF On-Demand Anodyne XIAP 42 34 COc1cc(Br)ccc1NC(=O)N[C@H]1CCN(C(C)C)C1=O ZINC000880631236 FF On-Demand Anodyne XIAP 42 34 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1(C)C ZINC000880631237 EF On-Demand Anodyne PDGFRB 28 44 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1(C)C ZINC000880631237 EF On-Demand Anodyne FAAH 20 40 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1(C)C ZINC000880631237 EF On-Demand Anodyne NPY5R 19 41 COc1cc(Br)ccc1NC(=O)NCCCn1cccn1 ZINC000880631238 FF On-Demand Anodyne QPCT 18 45 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2COC[C@H]2C1 ZINC000880631246 EE On-Demand Anodyne PDGFRB 22 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2COC[C@H]2C1 ZINC000880631246 EE On-Demand Anodyne RBP4 56 38 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2C[C@@]2(O)C1 ZINC000880631248 DD On-Demand Anodyne PDGFRB 23 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2C[C@]2(O)C1 ZINC000880631249 DD On-Demand Anodyne PDGFRB 23 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2C[C@@]2(O)C1 ZINC000880631250 DD On-Demand Anodyne PDGFRB 23 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2C[C@]2(O)C1 ZINC000880631251 DD On-Demand Anodyne PDGFRB 23 41 COc1cc(Br)ccc1NC(=O)N[C@H](C)Cn1cncn1 ZINC000880631256 FE On-Demand Anodyne HIS3 79 39 COc1cc(Br)ccc1NC(=O)N[C@@H](C)Cn1cncn1 ZINC000880631257 FE On-Demand Anodyne HIS3 79 39 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C(C)(C)C)CC1 ZINC000880631260 GG On-Demand Anodyne PDGFRB 21 43 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)C(C)(C)C)CC1 ZINC000880631260 GG On-Demand Anodyne RBP4 25 42 COc1cc(Br)ccc1NC(=O)NCC1CCN(C)CC1 ZINC000880631263 FF On-Demand Anodyne CACNA1I 63 35 COc1cc(Br)ccc1NC(=O)NCC1CCN(C)CC1 ZINC000880631263 FF On-Demand Anodyne ACKR3 59 31 COc1cc(Br)ccc1NC(=O)NCCNC(=O)C1CC1 ZINC000880631273 FE On-Demand Anodyne MTNR1A 33 43 COc1cc(Br)ccc1NC(=O)NCCNC(=O)C1CC1 ZINC000880631273 FE On-Demand Anodyne MTNR1B 29 43 COc1cc(Br)ccc1NC(=O)N1CCC(CCO)CC1 ZINC000880631274 FG On-Demand Anodyne PDGFRB 28 42 COc1cc(Br)ccc1NC(=O)N1CCC(CCO)CC1 ZINC000880631274 FG On-Demand Anodyne PTPN2 19 42 COc1cc(Br)ccc1NC(=O)N1CCC(CCO)CC1 ZINC000880631274 FG On-Demand Anodyne PTPN1 16 42 COc1cc(Br)ccc1NC(=O)N1CCC(CCO)CC1 ZINC000880631274 FG On-Demand Anodyne RBP4 28 42 O=C(NCC[C@@H](O)C(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631276 EE On-Demand Anodyne ADRB1 46 34 O=C(NCC[C@H](O)C(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631277 EE On-Demand Anodyne ADRB1 46 34 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne DRD2 21 46 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne DRD3 21 45 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne HTR4 53 50 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne CCR3 30 41 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne SLC6A5 16 40 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne EPHX2 36 44 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne PDK1 44 31 COc1cc(Br)ccc1NC(=O)NC1CCN(CCO)CC1 ZINC000880631278 FE On-Demand Anodyne MCHR1 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCC2(CC1)COC2 ZINC000880631280 FG On-Demand Anodyne EPHX2 34 42 C=CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631289 FG On-Demand Mild DRD2 15 45 C=CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631289 FG On-Demand Mild EPHX2 31 43 C=CCN1CCC(NC(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631289 FG On-Demand Mild PDK1 43 30 O=C(NC[C@H]1C[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631290 DE On-Demand Anodyne GRIN2B 17 40 CN1CCCC[C@H](N(C)C(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880631291 FF On-Demand Anodyne CPT1A 70 35 CN1CCCC[C@@H](N(C)C(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880631292 FF On-Demand Anodyne CPT1A 70 35 COc1cc(Br)ccc1NC(=O)NCC(=O)NC1CCCC1 ZINC000880631294 FF On-Demand Anodyne EPHX2 19 40 COc1cc(Br)ccc1NC(=O)N(C)C[C@@H]1CCCN(C)C1 ZINC000880631302 FG On-Demand Anodyne ACKR3 64 32 COc1cc(Br)ccc1NC(=O)N(C)C[C@H]1CCCN(C)C1 ZINC000880631303 FG On-Demand Anodyne ACKR3 64 32 COc1cc(Br)ccc1NC(=O)N1CCN(C2CC2)CC1 ZINC000880631305 FF On-Demand Anodyne ADRA1D 18 41 COc1cc(Br)ccc1NC(=O)N1CCN(C2CC2)CC1 ZINC000880631305 FF On-Demand Anodyne ADRA1B 15 41 COc1cc(Br)ccc1NC(=O)N1CCN(C2CC2)CC1 ZINC000880631305 FF On-Demand Anodyne PDGFRB 21 43 COc1cc(Br)ccc1NC(=O)N1CCN(C2CC2)CC1 ZINC000880631305 FF On-Demand Anodyne RBP4 22 42 COc1cc(Br)ccc1NC(=O)N1CCN(C2CC2)CC1 ZINC000880631305 FF On-Demand Anodyne L3MBTL3 41 34 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880631313 EH On-Demand Anodyne PDGFRB 22 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880631313 EH On-Demand Anodyne RBP4 56 38 COc1cc(Br)ccc1NC(=O)NC1CCN(C(C)=O)CC1 ZINC000880631314 FF On-Demand Anodyne DRD2 20 42 COc1cc(Br)ccc1NC(=O)NC1CCN(C(C)=O)CC1 ZINC000880631314 FF On-Demand Anodyne EPHX2 53 51 COc1cc(Br)ccc1NC(=O)N1CCC(NC(C)=O)CC1 ZINC000880631315 FF On-Demand Anodyne EPHX2 23 41 COc1cc(Br)ccc1NC(=O)N1CCC(NC(C)=O)CC1 ZINC000880631315 FF On-Demand Anodyne RBP4 23 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CC2(CSC2)C1 ZINC000880631316 EG On-Demand Anodyne EPHX2 31 44 COc1cc(Br)ccc1NC(=O)NCCCOC(C)C ZINC000880631317 EG On-Demand Anodyne FOLH1 15 49 COc1cc(Br)ccc1NC(=O)N1CCC(c2nc(C)no2)CC1 ZINC000880631319 GH On-Demand Anodyne SMO 40 56 COc1cc(Br)ccc1NC(=O)N1CCC(c2nc(C)no2)CC1 ZINC000880631319 GH On-Demand Anodyne ETHR 55 37 COc1cc(Br)ccc1NC(=O)NC1CCN(C2CC2)CC1 ZINC000880631322 FG On-Demand Anodyne ADRA1D 22 55 COc1cc(Br)ccc1NC(=O)NC1CCN(C2CC2)CC1 ZINC000880631322 FG On-Demand Anodyne ADRA1A 15 55 COc1cc(Br)ccc1NC(=O)NC1CCN(C2CC2)CC1 ZINC000880631322 FG On-Demand Anodyne ADRA1B 17 55 COc1cc(Br)ccc1NC(=O)NC1CCN(C2CC2)CC1 ZINC000880631322 FG On-Demand Anodyne EPHX2 38 44 COc1cc(Br)ccc1NC(=O)NCCCN1C(=O)CCC1=O ZINC000880631349 GE On-Demand Anodyne DRD3 15 41 COc1cc(Br)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880631353 GF On-Demand Anodyne PDGFRB 65 52 COc1cc(Br)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880631353 GF On-Demand Anodyne RBP4 27 48 COc1cc(Br)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880631353 GF On-Demand Anodyne LIMK2 15 43 COc1cc(Br)ccc1NC(=O)NCCNC(C)=O ZINC000880631363 ED On-Demand Anodyne FOLH1 15 52 COc1cc(Br)ccc1NC(=O)NCCNC(C)=O ZINC000880631363 ED On-Demand Anodyne NQO2 57 35 COc1cc(Br)ccc1NC(=O)NCCNC(C)=O ZINC000880631363 ED On-Demand Anodyne MTNR1A 64 41 COc1cc(Br)ccc1NC(=O)NCCNC(C)=O ZINC000880631363 ED On-Demand Anodyne MTNR1B 61 41 CC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631365 EG On-Demand Anodyne PDGFRB 32 45 CC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631365 EG On-Demand Anodyne CPT1A 40 37 CC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631365 EG On-Demand Anodyne FAAH 25 42 CC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631365 EG On-Demand Anodyne NPY5R 22 40 CC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631365 EG On-Demand Anodyne EPHX2 32 40 COCCN(Cc1ccccn1)C(=O)Nc1ccc(Br)cc1OC ZINC000880631366 GH On-Demand Anodyne GRM4 19 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC[C@H](O)CC1 ZINC000880631372 EF On-Demand Anodyne EPHX2 52 47 COc1cc(Br)ccc1NC(=O)N1CCOCC2(CC2)C1 ZINC000880631375 FG On-Demand Anodyne LRRK2 28 42 CCC1(O)CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631388 FG On-Demand Anodyne PDGFRB 25 41 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)CO)CC1 ZINC000880631393 FD On-Demand Anodyne PDGFRB 30 43 COc1cc(Br)ccc1NC(=O)N1CCN(C(=O)CO)CC1 ZINC000880631393 FD On-Demand Anodyne RBP4 20 42 COc1cc(Br)ccc1NC(=O)N[C@H](C)CCN1CCN(C)CC1 ZINC000880631462 GF On-Demand Anodyne DRD3 20 40 COc1cc(Br)ccc1NC(=O)N[C@@H](C)CCN1CCN(C)CC1 ZINC000880631463 GF On-Demand Anodyne DRD3 20 40 COc1cc(Br)ccc1NC(=O)N[C@@H](C)[C@@H]1CN(C)CCO1 ZINC000880631485 FE On-Demand Anodyne GPR35 47 35 COc1cc(Br)ccc1NC(=O)N[C@@H](C)[C@H]1CN(C)CCO1 ZINC000880631486 FE On-Demand Anodyne GPR35 47 35 COc1cc(Br)ccc1NC(=O)N[C@H](C)[C@H]1CN(C)CCO1 ZINC000880631487 FE On-Demand Anodyne GPR35 47 35 COc1cc(Br)ccc1NC(=O)N[C@H](C)[C@@H]1CN(C)CCO1 ZINC000880631488 FE On-Demand Anodyne GPR35 47 35 CNC(=O)CN1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631498 GD On-Demand Anodyne DRD4 20 41 CNC(=O)CN1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631498 GD On-Demand Anodyne PDGFRB 26 40 COc1cc(Br)ccc1NC(=O)N1CCN(CCO)CC1 ZINC000880631502 FD On-Demand Anodyne DRD3 33 42 COc1cc(Br)ccc1NC(=O)N1CCN(CCO)CC1 ZINC000880631502 FD On-Demand Anodyne PDGFRB 40 42 COc1cc(Br)ccc1NC(=O)N1CCN(CCO)CC1 ZINC000880631502 FD On-Demand Anodyne RBP4 19 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1C[C@H](C)O ZINC000880631516 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1C[C@H](C)O ZINC000880631516 FG On-Demand Anodyne ACKR3 69 36 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1C[C@H](C)O ZINC000880631517 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1C[C@H](C)O ZINC000880631517 FG On-Demand Anodyne ACKR3 69 36 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1C[C@@H](C)O ZINC000880631518 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1C[C@@H](C)O ZINC000880631518 FG On-Demand Anodyne ACKR3 69 36 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1C[C@@H](C)O ZINC000880631519 FG On-Demand Anodyne DRD2 28 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1C[C@@H](C)O ZINC000880631519 FG On-Demand Anodyne ACKR3 69 36 COc1cc(Br)ccc1NC(=O)N(C)CCCn1ccnc1 ZINC000880631521 FG On-Demand Anodyne TBXAS1 42 40 COc1cc(Br)ccc1NC(=O)N(C)CCCn1ccnc1 ZINC000880631521 FG On-Demand Anodyne HMOX2 18 41 COc1cc(Br)ccc1NC(=O)N(C)CCCn1ccnc1 ZINC000880631521 FG On-Demand Anodyne QPCT 43 52 COc1cc(Br)ccc1NC(=O)N1[C@H]2CCC[C@H]1CC2 ZINC000880631524 EI On-Demand Anodyne DRD2 25 40 COc1cc(Br)ccc1NC(=O)NNC(=O)C1CCCC1 ZINC000880631542 FF On-Demand Reactive STK17B 43 42 CC[C@@H](O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631562 DE On-Demand Anodyne ADRB1 48 37 CC[C@@H](O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631562 DE On-Demand Anodyne PDS 56 34 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880631563 EE On-Demand Anodyne PDGFRB 30 41 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880631564 EE On-Demand Anodyne PDGFRB 30 41 COC(=O)[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1C ZINC000880631571 FF On-Demand Anodyne PDGFRB 24 40 CO[C@@H](C)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631594 DE On-Demand Anodyne ADRB1 43 33 COC[C@@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)OC ZINC000880631604 EE On-Demand Anodyne ADRB1 44 33 O=C(NC[C@]1(O)C[C@H]2C=C[C@H]1C2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631614 FF On-Demand Anodyne EPHX2 22 43 O=C(NC[C@@]1(O)C[C@H]2C=C[C@H]1C2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631615 FF On-Demand Anodyne EPHX2 22 43 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631629 EF On-Demand Anodyne PDGFRB 25 42 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631629 EF On-Demand Anodyne RBP4 42 36 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631630 EF On-Demand Anodyne PDGFRB 25 42 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631630 EF On-Demand Anodyne RBP4 42 36 O=C1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]2N1 ZINC000880631637 FE On-Demand Anodyne PDGFRB 23 41 O=C1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]2N1 ZINC000880631637 FE On-Demand Anodyne RBP4 48 38 O=C1CC[C@@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]2N1 ZINC000880631638 FE On-Demand Anodyne PDGFRB 23 41 O=C1CC[C@@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]2N1 ZINC000880631638 FE On-Demand Anodyne RBP4 48 38 O=C1CC[C@@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]2N1 ZINC000880631639 FE On-Demand Anodyne PDGFRB 23 41 O=C1CC[C@@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]2N1 ZINC000880631639 FE On-Demand Anodyne RBP4 48 38 O=C1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]2N1 ZINC000880631640 FE On-Demand Anodyne PDGFRB 23 41 O=C1CC[C@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@H]2N1 ZINC000880631640 FE On-Demand Anodyne RBP4 48 38 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631641 FF On-Demand Anodyne HCRTR1 23 42 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631641 FF On-Demand Anodyne CHRNA7 17 41 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631641 FF On-Demand Anodyne CPT1A 108 41 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631641 FF On-Demand Anodyne CPT2 45 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880631649 FF On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880631650 FF On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880631651 FF On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880631652 FF On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880631653 FF On-Demand Anodyne RBP4 58 39 O=C(NCCC1(CO)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631654 EF On-Demand Anodyne ADRB1 41 32 O=C(NCCC1(CO)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631654 EF On-Demand Anodyne NAMPT 20 42 COc1cc(Br)ccc1NC(=O)N1CCC(N2CC=CC2)CC1 ZINC000880631698 GG On-Demand Anodyne L3MBTL3 49 33 COc1cc(Br)ccc1NC(=O)N1CCN(CC(=O)N(C)C)CC1 ZINC000880631702 GD On-Demand Anodyne PDGFRB 23 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CN1CCOCC1 ZINC000880631709 GF On-Demand Anodyne DRD2 25 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1CN1CCOCC1 ZINC000880631709 GF On-Demand Anodyne ACKR3 63 33 COc1cc(Br)ccc1NC(=O)NCC(=O)N1CCOCC1 ZINC000880631727 FD On-Demand Anodyne LRRK2 26 43 CNC(=O)CC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631732 GF On-Demand Anodyne PDGFRB 16 40 CNC(=O)CC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631732 GF On-Demand Anodyne PTPN2 18 40 CNC(=O)CC1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631732 GF On-Demand Anodyne PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CCC(C(F)F)CC1 ZINC000880631741 FH On-Demand Anodyne RBP4 35 42 COC(=O)C1(O)CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880631744 GD On-Demand Anodyne PDGFRB 22 42 CO[C@@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631787 DF On-Demand Anodyne EPHX2 36 43 CCC1(N(C)C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631790 FH On-Demand Anodyne PDGFRB 31 43 CCC1(N(C)C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631790 FH On-Demand Anodyne FAAH 24 41 CCC1(N(C)C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631790 FH On-Demand Anodyne NPY5R 39 43 CCC1(N(C)C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631790 FH On-Demand Anodyne S1PR2 30 47 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880631795 DF On-Demand Anodyne PDGFRB 25 42 CCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631801 EE On-Demand Anodyne PDGFRB 34 46 CCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631801 EE On-Demand Anodyne FAAH 28 43 CCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631801 EE On-Demand Anodyne S1PR2 26 41 CCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631801 EE On-Demand Anodyne EPHX2 18 46 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCN(CCCO)C1 ZINC000880631803 FE On-Demand Anodyne SLC6A1 77 35 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCN(CCCO)C1 ZINC000880631803 FE On-Demand Anodyne LTA4H 29 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCN(CCCO)C1 ZINC000880631803 FE On-Demand Anodyne CCR3 52 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCN(CCCO)C1 ZINC000880631803 FE On-Demand Anodyne EPHX2 39 45 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCN(CCCO)C1 ZINC000880631804 FE On-Demand Anodyne SLC6A1 77 35 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCN(CCCO)C1 ZINC000880631804 FE On-Demand Anodyne LTA4H 29 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCN(CCCO)C1 ZINC000880631804 FE On-Demand Anodyne CCR3 52 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCN(CCCO)C1 ZINC000880631804 FE On-Demand Anodyne EPHX2 39 45 COC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880631807 FF On-Demand Anodyne PDGFRB 25 41 O=C(NCCC1SCCS1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631818 FH On-Demand Anodyne ADRB1 44 34 CC1(CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631823 DE On-Demand Anodyne PDGFRB 28 42 CC1(CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631823 DE On-Demand Anodyne FAAH 23 42 CC1(CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631823 DE On-Demand Anodyne NPY5R 23 41 CC1(CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880631823 DE On-Demand Anodyne S1PR2 25 40 CCOC(=O)CCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631824 EF On-Demand Anodyne LTA4H 33 44 CCC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)COC1 ZINC000880631827 EF On-Demand Anodyne NAMPT 17 42 C[C@H](CCO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631829 DF On-Demand Anodyne TSPO 47 30 C[C@H](CCO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631829 DF On-Demand Anodyne NPY5R 41 51 C[C@@H](CCO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631830 DF On-Demand Anodyne TSPO 47 30 C[C@@H](CCO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631830 DF On-Demand Anodyne NPY5R 41 51 COc1cc(Br)ccc1NC(=O)N1CCn2ncnc2C1 ZINC000880631836 FE On-Demand Anodyne PDGFRB 43 45 COc1cc(Br)ccc1NC(=O)N1CCC(N(C)CCO)CC1 ZINC000880631844 GE On-Demand Anodyne RBP4 25 40 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCC1 ZINC000880631849 EG On-Demand Mild ADRB1 41 32 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCC1 ZINC000880631849 EG On-Demand Mild NAMPT 15 42 COc1cc(Br)ccc1NC(=O)N1CCC(c2cn[nH]c2)CC1 ZINC000880631858 GH On-Demand Anodyne RBP4 27 40 C[C@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880631860 EF On-Demand Anodyne ADRB1 42 32 C[C@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880631860 EF On-Demand Anodyne NPY5R 28 40 C[C@@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880631861 EF On-Demand Anodyne ADRB1 42 32 C[C@@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880631861 EF On-Demand Anodyne NPY5R 28 40 O=C(NCC1(CO)CCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631862 EF On-Demand Anodyne NAMPT 40 47 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)N1CC#N ZINC000880631864 FF On-Demand Mild RBP4 43 36 COc1cc(Br)ccc1NC(=O)N1CCOC[C@@H](C)C1 ZINC000880631865 EF On-Demand Anodyne LRRK2 25 40 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H](C)N1CC#N ZINC000880631866 FF On-Demand Mild RBP4 43 36 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)N1CC#N ZINC000880631867 FF On-Demand Mild RBP4 43 36 O=C(NC[C@H]1CCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631873 DF On-Demand Anodyne TNK2 56 38 COc1cc(Br)ccc1NC(=O)N1CCOC[C@H](C)C1 ZINC000880631888 EF On-Demand Anodyne LRRK2 25 40 C[C@@H](CCO)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631909 EF On-Demand Anodyne ADRB1 43 32 C[C@@H](CCO)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631909 EF On-Demand Anodyne LTA4H 15 42 C[C@H](CCO)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631910 EF On-Demand Anodyne ADRB1 43 32 C[C@H](CCO)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631910 EF On-Demand Anodyne LTA4H 15 42 N#C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C1CC1 ZINC000880631915 FE On-Demand Mild PDGFRB 24 42 N#C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C1CC1 ZINC000880631915 FE On-Demand Mild DPP4 20 40 N#C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C1CC1 ZINC000880631919 FE On-Demand Mild PDGFRB 24 42 N#C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C1CC1 ZINC000880631919 FE On-Demand Mild DPP4 20 40 CO[C@@H](C)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631925 DF On-Demand Anodyne ADRB1 43 32 O=C(NOC1CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631928 DF On-Demand Anodyne CA1 24 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880631933 EF On-Demand Anodyne PDGFRB 22 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880631933 EF On-Demand Anodyne RBP4 47 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880631934 EF On-Demand Anodyne PDGFRB 22 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880631934 EF On-Demand Anodyne RBP4 47 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880631936 EF On-Demand Anodyne PDGFRB 22 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880631936 EF On-Demand Anodyne RBP4 47 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1C[C@H](CO)C1 ZINC000880631939 DE On-Demand Anodyne EPHX2 27 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CC(CO)C1 ZINC000880631941 DE On-Demand Anodyne EPHX2 27 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCOC1 ZINC000880631942 DE On-Demand Anodyne EPHX2 33 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@H](CO)C1 ZINC000880631943 EF On-Demand Anodyne EPHX2 30 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@@H](CO)C1 ZINC000880631945 EF On-Demand Anodyne EPHX2 30 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@H](CO)C1 ZINC000880631946 EF On-Demand Anodyne EPHX2 30 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880631947 EF On-Demand Anodyne EPHX2 30 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCSC1 ZINC000880631948 EG On-Demand Anodyne EPHX2 28 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCSC1 ZINC000880631950 EG On-Demand Anodyne EPHX2 28 41 O=C(NC[C@H]1CCCC[C@@H]1O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631951 EF On-Demand Anodyne NAMPT 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(c2cccnc2)CC1 ZINC000880631953 GI On-Demand Anodyne CHRNA7 29 45 COc1cc(Br)ccc1NC(=O)N1CCC(c2cccnc2)CC1 ZINC000880631953 GI On-Demand Anodyne RBP4 37 42 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880631955 FF On-Demand Anodyne EPHX2 36 58 CN(C)C1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631956 FG On-Demand Anodyne EPHX2 49 46 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880631958 FF On-Demand Anodyne EPHX2 36 58 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1O ZINC000880631964 ED On-Demand Anodyne PDGFRB 30 43 COc1cc(Br)ccc1NC(=O)N1CCC(OCC2CC2)CC1 ZINC000880631966 GH On-Demand Anodyne PDGFRB 23 40 COc1cc(Br)ccc1NC(=O)N1CCC(OCC2CC2)CC1 ZINC000880631966 GH On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(OCC2CC2)CC1 ZINC000880631966 GH On-Demand Anodyne PTPN1 16 40 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)CC(F)F ZINC000880631968 EH On-Demand Anodyne ADRB1 43 32 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)CC(F)F ZINC000880631968 EH On-Demand Anodyne NPY5R 20 40 O=CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631971 ED On-Demand Anodyne PDGFRB 31 47 O=CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631971 ED On-Demand Anodyne FAAH 23 43 O=CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880631971 ED On-Demand Anodyne NPY5R 17 40 CC[C@@H](C)CONC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631980 DG On-Demand Anodyne PDS 52 33 CC[C@H](C)CONC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631981 DG On-Demand Anodyne PDS 52 33 COc1cc(Br)ccc1NC(=O)N1CCC(O)(C(F)(F)F)CC1 ZINC000880631986 GG On-Demand Anodyne PDGFRB 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(O)(C(F)(F)F)CC1 ZINC000880631986 GG On-Demand Anodyne RBP4 42 41 O=C(NCCCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631993 EG On-Demand Anodyne ADRB1 41 32 O=C(NCCCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631993 EG On-Demand Anodyne HRH2 21 40 O=C(NCCCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880631993 EG On-Demand Anodyne NAMPT 15 42 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](C)C1 ZINC000880631997 DG On-Demand Anodyne RBP4 34 40 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H](C)O1 ZINC000880631999 EG On-Demand Anodyne PDGFRB 24 41 COc1cc(Br)ccc1NC(=O)N1CC[C@H](C)C1 ZINC000880632001 DG On-Demand Anodyne RBP4 34 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC[C@H]1O ZINC000880632006 DD On-Demand Anodyne EPHX2 17 40 CC[C@H]1CN(C)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632011 EF On-Demand Anodyne CHRNA7 15 44 COc1cc(Br)ccc1NC(=O)N1CCCC[C@H]1c1cn[nH]c1 ZINC000880632012 GH On-Demand Anodyne ROCK2 40 38 CC[C@@H]1CN(C)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632013 EF On-Demand Anodyne CHRNA7 15 44 CN(C)CC(C)(C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632014 EF On-Demand Anodyne P2RY1 23 42 CN(C)C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1CN(C)C ZINC000880632015 GE On-Demand Anodyne PDGFRB 24 40 COc1cc(Br)ccc1NC(=O)N1CCCC[C@@H]1c1cn[nH]c1 ZINC000880632016 GH On-Demand Anodyne ROCK2 40 38 CNC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632017 ED On-Demand Anodyne PDGFRB 26 41 CNC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632017 ED On-Demand Anodyne LTA4H 15 41 CNC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632017 ED On-Demand Anodyne EPHX2 26 41 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632025 GD On-Demand Anodyne PDGFRB 42 44 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632025 GD On-Demand Anodyne FAAH 23 41 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632026 GD On-Demand Anodyne PDGFRB 42 44 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632026 GD On-Demand Anodyne FAAH 23 41 O=C(NCC1(CF)CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632028 FG On-Demand Anodyne NAMPT 22 40 COC(=O)[C@H]1CSCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632029 GF On-Demand Anodyne PDGFRB 24 40 COC(=O)[C@@H]1CSCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632030 GF On-Demand Anodyne PDGFRB 24 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632031 EE On-Demand Anodyne PDGFRB 26 41 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632031 EE On-Demand Anodyne LTA4H 21 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632031 EE On-Demand Anodyne EPHX2 36 44 CC(=O)N[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632032 EE On-Demand Anodyne PDGFRB 26 41 CC(=O)N[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632032 EE On-Demand Anodyne LTA4H 21 40 CC(=O)N[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632032 EE On-Demand Anodyne EPHX2 36 44 COc1cc(Br)ccc1NC(=O)N1CCC(c2ncc[nH]2)CC1 ZINC000880632060 GH On-Demand Anodyne RBP4 29 40 N#C[C@H]1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632100 DG On-Demand Mild EPHX2 28 41 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880632102 FG On-Demand Anodyne PDGFRB 26 42 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880632102 FG On-Demand Anodyne NPY5R 33 45 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880632102 FG On-Demand Anodyne S1PR2 27 42 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880632103 FG On-Demand Anodyne PDGFRB 26 42 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880632103 FG On-Demand Anodyne NPY5R 33 45 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880632103 FG On-Demand Anodyne S1PR2 27 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@](=O)C1 ZINC000880632104 FF On-Demand Anodyne PDGFRB 23 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@](=O)C1 ZINC000880632105 FF On-Demand Anodyne PDGFRB 23 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@](=O)C1 ZINC000880632106 FF On-Demand Anodyne PDGFRB 23 41 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@](=O)C1 ZINC000880632107 FF On-Demand Anodyne PDGFRB 23 41 Cn1ncc(C2CC2)c1CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632114 FG On-Demand Anodyne NAMPT 27 41 CON(C)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632115 DD On-Demand Anodyne ADRB1 40 31 COC[C@@H]1CCCN1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632117 EE On-Demand Anodyne CPT1A 70 36 COC[C@@H]1CCCN1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632117 EE On-Demand Anodyne CHRNA10 51 39 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632123 FG On-Demand Anodyne EPHX2 30 41 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632124 FG On-Demand Anodyne EPHX2 30 41 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632125 FG On-Demand Anodyne EPHX2 30 41 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632126 FG On-Demand Anodyne EPHX2 30 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2[C@H]3C=C[C@@H](C3)[C@H]2C1 ZINC000880632129 EH On-Demand Anodyne PDGFRB 21 40 N#CC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632130 EG On-Demand Mild PDGFRB 32 42 N#CC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632130 EG On-Demand Mild DPP4 15 41 N#CC[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632131 EG On-Demand Mild PDGFRB 32 42 N#CC[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632131 EG On-Demand Mild DPP4 15 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCOC2)CC1 ZINC000880632132 GF On-Demand Anodyne EPHX2 44 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCOC2)CC1 ZINC000880632132 GF On-Demand Anodyne HPGDS 15 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880632133 GF On-Demand Anodyne EPHX2 44 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880632133 GF On-Demand Anodyne HPGDS 15 42 C[C@H](O)CN(C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880632141 EF On-Demand Anodyne NPY5R 33 40 CN1C[C@@H]2CCCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)[C@@H]2C1 ZINC000880632154 FF On-Demand Anodyne PREP 41 33 CC(C)(CNC(=O)Nc1cnc(Oc2ccccc2)nc1)C(=O)N1CCCC1 ZINC000880632157 GG On-Demand Anodyne CPT1A 47 36 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632159 FE On-Demand Anodyne ADRB1 42 33 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632159 FE On-Demand Anodyne CCR3 22 40 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632159 FE On-Demand Anodyne MTOR 52 37 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632159 FE On-Demand Anodyne NAMPT 22 42 O=C(NCC[C@H]1C[C@H]2CC[C@H]1O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632161 FG On-Demand Anodyne ADRB1 40 31 O=C(NCC[C@@H]1C[C@H]2CC[C@H]1O2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632162 FG On-Demand Anodyne ADRB1 40 31 O=C(NCC1CSC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632164 DF On-Demand Anodyne GRIN2B 19 42 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CO1 ZINC000880632167 DF On-Demand Anodyne EPHX2 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@@H]1N1CC[C@H](O)C1 ZINC000880632169 GE On-Demand Anodyne CHRNA7 20 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@@H]1N1CC[C@@H](O)C1 ZINC000880632170 GE On-Demand Anodyne CHRNA7 20 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)C1=O ZINC000880632171 EF On-Demand Anodyne PDGFRB 23 42 CC(C)(C)N1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632176 FF On-Demand Anodyne CCKBR 42 39 CC(C)(C)N1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632176 FF On-Demand Anodyne EPHX2 28 40 CC(C)(C)N1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632177 FF On-Demand Anodyne CCKBR 42 39 CC(C)(C)N1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632177 FF On-Demand Anodyne EPHX2 28 40 C[C@H](O)CN(CC(F)F)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632179 FF On-Demand Anodyne NPY5R 34 42 C[C@@H]1CCC[C@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632180 EF On-Demand Anodyne KCNA3 40 36 C[C@@H]1CCC[C@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632180 EF On-Demand Anodyne NAMPT 19 40 C[C@H]1CCC[C@@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632182 EF On-Demand Anodyne KCNA3 40 36 C[C@H]1CCC[C@@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632182 EF On-Demand Anodyne NAMPT 19 40 C[C@H]1CCC[C@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632183 EF On-Demand Anodyne KCNA3 40 36 C[C@H]1CCC[C@]1(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632183 EF On-Demand Anodyne NAMPT 19 40 CCN(Cc1ccccn1)C(=O)Nc1ccc(Br)cc1OC ZINC000880632227 FH On-Demand Anodyne GRM4 16 40 COc1cc(Br)ccc1NC(=O)NCCc1cnc(C2CC2)nc1 ZINC000880632233 GG On-Demand Anodyne RAF1 18 41 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCN(C)C1 ZINC000880632234 EF On-Demand Anodyne CACNA1I 61 34 COc1cc(Br)ccc1NC(=O)NC[C@@H]1CCN(C)C1 ZINC000880632234 EF On-Demand Anodyne ACKR3 61 31 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCN(C)C1 ZINC000880632235 EF On-Demand Anodyne CACNA1I 61 34 COc1cc(Br)ccc1NC(=O)NC[C@H]1CCN(C)C1 ZINC000880632235 EF On-Demand Anodyne ACKR3 61 31 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)=O)C[C@@H]1C ZINC000880632246 FF On-Demand Anodyne RBP4 16 40 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)=O)C[C@H]1C ZINC000880632247 FF On-Demand Anodyne RBP4 16 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1Cn1ccnc1C ZINC000880632251 GH On-Demand Anodyne DRD2 23 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@H]1Cn1ccnc1C ZINC000880632251 GH On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1ccnc1C ZINC000880632252 GH On-Demand Anodyne DRD2 23 40 COc1cc(Br)ccc1NC(=O)N1CCC[C@@H]1Cn1ccnc1C ZINC000880632252 GH On-Demand Anodyne ACKR3 63 32 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](NC(=O)NC2CC2)C1 ZINC000880632253 GF On-Demand Anodyne EPHX2 40 45 COc1cc(Br)ccc1NC(=O)N1CC[C@H](NC(=O)NC2CC2)C1 ZINC000880632254 GF On-Demand Anodyne EPHX2 40 45 COC[C@@H]1CCCCN(C(=O)Nc2ccc(Br)cc2OC)C1 ZINC000880632301 FH On-Demand Anodyne PDGFRB 27 40 COC1(CCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1 ZINC000880632412 EG On-Demand Anodyne ADRB1 40 31 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880632416 DH On-Demand Anodyne PDGFRB 25 44 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880632416 DH On-Demand Anodyne RBP4 47 36 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632417 EF On-Demand Anodyne CPT1A 81 38 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632417 EF On-Demand Anodyne PREP 42 34 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632420 EF On-Demand Anodyne CPT1A 81 38 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632420 EF On-Demand Anodyne PREP 42 34 CN1CC[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)C1 ZINC000880632422 FF On-Demand Anodyne PDGFRB 23 41 CN1CC[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)C1 ZINC000880632422 FF On-Demand Anodyne FAAH 15 49 CN1CC[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)C1 ZINC000880632422 FF On-Demand Anodyne NPY5R 27 43 CN1CC[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)C1 ZINC000880632422 FF On-Demand Anodyne S1PR2 26 41 CN1CC[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)C1 ZINC000880632422 FF On-Demand Anodyne EPHX2 39 42 COC[C@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632423 EG On-Demand Anodyne PDGFRB 30 41 COC[C@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632423 EG On-Demand Anodyne FAAH 15 42 COC[C@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632423 EG On-Demand Anodyne NPY5R 28 42 COC[C@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632423 EG On-Demand Anodyne S1PR2 27 42 COC[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632424 EG On-Demand Anodyne PDGFRB 30 41 COC[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632424 EG On-Demand Anodyne FAAH 15 42 COC[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632424 EG On-Demand Anodyne NPY5R 28 42 COC[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632424 EG On-Demand Anodyne S1PR2 27 42 CCN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632427 EE On-Demand Anodyne CCKAR 32 41 CCN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632427 EE On-Demand Anodyne CHRNA7 18 40 CCN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632427 EE On-Demand Anodyne CCKBR 47 41 CCN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632427 EE On-Demand Anodyne EPHX2 28 47 CCN1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632428 EE On-Demand Anodyne CCKAR 32 41 CCN1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632428 EE On-Demand Anodyne CHRNA7 18 40 CCN1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632428 EE On-Demand Anodyne CCKBR 47 41 CCN1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880632428 EE On-Demand Anodyne EPHX2 28 47 CC(C)[C@H]1CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632433 DH On-Demand Anodyne CPT1A 72 36 CN(C)C(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632434 GF On-Demand Anodyne PDGFRB 29 44 CN(C)C(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632434 GF On-Demand Anodyne FAAH 22 40 CN(C)C(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632434 GF On-Demand Anodyne LIMK2 17 45 O=C(NC[C@H](O)C1CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632438 EF On-Demand Anodyne ADRB1 41 32 O=C(NC[C@@H](O)C1CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632439 EF On-Demand Anodyne ADRB1 41 32 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632445 GG On-Demand Anodyne EPHX2 66 55 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632445 GG On-Demand Anodyne CXCR3 15 48 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1C[C@H](O)C1 ZINC000880632447 DD On-Demand Anodyne EPHX2 36 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1C[C@H](O)C1 ZINC000880632448 DD On-Demand Anodyne EPHX2 36 42 COCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632450 ED On-Demand Anodyne PDGFRB 39 44 COCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632450 ED On-Demand Anodyne FAAH 19 41 COCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632450 ED On-Demand Anodyne S1PR2 27 43 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632453 EF On-Demand Anodyne LTA4H 31 44 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632453 EF On-Demand Anodyne CPT1A 42 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632453 EF On-Demand Anodyne CHRNA10 69 44 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632453 EF On-Demand Anodyne ACKR3 68 35 CN(C[C@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632454 EF On-Demand Anodyne LTA4H 31 44 CN(C[C@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632454 EF On-Demand Anodyne CPT1A 42 33 CN(C[C@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632454 EF On-Demand Anodyne CHRNA10 69 44 CN(C[C@H]1CCCN1C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632454 EF On-Demand Anodyne ACKR3 68 35 COC1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632473 GH On-Demand Anodyne PDGFRB 30 43 COC1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632473 GH On-Demand Anodyne NPY5R 33 43 COC1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632473 GH On-Demand Anodyne S1PR2 28 42 COC1(C(F)(F)F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632473 GH On-Demand Anodyne RBP4 45 33 CN(CC(=O)N1CCCC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632477 FE On-Demand Anodyne CPT1A 64 38 C[C@@H](F)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632540 DG On-Demand Anodyne ADRB1 44 33 C[C@@]1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1(F)F ZINC000880632545 EG On-Demand Anodyne NAMPT 19 43 COc1cc(Br)ccc1NC(=O)NC1CCC(C)(O)CC1 ZINC000880632548 FG On-Demand Anodyne EPHX2 26 40 COc1cc(Br)ccc1NC(=O)N1CCC(C)(O)CC1 ZINC000880632552 EF On-Demand Anodyne PDGFRB 21 43 COc1cc(Br)ccc1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880632575 FG On-Demand Anodyne RBP4 23 40 COc1cc(Br)ccc1NC(=O)N[C@@H]1CCCOCC1 ZINC000880632580 EG On-Demand Anodyne EPHX2 17 43 COc1cc(Br)ccc1NC(=O)N[C@H]1CCCOCC1 ZINC000880632582 EG On-Demand Anodyne EPHX2 17 43 O=C(NCCN1CCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632591 EE On-Demand Anodyne HRH2 24 40 O=C(NCCN1CCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632591 EE On-Demand Anodyne TYRO3 19 40 COc1cc(Br)ccc1NC(=O)NCCN1CCNC(=O)C1 ZINC000880632592 FD On-Demand Anodyne DRD3 15 47 O=C(NCC[C@@H]1CCSC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632597 EH On-Demand Anodyne ADRB1 40 32 O=C(NCC[C@H]1CCSC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632599 EH On-Demand Anodyne ADRB1 40 32 COc1cc(Br)ccc1NC(=O)N1CCC(S(C)(=O)=O)CC1 ZINC000880632672 GE On-Demand Anodyne PDGFRB 19 42 COc1cc(Br)ccc1NC(=O)N1CCC(S(C)(=O)=O)CC1 ZINC000880632672 GE On-Demand Anodyne RBP4 33 40 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632673 EF On-Demand Anodyne PDGFRB 34 44 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632673 EF On-Demand Anodyne FAAH 20 41 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632673 EF On-Demand Anodyne RBP4 41 35 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CCC2)CC1 ZINC000880632678 FG On-Demand Anodyne HRH3 31 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CCC2)CC1 ZINC000880632678 FG On-Demand Anodyne CHRNA7 21 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CCC2)CC1 ZINC000880632678 FG On-Demand Anodyne EPHX2 54 50 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CCC2)CC1 ZINC000880632678 FG On-Demand Anodyne CXCR3 17 46 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCC[C@H]1O ZINC000880632681 EF On-Demand Anodyne CPT1A 42 34 C[C@@H](CO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632682 FG On-Demand Anodyne PDGFRB 40 42 C[C@@H](CO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632682 FG On-Demand Anodyne FAAH 23 41 C[C@@H](CO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632682 FG On-Demand Anodyne S1PR2 27 42 C[C@@H](CO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632682 FG On-Demand Anodyne EPHX2 24 41 O=C(NCCOCCF)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632696 DE On-Demand Anodyne ADRB1 47 38 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne CHRM1 15 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne HTR3A 32 42 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne SLC6A3 34 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne HTR4 21 42 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne EPHX2 45 45 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880632703 FG On-Demand Anodyne GLRA1 47 38 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCC1 ZINC000880632704 CF On-Demand Anodyne FAAH 20 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCC1 ZINC000880632704 CF On-Demand Anodyne EPHX2 58 49 N#CC[C@@H]1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632710 EG On-Demand Mild EPHX2 26 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1C[C@H]2CCCCN2C1=O ZINC000880632719 FF On-Demand Anodyne CPT1A 52 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1C[C@@H]2CCCCN2C1=O ZINC000880632720 FF On-Demand Anodyne CPT1A 52 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1C[C@@H]2CCCCN2C1=O ZINC000880632721 FF On-Demand Anodyne CPT1A 52 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1C[C@H]2CCCCN2C1=O ZINC000880632722 FF On-Demand Anodyne CPT1A 52 33 C#C[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632723 DG On-Demand Mild PDGFRB 22 40 C#C[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632723 DG On-Demand Mild CPT1A 43 35 C#C[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632723 DG On-Demand Mild CPT2 40 33 C#C[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632723 DG On-Demand Mild PREP 47 37 C#C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632724 DG On-Demand Mild PDGFRB 22 40 C#C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632724 DG On-Demand Mild CPT1A 43 35 C#C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632724 DG On-Demand Mild CPT2 40 33 C#C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632724 DG On-Demand Mild PREP 47 37 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880632725 DG On-Demand Anodyne EPHX2 36 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1C[C@@H]2C[C@H]2C1 ZINC000880632726 DG On-Demand Anodyne EPHX2 36 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1C[C@H]2C[C@@H]2C1 ZINC000880632727 DG On-Demand Anodyne EPHX2 36 43 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880632731 DE On-Demand Anodyne ADRB1 40 31 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)N(C)C ZINC000880632731 DE On-Demand Anodyne NPY5R 32 41 C#CC[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632736 EH On-Demand Mild PDGFRB 27 43 C#CC[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632736 EH On-Demand Mild CPT1A 53 36 C#CC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632737 EH On-Demand Mild PDGFRB 27 43 C#CC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632737 EH On-Demand Mild CPT1A 53 36 O=C(NCC1(O)CCC(F)(F)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632738 GG On-Demand Anodyne NAMPT 17 43 O=C(NCC[C@@H]1CC1(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632740 EG On-Demand Anodyne ADRB1 40 30 O=C(NCC[C@H]1CC1(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632741 EG On-Demand Anodyne ADRB1 40 30 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632748 GF On-Demand Anodyne PDGFRB 23 40 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632748 GF On-Demand Anodyne EPHX2 20 42 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632749 GF On-Demand Anodyne PDGFRB 23 40 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632749 GF On-Demand Anodyne EPHX2 20 42 CC[C@@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880632753 EG On-Demand Anodyne EPHX2 27 44 CC[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880632754 EG On-Demand Anodyne EPHX2 27 44 CC[C@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880632756 EG On-Demand Anodyne EPHX2 27 44 COC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632763 EF On-Demand Anodyne CHRNA7 23 45 COC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632763 EF On-Demand Anodyne CPT1A 101 37 COC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632763 EF On-Demand Anodyne CPT2 44 36 COC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632763 EF On-Demand Anodyne PREP 52 34 COC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632763 EF On-Demand Anodyne CHRNA10 55 40 O=C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCCCCN1 ZINC000880632769 GG On-Demand Anodyne PDGFRB 24 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@H]1CO ZINC000880632771 EF On-Demand Anodyne CCR3 25 40 COc1cc(Br)ccc1NC(=O)NNC(=O)C1CCC1 ZINC000880632781 EE On-Demand Reactive STK17B 41 39 COC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880632795 FF On-Demand Anodyne PDGFRB 15 41 COC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880632795 FF On-Demand Anodyne RBP4 26 42 COC(=O)C1CCN(C(=O)Nc2ccc(Br)cc2OC)CC1 ZINC000880632795 FF On-Demand Anodyne PTR1 46 35 COc1cc(Br)ccc1NC(=O)N1CCCOCC1 ZINC000880632802 EF On-Demand Anodyne LRRK2 30 45 COc1cc(Br)ccc1NC(=O)NCc1cnn(C)c1C ZINC000880632846 FF On-Demand Anodyne HTR2A 23 44 COc1cc(Br)ccc1NC(=O)N1CCC(CCCO)CC1 ZINC000880632850 FG On-Demand Anodyne PDGFRB 27 40 COc1cc(Br)ccc1NC(=O)N1CCC(CCCO)CC1 ZINC000880632850 FG On-Demand Anodyne PTPN2 19 41 COc1cc(Br)ccc1NC(=O)N1CCC(CCCO)CC1 ZINC000880632850 FG On-Demand Anodyne PTPN1 16 41 COc1cc(Br)ccc1NC(=O)N1CCC(CCCO)CC1 ZINC000880632850 FG On-Demand Anodyne RBP4 25 41 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne HTR1A 15 40 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne DRD2 29 41 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne DRD4 42 32 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne DRD3 35 45 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne HTR4 56 36 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne NPY1R 21 40 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne CCR3 32 41 COc1cc(Br)ccc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880632852 GF On-Demand Anodyne MCHR1 15 41 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CCO)C1 ZINC000880632859 EF On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CCO)C1 ZINC000880632859 EF On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CCO)C1 ZINC000880632860 EF On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CCO)C1 ZINC000880632860 EF On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(OC(C)(C)C)CC1 ZINC000880632866 GI On-Demand Anodyne PDGFRB 16 41 COc1cc(Br)ccc1NC(=O)N1CCC(OC(C)(C)C)CC1 ZINC000880632866 GI On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(OC(C)(C)C)CC1 ZINC000880632866 GI On-Demand Anodyne PTPN1 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(OC(C)(C)C)CC1 ZINC000880632866 GI On-Demand Anodyne RBP4 26 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne DRD4 16 49 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne PDGFRB 38 43 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne PTPN2 19 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne GRM4 20 40 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne PTPN1 16 41 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne RBP4 52 46 COc1cc(Br)ccc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880632888 GI On-Demand Anodyne SMO 22 50 COc1cc(Br)ccc1NC(=O)N1CCCN(C)CC1 ZINC000880632889 EF On-Demand Anodyne PDGFRB 26 42 COc1cc(Br)ccc1NC(=O)N1CCCN(C)CC1 ZINC000880632889 EF On-Demand Anodyne RBP4 20 41 C=CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632904 DH On-Demand Mild PDGFRB 25 41 C=CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632904 DH On-Demand Mild FAAH 17 42 C=CC[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632905 DH On-Demand Mild PDGFRB 25 41 C=CC[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632905 DH On-Demand Mild FAAH 17 42 CCN1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1=O ZINC000880632909 EE On-Demand Anodyne EPHX2 32 45 C[C@@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632911 DG On-Demand Mild PDGFRB 24 40 C[C@@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632911 DG On-Demand Mild NPY5R 27 43 C[C@@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632911 DG On-Demand Mild S1PR2 26 40 C[C@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632912 DG On-Demand Mild PDGFRB 24 40 C[C@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632912 DG On-Demand Mild NPY5R 27 43 C[C@]1(C#N)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880632912 DG On-Demand Mild S1PR2 26 40 COC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632918 FE On-Demand Anodyne PDGFRB 37 43 COC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632918 FE On-Demand Anodyne FAAH 26 44 COC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632918 FE On-Demand Anodyne NPY5R 40 46 COC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632918 FE On-Demand Anodyne S1PR2 29 46 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1 ZINC000880632919 DG On-Demand Mild ADRB1 44 33 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1 ZINC000880632919 DG On-Demand Mild NAMPT 15 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)N1C ZINC000880632920 EF On-Demand Anodyne PDGFRB 24 42 O=C(NCCCCF)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632925 DG On-Demand Anodyne ADRB1 46 36 O=C(NCCCCF)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632925 DG On-Demand Anodyne HRH2 16 40 O=C(NCCCCF)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632925 DG On-Demand Anodyne NAMPT 20 46 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880632927 ED On-Demand Anodyne PDGFRB 49 50 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880632927 ED On-Demand Anodyne FAAH 28 44 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880632927 ED On-Demand Anodyne NPY5R 22 40 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632928 EF On-Demand Anodyne CPT1A 77 37 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632928 EF On-Demand Anodyne PREP 48 33 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632930 EF On-Demand Anodyne CPT1A 77 37 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632930 EF On-Demand Anodyne PREP 48 33 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632931 EF On-Demand Anodyne CPT1A 77 37 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632931 EF On-Demand Anodyne PREP 48 33 C[C@@H](CCCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632938 EF On-Demand Anodyne ADRB1 42 32 C[C@@H](CCCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632938 EF On-Demand Anodyne LTA4H 23 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)C1O ZINC000880632946 EF On-Demand Anodyne PDGFRB 23 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H](C)C1O ZINC000880632947 EF On-Demand Anodyne PDGFRB 23 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)[C@@H]1O ZINC000880632948 EF On-Demand Anodyne PDGFRB 23 42 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632952 FH On-Demand Anodyne PDGFRB 50 45 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632952 FH On-Demand Anodyne CPT1A 61 36 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632952 FH On-Demand Anodyne FAAH 21 43 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632952 FH On-Demand Anodyne DGAT1 15 41 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1=O ZINC000880632967 ED On-Demand Anodyne PDGFRB 37 48 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1=O ZINC000880632967 ED On-Demand Anodyne FAAH 26 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@H]3C=C[C@@H](O3)[C@H]2C1 ZINC000880632970 FF On-Demand Anodyne PDGFRB 21 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@@H](C1)[C@H]1C=C[C@H]2O1 ZINC000880632971 FF On-Demand Anodyne PDGFRB 21 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H]2[C@H]3C=C[C@@H](O3)[C@H]2C1 ZINC000880632972 FF On-Demand Anodyne PDGFRB 21 40 O=C(NOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632980 DF On-Demand Anodyne GRIN2B 20 43 O=C(NCC1CCC(O)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632983 EF On-Demand Anodyne GRIN2B 21 45 CCC1(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632986 CG On-Demand Anodyne EPHX2 17 41 O=C(NCCC1(CO)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632987 EF On-Demand Anodyne ADRB1 40 31 O=C(NCCC1(CO)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632987 EF On-Demand Anodyne NAMPT 21 43 C[C@@H](N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1)C(C)(C)O ZINC000880632988 EF On-Demand Anodyne NPY5R 36 44 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne HRH2 35 40 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne LTA4H 27 42 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne CCR3 52 44 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne CHRNA7 19 41 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne MCHR1 25 51 O=C(NCCN1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632990 ED On-Demand Anodyne HPGDS 15 40 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne HRH2 35 40 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne LTA4H 27 42 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne CCR3 52 44 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne CHRNA7 19 41 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne MCHR1 25 51 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880632991 ED On-Demand Anodyne HPGDS 15 40 CO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880632995 EG On-Demand Anodyne PDGFRB 31 43 COc1cc(Br)ccc1NC(=O)N1CCN(c2cnn(C)c2)CC1 ZINC000880633065 GF On-Demand Anodyne PDGFRB 44 45 COc1cc(Br)ccc1NC(=O)N1CCN(c2cnn(C)c2)CC1 ZINC000880633065 GF On-Demand Anodyne RBP4 22 42 COc1cc(Br)ccc1NC(=O)NNC(=O)OC(C)(C)C ZINC000880633075 FG On-Demand Reactive PAPA1_CARPA 22 40 COc1cc(Br)ccc1NC(=O)NNC(=O)Cn1nc(C)cc1C ZINC000880633081 GE On-Demand Reactive FPR2 15 40 COc1cc(Br)ccc1NC(=O)N1CC[C@H](CN2CCCC2)C1 ZINC000880633082 GG On-Demand Anodyne CCR3 15 47 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](CN2CCCC2)C1 ZINC000880633083 GG On-Demand Anodyne CCR3 15 47 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne HTR1A 19 42 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne DRD2 31 41 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne DRD4 43 32 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne DRD3 39 46 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne HTR4 49 37 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne CCR3 39 41 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne PLD1 52 39 COc1cc(Br)ccc1NC(=O)NCCN1CCC(OC)CC1 ZINC000880633088 GF On-Demand Anodyne PLD2 55 39 O=C(NCC[S@@](=O)CC(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633098 GF On-Demand Anodyne ADRB1 41 31 O=C(NCC[S@](=O)CC(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633100 GF On-Demand Anodyne ADRB1 41 31 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880633109 EE On-Demand Anodyne CCKAR 36 40 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880633109 EE On-Demand Anodyne CCKBR 52 36 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880633109 EE On-Demand Anodyne EPHX2 15 41 COC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633112 FE On-Demand Anodyne PDGFRB 27 41 COC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633112 FE On-Demand Anodyne FAAH 18 44 COC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633112 FE On-Demand Anodyne NPY5R 29 42 COC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633112 FE On-Demand Anodyne S1PR2 27 42 O=C(NOCCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633115 DG On-Demand Anodyne GRIN2B 18 45 C#CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633123 DG On-Demand Mild PDGFRB 26 44 C#CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633123 DG On-Demand Mild FAAH 24 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1CO ZINC000880633128 EF On-Demand Anodyne PDGFRB 25 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1CO ZINC000880633129 EF On-Demand Anodyne PDGFRB 25 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1CO ZINC000880633130 EF On-Demand Anodyne PDGFRB 25 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1CO ZINC000880633132 EF On-Demand Anodyne PDGFRB 25 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@@H]2[C@@H](CO)[C@@H]2C1 ZINC000880633134 ED On-Demand Anodyne PDGFRB 22 40 O=C(NC[C@@H]1C[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633138 DE On-Demand Anodyne GRIN2B 17 40 O=C(NCC1CC(O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633140 DE On-Demand Anodyne GRIN2B 17 40 CO[C@]1(CO)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633141 FE On-Demand Anodyne FAAH 17 41 CO[C@]1(CO)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633141 FE On-Demand Anodyne NPY5R 19 40 CO[C@]1(CO)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633141 FE On-Demand Anodyne EPHX2 30 43 COCCCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633148 EG On-Demand Anodyne LTA4H 25 42 C[C@@H]1C[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633157 CF On-Demand Anodyne EPHX2 21 40 O=C(NCCO[C@@H]1CC1(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633174 FF On-Demand Anodyne ADRB1 40 31 O=C(NCCO[C@H]1CC1(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633176 FF On-Demand Anodyne ADRB1 40 31 CCO[C@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633180 EF On-Demand Anodyne TIMP3 63 33 CCO[C@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633180 EF On-Demand Anodyne EPHX2 41 45 CCO[C@@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633181 EF On-Demand Anodyne TIMP3 63 33 CCO[C@@H]1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633181 EF On-Demand Anodyne EPHX2 41 45 O=C(NC[C@H]1CCC[C@@H]1O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633184 EF On-Demand Anodyne NAMPT 15 40 COc1cc(Br)ccc1NC(=O)N1CCC(CC#N)CC1 ZINC000880633211 FH On-Demand Mild PDGFRB 24 40 COc1cc(Br)ccc1NC(=O)N1CCC(CC#N)CC1 ZINC000880633211 FH On-Demand Mild PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(CC#N)CC1 ZINC000880633211 FH On-Demand Mild PTPN1 16 40 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)(C)C(N)=O)CC1 ZINC000880633215 GD On-Demand Anodyne PDGFRB 18 42 COc1cc(Br)ccc1NC(=O)N1CCN(C(C)(C)C(N)=O)CC1 ZINC000880633215 GD On-Demand Anodyne RBP4 32 43 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CS1 ZINC000880633220 EG On-Demand Anodyne EPHX2 26 41 COc1cc(Br)ccc1NC(=O)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880633224 GH On-Demand Anodyne CCR3 31 45 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633225 FF On-Demand Anodyne RBP4 49 34 COc1cc(Br)ccc1NC(=O)N1CC[C@H](Cc2ccncc2)C1 ZINC000880633228 GH On-Demand Anodyne CCR3 31 45 COc1cc(Br)ccc1NC(=O)N1CCC(CC(=O)N(C)C)CC1 ZINC000880633232 GG On-Demand Anodyne PTPN2 18 40 COc1cc(Br)ccc1NC(=O)N1CCC(CC(=O)N(C)C)CC1 ZINC000880633232 GG On-Demand Anodyne PTPN1 15 40 N#CCC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633264 DF On-Demand Mild PDGFRB 26 41 CC(=O)NCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633267 ED On-Demand Anodyne MTNR1A 38 45 CC(=O)NCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633267 ED On-Demand Anodyne MTNR1B 37 45 N#CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633270 DG On-Demand Mild PDGFRB 28 44 N#CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633270 DG On-Demand Mild FAAH 25 40 COC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633271 EG On-Demand Anodyne CHRNA7 22 44 COC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633271 EG On-Demand Anodyne CPT1A 123 41 COC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633271 EG On-Demand Anodyne CPT2 48 39 COC[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633271 EG On-Demand Anodyne CHRNA10 40 37 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633281 GG On-Demand Anodyne CCR3 23 41 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633281 GG On-Demand Anodyne EPHX2 15 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC[C@@H](O)CC1 ZINC000880633282 EF On-Demand Anodyne EPHX2 52 47 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633285 GG On-Demand Anodyne PDGFRB 26 40 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633285 GG On-Demand Anodyne TIMP3 64 33 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633285 GG On-Demand Anodyne S1PR2 28 43 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633287 GG On-Demand Anodyne PDGFRB 26 40 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633287 GG On-Demand Anodyne TIMP3 64 33 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633287 GG On-Demand Anodyne S1PR2 28 43 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633289 GG On-Demand Anodyne PDGFRB 26 40 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633289 GG On-Demand Anodyne TIMP3 64 33 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633289 GG On-Demand Anodyne S1PR2 28 43 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633292 GG On-Demand Anodyne PDGFRB 26 40 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633292 GG On-Demand Anodyne TIMP3 64 33 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633292 GG On-Demand Anodyne S1PR2 28 43 CN1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880633305 EE On-Demand Anodyne EPHX2 32 44 C[C@H]1[C@H](C)N(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C ZINC000880633306 EF On-Demand Anodyne CHRNA7 20 40 CN1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880633307 EE On-Demand Anodyne EPHX2 32 44 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633310 GG On-Demand Anodyne CCR3 23 41 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633310 GG On-Demand Anodyne EPHX2 15 41 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633313 GG On-Demand Anodyne CCR3 23 41 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633313 GG On-Demand Anodyne EPHX2 15 41 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633314 GG On-Demand Anodyne CCR3 23 41 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(Br)cc1OC ZINC000880633314 GG On-Demand Anodyne EPHX2 15 41 O=C(NCCCN1CCCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633315 FF On-Demand Anodyne HRH2 37 44 O=C(NCCCN1CCCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633315 FF On-Demand Anodyne CCR3 29 42 O=C(NCCCN1CCCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633315 FF On-Demand Anodyne TYRO3 21 43 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C ZINC000880633317 EF On-Demand Anodyne CHRNA7 20 40 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633324 FF On-Demand Anodyne PDGFRB 27 41 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633324 FF On-Demand Anodyne FAAH 17 41 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633324 FF On-Demand Anodyne NPY5R 27 43 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633324 FF On-Demand Anodyne S1PR2 26 41 CC[C@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633329 EF On-Demand Anodyne ADRB1 40 30 COc1cc(Br)ccc1NC(=O)NCCc1ccnn1C ZINC000880633330 FF On-Demand Anodyne HTR2A 26 41 CC[C@@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633332 EF On-Demand Anodyne ADRB1 40 30 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633339 GE On-Demand Anodyne PDGFRB 49 44 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633339 GE On-Demand Anodyne FAAH 23 42 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633339 GE On-Demand Anodyne S1PR2 25 40 CSCC[C@H](NC(=O)Nc1cnc(Oc2ccccc2)nc1)C(=O)N(C)C ZINC000880633340 GF On-Demand Anodyne FPR1 42 42 C[C@H]1C[C@@H](C)CN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633343 DH On-Demand Anodyne PDGFRB 17 40 C[C@H]1C[C@@H](C)N(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633345 DH On-Demand Anodyne PDGFRB 17 40 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880633349 EF On-Demand Anodyne EPHX2 26 42 COCCCOCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633365 FF On-Demand Anodyne LTA4H 20 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne LTA4H 29 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne P2RY1 34 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne CCR3 35 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne CHRNA7 18 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne SLC6A5 30 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne EPHX2 59 49 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne CXCR3 22 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)(F)F)CC1 ZINC000880633367 GG On-Demand Anodyne HPGDS 46 61 O=C(NCC1OCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633369 EE On-Demand Anodyne ADRB1 40 31 O=C(NCC1OCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633369 EE On-Demand Anodyne NAMPT 17 41 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633374 FF On-Demand Anodyne FKBP1A 20 43 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633374 FF On-Demand Anodyne CPT2 40 33 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633374 FF On-Demand Anodyne PREP 62 36 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633376 FF On-Demand Anodyne FKBP1A 20 43 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633376 FF On-Demand Anodyne CPT2 40 33 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633376 FF On-Demand Anodyne PREP 62 36 O=C(NC[C@H](O)C1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633378 DE On-Demand Anodyne ADRB1 43 34 O=C(NC[C@@H](O)C1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633379 DE On-Demand Anodyne ADRB1 43 34 C[C@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633381 DE On-Demand Anodyne ADRB1 41 31 C[C@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633381 DE On-Demand Anodyne LTA4H 16 40 C[C@@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633383 DE On-Demand Anodyne ADRB1 41 31 C[C@@H](CCO)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633383 DE On-Demand Anodyne LTA4H 16 40 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633386 GG On-Demand Anodyne PDGFRB 23 40 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633386 GG On-Demand Anodyne EPHX2 23 41 COCCOC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633387 EE On-Demand Anodyne PDGFRB 32 42 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633388 GG On-Demand Anodyne PDGFRB 23 40 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633388 GG On-Demand Anodyne EPHX2 23 41 CN(CCN1CCOCC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633393 FE On-Demand Anodyne CASR 64 51 CN(CCN1CCOCC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633393 FE On-Demand Anodyne MAP2K1 15 40 CN(CCN1CCOCC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633393 FE On-Demand Anodyne EPHX2 28 50 CN(CCN1CCOCC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633393 FE On-Demand Anodyne HPGDS 20 47 O=C(NCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633400 DE On-Demand Anodyne ADRB1 41 32 O=C(NCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633400 DE On-Demand Anodyne NAMPT 24 45 CC[C@H](C)N(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633419 EF On-Demand Anodyne NPY5R 33 42 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne HRH2 29 41 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne CASR 46 40 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne CCR3 21 40 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne PIK3CA 17 42 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne CHRNA7 20 48 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne HNMT 53 30 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne MTOR 35 42 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne EPHX2 32 51 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne PIK3CG 17 42 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne AURKA 16 43 O=C(NCCN1CCCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633420 FE On-Demand Anodyne HPGDS 24 46 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC(F)(F)C1 ZINC000880633422 EH On-Demand Anodyne EPHX2 39 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC(F)(F)C1 ZINC000880633423 EH On-Demand Anodyne EPHX2 39 41 CC(C)[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880633424 EG On-Demand Anodyne PDGFRB 24 40 CC[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)OC ZINC000880633428 DF On-Demand Anodyne ADRB1 40 31 CC[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)OC ZINC000880633428 DF On-Demand Anodyne PDS 73 39 O=C(NCC1(CO)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633429 EF On-Demand Anodyne NAMPT 38 46 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633430 FF On-Demand Anodyne CHRNA7 28 42 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633430 FF On-Demand Anodyne CPT1A 72 35 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633430 FF On-Demand Anodyne PREP 49 33 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633430 FF On-Demand Anodyne CHRNA10 40 37 COC(=O)C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633432 FF On-Demand Anodyne CHRNA7 28 42 COC(=O)C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633432 FF On-Demand Anodyne CPT1A 72 35 COC(=O)C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633432 FF On-Demand Anodyne PREP 49 33 COC(=O)C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633432 FF On-Demand Anodyne CHRNA10 40 37 O=C(NCCCCN1CCC[C@H]1CO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633434 GF On-Demand Anodyne HRH2 25 40 O=C(NCCCCN1CCC[C@H]1CO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633434 GF On-Demand Anodyne CCR3 40 44 O=C(NCCCCN1CCC[C@@H]1CO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633436 GF On-Demand Anodyne HRH2 25 40 O=C(NCCCCN1CCC[C@@H]1CO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633436 GF On-Demand Anodyne CCR3 40 44 CCOC[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633442 FH On-Demand Anodyne PDGFRB 48 43 COCC1(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633452 DF On-Demand Anodyne EPHX2 25 42 CC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633453 CF On-Demand Anodyne PDGFRB 30 46 CC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633453 CF On-Demand Anodyne FAAH 27 42 CC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633453 CF On-Demand Anodyne NPY5R 22 40 CC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633453 CF On-Demand Anodyne EPHX2 19 40 CC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633453 CF On-Demand Anodyne RBP4 55 37 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C ZINC000880633459 EF On-Demand Anodyne CHRNA7 26 40 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C ZINC000880633459 EF On-Demand Anodyne SLC6A5 32 41 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C ZINC000880633459 EF On-Demand Anodyne EPHX2 49 48 CC[C@@H](O)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633468 DF On-Demand Anodyne ADRB1 49 36 CC[C@@H](O)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633468 DF On-Demand Anodyne PDS 44 33 CC[C@H](O)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633469 DF On-Demand Anodyne ADRB1 49 36 CC[C@H](O)CCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633469 DF On-Demand Anodyne PDS 44 33 CCCN(C)C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633470 FG On-Demand Anodyne LTA4H 21 41 CCCN(C)C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633492 FG On-Demand Anodyne LTA4H 21 41 CCCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633493 EG On-Demand Anodyne INHA 59 37 CCCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633493 EG On-Demand Anodyne TSPO 24 40 CCCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633493 EG On-Demand Anodyne PLA2G4B 40 32 CCCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633493 EG On-Demand Anodyne SOAT1 50 44 C[C@H](O)CN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633496 DE On-Demand Anodyne NPY5R 36 43 O=C(NCC1(O)CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633502 EG On-Demand Anodyne HCN1 49 30 O=C(NCC1(O)CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633502 EG On-Demand Anodyne HCN4 47 30 O=C(NCC1(O)CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633502 EG On-Demand Anodyne NAMPT 22 44 O=C(NCCSCCCO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633532 EF On-Demand Anodyne ADRB1 41 31 Cc1nsc(N2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)n1 ZINC000880633535 GF On-Demand Anodyne PDGFRB 38 49 Cc1nsc(N2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)n1 ZINC000880633535 GF On-Demand Anodyne FAAH 29 57 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880633544 GF On-Demand Anodyne CCR3 33 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880633544 GF On-Demand Anodyne EPHX2 43 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880633544 GF On-Demand Anodyne CXCR3 15 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880633544 GF On-Demand Anodyne HPGDS 20 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880633545 GF On-Demand Anodyne CCR3 33 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880633545 GF On-Demand Anodyne EPHX2 43 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880633545 GF On-Demand Anodyne CXCR3 15 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880633545 GF On-Demand Anodyne HPGDS 20 41 CNC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633549 FF On-Demand Anodyne PDGFRB 34 44 CNC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633549 FF On-Demand Anodyne FAAH 21 44 CCOCCN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633554 FE On-Demand Anodyne PDGFRB 55 47 CCOCCN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633554 FE On-Demand Anodyne FAAH 32 47 CCOCCN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633554 FE On-Demand Anodyne S1PR2 26 40 CN1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633556 EF On-Demand Anodyne GRIN2B 32 40 CN1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633556 EF On-Demand Anodyne CCR3 57 44 CN1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633556 EF On-Demand Anodyne EPHX2 25 41 CN1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633556 EF On-Demand Anodyne CACNA1I 40 34 CN1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633556 EF On-Demand Anodyne DGAT1 15 40 C[C@@]1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880633559 EF On-Demand Anodyne NAMPT 15 40 O=C(NCC1CCSCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633564 EH On-Demand Anodyne GRIN2B 20 42 CN(C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CCCC1 ZINC000880633584 DH On-Demand Anodyne LTA4H 19 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880633585 EF On-Demand Anodyne PDGFRB 24 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880633586 EF On-Demand Anodyne PDGFRB 24 42 CC[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633619 FE On-Demand Anodyne PDGFRB 41 45 CC[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633619 FE On-Demand Anodyne ACOX1 53 41 CC[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633619 FE On-Demand Anodyne FAAH 30 47 CC[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633619 FE On-Demand Anodyne ABCB1 64 51 CC[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633619 FE On-Demand Anodyne S1PR2 30 44 CC[C@@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633620 FE On-Demand Anodyne PDGFRB 41 45 CC[C@@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633620 FE On-Demand Anodyne ACOX1 53 41 CC[C@@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633620 FE On-Demand Anodyne FAAH 30 47 CC[C@@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633620 FE On-Demand Anodyne ABCB1 64 51 CC[C@@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633620 FE On-Demand Anodyne S1PR2 30 44 CN(C)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633628 EE On-Demand Anodyne PDGFRB 27 43 CN(C)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633628 EE On-Demand Anodyne RBP4 48 35 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633630 CG On-Demand Anodyne PDGFRB 29 45 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633630 CG On-Demand Anodyne FAAH 24 41 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633630 CG On-Demand Anodyne EPHX2 29 45 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633630 CG On-Demand Anodyne RBP4 40 34 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633631 CG On-Demand Anodyne PDGFRB 29 45 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633631 CG On-Demand Anodyne FAAH 24 41 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633631 CG On-Demand Anodyne EPHX2 29 45 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633631 CG On-Demand Anodyne RBP4 40 34 COCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633632 ED On-Demand Anodyne ROCK2 18 43 C[C@H]1C(=O)NCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633634 ED On-Demand Anodyne CHRNA7 15 45 CCOC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633655 EG On-Demand Anodyne PDGFRB 36 43 CCOC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633655 EG On-Demand Anodyne CCR3 15 44 CCOC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633655 EG On-Demand Anodyne FAAH 16 41 CCOC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633655 EG On-Demand Anodyne DGAT1 17 40 CSC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCOCC1 ZINC000880633657 FG On-Demand Anodyne NAMPT 18 40 Cn1cc([C@@H]2CCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)cn1 ZINC000880633674 FG On-Demand Anodyne CPT1A 80 36 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne PDGFRB 31 44 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne CCR3 23 45 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne FAAH 24 44 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne S1PR2 25 40 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne EPHX2 30 43 CC[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633679 DH On-Demand Anodyne DGAT1 20 40 O=C(NCCCOC1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633682 FF On-Demand Anodyne EPHX2 16 40 Cn1cc(CN2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)cn1 ZINC000880633685 GE On-Demand Anodyne PDGFRB 46 43 Cn1cc(CN2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)cn1 ZINC000880633685 GE On-Demand Anodyne LTA4H 27 40 Cn1cc(CN2CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)cn1 ZINC000880633685 GE On-Demand Anodyne FAAH 40 55 C[C@H](CCO)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633691 DE On-Demand Anodyne LTA4H 24 40 C[C@H](CCO)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633691 DE On-Demand Anodyne ACACB 24 41 C[C@@H](CCO)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633692 DE On-Demand Anodyne LTA4H 24 40 C[C@@H](CCO)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633692 DE On-Demand Anodyne ACACB 24 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCOCC1 ZINC000880633694 DF On-Demand Anodyne EPHX2 47 46 Cn1nccc1C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633711 GG On-Demand Anodyne PDGFRB 25 42 Cn1nccc1C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633711 GG On-Demand Anodyne LIMK2 19 42 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633713 FE On-Demand Anodyne PDGFRB 26 40 O=C(NCCOC[C@@H]1CCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633715 FF On-Demand Anodyne ADRB1 41 31 O=C(NCCOC[C@H]1CCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633716 FF On-Demand Anodyne ADRB1 41 31 C[C@@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)[S@@](C)=O ZINC000880633730 EF On-Demand Anodyne ADRB1 42 32 C[C@@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)[S@](C)=O ZINC000880633731 EF On-Demand Anodyne ADRB1 42 32 C[C@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)[S@@](C)=O ZINC000880633732 EF On-Demand Anodyne ADRB1 42 32 C[C@H](CCNC(=O)Nc1cnc(Oc2ccccc2)nc1)[S@](C)=O ZINC000880633733 EF On-Demand Anodyne ADRB1 42 32 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1n1ccnc1 ZINC000880633736 GH On-Demand Anodyne PDGFRB 22 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1n1ccnc1 ZINC000880633737 GH On-Demand Anodyne PDGFRB 22 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1n1ccnc1 ZINC000880633738 GH On-Demand Anodyne PDGFRB 22 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1n1ccnc1 ZINC000880633739 GH On-Demand Anodyne PDGFRB 22 40 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880633745 EF On-Demand Anodyne PDGFRB 26 42 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880633745 EF On-Demand Anodyne DGAT1 18 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCC(F)(F)C1 ZINC000880633749 EH On-Demand Anodyne EPHX2 36 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCC(F)(F)C1 ZINC000880633750 EH On-Demand Anodyne EPHX2 36 40 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633759 DH On-Demand Anodyne PDGFRB 27 45 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633759 DH On-Demand Anodyne FAAH 20 44 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633759 DH On-Demand Anodyne NPY5R 39 47 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633759 DH On-Demand Anodyne S1PR2 28 44 CC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633759 DH On-Demand Anodyne EPHX2 41 42 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne PDGFRB 50 46 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne CCR3 17 42 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne CPT1A 59 35 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne FAAH 25 45 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne EPHX2 25 40 COCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633769 EG On-Demand Anodyne DGAT1 18 44 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633770 DG On-Demand Anodyne PDGFRB 26 44 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633770 DG On-Demand Anodyne FAAH 21 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1C ZINC000880633771 DG On-Demand Anodyne PDGFRB 26 44 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1C ZINC000880633771 DG On-Demand Anodyne FAAH 21 40 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633772 DG On-Demand Anodyne PDGFRB 26 44 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633772 DG On-Demand Anodyne FAAH 21 40 O=C(NCC1(O)CCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633776 EF On-Demand Anodyne NAMPT 25 45 CC(C)(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633779 DE On-Demand Anodyne P2RY1 36 41 CC(C)(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633779 DE On-Demand Anodyne RAF1 24 40 CC(C)(O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633779 DE On-Demand Anodyne NAMPT 23 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880633805 GF On-Demand Anodyne CHRNA7 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880633805 GF On-Demand Anodyne SLC18A3 64 38 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880633805 GF On-Demand Anodyne EPHX2 54 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880633806 GF On-Demand Anodyne CHRNA7 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880633806 GF On-Demand Anodyne SLC18A3 64 38 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880633806 GF On-Demand Anodyne EPHX2 54 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880633807 GF On-Demand Anodyne CHRNA7 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880633807 GF On-Demand Anodyne SLC18A3 64 38 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880633807 GF On-Demand Anodyne EPHX2 54 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880633808 GF On-Demand Anodyne CHRNA7 17 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880633808 GF On-Demand Anodyne SLC18A3 64 38 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880633808 GF On-Demand Anodyne EPHX2 54 48 CNC(=O)CCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633809 ED On-Demand Anodyne LTA4H 41 40 CCCCNC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633813 GG On-Demand Anodyne PDGFRB 33 43 CCCCNC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633813 GG On-Demand Anodyne TBK1 70 34 COCCn1cc([C@@H]2OCC[C@H]2NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cn1 ZINC000880633864 GD On-Demand Anodyne PANC 45 31 COCCn1cc([C@@H]2OCC[C@H]2NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cn1 ZINC000880633865 GD On-Demand Anodyne PANC 45 31 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633875 GG On-Demand Anodyne CACNA1H 44 36 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633875 GG On-Demand Anodyne PDGFRB 29 43 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633875 GG On-Demand Anodyne FAAH 26 41 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633875 GG On-Demand Anodyne NPY5R 35 43 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)CC2 ZINC000880633875 GG On-Demand Anodyne S1PR2 27 42 COCCN(CCN(C)C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633877 FE On-Demand Anodyne LTA4H 19 40 COCCN(CCN(C)C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633877 FE On-Demand Anodyne ROCK2 24 43 C=CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633880 DH On-Demand Mild PDGFRB 26 44 C=CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633880 DH On-Demand Mild FAAH 22 40 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633884 GG On-Demand Anodyne EPHX2 24 42 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633884 GG On-Demand Anodyne HCN1 80 43 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633884 GG On-Demand Anodyne HCN4 56 36 N#CCCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633885 DG On-Demand Mild ADRB1 50 38 COCCCOC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633897 FF On-Demand Anodyne PDGFRB 29 41 CCN(CC(C)(C)O)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633899 EF On-Demand Anodyne ROCK2 18 40 C[C@@H](CCN(C)C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633901 EF On-Demand Anodyne ROCK2 15 48 C[C@@H](CCN(C)C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633901 EF On-Demand Anodyne UTS2 65 37 CN(CC(C)(C)O)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633902 DF On-Demand Anodyne ROCK2 20 41 CN(C)C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880633918 FE On-Demand Anodyne PDGFRB 26 41 CCc1nnc2n1CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880633921 FE On-Demand Anodyne PDGFRB 26 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne F2 44 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne FKBP1A 29 44 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne ELANE 50 39 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne TRY1_BOVIN 63 32 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne UL80 46 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne CPT1A 53 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne CPT2 41 34 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633932 EE On-Demand Anodyne PREP 72 37 O=C(NCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633936 FE On-Demand Anodyne HRH2 28 41 O=C(NCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633936 FE On-Demand Anodyne CPT1A 59 36 O=C(NCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633936 FE On-Demand Anodyne PREP 30 41 O=C(NCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633936 FE On-Demand Anodyne PRMT3 26 48 O=C(NCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633936 FE On-Demand Anodyne NAMPT 26 41 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633937 FD On-Demand Anodyne PDGFRB 48 47 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633937 FD On-Demand Anodyne FAAH 31 48 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633937 FD On-Demand Anodyne ABCB1 36 49 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880633937 FD On-Demand Anodyne S1PR2 26 41 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1C ZINC000880633943 FE On-Demand Anodyne PDGFRB 36 42 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1C ZINC000880633943 FE On-Demand Anodyne FAAH 19 41 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633944 FE On-Demand Anodyne PDGFRB 36 42 C[C@H](O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1C ZINC000880633944 FE On-Demand Anodyne FAAH 19 41 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C[C@@H](C)O ZINC000880633946 FE On-Demand Anodyne PDGFRB 36 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1C[C@@H](C)O ZINC000880633946 FE On-Demand Anodyne FAAH 19 41 CN(CCC1CC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633953 DH On-Demand Anodyne GRIN2B 16 40 CN(CCC1CC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880633953 DH On-Demand Anodyne LTA4H 30 40 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633973 FF On-Demand Anodyne PDGFRB 28 42 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633973 FF On-Demand Anodyne CPT1A 47 36 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633973 FF On-Demand Anodyne PREP 45 38 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880633973 FF On-Demand Anodyne EPHX2 16 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633985 GG On-Demand Anodyne CCR3 16 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633985 GG On-Demand Anodyne CPT1A 60 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633985 GG On-Demand Anodyne EPHX2 52 52 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633986 GG On-Demand Anodyne CCR3 16 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633986 GG On-Demand Anodyne CPT1A 60 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880633986 GG On-Demand Anodyne EPHX2 52 52 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634004 EG On-Demand Anodyne PDGFRB 46 44 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634004 EG On-Demand Anodyne CCR3 16 51 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634004 EG On-Demand Anodyne CPT1A 80 37 COC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634004 EG On-Demand Anodyne EPHX2 17 44 CN1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1=O ZINC000880634005 ED On-Demand Anodyne EPHX2 25 43 CN1C[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1=O ZINC000880634006 ED On-Demand Anodyne EPHX2 25 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN(CC(F)(F)F)C1=O ZINC000880634011 GF On-Demand Anodyne EPHX2 36 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN(CC(F)(F)F)C1=O ZINC000880634011 GF On-Demand Anodyne HPGDS 31 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN(CC(F)(F)F)C1=O ZINC000880634012 GF On-Demand Anodyne EPHX2 36 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN(CC(F)(F)F)C1=O ZINC000880634012 GF On-Demand Anodyne HPGDS 31 43 CSCC[C@@H](C)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634013 EH On-Demand Anodyne NPY5R 37 48 CSCC[C@H](C)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634014 EH On-Demand Anodyne NPY5R 37 48 C[C@@H](C[C@@H]1CCOC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634024 EG On-Demand Anodyne ACACB 17 40 C[C@H](C[C@@H]1CCOC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634025 EG On-Demand Anodyne ACACB 17 40 C[C@@H](C[C@H]1CCOC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634026 EG On-Demand Anodyne ACACB 17 40 O=C(NCC[C@@H]1CCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634030 EF On-Demand Anodyne ADRB1 40 30 O=C(NCC[C@H]1CCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634031 EF On-Demand Anodyne ADRB1 40 30 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634039 FE On-Demand Anodyne PDGFRB 27 41 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634039 FE On-Demand Anodyne FAAH 15 41 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634039 FE On-Demand Anodyne NPY5R 29 43 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634039 FE On-Demand Anodyne S1PR2 27 40 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880634041 EG On-Demand Anodyne PDGFRB 26 42 CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634042 EG On-Demand Anodyne PDGFRB 38 46 CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634042 EG On-Demand Anodyne FAAH 27 42 CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634042 EG On-Demand Anodyne NPY5R 39 45 CCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634042 EG On-Demand Anodyne S1PR2 36 56 CCC(=O)N1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634044 FE On-Demand Anodyne CCR3 19 41 CCC(=O)N1CC[C@@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634044 FE On-Demand Anodyne EPHX2 56 67 CCC(=O)N1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634045 FE On-Demand Anodyne CCR3 19 41 CCC(=O)N1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634045 FE On-Demand Anodyne EPHX2 56 67 CC(C)(C)[C@@H](O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634065 EF On-Demand Anodyne ADRB1 43 33 O=C(NCC1(CO)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634075 DE On-Demand Anodyne EPHX2 20 42 O=C(NCC1(CO)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634075 DE On-Demand Anodyne NAMPT 40 48 O=C(NCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634077 EF On-Demand Anodyne ADRB1 42 32 O=C(NCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634077 EF On-Demand Anodyne GRIN2B 18 45 CC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634083 FF On-Demand Anodyne PDGFRB 33 46 CC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634083 FF On-Demand Anodyne FAAH 18 42 CC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634083 FF On-Demand Anodyne NPY5R 25 40 CC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634083 FF On-Demand Anodyne EPHX2 28 40 Cc1nn(C)cc1[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634090 GH On-Demand Anodyne CPT1A 70 37 Cc1nn(C)cc1[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634091 GH On-Demand Anodyne CPT1A 70 37 CCCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634093 FI On-Demand Anodyne PDGFRB 27 41 CCCO[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634095 FI On-Demand Anodyne PDGFRB 27 41 COCCCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634099 EG On-Demand Anodyne ADRB1 41 31 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCC[C@H]1CO ZINC000880634100 EF On-Demand Anodyne CPT1A 69 36 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCSCC1 ZINC000880634101 EG On-Demand Anodyne EPHX2 52 47 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCC[C@@H]1CO ZINC000880634102 EF On-Demand Anodyne CPT1A 69 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCC[C@@H]1CO ZINC000880634104 EF On-Demand Anodyne CPT1A 69 36 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCC[C@H]1CO ZINC000880634106 EF On-Demand Anodyne CPT1A 69 36 CC[C@H](C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634111 CG On-Demand Anodyne ACE2 39 40 COC(=O)CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634132 GG On-Demand Anodyne PDGFRB 39 44 COC(=O)CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634132 GG On-Demand Anodyne FAAH 26 43 COC(=O)CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634132 GG On-Demand Anodyne S1PR2 25 40 COC(=O)CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634132 GG On-Demand Anodyne EPHX2 28 41 COC(=O)CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634132 GG On-Demand Anodyne DGAT1 15 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880634133 GG On-Demand Anodyne CCR3 28 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880634133 GG On-Demand Anodyne CPT1A 50 34 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880634133 GG On-Demand Anodyne EPHX2 42 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880634133 GG On-Demand Anodyne CXCR3 17 47 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880634133 GG On-Demand Anodyne HPGDS 31 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880634135 GG On-Demand Anodyne CCR3 28 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880634135 GG On-Demand Anodyne CPT1A 50 34 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880634135 GG On-Demand Anodyne EPHX2 42 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880634135 GG On-Demand Anodyne CXCR3 17 47 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880634135 GG On-Demand Anodyne HPGDS 31 42 Cn1cccc1[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634140 FH On-Demand Anodyne CPT1A 94 38 Cn1cccc1[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634143 FH On-Demand Anodyne CPT1A 94 38 O=C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1 ZINC000880634144 ED On-Demand Anodyne PDGFRB 26 45 O=C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1 ZINC000880634144 ED On-Demand Anodyne FAAH 24 42 O=C(NC[C@H]1CCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634159 EF On-Demand Anodyne CPT1A 65 37 O=C(NC[C@H]1CCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634159 EF On-Demand Anodyne TNK2 49 36 C[C@@H](O)CCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634166 DF On-Demand Anodyne NPY5R 36 42 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H]1C ZINC000880634182 DH On-Demand Anodyne CPT1A 45 34 C[C@H]1[C@H](C)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634184 DH On-Demand Anodyne CPT1A 45 34 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H]1C ZINC000880634186 DH On-Demand Anodyne CPT1A 45 34 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H]1C ZINC000880634187 DH On-Demand Anodyne CPT1A 45 34 C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634188 DH On-Demand Anodyne PDGFRB 27 43 C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634188 DH On-Demand Anodyne CPT1A 43 36 C[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634188 DH On-Demand Anodyne EPHX2 22 53 CC[C@H](O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634189 EF On-Demand Anodyne ADRB1 47 35 CC[C@@H](O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634191 EF On-Demand Anodyne ADRB1 47 35 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne ADRA1D 22 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne ADRA1A 15 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne ADRA1B 17 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne CHRNA7 27 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne SLC6A5 22 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne EPHX2 52 52 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C2CC2)CC1 ZINC000880634223 FG On-Demand Anodyne CXCR3 18 45 C[C@H](NC(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880634224 CG On-Demand Anodyne ACACB 48 37 C[C@H](NC(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880634224 CG On-Demand Anodyne DGAT1 16 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@@H](O)C1 ZINC000880634225 EF On-Demand Anodyne EPHX2 40 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@H](O)C1 ZINC000880634226 EF On-Demand Anodyne EPHX2 40 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@H](O)C1 ZINC000880634227 EF On-Demand Anodyne EPHX2 40 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@@H](O)C1 ZINC000880634228 EF On-Demand Anodyne EPHX2 40 42 CCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634232 EF On-Demand Anodyne INHA 47 36 CCCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634232 EF On-Demand Anodyne SOAT1 36 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880634238 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880634238 FG On-Demand Anodyne CHRNA7 15 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880634238 FG On-Demand Anodyne EPHX2 39 45 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880634239 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880634239 FG On-Demand Anodyne CHRNA7 15 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880634239 FG On-Demand Anodyne EPHX2 39 45 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880634240 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880634240 FG On-Demand Anodyne CHRNA7 15 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880634240 FG On-Demand Anodyne EPHX2 39 45 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880634241 FG On-Demand Anodyne HRH3 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880634241 FG On-Demand Anodyne CHRNA7 15 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880634241 FG On-Demand Anodyne EPHX2 39 45 CCOCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634248 DF On-Demand Anodyne ADRB1 41 31 CCOCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634248 DF On-Demand Anodyne HRH2 26 42 CCOC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634249 GF On-Demand Anodyne P2RY12 94 46 CCOC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634249 GF On-Demand Anodyne PDGFRB 39 48 CCOC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634249 GF On-Demand Anodyne FAAH 31 46 CCOC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634249 GF On-Demand Anodyne S1PR2 27 43 CCOC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634249 GF On-Demand Anodyne DGAT1 18 40 O=C(NCCOCC(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634250 FF On-Demand Anodyne ADRB1 43 32 C[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634258 DH On-Demand Anodyne CPT1A 116 41 C[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634258 DH On-Demand Anodyne CPT2 46 36 C[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634259 DH On-Demand Anodyne CPT1A 116 41 C[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634259 DH On-Demand Anodyne CPT2 46 36 COCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634290 DE On-Demand Anodyne ADRB1 42 32 COCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634290 DE On-Demand Anodyne HRH2 28 43 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne P2RY12 21 43 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne PDGFRB 30 44 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne CPT1A 56 35 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne FAAH 30 43 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne S1PR2 26 42 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne EPHX2 24 41 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne DGAT1 19 43 CCOC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634300 FG On-Demand Anodyne PTR1 47 34 O=C(NC[C@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634311 FE On-Demand Anodyne ADRB1 42 32 O=C(NC[C@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634311 FE On-Demand Anodyne HRH2 27 43 O=C(NC[C@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634311 FE On-Demand Anodyne ACOX1 47 40 O=C(NC[C@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634311 FE On-Demand Anodyne ABCB1 49 41 O=C(NC[C@@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634312 FE On-Demand Anodyne ADRB1 42 32 O=C(NC[C@@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634312 FE On-Demand Anodyne HRH2 27 43 O=C(NC[C@@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634312 FE On-Demand Anodyne ACOX1 47 40 O=C(NC[C@@H](O)CN1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634312 FE On-Demand Anodyne ABCB1 49 41 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)N1CCOCC1 ZINC000880634314 FE On-Demand Anodyne MTOR 52 37 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)N1CCOCC1 ZINC000880634314 FE On-Demand Anodyne EPHX2 15 42 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)on1 ZINC000880634317 FH On-Demand Anodyne CPT1A 107 45 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634322 FF On-Demand Anodyne F2 18 40 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634322 FF On-Demand Anodyne PDGFRB 30 43 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634322 FF On-Demand Anodyne CCR3 24 47 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634322 FF On-Demand Anodyne EPHX2 17 42 COCCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634334 DF On-Demand Anodyne LTA4H 33 45 C[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)CN1CCN(C)CC1 ZINC000880634347 GE On-Demand Anodyne ACOX1 47 39 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634348 GG On-Demand Anodyne CCR3 62 39 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634348 GG On-Demand Anodyne CACNA1I 42 32 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634348 GG On-Demand Anodyne HPGDS 34 46 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634349 GG On-Demand Anodyne CCR3 62 39 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634349 GG On-Demand Anodyne CACNA1I 42 32 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634349 GG On-Demand Anodyne HPGDS 34 46 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880634356 EF On-Demand Anodyne EPHX2 49 47 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC[C@H](CO)CC1 ZINC000880634359 EF On-Demand Anodyne EPHX2 49 47 C=CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634368 FG On-Demand Mild CCR3 27 42 C=CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634368 FG On-Demand Mild CHRNA7 16 40 C=CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634368 FG On-Demand Mild EPHX2 46 49 C=CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634368 FG On-Demand Mild CXCR3 18 48 C=CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634368 FG On-Demand Mild HPGDS 31 43 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880634374 FG On-Demand Anodyne HTR3A 38 46 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880634374 FG On-Demand Anodyne EPHX2 44 44 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880634374 FG On-Demand Anodyne GLRA1 43 34 CCCN(CC)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634391 DH On-Demand Anodyne INHA 40 33 CCCN(CC)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634391 DH On-Demand Anodyne ROCK2 18 40 CCOCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634398 DE On-Demand Anodyne ADRB1 42 32 O=C1CC2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CN1 ZINC000880634416 FE On-Demand Anodyne PDGFRB 24 43 O=C1CC2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CN1 ZINC000880634416 FE On-Demand Anodyne FAAH 17 43 O=C1CC2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CN1 ZINC000880634416 FE On-Demand Anodyne NPY5R 30 44 O=C1CC2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC2)CN1 ZINC000880634416 FE On-Demand Anodyne S1PR2 27 40 O=C(NCCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634417 EG On-Demand Anodyne ADRB1 42 31 O=C(NCCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634417 EG On-Demand Anodyne HRH2 26 42 O=C(NCCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634417 EG On-Demand Anodyne GRIN2B 17 44 O=C(NCCCOCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634417 EG On-Demand Anodyne CCR3 27 41 CC(C)c1nnc2n1CCN(C(=O)Nc1cnc(Oc3ccccc3)nc1)C2 ZINC000880634422 GG On-Demand Anodyne PDGFRB 26 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CC(=O)N(C2CC2)C1 ZINC000880634426 FE On-Demand Anodyne EPHX2 23 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CC(=O)N(C2CC2)C1 ZINC000880634427 FE On-Demand Anodyne EPHX2 23 42 O=C(NCCCN1CCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634430 FE On-Demand Anodyne HRH2 31 43 O=C(NCCCN1CCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634430 FE On-Demand Anodyne CCR3 27 42 O=C(NCCCN1CCCC1=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634430 FE On-Demand Anodyne TYRO3 22 46 COCCCOC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634431 GG On-Demand Anodyne PDGFRB 42 44 O=C(NCc1cn2c(n1)CCCC2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634434 FG On-Demand Anodyne NAMPT 31 41 C=CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634448 GD On-Demand Mild PDGFRB 29 43 C=CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634448 GD On-Demand Mild LTA4H 21 42 C=CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634448 GD On-Demand Mild FAAH 26 47 C[C@@]1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCOC1 ZINC000880634449 EF On-Demand Anodyne NAMPT 19 40 C[C@H]1C[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634455 CF On-Demand Anodyne EPHX2 21 40 C[C@@H]1C[C@@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634456 CF On-Demand Anodyne EPHX2 21 40 C[S@@](=O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634458 EE On-Demand Anodyne ADRB1 40 31 C[S@@](=O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634458 EE On-Demand Anodyne CCR3 16 40 CC(C)(C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634462 CG On-Demand Anodyne P2RY1 28 42 CC(C)(C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634462 CG On-Demand Anodyne RAF1 25 43 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H](C)C1 ZINC000880634463 FE On-Demand Anodyne PDGFRB 23 41 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H](C)C1 ZINC000880634463 FE On-Demand Anodyne LIMK1 16 40 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H](C)C1 ZINC000880634463 FE On-Demand Anodyne LIMK2 29 41 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H](C)C1 ZINC000880634464 FE On-Demand Anodyne PDGFRB 23 41 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H](C)C1 ZINC000880634464 FE On-Demand Anodyne LIMK1 16 40 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H](C)C1 ZINC000880634464 FE On-Demand Anodyne LIMK2 29 41 CN1CCN(C)[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634466 FD On-Demand Anodyne CHRNA10 40 37 CN1CCN(C)[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634467 FD On-Demand Anodyne CHRNA10 40 37 C[C@@H](CC#N)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634477 DG On-Demand Mild NPY5R 38 49 O=C(NC[C@H]1CCC[C@H]1O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634480 EF On-Demand Anodyne NAMPT 15 40 CC[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634482 DH On-Demand Anodyne FKBP1A 24 40 CC[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634482 DH On-Demand Anodyne CHRNA7 24 44 CC[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634482 DH On-Demand Anodyne CPT1A 87 38 CC[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634482 DH On-Demand Anodyne PREP 64 34 CC[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634482 DH On-Demand Anodyne CHRNA10 48 39 CC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634483 DH On-Demand Anodyne FKBP1A 24 40 CC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634483 DH On-Demand Anodyne CHRNA7 24 44 CC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634483 DH On-Demand Anodyne CPT1A 87 38 CC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634483 DH On-Demand Anodyne PREP 64 34 CC[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634483 DH On-Demand Anodyne CHRNA10 48 39 CCC[C@@H](O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634487 DF On-Demand Anodyne ADRB1 45 34 CCC[C@H](O)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634488 DF On-Demand Anodyne ADRB1 45 34 CNC(=O)[C@@H](C)CN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634497 EE On-Demand Anodyne NPY5R 29 40 CCOC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634498 GG On-Demand Anodyne PDGFRB 27 42 CCOC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634498 GG On-Demand Anodyne FAAH 18 41 CCOC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634498 GG On-Demand Anodyne S1PR2 25 41 CCOC(=O)N(C)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634498 GG On-Demand Anodyne LIMK2 28 43 COC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634502 FF On-Demand Anodyne PDGFRB 38 46 COC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634502 FF On-Demand Anodyne FAAH 34 43 COC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634502 FF On-Demand Anodyne PTR1 48 36 C[C@@H](CCCO)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634505 DF On-Demand Anodyne LTA4H 27 41 CNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634522 FD On-Demand Anodyne PDGFRB 43 46 CNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634522 FD On-Demand Anodyne LTA4H 28 43 CNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634522 FD On-Demand Anodyne FAAH 33 51 CN1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634527 EF On-Demand Anodyne CCR3 66 45 CN1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634527 EF On-Demand Anodyne EPHX2 16 41 CN1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634527 EF On-Demand Anodyne NAMPT 26 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne DRD4 18 51 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne LTA4H 42 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne SIGMAR1 19 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne CCR3 50 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne CHRNA7 36 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne SLC6A5 30 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne EPHX2 61 52 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne CXCR3 21 50 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne MCHR1 29 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CCO)CC1 ZINC000880634529 FD On-Demand Anodyne HPGDS 32 45 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634541 FH On-Demand Anodyne PDGFRB 30 42 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634541 FH On-Demand Anodyne NPY5R 33 43 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634541 FH On-Demand Anodyne S1PR2 27 42 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634541 FH On-Demand Anodyne EPHX2 28 41 O=C(C1CC1)[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880634547 FE On-Demand Anodyne PDGFRB 20 43 O=C(C1CC1)[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880634548 FE On-Demand Anodyne PDGFRB 20 43 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634577 EE On-Demand Anodyne CCR3 38 40 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634577 EE On-Demand Anodyne SLC6A5 17 41 CN1CCC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634577 EE On-Demand Anodyne EPHX2 50 47 COC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634611 EE On-Demand Anodyne PDGFRB 30 43 COC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634611 EE On-Demand Anodyne FAAH 27 40 COC(=O)[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634611 EE On-Demand Anodyne PTR1 45 33 COC(=O)[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634612 EE On-Demand Anodyne PDGFRB 30 43 COC(=O)[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634612 EE On-Demand Anodyne FAAH 27 40 COC(=O)[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634612 EE On-Demand Anodyne PTR1 45 33 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne HTR1A 16 44 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne DRD2 24 47 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne DRD4 29 47 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne LTA4H 48 46 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne HTR7 18 44 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne SIGMAR1 22 44 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne SSTR5 40 37 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne CCR3 46 43 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne CHRNA7 36 41 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne EPHX2 59 51 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne CXCR3 23 47 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne MCHR1 37 44 COCCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634619 FF On-Demand Anodyne HPGDS 33 44 COCC[C@@H](C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634620 DF On-Demand Anodyne ACACB 45 39 COCC[C@@H](C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634620 DF On-Demand Anodyne GCK 28 42 COCC[C@H](C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634621 DF On-Demand Anodyne ACACB 45 39 COCC[C@H](C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634621 DF On-Demand Anodyne GCK 28 42 Cn1cnnc1C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634627 GF On-Demand Anodyne PDGFRB 25 41 CC(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634629 FE On-Demand Anodyne PDGFRB 24 41 CC(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634629 FE On-Demand Anodyne LTA4H 18 42 CC(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634629 FE On-Demand Anodyne CCR3 16 42 CC(=O)N[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634629 FE On-Demand Anodyne EPHX2 21 42 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634630 FE On-Demand Anodyne PDGFRB 24 41 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634630 FE On-Demand Anodyne LTA4H 18 42 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634630 FE On-Demand Anodyne CCR3 16 42 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634630 FE On-Demand Anodyne EPHX2 21 42 CCC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634631 FF On-Demand Anodyne PDGFRB 40 48 CCC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634631 FF On-Demand Anodyne FAAH 28 45 CCC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634631 FF On-Demand Anodyne S1PR2 27 42 CCC(=O)N1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634631 FF On-Demand Anodyne EPHX2 26 48 CN(CC1CC1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634646 CG On-Demand Anodyne LTA4H 27 44 COC1(C)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634689 DF On-Demand Anodyne PDGFRB 28 42 COC1(C)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634689 DF On-Demand Anodyne FAAH 18 41 COC1(C)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634689 DF On-Demand Anodyne NPY5R 20 41 C[C@@]1(CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634711 EF On-Demand Anodyne SLC12A5 40 33 C[C@]1(CO)CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634712 EF On-Demand Anodyne SLC12A5 40 33 O=C(NC[C@H]1CCn2ccnc2C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634713 FF On-Demand Anodyne NAMPT 17 47 O=C(NC[C@@H]1CCn2ccnc2C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634714 FF On-Demand Anodyne NAMPT 17 47 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880634718 DF On-Demand Anodyne PDGFRB 25 42 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1O ZINC000880634720 DE On-Demand Anodyne PDGFRB 23 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1O ZINC000880634721 DE On-Demand Anodyne PDGFRB 23 42 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1O ZINC000880634722 DE On-Demand Anodyne PDGFRB 23 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1O ZINC000880634723 DE On-Demand Anodyne PDGFRB 23 42 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1C ZINC000880634724 EG On-Demand Anodyne PDGFRB 27 41 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1C ZINC000880634724 EG On-Demand Anodyne RBP4 40 34 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1C ZINC000880634725 EG On-Demand Anodyne PDGFRB 27 41 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1C ZINC000880634725 EG On-Demand Anodyne RBP4 40 34 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1C ZINC000880634726 EG On-Demand Anodyne PDGFRB 27 41 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1C ZINC000880634726 EG On-Demand Anodyne RBP4 40 34 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1C ZINC000880634727 EG On-Demand Anodyne PDGFRB 27 41 CO[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1C ZINC000880634727 EG On-Demand Anodyne RBP4 40 34 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCOC1 ZINC000880634728 DF On-Demand Anodyne EPHX2 29 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCOC1 ZINC000880634729 DF On-Demand Anodyne EPHX2 29 41 CO[C@@H](C)CN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634739 DF On-Demand Anodyne TSPO 46 30 CO[C@@H](C)CN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634739 DF On-Demand Anodyne NPY5R 33 42 N#CCC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634740 DG On-Demand Mild ADRB1 41 32 CC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634745 EF On-Demand Anodyne PDGFRB 34 45 CC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634745 EF On-Demand Anodyne FAAH 28 43 CC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634745 EF On-Demand Anodyne NPY5R 41 45 CC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634745 EF On-Demand Anodyne S1PR2 30 47 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634764 FG On-Demand Anodyne NPY5R 34 42 C[C@@H](O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634766 DF On-Demand Anodyne ADRB1 45 34 C[C@@H](O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634766 DF On-Demand Anodyne LTA4H 21 41 CCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634768 DE On-Demand Anodyne PDGFRB 30 44 CCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634768 DE On-Demand Anodyne FAAH 23 42 CCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634768 DE On-Demand Anodyne NPY5R 21 40 CCC1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634768 DE On-Demand Anodyne S1PR2 29 46 O=C(NCC1(N2CCOCC2)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634770 FE On-Demand Anodyne MTOR 40 38 O=C(NCC1(N2CCOCC2)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634770 FE On-Demand Anodyne EPHX2 26 45 O=C(NCC1(N2CCOCC2)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634770 FE On-Demand Anodyne HCN1 79 40 O=C(NCC1(N2CCOCC2)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634770 FE On-Demand Anodyne HCN4 54 35 O=C(NCC1(N2CCOCC2)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634770 FE On-Demand Anodyne NAMPT 24 40 O=C(NCc1cnc2n1CCCC2)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634794 FG On-Demand Anodyne NAMPT 29 41 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne DRD4 20 51 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne CHRM3 24 41 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne LTA4H 37 41 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne SIGMAR1 17 47 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne SSTR5 46 37 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne CCR3 39 44 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne CHRNA7 24 41 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne SLC6A5 29 42 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne EPHX2 63 57 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne CXCR3 23 50 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne MCHR1 31 41 CCN1CCC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634803 EF On-Demand Anodyne HPGDS 33 45 CN(C)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634804 FF On-Demand Anodyne PDGFRB 29 44 CN(C)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634804 FF On-Demand Anodyne FAAH 20 40 CN(C)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634804 FF On-Demand Anodyne LIMK2 15 43 COCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634819 FD On-Demand Anodyne PDGFRB 49 47 COCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634819 FD On-Demand Anodyne CPT1A 74 37 COCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634819 FD On-Demand Anodyne FAAH 32 45 COCC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634819 FD On-Demand Anodyne S1PR2 26 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCC2(CC1)OCCO2 ZINC000880634823 FG On-Demand Anodyne EPHX2 34 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne DRD4 18 51 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne CHRM3 18 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne LTA4H 31 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne SIGMAR1 27 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne CCR3 61 44 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne CHRNA7 20 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne EPHX2 58 52 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne CXCR3 22 50 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne MCHR1 25 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC2CC2)CC1 ZINC000880634827 FG On-Demand Anodyne HPGDS 32 45 CCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634841 EG On-Demand Anodyne PDGFRB 26 40 CCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634841 EG On-Demand Anodyne TIMP3 69 33 CCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634841 EG On-Demand Anodyne EPHX2 22 41 CC(=O)NCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634843 FF On-Demand Anodyne PDGFRB 35 45 CC(=O)NCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634843 FF On-Demand Anodyne GRIN2B 44 39 CC(=O)NCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634843 FF On-Demand Anodyne CCR3 22 40 CC(=O)NCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634843 FF On-Demand Anodyne FAAH 24 45 CC(=O)NCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634843 FF On-Demand Anodyne EPHX2 32 40 CN(C[C@@H]1CCCO1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634848 EF On-Demand Anodyne TNK2 41 37 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)O1 ZINC000880634852 EF On-Demand Anodyne PDGFRB 23 42 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)O1 ZINC000880634853 EF On-Demand Anodyne PDGFRB 23 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H](C)O1 ZINC000880634854 EF On-Demand Anodyne PDGFRB 23 42 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne HTR2C 15 43 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne PDGFRB 49 51 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne FAAH 38 47 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne NPY5R 29 42 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne S1PR2 26 42 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880634863 DE On-Demand Anodyne EPHX2 22 43 O=C(NC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1)C1CC1 ZINC000880634898 FE On-Demand Anodyne PDGFRB 21 41 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1O ZINC000880634903 EF On-Demand Anodyne PDGFRB 26 41 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1O ZINC000880634904 EF On-Demand Anodyne PDGFRB 26 41 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCOC1 ZINC000880634908 DE On-Demand Anodyne EPHX2 33 42 COCCO[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634909 FF On-Demand Anodyne PDGFRB 33 43 COCCO[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634909 FF On-Demand Anodyne CPT1A 42 34 COCCO[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634909 FF On-Demand Anodyne EPHX2 26 40 COCCO[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634910 FF On-Demand Anodyne PDGFRB 33 43 COCCO[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634910 FF On-Demand Anodyne CPT1A 42 34 COCCO[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880634910 FF On-Demand Anodyne EPHX2 26 40 CN(C(=O)Nc1cnc(Oc2ccccc2)nc1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880634925 FG On-Demand Anodyne SLC6A3 30 40 CN(C(=O)Nc1cnc(Oc2ccccc2)nc1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880634925 FG On-Demand Anodyne GLRA1 47 39 C[C@H]1C[C@H](O)CN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634926 DE On-Demand Anodyne CFTR 35 40 C[C@@H]1C[C@H](O)CN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634929 DE On-Demand Anodyne CFTR 35 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634932 EH On-Demand Anodyne PDGFRB 23 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634932 EH On-Demand Anodyne NPY5R 27 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634932 EH On-Demand Anodyne S1PR2 27 41 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634933 EH On-Demand Anodyne PDGFRB 23 41 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634933 EH On-Demand Anodyne NPY5R 27 41 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1(F)F ZINC000880634933 EH On-Demand Anodyne S1PR2 27 41 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634934 GE On-Demand Anodyne CCR3 47 39 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634934 GE On-Demand Anodyne EPHX2 23 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H](O)CC(F)(F)C1 ZINC000880634939 FF On-Demand Anodyne PDGFRB 18 40 CCC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880634946 EG On-Demand Anodyne PDGFRB 25 40 CCC[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880634947 EG On-Demand Anodyne PDGFRB 25 40 O=C(NCCCCO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634949 DE On-Demand Anodyne ADRB1 43 32 O=C(NCCCCO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634949 DE On-Demand Anodyne HRH2 17 40 COC[C@H](C)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634967 DF On-Demand Anodyne ADRB1 43 32 COC[C@@H](C)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634968 DF On-Demand Anodyne ADRB1 43 32 O=C(NCC1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634972 EF On-Demand Anodyne GRIN2B 18 42 O=C(NCC1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634972 EF On-Demand Anodyne EPHX2 15 40 O=C(NCC1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634972 EF On-Demand Anodyne NAMPT 16 41 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne HTR1A 28 40 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne HRH2 29 43 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne HTR2A 27 49 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne DRD3 49 40 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne PDGFRB 16 40 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne CASR 51 41 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne TACR2 17 57 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne CCR3 39 49 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne CHRNA7 29 56 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne MTOR 41 36 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne MAP2K1 15 46 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne EPHX2 40 58 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne FLT3 16 42 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne MCHR1 15 56 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne AURKA 17 45 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne HPGDS 22 47 O=C(NCCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634985 FE On-Demand Anodyne NAMPT 27 42 C[C@H](CN1CCOCC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634987 FE On-Demand Anodyne CASR 45 41 C[C@H](CN1CCOCC1)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880634987 FE On-Demand Anodyne EPHX2 25 47 C[C@H](CO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635004 DE On-Demand Anodyne NPY5R 42 53 C[C@@H](CO)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635005 DE On-Demand Anodyne NPY5R 42 53 O=C1C[C@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635013 FE On-Demand Anodyne NPY5R 22 41 O=C1C[C@@]2(CCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635017 FE On-Demand Anodyne NPY5R 22 41 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635024 GF On-Demand Anodyne LIMK2 29 40 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635035 GF On-Demand Anodyne PDGFRB 37 48 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635035 GF On-Demand Anodyne FAAH 27 45 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635035 GF On-Demand Anodyne NPY5R 23 40 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635035 GF On-Demand Anodyne S1PR2 25 40 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635035 GF On-Demand Anodyne EPHX2 23 43 O=C(CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1)NC1CC1 ZINC000880635039 GD On-Demand Anodyne PDGFRB 26 45 O=C(CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1)NC1CC1 ZINC000880635039 GD On-Demand Anodyne FAAH 30 46 O=C(CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1)NC1CC1 ZINC000880635039 GD On-Demand Anodyne EPHX2 26 40 CCN(CC)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635048 GG On-Demand Anodyne PDGFRB 29 42 CCN(CC)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635048 GG On-Demand Anodyne FAAH 20 40 CCN(CC)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635048 GG On-Demand Anodyne S1PR2 25 40 CCN(CC)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635048 GG On-Demand Anodyne EPHX2 19 40 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CC(C)(C)O ZINC000880635064 GF On-Demand Anodyne PDGFRB 27 43 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CC(C)(C)O ZINC000880635067 GF On-Demand Anodyne PDGFRB 27 43 CN(C(=O)Nc1cnc(Oc2ccccc2)nc1)C(C1CC1)C1CC1 ZINC000880635073 EH On-Demand Anodyne NPY5R 34 42 CN(C)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635085 FG On-Demand Anodyne PDGFRB 27 43 CN(C)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635085 FG On-Demand Anodyne LTA4H 16 40 CN(C)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635085 FG On-Demand Anodyne EPHX2 26 40 CN(C)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635085 FG On-Demand Anodyne WNT3 40 31 CCCN(CCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635113 DF On-Demand Anodyne ROCK2 15 42 COCCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635117 DF On-Demand Anodyne ADRB1 42 31 COCCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635117 DF On-Demand Anodyne HRH2 25 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880635132 GF On-Demand Anodyne PDGFRB 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880635132 GF On-Demand Anodyne CHRNA7 17 42 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880635132 GF On-Demand Anodyne EPHX2 67 61 CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635137 GD On-Demand Anodyne PDGFRB 36 44 CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635137 GD On-Demand Anodyne LTA4H 22 42 CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635137 GD On-Demand Anodyne FAAH 30 49 CCNC(=O)CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635137 GD On-Demand Anodyne S1PR2 26 40 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne DRD4 43 34 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne HRH2 21 40 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne CASR 49 42 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne CCR3 25 41 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne PIK3CA 24 40 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne CHRNA7 21 51 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne MTOR 52 40 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne MAP2K1 15 51 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne EPHX2 36 54 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne PIK3CG 22 40 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne AURKA 18 43 O=C(NCCN1CCOCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635138 ED On-Demand Anodyne HPGDS 25 48 COCCN(CCOC)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635144 EE On-Demand Anodyne LTA4H 27 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne DRD4 15 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne SIGMAR1 15 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne CCR3 53 46 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne CHRNA7 18 40 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne EPHX2 60 54 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne CXCR3 21 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(CC(F)F)CC1 ZINC000880635146 GG On-Demand Anodyne HPGDS 34 45 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne P2RY12 20 42 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne PDGFRB 32 45 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne CPT1A 41 34 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne FAAH 21 43 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne S1PR2 25 41 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne EPHX2 22 42 CCOC(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635165 GG On-Demand Anodyne DGAT1 24 44 O=C(NCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635175 CF On-Demand Anodyne GRIN2B 25 48 O=C(NCC1CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635175 CF On-Demand Anodyne NAMPT 26 44 C[C@@H](C1CC1)N(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635179 DH On-Demand Anodyne NPY5R 36 43 CCOCCCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635204 EG On-Demand Anodyne ADRB1 40 30 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635218 ED On-Demand Anodyne PDGFRB 44 52 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635218 ED On-Demand Anodyne FAAH 36 47 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635218 ED On-Demand Anodyne NPY5R 32 43 CC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635218 ED On-Demand Anodyne S1PR2 26 42 CCN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635248 EF On-Demand Anodyne HTR4 54 36 CCN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635248 EF On-Demand Anodyne CCR3 71 43 CCN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635248 EF On-Demand Anodyne CACNA1I 53 33 CCN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635248 EF On-Demand Anodyne NAMPT 27 40 CN(C)C(=O)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635254 EE On-Demand Anodyne ADRB1 41 31 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635261 GG On-Demand Anodyne CPT1A 44 34 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635261 GG On-Demand Anodyne TBK1 46 32 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635262 GG On-Demand Anodyne CPT1A 44 34 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635262 GG On-Demand Anodyne TBK1 46 32 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635287 GG On-Demand Anodyne F2 15 40 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635287 GG On-Demand Anodyne PDGFRB 27 41 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635287 GG On-Demand Anodyne CPT1A 44 33 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635288 GG On-Demand Anodyne F2 15 40 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635288 GG On-Demand Anodyne PDGFRB 27 41 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635288 GG On-Demand Anodyne CPT1A 44 33 CN(C[C@@H]1CCCCO1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635291 EG On-Demand Anodyne CPT1A 55 35 CN(C[C@H]1CCCCO1)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635292 EG On-Demand Anodyne CPT1A 55 35 O=C(NCCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635293 EF On-Demand Anodyne ADRB1 42 32 O=C(NCCC1(O)CCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635293 EF On-Demand Anodyne NAMPT 19 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@H]1CCO ZINC000880635297 EF On-Demand Anodyne CPT1A 45 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCC[C@@H]1CCO ZINC000880635298 EF On-Demand Anodyne CPT1A 45 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@@H]1CCO ZINC000880635299 EF On-Demand Anodyne CPT1A 45 33 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCC[C@H]1CCO ZINC000880635300 EF On-Demand Anodyne CPT1A 45 33 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635301 DF On-Demand Mild ADRB1 43 32 N#CC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635301 DF On-Demand Mild NAMPT 17 43 O=C(NCCCCCO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635303 DF On-Demand Anodyne ADRB1 43 32 CN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880635318 ED On-Demand Anodyne CCKBR 53 37 CN1CC[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C1=O ZINC000880635318 ED On-Demand Anodyne EPHX2 30 42 O=C1C[C@@H]([C@@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635324 GF On-Demand Anodyne CHRNA7 22 40 O=C1C[C@@H]([C@@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635324 GF On-Demand Anodyne CPT1A 109 35 O=C1C[C@@H]([C@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635325 GF On-Demand Anodyne CHRNA7 22 40 O=C1C[C@@H]([C@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635325 GF On-Demand Anodyne CPT1A 109 35 O=C1C[C@H]([C@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635326 GF On-Demand Anodyne CHRNA7 22 40 O=C1C[C@H]([C@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635326 GF On-Demand Anodyne CPT1A 109 35 O=C1C[C@H]([C@@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635327 GF On-Demand Anodyne CHRNA7 22 40 O=C1C[C@H]([C@@H]2CCCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)CN1 ZINC000880635327 GF On-Demand Anodyne CPT1A 109 35 CCC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635328 FG On-Demand Anodyne FAAH 19 43 CCC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635328 FG On-Demand Anodyne NPY5R 30 42 CCC[C@]1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635328 FG On-Demand Anodyne S1PR2 28 43 O=C(NCCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635336 FF On-Demand Anodyne HRH2 34 44 O=C(NCCC(=O)N1CCCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635336 FF On-Demand Anodyne CPT1A 54 35 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCSC1 ZINC000880635343 DF On-Demand Anodyne EPHX2 31 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCSC1 ZINC000880635344 DF On-Demand Anodyne EPHX2 31 42 CN(C)C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635345 EF On-Demand Anodyne PDGFRB 28 43 CN(C)C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635345 EF On-Demand Anodyne CCR3 17 44 CN(C)C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635345 EF On-Demand Anodyne FAAH 17 42 C[C@@H]1CN(CCCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635349 GF On-Demand Anodyne HRH2 42 41 C[C@@H]1CN(CCCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635349 GF On-Demand Anodyne NPY1R 18 40 C[C@@H]1CN(CCCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635349 GF On-Demand Anodyne CCR3 45 49 C[C@@H]1CN(CCCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635349 GF On-Demand Anodyne CHRNA7 17 46 C[C@@H]1CN(CCCNC(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635349 GF On-Demand Anodyne EPHX2 22 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1CCCOCC1 ZINC000880635353 EF On-Demand Anodyne EPHX2 36 44 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCOCC1 ZINC000880635354 EF On-Demand Anodyne EPHX2 36 44 C[C@@H]1CCOCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635355 EF On-Demand Anodyne CPT1A 44 36 C[C@H]1CCOCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635356 EF On-Demand Anodyne CPT1A 44 36 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635359 EG On-Demand Anodyne PDGFRB 33 46 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635359 EG On-Demand Anodyne FAAH 22 40 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635359 EG On-Demand Anodyne NPY5R 35 44 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635359 EG On-Demand Anodyne S1PR2 29 46 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635359 EG On-Demand Anodyne EPHX2 32 42 C[C@@]1(C#N)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635361 EG On-Demand Mild NPY5R 17 40 C[C@@]1(C#N)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635361 EG On-Demand Mild EPHX2 30 44 CS[C@H](C)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635367 DG On-Demand Anodyne ADRB1 40 31 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1c1ncc[nH]1 ZINC000880635382 GF On-Demand Anodyne PDGFRB 25 40 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1c1ncc[nH]1 ZINC000880635383 GF On-Demand Anodyne PDGFRB 25 40 O=C(NC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1)C1CC1 ZINC000880635390 GF On-Demand Anodyne PDGFRB 27 47 O=C(NC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1)C1CC1 ZINC000880635390 GF On-Demand Anodyne EPHX2 56 47 O=C(NCCCOC(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635426 EG On-Demand Anodyne ADRB1 44 34 O=C(NCCCOC(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635426 EG On-Demand Anodyne HRH2 22 41 Cc1n[nH]c(C)c1[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635440 GH On-Demand Anodyne CPT1A 98 38 C[C@H]1[C@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635445 FG On-Demand Anodyne UL80 45 40 C[C@H]1[C@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635445 FG On-Demand Anodyne CPT1A 78 35 C[C@@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635446 FG On-Demand Anodyne UL80 45 40 C[C@@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635446 FG On-Demand Anodyne CPT1A 78 35 C[C@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635447 FG On-Demand Anodyne UL80 45 40 C[C@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635447 FG On-Demand Anodyne CPT1A 78 35 CCOCCOC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635449 FF On-Demand Anodyne PDGFRB 23 43 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635450 EG On-Demand Anodyne PDGFRB 26 41 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635450 EG On-Demand Anodyne CPT1A 73 36 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635450 EG On-Demand Anodyne CPT2 40 33 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635450 EG On-Demand Anodyne P2RY14 42 32 CC[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCCO1 ZINC000880635450 EG On-Demand Anodyne DGAT1 20 42 O=C(NCC1(CCO)CC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635454 EF On-Demand Anodyne NAMPT 18 43 COC[C@@H]1CCCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635456 FH On-Demand Anodyne PDGFRB 44 44 COC[C@@H]1CCCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635456 FH On-Demand Anodyne CPT1A 112 40 COC[C@@H]1CCCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635456 FH On-Demand Anodyne CPT2 48 39 COC[C@@H]1CCCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635456 FH On-Demand Anodyne EPHX2 18 41 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H]1CO ZINC000880635457 EF On-Demand Anodyne CPT1A 50 35 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H]1CO ZINC000880635458 EF On-Demand Anodyne CPT1A 50 35 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@@H]1CO ZINC000880635459 EF On-Demand Anodyne CPT1A 50 35 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)[C@H]1CO ZINC000880635460 EF On-Demand Anodyne CPT1A 50 35 C#CCNC(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635461 GE On-Demand Mild PDGFRB 28 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H](F)C[C@@H]1CO ZINC000880635468 EE On-Demand Anodyne ITGA4 42 37 O=C(Nc1cnc(Oc2ccccc2)nc1)N1C[C@H](F)C[C@H]1CO ZINC000880635470 EE On-Demand Anodyne ITGA4 42 37 CO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635471 EF On-Demand Anodyne PDGFRB 27 41 CO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635471 EF On-Demand Anodyne EPHX2 22 43 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CC(F)(F)C1 ZINC000880635473 DG On-Demand Anodyne EPHX2 37 41 O=C(NC[C@@H]1CCc2nccn2C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635483 FF On-Demand Anodyne NAMPT 16 66 O=C(NC[C@H]1CCc2nccn2C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635484 FF On-Demand Anodyne NAMPT 16 66 C[C@@H](O)C(C)(C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635488 DF On-Demand Anodyne P2RY1 33 41 C[C@@H](O)C(C)(C)NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635488 DF On-Demand Anodyne RAF1 18 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCC(F)(F)CC1 ZINC000880635491 EH On-Demand Anodyne EPHX2 54 45 CC[C@]1(C)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCO1 ZINC000880635494 EG On-Demand Anodyne FAAH 15 40 O=C(NCC1CC(F)(F)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635502 EG On-Demand Anodyne NAMPT 16 42 CC(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635503 FF On-Demand Anodyne PDGFRB 31 45 CC(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635503 FF On-Demand Anodyne FAAH 23 41 CC(=O)OC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635503 FF On-Demand Anodyne EPHX2 31 40 CN1C(=O)N[C@@H]2CN(C(=O)Nc3cnc(Oc4ccccc4)nc3)CC[C@@H]21 ZINC000880635506 FD On-Demand Anodyne PDGFRB 24 42 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635512 GG On-Demand Anodyne PDGFRB 25 40 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635512 GG On-Demand Anodyne FAAH 15 40 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635512 GG On-Demand Anodyne S1PR2 25 40 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635513 GG On-Demand Anodyne PDGFRB 25 40 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635513 GG On-Demand Anodyne FAAH 15 40 CCC1(CC)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635513 GG On-Demand Anodyne S1PR2 25 40 CN(C)C(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635572 GF On-Demand Anodyne PDGFRB 35 44 CN(C)C(=O)CC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635572 GF On-Demand Anodyne FAAH 22 44 CCCCN(CCCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635573 EG On-Demand Anodyne INHA 47 36 CCCCN(CCCO)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635573 EG On-Demand Anodyne SOAT1 38 41 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1c1nccn1C ZINC000880635574 GF On-Demand Anodyne PDGFRB 25 41 CN1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1c1nccn1C ZINC000880635575 GF On-Demand Anodyne PDGFRB 25 41 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880635580 EF On-Demand Anodyne PDGFRB 26 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1=O ZINC000880635581 EF On-Demand Anodyne PDGFRB 26 42 COCCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635584 FF On-Demand Anodyne PDGFRB 33 42 COCCO[C@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635584 FF On-Demand Anodyne CPT1A 66 35 COCCO[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635585 FF On-Demand Anodyne PDGFRB 33 42 COCCO[C@@H]1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635585 FF On-Demand Anodyne CPT1A 66 35 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635586 FF On-Demand Anodyne PDGFRB 31 45 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635586 FF On-Demand Anodyne FAAH 15 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635586 FF On-Demand Anodyne EPHX2 19 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635586 FF On-Demand Anodyne SCD1 15 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635587 FF On-Demand Anodyne PDGFRB 31 45 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635587 FF On-Demand Anodyne FAAH 15 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635587 FF On-Demand Anodyne EPHX2 19 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@@]1=O ZINC000880635587 FF On-Demand Anodyne SCD1 15 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635588 FF On-Demand Anodyne PDGFRB 31 45 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635588 FF On-Demand Anodyne FAAH 15 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635588 FF On-Demand Anodyne EPHX2 19 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635588 FF On-Demand Anodyne SCD1 15 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635589 FF On-Demand Anodyne PDGFRB 31 45 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635589 FF On-Demand Anodyne FAAH 15 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635589 FF On-Demand Anodyne EPHX2 19 40 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[S@]1=O ZINC000880635589 FF On-Demand Anodyne SCD1 15 40 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635592 GH On-Demand Anodyne CPT1A 121 42 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635592 GH On-Demand Anodyne CPT2 42 33 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635593 GH On-Demand Anodyne CPT1A 121 42 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635593 GH On-Demand Anodyne CPT2 42 33 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635597 GF On-Demand Anodyne PDGFRB 37 48 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635597 GF On-Demand Anodyne FAAH 28 45 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635597 GF On-Demand Anodyne NPY5R 22 40 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635597 GF On-Demand Anodyne S1PR2 25 40 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635597 GF On-Demand Anodyne RBP4 46 34 CN1CC=C(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635600 EF On-Demand Anodyne NAMPT 34 42 CC(C)(C#N)CNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635606 DF On-Demand Mild ADRB1 42 32 CCn1ccnc1[C@H]1CCCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635615 GI On-Demand Anodyne CPT1A 116 43 O=C(NC1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1)C1CCC1 ZINC000880635619 FE On-Demand Anodyne EPHX2 21 40 CN(CCO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635620 FE On-Demand Anodyne PDGFRB 27 42 CN(CCO)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635620 FE On-Demand Anodyne FAAH 21 42 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1CCCC[C@@H]1O ZINC000880635622 EF On-Demand Anodyne CPT1A 42 34 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CCO ZINC000880635632 FD On-Demand Anodyne PDGFRB 27 42 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CCO ZINC000880635632 FD On-Demand Anodyne FAAH 16 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CCO ZINC000880635633 FD On-Demand Anodyne PDGFRB 27 42 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCN1CCO ZINC000880635633 FD On-Demand Anodyne FAAH 16 40 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635650 EF On-Demand Anodyne PDGFRB 28 43 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635650 EF On-Demand Anodyne FAAH 15 42 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635650 EF On-Demand Anodyne NPY5R 27 42 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635650 EF On-Demand Anodyne S1PR2 26 41 C[C@]1(O)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635650 EF On-Demand Anodyne EPHX2 37 47 COC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635659 EG On-Demand Anodyne PDGFRB 35 45 COC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635659 EG On-Demand Anodyne FAAH 23 41 COC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635659 EG On-Demand Anodyne NPY5R 37 45 COC1(C)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635659 EG On-Demand Anodyne S1PR2 28 45 O=C(NCC[C@@H](O)C(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635661 FF On-Demand Anodyne ADRB1 46 36 O=C(NCC[C@H](O)C(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635662 FF On-Demand Anodyne ADRB1 46 36 C[C@H]1C[C@H](NC(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)O1 ZINC000880635673 EG On-Demand Anodyne EPHX2 26 42 C[C@@H]1CC(NC(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H](C)O1 ZINC000880635674 EG On-Demand Anodyne EPHX2 26 42 O=C(NC[C@H]1CCSC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635677 EG On-Demand Anodyne GRIN2B 18 40 O=C(NC[C@@H]1CCSC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635678 EG On-Demand Anodyne GRIN2B 18 40 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635696 EG On-Demand Anodyne PDGFRB 26 40 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635696 EG On-Demand Anodyne NPY5R 23 41 CO[C@@]1(C)CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635696 EG On-Demand Anodyne EPHX2 33 45 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(c2nccs2)CC1 ZINC000880635697 GH On-Demand Anodyne CHRNA7 16 41 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CCN(c2nccs2)CC1 ZINC000880635697 GH On-Demand Anodyne EPHX2 45 48 C[C@@H]1CSCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635701 EG On-Demand Anodyne PDGFRB 24 41 O=C(NCCCC(F)(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635708 EH On-Demand Anodyne ADRB1 42 31 N#CC1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635709 FH On-Demand Mild ADRB1 42 32 N#CC1CCC(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635709 FH On-Demand Mild GRIN2B 21 43 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@@H]1[C@H]2CCC[C@H]21 ZINC000880635717 DG On-Demand Anodyne EPHX2 22 40 O=C(Nc1cnc(Oc2ccccc2)nc1)N[C@H]1[C@H]2CCC[C@H]21 ZINC000880635718 DG On-Demand Anodyne EPHX2 22 40 CON(C)C(=O)C1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635735 GF On-Demand Anodyne PDGFRB 35 44 CC(C)C1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635736 EF On-Demand Anodyne PDGFRB 29 44 CC(C)C1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635736 EF On-Demand Anodyne FAAH 15 40 CC(C)C1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635736 EF On-Demand Anodyne NPY5R 23 40 CC(C)C1(O)CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635736 EF On-Demand Anodyne S1PR2 28 44 COCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635742 FE On-Demand Anodyne PDGFRB 51 46 COCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635742 FE On-Demand Anodyne FAAH 26 42 COCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635742 FE On-Demand Anodyne NPY5R 37 44 COCC1(O)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635742 FE On-Demand Anodyne S1PR2 34 52 O=C(NCC[C@@H]1CCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635761 EG On-Demand Anodyne CPT1A 51 36 O=C(NCC[C@H]1CCCCO1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635762 EG On-Demand Anodyne CPT1A 51 36 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1OC ZINC000880635764 EE On-Demand Anodyne PDGFRB 29 43 CO[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1OC ZINC000880635764 EE On-Demand Anodyne RBP4 48 37 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1F ZINC000880635767 EG On-Demand Anodyne PDGFRB 24 42 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1F ZINC000880635767 EG On-Demand Anodyne RBP4 40 34 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1F ZINC000880635768 EG On-Demand Anodyne PDGFRB 24 42 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1F ZINC000880635768 EG On-Demand Anodyne RBP4 40 34 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1F ZINC000880635769 EG On-Demand Anodyne PDGFRB 24 42 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@H]1F ZINC000880635769 EG On-Demand Anodyne RBP4 40 34 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1F ZINC000880635770 EG On-Demand Anodyne PDGFRB 24 42 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C[C@@H]1F ZINC000880635770 EG On-Demand Anodyne RBP4 40 34 O=C1C[C@H]([C@@H]2CCCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635771 GF On-Demand Anodyne PDGFRB 19 41 O=C1C[C@H]([C@H]2CCCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635772 GF On-Demand Anodyne PDGFRB 19 41 O=C1C[C@@H]([C@@H]2CCCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635773 GF On-Demand Anodyne PDGFRB 19 41 O=C1C[C@@H]([C@H]2CCCN(C(=O)Nc3cnc(Oc4ccccc4)nc3)C2)CN1 ZINC000880635774 GF On-Demand Anodyne PDGFRB 19 41 CCC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635778 FG On-Demand Anodyne PDGFRB 30 43 CCC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635778 FG On-Demand Anodyne FAAH 25 42 CCC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635778 FG On-Demand Anodyne NPY5R 39 44 CCC1(CO)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635778 FG On-Demand Anodyne S1PR2 31 48 CSC1(CNC(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635786 EG On-Demand Anodyne NAMPT 23 44 C[C@@H](CO)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635794 EF On-Demand Anodyne ADRB1 43 33 C[C@@H](CO)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635794 EF On-Demand Anodyne LTA4H 17 40 C[C@H](CO)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635795 EF On-Demand Anodyne ADRB1 43 33 C[C@H](CO)CCCNC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635795 EF On-Demand Anodyne LTA4H 17 40 COCC1(NC(=O)Nc2cnc(Oc3ccccc3)nc2)CCC1 ZINC000880635798 EF On-Demand Anodyne EPHX2 21 41 CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635802 EE On-Demand Anodyne PDGFRB 42 48 CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635802 EE On-Demand Anodyne FAAH 25 44 CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635802 EE On-Demand Anodyne NPY5R 20 40 CN1CCCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635802 EE On-Demand Anodyne EPHX2 19 40 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880635806 EH On-Demand Anodyne PDGFRB 31 43 C[C@@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880635806 EH On-Demand Anodyne FAAH 20 41 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880635807 EH On-Demand Anodyne PDGFRB 31 43 C[C@H]1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CCS1 ZINC000880635807 EH On-Demand Anodyne FAAH 20 41 CC(=O)N(C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880635808 GG On-Demand Anodyne CPT1A 51 35 CC(=O)N(C[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880635808 GG On-Demand Anodyne ACKR3 60 32 CC(=O)N(C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880635809 GG On-Demand Anodyne CPT1A 51 35 CC(=O)N(C[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1)C1CC1 ZINC000880635809 GG On-Demand Anodyne ACKR3 60 32 O=C(NOC1CCCC1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635811 DG On-Demand Anodyne CA1 23 40 COCC1=CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635823 EG On-Demand Anodyne PDGFRB 29 40 O=C(NCCCCCCO)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635835 EF On-Demand Anodyne ADRB1 43 32 Cn1cnnc1[C@@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635841 FF On-Demand Anodyne CPT1A 80 40 Cn1cnnc1[C@H]1CCCN1C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635842 FF On-Demand Anodyne CPT1A 80 40 O=C(NCCOCC(F)F)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635843 EF On-Demand Anodyne ADRB1 47 36 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635844 FF On-Demand Anodyne F2 18 40 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635844 FF On-Demand Anodyne CCR3 61 43 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635844 FF On-Demand Anodyne EPHX2 16 40 CC(=O)N1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635845 FF On-Demand Anodyne F2 18 40 CC(=O)N1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635845 FF On-Demand Anodyne CCR3 61 43 CC(=O)N1CCC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880635845 FF On-Demand Anodyne EPHX2 16 40 O=C(NC[C@H]1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635948 EF On-Demand Anodyne GRIN2B 18 43 O=C(NC[C@H]1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635949 EF On-Demand Anodyne GRIN2B 18 43 O=C(NC[C@@H]1CC[C@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635950 EF On-Demand Anodyne GRIN2B 18 43 O=C(NC[C@@H]1CC[C@@H](O)C1)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635951 EF On-Demand Anodyne GRIN2B 18 43 CNC(=O)CCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880635952 EE On-Demand Anodyne LTA4H 37 43 COC[C@@H](CNC(=O)Nc1cnc(Oc2ccccc2)nc1)OC ZINC000880635976 EE On-Demand Anodyne ADRB1 43 32 N#CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635984 EG On-Demand Mild PDGFRB 34 44 N#CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635984 EG On-Demand Mild FAAH 21 45 N#CCC1CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC1 ZINC000880635984 EG On-Demand Mild EPHX2 20 40 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1O ZINC000880635985 EF On-Demand Anodyne PDGFRB 26 43 C[C@@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1O ZINC000880635986 EF On-Demand Anodyne PDGFRB 26 43 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@H]1O ZINC000880635987 EF On-Demand Anodyne PDGFRB 26 43 C[C@H]1CN(C(=O)Nc2cnc(Oc3ccccc3)nc2)CC[C@@H]1O ZINC000880635988 EF On-Demand Anodyne PDGFRB 26 43 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)no1 ZINC000880635997 FH On-Demand Anodyne CPT1A 122 47 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnc(Oc3ccccc3)nc2)no1 ZINC000880635997 FH On-Demand Anodyne CPT2 40 33 CCOCCN(C)C(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636013 DF On-Demand Anodyne LTA4H 24 40 N#C[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636018 EF On-Demand Mild PDGFRB 22 42 N#C[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636018 EF On-Demand Mild FAAH 15 41 N#C[C@@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636018 EF On-Demand Mild NPY5R 29 43 N#C[C@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636019 EF On-Demand Mild PDGFRB 22 42 N#C[C@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636019 EF On-Demand Mild FAAH 15 41 N#C[C@]1(F)CCN(C(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636019 EF On-Demand Mild NPY5R 29 43 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636021 GG On-Demand Anodyne CCR3 40 39 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636021 GG On-Demand Anodyne EPHX2 32 48 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636022 GG On-Demand Anodyne CCR3 40 39 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636022 GG On-Demand Anodyne EPHX2 32 48 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636023 GG On-Demand Anodyne CCR3 40 39 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636023 GG On-Demand Anodyne EPHX2 32 48 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636024 GG On-Demand Anodyne CCR3 40 39 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnc(Oc2ccccc2)nc1 ZINC000880636024 GG On-Demand Anodyne EPHX2 32 48 O=C(Nc1cnc(Oc2ccccc2)nc1)NC1CC(N2CCCCC2)C1 ZINC000880636028 FG On-Demand Anodyne EPHX2 32 42 CN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636029 EE On-Demand Anodyne CCR3 57 43 CN1CC[C@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636029 EE On-Demand Anodyne NAMPT 34 41 CN1CC[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636030 EE On-Demand Anodyne CCR3 57 43 CN1CC[C@@H](CNC(=O)Nc2cnc(Oc3ccccc3)nc2)C1 ZINC000880636030 EE On-Demand Anodyne NAMPT 34 41 Cc1ccncc1CNC(=O)Nc1cccc2c1OC(C)(C)C=C2 ZINC000880636390 DH On-Demand Anodyne TRPV1 15 40 Cc1ccncc1CNC(=O)Nc1cccc2c1OC(C)(C)C=C2 ZINC000880636390 DH On-Demand Anodyne NAMPT 15 52 CN1CCN(C(=O)Nc2cccc3c2OC(C)(C)C=C3)C[C@H]1c1ncc[nH]1 ZINC000880636805 FG On-Demand Anodyne G2YM83_BOTF4 40 36 CN1CCN(C(=O)Nc2cccc3c2OC(C)(C)C=C3)C[C@@H]1c1ncc[nH]1 ZINC000880636806 FG On-Demand Anodyne G2YM83_BOTF4 40 36 COC(=O)N1CCC(NC(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880637833 FG On-Demand Anodyne EPHX2 39 40 Cn1cc(CNC(=O)Nc2cccc3c2OC(C)(C)C=C3)cn1 ZINC000880637885 DF On-Demand Anodyne NAMPT 27 42 C[C@@H](Cn1cncn1)NC(=O)Nc1cccc2c1OC(C)(C)C=C2 ZINC000880637956 EF On-Demand Anodyne HIS3 66 36 COCCC(=O)N1CCC(NC(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880638054 GG On-Demand Anodyne EPHX2 34 42 COCCC(=O)N1CCC(NC(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880638054 GG On-Demand Anodyne CCR8 48 37 Cc1cncc(CNC(=O)Nc2cccc3c2OC(C)(C)C=C3)c1 ZINC000880638097 DH On-Demand Anodyne NAMPT 30 52 NC(=O)COc1cccc(NC(=O)/C(=C\c2ccc(Cl)cc2)c2ccc(F)cc2)c1 ZINC000880638209 HJ On-Demand Anodyne TAAR1 15 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc2c1OC(C)(C)C=C2 ZINC000880638318 EF On-Demand Anodyne LGMN 42 30 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2csc(C)c2)C1 ZINC000880638427 DG On-Demand Anodyne EPHX2 33 41 Cc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)cs1 ZINC000880638451 CE On-Demand Anodyne CXCR3 20 40 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne CA2 20 47 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne LPL 48 35 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne CA1 54 41 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne CA12 34 47 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne CA9 34 47 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne NCE103 21 47 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne MTCA1 36 47 Cc1cc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cs1 ZINC000880638488 FG On-Demand Anodyne P96878_MYCTU 41 47 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OC(C)(C)C=C3)C1 ZINC000880638781 EG On-Demand Anodyne EPHX2 28 45 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OC(C)(C)C=C3)C1 ZINC000880638781 EG On-Demand Anodyne CCR8 25 40 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OC(C)(C)C=C3)C1 ZINC000880638782 EG On-Demand Anodyne EPHX2 28 45 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OC(C)(C)C=C3)C1 ZINC000880638782 EG On-Demand Anodyne CCR8 25 40 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2csc(C)c2)C1 ZINC000880638835 EG On-Demand Anodyne EPHX2 34 41 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2csc(C)c2)C1 ZINC000880638943 EG On-Demand Anodyne EPHX2 33 44 CCn1nc2c(cc1=O)CN(C(=O)Nc1cccc3c1OC(C)(C)C=C3)CC2 ZINC000880639034 GG On-Demand Anodyne P2RY14 45 34 Cc1cc(NC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)cs1 ZINC000880639062 EG On-Demand Anodyne CACNA1I 48 33 Cc1cc(NC(=O)NCCC(=O)OCc2ccccc2)cs1 ZINC000880639105 DG On-Demand Anodyne NPR 41 33 CCOC(=O)N1CC[C@H](NC(=O)Nc2csc(C)c2)C1 ZINC000880639207 CE On-Demand Anodyne EPHX2 46 45 CCOC(=O)N1CC[C@@H](NC(=O)Nc2csc(C)c2)C1 ZINC000880639209 CE On-Demand Anodyne EPHX2 46 45 Cc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)cs1 ZINC000880639291 DG On-Demand Anodyne CTSV 29 40 Cc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)cs1 ZINC000880639293 DG On-Demand Anodyne CTSV 29 40 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1csc(C)c1)CC2 ZINC000880639295 EI On-Demand Anodyne SLC18A2 46 34 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1csc(C)c1)CC2 ZINC000880639298 EI On-Demand Anodyne SLC18A2 46 34 Cc1cc(NC(=O)NCCc2ccns2)cs1 ZINC000880639325 CF On-Demand Anodyne PRMT3 44 32 Cc1cc(NC(=O)N[C@H](COC(=N)O)Cc2ccccc2)cs1 ZINC000880639381 EG On-Demand Anodyne MME 44 37 Cc1cc(NC(=O)N[C@H](COC(=N)O)Cc2ccccc2)cs1 ZINC000880639381 EG On-Demand Anodyne ANPEP 56 32 Cc1cc(NC(=O)N[C@H](COC(=N)O)Cc2ccccc2)cs1 ZINC000880639381 EG On-Demand Anodyne PLAU 43 36 COC(=O)Cc1ccccc1CNC(=O)Nc1csc(C)c1 ZINC000880639447 DG On-Demand Anodyne ROCK2 15 40 COC(=O)N1CCC(NC(=O)Nc2csc(C)c2)CC1 ZINC000880639453 CE On-Demand Anodyne MTOR 20 40 COC(=O)N1CCC(NC(=O)Nc2csc(C)c2)CC1 ZINC000880639453 CE On-Demand Anodyne EPHX2 55 46 COC(=O)N1CCC(NC(=O)Nc2csc(C)c2)CC1 ZINC000880639453 CE On-Demand Anodyne CXCR3 17 40 Cc1cc(NC(=O)Nc2ccc(N3CCC(O)CC3)c(C#N)c2)cs1 ZINC000880639454 FH On-Demand Mild NPY2R 40 37 COc1cc(C(=O)NNC(=O)Nc2csc(C)c2)cc(OC)c1OC ZINC000880639461 FF On-Demand Reactive SMO 18 45 CC[C@@H](C(=O)NNC(=O)Nc1csc(C)c1)c1ccccc1 ZINC000880639488 DG On-Demand Reactive KCNQ2 47 42 Cc1cc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)cs1 ZINC000880639623 EF On-Demand Anodyne EPHX2 34 51 Cc1cc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)cs1 ZINC000880639623 EF On-Demand Anodyne CACNA1I 58 36 Cc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)cs1 ZINC000880639647 EG On-Demand Anodyne EPHX2 43 39 Cc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)cs1 ZINC000880639647 EG On-Demand Anodyne GPR119 30 40 Cc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C[C@H]2O)cs1 ZINC000880639657 FF On-Demand Anodyne GPR119 27 41 Cc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C[C@@H]2O)cs1 ZINC000880639660 FF On-Demand Anodyne GPR119 27 41 COc1ccc(CN(CCO)C(=O)Nc2csc(C)c2)cc1 ZINC000880639665 DG On-Demand Anodyne BMP1 53 42 COc1ccc(CN(CCO)C(=O)Nc2csc(C)c2)cc1 ZINC000880639665 DG On-Demand Anodyne ROCK2 16 46 Cc1cc(NC(=O)N[C@H]2CCOC2=O)cs1 ZINC000880639669 BD On-Demand Anodyne LUXR 76 41 Cc1cc(NC(=O)N[C@H]2CCOC2=O)cs1 ZINC000880639669 BD On-Demand Anodyne TRAR 89 40 Cc1cc(NC(=O)N[C@H]2CCOC2=O)cs1 ZINC000880639669 BD On-Demand Anodyne LASR 65 40 Cc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)cs1 ZINC000880639702 EH On-Demand Anodyne EPHX2 19 41 Cc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)cs1 ZINC000880639705 EH On-Demand Anodyne EPHX2 19 41 CN(CCN1CCOCC1)C(=O)Nc1cccc2c1OC(C)(C)C=C2 ZINC000880639707 EF On-Demand Anodyne CASR 50 37 CC(=O)Nc1cccc2c1CN(C(=O)Nc1csc(C)c1)CC2 ZINC000880639750 EH On-Demand Anodyne P2RY14 49 35 COc1ccc(N2CC[C@H](CNC(=O)Nc3csc(C)c3)C2)cc1 ZINC000880639842 EH On-Demand Clean CCR3 23 41 COc1ccc(N2CC[C@H](NC(=O)Nc3csc(C)c3)C2)cc1 ZINC000880639903 EG On-Demand Clean EPHX2 42 37 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)/C=C\c3ccc4c(c3)OCO4)sc2C1 ZINC000880639907 IH On-Demand Anodyne DYRK2 46 31 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)/C=C/c3ccc4c(c3)OCO4)sc2C1 ZINC000880639909 IH On-Demand Anodyne DYRK2 46 31 CN1CCN(C(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880639921 DF On-Demand Anodyne TRPM8 28 40 C[C@H](NC(=O)Nc1cccc2c1OC(C)(C)C=C2)c1cccnc1 ZINC000880639967 DI On-Demand Anodyne KCNA5 16 41 Cc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)cs1 ZINC000880640084 CG On-Demand Anodyne PRMT3 26 41 Cc1cc(NC(=O)NCC[C@H](O)C2CCCC2)cs1 ZINC000880640085 CG On-Demand Anodyne PRMT3 26 41 Cc1noc(C2CCN(C(=O)Nc3cccc4c3OC(C)(C)C=C4)CC2)n1 ZINC000880640208 FH On-Demand Anodyne SMO 41 47 Cc1cc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)cs1 ZINC000880640245 EG On-Demand Anodyne NAMPT 55 38 COc1ccccc1[C@@H](O)CNC(=O)Nc1csc(C)c1 ZINC000880640361 DF On-Demand Anodyne ADRB2 23 43 COc1ccccc1[C@@H](O)CNC(=O)Nc1csc(C)c1 ZINC000880640361 DF On-Demand Anodyne ADRB1 41 32 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)c3c4c(nc5ccccc35)CCC4)sc2C1 ZINC000880640460 JJ On-Demand Anodyne ACHE 60 39 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)c3c4c(nc5ccccc35)CCC4)sc2C1 ZINC000880640460 JJ On-Demand Anodyne BCHE 91 39 Cc1cc(NC(=O)N[C@H](CCO)Cc2ccccc2)cs1 ZINC000880640639 DG On-Demand Anodyne MME 56 39 Cc1cc(NC(=O)N[C@H](CCO)Cc2ccccc2)cs1 ZINC000880640639 DG On-Demand Anodyne ANPEP 57 32 Cc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccc(F)cc2)cs1 ZINC000880640684 DH On-Demand Anodyne CCR3 51 38 Cc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccc(F)cc2)cs1 ZINC000880640686 DH On-Demand Anodyne CCR3 51 38 COC(=O)CCCCCCNC(=O)Nc1csc(C)c1 ZINC000880640764 CG On-Demand Anodyne EPHX2 18 45 COc1ccc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc1F ZINC000880640780 EH On-Demand Clean HTR1B 15 53 COc1ccc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc1F ZINC000880640780 EH On-Demand Clean PDGFRB 48 41 COc1ccc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc1F ZINC000880640780 EH On-Demand Clean RBP4 18 42 Cc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)cs1 ZINC000880640783 DH On-Demand Anodyne TRPV1 18 42 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cs1 ZINC000880640790 CH On-Demand Anodyne IMDH_CRYPV 57 34 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cs1 ZINC000880640790 CH On-Demand Anodyne KCNK3 65 39 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cs1 ZINC000880640790 CH On-Demand Anodyne KCNK9 58 36 Cc1cc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)cs1 ZINC000880640800 EG On-Demand Anodyne CACNA1I 64 37 Cc1cc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)cs1 ZINC000880640801 EG On-Demand Anodyne CACNA1I 64 37 COCCN1CCC(NC(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880640815 FG On-Demand Anodyne CCR3 17 40 Cc1cc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)cs1 ZINC000880640826 EH On-Demand Anodyne F7 20 41 Cc1cc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)cs1 ZINC000880640827 EH On-Demand Anodyne F7 20 41 CN(C)C(=O)c1cccc(CNC(=O)Nc2cccc3c2OC(C)(C)C=C3)c1 ZINC000880640852 GH On-Demand Anodyne ROCK2 19 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cccc3c2OC(C)(C)C=C3)CC1 ZINC000880640898 GF On-Demand Anodyne CCR8 84 39 COC[C@@H](O)CNC(=O)Nc1csc(C)c1 ZINC000880640959 BD On-Demand Anodyne ADRB1 41 32 COc1cc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc(OC)c1OC ZINC000880640969 GG On-Demand Clean PDGFRB 55 42 Cc1cc(NC(=O)NCC[C@H](O)c2ccccc2)cs1 ZINC000880640971 CG On-Demand Anodyne F7 18 40 Cc1cc(NC(=O)NCC[C@@H](O)c2ccccc2)cs1 ZINC000880640972 CG On-Demand Anodyne F7 18 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640981 EI On-Demand Mild ROCK1 15 41 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640981 EI On-Demand Mild ROCK2 28 45 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640981 EI On-Demand Mild PDS 44 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640982 EI On-Demand Mild ROCK1 15 41 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640982 EI On-Demand Mild ROCK2 28 45 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2csc(C)c2)c1 ZINC000880640982 EI On-Demand Mild PDS 44 36 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne ACE 35 41 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne F10 22 42 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne MME 23 41 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne SIGMAR1 15 40 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne NPY1R 29 43 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne CCKAR 36 40 Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)cs1 ZINC000880640985 EG On-Demand Anodyne CCKBR 50 40 COc1ccc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc1 ZINC000880640996 EG On-Demand Clean HTR1B 17 47 COc1ccc(N2CCN(C(=O)Nc3csc(C)c3)CC2)cc1 ZINC000880640996 EG On-Demand Clean PDGFRB 52 42 COc1cccc(C2(NC(=O)C3CCC(S(C)(=O)=O)CC3)CC2)c1 ZINC000880641119 FE On-Demand Anodyne MTNR1A 34 46 COc1cccc(C2(NC(=O)C3CCC(S(C)(=O)=O)CC3)CC2)c1 ZINC000880641119 FE On-Demand Anodyne MTNR1B 28 46 Cn1nnc(C(=O)NC2(Cc3ccccc3)CCC2)n1 ZINC000880641132 CD On-Demand Anodyne SLC12A5 50 36 Cn1ncc(Br)c1CC(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641134 FG On-Demand Anodyne SLC12A5 42 36 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc(N=S(C)(C)=O)cc1)C2 ZINC000880641152 FH On-Demand Anodyne MTNR1A 24 47 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc(N=S(C)(C)=O)cc1)C2 ZINC000880641152 FH On-Demand Anodyne MTNR1B 27 47 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc(N=S(C)(C)=O)cc1)C2 ZINC000880641152 FH On-Demand Anodyne ROCK2 16 42 Cc1cc(NC(=O)NCC2CCN(S(=O)(=O)C(F)F)CC2)cs1 ZINC000880641177 FE On-Demand Anodyne CACNA1I 44 33 Cc1cc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)cs1 ZINC000880641180 EF On-Demand Anodyne CA1 25 41 CCn1c(CNC(=O)Nc2csc(C)c2)nc2ccccc21 ZINC000880641200 DH On-Demand Anodyne PYGM 21 40 COc1cccc(C2(NC(=O)c3nnn(C)n3)CC2)c1 ZINC000880641214 CC On-Demand Anodyne DRD4 41 31 Cc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)cs1 ZINC000880641218 EH On-Demand Anodyne AVPR2 18 42 Cc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)cs1 ZINC000880641218 EH On-Demand Anodyne L3MBTL3 66 35 Cc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)cs1 ZINC000880641218 EH On-Demand Anodyne NAMPT 25 53 COC(=O)N1CCC[C@H](NC(=O)Nc2csc(C)c2)C1 ZINC000880641233 CE On-Demand Anodyne EPHX2 30 40 COC(=O)N1CCC[C@@H](NC(=O)Nc2csc(C)c2)C1 ZINC000880641234 CE On-Demand Anodyne EPHX2 30 40 O=C(CN1CCCCS1(=O)=O)NC1(Cc2ccccc2)CCC1 ZINC000880641235 ED On-Demand Anodyne SLC12A5 45 36 Cc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)cs1 ZINC000880641236 DF On-Demand Anodyne ADRB2 32 47 Cc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)cs1 ZINC000880641236 DF On-Demand Anodyne ADRB1 64 41 Cc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)cs1 ZINC000880641236 DF On-Demand Anodyne ADRB3 31 40 Cc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)cs1 ZINC000880641236 DF On-Demand Anodyne ACOX1 47 36 Cc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)cs1 ZINC000880641236 DF On-Demand Anodyne PDS 42 41 Cc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)cs1 ZINC000880641237 DF On-Demand Anodyne ADRB2 32 47 Cc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)cs1 ZINC000880641237 DF On-Demand Anodyne ADRB1 64 41 Cc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)cs1 ZINC000880641237 DF On-Demand Anodyne ADRB3 31 40 Cc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)cs1 ZINC000880641237 DF On-Demand Anodyne ACOX1 47 36 Cc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)cs1 ZINC000880641237 DF On-Demand Anodyne PDS 42 41 O=C(NC1(C2CC2)CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880641260 DH On-Demand Anodyne PDE4D 19 45 COc1cccc(C2(NC(=O)COC3CC3)CC2)c1 ZINC000880641275 CD On-Demand Anodyne MTNR1A 41 40 COc1cccc(C2(NC(=O)COC3CC3)CC2)c1 ZINC000880641275 CD On-Demand Anodyne MTNR1B 40 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(C2CC2)CC1 ZINC000880641279 DD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(C2CC2)CC1 ZINC000880641279 DD On-Demand Anodyne CTSK 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(C2CC2)CC1 ZINC000880641280 DD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(C2CC2)CC1 ZINC000880641280 DD On-Demand Anodyne CTSK 15 46 COc1ccc(O)c([C@H](C)NC(=O)Nc2csc(C)c2)c1 ZINC000880641283 DH On-Demand Clean THRB 45 37 COc1ccc(O)c([C@@H](C)NC(=O)Nc2csc(C)c2)c1 ZINC000880641284 DH On-Demand Clean THRB 45 37 Cc1cc(NC(=O)NCCS(=O)(=O)N2CCOCC2)cs1 ZINC000880641285 EC On-Demand Anodyne LPL 32 41 COc1cccc(C2(NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)CC2)c1 ZINC000880641294 FG On-Demand Anodyne DRD4 41 32 COc1cccc(C2(NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)CC2)c1 ZINC000880641295 FG On-Demand Anodyne DRD4 41 32 COc1cccc(C2(NC(=O)[C@H]3C[C@@H]4CC[C@H](C3)S4(=O)=O)CC2)c1 ZINC000880641296 EE On-Demand Anodyne MTNR1A 22 41 COc1cccc(C2(NC(=O)[C@H]3C[C@@H]4CC[C@H](C3)S4(=O)=O)CC2)c1 ZINC000880641296 EE On-Demand Anodyne MTNR1B 25 41 Cc1cc(NC(=O)NC[C@@H](O)c2ccccc2C(F)(F)F)cs1 ZINC000880641309 EH On-Demand Anodyne SOAT1 17 41 Cc1cc(NC(=O)NC[C@H](O)c2ccccc2C(F)(F)F)cs1 ZINC000880641310 EH On-Demand Anodyne SOAT1 17 41 COc1cccc(C2(NC(=O)c3c4c(nn3C)CCSC4)CC2)c1 ZINC000880641333 EF On-Demand Anodyne DRD4 41 31 COc1cccc(C2(NC(=O)c3cc(C)cnc3Cl)CC2)c1 ZINC000880641335 DG On-Demand Anodyne DRD4 43 32 COc1ccc([C@@H](O)CNC(=O)Nc2csc(C)c2)cc1 ZINC000880641359 DF On-Demand Anodyne MTNR1A 20 40 COc1ccc([C@@H](O)CNC(=O)Nc2csc(C)c2)cc1 ZINC000880641359 DF On-Demand Anodyne F7 21 43 COc1cccc(C2(NC(=O)CN3CCCCS3(=O)=O)CC2)c1 ZINC000880641373 ED On-Demand Anodyne DRD4 40 31 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)C3(c4ccccc4)CCCC3)sc2C1 ZINC000880641378 IJ On-Demand Anodyne SLC27A1 28 40 COc1cccc(C2(NC(=O)c3ccc(CN4CCOCC4)o3)CC2)c1 ZINC000880641393 FF On-Demand Anodyne DRD4 43 34 COc1cccc(C2(NC(=O)c3ccc(CN4CCOCC4)o3)CC2)c1 ZINC000880641393 FF On-Demand Anodyne MMP13 16 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2cccc(OC)c2)CC1 ZINC000880641403 GF On-Demand Anodyne FPR1 44 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2cccc(OC)c2)CC1 ZINC000880641404 GF On-Demand Anodyne FPR1 44 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C1CC1 ZINC000880641425 DE On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C1CC1 ZINC000880641425 DE On-Demand Anodyne CTSK 15 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C1CC1 ZINC000880641426 DE On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)C1CC1 ZINC000880641426 DE On-Demand Anodyne CTSK 15 49 COc1cccc(C2(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880641444 EE On-Demand Anodyne DRD4 42 32 COc1cccc(C2(NC(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880641444 EE On-Demand Anodyne MTNR1B 15 40 COc1cccc(C2(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880641445 EE On-Demand Anodyne DRD4 42 32 COc1cccc(C2(NC(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880641445 EE On-Demand Anodyne MTNR1B 15 40 O=C(COC1CC1)NC1(Cc2ccccc2)CCC1 ZINC000880641458 CE On-Demand Anodyne TIMP3 82 38 O=C(NC1(C2CC2)CC1)c1ccnc(Cl)c1I ZINC000880641469 FG On-Demand Anodyne G2YM83_BOTF4 54 34 O=C(NC1(Cc2ccccc2)CCC1)[C@H]1CCc2nncn2CC1 ZINC000880641537 DF On-Demand Anodyne CACNA1G 16 40 O=C(NC1(Cc2ccccc2)CCC1)[C@@H]1CCc2nncn2CC1 ZINC000880641538 DF On-Demand Anodyne CACNA1G 16 40 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2csc(C)c2)c1 ZINC000880641540 EF On-Demand Anodyne MTNR1A 21 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne PGC 55 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne KLK3 61 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne PAPA1_CARPA 53 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne CCKAR 46 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne CTSK 38 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne CTSL 30 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne REN 66 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne CTSS 18 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne CAPN1 36 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641542 GG On-Demand Anodyne FPR1 57 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne PGC 55 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne KLK3 61 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne PAPA1_CARPA 53 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne CCKAR 46 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne CTSK 38 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne CTSL 30 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne REN 66 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne CTSS 18 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne CAPN1 36 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(Cc2ccccc2)CCC1 ZINC000880641543 GG On-Demand Anodyne FPR1 57 42 N#C[C@H](c1ccc(F)cc1)N1CCN(C(=O)/C=C\c2cccnc2)CC1 ZINC000880641548 FF On-Demand Mild PTAFR 47 56 N#C[C@@H](c1ccc(F)cc1)N1CCN(C(=O)/C=C\c2cccnc2)CC1 ZINC000880641549 FF On-Demand Mild PTAFR 47 56 CCOC(=O)N1CCN(C(=O)Nc2csc(C)c2)CC1 ZINC000880641550 CE On-Demand Anodyne P2RY12 46 40 CCOC(=O)N1CCN(C(=O)Nc2csc(C)c2)CC1 ZINC000880641550 CE On-Demand Anodyne TGM2 21 43 CCOC(=O)N1CCN(C(=O)Nc2csc(C)c2)CC1 ZINC000880641550 CE On-Demand Anodyne F13A1 36 43 O=C(NC1(C2CC2)CC1)c1cccn2nccc12 ZINC000880641571 BE On-Demand Anodyne JAK3 19 40 O=C(NC1(C2CC2)CC1)c1cccn2nccc12 ZINC000880641571 BE On-Demand Anodyne JAK1 15 40 O=C(NC1(C2CC2)CC1)c1cccn2nccc12 ZINC000880641571 BE On-Demand Anodyne TYK2 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2ccc(Cl)cc2)CC1 ZINC000880641572 GG On-Demand Anodyne FPR1 46 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2ccc(Cl)cc2)CC1 ZINC000880641573 GG On-Demand Anodyne FPR1 46 43 O=C(NC1(c2ccc(Cl)cc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880641583 FG On-Demand Anodyne DRD4 19 42 O=C(NC1(c2ccc(Cl)cc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880641583 FG On-Demand Anodyne DPOL_VZVD 23 40 Cc1cc(NC(=O)NCC2CCN(S(=O)(=O)C(F)(F)F)CC2)cs1 ZINC000880641591 GF On-Demand Anodyne CACNA1I 57 36 Cc1cc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)cs1 ZINC000880641593 EH On-Demand Clean PIK3CA 27 41 Cc1cc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)cs1 ZINC000880641593 EH On-Demand Clean MTOR 42 41 Cc1cc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)cs1 ZINC000880641593 EH On-Demand Clean PIK3CG 22 41 COc1ccc(N2CCCN(C(=O)Nc3csc(C)c3)CC2)cc1 ZINC000880641616 EH On-Demand Clean PDGFRB 49 39 O=C(CC[C@@H]1CCc2ccccc21)NC1(C2CC2)CC1 ZINC000880641626 CH On-Demand Anodyne MTNR1A 15 42 O=C(CC[C@@H]1CCc2ccccc21)NC1(C2CC2)CC1 ZINC000880641626 CH On-Demand Anodyne MTNR1B 16 42 O=C(CC[C@H]1CCc2ccccc21)NC1(C2CC2)CC1 ZINC000880641627 CH On-Demand Anodyne MTNR1A 15 42 O=C(CC[C@H]1CCc2ccccc21)NC1(C2CC2)CC1 ZINC000880641627 CH On-Demand Anodyne MTNR1B 16 42 O=C(NC1(C2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880641634 CF On-Demand Anodyne GABRA1 16 44 O=C(NC1(C2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880641634 CF On-Demand Anodyne GABRA2 16 44 CCOC(=O)N1CCC(NC(=O)Nc2csc(C)c2)CC1 ZINC000880641643 DF On-Demand Anodyne EPHX2 58 49 CCOC(=O)N1CCC(NC(=O)Nc2csc(C)c2)CC1 ZINC000880641643 DF On-Demand Anodyne CXCR3 18 43 CO/C(=C\c1ccccc1)C(=O)NC1(C2CC2)CC1 ZINC000880641645 CF On-Demand Anodyne TLR4 25 43 CO/C(=C/c1ccccc1)C(=O)NC1(C2CC2)CC1 ZINC000880641646 CF On-Demand Anodyne TLR4 25 43 Cc1cc(NC(=O)NCc2ccc(N3CCC(O)CC3)c(F)c2)cs1 ZINC000880641648 FG On-Demand Clean NPY2R 43 37 COc1ccc(N2CCC(NC(=O)Nc3csc(C)c3)CC2)cc1 ZINC000880641649 EH On-Demand Clean EPHX2 51 40 COc1ccc(N2CCC(NC(=O)Nc3csc(C)c3)CC2)cc1 ZINC000880641649 EH On-Demand Clean PDK1 45 31 Cn1nnc(C(=O)NCc2cccc(C3(C)OCCO3)c2)n1 ZINC000880641685 DC On-Demand Anodyne CARM1 40 34 COc1cccc(C2(NC(=O)Cc3ccccc3N3CCCC3=O)CC2)c1 ZINC000880641692 FG On-Demand Anodyne DRD4 42 35 COc1cccc(C2(NC(=O)Cc3ccccc3N3CCCC3=O)CC2)c1 ZINC000880641692 FG On-Demand Anodyne MTNR1A 19 40 O=C(NC1(Cc2ccccc2)CCC1)c1ccc(CN2CCOCC2)o1 ZINC000880641694 FG On-Demand Anodyne TACR2 49 36 O=C(NC1(Cc2ccccc2)CCC1)c1ccc(CN2CCOCC2)o1 ZINC000880641694 FG On-Demand Anodyne SLC12A5 44 32 O=C(NC1(C2CC2)CC1)c1cccnc1I ZINC000880641709 EE On-Demand Anodyne G2YM83_BOTF4 57 36 CCOC(=O)N1CCCN(C(=O)Nc2csc(C)c2)CC1 ZINC000880641712 DF On-Demand Anodyne P2RY12 42 38 CCOC(=O)N1CCCN(C(=O)Nc2csc(C)c2)CC1 ZINC000880641712 DF On-Demand Anodyne F13A1 26 41 CC(=O)N(CC(=O)NC1(Cc2ccccc2)CCC1)c1ccccc1 ZINC000880641722 EG On-Demand Anodyne SLC12A5 43 35 CON(C)CCNC(=O)[C@H](C)Oc1ccc(F)cc1 ZINC000880641766 CD On-Demand Anodyne SLC6A9 23 40 CON(C)CCNC(=O)[C@@H](C)Oc1ccc(F)cc1 ZINC000880641767 CD On-Demand Anodyne SLC6A9 23 40 CON(C)CCNC(=O)CCc1nc2ccccc2[nH]1 ZINC000880641769 CD On-Demand Anodyne CACNA1G 24 44 CON(C)CCNC(=O)CCc1nc2ccccc2[nH]1 ZINC000880641769 CD On-Demand Anodyne PARP3 23 40 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne PAPA1_CARPA 27 45 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne CTSK 17 46 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne CTSL 36 46 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne FURIN 21 40 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne CTSS 26 46 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne CTSV 18 40 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1 ZINC000880641779 ED On-Demand Anodyne UTS2 70 38 CON(C)CCNC(=O)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880641793 ED On-Demand Anodyne P2RX7 35 52 CON(C)CCNC(=O)CCc1ccc2ccccc2n1 ZINC000880641799 CD On-Demand Anodyne CYSLTR1 51 42 CON(C)CCNC(=O)CCc1ccc2ccccc2n1 ZINC000880641799 CD On-Demand Anodyne MTNR1A 43 37 CCOC(=O)Nc1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880641801 CD On-Demand Anodyne ACR 44 33 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne MMP13 22 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne MMP3 30 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne MMP9 20 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne EPHX2 47 54 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne TGM2 67 43 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne MMP7 30 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne MMP1 27 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880641822 FC On-Demand Anodyne F13A1 58 38 CON(C)CCNC(=O)C1CCN(c2ccc(C(F)(F)F)cn2)CC1 ZINC000880641826 FD On-Demand Anodyne DGAT1 19 40 CON(C)CCNC(=O)CCCNS(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000880641830 GD On-Demand Anodyne CACNA1B 46 34 COc1ccc(C(=O)N2CCC[C@H](C(=O)NCCN(C)OC)C2)c2ccccc12 ZINC000880641835 GE On-Demand Anodyne ACKR3 64 33 COc1ccc(C(=O)N2CCC[C@@H](C(=O)NCCN(C)OC)C2)c2ccccc12 ZINC000880641836 GE On-Demand Anodyne ACKR3 64 33 CON(C)CCNC(=O)CNC(=O)CC12CC3CC(CC(C3)C1)C2 ZINC000880641837 ED On-Demand Anodyne EPHX2 19 51 CON(C)CCNC(=O)CNC(=O)CC12CC3CC(CC(C3)C1)C2 ZINC000880641837 ED On-Demand Anodyne BOTA 29 44 CCOc1ccc(SCC(=O)NCCN(C)OC)cc1 ZINC000880641840 CD On-Demand Anodyne MTNR1A 24 40 CCOc1ccc(SCC(=O)NCCN(C)OC)cc1 ZINC000880641840 CD On-Demand Anodyne FAS 43 40 CON(C)CCNC(=O)CCCOc1cccc(Br)c1 ZINC000880641841 EE On-Demand Anodyne MTNR1A 47 47 CON(C)CCNC(=O)CCCOc1cccc(Br)c1 ZINC000880641841 EE On-Demand Anodyne MTNR1B 37 47 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccccc2F)CC1 ZINC000880641843 FC On-Demand Anodyne EPHX2 46 58 CON(C)CCNC(=O)CCc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880641849 FD On-Demand Anodyne TGM2 59 39 CON(C)CCNC(=O)CCc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880641849 FD On-Demand Anodyne F13A1 60 38 CON(C)CCNC(=O)CCc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880641849 FD On-Demand Anodyne NAMPT 38 41 CON(C)CCNC(=O)CNC(=O)c1ccc(Oc2ccccc2)cc1 ZINC000880641858 FD On-Demand Anodyne LTA4H 42 43 CON(C)CCNC(=O)CNC(=O)c1ccc(Oc2ccccc2)cc1 ZINC000880641858 FD On-Demand Anodyne CRTM 41 37 CON(C)CCNC(=O)Cc1coc2ccc3ccccc3c12 ZINC000880641881 DF On-Demand Anodyne NQO2 43 37 CON(C)CCNC(=O)C1CCN(c2ncnc3sc(C)c(C)c23)CC1 ZINC000880641882 GE On-Demand Anodyne SIRT3 68 37 CON(C)CCNC(=O)C1CCN(c2ncnc3sc(C)c(C)c23)CC1 ZINC000880641882 GE On-Demand Anodyne SIRT2 52 33 CON(C)CCNC(=O)C1CCN(c2ncnc3sc(C)c(C)c23)CC1 ZINC000880641882 GE On-Demand Anodyne SIRT1 50 31 CON(C)CCNC(=O)C1CCN(c2ncnc3sc(C)c(C)c23)CC1 ZINC000880641882 GE On-Demand Anodyne LIMK2 27 40 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000880641883 GD On-Demand Anodyne CCR5 18 40 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000880641883 GD On-Demand Anodyne PTR1 41 36 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000880641883 GD On-Demand Anodyne L3MBTL3 80 41 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne OPRM1 24 46 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne OPRD1 74 46 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne PREP 15 40 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne MMP3 19 40 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne CFTR 84 48 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne ADAM9 67 40 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880641892 FD On-Demand Anodyne MMP1 15 40 CON(C)CCNC(=O)C(O)(c1ccccc1)c1ccccc1 ZINC000880641894 DD On-Demand Anodyne AMY2 58 37 CON(C)CCNC(=O)CCc1ccccc1F ZINC000880641899 CD On-Demand Anodyne MTNR1A 44 42 CON(C)CCNC(=O)CCc1nc2ccccc2o1 ZINC000880641901 CD On-Demand Anodyne MTNR1A 32 42 CON(C)CCNC(=O)CCc1nc2ccccc2o1 ZINC000880641901 CD On-Demand Anodyne MTNR1B 34 42 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1 ZINC000880641902 GD On-Demand Anodyne EPHX2 36 48 CON(C)CCNC(=O)CCc1nc(O)c2ccccc2n1 ZINC000880641907 DC On-Demand Anodyne TNKS 56 32 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(C(C)C)cc2)CC1 ZINC000880641924 GD On-Demand Anodyne EPHX2 38 59 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(C(C)C)cc2)CC1 ZINC000880641924 GD On-Demand Anodyne TGM2 46 39 CON(C)CCNC(=O)C[C@H]1c2ccccc2CCN1C(C)=O ZINC000880641928 DD On-Demand Anodyne MTNR1A 17 42 CON(C)CCNC(=O)C[C@H]1c2ccccc2CCN1C(C)=O ZINC000880641928 DD On-Demand Anodyne MTNR1B 27 51 CON(C)CCNC(=O)C[C@@H]1c2ccccc2CCN1C(C)=O ZINC000880641929 DD On-Demand Anodyne MTNR1A 17 42 CON(C)CCNC(=O)C[C@@H]1c2ccccc2CCN1C(C)=O ZINC000880641929 DD On-Demand Anodyne MTNR1B 27 51 CCn1c(S)nc2cc(C(=O)NCCN(C)OC)ccc2c1=O ZINC000880641949 EC On-Demand Anodyne POLR1A 64 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PRSS1 18 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne ACE 50 47 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne OPRM1 34 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne OPRD1 32 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MME 146 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne ANPEP 73 37 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne TACR1 22 49 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSD 24 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CMA1 24 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTRA_BOVIN 18 60 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne FCER2 96 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSB 79 51 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PAPA1_CARPA 89 67 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CYSP_TRYCR 66 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSG 34 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSK 38 60 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSL 94 67 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CPA1 37 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CACNA1B 46 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne NPFFR2 53 48 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne TIMP3 81 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PYGL 15 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTRB1 56 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne TACR3 30 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CAPNS1 69 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MMP2 25 50 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MMP3 42 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MMP8 28 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne GRIA1 56 53 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne HLA-DRB1 59 37 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CELA2A 30 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne FURIN 46 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PTPRA 58 32 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSS 50 67 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CAPN1 97 48 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MMP9 33 47 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CAPN2 89 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne ACE2 77 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTSV 63 56 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PIN1 23 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne MMP1 50 47 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne FPR1 76 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne CTRB_BOVIN 60 37 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne NPR 82 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne AMP1_PLAFQ 49 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PSMB5 34 53 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne BLA1_STEMA 70 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne KISS1R 76 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne QRFPR 46 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne UTS2 73 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne PSMB8 53 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1 ZINC000880641952 FD On-Demand Anodyne NPFFR1 70 48 CON(C)CCNC(=O)CSc1ccc(F)cc1 ZINC000880641955 CD On-Demand Anodyne FAS 48 38 COc1ccc(OCC(=O)NCCN(C)OC)cc1 ZINC000880641971 CC On-Demand Anodyne MTNR1A 94 44 COc1ccc(OCC(=O)NCCN(C)OC)cc1 ZINC000880641971 CC On-Demand Anodyne MTNR1B 71 44 COc1ccc(OCC(=O)NCCN(C)OC)cc1 ZINC000880641971 CC On-Demand Anodyne CA9 15 41 CON(C)CCNC(=O)CCc1nnc(-c2ccccc2)o1 ZINC000880641974 DD On-Demand Anodyne MTNR1A 15 42 CON(C)CCNC(=O)CCc1nnc(-c2ccccc2)o1 ZINC000880641974 DD On-Demand Anodyne FAAH 18 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne F2 15 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne ACE 49 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne OPRM1 62 47 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne OPRD1 61 47 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MME 148 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne ANPEP 76 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne TACR1 30 50 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSD 21 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CMA1 19 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne FCER2 106 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne GRB2 40 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne KLK3 55 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSB 76 48 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne PAPA1_CARPA 95 52 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CYSP_TRYCR 66 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CCKAR 54 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSK 36 52 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSL 87 52 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CPA1 40 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CACNA1B 42 37 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne NPFFR2 61 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne TIMP3 82 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne TACR3 31 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MC3R 41 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CAPNS1 74 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MMP2 25 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MMP3 44 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MMP8 29 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne GRIA1 67 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne HLA-DRB1 90 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne FURIN 62 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne PTPRA 64 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSS 41 52 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CAPN1 118 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MMP9 34 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CAPN2 121 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne ACE2 74 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MC1R 65 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTSV 56 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne PROC 19 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne MMP1 53 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne FPR1 76 54 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne CTRB_BOVIN 45 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne NPR 82 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne AMP1_PLAFQ 46 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne BLA1_STEMA 54 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne KISS1R 64 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne POLG_WNV 68 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne QRFPR 54 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne PSMB8 50 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(N)=O ZINC000880641975 CB On-Demand Anodyne NPFFR1 76 40 CON(C)CCNC(=O)Cn1c(-c2cscn2)nc2ccccc21 ZINC000880641981 ED On-Demand Anodyne IMDH_CRYPV 47 61 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP13 40 45 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP2 42 49 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP3 21 45 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP8 25 49 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP14 24 40 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP9 28 49 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne MMP7 17 40 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000880641990 EC On-Demand Anodyne LEF 25 41 CON(C)CCNC(=O)Cn1c(C(F)(F)F)nc2ccccc21 ZINC000880641992 ED On-Demand Anodyne IMDH_CRYPV 31 41 CON(C)CCNC(=O)CSCc1ccc(F)cc1 ZINC000880641993 CD On-Demand Anodyne PLA2G7 42 33 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(Cl)cc1 ZINC000880641998 EC On-Demand Anodyne TBXA2R 52 42 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(Cl)cc1 ZINC000880641998 EC On-Demand Anodyne TBXAS1 25 42 CON(C)CCNC(=O)CCCOc1ccc(C)cc1 ZINC000880642012 CD On-Demand Anodyne LTA4H 23 42 CON(C)CCNC(=O)CCC(=O)c1ccc(-c2ccccc2)cc1 ZINC000880642013 EF On-Demand Anodyne HDAC8 19 46 CON(C)CCNC(=O)CCC(=O)c1ccc(-c2ccccc2)cc1 ZINC000880642013 EF On-Demand Anodyne FAAH 15 40 CON(C)CCNC(=O)CCC(=O)c1ccc(-c2ccccc2)cc1 ZINC000880642013 EF On-Demand Anodyne UTS2 48 36 CON(C)CCNC(=O)CNC(=O)Cc1ccccc1 ZINC000880642018 CB On-Demand Anodyne MME 22 40 CON(C)CCNC(=O)CNC(=O)Cc1ccccc1 ZINC000880642018 CB On-Demand Anodyne CA5B 32 41 CON(C)CCNC(=O)CNC(=O)Cc1ccccc1 ZINC000880642018 CB On-Demand Anodyne CA5A 36 41 CON(C)CCNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880642033 DC On-Demand Anodyne KCNQ2 42 34 CON(C)CCNC(=O)CNC(=O)c1ccccc1OC(F)F ZINC000880642037 EC On-Demand Anodyne KCNK3 40 33 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne MME 41 36 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne CTSB 22 44 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne PAPA1_CARPA 23 43 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne CTSK 20 47 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne CTSL 33 47 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne CTRB1 43 39 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne CTSS 23 47 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne NPR 71 40 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000880642061 CC On-Demand Anodyne UTS2 71 38 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne MME 41 36 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne CTSB 22 44 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne PAPA1_CARPA 23 43 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne CTSK 20 47 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne CTSL 33 47 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne CTRB1 43 39 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne CTSS 23 47 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne NPR 71 40 CON(C)CCNC(=O)[C@H](C)NC(=O)c1ccccc1 ZINC000880642062 CC On-Demand Anodyne UTS2 71 38 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(Br)cc1 ZINC000880642063 GC On-Demand Anodyne MMP14 16 58 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(Br)cc1 ZINC000880642063 GC On-Demand Anodyne IDO1 17 40 CC[C@@H](Nc1ccccc1)C(=O)NCCN(C)OC ZINC000880642068 CD On-Demand Anodyne CAPN2 51 33 CC[C@@H](Nc1ccccc1)C(=O)NCCN(C)OC ZINC000880642068 CD On-Demand Anodyne NPR 52 36 CC[C@H](Nc1ccccc1)C(=O)NCCN(C)OC ZINC000880642069 CD On-Demand Anodyne CAPN2 51 33 CC[C@H](Nc1ccccc1)C(=O)NCCN(C)OC ZINC000880642069 CD On-Demand Anodyne NPR 52 36 CCCN(CC)C(=O)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880642074 DD On-Demand Anodyne OPRD1 15 43 CCCN(CCC)C(=O)c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880642084 EE On-Demand Anodyne DRD4 45 34 CCCN(CCC)C(=O)c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880642084 EE On-Demand Anodyne BACE1 15 44 CON(C)CCNC(=O)CCCn1ccnc1 ZINC000880642086 BC On-Demand Anodyne TBXAS1 49 46 CON(C)CCNC(=O)CCCn1ccnc1 ZINC000880642086 BC On-Demand Anodyne QPCT 40 44 CON(C)CCNC(=O)CCc1ccccc1C ZINC000880642092 CD On-Demand Anodyne MTNR1A 41 40 CON(C)CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1[N+](=O)[O-] ZINC000880642093 ED On-Demand Bother COLA 66 36 CON(C)CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1[N+](=O)[O-] ZINC000880642094 ED On-Demand Bother COLA 66 36 CON(C)CCNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880642100 FC On-Demand Anodyne Q9NAW4_PLAFA 46 56 CON(C)CCNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880642100 FC On-Demand Anodyne VHL 62 36 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642101 DD On-Demand Anodyne CTSD 28 47 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642101 DD On-Demand Anodyne PAPA1_CARPA 35 40 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642101 DD On-Demand Anodyne CTSK 17 45 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642101 DD On-Demand Anodyne ECE1 43 47 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642101 DD On-Demand Anodyne POLG_HCV1 21 44 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642104 DD On-Demand Anodyne CTSD 28 47 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642104 DD On-Demand Anodyne PAPA1_CARPA 35 40 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642104 DD On-Demand Anodyne CTSK 17 45 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642104 DD On-Demand Anodyne ECE1 43 47 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642104 DD On-Demand Anodyne POLG_HCV1 21 44 CON(C)CCNC(=O)[C@@H](C)c1ccccc1F ZINC000880642125 CD On-Demand Anodyne CXCL8 28 42 CON(C)CCNC(=O)C(=O)c1ccc(Br)cc1 ZINC000880642133 DD On-Demand Anodyne SHC 43 33 CCOc1ccccc1CCC(=O)NCCN(C)OC ZINC000880642142 CD On-Demand Anodyne MTNR1A 44 40 CCOc1ccccc1CCC(=O)NCCN(C)OC ZINC000880642142 CD On-Demand Anodyne MBTPS1 40 33 CON(C)CCNC(=O)CCC(=O)c1ccc2ccccc2c1 ZINC000880642151 DE On-Demand Anodyne MTNR1A 63 38 CON(C)CCNC(=O)CCC(=O)c1ccc2ccccc2c1 ZINC000880642151 DE On-Demand Anodyne MTNR1B 43 37 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880642153 FC On-Demand Anodyne F2 22 40 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880642153 FC On-Demand Anodyne FKBP1A 24 45 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880642153 FC On-Demand Anodyne SLC6A1 51 33 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880642153 FC On-Demand Anodyne TMPRSS11D 44 32 CON(C)CCNC(=O)COc1ccc(C(C)(C)C)cc1 ZINC000880642158 CD On-Demand Anodyne MT-ND1 27 41 CON(C)CCNC(=O)Cc1c(C)noc1Cl ZINC000880642192 CC On-Demand Anodyne P2RX7 28 46 CON(C)CCNC(=O)[C@@H](CCSC)NC(=O)c1ccccc1Cl ZINC000880642209 FD On-Demand Anodyne UTS2 41 33 COc1ccc(-c2nc(C)c(C(=O)NCCN(C)OC)s2)cc1 ZINC000880642213 EE On-Demand Anodyne PPARA 15 58 COc1ccc(-c2nc(C)c(C(=O)NCCN(C)OC)s2)cc1 ZINC000880642213 EE On-Demand Anodyne CHRM4 15 41 COc1ccc(-c2nc(C)c(C(=O)NCCN(C)OC)s2)cc1 ZINC000880642213 EE On-Demand Anodyne SCD1 24 46 COc1ccc(-c2nc(C)c(C(=O)NCCN(C)OC)s2)cc1 ZINC000880642213 EE On-Demand Anodyne SCD 24 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne MMP13 27 41 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne APP 52 36 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne MMP3 29 41 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne LSS 15 42 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne MMP9 22 41 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne EPHX2 43 54 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne TGM2 49 42 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne MMP7 29 41 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880642215 GD On-Demand Anodyne MMP1 28 41 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(F)cc2)C1 ZINC000880642216 FC On-Demand Anodyne GPBAR1 17 41 CON(C)CCNC(=O)COc1ccc2c(C)cc(=O)oc2c1 ZINC000880642218 DD On-Demand Anodyne MAOA 84 67 CON(C)CCNC(=O)COc1ccc2c(C)cc(=O)oc2c1 ZINC000880642218 DD On-Demand Anodyne ACHE 16 44 CON(C)CCNC(=O)COc1ccc2c(C)cc(=O)oc2c1 ZINC000880642218 DD On-Demand Anodyne MAOB 61 67 CON(C)CCNC(=O)COc1ccc2c(C)cc(=O)oc2c1 ZINC000880642218 DD On-Demand Anodyne MTNR1A 47 35 CON(C)CCNC(=O)CCCn1c(=O)oc2ccccc21 ZINC000880642224 DC On-Demand Anodyne TSPO 17 48 CON(C)CCNC(=O)CCc1cccnc1 ZINC000880642228 BC On-Demand Anodyne TBXAS1 45 45 CON(C)CCNC(=O)CCc1cccnc1 ZINC000880642228 BC On-Demand Anodyne PTAFR 36 47 CON(C)CCNC(=O)CCc1cccnc1 ZINC000880642228 BC On-Demand Anodyne KCNA5 15 44 CON(C)CCNC(=O)CCc1cccnc1 ZINC000880642228 BC On-Demand Anodyne NAMPT 29 45 COc1cn(-c2ccccc2)nc1C(=O)NCCN(C)OC ZINC000880642231 DD On-Demand Anodyne CTSA 18 54 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne FKBP1A 17 49 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP13 68 50 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne ADAM17 45 44 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne ITGA4 35 49 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne CAPNS1 25 51 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP2 32 44 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP3 75 50 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP8 34 43 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne CAPN1 15 51 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP9 35 43 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne CASP7 40 36 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP7 70 50 CON(C)CCNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1 ZINC000880642244 FC On-Demand Anodyne MMP1 73 54 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne CA2 22 48 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne ADRB2 15 41 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne ADRB3 44 41 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne TBXA2R 23 44 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne CA1 22 48 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne CA4 24 44 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne PTPRB 44 33 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne CA12 18 41 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne CA9 24 41 CON(C)CCNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 ZINC000880642259 GD On-Demand Anodyne LIMK2 37 52 CON(C)CCNC(=O)[C@@H](O)c1cccnc1 ZINC000880642264 BB On-Demand Anodyne ADRB3 46 41 CON(C)CCNC(=O)[C@@H](O)c1cccnc1 ZINC000880642264 BB On-Demand Anodyne KCNA5 25 43 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642287 DD On-Demand Anodyne PAPA1_CARPA 44 64 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880642287 DD On-Demand Anodyne CTSK 24 48 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne DRD4 44 35 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne MTNR1A 51 43 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne MTNR1B 49 43 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne TAAR1 30 40 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne AKR1C3 40 61 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne AKR1C2 74 43 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne KCNK3 56 39 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne KCNK9 46 39 COc1cccc(Nc2ccccc2C(=O)NCCN(C)OC)c1 ZINC000880642290 EF On-Demand Anodyne POLR1A 40 39 CON(C)CCNC(=O)CCCCOc1ccc(Br)cc1 ZINC000880642304 FF On-Demand Anodyne LTA4H 21 41 CON(C)CCNC(=O)CCCCOc1ccc(Br)cc1 ZINC000880642304 FF On-Demand Anodyne SHC 61 46 CON(C)CCNC(=O)CCCCOc1ccc(Br)cc1 ZINC000880642304 FF On-Demand Anodyne PLA2G4B 50 33 CON(C)CCNC(=O)CCCCOc1ccc(Br)cc1 ZINC000880642304 FF On-Demand Anodyne LSS 72 46 CON(C)CCNC(=O)CCCCOc1ccc(Br)cc1 ZINC000880642304 FF On-Demand Anodyne ERG7 29 40 COCCn1cc(C(=O)NCCN(C)OC)c2ccccc21 ZINC000880642316 DD On-Demand Anodyne CNR1 21 57 COCCn1cc(C(=O)NCCN(C)OC)c2ccccc21 ZINC000880642316 DD On-Demand Anodyne CNR2 30 59 CON(C)CCNC(=O)Cn1c(Cc2ccccc2)nc2ccccc21 ZINC000880642336 FE On-Demand Anodyne MAOA 21 46 CCN(CC)S(=O)(=O)c1cc(C(=O)NCCN(C)OC)ccc1OC ZINC000880642342 FC On-Demand Anodyne CPT1A 51 35 CCN(CC)S(=O)(=O)c1cc(C(=O)NCCN(C)OC)ccc1OC ZINC000880642342 FC On-Demand Anodyne CPT1B 55 35 CON(C)CCNC(=O)Cc1ccc(OCc2c(C)noc2C)cc1 ZINC000880642353 EE On-Demand Anodyne RORC 15 50 CON(C)CCNC(=O)Cc1nn(C)c(=O)c2ccccc12 ZINC000880642364 DC On-Demand Anodyne IMDH_CRYPV 36 58 CON(C)CCNC(=O)CSc1ccc(Cl)cc1 ZINC000880642365 CE On-Demand Anodyne UTS2 41 32 CON(C)CCNC(=O)CSc1ccc(Cl)cc1 ZINC000880642365 CE On-Demand Anodyne FAS 55 43 COc1ccc(Nc2nc(C(=O)NCCN(C)OC)cs2)cc1 ZINC000880642378 EE On-Demand Anodyne TRPC6 58 50 COc1ccc(Nc2nc(C(=O)NCCN(C)OC)cs2)cc1 ZINC000880642378 EE On-Demand Anodyne TRPC3 55 50 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP13 57 55 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP2 46 55 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP3 22 55 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP8 30 51 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP14 22 44 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP9 28 51 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP12 89 42 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne MMP7 20 48 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne ADAMTS4 45 45 CON(C)CCNC(=O)[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(C)C ZINC000880642387 FC On-Demand Anodyne LEF 26 51 COC(=O)N1CCC(NC(=O)Nc2ccc(C(=O)N(C)C)cc2F)CC1 ZINC000880642388 FD On-Demand Anodyne EPHX2 49 40 CON(C)CCNC(=O)CC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880642397 CD On-Demand Anodyne BOTA 27 40 CON(C)CCNC(=O)[C@@H]1CCCN(c2nc3ccccc3s2)C1 ZINC000880642398 EE On-Demand Anodyne TRY1_BOVIN 42 38 CON(C)CCNC(=O)[C@@H]1CCCN(c2nc3ccccc3s2)C1 ZINC000880642398 EE On-Demand Anodyne GPBAR1 21 41 CON(C)CCNC(=O)CSc1cccc(C(F)(F)F)c1 ZINC000880642410 DE On-Demand Anodyne PDS 43 34 CON(C)CCNC(=O)CSc1ccc2ccccc2c1 ZINC000880642417 DF On-Demand Anodyne MTNR1A 49 39 CON(C)CCNC(=O)CSc1ccc2ccccc2c1 ZINC000880642417 DF On-Demand Anodyne FAS 66 40 CON(C)CCNC(=O)CCNS(=O)(=O)c1cccc(Cl)c1 ZINC000880642418 EC On-Demand Anodyne TBXA2R 40 37 CON(C)CCNC(=O)CCNS(=O)(=O)c1cccc(Cl)c1 ZINC000880642418 EC On-Demand Anodyne FBP1 25 40 CCNS(=O)(=O)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880642420 DC On-Demand Anodyne CA2 21 44 CON(C)CCNC(=O)CCNC(=O)C12CC3CC(CC(C3)C1)C2 ZINC000880642436 ED On-Demand Anodyne EPHX2 26 46 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne CHRM2 27 45 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne MTNR1A 28 43 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne MTNR1B 22 40 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne EPHX2 15 41 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne CCR8 46 33 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne L3MBTL3 23 40 CON(C)CCNC(=O)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880642437 FE On-Demand Anodyne POLR1A 47 35 CON(C)CCNC(=O)Cn1c(S)nc2ccccc2c1=O ZINC000880642438 DC On-Demand Anodyne POLR1A 45 38 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880642448 FD On-Demand Anodyne F2 21 42 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880642448 FD On-Demand Anodyne HTR7 15 42 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880642448 FD On-Demand Anodyne NQO2 23 42 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880642448 FD On-Demand Anodyne TRY2_BOVIN 63 42 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880642448 FD On-Demand Anodyne MTNR1A 38 40 CON(C)CCNC(=O)C1CCN(c2ccc3cccc(O)c3n2)CC1 ZINC000880642464 FD On-Demand Anodyne MTNR1A 17 41 CCOc1cn(-c2ccccc2)nc1C(=O)NCCN(C)OC ZINC000880642476 DD On-Demand Anodyne CTSA 15 47 CCOc1cn(-c2ccccc2)nc1C(=O)NCCN(C)OC ZINC000880642476 DD On-Demand Anodyne HCN1 48 32 CON(C)CCNC(=O)C[C@@H](C)c1cccnc1 ZINC000880642486 CD On-Demand Anodyne KCNA5 28 51 CON(C)CCNC(=O)C[C@H](C)c1cccnc1 ZINC000880642487 CD On-Demand Anodyne KCNA5 28 51 CON(C)CCNC(=O)[C@@H](c1ccccc1)N1CCC(O)CC1 ZINC000880642501 DC On-Demand Anodyne NPY2R 35 42 CON(C)CCNC(=O)[C@@H](c1ccccc1)N1CCC(O)CC1 ZINC000880642501 DC On-Demand Anodyne XIAP 45 32 CON(C)CCNC(=O)[C@@H](c1ccccc1)N1CCC(O)CC1 ZINC000880642501 DC On-Demand Anodyne BIRC2 41 31 CON(C)CCNC(=O)C[C@@H]1CCc2ccccc2C1 ZINC000880642509 CD On-Demand Anodyne PTGIR 15 44 CON(C)CCNC(=O)C[C@H]1CCc2ccccc2C1 ZINC000880642510 CD On-Demand Anodyne PTGIR 15 44 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MME 59 38 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne TBXAS1 43 43 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne PTAFR 31 46 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTRA_BOVIN 15 48 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne FCER2 61 35 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSB 42 43 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne PAPA1_CARPA 67 55 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CYSP_TRYCR 45 42 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSG 25 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSK 21 49 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSL 65 55 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne NPFFR2 33 40 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne TIMP3 40 40 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTRB1 37 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CAPNS1 43 32 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MMP3 23 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MMP8 21 46 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne GRIA1 16 49 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSS 37 60 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CAPN1 38 40 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MMP9 26 46 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTSV 59 49 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MMP7 19 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne MMP1 35 46 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne CTRB_BOVIN 44 32 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne NPR 56 33 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne PSMB5 45 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne KISS1R 58 39 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne UTS2 54 35 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne PSMB8 29 41 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)NC(=O)c1ccccc1 ZINC000880642517 FD On-Demand Anodyne NPFFR1 41 40 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(C)cc2C)CC1 ZINC000880642518 GD On-Demand Anodyne EPHX2 52 67 CCCN(CCC)S(=O)(=O)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880642519 FD On-Demand Anodyne CA2 19 57 CCCN(CCC)S(=O)(=O)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880642519 FD On-Demand Anodyne BMP1 19 40 CON(C)CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880642528 CE On-Demand Anodyne NQO2 23 49 CON(C)CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880642528 CE On-Demand Anodyne MTNR1A 29 42 CON(C)CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880642528 CE On-Demand Anodyne MTNR1B 32 42 CON(C)CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880642529 CE On-Demand Anodyne NQO2 23 49 CON(C)CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880642529 CE On-Demand Anodyne MTNR1A 29 42 CON(C)CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880642529 CE On-Demand Anodyne MTNR1B 32 42 CON(C)CCNC(=O)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880642543 GD On-Demand Anodyne EPHX2 28 43 CON(C)CCNC(=O)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880642544 GD On-Demand Anodyne EPHX2 28 43 CON(C)CCNC(=O)C1CCN(C2=NS(=O)(=O)c3ccccc32)CC1 ZINC000880642549 GC On-Demand Anodyne KCNA3 17 40 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc(C(C)(C)C)cc1 ZINC000880642570 FD On-Demand Anodyne CYNT 46 36 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(Cl)s1 ZINC000880642571 EC On-Demand Anodyne CCR4 62 36 CON(C)CCNC(=O)CCn1c(S)nc2ccccc2c1=O ZINC000880642581 EC On-Demand Anodyne POLR1A 49 37 CCc1ccc([C@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880642603 CD On-Demand Anodyne TRPV1 16 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne ACE 42 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne OPRM1 28 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne OPRD1 28 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne MME 122 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne ANPEP 64 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne TACR1 23 52 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSD 25 50 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne PGC 66 50 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne FCER2 89 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSB 80 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne PAPA1_CARPA 113 71 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CYSP_TRYCR 71 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CCKAR 71 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSK 50 67 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSL 88 71 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CACNA1B 56 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne PGA 42 50 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne NPFFR2 41 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne TIMP3 74 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne TACR3 34 57 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CAPNS1 69 39 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne MMP2 19 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne MMP3 32 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne GRIA1 52 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne HLA-DRB1 74 51 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne REN 98 54 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne REN1 35 49 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CCKBR 26 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSS 43 71 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CAPN1 103 57 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne MMP9 27 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CAPN2 119 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne ACE2 58 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne SCN10A 21 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne KLK5 23 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTSV 53 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne MMP1 43 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne FPR1 94 55 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne CTRB_BOVIN 57 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne NPR 76 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne AMP1_PLAFQ 43 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne PSMB5 41 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne QRFPR 44 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne PSMB8 48 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C ZINC000880642610 FD On-Demand Anodyne NPFFR1 58 33 CON(C)CCNC(=O)CC1(CC(=O)Nc2nccs2)CCCCC1 ZINC000880642611 FE On-Demand Anodyne MAP1 102 36 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000880642612 GC On-Demand Anodyne MMP13 23 42 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000880642612 GC On-Demand Anodyne MMP2 26 42 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000880642612 GC On-Demand Anodyne MMP8 15 49 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000880642612 GC On-Demand Anodyne MMP14 21 49 CON(C)CCNC(=O)CCc1cccc(C)c1 ZINC000880642622 CD On-Demand Anodyne MTNR1A 37 42 CON(C)CCNC(=O)CCc1cccc(C)c1 ZINC000880642622 CD On-Demand Anodyne MTNR1B 28 42 CON(C)CCNC(=O)CSCC(=O)Nc1ccc(F)cc1 ZINC000880642625 ED On-Demand Anodyne ENPP1 59 31 CON(C)CCNC(=O)CCNS(=O)(=O)c1ccc(F)c(F)c1 ZINC000880642627 FC On-Demand Anodyne TBXA2R 51 36 CON(C)CCNC(=O)CCCNS(=O)(=O)c1ccc(F)cc1 ZINC000880642629 EC On-Demand Anodyne TBXA2R 45 39 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(C)c(C)c2)CC1 ZINC000880642632 GD On-Demand Anodyne EPHX2 46 52 CON(C)CCNC(=O)C1CCN(S(=O)(=O)c2ccc(C)c(C)c2)CC1 ZINC000880642632 GD On-Demand Anodyne TGM2 38 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MME 94 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne ANPEP 64 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne TBXAS1 48 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne PTAFR 27 41 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTRA_BOVIN 19 48 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne FCER2 76 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSB 50 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne PAPA1_CARPA 73 55 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CYSP_TRYCR 59 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSG 17 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSK 23 49 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSL 74 55 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne NPFFR2 38 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne TIMP3 60 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTRB1 30 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CAPNS1 58 32 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP2 15 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP3 23 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP8 22 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne GRIA1 48 55 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne HLA-DRB1 48 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSS 38 57 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CAPN1 60 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP9 27 42 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CAPN2 45 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne ACE2 49 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MC1R 15 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTSV 58 46 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP7 20 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne MMP1 36 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne FPR1 56 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne CTRB_BOVIN 43 32 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne NPR 57 35 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne PSMB5 47 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne BLA1_STEMA 43 37 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne KISS1R 63 44 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne UTS2 40 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne PSMB8 42 43 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne NPFFR1 49 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cccnc1 ZINC000880642658 FD On-Demand Anodyne GPR142 45 33 CON(C)CCNC(=O)[C@@]1(C)CCCN1C(=O)c1ccccc1 ZINC000880642661 DD On-Demand Anodyne SLC12A5 53 36 CON(C)CCNC(=O)[C@@H](OC1CCCC1)c1ccccc1 ZINC000880642667 DE On-Demand Anodyne AMY2 49 34 CON(C)CCNC(=O)CNc1cccc(C(F)(F)F)c1 ZINC000880642670 DD On-Demand Anodyne CCR2 49 39 COc1ccc(Cn2cc(C(=O)NCCN(C)OC)cn2)cc1 ZINC000880642671 DD On-Demand Anodyne DRD4 41 31 COc1ccc(Cn2cc(C(=O)NCCN(C)OC)cn2)cc1 ZINC000880642671 DD On-Demand Anodyne PROKR1 63 34 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne ACE 31 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne MME 108 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne ANPEP 51 45 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne FCER2 41 32 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne PAPA1_CARPA 61 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne CPA1 46 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne CAPNS1 54 33 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne MMP3 23 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne MMP8 18 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne CAPN1 52 40 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne CAPN2 46 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne ACE2 42 36 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne NPR 56 38 CON(C)CCNC(=O)[C@@H](Cc1ccccc1)N(C)C ZINC000880642679 CC On-Demand Anodyne AMP1_PLAFQ 54 42 CON(C)CCNC(=O)[C@@H](C)SCc1ncc(-c2ccc(Cl)cc2)o1 ZINC000880642697 GG On-Demand Anodyne NPPA 20 40 CON(C)CCNC(=O)[C@H](C)SCc1ncc(-c2ccc(Cl)cc2)o1 ZINC000880642698 GG On-Demand Anodyne NPPA 20 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccc2ccccc2c1O ZINC000880642710 FD On-Demand Anodyne TRY1_BOVIN 40 35 CON(C)CCNC(=O)C[C@H]1CCc2ccccc21 ZINC000880642712 CD On-Demand Anodyne NQO2 21 42 CON(C)CCNC(=O)C[C@@H]1CCc2ccccc21 ZINC000880642713 CD On-Demand Anodyne NQO2 21 42 CON(C)CCNC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000880642719 FG On-Demand Anodyne F10 40 31 CON(C)CCNC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000880642719 FG On-Demand Anodyne ALPL 47 41 CON(C)CCNC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000880642719 FG On-Demand Anodyne DPP8 74 34 CON(C)CCNC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000880642719 FG On-Demand Anodyne DPP9 71 34 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2N1C(C)=O ZINC000880642723 CC On-Demand Anodyne ACE 19 41 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2N1C(C)=O ZINC000880642723 CC On-Demand Anodyne ADAM9 58 33 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2N1C(C)=O ZINC000880642723 CC On-Demand Anodyne TPP2 61 52 CON(C)CCNC(=O)CN(Cc1cccnc1)c1ccccc1 ZINC000880642725 ED On-Demand Anodyne NAMPT 36 42 CON(C)CCNC(=O)CCCCCc1ccc(O)cc1 ZINC000880642741 CE On-Demand Anodyne GRIA1 50 37 CON(C)CCNC(=O)CCCCCc1ccc(O)cc1 ZINC000880642741 CE On-Demand Anodyne FAAH 19 41 CON(C)CCNC(=O)CCCOCc1ccccc1 ZINC000880642757 CD On-Demand Anodyne LTA4H 28 41 CON(C)CCNC(=O)Cc1cccc(NS(C)(=O)=O)c1 ZINC000880642767 DC On-Demand Anodyne RAF1 17 43 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne MAOB 44 42 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne PTGER3 54 40 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne MTNR1A 35 44 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne MTNR1B 29 44 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne FFAR1 36 43 CON(C)CCNC(=O)Cc1cccc(OCc2cccc(C)c2)c1 ZINC000880642779 EF On-Demand Anodyne CRTM 40 34 CON(C)CCNC(=O)Cc1cccc(OCc2ccccc2C)c1 ZINC000880642785 EF On-Demand Anodyne MAOB 27 41 CON(C)CCNC(=O)Cc1cccc(OCc2ccccc2C)c1 ZINC000880642785 EF On-Demand Anodyne MTNR1A 52 41 CON(C)CCNC(=O)Cc1cccc(OCc2ccccc2C)c1 ZINC000880642785 EF On-Demand Anodyne MTNR1B 42 41 CON(C)CCNC(=O)Cc1cccc(OCc2ccccc2C)c1 ZINC000880642785 EF On-Demand Anodyne CRTM 47 38 CON(C)CCNC(=O)Cc1cccc(OCc2ccccc2C)c1 ZINC000880642785 EF On-Demand Anodyne PDS 44 33 CON(C)CCNC(=O)CCc1nc2cc(C(F)(F)F)ccc2s1 ZINC000880642787 FF On-Demand Anodyne AKR1B1 15 44 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880642790 EC On-Demand Anodyne F2 41 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880642790 EC On-Demand Anodyne PREP 27 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880642790 EC On-Demand Anodyne NOS2 20 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880642790 EC On-Demand Anodyne TMPRSS11D 45 32 CON(C)CCNC(=O)[C@@H](Sc1ccccc1)C(C)C ZINC000880642791 CE On-Demand Anodyne NPR 47 33 CON(C)CCNC(=O)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880642821 DC On-Demand Anodyne FKBP1A 18 41 CON(C)CCNC(=O)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880642821 DC On-Demand Anodyne ACHE 15 41 CON(C)CCNC(=O)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880642821 DC On-Demand Anodyne SLC6A1 95 35 CON(C)CCNC(=O)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880642821 DC On-Demand Anodyne CHRNA7 40 36 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne HTR1A 138 57 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne DRD2 99 50 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne DRD1 20 41 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne DRD4 74 48 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne ADRA1D 63 52 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne HTR2A 81 50 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne HTR2C 43 48 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne SLC6A4 21 41 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne ADRA1A 82 52 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne ADRA1B 54 52 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne DRD3 125 50 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne HTR4 24 42 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne DRD5 17 43 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne HTR7 155 51 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne SIGMAR1 25 45 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne CACNA1G 25 43 CON(C)CCNC(=O)CCCN1CCN(c2ccccc2)CC1 ZINC000880642834 ED On-Demand Anodyne CYP2J2 44 31 CON(C)CCNC(=O)CCNC(=O)c1n[nH]c2ccccc12 ZINC000880642835 DC On-Demand Anodyne ITK 15 41 CON(C)CCNC(=O)[C@@H]1CCC(=O)N(C)[C@@H]1c1ccccc1 ZINC000880642855 DD On-Demand Anodyne P2RX7 20 40 CON(C)CCNC(=O)[C@@H]1CCC(=O)N(C)[C@H]1c1ccccc1 ZINC000880642860 DD On-Demand Anodyne P2RX7 20 40 CON(C)CCNC(=O)C1CCN(C(=O)N(C)Cc2ccccc2)CC1 ZINC000880642937 FD On-Demand Anodyne TACR1 23 43 CON(C)CCNC(=O)C1CCN(C(=O)N(C)Cc2ccccc2)CC1 ZINC000880642937 FD On-Demand Anodyne CCR5 17 40 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne SIGMAR1 18 42 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne SCN2A 20 42 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne MTNR1A 44 45 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne MTNR1B 44 45 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne FAAH 34 40 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne CAPN2 27 41 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne AMP1_PLAFQ 33 50 CON(C)CCNC(=O)C(=O)NCCCc1ccccc1 ZINC000880642943 CC On-Demand Anodyne CRTM 50 40 CON(C)CCNC(=O)[C@@H]1CCCN1c1ccc(C#N)cc1 ZINC000880642945 DD On-Demand Mild GPBAR1 30 45 CON(C)CCNC(=O)Cc1cn(C)c2ccccc12 ZINC000880642960 CD On-Demand Anodyne MTNR1A 16 42 COCCOc1ncccc1C(=O)NCCN(C)OC ZINC000880642989 CC On-Demand Anodyne POLR1A 32 40 CON(C)CCNC(=O)C[C@H](c1ccccc1)C(C)C ZINC000880642990 CE On-Demand Anodyne KCNA5 16 43 CON(C)CCNC(=O)C[C@@H](c1ccccc1)C(C)C ZINC000880642991 CE On-Demand Anodyne KCNA5 16 43 CON(C)CCNC(=O)CNC(=O)c1ccc(C#N)cc1 ZINC000880643002 CB On-Demand Mild CTRB_BOVIN 45 34 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(Cl)cc1Cl ZINC000880643013 DF On-Demand Anodyne UGCG 20 43 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(Cl)cc1Cl ZINC000880643013 DF On-Demand Anodyne MC4R 53 38 CON(C)CCNC(=O)[C@H](C)Cc1ccc(Cl)cc1Cl ZINC000880643014 DF On-Demand Anodyne UGCG 20 43 CON(C)CCNC(=O)[C@H](C)Cc1ccc(Cl)cc1Cl ZINC000880643014 DF On-Demand Anodyne MC4R 53 38 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne ACE 19 41 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne MME 58 42 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne PAPA1_CARPA 24 43 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne CTSL 15 43 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne NPY5R 15 40 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne ACE2 53 41 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)cc1 ZINC000880643032 CD On-Demand Anodyne LEF 64 36 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne ACE 19 41 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne MME 58 42 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne PAPA1_CARPA 24 43 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne CTSL 15 43 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne NPY5R 15 40 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne ACE2 53 41 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)cc1 ZINC000880643033 CD On-Demand Anodyne LEF 64 36 CON(C)CCNC(=O)CNC(=O)c1cc(-c2ccccc2)on1 ZINC000880643038 EC On-Demand Anodyne HDAC10 17 53 COc1ccc(CC(=O)NCCN(C)OC)cc1[N+](=O)[O-] ZINC000880643040 CC On-Demand Bother MTNR1B 15 40 CON(C)CCNC(=O)[C@H](C)c1c(Cl)cccc1Cl ZINC000880643044 DF On-Demand Anodyne CXCL8 51 45 CON(C)CCNC(=O)[C@@H](C)c1c(Cl)cccc1Cl ZINC000880643045 DF On-Demand Anodyne CXCL8 51 45 CON(C)CCNC(=O)Cc1cccc(OCC(F)(F)F)c1 ZINC000880643069 DD On-Demand Anodyne MTNR1A 40 40 CON(C)CCNC(=O)Cc1cccc(OCC(F)(F)F)c1 ZINC000880643069 DD On-Demand Anodyne MTNR1B 30 40 CON(C)CCNC(=O)Cc1cccc(OCC(F)(F)F)c1 ZINC000880643069 DD On-Demand Anodyne CRTM 41 35 CON(C)CCNC(=O)Cc1cccc(OCC(F)(F)F)c1 ZINC000880643069 DD On-Demand Anodyne PDS 63 37 CON(C)CCNC(=O)CCCc1csc2ccccc12 ZINC000880643071 DF On-Demand Anodyne MTNR1A 29 50 CON(C)CCNC(=O)CCCc1csc2ccccc12 ZINC000880643071 DF On-Demand Anodyne FFAR2 54 34 CON(C)CCNC(=O)[C@@H](C)c1cccc(C)c1 ZINC000880643090 CD On-Demand Anodyne TRPV1 15 42 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne ACHE 17 43 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne HRH2 30 42 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne UPP1 51 40 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne MTNR1A 66 50 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne MTNR1B 55 45 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne ROCK2 17 40 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne PLA2G4B 30 43 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne CRTM 51 36 CCCOc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643095 CD On-Demand Anodyne PDS 60 33 COc1cc2c(cc1OC)CN(C(=O)CCC(=O)NCCN(C)OC)CC2 ZINC000880643096 GC On-Demand Anodyne ABCB1 15 48 CON(C)CCNC(=O)CCCOc1ccc2c(c1)OCO2 ZINC000880643101 DD On-Demand Anodyne EDNRB 72 40 CON(C)CCNC(=O)CCCOc1ccc2c(c1)OCO2 ZINC000880643101 DD On-Demand Anodyne EDNRA 73 41 CON(C)CCNC(=O)CCCOc1ccc2c(c1)OCO2 ZINC000880643101 DD On-Demand Anodyne BMP1 53 38 CON(C)CCNC(=O)CCCOc1ccc2c(c1)OCO2 ZINC000880643101 DD On-Demand Anodyne MTNR1A 52 38 CON(C)CCNC(=O)CCCOc1ccc2c(c1)OCO2 ZINC000880643101 DD On-Demand Anodyne DYRK2 41 34 CON(C)CCNC(=O)Cc1c[nH]c2cc(Br)ccc12 ZINC000880643123 EE On-Demand Anodyne TPR 17 54 COc1cccc(C(=O)NCCN(C)OC)n1 ZINC000880643127 BC On-Demand Anodyne ALS 61 31 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880643132 EC On-Demand Anodyne SLC6A1 55 33 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880643132 EC On-Demand Anodyne CPT1A 123 46 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880643132 EC On-Demand Anodyne CPT2 48 38 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880643132 EC On-Demand Anodyne ACKR3 62 35 CON(C)CCNC(=O)C[C@H](C)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880643141 FE On-Demand Anodyne GPR119 32 48 CON(C)CCNC(=O)C[C@@H](C)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880643142 FE On-Demand Anodyne GPR119 32 48 CC[C@@H](C)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880643144 CE On-Demand Anodyne SCN2A 16 41 CC[C@@H](C)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880643144 CE On-Demand Anodyne UTS2 43 34 CON(C)CCNC(=O)Cc1coc2cc(F)ccc12 ZINC000880643148 CD On-Demand Anodyne MTNR1A 23 40 CON(C)CCNC(=O)CN(C)c1ccccc1[N+](=O)[O-] ZINC000880643149 CC On-Demand Bother COLA 70 33 CON(C)CCNC(=O)[C@H](C)c1ccc(Cl)c(Cl)c1 ZINC000880643162 DF On-Demand Anodyne TRPV1 57 38 CON(C)CCNC(=O)[C@@H](C)c1ccc(Cl)c(Cl)c1 ZINC000880643163 DF On-Demand Anodyne TRPV1 57 38 CON(C)CCNC(=O)[C@@H](CNC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643170 FD On-Demand Anodyne PAPA1_CARPA 38 42 CON(C)CCNC(=O)[C@@H](CNC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643170 FD On-Demand Anodyne CTSK 17 43 CON(C)CCNC(=O)[C@@H](CNC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643170 FD On-Demand Anodyne FPR1 47 37 COc1ccccc1-c1nn(C)cc1C(=O)NCCN(C)OC ZINC000880643180 DD On-Demand Anodyne DRD2 23 43 COc1ccccc1-c1nn(C)cc1C(=O)NCCN(C)OC ZINC000880643180 DD On-Demand Anodyne DRD4 19 40 COc1ccccc1-c1nn(C)cc1C(=O)NCCN(C)OC ZINC000880643180 DD On-Demand Anodyne DRD3 37 40 CON(C)CCNC(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643193 FE On-Demand Anodyne PAPA1_CARPA 43 44 CON(C)CCNC(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643193 FE On-Demand Anodyne CTSK 21 45 CON(C)CCNC(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643193 FE On-Demand Anodyne CTSL 15 44 CON(C)CCNC(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643193 FE On-Demand Anodyne TACR3 18 40 CON(C)CCNC(=O)[C@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643193 FE On-Demand Anodyne FPR1 49 38 CON(C)CCNC(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643194 FE On-Demand Anodyne PAPA1_CARPA 43 44 CON(C)CCNC(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643194 FE On-Demand Anodyne CTSK 21 45 CON(C)CCNC(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643194 FE On-Demand Anodyne CTSL 15 44 CON(C)CCNC(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643194 FE On-Demand Anodyne TACR3 18 40 CON(C)CCNC(=O)[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643194 FE On-Demand Anodyne FPR1 49 38 CON(C)CCNC(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643195 FE On-Demand Anodyne PAPA1_CARPA 43 44 CON(C)CCNC(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643195 FE On-Demand Anodyne CTSK 21 45 CON(C)CCNC(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643195 FE On-Demand Anodyne CTSL 15 44 CON(C)CCNC(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643195 FE On-Demand Anodyne TACR3 18 40 CON(C)CCNC(=O)[C@@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643195 FE On-Demand Anodyne FPR1 49 38 CON(C)CCNC(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643196 FE On-Demand Anodyne PAPA1_CARPA 43 44 CON(C)CCNC(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643196 FE On-Demand Anodyne CTSK 21 45 CON(C)CCNC(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643196 FE On-Demand Anodyne CTSL 15 44 CON(C)CCNC(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643196 FE On-Demand Anodyne TACR3 18 40 CON(C)CCNC(=O)[C@H](C)[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880643196 FE On-Demand Anodyne FPR1 49 38 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccc2)CC1 ZINC000880643208 EC On-Demand Anodyne HTR1A 20 42 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccc2)CC1 ZINC000880643208 EC On-Demand Anodyne DRD3 21 40 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccc2)CC1 ZINC000880643208 EC On-Demand Anodyne SSTR1 48 46 CON(C)CCNC(=O)COc1ccc2c(c1)CCCC2 ZINC000880643228 CD On-Demand Anodyne MTNR1A 46 39 COCCCOc1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880643230 CD On-Demand Anodyne LTA4H 23 40 COCCCOc1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880643230 CD On-Demand Anodyne PLA2G4B 41 35 COCCCOc1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880643230 CD On-Demand Anodyne ESRRG 43 31 COCCCOc1cccc(C(=O)NCCN(C)OC)c1 ZINC000880643231 CD On-Demand Anodyne DRD4 52 40 COCCCOc1cccc(C(=O)NCCN(C)OC)c1 ZINC000880643231 CD On-Demand Anodyne DRD3 15 45 COCCCOc1cccc(C(=O)NCCN(C)OC)c1 ZINC000880643231 CD On-Demand Anodyne MTNR1A 38 52 COCCCOc1cccc(C(=O)NCCN(C)OC)c1 ZINC000880643231 CD On-Demand Anodyne MTNR1B 32 49 COCCCOc1cccc(C(=O)NCCN(C)OC)c1 ZINC000880643231 CD On-Demand Anodyne TAAR1 15 41 CON(C)CCNC(=O)[C@@]1(C)CCc2ccccc2C1 ZINC000880643250 CD On-Demand Anodyne MME 15 47 CON(C)CCNC(=O)Cc1ccncc1 ZINC000880643261 BC On-Demand Anodyne CA5B 18 47 CON(C)CCNC(=O)Cc1ccncc1 ZINC000880643261 BC On-Demand Anodyne CA5A 16 47 CON(C)CCNC(=O)Cc1ccc(S(=O)(=O)CC(F)(F)F)cc1 ZINC000880643277 FD On-Demand Anodyne CA9 22 43 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne FCER2 42 35 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CTSK 40 55 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CTSL 25 52 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CAPNS1 49 32 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CTSS 17 40 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CAPN1 62 39 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne CAPN2 91 36 CON(C)CCNC(=O)[C@@H](CC(C)C)c1ccccc1 ZINC000880643278 CE On-Demand Anodyne NPR 77 37 CON(C)CCNC(=O)CCCN(C)C1=NS(=O)(=O)c2ccccc21 ZINC000880643285 FC On-Demand Anodyne KCNA3 35 49 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncnc3sccc23)C1 ZINC000880643287 ED On-Demand Anodyne SIRT3 55 31 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncnc3sccc23)C1 ZINC000880643287 ED On-Demand Anodyne SIRT2 50 31 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncnc3sccc23)C1 ZINC000880643287 ED On-Demand Anodyne SIRT1 49 31 CON(C)CCNC(=O)Cc1ccc(NC(=O)C2CC2)cc1 ZINC000880643295 DD On-Demand Anodyne MTNR1A 19 45 CON(C)CCNC(=O)Cc1ccc(NC(=O)C2CC2)cc1 ZINC000880643295 DD On-Demand Anodyne MTNR1B 15 45 CON(C)CCNC(=O)Cc1cccc([N+](=O)[O-])c1C ZINC000880643299 CD On-Demand Bother COLA 111 35 CNC(=O)COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643320 DB On-Demand Anodyne UPP1 48 32 CNC(=O)COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643320 DB On-Demand Anodyne MTNR1A 47 42 CNC(=O)COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643320 DB On-Demand Anodyne MTNR1B 38 42 CNC(=O)COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643320 DB On-Demand Anodyne CRTM 49 38 CNC(=O)COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880643320 DB On-Demand Anodyne PDS 41 33 CON(C)CCNC(=O)CCCc1cccc(Br)c1 ZINC000880643345 EE On-Demand Anodyne MTNR1A 41 44 CON(C)CCNC(=O)CCCc1cccc(Br)c1 ZINC000880643345 EE On-Demand Anodyne MTNR1B 33 44 CON(C)CCNC(=O)CCCc1cccc(Br)c1 ZINC000880643345 EE On-Demand Anodyne CRTM 46 36 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne EDNRB 49 35 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne TACR1 18 45 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MC4R 35 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne CCKAR 74 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MPO 52 37 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne BRS3 27 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne NMBR 16 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MC3R 48 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MC5R 48 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne GRPR 68 38 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne GHSR 15 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MC1R 71 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne MMP1 18 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2cc(F)ccc12)NC(C)=O ZINC000880643351 FC On-Demand Anodyne KISS1R 69 37 CCOC(=O)N[C@H](C(=O)NCCN(C)OC)C(C)C ZINC000880643356 CC On-Demand Anodyne HLA-DRB1 63 40 CCOC(=O)N[C@@H](C(=O)NCCN(C)OC)C(C)C ZINC000880643357 CC On-Demand Anodyne HLA-DRB1 63 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)c(OC)c1 ZINC000880643358 FC On-Demand Anodyne F2 24 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)c(OC)c1 ZINC000880643358 FC On-Demand Anodyne ACKR3 43 30 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)c(OC)c1 ZINC000880643359 FC On-Demand Anodyne F2 24 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)c(OC)c1 ZINC000880643359 FC On-Demand Anodyne ACKR3 43 30 CON(C)CCNC(=O)Cc1csc2ccccc12 ZINC000880643363 CE On-Demand Anodyne FFAR2 51 34 CCCCCCC(=O)NCCN(C)OC ZINC000880643374 BD On-Demand Anodyne CNR1 17 57 CCCCCCC(=O)NCCN(C)OC ZINC000880643374 BD On-Demand Anodyne NOD1 59 39 CCCCCCC(=O)NCCN(C)OC ZINC000880643374 BD On-Demand Anodyne CQSS 54 33 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880643380 EC On-Demand Anodyne F2 41 39 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880643380 EC On-Demand Anodyne PREP 75 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880643380 EC On-Demand Anodyne XIAP 23 46 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne F2 71 43 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne ACE 42 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne FKBP1A 40 45 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne CELA1 40 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne ELANE 63 39 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne TACR1 21 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne TRY1_BOVIN 78 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne DPP4 16 46 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne PREP 96 46 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne LGMN 51 38 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne XIAP 53 46 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne BRCA1 51 32 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne TMPRSS11D 69 37 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880643383 DC On-Demand Anodyne ACKR3 47 33 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne HTR1A 20 42 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne DRD2 36 43 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne DRD4 75 47 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne ACHE 45 45 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne LTA4H 25 45 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne SIGMAR1 68 45 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne BCHE 16 40 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne FAAH 20 42 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne MCHR1 15 42 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne CACNA1G 40 37 CON(C)CCNC(=O)CN1CCN(Cc2ccccc2)CC1 ZINC000880643388 DC On-Demand Anodyne NPFFR1 43 38 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CTSD 28 41 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne PGC 23 41 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne PAPA1_CARPA 53 47 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CTSK 52 64 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CTSL 34 46 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne PGA 25 41 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CAPNS1 54 33 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne ECE1 37 40 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne HLA-DRB1 25 43 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne REN 42 43 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne REN1 21 40 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CTSS 25 64 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CAPN1 64 58 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne CAPN2 85 37 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne POLG_HCV1 26 44 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne FPR1 64 47 CON(C)CCNC(=O)[C@@H](CC(C)C)NC(=O)OC(C)(C)C ZINC000880643390 DD On-Demand Anodyne NPR 70 37 CON(C)CCNC(=O)Cc1ccc(F)cc1F ZINC000880643399 CD On-Demand Anodyne P2RX7 45 44 CON(C)CCNC(=O)[C@@H](C)c1cccc(Cl)c1 ZINC000880643402 CE On-Demand Anodyne TRPV1 17 41 CON(C)CCNC(=O)[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000880643408 DC On-Demand Anodyne TRPV1 98 36 CON(C)CCNC(=O)Cc1ccc(F)cc1Cl ZINC000880643411 CD On-Demand Anodyne P2RX7 80 48 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880643413 FD On-Demand Anodyne TRPV1 28 46 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880643413 FD On-Demand Anodyne RBP4 21 43 CON(C)CCNC(=O)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880643413 FD On-Demand Anodyne GPBAR1 25 45 CON(C)CCNC(=O)Cn1c(-c2scnc2C)nc2ccccc21 ZINC000880643435 FE On-Demand Anodyne IMDH_CRYPV 39 42 CON(C)CCNC(=O)[C@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643438 GD On-Demand Anodyne MMP13 19 43 CON(C)CCNC(=O)[C@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643438 GD On-Demand Anodyne MMP2 19 44 CON(C)CCNC(=O)[C@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643438 GD On-Demand Anodyne MMP9 16 43 CON(C)CCNC(=O)[C@@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643440 GD On-Demand Anodyne MMP13 19 43 CON(C)CCNC(=O)[C@@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643440 GD On-Demand Anodyne MMP2 19 44 CON(C)CCNC(=O)[C@@H](C)CS(=O)(=O)c1ccc(Br)cc1 ZINC000880643440 GD On-Demand Anodyne MMP9 16 43 CON(C)CCNC(=O)CCCC(C)=O ZINC000880643465 BC On-Demand Anodyne PAOX 26 40 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(F)c(Br)c1 ZINC000880643466 EE On-Demand Anodyne LEF 73 34 CON(C)CCNC(=O)[C@H](C)Cc1ccc(F)c(Br)c1 ZINC000880643468 EE On-Demand Anodyne LEF 73 34 CON(C)CCNC(=O)COc1ccc(O)cc1 ZINC000880643472 CC On-Demand Anodyne ESRRG 43 32 CON(C)CCNC(=O)CCCCC(=O)c1ccccc1 ZINC000880643493 CE On-Demand Anodyne HDAC8 33 45 CON(C)CCNC(=O)CCCCC(=O)c1ccccc1 ZINC000880643493 CE On-Demand Anodyne HDAC1 17 52 CON(C)CCNC(=O)CCCCC(=O)c1ccccc1 ZINC000880643493 CE On-Demand Anodyne HDAC2 16 40 CON(C)CCNC(=O)[C@@H](C)NC(=O)c1cccc(Cl)c1Cl ZINC000880643511 ED On-Demand Anodyne ECR 45 45 CON(C)CCNC(=O)[C@H](C)NC(=O)c1cccc(Cl)c1Cl ZINC000880643514 ED On-Demand Anodyne ECR 45 45 CON(C)CCNC(=O)CNC(=O)c1ccccc1C(F)(F)F ZINC000880643524 ED On-Demand Anodyne ECR 18 42 CON(C)CCNC(=O)CNC(=O)c1ccccc1C(F)(F)F ZINC000880643524 ED On-Demand Anodyne E3UJZ5_SPOLI 19 42 CON(C)CCNC(=O)CNC(=O)c1ccccc1C(F)(F)F ZINC000880643524 ED On-Demand Anodyne KCNK3 18 40 CON(C)CCNC(=O)CCc1c[nH]c2cc(C)ccc12 ZINC000880643528 CE On-Demand Anodyne MTNR1A 15 47 COc1cc2c(cc1OC)CN(CC(=O)NCCN(C)OC)CC2 ZINC000880643530 EC On-Demand Anodyne SLC18A2 40 33 COc1cc2c(cc1OC)CN(CC(=O)NCCN(C)OC)CC2 ZINC000880643530 EC On-Demand Anodyne ABCB1B 67 39 COc1cc2c(cc1OC)CN(CC(=O)NCCN(C)OC)CC2 ZINC000880643530 EC On-Demand Anodyne ABCB1 25 46 CON(C)CCNC(=O)Cc1ccc(C)cc1Cl ZINC000880643537 CD On-Demand Anodyne P2RX7 47 38 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)cc1 ZINC000880643551 DD On-Demand Anodyne CYP11B1 15 52 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)cc1 ZINC000880643551 DD On-Demand Anodyne DRD4 42 32 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)cc1 ZINC000880643551 DD On-Demand Anodyne SCN2A 27 43 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)cc1 ZINC000880643551 DD On-Demand Anodyne CYP11B2 29 52 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)cc1 ZINC000880643551 DD On-Demand Anodyne SCN10A 63 44 CON(C)CCNC(=O)[C@@H](C)c1ccc(S(=O)(=O)N(C)C)cc1 ZINC000880643555 EC On-Demand Anodyne BMP1 24 40 CON(C)CCNC(=O)[C@@H](C)c1ccc(S(=O)(=O)N(C)C)cc1 ZINC000880643555 EC On-Demand Anodyne TRPV1 81 34 CON(C)CCNC(=O)CCCNC(=O)c1cccnc1 ZINC000880643556 CC On-Demand Anodyne TBXAS1 68 42 CON(C)CCNC(=O)CCCNC(=O)c1cccnc1 ZINC000880643556 CC On-Demand Anodyne PTAFR 22 44 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccn2)CC1 ZINC000880643557 EC On-Demand Anodyne HTR1A 15 44 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccn2)CC1 ZINC000880643557 EC On-Demand Anodyne DRD4 29 44 CON(C)CCNC(=O)CCC(=O)N1CCN(c2ccccn2)CC1 ZINC000880643557 EC On-Demand Anodyne SSTR1 48 39 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne GRIN2B 20 42 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne TGM2 45 40 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne NPR 57 34 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne F13A1 40 40 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne Q6PRC7_IXORI 38 40 CON(C)CCNC(=O)CN1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880643567 FC On-Demand Anodyne SLC12A5 46 38 CON(C)CCNC(=O)[C@@H]1Cc2ccccc21 ZINC000880643575 BC On-Demand Anodyne ADAM9 41 32 CON(C)CCNC(=O)COc1cccc(OCC(C)C)c1 ZINC000880643580 DD On-Demand Anodyne MTNR1A 49 40 CON(C)CCNC(=O)COc1cccc(OCC(C)C)c1 ZINC000880643580 DD On-Demand Anodyne MTNR1B 42 43 CON(C)CCNC(=O)COc1cccc(OCC(C)C)c1 ZINC000880643580 DD On-Demand Anodyne PDS 72 37 CCOc1ccccc1Oc1ccccc1C(=O)NCCN(C)OC ZINC000880643601 EG On-Demand Anodyne KCNA3 40 42 CCOc1ccccc1Oc1ccccc1C(=O)NCCN(C)OC ZINC000880643601 EG On-Demand Anodyne HCN1 83 40 CCOc1ccccc1Oc1ccccc1C(=O)NCCN(C)OC ZINC000880643601 EG On-Demand Anodyne HCN4 59 39 CCOc1ccccc1Oc1ccccc1C(=O)NCCN(C)OC ZINC000880643601 EG On-Demand Anodyne KCNK3 46 44 CCOc1ccccc1Oc1ccccc1C(=O)NCCN(C)OC ZINC000880643601 EG On-Demand Anodyne KCNK9 39 44 COc1ccc(OCC(=O)NCCN(C)OC)cc1C ZINC000880643602 CC On-Demand Anodyne MTNR1A 49 41 COc1ccc(OCC(=O)NCCN(C)OC)cc1C ZINC000880643602 CC On-Demand Anodyne MTNR1B 38 41 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne HTR1A 15 46 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne HTR1D 64 47 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne HTR1B 38 46 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne MPO 74 45 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne HTR5A 19 43 CON(C)CCNC(=O)CCc1c[nH]c2ccc(C)cc12 ZINC000880643605 CE On-Demand Anodyne MTNR1A 18 54 CON(C)CCNC(=O)CCc1ncc(-c2ccc(Cl)cc2Cl)o1 ZINC000880643611 FG On-Demand Anodyne ALPL 42 37 CON(C)CCNC(=O)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880643618 FD On-Demand Anodyne LTA4H 36 45 CON(C)CCNC(=O)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880643618 FD On-Demand Anodyne CPT1A 54 34 CON(C)CCNC(=O)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880643618 FD On-Demand Anodyne CACNA1G 35 44 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne F2 84 47 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne PLG 33 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne PRSS1 29 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne ACE 52 48 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne FKBP1A 73 47 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne OPRM1 34 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne OPRD1 21 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CELA1 52 57 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne ELANE 53 46 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne TACR1 23 43 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CMA1 36 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CTRA_BOVIN 66 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne TRY1_BOVIN 100 43 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne NTSR1 89 35 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne NTSR2 88 33 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CTSG 45 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CTSK 19 55 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne HLA-A 57 34 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne DPP4 17 43 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne PREP 88 57 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne CELA2A 54 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne LGMN 106 55 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne SORT1 48 33 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne GHSR 18 47 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne ACE2 22 43 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne KLK5 47 51 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne XIAP 62 47 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne BRCA1 62 33 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne SLC12A5 68 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880643655 ED On-Demand Anodyne TMPRSS11D 74 42 CON(C)CCNC(=O)CSc1nnc(-c2ccco2)n1Cc1ccco1 ZINC000880643679 GD On-Demand Anodyne HCRTR2 17 53 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne F2 23 52 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne NQO2 27 41 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne MMP13 19 60 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne TRY2_BOVIN 67 52 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne MTNR1A 38 41 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne MMP2 17 60 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne MMP14 16 46 CON(C)CCNC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 ZINC000880643680 FC On-Demand Anodyne MMP12 21 46 CCOc1cccnc1C(=O)NCCN(C)OC ZINC000880643684 CC On-Demand Anodyne MAP1 31 40 CCOc1cccnc1C(=O)NCCN(C)OC ZINC000880643684 CC On-Demand Anodyne HCN1 46 31 CON(C)CCNC(=O)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880643698 FC On-Demand Anodyne FKBP1A 22 47 CON(C)CCNC(=O)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880643698 FC On-Demand Anodyne MMP13 18 43 CON(C)CCNC(=O)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880643698 FC On-Demand Anodyne MMP3 15 43 CON(C)CCNC(=O)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880643698 FC On-Demand Anodyne MMP7 23 43 CON(C)CCNC(=O)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880643698 FC On-Demand Anodyne MMP1 22 43 CON(C)CCNC(=O)Cc1csc(NC(=O)c2ccccc2)n1 ZINC000880643711 ED On-Demand Anodyne CPT1A 29 45 CON(C)CCNC(=O)CCc1c(C)n[nH]c1C ZINC000880643712 CC On-Demand Anodyne HAO2 49 33 CON(C)CCNC(=O)COc1cccc(C(C)C)c1 ZINC000880643734 CD On-Demand Anodyne MTNR1A 49 40 CON(C)CCNC(=O)COc1cccc(C(C)C)c1 ZINC000880643734 CD On-Demand Anodyne MTNR1B 41 40 CON(C)CCNC(=O)COc1cccc(C(C)C)c1 ZINC000880643734 CD On-Demand Anodyne PDS 28 43 CON(C)CCNC(=O)CCCC[C@@H](C)C(C)=O ZINC000880643774 CD On-Demand Anodyne NOD1 53 38 CON(C)CCNC(=O)CCCC[C@H](C)C(C)=O ZINC000880643775 CD On-Demand Anodyne NOD1 53 38 CON(C)CCNC(=O)C[C@H](Cc1ccccc1)c1ccccc1 ZINC000880643803 EG On-Demand Anodyne MME 59 39 CON(C)CCNC(=O)C[C@@H](Cc1ccccc1)c1ccccc1 ZINC000880643806 EG On-Demand Anodyne MME 59 39 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880643810 FD On-Demand Anodyne CACNA1G 40 39 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880643810 FD On-Demand Anodyne GPBAR1 20 44 CON(C)CCNC(=O)[C@H](C)NS(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000880643821 GC On-Demand Anodyne CACNA1B 47 35 CON(C)CCNC(=O)[C@@H](C)NS(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000880643827 GC On-Demand Anodyne CACNA1B 47 35 CON(C)CCNC(=O)CCCc1ccccc1Br ZINC000880643843 EE On-Demand Anodyne MTNR1A 42 40 CON(C)CCNC(=O)C1(c2ccc(Cl)c(Cl)c2)CCC1 ZINC000880643847 EG On-Demand Anodyne SLC6A2 15 43 CON(C)CCNC(=O)C1(c2ccc(Cl)c(Cl)c2)CCC1 ZINC000880643847 EG On-Demand Anodyne SLC6A3 15 43 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NCCN(C)OC ZINC000880643852 ED On-Demand Anodyne F2 43 37 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NCCN(C)OC ZINC000880643852 ED On-Demand Anodyne FKBP1A 19 41 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NCCN(C)OC ZINC000880643852 ED On-Demand Anodyne TRY1_BOVIN 43 34 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NCCN(C)OC ZINC000880643852 ED On-Demand Anodyne HCN1 66 39 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NCCN(C)OC ZINC000880643852 ED On-Demand Anodyne HCN4 58 39 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NCCN(C)OC ZINC000880643853 ED On-Demand Anodyne F2 43 37 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NCCN(C)OC ZINC000880643853 ED On-Demand Anodyne FKBP1A 19 41 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NCCN(C)OC ZINC000880643853 ED On-Demand Anodyne TRY1_BOVIN 43 34 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NCCN(C)OC ZINC000880643853 ED On-Demand Anodyne HCN1 66 39 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NCCN(C)OC ZINC000880643853 ED On-Demand Anodyne HCN4 58 39 CON(C)CCNC(=O)C1CCN(C(=O)c2ccoc2)CC1 ZINC000880643855 DC On-Demand Anodyne L3MBTL3 46 36 COCC[C@@H](Cc1cccc(Br)c1)C(=O)NCCN(C)OC ZINC000880643856 FE On-Demand Anodyne MME 30 41 COCC[C@H](Cc1cccc(Br)c1)C(=O)NCCN(C)OC ZINC000880643857 FE On-Demand Anodyne MME 30 41 CON(C)CCNC(=O)Cn1c(C)nc2ccccc2c1=O ZINC000880643866 DC On-Demand Anodyne AVPR1B 48 40 CON(C)CCNC(=O)Cn1c(C)nc2ccccc2c1=O ZINC000880643866 DC On-Demand Anodyne POLR1A 45 38 COCCOc1ccc(Cl)cc1C(=O)NCCN(C)OC ZINC000880643870 DD On-Demand Anodyne ALPL 31 42 CON(C)CCNC(=O)Cc1ccc(C(C)(C)C)cc1 ZINC000880643880 CE On-Demand Anodyne TRPV1 37 47 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1 ZINC000880643899 GD On-Demand Anodyne SLC6A1 42 33 CON(C)CCNC(=O)Cc1c(C)n[nH]c1C ZINC000880643930 BC On-Demand Anodyne P2RX7 15 53 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000880643935 CC On-Demand Anodyne FKBP1A 17 41 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000880643935 CC On-Demand Anodyne CELA1 44 33 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000880643935 CC On-Demand Anodyne TPP2 31 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(C)(C)C ZINC000880643935 CC On-Demand Anodyne XIAP 23 42 CON(C)CCNC(=O)CCCOc1ccc2c(c1)CCC2 ZINC000880643988 DD On-Demand Anodyne NQO2 19 40 CON(C)CCNC(=O)CCCOc1ccc2c(c1)CCC2 ZINC000880643988 DD On-Demand Anodyne MTNR1A 40 38 CON(C)CCNC(=O)CCCOc1cccnc1 ZINC000880643989 CC On-Demand Anodyne LTA4H 17 49 CON(C)CCNC(=O)CCCOc1cccnc1 ZINC000880643989 CC On-Demand Anodyne PTAFR 16 47 CON(C)CCNC(=O)CCCOc1cccnc1 ZINC000880643989 CC On-Demand Anodyne MTNR1A 25 40 CON(C)CCNC(=O)CCCOc1cccnc1 ZINC000880643989 CC On-Demand Anodyne MTNR1B 20 40 CON(C)CCNC(=O)CCCn1cncn1 ZINC000880643991 BB On-Demand Anodyne HIS3 40 39 CON(C)CCNC(=O)[C@@H]1CCCN(S(=O)(=O)c2ccc(C)cc2)C1 ZINC000880644008 FD On-Demand Anodyne EPHX2 26 46 CON(C)CCNC(=O)C[C@@H](NC(=O)c1ccc(O)cc1)c1ccccc1 ZINC000880644012 FD On-Demand Anodyne UTS2 81 43 CON(C)CCNC(=O)C[C@H](NC(=O)c1ccc(O)cc1)c1ccccc1 ZINC000880644013 FD On-Demand Anodyne UTS2 81 43 COc1ccc(O[C@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644020 CD On-Demand Anodyne BMP1 41 37 COc1ccc(O[C@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644020 CD On-Demand Anodyne NQO2 25 44 COc1ccc(O[C@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644020 CD On-Demand Anodyne MTNR1A 77 44 COc1ccc(O[C@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644020 CD On-Demand Anodyne MTNR1B 61 42 COc1ccc(O[C@@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644021 CD On-Demand Anodyne BMP1 41 37 COc1ccc(O[C@@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644021 CD On-Demand Anodyne NQO2 25 44 COc1ccc(O[C@@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644021 CD On-Demand Anodyne MTNR1A 77 44 COc1ccc(O[C@@H](C)C(=O)NCCN(C)OC)cc1 ZINC000880644021 CD On-Demand Anodyne MTNR1B 61 42 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne LSS 16 41 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne MTTP 17 42 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne SLC6A5 31 42 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne EPHX2 35 43 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne MCHR1 18 44 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne SFRP1 22 40 CON(C)CCNC(=O)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880644025 GE On-Demand Anodyne L3MBTL3 69 41 CON(C)CCNC(=O)CSc1nc(C)c(Cc2ccccc2)[nH]1 ZINC000880644031 EE On-Demand Anodyne ENPP1 73 36 CON(C)CCNC(=O)Cn1cc(C(N)=O)c2ccccc21 ZINC000880644049 DC On-Demand Anodyne CNR2 20 40 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne MME 55 36 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne KLK3 45 29 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CTSB 41 39 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne PAPA1_CARPA 55 36 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CTSK 28 40 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CTSL 26 40 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CAPNS1 61 37 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CAPN1 68 41 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne CAPN2 97 38 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne NPR 84 41 CON(C)CCNC(=O)[C@@H](C)OCc1ccccc1 ZINC000880644051 CD On-Demand Anodyne AMP1_PLAFQ 43 37 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne MME 55 36 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne KLK3 45 29 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CTSB 41 39 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne PAPA1_CARPA 55 36 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CTSK 28 40 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CTSL 26 40 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CAPNS1 61 37 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CAPN1 68 41 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne CAPN2 97 38 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne NPR 84 41 CON(C)CCNC(=O)[C@H](C)OCc1ccccc1 ZINC000880644052 CD On-Demand Anodyne AMP1_PLAFQ 43 37 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne ACE 25 56 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne TYR 15 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne SSTR2 67 45 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne OPRM1 16 55 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MME 40 52 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne EDNRB 62 47 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne EDNRA 46 57 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne TACR1 38 59 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MC4R 57 47 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CTSB 24 44 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne PAPA1_CARPA 36 40 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CCKAR 141 56 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CTSL 39 56 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne BRS3 37 60 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne TIMP3 18 55 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne NMBR 48 58 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MC3R 78 45 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MC5R 77 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP2 39 56 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP8 61 55 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne GRIA1 27 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP14 30 53 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne GRPR 88 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne ECE1 74 52 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne LNPEP 22 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne SSTR3 21 40 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP11 102 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne FURIN 24 45 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CCKBR 109 51 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne GHSR 71 50 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CAPN1 22 48 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP9 40 56 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne CAPN2 26 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MC1R 110 45 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP7 24 54 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne MMP1 39 59 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne FPR1 28 49 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne NPR 46 52 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne ADAM12 18 53 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne KISS1R 93 43 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne ERAP2 46 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne PSMB8 28 41 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne TMPRSS6 17 42 CON(C)CCNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000880644057 FD On-Demand Anodyne HPN 22 43 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880644070 ED On-Demand Anodyne SLC6A1 77 36 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880644070 ED On-Demand Anodyne PREP 48 37 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880644070 ED On-Demand Anodyne DPP7 41 36 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880644070 ED On-Demand Anodyne BIRC2 20 46 CON(C)CCNC(=O)[C@@H](C)Oc1ccccc1C#N ZINC000880644081 CC On-Demand Mild ADRB1 45 35 CON(C)CCNC(=O)[C@H](C)Oc1ccccc1C#N ZINC000880644082 CC On-Demand Mild ADRB1 45 35 CON(C)CCNC(=O)CCCc1ccc(Cl)cc1 ZINC000880644083 CE On-Demand Anodyne MMP2 39 40 CON(C)CCNC(=O)CCC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880644091 EE On-Demand Anodyne GPR119 40 44 CON(C)CCNC(=O)C(C)(C)C1CCCCC1 ZINC000880644098 CE On-Demand Anodyne AMY2 49 35 CON(C)CCNC(=O)CC[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880644117 ED On-Demand Anodyne GPR119 31 40 CON(C)CCNC(=O)CC[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880644118 ED On-Demand Anodyne GPR119 31 40 CON(C)CCNC(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C ZINC000880644140 ED On-Demand Anodyne PAPA1_CARPA 46 46 CON(C)CCNC(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C ZINC000880644140 ED On-Demand Anodyne CTSK 22 50 CON(C)CCNC(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C ZINC000880644140 ED On-Demand Anodyne POLG_HCV1 32 49 CON(C)CCNC(=O)[C@@H](CC(F)F)NC(=O)OC(C)(C)C ZINC000880644140 ED On-Demand Anodyne FPR1 47 37 CON(C)CCNC(=O)Cc1ccc(OCc2ccccn2)cc1 ZINC000880644154 ED On-Demand Anodyne CYSLTR1 27 47 CON(C)CCNC(=O)Cc1ccc(OCc2ccccn2)cc1 ZINC000880644154 ED On-Demand Anodyne LPAR1 20 41 CON(C)CCNC(=O)Cc1ccc(OCc2ccccn2)cc1 ZINC000880644154 ED On-Demand Anodyne MTNR1B 16 45 CON(C)CCNC(=O)Cc1ccc(OCc2ccccn2)cc1 ZINC000880644154 ED On-Demand Anodyne LPAR3 23 41 CON(C)CCNC(=O)Cc1ccc(OCc2ccccn2)cc1 ZINC000880644154 ED On-Demand Anodyne SMO 22 45 COCCc1nnc(-c2cccc(C(=O)NCCN(C)OC)c2)o1 ZINC000880644160 ED On-Demand Anodyne DRD4 41 31 CON(C)CCNC(=O)Cc1cccc(NC(=O)OC(C)(C)C)c1 ZINC000880644163 EE On-Demand Anodyne NQO2 25 40 CC[C@@H](CC(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644167 CE On-Demand Anodyne MTNR1A 40 39 CON(C)CCNC(=O)CCc1cc2ccccc2nc1O ZINC000880644168 DD On-Demand Anodyne MTNR1A 39 40 COC(=O)c1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880644169 CC On-Demand Anodyne NQO2 26 41 CCCc1c(C(=O)NCCN(C)OC)cnn1-c1cccc(F)c1 ZINC000880644186 EE On-Demand Anodyne GPR142 40 31 CON(C)CCNC(=O)COc1cccc(NC(=O)C2CC2)c1 ZINC000880644242 DD On-Demand Anodyne MTNR1A 48 49 CON(C)CCNC(=O)COc1cccc(NC(=O)C2CC2)c1 ZINC000880644242 DD On-Demand Anodyne MTNR1B 42 49 CON(C)CCNC(=O)COc1cccc(NC(=O)C2CC2)c1 ZINC000880644242 DD On-Demand Anodyne EPHX2 19 43 COc1ccc([C@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644244 DC On-Demand Anodyne MTNR1A 58 37 COc1ccc([C@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644244 DC On-Demand Anodyne MTNR1B 45 36 COc1ccc([C@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644244 DC On-Demand Anodyne UTS2 36 42 COc1ccc([C@@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644245 DC On-Demand Anodyne MTNR1A 58 37 COc1ccc([C@@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644245 DC On-Demand Anodyne MTNR1B 45 36 COc1ccc([C@@H](CC(=O)NCCN(C)OC)NC(C)=O)cc1 ZINC000880644245 DC On-Demand Anodyne UTS2 36 42 CN(C)C(=O)c1ccc(NC(=O)NOCCO)c(F)c1 ZINC000880644266 CC On-Demand Anodyne MAP2K1 24 40 CON(C)CCNC(=O)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000880644279 CB On-Demand Anodyne INHA 21 43 CON(C)CCNC(=O)CCn1ccnc1 ZINC000880644281 BB On-Demand Anodyne TBXAS1 39 41 CON(C)CCNC(=O)CCn1ccnc1 ZINC000880644281 BB On-Demand Anodyne QPCT 35 41 CON(C)CCNC(=O)Cc1c(C)nn(-c2ccc(F)cc2)c1C ZINC000880644287 ED On-Demand Anodyne P2RX7 46 57 CON(C)CCNC(=O)CCCOc1ccc(Cl)cc1 ZINC000880644291 DE On-Demand Anodyne FDPS 15 42 CON(C)CCNC(=O)CCCOc1ccc(Cl)cc1 ZINC000880644291 DE On-Demand Anodyne LTA4H 26 42 CON(C)CCNC(=O)Cc1ccc(-n2nc(C)cc2C)cc1 ZINC000880644297 DD On-Demand Anodyne ADORA2A 35 41 CON(C)CCNC(=O)[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880644298 CC On-Demand Anodyne INHA 25 50 COc1ccc2c(c1)C[C@@H](C(=O)NCCN(C)OC)CO2 ZINC000880644300 CC On-Demand Anodyne NQO2 32 43 COc1ccc2c(c1)C[C@@H](C(=O)NCCN(C)OC)CO2 ZINC000880644300 CC On-Demand Anodyne MTNR1A 70 57 COc1ccc2c(c1)C[C@@H](C(=O)NCCN(C)OC)CO2 ZINC000880644300 CC On-Demand Anodyne MTNR1B 51 39 COc1ccc2c(c1)C[C@@H](C(=O)NCCN(C)OC)CO2 ZINC000880644300 CC On-Demand Anodyne ROCK2 45 53 COc1ccc2c(c1)C[C@H](C(=O)NCCN(C)OC)CO2 ZINC000880644301 CC On-Demand Anodyne NQO2 32 43 COc1ccc2c(c1)C[C@H](C(=O)NCCN(C)OC)CO2 ZINC000880644301 CC On-Demand Anodyne MTNR1A 70 57 COc1ccc2c(c1)C[C@H](C(=O)NCCN(C)OC)CO2 ZINC000880644301 CC On-Demand Anodyne MTNR1B 51 39 COc1ccc2c(c1)C[C@H](C(=O)NCCN(C)OC)CO2 ZINC000880644301 CC On-Demand Anodyne ROCK2 45 53 COc1cccc([C@@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644312 CD On-Demand Anodyne DRD4 42 32 COc1cccc([C@@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644312 CD On-Demand Anodyne NQO2 25 46 COc1cccc([C@@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644312 CD On-Demand Anodyne TRPV1 17 41 COc1cccc([C@@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644312 CD On-Demand Anodyne MTNR1A 90 46 COc1cccc([C@@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644312 CD On-Demand Anodyne MTNR1B 80 45 COc1cccc([C@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644313 CD On-Demand Anodyne DRD4 42 32 COc1cccc([C@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644313 CD On-Demand Anodyne NQO2 25 46 COc1cccc([C@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644313 CD On-Demand Anodyne TRPV1 17 41 COc1cccc([C@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644313 CD On-Demand Anodyne MTNR1A 90 46 COc1cccc([C@H](C)C(=O)NCCN(C)OC)c1 ZINC000880644313 CD On-Demand Anodyne MTNR1B 80 45 CON(C)CCNC(=O)CS(=O)(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000880644328 GC On-Demand Anodyne DRD4 42 37 CON(C)CCNC(=O)Cc1ccc(O)cc1 ZINC000880644331 BC On-Demand Anodyne GRIA1 45 34 CON(C)CCNC(=O)Cc1ccc(O)cc1 ZINC000880644331 BC On-Demand Anodyne CA9 17 40 CON(C)CCNC(=O)CCc1cccc(C(F)(F)F)c1 ZINC000880644337 DE On-Demand Anodyne TACR1 20 40 CON(C)CCNC(=O)CCc1cccc(C(F)(F)F)c1 ZINC000880644337 DE On-Demand Anodyne MTNR1A 21 42 CON(C)CCNC(=O)CCc1cccc(C(F)(F)F)c1 ZINC000880644337 DE On-Demand Anodyne MTNR1B 18 42 CON(C)CCNC(=O)CCc1cccc(C(F)(F)F)c1 ZINC000880644337 DE On-Demand Anodyne LUXR 15 47 CON(C)CCNC(=O)CCc1cccc(C(F)(F)F)c1 ZINC000880644337 DE On-Demand Anodyne PDS 43 39 CON(C)CCNC(=O)Cc1cccc(OCc2cccnc2)c1 ZINC000880644352 ED On-Demand Anodyne PTAFR 30 41 CON(C)CCNC(=O)Cc1cccc(OCc2cccnc2)c1 ZINC000880644352 ED On-Demand Anodyne MTNR1A 29 40 CON(C)CCNC(=O)Cc1cccc(OCc2cccnc2)c1 ZINC000880644352 ED On-Demand Anodyne MTNR1B 25 40 CON(C)CCNC(=O)COc1cccc(C#N)c1 ZINC000880644358 CC On-Demand Mild MTNR1A 40 40 CON(C)CCNC(=O)COc1cccc(C#N)c1 ZINC000880644358 CC On-Demand Mild MTNR1B 30 40 CON(C)CCNC(=O)[C@@H](c1ccc(F)cc1)C(C)C ZINC000880644381 CE On-Demand Anodyne LEF 42 42 CON(C)CCNC(=O)C1=Cc2cc(F)ccc2OC1 ZINC000880644392 CD On-Demand Anodyne ALOX12 16 45 CON(C)CCNC(=O)[C@@H](C)Oc1cccc(CO)c1 ZINC000880644417 CC On-Demand Anodyne MTNR1A 47 42 CON(C)CCNC(=O)[C@@H](C)Oc1cccc(CO)c1 ZINC000880644417 CC On-Demand Anodyne MTNR1B 43 42 CON(C)CCNC(=O)[C@H](C)Oc1cccc(CO)c1 ZINC000880644418 CC On-Demand Anodyne MTNR1A 47 42 CON(C)CCNC(=O)[C@H](C)Oc1cccc(CO)c1 ZINC000880644418 CC On-Demand Anodyne MTNR1B 43 42 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne ACE 34 40 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne MME 111 42 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne ANPEP 48 37 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne FCER2 41 34 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne PAPA1_CARPA 59 40 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne CPA1 46 36 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne CAPNS1 53 33 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne MMP8 20 40 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne CAPN1 56 40 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne CAPN2 45 36 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne ACE2 42 36 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne NPR 57 38 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne AMP1_PLAFQ 56 42 CON(C)CCNC(=O)[C@@H](F)Cc1ccccc1 ZINC000880644427 CD On-Demand Anodyne NPFFR1 51 31 CON(C)CCNC(=O)CCCc1cc(F)ccc1F ZINC000880644428 CD On-Demand Anodyne MPO 21 42 CON(C)CCNC(=O)Cn1cnc2c(cnn2C)c1=O ZINC000880644440 CA On-Demand Anodyne Q9M629_MAIZE 42 35 CCCCSCC(=O)NCCN(C)OC ZINC000880644449 BD On-Demand Anodyne EST1_PIG 45 39 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne NQO2 24 46 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne MMP13 17 43 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne MTNR1A 61 38 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne MTNR1B 44 37 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne MT-ND1 24 41 COc1ccc(CC(=O)NCc2ccc(C(=O)NCCN(C)OC)cc2)cc1 ZINC000880644460 GD On-Demand Anodyne CA9 24 54 CON(C)CCNC(=O)C[C@@H](NC(N)=O)c1ccccc1C ZINC000880644467 DC On-Demand Anodyne CTSA 65 39 CON(C)CCNC(=O)C[C@H](NC(N)=O)c1ccccc1C ZINC000880644470 DC On-Demand Anodyne CTSA 65 39 CON(C)CCNC(=O)Cc1csc(-c2ccc(C(F)(F)F)cc2)n1 ZINC000880644473 FF On-Demand Anodyne PPARA 19 45 CON(C)CCNC(=O)[C@@H](Oc1ccccc1C#N)C(C)C ZINC000880644480 DD On-Demand Mild ADRB1 43 34 CON(C)CCNC(=O)CCc1cccc(Br)c1 ZINC000880644482 DD On-Demand Anodyne MTNR1A 32 41 CON(C)CCNC(=O)CCc1cccc(Br)c1 ZINC000880644482 DD On-Demand Anodyne MTNR1B 23 41 CON(C)CCNC(=O)CCc1cccc(Br)c1 ZINC000880644482 DD On-Demand Anodyne LUXR 15 44 CON(C)CCNC(=O)C[C@@H](C)NC(=O)c1ccccc1 ZINC000880644491 CC On-Demand Anodyne CTSL 15 42 CON(C)CCNC(=O)C[C@@H](C)NC(=O)c1ccccc1 ZINC000880644491 CC On-Demand Anodyne UTS2 65 36 CON(C)CCNC(=O)C[C@H](C)NC(=O)c1ccccc1 ZINC000880644493 CC On-Demand Anodyne CTSL 15 42 CON(C)CCNC(=O)C[C@H](C)NC(=O)c1ccccc1 ZINC000880644493 CC On-Demand Anodyne UTS2 65 36 CON(C)CCNC(=O)[C@@H](C)c1cccc(C(=O)c2ccccc2)c1 ZINC000880644498 EF On-Demand Anodyne CXCL8 20 56 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne F2 52 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne FKBP1A 20 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne TRY1_BOVIN 51 36 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne PREP 59 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne XIAP 42 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880644541 DC On-Demand Anodyne TMPRSS11D 43 32 CON(C)CCNC(=O)CCc1nc(-c2ccncc2)no1 ZINC000880644544 DC On-Demand Anodyne HCAR2 19 42 CON(C)CCNC(=O)Cc1c(C)nn(-c2ccc(C(F)(F)F)cn2)c1C ZINC000880644554 GE On-Demand Anodyne P2RX7 27 47 COCCOc1cc(C(=O)NCCN(C)OC)nc2ccccc12 ZINC000880644556 ED On-Demand Anodyne BCHE 49 35 COCCOc1cc(C(=O)NCCN(C)OC)nc2ccccc12 ZINC000880644556 ED On-Demand Anodyne POLR1A 39 40 CON(C)CCNC(=O)CCCc1ccc(Cl)c(Cl)c1 ZINC000880644559 DF On-Demand Anodyne CRTM 32 40 COC[C@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880644581 EG On-Demand Anodyne KCNK3 48 43 COC[C@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880644581 EG On-Demand Anodyne KCNK9 43 40 CON(C)CCNC(=O)CCC(=O)c1ccc2c(c1)CCC(=O)N2 ZINC000880644587 ED On-Demand Anodyne HDAC9 19 49 CON(C)CCNC(=O)C[C@H](NC(C)=O)c1ccccc1 ZINC000880644596 CC On-Demand Anodyne UTS2 42 38 CON(C)CCNC(=O)C[C@@H](NC(C)=O)c1ccccc1 ZINC000880644597 CC On-Demand Anodyne UTS2 42 38 COc1ccc2c(=O)c(C(=O)NCCN(C)OC)c[nH]c2c1 ZINC000880644602 DC On-Demand Anodyne NQO2 32 42 COc1ccc2c(=O)c(C(=O)NCCN(C)OC)c[nH]c2c1 ZINC000880644602 DC On-Demand Anodyne MTNR1A 61 42 COc1ccc2c(=O)c(C(=O)NCCN(C)OC)c[nH]c2c1 ZINC000880644602 DC On-Demand Anodyne MTNR1B 45 42 COc1ccc2c(=O)c(C(=O)NCCN(C)OC)c[nH]c2c1 ZINC000880644602 DC On-Demand Anodyne CFTR 34 41 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880644607 CC On-Demand Anodyne PAPA1_CARPA 46 50 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880644607 CC On-Demand Anodyne CTSK 19 47 CON(C)CCNC(=O)Cc1csc(NC(=O)Cc2cccs2)n1 ZINC000880644614 FD On-Demand Anodyne CA5B 31 41 CON(C)CCNC(=O)Cc1csc(NC(=O)Cc2cccs2)n1 ZINC000880644614 FD On-Demand Anodyne CA5A 30 41 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne SLC6A1 52 33 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne GRIN2B 22 43 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne CTSK 20 40 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne PREP 50 48 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne AMY2 44 31 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne LGMN 59 38 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne TGM2 45 43 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne DPP7 62 39 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne XIAP 18 41 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne BIRC2 20 49 CON(C)CCNC(=O)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880644618 ED On-Demand Anodyne SLC12A5 46 37 CON(C)CCNC(=O)CCc1cccc(Cl)c1 ZINC000880644619 CD On-Demand Anodyne MTNR1A 33 41 CON(C)CCNC(=O)CCc1cccc(Cl)c1 ZINC000880644619 CD On-Demand Anodyne MTNR1B 26 41 CCOc1ccccc1-c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880644648 EF On-Demand Anodyne DRD4 41 32 CCOc1ccccc1-c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880644648 EF On-Demand Anodyne PTGER1 20 41 CCOc1ccccc1-c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880644648 EF On-Demand Anodyne KCNK3 37 40 CCOc1ccccc1-c1cccc(C(=O)NCCN(C)OC)c1 ZINC000880644648 EF On-Demand Anodyne KCNK9 28 40 CON(C)CCNC(=O)[C@@H]1CC(=O)N(c2ccc(Cl)c(F)c2)C1 ZINC000880644662 ED On-Demand Anodyne P2RX7 17 41 CON(C)CCNC(=O)Cc1cccc(OCC#N)c1 ZINC000880644663 CC On-Demand Mild MTNR1A 38 40 CON(C)CCNC(=O)Cc1cccc(OCC#N)c1 ZINC000880644663 CC On-Demand Mild MTNR1B 29 40 CON(C)CCNC(=O)Cc1cccc(OCC#N)c1 ZINC000880644663 CC On-Demand Mild CRTM 45 35 CON(C)CCNC(=O)[C@H](C)Cc1cccc(Cl)c1 ZINC000880644666 CE On-Demand Anodyne CTSB 21 49 CON(C)CCNC(=O)[C@H](C)Cc1cccc(Cl)c1 ZINC000880644666 CE On-Demand Anodyne CTSL 30 48 CON(C)CCNC(=O)[C@H](C)Cc1cccc(Cl)c1 ZINC000880644666 CE On-Demand Anodyne CTSS 18 47 CON(C)CCNC(=O)[C@H](C)Cc1cccc(Cl)c1 ZINC000880644666 CE On-Demand Anodyne CTSV 42 47 CON(C)CCNC(=O)[C@H](C)Cc1cccc(Cl)c1 ZINC000880644666 CE On-Demand Anodyne PDS 45 36 CON(C)CCNC(=O)[C@@H](C)Cc1cccc(Cl)c1 ZINC000880644667 CE On-Demand Anodyne CTSB 21 49 CON(C)CCNC(=O)[C@@H](C)Cc1cccc(Cl)c1 ZINC000880644667 CE On-Demand Anodyne CTSL 30 48 CON(C)CCNC(=O)[C@@H](C)Cc1cccc(Cl)c1 ZINC000880644667 CE On-Demand Anodyne CTSS 18 47 CON(C)CCNC(=O)[C@@H](C)Cc1cccc(Cl)c1 ZINC000880644667 CE On-Demand Anodyne CTSV 42 47 CON(C)CCNC(=O)[C@@H](C)Cc1cccc(Cl)c1 ZINC000880644667 CE On-Demand Anodyne PDS 45 36 CON(C)CCNC(=O)[C@H](C)CC(=O)c1ccc(Cl)cc1 ZINC000880644740 DE On-Demand Anodyne UTS2 46 35 CON(C)CCNC(=O)[C@@H](C)CC(=O)c1ccc(Cl)cc1 ZINC000880644741 DE On-Demand Anodyne UTS2 46 35 CC[C@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644751 CD On-Demand Anodyne NQO2 21 40 CC[C@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644751 CD On-Demand Anodyne KCNQ2 26 47 CC[C@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644751 CD On-Demand Anodyne MTNR1A 59 40 CC[C@@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644752 CD On-Demand Anodyne NQO2 21 40 CC[C@@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644752 CD On-Demand Anodyne KCNQ2 26 47 CC[C@@H](C(=O)NCCN(C)OC)c1ccc(OC)cc1 ZINC000880644752 CD On-Demand Anodyne MTNR1A 59 40 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne PPARG 21 41 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne CSNK1D 16 40 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne MTNR1A 38 42 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne MTNR1B 29 42 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne CRTM 47 38 CON(C)CCNC(=O)Cc1cccc(OC(F)(F)F)c1 ZINC000880644756 DD On-Demand Anodyne PDS 45 33 CON(C)CCNC(=O)C1=NOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 ZINC000880644772 FD On-Demand Anodyne GPR119 18 54 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880644798 GG On-Demand Mild HTR1B 15 48 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880644798 GG On-Demand Mild PDGFRB 54 43 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880644798 GG On-Demand Mild ABCB1 17 43 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880644798 GG On-Demand Mild S1PR2 27 40 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne ACE 29 51 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne MME 61 51 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne LTA4H 26 45 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne FCER2 68 44 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne PAPA1_CARPA 62 38 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne CTSK 26 41 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne CAPNS1 53 33 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne HLA-DRB1 27 41 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne GSTP1 15 43 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne CAPN1 56 42 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne CAPN2 86 42 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne MMP1 24 44 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne FPR1 50 33 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne NPR 74 35 CON(C)CCNC(=O)[C@H](C)CSCc1ccccc1 ZINC000880644804 CE On-Demand Anodyne PDS 44 33 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne ACE 29 51 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne MME 61 51 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne LTA4H 26 45 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne FCER2 68 44 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne PAPA1_CARPA 62 38 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne CTSK 26 41 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne CAPNS1 53 33 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne HLA-DRB1 27 41 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne GSTP1 15 43 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne CAPN1 56 42 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne CAPN2 86 42 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne MMP1 24 44 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne FPR1 50 33 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne NPR 74 35 CON(C)CCNC(=O)[C@@H](C)CSCc1ccccc1 ZINC000880644805 CE On-Demand Anodyne PDS 44 33 CON(C)CCNC(=O)[C@@H](C)CC(C)C ZINC000880644823 BD On-Demand Anodyne CAPN2 45 30 CON(C)CCNC(=O)[C@@H](C)CC(C)C ZINC000880644823 BD On-Demand Anodyne NPR 65 35 CON(C)CCNC(=O)[C@H](C)CC(C)C ZINC000880644824 BD On-Demand Anodyne CAPN2 45 30 CON(C)CCNC(=O)[C@H](C)CC(C)C ZINC000880644824 BD On-Demand Anodyne NPR 65 35 CON(C)CCNC(=O)[C@@H]1CCc2c(Cl)cccc21 ZINC000880644831 CD On-Demand Anodyne MTNR1A 17 40 CON(C)CCNC(=O)CCc1cncc2ccccc12 ZINC000880644834 CD On-Demand Anodyne MTNR1A 30 42 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne DRD2 18 47 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne DRD4 39 47 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne ACHE 38 42 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne DRD3 15 47 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne SIGMAR1 77 42 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne NPFFR2 38 40 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne FAAH 15 40 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne MCHR2 46 35 CON(C)CCNC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000880644860 DD On-Demand Anodyne NPFFR1 51 47 CON(C)CCNC(=O)C[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880644864 FE On-Demand Anodyne PAPA1_CARPA 35 42 CON(C)CCNC(=O)C[C@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880644864 FE On-Demand Anodyne FPR1 43 35 CON(C)CCNC(=O)C[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880644865 FE On-Demand Anodyne PAPA1_CARPA 35 42 CON(C)CCNC(=O)C[C@@H](NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880644865 FE On-Demand Anodyne FPR1 43 35 CON(C)CCNC(=O)C[C@@H](C)C(=O)c1ccc(Cl)cc1 ZINC000880644873 DE On-Demand Anodyne UTS2 45 35 CON(C)CCNC(=O)C[C@H](C)C(=O)c1ccc(Cl)cc1 ZINC000880644874 DE On-Demand Anodyne UTS2 45 35 CON(C)CCNC(=O)[C@@H]1CC[C@@H](C(=O)NCCN(C)OC)CC1 ZINC000880644901 EC On-Demand Anodyne MTNR1A 23 43 CON(C)CCNC(=O)C[C@@H](NC(=O)OC(C)(C)C)C1CC1 ZINC000880644911 DD On-Demand Anodyne ECE1 17 40 CON(C)CCNC(=O)C[C@H](NC(=O)OC(C)(C)C)C1CC1 ZINC000880644912 DD On-Demand Anodyne ECE1 17 40 CON(C)CCNC(=O)CCc1cccc2c1OCO2 ZINC000880644934 CC On-Demand Anodyne MTNR1A 39 48 CON(C)CCNC(=O)CCc1cccc2c1OCO2 ZINC000880644934 CC On-Demand Anodyne MTNR1B 21 40 COC(=O)C1CCC(C(=O)NCCN(C)OC)CC1 ZINC000880644935 CC On-Demand Anodyne MTNR1A 18 40 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne ACE 51 35 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne GHRHR 42 34 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MME 73 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne ANPEP 49 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne SIGMAR1 15 40 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne KLK3 49 32 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne PAPA1_CARPA 63 35 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne CTSK 33 40 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne NPFFR2 45 34 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne CAPNS1 44 35 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MTNR1A 34 42 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MTNR1B 33 42 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MMP2 44 41 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MMP3 79 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MMP8 26 47 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne FAAH 40 41 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne FURIN 54 36 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne CAPN1 52 38 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MMP9 22 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne CAPN2 77 38 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne ACE2 40 34 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne LAP3 43 34 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne MMP1 34 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne NPR 85 39 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne AMP1_PLAFQ 41 44 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne POLG_WNV 52 33 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne DAGLA 19 41 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne CRTM 45 36 CON(C)CCNC(=O)[C@@H](C)CCCc1ccccc1 ZINC000880644936 CE On-Demand Anodyne NPFFR1 61 34 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne ACE 51 35 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne GHRHR 42 34 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MME 73 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne ANPEP 49 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne SIGMAR1 15 40 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne KLK3 49 32 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne PAPA1_CARPA 63 35 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne CTSK 33 40 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne NPFFR2 45 34 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne CAPNS1 44 35 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MTNR1A 34 42 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MTNR1B 33 42 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MMP2 44 41 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MMP3 79 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MMP8 26 47 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne FAAH 40 41 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne FURIN 54 36 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne CAPN1 52 38 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MMP9 22 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne CAPN2 77 38 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne ACE2 40 34 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne LAP3 43 34 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne MMP1 34 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne NPR 85 39 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne AMP1_PLAFQ 41 44 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne POLG_WNV 52 33 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne DAGLA 19 41 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne CRTM 45 36 CON(C)CCNC(=O)[C@H](C)CCCc1ccccc1 ZINC000880644937 CE On-Demand Anodyne NPFFR1 61 34 CON(C)CCNC(=O)[C@@H]1CCC(=O)N1C ZINC000880644942 BB On-Demand Anodyne P2RX7 39 52 CON(C)CCNC(=O)CCCc1cccc(C(F)(F)F)c1 ZINC000880644956 DF On-Demand Anodyne MTNR1A 27 42 CON(C)CCNC(=O)CCCc1cccc(C(F)(F)F)c1 ZINC000880644956 DF On-Demand Anodyne MTNR1B 22 42 CON(C)CCNC(=O)CCCc1cccc(C(F)(F)F)c1 ZINC000880644956 DF On-Demand Anodyne PDS 42 41 C=CCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880644979 CD On-Demand Mild MTNR1A 52 36 C=CCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880644979 CD On-Demand Mild MTNR1B 41 36 C=CCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880644979 CD On-Demand Mild LSS 29 40 C=CCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880644979 CD On-Demand Mild LUCI_LUCLA 15 40 CON(C)CCNC(=O)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880645013 DD On-Demand Anodyne TACR1 23 42 CON(C)CCNC(=O)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880645013 DD On-Demand Anodyne CCR2 37 41 CON(C)CCNC(=O)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880645013 DD On-Demand Anodyne PDS 44 38 CON(C)CCNC(=O)CC[C@H]1CCCCN1C ZINC000880645025 CC On-Demand Anodyne ACKR3 71 37 CON(C)CCNC(=O)CC[C@@H]1CCCCN1C ZINC000880645026 CC On-Demand Anodyne ACKR3 71 37 CON(C)CCNC(=O)CCCc1nnc(-c2ccc(Cl)cc2Cl)o1 ZINC000880645043 GF On-Demand Anodyne ALPL 42 37 CON(C)CCNC(=O)CC[C@@H](C)NC(=O)OC(C)(C)C ZINC000880645044 DD On-Demand Anodyne CTSK 17 40 CON(C)CCNC(=O)CC[C@H](C)NC(=O)OC(C)(C)C ZINC000880645045 DD On-Demand Anodyne CTSK 17 40 CON(C)CCNC(=O)Cc1ccc(C(N)=O)cc1 ZINC000880645051 CB On-Demand Anodyne CA9 20 40 CON(C)CCNC(=O)Cc1ccc(F)cc1Br ZINC000880645078 DD On-Demand Anodyne P2RX7 35 46 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne GRIN2B 34 47 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne PREP 30 42 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne GHSR 15 43 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne CAPN2 43 32 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne TGM2 46 41 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne F13A1 38 41 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880645122 ED On-Demand Anodyne BIRC2 18 47 CON(C)CCNC(=O)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000880645124 CD On-Demand Bother CACNA1C 61 41 CON(C)CCNC(=O)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000880645124 CD On-Demand Bother CACNA1D 88 39 CON(C)CCNC(=O)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000880645124 CD On-Demand Bother COLA 89 39 CON(C)CCNC(=O)CCn1c(C)nc2ccccc21 ZINC000880645157 CD On-Demand Anodyne PTAFR 32 42 CON(C)CCNC(=O)CCn1c(C)nc2ccccc21 ZINC000880645157 CD On-Demand Anodyne PDE6D 28 40 CON(C)CCNC(=O)C1Cc2ccccc2C1 ZINC000880645221 BD On-Demand Anodyne MTNR1A 38 41 CON(C)CCNC(=O)C1Cc2ccccc2C1 ZINC000880645221 BD On-Demand Anodyne MTNR1B 33 41 CON(C)CCNC(=O)C1Cc2ccccc2C1 ZINC000880645221 BD On-Demand Anodyne ADAM9 60 35 CON(C)CCNC(=O)Cc1c(C)oc2ccccc12 ZINC000880645234 CD On-Demand Anodyne MTNR1A 25 40 CON(C)CCNC(=O)Cc1c(C)oc2ccccc12 ZINC000880645234 CD On-Demand Anodyne MTNR1B 23 40 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880645253 CC On-Demand Anodyne CELA1 54 37 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880645253 CC On-Demand Anodyne ELANE 47 42 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880645253 CC On-Demand Anodyne TPP2 30 41 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne DRD4 58 44 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne DRD3 17 46 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne NQO2 21 49 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne MTNR1A 64 43 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne MTNR1B 57 51 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne TUBB2B 25 40 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne HSD17B2 24 41 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne TAAR1 31 44 COc1cccc(C(=O)c2ccc(C(=O)NCCN(C)OC)cc2)c1 ZINC000880645260 EE On-Demand Anodyne KCNK3 17 45 CON(C)CCNC(=O)Cc1c(C)cccc1Cl ZINC000880645263 CD On-Demand Anodyne P2RX7 31 48 CON(C)CCNC(=O)CCCCN1CCOCC1 ZINC000880645335 CC On-Demand Anodyne PAOX 19 47 CON(C)CCNC(=O)CCCCN1CCOCC1 ZINC000880645335 CC On-Demand Anodyne EPHX2 19 40 CON(C)CCNC(=O)CCCCCc1ccc(F)cc1 ZINC000880645342 CF On-Demand Anodyne FAAH 18 40 CON(C)CCNC(=O)CCCCCc1ccc(F)cc1 ZINC000880645342 CF On-Demand Anodyne LEF 27 40 CON(C)CCNC(=O)[C@@](C)(OC)c1ccccc1 ZINC000880645362 CD On-Demand Anodyne AMY2 57 36 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NCCN(C)OC)c1 ZINC000880645376 DD On-Demand Anodyne MTNR1A 58 53 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NCCN(C)OC)c1 ZINC000880645376 DD On-Demand Anodyne MTNR1B 49 53 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NCCN(C)OC)c1 ZINC000880645377 DD On-Demand Anodyne MTNR1A 58 53 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NCCN(C)OC)c1 ZINC000880645377 DD On-Demand Anodyne MTNR1B 49 53 CON(C)CCNC(=O)[C@@H]1CCCc2cccnc21 ZINC000880645432 CD On-Demand Anodyne CXCR4 76 43 CCN1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645434 GF On-Demand Anodyne TSHR 49 32 CCN1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645434 GF On-Demand Anodyne CCKAR 42 41 CCN1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645434 GF On-Demand Anodyne CCKBR 65 38 CCN1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645435 GF On-Demand Anodyne TSHR 49 32 CCN1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645435 GF On-Demand Anodyne CCKAR 42 41 CCN1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1=O ZINC000880645435 GF On-Demand Anodyne CCKBR 65 38 COc1ccc(O)cc1C(=O)NCCN(C)OC ZINC000880645448 CC On-Demand Anodyne AKR1B10 61 38 CON(C)CCNC(=O)[C@@H]1CCC(=O)N1Cc1ccc(Br)cc1 ZINC000880645449 GD On-Demand Anodyne P2RX7 36 48 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne DRD3 15 50 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne NQO2 29 41 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne PYGL 73 48 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne ROCK1 15 42 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne MTNR1A 92 41 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne MTNR1B 72 41 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne ROCK2 15 42 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne TUBB2B 55 52 COc1ccc2[nH]c(C(=O)NCCN(C)OC)cc2c1 ZINC000880645471 CD On-Demand Anodyne PYK 30 44 CON(C)CCNC(=O)Cc1cncn1Cc1ccccc1 ZINC000880645490 DD On-Demand Anodyne CYP11B1 15 58 CON(C)CCNC(=O)[C@@H](C)Oc1cccc2ccccc12 ZINC000880645496 DE On-Demand Anodyne NQO2 25 40 CON(C)CCNC(=O)[C@@H](C)Oc1cccc2ccccc12 ZINC000880645496 DE On-Demand Anodyne MTNR1A 46 42 CON(C)CCNC(=O)[C@@H](C)Oc1cccc2ccccc12 ZINC000880645496 DE On-Demand Anodyne IMDH_CRYPV 19 45 CON(C)CCNC(=O)[C@H](C)Oc1cccc2ccccc12 ZINC000880645497 DE On-Demand Anodyne NQO2 25 40 CON(C)CCNC(=O)[C@H](C)Oc1cccc2ccccc12 ZINC000880645497 DE On-Demand Anodyne MTNR1A 46 42 CON(C)CCNC(=O)[C@H](C)Oc1cccc2ccccc12 ZINC000880645497 DE On-Demand Anodyne IMDH_CRYPV 19 45 CCCc1c(C(=O)NCCN(C)OC)cnn1-c1ccc(C)cc1 ZINC000880645529 EE On-Demand Anodyne GPR142 50 33 CCCC[C@H](C)C(=O)NCCN(C)OC ZINC000880645551 BD On-Demand Anodyne NOD1 60 33 CCCC[C@@H](C)C(=O)NCCN(C)OC ZINC000880645552 BD On-Demand Anodyne NOD1 60 33 CON(C)CCNC(=O)Cc1ccc(Cl)c(F)c1 ZINC000880645567 CD On-Demand Anodyne NCE103 16 49 COCCOc1ccc(CC(=O)NCCN(C)OC)cc1 ZINC000880645641 CC On-Demand Anodyne LTA4H 35 44 COCCOc1ccc(CC(=O)NCCN(C)OC)cc1 ZINC000880645641 CC On-Demand Anodyne MTNR1A 44 37 COCCOc1ccc(CC(=O)NCCN(C)OC)cc1 ZINC000880645641 CC On-Demand Anodyne CA9 18 42 CON(C)CCNC(=O)COC1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880645642 ED On-Demand Anodyne GPR119 35 40 CCCOc1cccnc1C(=O)NCCN(C)OC ZINC000880645647 CD On-Demand Anodyne MAP1 29 41 CON(C)CCNC(=O)CCc1cccc(N(C)C)c1 ZINC000880645659 CD On-Demand Anodyne MTNR1A 35 41 CON(C)CCNC(=O)CCc1cccc(N(C)C)c1 ZINC000880645659 CD On-Demand Anodyne MTNR1B 26 41 CON(C)CCNC(=O)C[C@H]1CCCN(C(=O)OC(C)(C)C)CC1 ZINC000880645664 EE On-Demand Anodyne GPR119 34 40 CON(C)CCNC(=O)C[C@@H]1CCCN(C(=O)OC(C)(C)C)CC1 ZINC000880645665 EE On-Demand Anodyne GPR119 34 40 CCCCS(=O)(=O)c1ccc(C(=O)NCCN(C)OC)cc1 ZINC000880645671 ED On-Demand Anodyne CA2 17 50 CCCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880645683 CD On-Demand Anodyne MTNR1A 74 48 CCCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880645683 CD On-Demand Anodyne MTNR1B 57 48 COCCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880645695 DC On-Demand Anodyne MTNR1A 72 42 COCCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880645695 DC On-Demand Anodyne MTNR1B 55 42 COCCOc1cc(OC)ccc1C(=O)NCCN(C)OC ZINC000880645695 DC On-Demand Anodyne LUCI_LUCLA 15 42 CNc1ccccc1C(=O)NCCN(C)OC ZINC000880645706 BC On-Demand Anodyne KCNA3 17 44 CNc1ccccc1C(=O)NCCN(C)OC ZINC000880645706 BC On-Demand Anodyne POLR1A 58 41 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880645713 FE On-Demand Anodyne PDGFRB 47 41 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880645713 FE On-Demand Anodyne ABCB1 19 43 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880645713 FE On-Demand Anodyne ENPP1 57 33 COCCn1ccc(C(=O)NCCN(C)OC)n1 ZINC000880645715 CB On-Demand Anodyne POLR1A 33 40 CON(C)CCNC(=O)Cc1ccc(Br)c(Cl)c1 ZINC000880645742 EE On-Demand Anodyne NCE103 17 52 CON(C)CCNC(=O)CCN(C)C(=O)OCc1ccccc1 ZINC000880645764 DD On-Demand Anodyne CAPN2 52 32 CON(C)CCNC(=O)CCN(C)C(=O)OCc1ccccc1 ZINC000880645764 DD On-Demand Anodyne NPR 64 35 CON(C)CCNC(=O)Cc1ccc(Cl)cn1 ZINC000880645791 CC On-Demand Anodyne F10 48 33 COc1ccc(CC(=O)NCCN(C)OC)nc1 ZINC000880645815 CC On-Demand Anodyne MTNR1A 50 40 COc1ccc(CC(=O)NCCN(C)OC)nc1 ZINC000880645815 CC On-Demand Anodyne MTNR1B 32 40 COc1ccccc1-n1ncc(C(=O)NCCN(C)OC)c1C ZINC000880645818 DD On-Demand Anodyne HTR1A 25 44 COc1ccccc1-n1ncc(C(=O)NCCN(C)OC)c1C ZINC000880645818 DD On-Demand Anodyne DRD2 27 45 COc1ccccc1-n1ncc(C(=O)NCCN(C)OC)c1C ZINC000880645818 DD On-Demand Anodyne DRD4 19 45 COc1ccccc1-n1ncc(C(=O)NCCN(C)OC)c1C ZINC000880645818 DD On-Demand Anodyne DRD3 46 44 CON(C)CCNC(=O)CCSCc1ccccc1 ZINC000880645820 CD On-Demand Anodyne CACNA2D1 20 42 CON(C)CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1 ZINC000880645843 CD On-Demand Anodyne UTS2 42 37 CCCc1c(C(=O)NCCN(C)OC)cnn1-c1cccc(C)c1 ZINC000880645852 EE On-Demand Anodyne GPR142 50 33 CCCc1c(C(=O)NCCN(C)OC)cnn1-c1ccccc1C ZINC000880645854 EE On-Demand Anodyne GPR142 55 37 CC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645871 EF On-Demand Anodyne ADRB1 44 35 CC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645871 EF On-Demand Anodyne TSHR 47 31 CC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645871 EF On-Demand Anodyne KCNK3 52 42 CC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645871 EF On-Demand Anodyne KCNK9 52 38 CON(C)CCNC(=O)CN(C)C(=O)OCc1ccccc1 ZINC000880645883 DC On-Demand Anodyne CAPNS1 43 33 CON(C)CCNC(=O)CN(C)C(=O)OCc1ccccc1 ZINC000880645883 DC On-Demand Anodyne CAPN2 59 33 CON(C)CCNC(=O)CN(C)C(=O)OCc1ccccc1 ZINC000880645883 DC On-Demand Anodyne NPR 65 37 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne F2 38 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne ELANE 43 42 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne MMP13 27 43 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne PREP 37 43 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne MMP3 39 43 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne TPP2 27 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne MMP1 34 43 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645899 EC On-Demand Anodyne TMPRSS11D 41 32 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne F2 38 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne ELANE 43 42 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne MMP13 27 43 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne PREP 37 43 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne MMP3 39 43 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne TPP2 27 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne MMP1 34 43 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NCCN(C)OC)cc1 ZINC000880645900 EC On-Demand Anodyne TMPRSS11D 41 32 CCNC(=O)C(C)(C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645903 GF On-Demand Anodyne IMDH_CRYPV 60 39 CCNC(=O)C(C)(C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880645903 GF On-Demand Anodyne KCNK3 44 37 COc1cccc([C@@H](C)CCCC(=O)NCCN(C)OC)c1 ZINC000880645914 DF On-Demand Anodyne MTNR1A 63 43 COc1cccc([C@@H](C)CCCC(=O)NCCN(C)OC)c1 ZINC000880645914 DF On-Demand Anodyne MTNR1B 58 43 COc1cccc([C@H](C)CCCC(=O)NCCN(C)OC)c1 ZINC000880645915 DF On-Demand Anodyne MTNR1A 63 43 COc1cccc([C@H](C)CCCC(=O)NCCN(C)OC)c1 ZINC000880645915 DF On-Demand Anodyne MTNR1B 58 43 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne ACE 49 48 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne FOLH1 16 42 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne MME 166 52 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne LTA4H 26 47 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne ANPEP 112 45 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne FCER2 64 36 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CTSB 43 39 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne PAPA1_CARPA 64 43 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CTSK 17 40 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CTSL 42 43 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CPA1 84 41 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CTRB1 35 40 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CAPNS1 63 34 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne MMP8 25 42 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne ECE1 15 48 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CTSS 20 43 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CAPN1 71 41 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne CAPN2 66 38 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne ACE2 67 37 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne LAP3 63 41 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne FPR1 46 34 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne NPR 83 45 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne AMP1_PLAFQ 58 43 CON(C)CCNC(=O)C(Cc1ccccc1)Cc1ccccc1 ZINC000880645990 EF On-Demand Anodyne NPFFR1 47 34 CON(C)CCNC(=O)[C@@H]1CCCN1c1ccccc1 ZINC000880645993 CD On-Demand Anodyne FKBP1A 22 40 CON(C)CCNC(=O)[C@@H]1CCCN1c1ccccc1 ZINC000880645993 CD On-Demand Anodyne PREP 46 36 CON(C)CCNC(=O)[C@@H]1CCCN1c1ccccc1 ZINC000880645993 CD On-Demand Anodyne XIAP 32 43 CON(C)CCNC(=O)Cn1ccc2ccccc2c1=O ZINC000880646029 CC On-Demand Anodyne MTNR1A 15 41 CON(C)CCNC(=O)Cn1ccc2ccccc2c1=O ZINC000880646029 CC On-Demand Anodyne PSMB5 17 51 CON(C)CCNC(=O)Cn1ccc2ccccc2c1=O ZINC000880646029 CC On-Demand Anodyne PSMB1 18 51 CON(C)CCNC(=O)Cn1ccc2ccccc2c1=O ZINC000880646029 CC On-Demand Anodyne NR5A1 26 43 CON(C)CCNC(=O)Cn1ccc2ccccc2c1=O ZINC000880646029 CC On-Demand Anodyne POLR1A 46 39 CON(C)CCNC(=O)Cc1coc2ccccc12 ZINC000880646047 CD On-Demand Anodyne NQO2 25 40 CON(C)CCNC(=O)Cc1coc2ccccc12 ZINC000880646047 CD On-Demand Anodyne MTNR1A 28 43 CON(C)CCNC(=O)C1CCC(O)CC1 ZINC000880646051 BC On-Demand Anodyne MTNR1A 18 40 CON(C)CCNC(=O)[C@@H](CNC(=O)OC(C)(C)C)c1ccc(F)cc1 ZINC000880646060 FE On-Demand Anodyne PAPA1_CARPA 32 43 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne MME 67 39 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne PAPA1_CARPA 48 34 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne PGA 44 36 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne BRS3 20 41 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne CTRB1 22 40 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne MMP3 46 39 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne HLA-DRB1 53 35 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne CAPN1 45 37 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne CASP1 30 50 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne CAPN2 58 34 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne NPR 81 42 CON(C)CCNC(=O)[C@@H](C)NC(=O)CCc1ccccc1 ZINC000880646076 DC On-Demand Anodyne PSMB5 26 46 CC[C@@H](NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1)C(=O)NC ZINC000880646090 FF On-Demand Anodyne ANPEP 15 41 CC[C@@H](NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1)C(=O)NC ZINC000880646090 FF On-Demand Anodyne KCNK3 40 38 CON(C)CCNC(=O)[C@@H]1CCc2cccnc21 ZINC000880646110 BC On-Demand Anodyne CXCR4 45 39 COCCCCN(C)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646128 FH On-Demand Anodyne KCNK3 49 43 COCCCCN(C)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646128 FH On-Demand Anodyne KCNK9 43 39 COc1cccc(C2=NO[C@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646158 DC On-Demand Anodyne DRD4 40 31 COc1cccc(C2=NO[C@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646158 DC On-Demand Anodyne MTNR1A 53 39 COc1cccc(C2=NO[C@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646158 DC On-Demand Anodyne MTNR1B 47 39 COc1cccc(C2=NO[C@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646158 DC On-Demand Anodyne LUCI_PHOPY 40 48 COc1cccc(C2=NO[C@@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646159 DC On-Demand Anodyne DRD4 40 31 COc1cccc(C2=NO[C@@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646159 DC On-Demand Anodyne MTNR1A 53 39 COc1cccc(C2=NO[C@@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646159 DC On-Demand Anodyne MTNR1B 47 39 COc1cccc(C2=NO[C@@H](C(=O)NCCN(C)OC)C2)c1 ZINC000880646159 DC On-Demand Anodyne LUCI_PHOPY 40 48 CON(C)CCNC(=O)CCCC(=O)c1ccc(Br)cc1 ZINC000880646162 FE On-Demand Anodyne HDAC8 20 49 CON(C)CCNC(=O)[C@@H](c1cccnc1)C(C)C ZINC000880646193 CD On-Demand Anodyne KCNA5 27 49 CON(C)CCNC(=O)[C@@H](C)c1ccc(C(F)(F)F)cc1 ZINC000880646199 DE On-Demand Anodyne TRPV1 88 37 CON(C)CCNC(=O)[C@H](C)c1ccc(C(F)(F)F)cc1 ZINC000880646200 DE On-Demand Anodyne TRPV1 88 37 CON(C)CCNC(=O)COc1cccc(I)c1 ZINC000880646215 FD On-Demand Anodyne MTNR1A 57 42 CON(C)CCNC(=O)COc1cccc(I)c1 ZINC000880646215 FD On-Demand Anodyne MTNR1B 44 42 CON(C)CCNC(=O)C[C@@H](C)c1c[nH]c2ccccc12 ZINC000880646221 CE On-Demand Anodyne SSTR2 46 36 CON(C)CCNC(=O)C[C@@H](C)c1c[nH]c2ccccc12 ZINC000880646221 CE On-Demand Anodyne GRIA1 15 41 CON(C)CCNC(=O)C[C@@H](C)c1c[nH]c2ccccc12 ZINC000880646221 CE On-Demand Anodyne MMP1 21 40 CON(C)CCNC(=O)C[C@H](C)c1c[nH]c2ccccc12 ZINC000880646222 CE On-Demand Anodyne SSTR2 46 36 CON(C)CCNC(=O)C[C@H](C)c1c[nH]c2ccccc12 ZINC000880646222 CE On-Demand Anodyne GRIA1 15 41 CON(C)CCNC(=O)C[C@H](C)c1c[nH]c2ccccc12 ZINC000880646222 CE On-Demand Anodyne MMP1 21 40 CON(C)CCNC(=O)[C@@H]1CCc2nn[nH]c2C1 ZINC000880646225 CB On-Demand Anodyne MKNK1 45 38 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880646259 ED On-Demand Anodyne ACHE 22 41 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880646259 ED On-Demand Anodyne SIGMAR1 54 41 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880646259 ED On-Demand Anodyne NPFFR1 43 38 CON(C)CCNC(=O)[C@@]1(C)CCN(C(=O)OCc2ccccc2)C1 ZINC000880646282 ED On-Demand Anodyne SLC12A5 68 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880646315 GF On-Demand Anodyne ABCB1 17 42 CON(C)CCNC(=O)[C@H](C)Oc1ccc2ccccc2c1 ZINC000880646320 DE On-Demand Anodyne NQO2 32 46 CON(C)CCNC(=O)[C@H](C)Oc1ccc2ccccc2c1 ZINC000880646320 DE On-Demand Anodyne MTNR1A 68 46 CON(C)CCNC(=O)[C@H](C)Oc1ccc2ccccc2c1 ZINC000880646320 DE On-Demand Anodyne MTNR1B 52 43 CON(C)CCNC(=O)[C@H](C)Oc1ccc2ccccc2c1 ZINC000880646320 DE On-Demand Anodyne UTS2 39 40 CON(C)CCNC(=O)[C@H](C)Oc1ccc2ccccc2c1 ZINC000880646320 DE On-Demand Anodyne POLR1A 41 34 CON(C)CCNC(=O)[C@@H](C)n1ccc2ccccc2c1=O ZINC000880646325 DD On-Demand Anodyne POLR1A 46 38 CON(C)CCNC(=O)C(C)(C)Cc1nc2ccccc2[nH]1 ZINC000880646327 DD On-Demand Anodyne CACNA1G 22 41 CON(C)CCNC(=O)[C@@H]1CCN(c2ccc(C#N)cc2F)C1 ZINC000880646345 DD On-Demand Mild GPBAR1 32 43 COC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880646353 DC On-Demand Anodyne PAPA1_CARPA 45 47 COC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880646353 DC On-Demand Anodyne CTSK 15 47 CON(C)CCNC(=O)Cc1cccc(Cl)c1Cl ZINC000880646359 CE On-Demand Anodyne P2RX7 36 45 COc1cccc(C2(C(=O)NCCN(C)OC)CC2)c1 ZINC000880646382 CD On-Demand Anodyne DRD4 43 33 COc1cccc(C2(C(=O)NCCN(C)OC)CC2)c1 ZINC000880646382 CD On-Demand Anodyne MTNR1A 66 45 COc1cccc(C2(C(=O)NCCN(C)OC)CC2)c1 ZINC000880646382 CD On-Demand Anodyne MTNR1B 58 45 CON(C)CCNC(=O)[C@@H](NC(N)=O)C(C)(C)C ZINC000880646393 CB On-Demand Anodyne PDF 42 30 COCC[C@@H](CO)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646431 FE On-Demand Anodyne KCNK3 59 43 COCC[C@@H](CO)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646431 FE On-Demand Anodyne KCNK9 49 40 COCC[C@H](CO)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646432 FE On-Demand Anodyne KCNK3 59 43 COCC[C@H](CO)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646432 FE On-Demand Anodyne KCNK9 49 40 CON(C)CCNC(=O)[C@@H]1CCc2ccccc2C1 ZINC000880646436 CD On-Demand Anodyne MTNR1A 34 40 CON(C)CCNC(=O)[C@@H]1CCc2ccccc2C1 ZINC000880646436 CD On-Demand Anodyne MTNR1B 34 40 CON(C)CCNC(=O)[C@@H]1CCc2ccccc2C1 ZINC000880646436 CD On-Demand Anodyne ADAM9 49 33 COc1ccc(OC(F)(F)F)c(C(=O)NCCN(C)OC)c1 ZINC000880646437 DD On-Demand Anodyne MTNR1A 46 37 COc1ccc(OC(F)(F)F)c(C(=O)NCCN(C)OC)c1 ZINC000880646437 DD On-Demand Anodyne KCNK3 19 40 COc1ccc(OC(F)(F)F)c(C(=O)NCCN(C)OC)c1 ZINC000880646437 DD On-Demand Anodyne KCNK9 20 40 CON(C)CCNC(=O)Cc1cccc(NC(C)=O)c1 ZINC000880646452 CC On-Demand Anodyne NQO2 42 41 CON(C)CCNC(=O)Cc1cccc(NC(C)=O)c1 ZINC000880646452 CC On-Demand Anodyne MTNR1A 58 41 CON(C)CCNC(=O)Cc1cccc(NC(C)=O)c1 ZINC000880646452 CC On-Demand Anodyne MTNR1B 52 41 CON(C)CCNC(=O)Cc1cccc(NC(C)=O)c1 ZINC000880646452 CC On-Demand Anodyne KCNK3 63 35 CON(C)CCNC(=O)Cc1cccc(NC(C)=O)c1 ZINC000880646452 CC On-Demand Anodyne KCNK9 53 35 CON(C)CCNC(=O)CN(C)C1CCC1 ZINC000880646472 BC On-Demand Anodyne ACE 42 35 CON(C)CCNC(=O)CCc1cccc(OC(F)F)c1 ZINC000880646502 DD On-Demand Anodyne MTNR1A 38 45 CON(C)CCNC(=O)CCc1cccc(OC(F)F)c1 ZINC000880646502 DD On-Demand Anodyne MTNR1B 30 45 CON(C)CCNC(=O)CCc1cccc(OC(F)F)c1 ZINC000880646502 DD On-Demand Anodyne CRTM 48 37 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1cccnc1 ZINC000880646540 BC On-Demand Anodyne NAMPT 32 57 CON(C)CCNC(=O)[C@@H]1CCCN1C(=O)C1CC1 ZINC000880646544 CB On-Demand Anodyne TPP2 31 43 CON(C)CCNC(=O)[C@@H](CC(C)C)C(N)=O ZINC000880646553 BB On-Demand Anodyne NPR 20 40 CON(C)CCNC(=O)Cc1nn(C)c2ccccc12 ZINC000880646556 CC On-Demand Anodyne IMDH_CRYPV 26 43 CON(C)CCNC(=O)Cc1ccccc1OC1CCCC1 ZINC000880646563 DE On-Demand Anodyne PDE4A 18 42 CON(C)CCNC(=O)Cc1ccccc1OC1CCCC1 ZINC000880646563 DE On-Demand Anodyne MBTPS1 45 35 CON(C)CCNC(=O)Cc1ccc(O)c(F)c1 ZINC000880646570 CC On-Demand Anodyne NCE103 16 50 CON(C)CCNC(=O)CCc1ccc2ccccc2c1O ZINC000880646591 DE On-Demand Anodyne ALOX5 15 55 CON(C)CCNC(=O)CCc1ccc2ccccc2c1O ZINC000880646591 DE On-Demand Anodyne MTNR1A 50 44 CON(C)CCNC(=O)[C@@H]1CCc2nc(C)[nH]c2C1 ZINC000880646601 CC On-Demand Anodyne MKNK1 44 37 CCn1nc(C)c(CC(=O)NCCN(C)OC)c1C ZINC000880646632 CC On-Demand Anodyne P2RX7 25 50 CNC(=O)C[C@@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646666 FF On-Demand Anodyne ENPP1 67 32 CNC(=O)C[C@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646667 FF On-Demand Anodyne ENPP1 67 32 CON(C)CCNC(=O)C[C@@H]1COc2ccccc2O1 ZINC000880646672 CC On-Demand Anodyne ADRA2B 15 44 CON(C)CCNC(=O)C[C@H]1COc2ccccc2O1 ZINC000880646673 CC On-Demand Anodyne ADRA2B 15 44 CON(C)CCNC(=O)[C@@H](C)c1cccc(Br)c1 ZINC000880646686 DE On-Demand Anodyne TRPV1 24 43 CON(C)CCNC(=O)CCCc1ccccc1Cl ZINC000880646750 CE On-Demand Anodyne MTNR1A 43 43 CON(C)CCNC(=O)C(C)(C)c1ccccc1[N+](=O)[O-] ZINC000880646751 CD On-Demand Bother COLA 87 33 CON(C)CCNC(=O)C1CCN(c2noc3ccc(Cl)cc23)CC1 ZINC000880646753 FE On-Demand Anodyne PTGES 20 41 CON(C)CCNC(=O)[C@@H](NC(=O)OC(C)(C)C)c1c(F)cccc1F ZINC000880646793 FE On-Demand Anodyne PAPA1_CARPA 36 46 CON(C)CCNC(=O)[C@@H]1CCc2nc[nH]c2C1 ZINC000880646824 CC On-Demand Anodyne MKNK1 43 36 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc(C)cc1 ZINC000880646845 CD On-Demand Anodyne SLC6A3 19 40 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2F)C1 ZINC000880646849 CD On-Demand Anodyne HTR1A 19 43 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2F)C1 ZINC000880646849 CD On-Demand Anodyne DRD2 19 42 CON(C)CCNC(=O)[C@@H]1C[C@@H]1c1ccc(C)cc1 ZINC000880646850 CD On-Demand Anodyne SLC6A3 19 40 CON(C)CCNC(=O)COCc1cccnc1 ZINC000880646867 CC On-Demand Anodyne PTAFR 27 42 CON(C)CCNC(=O)[C@@H](OC(C)C)c1ccccc1 ZINC000880646879 CD On-Demand Anodyne UTS2 26 40 CON(C)CCNC(=O)Cc1ccc2c(c1)CCCO2 ZINC000880646907 CD On-Demand Anodyne MTNR1A 15 40 CON(C)CCNC(=O)Cn1c(-c2ccccc2)nc2ccccc21 ZINC000880646930 EE On-Demand Anodyne AVPR1B 50 44 CON(C)CCNC(=O)Cn1c(-c2ccccc2)nc2ccccc21 ZINC000880646930 EE On-Demand Anodyne PDE6D 88 41 CON(C)CCNC(=O)Cn1c(-c2ccccc2)nc2ccccc21 ZINC000880646930 EE On-Demand Anodyne IMDH_CRYPV 38 54 CON(C)CCNC(=O)COc1ccc(Cl)c(F)c1 ZINC000880646941 CD On-Demand Anodyne MTNR1A 48 39 CON(C)CCNC(=O)[C@@H](C)CNC(=O)OC(C)(C)C ZINC000880646956 CC On-Demand Anodyne PAPA1_CARPA 38 40 CON(C)CCNC(=O)[C@H](C)CNC(=O)OC(C)(C)C ZINC000880646957 CC On-Demand Anodyne PAPA1_CARPA 38 40 COCCCONC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646959 FG On-Demand Anodyne KCNK3 72 45 COCCCONC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880646959 FG On-Demand Anodyne KCNK9 49 42 CCCOc1ccc(C(=O)NCCN(C)OC)c(OC)c1 ZINC000880646970 CD On-Demand Anodyne MTNR1B 25 40 CCCOc1ccc(C(=O)NCCN(C)OC)c(OC)c1 ZINC000880646970 CD On-Demand Anodyne LSS 19 42 CON(C)CCNC(=O)Cc1cccc(Cl)c1F ZINC000880646980 CD On-Demand Anodyne P2RX7 36 46 CON(C)CCNC(=O)Cc1cccc(Cl)c1F ZINC000880646980 CD On-Demand Anodyne ECR 40 32 CCC(=O)Nc1ccccc1C(=O)NCCN(C)OC ZINC000880646982 CD On-Demand Anodyne FAS 17 40 C/C=C\COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646990 CD On-Demand Anodyne MTNR1A 42 42 C/C=C\COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646990 CD On-Demand Anodyne MTNR1B 32 42 C/C=C\COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646990 CD On-Demand Anodyne CRTM 42 37 C/C=C/COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646991 CD On-Demand Anodyne MTNR1A 42 42 C/C=C/COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646991 CD On-Demand Anodyne MTNR1B 32 42 C/C=C/COc1cccc(CC(=O)NCCN(C)OC)c1 ZINC000880646991 CD On-Demand Anodyne CRTM 42 37 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne MME 32 42 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne MTNR1A 28 41 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne MTNR1B 25 41 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne ACE2 41 33 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne NPR 43 32 CON(C)CCNC(=O)[C@H](C)COc1ccccc1 ZINC000880647026 CD On-Demand Anodyne PDS 75 40 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne MME 32 42 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne MTNR1A 28 41 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne MTNR1B 25 41 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne ACE2 41 33 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne NPR 43 32 CON(C)CCNC(=O)[C@@H](C)COc1ccccc1 ZINC000880647027 CD On-Demand Anodyne PDS 75 40 CON(C)CCNC(=O)[C@H](C)Cc1cncc2ccccc12 ZINC000880647043 DE On-Demand Anodyne MTNR1A 17 41 CON(C)CCNC(=O)[C@@H](C)Cc1cncc2ccccc12 ZINC000880647044 DE On-Demand Anodyne MTNR1A 17 41 COC[C@@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647141 EG On-Demand Anodyne KCNK3 48 43 COC[C@@H](C)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647141 EG On-Demand Anodyne KCNK9 43 40 CON(C)CCNC(=O)C[C@H](C)n1ccnc1 ZINC000880647143 BC On-Demand Anodyne CYP26A1 90 37 CON(C)CCNC(=O)C[C@@H](C)n1ccnc1 ZINC000880647144 BC On-Demand Anodyne CYP26A1 90 37 CON(C)CCNC(=O)Cc1cccc(OCC=C(C)C)c1 ZINC000880647165 DE On-Demand Anodyne MTNR1A 47 41 CON(C)CCNC(=O)Cc1cccc(OCC=C(C)C)c1 ZINC000880647165 DE On-Demand Anodyne MTNR1B 39 41 CON(C)CCNC(=O)Cc1cccc(OCC=C(C)C)c1 ZINC000880647165 DE On-Demand Anodyne CRTM 44 34 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc(Cl)cc1 ZINC000880647178 CE On-Demand Anodyne SLC6A4 18 50 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc(Cl)cc1 ZINC000880647178 CE On-Demand Anodyne SLC6A3 31 50 CON(C)CCNC(=O)Cc1c(C)nn(CC2CC2)c1C ZINC000880647205 CD On-Demand Anodyne P2RX7 23 49 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc([N+](=O)[O-])cc1 ZINC000880647211 CD On-Demand Bother SLC27A4 55 37 CCc1ccccc1-n1cc(C(=O)NCCN(C)OC)nn1 ZINC000880647212 DD On-Demand Anodyne DRD3 18 43 CON(C)CCNC(=O)[C@@H](C)c1ccc(Cl)cc1 ZINC000880647217 CE On-Demand Anodyne TRPV1 22 43 CON(C)CCNC(=O)[C@@H](C)c1ccc(Cl)cc1 ZINC000880647217 CE On-Demand Anodyne UTS2 48 38 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne MME 60 42 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne ANPEP 53 33 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne PAPA1_CARPA 52 35 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne MMP3 59 38 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne MMP8 21 42 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne CASP1 29 41 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne CAPN2 52 34 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne LAP3 45 38 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne NPR 81 37 CON(C)CCNC(=O)[C@@H](CCc1ccccc1)C(C)C ZINC000880647230 CF On-Demand Anodyne AMP1_PLAFQ 36 41 COCC[C@@H]1COCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647233 GG On-Demand Anodyne ACKR3 67 34 COCC[C@H]1COCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647234 GG On-Demand Anodyne ACKR3 67 34 CON(C)CCNC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1C ZINC000880647260 FE On-Demand Anodyne PAPA1_CARPA 37 42 CON(C)CCNC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1C ZINC000880647260 FE On-Demand Anodyne FPR1 44 36 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880647271 DD On-Demand Anodyne HTR1A 19 44 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880647271 DD On-Demand Anodyne DRD2 29 43 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880647271 DD On-Demand Anodyne DRD3 47 40 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880647271 DD On-Demand Anodyne GPBAR1 15 40 CON(C)CCNC(=O)C1(c2ccccc2)CC(=O)C1 ZINC000880647280 CC On-Demand Anodyne KCNA3 43 38 CON(C)CCNC(=O)Cn1nc(C(F)(F)F)c(Cl)c1C ZINC000880647283 ED On-Demand Anodyne CCR1 23 44 CON(C)CCNC(=O)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880647286 FC On-Demand Anodyne CELA1 20 42 CON(C)CCNC(=O)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880647286 FC On-Demand Anodyne PREP 29 43 CON(C)CCNC(=O)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880647286 FC On-Demand Anodyne LGMN 66 40 CON(C)CCNC(=O)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880647286 FC On-Demand Anodyne KLK5 43 42 CON(C)CCNC(=O)Cc1c(C)nn(C(C)C)c1C ZINC000880647290 CD On-Demand Anodyne P2RX7 25 51 CON(C)CCNC(=O)C(C)(C)c1cccc2ccccc12 ZINC000880647292 DF On-Demand Anodyne MTNR1A 22 40 CON(C)CCNC(=O)[C@H](C)c1ccc(Cl)cc1 ZINC000880647318 CE On-Demand Anodyne TRPV1 22 43 CON(C)CCNC(=O)[C@H](C)c1ccc(Cl)cc1 ZINC000880647318 CE On-Demand Anodyne UTS2 48 38 CON(C)CCNC(=O)[C@@H]1CSCN1C(=O)OC(C)(C)C ZINC000880647323 DC On-Demand Anodyne CACNA1B 16 42 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000880647359 CE On-Demand Anodyne MDM2 40 31 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP13 44 47 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne ADAM17 16 47 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP2 44 46 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP3 19 46 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP8 22 46 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP14 42 46 CON(C)CCNC(=O)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880647382 ED On-Demand Anodyne MMP10 85 38 COC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647390 FE On-Demand Anodyne ADRB1 49 41 COC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647390 FE On-Demand Anodyne TSHR 41 30 COC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647390 FE On-Demand Anodyne ABCB1 20 40 CO/C(=C/c1ccccc1)C(=O)NCCN(C)OC ZINC000880647396 CD On-Demand Anodyne TLR4 26 44 CO/C(=C\c1ccccc1)C(=O)NCCN(C)OC ZINC000880647397 CD On-Demand Anodyne TLR4 26 44 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1C(F)(F)F ZINC000880647429 FD On-Demand Anodyne ACHE 22 40 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1C(F)(F)F ZINC000880647429 FD On-Demand Anodyne SIGMAR1 23 41 CON(C)CCNC(=O)[C@H](C)Cc1ccc(OC(F)(F)F)cc1 ZINC000880647430 EE On-Demand Anodyne GCGR 22 43 CON(C)CCNC(=O)[C@H](C)Cc1ccc(OC(F)(F)F)cc1 ZINC000880647430 EE On-Demand Anodyne ACE2 46 36 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(OC(F)(F)F)cc1 ZINC000880647431 EE On-Demand Anodyne GCGR 22 43 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(OC(F)(F)F)cc1 ZINC000880647431 EE On-Demand Anodyne ACE2 46 36 CCC[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)NCCN(C)OC ZINC000880647432 EE On-Demand Anodyne DRD4 18 47 CCC[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)NCCN(C)OC ZINC000880647432 EE On-Demand Anodyne ACHE 23 41 CCC[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)NCCN(C)OC ZINC000880647432 EE On-Demand Anodyne SIGMAR1 20 41 CON(C)CCNC(=O)[C@@H](CC(C)C)n1ccnc1 ZINC000880647443 CD On-Demand Anodyne CYP26A1 81 35 COc1cccc(C(=O)NCCN(C)OC)c1OC(C)C ZINC000880647451 CD On-Demand Anodyne KCNA3 39 41 COc1cccc(C(=O)NCCN(C)OC)c1OC(C)C ZINC000880647451 CD On-Demand Anodyne KCNK3 45 39 CON(C)CCNC(=O)[C@@H]1CCc2nnc(-c3ccccc3)n2C1 ZINC000880647452 ED On-Demand Anodyne PDE8B 48 34 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild PAPA1_CARPA 45 37 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild CTSK 24 42 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild CTSL 24 42 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild CTSS 18 42 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild ACE2 46 32 CON(C)CCNC(=O)[C@H](C)Cc1ccc(C#N)cc1 ZINC000880647465 CD On-Demand Mild CTRB_BOVIN 47 34 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild PAPA1_CARPA 45 37 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild CTSK 24 42 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild CTSL 24 42 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild CTSS 18 42 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild ACE2 46 32 CON(C)CCNC(=O)[C@@H](C)Cc1ccc(C#N)cc1 ZINC000880647466 CD On-Demand Mild CTRB_BOVIN 47 34 CON(C)CCNC(=O)Cc1c(Cl)cccc1Br ZINC000880647468 EE On-Demand Anodyne P2RX7 29 43 CON(C)CCNC(=O)[C@@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880647483 FD On-Demand Anodyne GHSR 15 40 CON(C)CCNC(=O)[C@@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880647483 FD On-Demand Anodyne SLC12A5 55 40 CON(C)CCNC(=O)[C@@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880647484 FD On-Demand Anodyne GHSR 15 40 CON(C)CCNC(=O)[C@@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880647484 FD On-Demand Anodyne SLC12A5 55 40 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1C1CC1 ZINC000880647489 ED On-Demand Anodyne ACHE 23 40 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1C1CC1 ZINC000880647489 ED On-Demand Anodyne SIGMAR1 28 41 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000880647589 DF On-Demand Anodyne SLC6A4 21 45 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccc(Cl)c(Cl)c1 ZINC000880647589 DF On-Demand Anodyne SLC6A3 27 45 CON(C)CCNC(=O)Cc1cc2cc(Cl)ccc2[nH]1 ZINC000880647599 CD On-Demand Anodyne PYGL 81 47 CON(C)CCNC(=O)Cn1cncc1C ZINC000880647618 BB On-Demand Anodyne QPCT 52 35 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccncc1 ZINC000880647687 FD On-Demand Anodyne ACHE 15 40 CON(C)CCNC(=O)[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccncc1 ZINC000880647687 FD On-Demand Anodyne SIGMAR1 17 48 COc1cccc([C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC)c1 ZINC000880647690 FD On-Demand Anodyne CTSL 21 41 COc1cccc([C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC)c1 ZINC000880647690 FD On-Demand Anodyne MTNR1A 60 42 COc1cccc([C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC)c1 ZINC000880647690 FD On-Demand Anodyne MTNR1B 54 39 COc1cccc([C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC)c1 ZINC000880647690 FD On-Demand Anodyne CTSS 15 41 COc1ccccc1Cn1cnc2cc(C(=O)NCCN(C)OC)ccc21 ZINC000880647694 FE On-Demand Anodyne DRD3 21 40 COc1ccccc1Cn1cnc2cc(C(=O)NCCN(C)OC)ccc21 ZINC000880647694 FE On-Demand Anodyne NR1I2 42 32 CON(C)CCNC(=O)[C@@H]1CC[C@@H](C)CC1 ZINC000880647706 BD On-Demand Anodyne MTNR1A 17 40 CO[C@H]1CN(C(=O)OCc2ccccc2)[C@](C)(C(=O)NCCN(C)OC)C1 ZINC000880647713 GD On-Demand Anodyne SLC12A5 49 36 CO[C@@H]1CN(C(=O)OCc2ccccc2)[C@](C)(C(=O)NCCN(C)OC)C1 ZINC000880647714 GD On-Demand Anodyne SLC12A5 49 36 CO[C@@H]1CN(C(=O)OCc2ccccc2)[C@@](C)(C(=O)NCCN(C)OC)C1 ZINC000880647715 GD On-Demand Anodyne SLC12A5 49 36 CO[C@H]1CN(C(=O)OCc2ccccc2)[C@@](C)(C(=O)NCCN(C)OC)C1 ZINC000880647716 GD On-Demand Anodyne SLC12A5 49 36 CON(C)CCNC(=O)CN1c2ccccc2Sc2ccccc21 ZINC000880647722 EF On-Demand Anodyne BCHE 15 48 CON(C)CCNC(=O)Cc1cc2ccccc2c(O)n1 ZINC000880647748 CD On-Demand Anodyne POLR1A 42 36 COc1cccc(Oc2ccc(C(=O)NCCN(C)OC)nc2)c1 ZINC000880647802 EE On-Demand Anodyne DRD4 45 34 COc1cccc(Oc2ccc(C(=O)NCCN(C)OC)nc2)c1 ZINC000880647802 EE On-Demand Anodyne MTNR1A 67 43 COc1cccc(Oc2ccc(C(=O)NCCN(C)OC)nc2)c1 ZINC000880647802 EE On-Demand Anodyne MTNR1B 61 43 COc1cccc(Oc2ccc(C(=O)NCCN(C)OC)nc2)c1 ZINC000880647802 EE On-Demand Anodyne ROCK2 42 36 CON(C)CCNC(=O)C(=O)N1CCN(c2ccccc2)CC1 ZINC000880647812 DB On-Demand Anodyne HTR1A 23 43 CON(C)CCNC(=O)C(=O)N1CCN(c2ccccc2)CC1 ZINC000880647812 DB On-Demand Anodyne DRD3 24 41 CON(C)CCNC(=O)[C@@H](C)c1ccc2c(c1)OCO2 ZINC000880647823 CD On-Demand Anodyne EDNRB 60 38 CON(C)CCNC(=O)[C@@H](C)c1ccc2c(c1)OCO2 ZINC000880647823 CD On-Demand Anodyne EDNRA 59 37 CON(C)CCNC(=O)[C@@H](C)c1ccc2c(c1)OCO2 ZINC000880647823 CD On-Demand Anodyne BMP1 50 37 CON(C)CCNC(=O)[C@@H](C)c1ccc2c(c1)OCO2 ZINC000880647823 CD On-Demand Anodyne TRPV1 45 32 CON(C)CCNC(=O)[C@@H](C)c1ccc2c(c1)OCO2 ZINC000880647823 CD On-Demand Anodyne DYRK2 52 36 CON(C)CCNC(=O)/C(C)=C\c1ccccc1Cl ZINC000880647855 CE On-Demand Anodyne ECR 50 35 CON(C)CCNC(=O)/C(C)=C\c1ccccc1Cl ZINC000880647855 CE On-Demand Anodyne TLR4 17 48 CON(C)CCNC(=O)/C(C)=C/c1ccccc1Cl ZINC000880647856 CE On-Demand Anodyne ECR 50 35 CON(C)CCNC(=O)/C(C)=C/c1ccccc1Cl ZINC000880647856 CE On-Demand Anodyne TLR4 17 48 CON(C)CCNC(=O)[C@@H](NC(C)=O)C(C)(C)C ZINC000880647864 CC On-Demand Anodyne PDF 52 31 CON(C)CCNC(=O)[C@@H]1C[C@H]1C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880647865 FD On-Demand Anodyne GPR119 30 42 CCN(C)C(=O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647883 FF On-Demand Anodyne TSHR 46 30 CCN(C)C(=O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647883 FF On-Demand Anodyne KCNK3 45 39 CCN(C)C(=O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880647883 FF On-Demand Anodyne KCNK9 43 39 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne ALOX5 20 61 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne TSHR 40 31 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MAOB 35 45 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne CYSLTR1 18 43 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MME 15 40 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne LTA4H 65 47 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne PTGER3 56 37 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MMP13 16 42 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne ADAM17 25 42 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne CA5B 16 40 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne CA5A 19 40 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MTNR1A 42 38 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MTNR1B 35 42 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne FAAH 17 40 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne SLC6A5 42 38 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MMP9 15 42 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne ACE2 17 40 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne ADAMTS4 27 42 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne NPR 45 33 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne TAAR1 21 51 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne FFAR1 48 47 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne FFAR4 47 38 CON(C)CCNC(=O)Cc1ccc(OCc2ccccc2)cc1 ZINC000880647886 EE On-Demand Anodyne MBTPS1 18 41 CON(C)CCNC(=O)Cc1ccc(F)c(Cl)c1 ZINC000880647887 CD On-Demand Anodyne NCE103 17 52 CON(C)CCNC(=O)[C@H](C)Cc1ccccc1C ZINC000880647892 CD On-Demand Anodyne ANPEP 28 43 CON(C)CCNC(=O)[C@H](C)Cc1ccccc1C ZINC000880647892 CD On-Demand Anodyne ACE2 41 33 CON(C)CCNC(=O)[C@H](C)Cc1ccccc1C ZINC000880647892 CD On-Demand Anodyne AMP1_PLAFQ 30 41 CON(C)CCNC(=O)[C@@H](C)Cc1ccccc1C ZINC000880647893 CD On-Demand Anodyne ANPEP 28 43 CON(C)CCNC(=O)[C@@H](C)Cc1ccccc1C ZINC000880647893 CD On-Demand Anodyne ACE2 41 33 CON(C)CCNC(=O)[C@@H](C)Cc1ccccc1C ZINC000880647893 CD On-Demand Anodyne AMP1_PLAFQ 30 41 CON(C)CCNC(=O)[C@@H](F)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880647898 ED On-Demand Anodyne GPR119 28 45 CON(C)CCNC(=O)[C@@H](F)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880647902 ED On-Demand Anodyne GPR119 28 45 COc1cccc(C(=O)NCCN(C)OC)c1C ZINC000880647918 CD On-Demand Anodyne ECR 28 50 COc1cccc(C(=O)NCCN(C)OC)c1C ZINC000880647918 CD On-Demand Anodyne KCNA3 42 40 COc1cccc(C(=O)NCCN(C)OC)c1C ZINC000880647918 CD On-Demand Anodyne E3UJZ5_SPOLI 20 49 COc1cccc(C(=O)NCCN(C)OC)c1C ZINC000880647918 CD On-Demand Anodyne KCNK3 59 43 COc1cccc(C(=O)NCCN(C)OC)c1C ZINC000880647918 CD On-Demand Anodyne KCNK9 53 43 CON(C)CCNC(=O)[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000880647934 EG On-Demand Anodyne NPY1R 20 43 CON(C)CCNC(=O)[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000880647934 EG On-Demand Anodyne UTS2 64 51 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne ELANE 32 44 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CASP3 18 42 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne BMP1 20 41 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne KLK3 85 38 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CTSB 87 49 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne PAPA1_CARPA 95 46 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CYSP_TRYCR 57 44 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CTSK 46 51 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CTSL 57 49 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne PGA 29 41 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne AMY2 55 32 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CAPNS1 73 43 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne MMP2 24 40 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne MMP3 38 40 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne MMP8 15 40 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne MMP11 51 31 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CTSS 34 51 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CAPN1 98 56 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CASP1 26 44 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CAPN2 146 44 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CASP6 15 42 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne CASP9 31 42 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne TPSAB1 42 38 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne NPR 90 48 CON(C)CCNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C ZINC000880647946 FD On-Demand Anodyne PSMB5 45 42 CNc1ccc(C(F)(F)F)cc1C(=O)NCCN(C)OC ZINC000880647951 DD On-Demand Anodyne LIPG 20 40 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne MME 42 38 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne PAPA1_CARPA 43 33 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne MTNR1A 37 42 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne MTNR1B 34 42 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne CAPN2 55 33 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne NPR 70 37 CON(C)CCNC(=O)[C@@H](C)OCCc1ccccc1 ZINC000880647956 CD On-Demand Anodyne AMP1_PLAFQ 34 40 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne MME 42 38 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne PAPA1_CARPA 43 33 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne MTNR1A 37 42 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne MTNR1B 34 42 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne CAPN2 55 33 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne NPR 70 37 CON(C)CCNC(=O)[C@H](C)OCCc1ccccc1 ZINC000880647960 CD On-Demand Anodyne AMP1_PLAFQ 34 40 CON(C)CCNC(=O)Cc1coc2ccc(C)cc12 ZINC000880647966 CD On-Demand Anodyne NQO2 22 44 CON(C)CCNC(=O)Cc1coc2ccc(C)cc12 ZINC000880647966 CD On-Demand Anodyne MTNR1A 16 48 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne DRD2 18 40 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne TSHR 41 31 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne DRD4 19 40 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne HTR1D 15 43 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne HTR1B 17 43 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne DRD3 18 40 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne PDGFRB 46 40 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647988 GG On-Demand Anodyne ABCB1 20 41 CON(C)CCNC(=O)[C@@H]1CC(=O)N(c2ccc(C#N)c(Cl)c2)C1 ZINC000880647989 FD On-Demand Mild AR 16 42 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne DRD2 18 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne TSHR 41 31 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne DRD4 19 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne HTR1D 15 43 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne HTR1B 17 43 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne DRD3 18 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne PDGFRB 46 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880647990 GG On-Demand Anodyne ABCB1 20 41 COC[C@]1(CO)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648019 GF On-Demand Anodyne ABCB1 15 41 COC[C@]1(CO)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648019 GF On-Demand Anodyne EPHX2 30 40 CCC1(CNC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)COC1 ZINC000880648032 FG On-Demand Anodyne KCNK3 48 42 COC[C@]1(C)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648087 GH On-Demand Anodyne ABCB1 19 41 COC[C@@]1(C)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648089 GH On-Demand Anodyne ABCB1 19 41 CON(C)CCNC(=O)[C@@H]1CCCC[C@@H]1c1ccccc1 ZINC000880648094 CF On-Demand Anodyne AMY2 45 32 CON(C)CCNC(=O)[C@@H]1CCN(c2ccccc2)C1 ZINC000880648155 CD On-Demand Anodyne SLC6A1 40 32 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne ACE 34 40 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne PPARA 16 40 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne MME 112 44 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne ANPEP 48 39 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne FCER2 41 32 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne PAPA1_CARPA 59 40 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne CPA1 46 36 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne CAPNS1 53 33 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne MMP8 16 40 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne CAPN1 51 40 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne CAPN2 47 33 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne ACE2 42 36 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne FPR1 40 33 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne NPR 56 38 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne AMP1_PLAFQ 54 42 CO[C@@H](Cc1ccccc1)C(=O)NCCN(C)OC ZINC000880648164 CC On-Demand Anodyne NPFFR1 41 31 CON(C)CCNC(=O)[C@@H](NC(=O)OC(C)(C)C)C(F)(F)F ZINC000880648167 ED On-Demand Anodyne PAPA1_CARPA 38 40 COCC(COC)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648208 FF On-Demand Anodyne KCNK3 47 44 COCC(COC)NC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648208 FF On-Demand Anodyne KCNK9 35 40 C=CCOc1ccc(CC(=O)NCCN(C)OC)cc1 ZINC000880648209 CD On-Demand Mild MTNR1A 27 46 C=CCOc1ccc(CC(=O)NCCN(C)OC)cc1 ZINC000880648209 CD On-Demand Mild CA9 15 40 CC[C@H](Nc1cccnc1Cl)C(=O)NCCN(C)OC ZINC000880648236 DD On-Demand Anodyne G2YM83_BOTF4 62 32 CC[C@@H](Nc1cccnc1Cl)C(=O)NCCN(C)OC ZINC000880648237 DD On-Demand Anodyne G2YM83_BOTF4 62 32 CON(C)CCNC(=O)C1CCc2ccccc2CC1 ZINC000880648250 CD On-Demand Anodyne MTNR1A 36 41 CON(C)CCNC(=O)C1CCc2ccccc2CC1 ZINC000880648250 CD On-Demand Anodyne MTNR1B 37 40 CON(C)CCNC(=O)[C@@H](c1ccc(Cl)cc1)N(C)C ZINC000880648283 CD On-Demand Anodyne UTS2 47 37 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)c(C)c1 ZINC000880648296 EE On-Demand Anodyne DRD4 41 32 COc1ccc(-c2cncc(C(=O)NCCN(C)OC)c2)c(C)c1 ZINC000880648296 EE On-Demand Anodyne CYP11B2 18 42 CON(C)CCNC(=O)CCCc1cccnc1 ZINC000880648299 CD On-Demand Anodyne TBXAS1 63 47 CON(C)CCNC(=O)CCCc1cccnc1 ZINC000880648299 CD On-Demand Anodyne PTAFR 41 53 CON(C)CCNC(=O)COc1cc(Cl)ccc1C ZINC000880648381 CD On-Demand Anodyne MCHR2 25 41 CON(C)CCNC(=O)COc1cc(Cl)ccc1C ZINC000880648381 CD On-Demand Anodyne PTGDR2 22 40 CON(C)CCNC(=O)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880648382 DE On-Demand Anodyne C3AR1 45 44 COCC1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648406 GH On-Demand Anodyne TSHR 46 30 COCC1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648406 GH On-Demand Anodyne HTR1B 15 48 COCC1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648406 GH On-Demand Anodyne PDGFRB 55 44 COCC1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648406 GH On-Demand Anodyne CCR3 24 42 COCC1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648406 GH On-Demand Anodyne ABCB1 20 44 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648408 GG On-Demand Anodyne DRD2 15 41 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648408 GG On-Demand Anodyne DRD4 23 40 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648408 GG On-Demand Anodyne EPHX2 49 56 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648408 GG On-Demand Anodyne CCR8 43 34 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648409 GG On-Demand Anodyne DRD2 15 41 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648409 GG On-Demand Anodyne DRD4 23 40 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648409 GG On-Demand Anodyne EPHX2 49 56 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648409 GG On-Demand Anodyne CCR8 43 34 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880648422 ED On-Demand Mild PAPA1_CARPA 40 43 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN(C)OC ZINC000880648435 ED On-Demand Mild PAPA1_CARPA 40 43 CON(C)CCNC(=O)C1CCC(C2CC2)CC1 ZINC000880648442 CD On-Demand Anodyne MTNR1A 19 40 COCCOC1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648455 GF On-Demand Anodyne TSHR 40 30 COCCOC1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648455 GF On-Demand Anodyne PDGFRB 40 39 COCCOC1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648455 GF On-Demand Anodyne ABCB1 19 41 COCCOC1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648455 GF On-Demand Anodyne KCNK3 43 42 COc1ccc2c(c1)CC[C@H]2C(=O)NCCN(C)OC ZINC000880648486 CD On-Demand Anodyne NQO2 40 45 COc1ccc2c(c1)CC[C@H]2C(=O)NCCN(C)OC ZINC000880648486 CD On-Demand Anodyne PPARD 37 42 COc1ccc2c(c1)CC[C@H]2C(=O)NCCN(C)OC ZINC000880648486 CD On-Demand Anodyne MTNR1A 79 44 COc1ccc2c(c1)CC[C@H]2C(=O)NCCN(C)OC ZINC000880648486 CD On-Demand Anodyne MTNR1B 64 39 COc1ccc2c(c1)CC[C@H]2C(=O)NCCN(C)OC ZINC000880648486 CD On-Demand Anodyne GHSR 22 44 CON(C)CCNC(=O)C(C)(C)c1ccc(C#N)cc1 ZINC000880648502 CD On-Demand Mild CTRB_BOVIN 45 33 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne HTR1B 16 48 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne PDGFRB 56 45 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne NPY5R 23 40 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne ABCB1 22 47 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne S1PR2 28 42 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648513 GF On-Demand Anodyne ENPP1 55 32 O=C(COC1CC1)NC1(c2cccc(C(F)(F)F)c2)CC1 ZINC000880648555 CF On-Demand Anodyne TACR1 35 40 O=C(COC1CC1)NC1(c2cccc(C(F)(F)F)c2)CC1 ZINC000880648555 CF On-Demand Anodyne CCR2 50 38 COCC1=CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880648563 GH On-Demand Anodyne ABCB1 20 41 CON(C)CCNC(=O)[C@@H]1COc2cc(F)ccc2C1 ZINC000880648571 CC On-Demand Anodyne ROCK2 27 42 CON(C)CCNC(=O)[C@@H]1CC[C@@H](c2ccccc2)C1 ZINC000880648690 CE On-Demand Anodyne MTNR1A 20 43 CON(C)CCNC(=O)[C@@H]1CC[C@@H](c2ccccc2)C1 ZINC000880648690 CE On-Demand Anodyne MTNR1B 17 43 COc1ccccc1-c1ccc(C(=O)NCCN(C)OC)s1 ZINC000880648745 DF On-Demand Anodyne DRD3 22 43 COc1ccccc1-c1ccc(C(=O)NCCN(C)OC)s1 ZINC000880648745 DF On-Demand Anodyne HSD17B2 38 44 CNC(=O)CCCN(C)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648769 GF On-Demand Anodyne ENPP1 64 31 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne TSHR 48 31 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne PDGFRB 52 42 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne CCR3 18 50 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne ABCB1 20 42 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne QRFPR 40 40 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880648792 GH On-Demand Anodyne ACKR3 57 33 CON(C)CCNC(=O)Cc1cccc2ncccc12 ZINC000880648796 CD On-Demand Anodyne MTNR1A 39 41 CON(C)CCNC(=O)Cc1cccc2ncccc12 ZINC000880648796 CD On-Demand Anodyne MTNR1B 30 41 CON(C)CCNC(=O)C[C@@H](n1ccnc1)C(F)(F)F ZINC000880648810 CC On-Demand Anodyne CYP26A1 86 35 CON(C)CCNC(=O)C[C@H](n1ccnc1)C(F)(F)F ZINC000880648811 CC On-Demand Anodyne CYP26A1 86 35 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne F2 33 42 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne FKBP1A 45 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne ELANE 50 37 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne PREP 51 35 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne TMPRSS11D 43 32 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648816 GF On-Demand Anodyne ACKR3 57 33 COc1cccc(C(C)(C)C(=O)NCCN(C)OC)c1 ZINC000880648824 CD On-Demand Anodyne DRD4 42 32 COc1cccc(C(C)(C)C(=O)NCCN(C)OC)c1 ZINC000880648824 CD On-Demand Anodyne MTNR1A 69 44 COc1cccc(C(C)(C)C(=O)NCCN(C)OC)c1 ZINC000880648824 CD On-Demand Anodyne MTNR1B 61 44 CON(C)CCNC(=O)[C@@H]1Cc2ccccc2CO1 ZINC000880648832 CC On-Demand Anodyne ADAM9 48 31 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880648835 DC On-Demand Anodyne SLC18A3 21 46 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880648835 DC On-Demand Anodyne EPHX2 20 47 CON(C)CCNC(=O)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880648835 DC On-Demand Anodyne L3MBTL3 62 36 CON(C)CCNC(=O)Cc1cccc2cnccc12 ZINC000880648849 CD On-Demand Anodyne TRPV1 18 46 CON(C)CCNC(=O)Cc1cccc2cnccc12 ZINC000880648849 CD On-Demand Anodyne MTNR1A 39 40 COC[C@@H](CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1)OC ZINC000880648863 FF On-Demand Anodyne ADRB1 40 31 COC[C@@H](CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1)OC ZINC000880648863 FF On-Demand Anodyne TSHR 40 30 COCC[C@](C)(O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648886 GF On-Demand Anodyne KCNK3 43 42 COCC[C@@](C)(O)CNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880648887 GF On-Demand Anodyne KCNK3 43 42 CON(C)CCNC(=O)[C@@]1(C)CC(c2ccccc2)=NO1 ZINC000880648907 CD On-Demand Anodyne NPPA 43 33 CON(C)CCNC(=O)Cc1coc2cc(Cl)ccc12 ZINC000880648910 CE On-Demand Anodyne MTNR1A 16 40 CON(C)CCNC(=O)Cc1ccc(O)c(Cl)c1 ZINC000880648926 CD On-Demand Anodyne NCE103 23 71 CON(C)CCNC(=O)Cc1ccc(O)c(Cl)c1 ZINC000880648926 CD On-Demand Anodyne P96878_MYCTU 18 61 COC(=O)c1cc(C(=O)NCCN(C)OC)ccc1C ZINC000880648945 CD On-Demand Anodyne DRD4 40 32 COC(=O)c1cc(C(=O)NCCN(C)OC)ccc1C ZINC000880648945 CD On-Demand Anodyne MAPK14 18 40 CON(C)CCNC(=O)C1(c2ccc([N+](=O)[O-])cc2)CCC1 ZINC000880648949 DD On-Demand Bother SLC27A4 53 35 CON(C)CCNC(=O)[C@@H](C)n1ccc(C(F)(F)F)n1 ZINC000880649016 CD On-Demand Anodyne CARM1 58 34 CON(C)CCNC(=O)C1(O)CN(C(=O)OCc2ccccc2)C1 ZINC000880649023 EB On-Demand Anodyne SLC12A5 56 38 CS(=O)(=O)C1CCC(C(=O)NC2(c3cccc(C(F)(F)F)c3)CC2)CC1 ZINC000880649056 GG On-Demand Anodyne CACNA1B 52 33 CON(C)CCNC(=O)CCc1cccc2ccccc12 ZINC000880649062 CE On-Demand Anodyne NQO2 42 43 CON(C)CCNC(=O)CCc1cccc2ccccc12 ZINC000880649062 CE On-Demand Anodyne MTNR1A 94 53 CON(C)CCNC(=O)CCc1cccc2ccccc12 ZINC000880649062 CE On-Demand Anodyne MTNR1B 70 42 COCCN(CCO)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880649064 FE On-Demand Anodyne KCNK3 49 43 COCCN(CCO)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880649064 FE On-Demand Anodyne KCNK9 43 39 CON(C)CCNC(=O)Cc1ccccc1C(=O)OC(C)(C)C ZINC000880649089 DD On-Demand Anodyne ECR 41 36 CCOC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649093 GH On-Demand Anodyne PDGFRB 49 41 CCOC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649093 GH On-Demand Anodyne CCR3 20 45 CCOC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649093 GH On-Demand Anodyne ABCB1 16 41 CON(C)CCNC(=O)CCc1ccc(N2CCCS2(=O)=O)cc1 ZINC000880649095 FC On-Demand Anodyne CDK1 17 42 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649163 GH On-Demand Anodyne HTR1B 15 48 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649163 GH On-Demand Anodyne PDGFRB 56 45 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649163 GH On-Demand Anodyne NPY5R 21 40 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649163 GH On-Demand Anodyne ABCB1 22 45 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649163 GH On-Demand Anodyne S1PR2 30 44 COc1ccccc1-n1nccc1[C@@H]1OCC[C@H]1C(=O)NCCN(C)OC ZINC000880649208 FD On-Demand Anodyne HTR1A 21 41 CON(C)CCNC(=O)[C@@H]1CC[C@H]1c1ccc(F)cc1 ZINC000880649215 CD On-Demand Anodyne SLC6A4 18 41 CON(C)CCNC(=O)[C@@H]1CC[C@H]1c1ccc(F)cc1 ZINC000880649215 CD On-Demand Anodyne SLC6A3 30 41 CON(C)CCNC(=O)[C@@H]1CC[C@@H]1c1ccc(F)cc1 ZINC000880649216 CD On-Demand Anodyne SLC6A4 18 41 CON(C)CCNC(=O)[C@@H]1CC[C@@H]1c1ccc(F)cc1 ZINC000880649216 CD On-Demand Anodyne SLC6A3 30 41 COC[C@@H](O)CCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880649239 FE On-Demand Anodyne ADRB1 47 36 CNC(=O)CCN(C)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880649278 FF On-Demand Anodyne KCNK3 60 44 CNC(=O)CCN(C)C(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880649278 FF On-Demand Anodyne KCNK9 44 40 CON(C)CCNC(=O)[C@@](C)(Cc1ccccc1)C(C)C ZINC000880649305 CF On-Demand Anodyne PAPA1_CARPA 50 38 CON(C)CCNC(=O)[C@@](C)(Cc1ccccc1)C(C)C ZINC000880649305 CF On-Demand Anodyne TACR3 19 41 CON(C)CCNC(=O)[C@@](C)(Cc1ccccc1)C(C)C ZINC000880649305 CF On-Demand Anodyne NPR 51 33 CON(C)CCNC(=O)Cc1ccc(OCc2ccncc2)cc1 ZINC000880649312 ED On-Demand Anodyne CYP26A1 28 40 CON(C)CCNC(=O)[C@@H]1C[C@H]1c1ccsc1 ZINC000880649323 CD On-Demand Anodyne NPBWR1 79 32 CON(C)CCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880649331 CD On-Demand Anodyne GABRA1 16 50 CON(C)CCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880649331 CD On-Demand Anodyne MPO 64 38 CON(C)CCNC(=O)[C@@H]1CCC(=O)N1C(C)C ZINC000880649366 CB On-Demand Anodyne P2RX7 30 51 CON(C)CCNC(=O)[C@@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880649412 ED On-Demand Anodyne HSD11B1 19 41 CON(C)CCNC(=O)[C@@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880649412 ED On-Demand Anodyne P2RX7 25 40 CON(C)CCNC(=O)[C@@H]1CCCN1Cc1ccc(Cl)cc1 ZINC000880649412 ED On-Demand Anodyne CCR1 15 44 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649416 GG On-Demand Anodyne TSHR 42 31 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649416 GG On-Demand Anodyne HTR1B 16 49 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649416 GG On-Demand Anodyne PDGFRB 50 44 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649416 GG On-Demand Anodyne ABCB1 18 44 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)CC1 ZINC000880649416 GG On-Demand Anodyne RBP4 26 42 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne INHA 40 32 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne TRPV1 19 52 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne MTNR1A 27 40 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne MTNR1B 26 40 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne HDAC1 15 40 COc1ccc(CC(=O)NCCN(C)OC)cc1O ZINC000880649433 CC On-Demand Anodyne NCE103 15 52 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C[C@H]1O ZINC000880649436 FG On-Demand Anodyne PDGFRB 34 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C[C@H]1O ZINC000880649436 FG On-Demand Anodyne ABCB1 17 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C[C@@H]1O ZINC000880649438 FG On-Demand Anodyne PDGFRB 34 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C[C@@H]1O ZINC000880649438 FG On-Demand Anodyne ABCB1 17 42 CON(C)CCNC(=O)CCNC(=O)c1cc2ccccc2[nH]1 ZINC000880649446 DC On-Demand Anodyne PYGL 60 44 CON(C)CCNC(=O)CCNC(=O)c1cc2ccccc2[nH]1 ZINC000880649446 DC On-Demand Anodyne PLD2 27 41 CON(C)CCNC(=O)[C@H](C)CCc1ccc(F)cc1 ZINC000880649463 CE On-Demand Anodyne LEF 58 39 CON(C)CCNC(=O)[C@@H](C)CCc1ccc(F)cc1 ZINC000880649464 CE On-Demand Anodyne LEF 58 39 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649478 GF On-Demand Anodyne SLC6A1 53 40 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649478 GF On-Demand Anodyne NPY2R 27 41 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649478 GF On-Demand Anodyne ABCB1 17 41 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880649478 GF On-Demand Anodyne ACKR3 57 33 COC(=O)[C@@H](CC(C)C)N(C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880649490 EF On-Demand Anodyne MPO 57 34 Cc1ccc(NC(=O)N2CC3(CC3)C2)cc1C(=O)c1ccccc1 ZINC000880649492 DH On-Demand Anodyne NPY5R 19 42 Cc1ccc(NC(=O)N2CC3(CC3)C2)cc1C(=O)c1ccccc1 ZINC000880649492 DH On-Demand Anodyne EPHX2 29 44 Cc1ccc(NC(=O)N2CC3(CC3)C2)cc1C(=O)c1ccccc1 ZINC000880649492 DH On-Demand Anodyne P2RY14 42 33 Cc1ccc(NC(=O)N2CC3(CC3)C2)cc1C(=O)c1ccccc1 ZINC000880649492 DH On-Demand Anodyne KCNK3 45 40 Cc1ccc(NC(=O)N2CCC3(CCNC3=O)CC2)cc1C(=O)c1ccccc1 ZINC000880649497 GG On-Demand Anodyne CACNA1H 46 38 Cc1ccc(NC(=O)N2CCC3(CCNC3=O)CC2)cc1C(=O)c1ccccc1 ZINC000880649497 GG On-Demand Anodyne NPY5R 28 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nnc(O)n1C)C2 ZINC000880649501 DC On-Demand Anodyne NQO2 33 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nnc(O)n1C)C2 ZINC000880649501 DC On-Demand Anodyne MTNR1A 46 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nnc(O)n1C)C2 ZINC000880649501 DC On-Demand Anodyne MTNR1B 40 40 Cc1ccc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)cc1C(=O)c1ccccc1 ZINC000880649521 GG On-Demand Anodyne NPY2R 42 35 Cc1ccc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)cc1C(=O)c1ccccc1 ZINC000880649522 GG On-Demand Anodyne NPY2R 42 35 CCCCCCCC[C@@H](C)C(=O)NCc1nnc(O)n1C ZINC000880649567 CF On-Demand Mild NOD1 67 37 CCCCCCCC[C@H](C)C(=O)NCc1nnc(O)n1C ZINC000880649568 CF On-Demand Mild NOD1 67 37 COc1cccc(C(C)(C)C(=O)NCc2nnc(O)n2C)c1 ZINC000880649573 DD On-Demand Anodyne DRD4 42 32 C=CC(C)(C)CC(=O)N1CCCC[C@@H]1c1n[nH]c(COC)n1 ZINC000880649578 DF On-Demand Mild CPT1A 95 38 C=CC(C)(C)CC(=O)N1CCCC[C@H]1c1n[nH]c(COC)n1 ZINC000880649579 DF On-Demand Mild CPT1A 95 38 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880649589 EE On-Demand Mild ITK 18 51 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880649589 EE On-Demand Mild PANC 58 39 C[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649596 DG On-Demand Mild ITK 28 49 C[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649596 DG On-Demand Mild PANC 55 39 C[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649597 DG On-Demand Mild ITK 28 49 C[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649597 DG On-Demand Mild PANC 55 39 CCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649598 CE On-Demand Mild ITK 24 55 CCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649598 CE On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4OCCO4)CC3)cn2)cc1 ZINC000880649613 GE On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4OCCO4)CC3)cn2)cc1 ZINC000880649613 GE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C(=O)C4CC4)CC3)cn2)cc1 ZINC000880649615 GD On-Demand Mild ITK 19 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C(=O)C4CC4)CC3)cn2)cc1 ZINC000880649615 GD On-Demand Mild MLNR 23 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C(=O)C4CC4)CC3)cn2)cc1 ZINC000880649615 GD On-Demand Mild PANC 55 38 CC(C)(C)N1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649616 GG On-Demand Mild ITK 15 48 CC(C)(C)N1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649616 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N(Cc3cccs3)C3CC3)cn2)cc1 ZINC000880649625 GI On-Demand Mild ITK 19 48 N#Cc1ccc(Cn2cc(NC(=O)N(Cc3cccs3)C3CC3)cn2)cc1 ZINC000880649625 GI On-Demand Mild PANC 53 35 CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649627 EG On-Demand Mild ITK 19 48 CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649627 EG On-Demand Mild PANC 54 38 CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649628 EG On-Demand Mild ITK 19 48 CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649628 EG On-Demand Mild PANC 54 38 Cc1ccc(N2CCCC2)c(C(=O)NCc2nnc(O)n2C)c1 ZINC000880649634 DD On-Demand Anodyne KCNQ2 45 36 CN(C[C@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649637 FF On-Demand Mild ITK 34 45 CN(C[C@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649637 FF On-Demand Mild PANC 62 43 CN(C[C@@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649638 FF On-Demand Mild ITK 34 45 CN(C[C@@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649638 FF On-Demand Mild PANC 62 43 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)on1 ZINC000880649643 GG On-Demand Mild ITK 16 43 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)on1 ZINC000880649643 GG On-Demand Mild PANC 60 41 COc1cccc(OC)c1C(=O)NCc1nnc(O)n1C ZINC000880649645 CC On-Demand Anodyne DRD2 22 43 COc1cccc(OC)c1C(=O)NCc1nnc(O)n1C ZINC000880649645 CC On-Demand Anodyne DRD4 41 31 COc1cccc(OC)c1C(=O)NCc1nnc(O)n1C ZINC000880649645 CC On-Demand Anodyne ALS 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880649646 GF On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880649646 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880649647 GF On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880649647 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCCSCC3)cn2)cc1 ZINC000880649667 EF On-Demand Mild ITK 15 51 CC[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649670 DG On-Demand Mild DPP4 15 42 CC[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649670 DG On-Demand Mild ITK 18 49 CC[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649670 DG On-Demand Mild PANC 55 38 CC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649671 DG On-Demand Mild DPP4 15 42 CC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649671 DG On-Demand Mild ITK 18 49 CC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649671 DG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)(F)F)CC3)cn2)cc1 ZINC000880649680 GF On-Demand Mild ITK 15 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)(F)F)CC3)cn2)cc1 ZINC000880649680 GF On-Demand Mild FAAH 17 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)(F)F)CC3)cn2)cc1 ZINC000880649680 GF On-Demand Mild PANC 40 35 Cc1ccc(NC(=O)N2CCCNC(=O)C2)cc1C(=O)c1ccccc1 ZINC000880649810 FF On-Demand Anodyne P2RY14 50 37 COC(=O)[C@@H](CC(C)C)N(C)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880649839 FE On-Demand Anodyne KCNQ2 44 34 CCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649869 CD On-Demand Mild ASAH1 48 35 CCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649869 CD On-Demand Mild LASR 47 33 CCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649869 CD On-Demand Mild NOD1 61 39 CCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649869 CD On-Demand Mild CQSS 55 35 CCCN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649870 DG On-Demand Mild ITK 17 52 N#Cc1ccc(Cn2cc(NC(=O)N(C[C@@H]3CCOC3)C3CC3)cn2)cc1 ZINC000880649872 FF On-Demand Mild ITK 16 46 N#Cc1ccc(Cn2cc(NC(=O)N(C[C@@H]3CCOC3)C3CC3)cn2)cc1 ZINC000880649872 FF On-Demand Mild PANC 52 35 N#Cc1ccc(Cn2cc(NC(=O)N(C[C@H]3CCOC3)C3CC3)cn2)cc1 ZINC000880649874 FF On-Demand Mild ITK 16 46 N#Cc1ccc(Cn2cc(NC(=O)N(C[C@H]3CCOC3)C3CC3)cn2)cc1 ZINC000880649874 FF On-Demand Mild PANC 52 35 C/C(=C\C(=O)NCc1nnc(O)n1C)c1cccc(C(F)(F)F)c1 ZINC000880649896 EE On-Demand Anodyne CCR2 66 36 C/C(=C/C(=O)NCc1nnc(O)n1C)c1cccc(C(F)(F)F)c1 ZINC000880649897 EE On-Demand Anodyne CCR2 66 36 CCCN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649898 EE On-Demand Mild ITK 16 51 Cc1cc(-c2nc(C)c(C(=O)NCc3nnc(O)n3C)s2)ccc1F ZINC000880649911 FE On-Demand Anodyne CHRM4 16 42 Cc1cc(-c2nc(C)c(C(=O)NCc3nnc(O)n3C)s2)ccc1F ZINC000880649911 FE On-Demand Anodyne SCD1 32 42 Cc1cc(-c2nc(C)c(C(=O)NCc3nnc(O)n3C)s2)ccc1F ZINC000880649911 FE On-Demand Anodyne SCD 33 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3c3cccs3)cn2)cc1 ZINC000880649919 GI On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3c3cccs3)cn2)cc1 ZINC000880649919 GI On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3c3cccs3)cn2)cc1 ZINC000880649920 GI On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3c3cccs3)cn2)cc1 ZINC000880649920 GI On-Demand Mild PANC 55 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC(C)(C)O1 ZINC000880649923 FF On-Demand Mild ITK 15 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC(C)(C)O1 ZINC000880649923 FF On-Demand Mild PANC 54 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC(C)(C)O1 ZINC000880649924 FF On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC(C)(C)O1 ZINC000880649924 FF On-Demand Mild PANC 54 37 COCCN(CC(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649926 FF On-Demand Mild ITK 21 49 COCCN(CC(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649926 FF On-Demand Mild PANC 41 35 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649931 EG On-Demand Mild ITK 19 52 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649931 EG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CC3)OCCO4)cn2)cc1 ZINC000880649933 FE On-Demand Mild ITK 15 49 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)C(C)(C)c3ccccc3)sc2C1 ZINC000880649934 HI On-Demand Anodyne NPY2R 25 40 CCCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649947 CE On-Demand Mild ASAH1 48 35 CCCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649947 CE On-Demand Mild LASR 47 33 CCCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649947 CE On-Demand Mild NOD1 61 39 CCCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880649947 CE On-Demand Mild CQSS 55 35 CCO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649955 FF On-Demand Mild ITK 18 48 CCO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649955 FF On-Demand Mild MLNR 24 41 CCO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649955 FF On-Demand Mild PANC 55 38 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649962 DG On-Demand Mild ITK 19 50 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649962 DG On-Demand Mild MLNR 37 42 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880649962 DG On-Demand Mild PANC 56 39 CN(C)C(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649963 GE On-Demand Mild ITK 33 48 CN(C)C(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649963 GE On-Demand Mild MLNR 30 48 CN(C)C(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649963 GE On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3C4CCC3CC4)cn2)cc1 ZINC000880649967 DF On-Demand Mild ITK 19 55 N#Cc1ccc(Cn2cc(NC(=O)N3C4CCC3CC4)cn2)cc1 ZINC000880649967 DF On-Demand Mild PANC 58 41 CC(C)[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649970 EG On-Demand Mild DPP4 18 42 CC(C)[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649970 EG On-Demand Mild ITK 18 49 CC(C)[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880649970 EG On-Demand Mild PANC 55 38 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649975 GF On-Demand Mild ITK 16 51 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649975 GF On-Demand Mild MLNR 21 41 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880649975 GF On-Demand Mild PANC 57 40 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(C)c(C(=O)c3ccccc3)c2)C1 ZINC000880650014 GE On-Demand Anodyne NPY5R 15 40 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(C)c(C(=O)c3ccccc3)c2)C1 ZINC000880650014 GE On-Demand Anodyne EPHX2 31 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)CC3)cn2)cc1 ZINC000880650015 ED On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)CC3)cn2)cc1 ZINC000880650015 ED On-Demand Mild MLNR 22 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)CC3)cn2)cc1 ZINC000880650015 ED On-Demand Mild PANC 56 39 C[C@H](NC(=O)c1ncsc1C1CC1)c1cnccn1 ZINC000880650016 CE On-Demand Anodyne MAP1 47 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@H]3C4)cn2)cc1 ZINC000880650027 DF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@H]3C4)cn2)cc1 ZINC000880650027 DF On-Demand Mild PANC 53 35 Cc1noc(C)c1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650031 FG On-Demand Mild ITK 15 47 Cc1noc(C)c1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650031 FG On-Demand Mild PANC 56 38 CCOc1ccccc1C(F)(F)C(=O)NCc1nnc(O)n1C ZINC000880650043 ED On-Demand Anodyne PLK1 43 33 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C ZINC000880650069 DC On-Demand Anodyne PPARG 30 40 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C ZINC000880650069 DC On-Demand Anodyne NQO2 33 41 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C ZINC000880650069 DC On-Demand Anodyne PPARD 39 41 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1nnc(O)n1C ZINC000880650069 DC On-Demand Anodyne MTNR1A 43 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)F)CC3)cn2)cc1 ZINC000880650083 FE On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)F)CC3)cn2)cc1 ZINC000880650083 FE On-Demand Mild MLNR 32 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC(F)F)CC3)cn2)cc1 ZINC000880650083 FE On-Demand Mild FAAH 16 43 CCCOc1ccc(OCC(=O)NCc2nnc(O)n2C)cc1 ZINC000880650090 DD On-Demand Anodyne ADORA1 19 40 CCCOc1ccc(OCC(=O)NCc2nnc(O)n2C)cc1 ZINC000880650090 DD On-Demand Anodyne ADORA2B 39 40 CCCOc1ccc(OCC(=O)NCc2nnc(O)n2C)cc1 ZINC000880650090 DD On-Demand Anodyne MTNR1A 23 41 CCCOc1ccc(OCC(=O)NCc2nnc(O)n2C)cc1 ZINC000880650090 DD On-Demand Anodyne PLA2G4B 76 35 Cc1ccc(NC(=O)N2CCC3(CC2)OCCCO3)cc1C(=O)c1ccccc1 ZINC000880650092 GH On-Demand Anodyne NPY5R 24 41 Cc1ccc(NC(=O)N2CCC3(CC2)OCCCO3)cc1C(=O)c1ccccc1 ZINC000880650092 GH On-Demand Anodyne EPHX2 31 40 COCCCONC(=O)Nc1ccc(C)c(C(=O)c2ccccc2)c1 ZINC000880650109 EG On-Demand Anodyne KCNK3 73 40 COCCCONC(=O)Nc1ccc(C)c(C(=O)c2ccccc2)c1 ZINC000880650109 EG On-Demand Anodyne KCNK9 46 36 C[C@@H](CCc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650113 DD On-Demand Anodyne LEF 40 35 C[C@H](CCc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650114 DD On-Demand Anodyne LEF 40 35 COc1cccc(C(C)(C)C(=O)NCc2cc(O)nc(SC)n2)c1 ZINC000880650127 EF On-Demand Anodyne LHCGR 17 40 CCCCN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650128 EG On-Demand Mild ITK 16 52 CCCCN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650128 EG On-Demand Mild PANC 41 35 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650139 DD On-Demand Mild ITK 22 53 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650139 DD On-Demand Mild MLNR 17 40 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650139 DD On-Demand Mild PANC 53 38 Cn1cccc1[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650152 FH On-Demand Mild ITK 18 46 Cn1cccc1[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650152 FH On-Demand Mild PANC 57 38 Cn1cccc1[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650154 FH On-Demand Mild ITK 18 46 Cn1cccc1[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650154 FH On-Demand Mild PANC 57 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](O)C3)cn2)cc1 ZINC000880650159 ED On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](O)C3)cn2)cc1 ZINC000880650159 ED On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](O)C3)cn2)cc1 ZINC000880650163 ED On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](O)C3)cn2)cc1 ZINC000880650163 ED On-Demand Mild PANC 54 38 CCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650173 CD On-Demand Mild ASAH1 48 35 CCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650173 CD On-Demand Mild LASR 47 33 CCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650173 CD On-Demand Mild NOD1 61 39 CCCCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650173 CD On-Demand Mild CQSS 55 35 CCCN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650179 EG On-Demand Mild ITK 19 49 CCCN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650179 EG On-Demand Mild PANC 54 37 CN(C[C@@H]1CCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650182 EE On-Demand Mild ITK 35 46 CN(C[C@@H]1CCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650182 EE On-Demand Mild PANC 63 43 CC[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650184 EH On-Demand Mild ITK 25 48 CC[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650184 EH On-Demand Mild PANC 54 38 CC[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650185 EH On-Demand Mild ITK 25 48 CC[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650185 EH On-Demand Mild PANC 54 38 CN(C)CCc1ccc(C(=O)NCc2nnc(O)n2C)cc1 ZINC000880650189 DC On-Demand Anodyne UTS2 40 31 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C(F)(F)F)C3)cn2)cc1 ZINC000880650203 GH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C(F)(F)F)C3)cn2)cc1 ZINC000880650203 GH On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C(F)(F)F)C3)cn2)cc1 ZINC000880650204 GH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C(F)(F)F)C3)cn2)cc1 ZINC000880650204 GH On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880650205 FF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880650205 FF On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880650205 FF On-Demand Mild L3MBTL3 74 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880650206 FF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880650206 FF On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880650206 FF On-Demand Mild L3MBTL3 74 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CO)C3)cn2)cc1 ZINC000880650208 EE On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CO)C3)cn2)cc1 ZINC000880650208 EE On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CO)C3)cn2)cc1 ZINC000880650209 EE On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CO)C3)cn2)cc1 ZINC000880650209 EE On-Demand Mild PANC 49 37 CCOc1ccccc1OCC(=O)NCc1nnc(O)n1C ZINC000880650212 DC On-Demand Anodyne HCN1 49 33 CCOc1ccccc1OCC(=O)NCc1nnc(O)n1C ZINC000880650212 DC On-Demand Anodyne HCN4 40 31 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650222 EG On-Demand Mild ITK 18 49 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650222 EG On-Demand Mild MLNR 34 43 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650222 EG On-Demand Mild PANC 55 38 Cc1nc(CNC(=O)CC[C@H]2CCc3ccccc32)sc1C(N)=O ZINC000880650228 EF On-Demand Anodyne NQO2 17 40 Cc1nc(CNC(=O)CC[C@H]2CCc3ccccc32)sc1C(N)=O ZINC000880650228 EF On-Demand Anodyne MTNR1B 16 42 Cc1nc(CNC(=O)CC[C@@H]2CCc3ccccc32)sc1C(N)=O ZINC000880650230 EF On-Demand Anodyne NQO2 17 40 Cc1nc(CNC(=O)CC[C@@H]2CCc3ccccc32)sc1C(N)=O ZINC000880650230 EF On-Demand Anodyne MTNR1B 16 42 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650235 GF On-Demand Anodyne TSHR 42 31 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650235 GF On-Demand Anodyne HTR1B 15 46 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650235 GF On-Demand Anodyne PDGFRB 35 41 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650235 GF On-Demand Anodyne ABCB1 20 41 CCCCSCC(=O)NCc1nnc(O)n1C ZINC000880650236 CC On-Demand Anodyne EST1_PIG 42 36 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650237 GF On-Demand Anodyne TSHR 42 31 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650237 GF On-Demand Anodyne HTR1B 15 46 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650237 GF On-Demand Anodyne PDGFRB 35 41 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C(=O)c3ccccc3)c2)C1 ZINC000880650237 GF On-Demand Anodyne ABCB1 20 41 CCCCN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650273 EE On-Demand Mild ITK 16 50 CCCCN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650273 EE On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CCC3)cn2)cc1 ZINC000880650293 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CCC3)cn2)cc1 ZINC000880650293 EH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CCC3)cn2)cc1 ZINC000880650295 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CCC3)cn2)cc1 ZINC000880650295 EH On-Demand Mild PANC 53 37 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650301 CD On-Demand Anodyne ACE 15 42 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650301 CD On-Demand Anodyne MME 30 42 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650301 CD On-Demand Anodyne ACE2 42 39 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650301 CD On-Demand Anodyne AMP1_PLAFQ 23 41 C[C@@H](Cc1ccc(F)cc1)C(=O)NCc1nnc(O)n1C ZINC000880650301 CD On-Demand Anodyne LEF 42 32 C[C@@H](Cc1ccccc1)n1cccc1C(=O)NCc1nnc(O)n1C ZINC000880650311 EE On-Demand Anodyne MME 63 36 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650313 FD On-Demand Mild ITK 18 54 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650313 FD On-Demand Mild MLNR 20 41 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650313 FD On-Demand Mild PANC 55 38 CN(CC1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650322 EG On-Demand Mild ITK 29 50 CN(CC1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650322 EG On-Demand Mild PANC 59 41 COc1cc(C(=O)NCc2nnc(O)n2C)cc2c1O[C@H](C)C2 ZINC000880650325 DC On-Demand Anodyne SLC5A7 31 40 COc1cc(C(=O)NCc2nnc(O)n2C)cc2c1O[C@@H](C)C2 ZINC000880650327 DC On-Demand Anodyne SLC5A7 31 40 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne ADRB1 40 30 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne DRD2 18 41 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne TSHR 40 29 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne DRD3 31 41 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne KCNA3 24 40 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne KCNK3 75 45 COCCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650330 EG On-Demand Anodyne KCNK9 54 42 C#CCC1(O)CCN(C(=O)Nc2ccc(C)c(C(=O)c3ccccc3)c2)CC1 ZINC000880650348 GH On-Demand Mild S1PR2 27 44 Cc1ccc(NC(=O)N2CC3(CCOC3)C2)cc1C(=O)c1ccccc1 ZINC000880650357 FG On-Demand Anodyne EPHX2 31 41 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650379 EG On-Demand Mild ITK 18 52 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650379 EG On-Demand Mild MLNR 31 41 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650379 EG On-Demand Mild PANC 55 38 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650381 EG On-Demand Mild ITK 18 52 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650381 EG On-Demand Mild MLNR 31 41 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650381 EG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC4CC4)CC3)cn2)cc1 ZINC000880650383 FE On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC4CC4)CC3)cn2)cc1 ZINC000880650383 FE On-Demand Mild MLNR 29 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC4CC4)CC3)cn2)cc1 ZINC000880650383 FE On-Demand Mild FAAH 20 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CC4CC4)CC3)cn2)cc1 ZINC000880650383 FE On-Demand Mild PANC 53 37 CCC(CC)(C(=O)NCc1nnc(O)n1C)c1ccc(OC)c(OC)c1 ZINC000880650394 FD On-Demand Anodyne MT-ND1 23 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(Cc4ccco4)CC3)cn2)cc1 ZINC000880650395 GF On-Demand Mild ITK 15 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(Cc4ccco4)CC3)cn2)cc1 ZINC000880650395 GF On-Demand Mild FAAH 22 44 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C ZINC000880650399 ED On-Demand Anodyne ST14 41 35 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C ZINC000880650399 ED On-Demand Anodyne TMPRSS6 58 35 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C ZINC000880650400 ED On-Demand Anodyne ST14 41 35 C[C@H](Sc1nc2ccccc2s1)C(=O)NCc1nnc(O)n1C ZINC000880650400 ED On-Demand Anodyne TMPRSS6 58 35 CCCN(CC(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650402 EH On-Demand Mild ITK 15 49 CCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650406 BD On-Demand Anodyne ASAH1 48 35 CCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650406 BD On-Demand Anodyne LASR 47 33 CCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650406 BD On-Demand Anodyne NOD1 61 39 CCCCCCC(=O)NCc1nnc(O)n1C ZINC000880650406 BD On-Demand Anodyne CQSS 55 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880650410 EE On-Demand Mild ITK 18 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880650410 EE On-Demand Mild PANC 55 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880650411 EE On-Demand Mild ITK 18 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880650411 EE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCCC3)cn2)cc1 ZINC000880650414 EH On-Demand Mild ITK 20 55 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCCC3)cn2)cc1 ZINC000880650414 EH On-Demand Mild PANC 42 37 CN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650424 DF On-Demand Mild ITK 28 52 CN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650424 DF On-Demand Mild PANC 60 42 Cc1c(Br)cccc1CC(=O)NCc1nnc(O)n1C ZINC000880650425 ED On-Demand Anodyne P2RX7 23 41 CC(=O)N(C)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650427 GE On-Demand Mild ITK 20 48 CC(=O)N(C)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650427 GE On-Demand Mild MLNR 42 40 CC(=O)N(C)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650427 GE On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCC3)cn2)cc1 ZINC000880650439 DG On-Demand Mild ITK 20 55 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCC3)cn2)cc1 ZINC000880650439 DG On-Demand Mild PANC 42 37 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CC3)cn2)cc1 ZINC000880650440 ED On-Demand Mild ITK 19 51 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CC3)cn2)cc1 ZINC000880650440 ED On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CO)CC3)cn2)cc1 ZINC000880650447 EE On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CO)CC3)cn2)cc1 ZINC000880650447 EE On-Demand Mild MLNR 19 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CO)CC3)cn2)cc1 ZINC000880650447 EE On-Demand Mild PANC 54 38 COCCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650457 EE On-Demand Mild ITK 23 52 COCCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650457 EE On-Demand Mild PANC 56 38 CCCN(CCC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650460 EG On-Demand Mild ITK 18 54 CCCN(CCC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650460 EG On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCCC4)CC3)cn2)cc1 ZINC000880650466 GF On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCCC4)CC3)cn2)cc1 ZINC000880650466 GF On-Demand Mild PANC 53 37 COc1ccc(CC(=O)NCc2nnc(O)n2C)cc1F ZINC000880650469 CC On-Demand Anodyne TRPV1 26 43 COc1ccc(CC(=O)NCc2nnc(O)n2C)cc1F ZINC000880650469 CC On-Demand Anodyne DRTS_TRYCR 44 30 C=CC(C)(C)CC(=O)N1CCCC[C@@H]1c1n[nH]c(C(C)C)n1 ZINC000880650544 DH On-Demand Mild CPT1A 56 35 C=CC(C)(C)CC(=O)N1CCCC[C@H]1c1n[nH]c(C(C)C)n1 ZINC000880650545 DH On-Demand Mild CPT1A 56 35 Cc1ccc(NC(=O)N2CCC3(C2)OCCO3)cc1C(=O)c1ccccc1 ZINC000880650554 FG On-Demand Anodyne NPY5R 19 41 Cc1ccc(NC(=O)N2CCC3(C2)OCCO3)cc1C(=O)c1ccccc1 ZINC000880650554 FG On-Demand Anodyne EPHX2 36 44 COCCN(Cc1ccco1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650576 GG On-Demand Mild ITK 17 47 COCCN(Cc1ccco1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650576 GG On-Demand Mild PANC 48 34 CC(C)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650577 FF On-Demand Mild ITK 16 51 CC(C)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650577 FF On-Demand Mild MLNR 29 43 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650585 DF On-Demand Mild ITK 19 52 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650585 DF On-Demand Mild MLNR 53 45 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650585 DF On-Demand Mild PANC 57 40 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650586 DF On-Demand Mild ITK 19 52 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650586 DF On-Demand Mild MLNR 53 45 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650586 DF On-Demand Mild PANC 57 40 C[C@@H]1C[C@@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650602 CE On-Demand Mild ITK 19 52 C[C@@H]1C[C@@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650602 CE On-Demand Mild PANC 55 38 C[C@H]1C[C@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650604 CE On-Demand Mild ITK 19 52 C[C@H]1C[C@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650604 CE On-Demand Mild PANC 55 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880650618 EE On-Demand Mild ITK 25 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880650618 EE On-Demand Mild PANC 56 39 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880650619 EE On-Demand Mild ITK 25 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880650619 EE On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCCOCC3)cn2)cc1 ZINC000880650623 EE On-Demand Mild ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCCOCC3)cn2)cc1 ZINC000880650623 EE On-Demand Mild PANC 41 36 C=CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)C ZINC000880650624 DG On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCSCC3)cn2)cc1 ZINC000880650625 EE On-Demand Mild ITK 16 53 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3c3ccsc3)cn2)cc1 ZINC000880650627 GI On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3c3ccsc3)cn2)cc1 ZINC000880650628 GI On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4nccs4)CC3)cn2)cc1 ZINC000880650630 GH On-Demand Mild ITK 17 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CCCCC4)CC3)cn2)cc1 ZINC000880650636 GG On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CCCCC4)CC3)cn2)cc1 ZINC000880650636 GG On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CCCCC4)CC3)cn2)cc1 ZINC000880650636 GG On-Demand Mild L3MBTL3 101 44 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)no1 ZINC000880650639 GG On-Demand Mild ITK 17 47 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)no1 ZINC000880650639 GG On-Demand Mild PANC 62 42 C[C@@H](C1CC1)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650644 DG On-Demand Mild ITK 25 51 C[C@@H](C1CC1)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650644 DG On-Demand Mild PANC 58 39 COCCN(Cc1cccs1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650652 GH On-Demand Mild ITK 18 47 COCCN(Cc1cccs1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650652 GH On-Demand Mild PANC 48 34 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C1CC1)C1CC1 ZINC000880650653 EG On-Demand Mild ITK 27 52 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C1CC1)C1CC1 ZINC000880650653 EG On-Demand Mild PANC 58 39 C/C=C\c1ccc(OCC(=O)NCc2nnc(O)n2C)c(OC)c1 ZINC000880650659 ED On-Demand Anodyne TUBB1 50 37 C/C=C/c1ccc(OCC(=O)NCc2nnc(O)n2C)c(OC)c1 ZINC000880650660 ED On-Demand Anodyne TUBB1 50 37 CCC(=O)N1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650695 GE On-Demand Mild ITK 16 49 CCC(=O)N1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880650695 GE On-Demand Mild MLNR 26 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCCC4)CC3)cn2)cc1 ZINC000880650698 GH On-Demand Mild ITK 20 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCCC4)CC3)cn2)cc1 ZINC000880650698 GH On-Demand Mild MLNR 25 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCCC4)CC3)cn2)cc1 ZINC000880650698 GH On-Demand Mild PANC 55 39 COCCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650726 FD On-Demand Mild ITK 23 54 COCCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650726 FD On-Demand Mild PANC 55 38 Cc1ccc(NC(=O)N2CCC3(CC2)CNC(=O)O3)cc1C(=O)c1ccccc1 ZINC000880650742 GG On-Demand Anodyne TRPM8 29 41 Cc1ccc(NC(=O)N2CCC3(CC2)OCCO3)cc1C(=O)c1ccccc1 ZINC000880650776 GH On-Demand Anodyne NPY5R 27 42 Cc1ccc(NC(=O)N2CCC3(CC2)OCCO3)cc1C(=O)c1ccccc1 ZINC000880650776 GH On-Demand Anodyne EPHX2 34 41 CCOCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650788 EG On-Demand Anodyne KCNK3 47 43 CCOCCNC(=O)Nc1ccc(OC)c(C(=O)c2ccccc2)c1 ZINC000880650788 EG On-Demand Anodyne KCNK9 40 43 Cc1ccc(NC(=O)N2CCC3=C(CCC(=O)N3)C2)cc1C(=O)c1ccccc1 ZINC000880650796 GH On-Demand Anodyne P2RY14 48 35 Cc1ccc(NC(=O)N2CCC3(CC2)COCCO3)cc1C(=O)c1ccccc1 ZINC000880650850 GH On-Demand Anodyne EPHX2 28 45 Cc1ccc(NC(=O)N2CCC3(CC2)COCCO3)cc1C(=O)c1ccccc1 ZINC000880650850 GH On-Demand Anodyne TRPM8 27 40 CC(=O)C1CCN(C(=O)Nc2ccc(C)c(C(=O)c3ccccc3)c2)CC1 ZINC000880650857 FI On-Demand Anodyne NPY5R 15 40 CC(=O)C1CCN(C(=O)Nc2ccc(C)c(C(=O)c3ccccc3)c2)CC1 ZINC000880650857 FI On-Demand Anodyne CCR8 47 34 Cc1ccc(NC(=O)N2CCC(CO)(CO)CC2)cc1C(=O)c1ccccc1 ZINC000880650862 GF On-Demand Anodyne NPY5R 26 43 Cc1ccc(NC(=O)N2CCC(CO)(CO)CC2)cc1C(=O)c1ccccc1 ZINC000880650862 GF On-Demand Anodyne S1PR2 25 41 Cc1cnc(Cl)c(C(=O)N2CCCC[C@@H]2c2n[nH]c(C(C)C)n2)c1 ZINC000880650894 EH On-Demand Anodyne CPT1A 47 36 Cc1cnc(Cl)c(C(=O)N2CCCC[C@H]2c2n[nH]c(C(C)C)n2)c1 ZINC000880650895 EH On-Demand Anodyne CPT1A 47 36 COC[C@@H](O)CNC(=O)Nc1ccc(C)c(C(=O)c2ccccc2)c1 ZINC000880650912 EE On-Demand Anodyne ADRB1 49 41 CCN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650915 EE On-Demand Mild ITK 15 50 CCN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650915 EE On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCSC[C@@H]3CO)cn2)cc1 ZINC000880650917 FD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCSC[C@H]3CO)cn2)cc1 ZINC000880650918 FD On-Demand Mild ITK 15 47 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1=O ZINC000880650919 ED On-Demand Mild ITK 16 49 C[C@H](CO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650928 DD On-Demand Mild ITK 20 52 C[C@H](CO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650928 DD On-Demand Mild PANC 40 34 C[C@@H](CO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650929 DD On-Demand Mild ITK 20 52 C[C@@H](CO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650929 DD On-Demand Mild PANC 40 34 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1n1ccnc1 ZINC000880650930 GG On-Demand Mild MLNR 27 41 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1n1ccnc1 ZINC000880650931 GG On-Demand Mild MLNR 27 41 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1n1ccnc1 ZINC000880650932 GG On-Demand Mild MLNR 27 41 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1n1ccnc1 ZINC000880650933 GG On-Demand Mild MLNR 27 41 CN(CCOCC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650938 FF On-Demand Mild ITK 20 47 CN(CCOCC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650938 FF On-Demand Mild PANC 58 39 CN(C)[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650940 ED On-Demand Mild ITK 23 49 CN(C)[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650940 ED On-Demand Mild MLNR 41 41 CN(C)[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880650940 ED On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC=C(C(F)(F)F)CC3)cn2)cc1 ZINC000880650942 GH On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC=C(C(F)(F)F)CC3)cn2)cc1 ZINC000880650942 GH On-Demand Mild PANC 42 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](N4CCCC4=O)C3)cn2)cc1 ZINC000880650943 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](N4CCCC4=O)C3)cn2)cc1 ZINC000880650944 GE On-Demand Mild PANC 53 37 CC[C@H]1C[C@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650952 EG On-Demand Mild ITK 15 48 CC[C@H]1C[C@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650952 EG On-Demand Mild PANC 41 35 CC[C@@H]1C[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650953 EG On-Demand Mild ITK 15 48 CC[C@@H]1C[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650953 EG On-Demand Mild PANC 41 35 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)O1 ZINC000880650961 FF On-Demand Mild ITK 15 49 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)O1 ZINC000880650961 FF On-Demand Mild PANC 53 35 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)O1 ZINC000880650962 FF On-Demand Mild ITK 15 49 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)O1 ZINC000880650962 FF On-Demand Mild PANC 53 35 C[C@@H]1SCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880650964 FG On-Demand Mild ITK 15 48 C[C@@H]1SCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880650964 FG On-Demand Mild PANC 41 36 C[C@@H]1SCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880650965 FG On-Demand Mild ITK 15 48 C[C@@H]1SCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880650965 FG On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C(C)(C)C1 ZINC000880650970 EG On-Demand Mild ITK 15 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C(C)(C)C1 ZINC000880650970 EG On-Demand Mild PANC 48 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C(C)(C)C1 ZINC000880650971 EG On-Demand Mild ITK 15 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C(C)(C)C1 ZINC000880650971 EG On-Demand Mild PANC 48 35 CN(C[C@@H]1CCCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650973 FF On-Demand Mild ITK 27 45 CN(C[C@@H]1CCCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880650973 FF On-Demand Mild PANC 57 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CCCO)cn2)cc1 ZINC000880650975 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CCCO)cn2)cc1 ZINC000880650975 FF On-Demand Mild PANC 41 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CCCO)cn2)cc1 ZINC000880650976 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CCCO)cn2)cc1 ZINC000880650976 FF On-Demand Mild PANC 41 37 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCCC1 ZINC000880650979 DG On-Demand Mild ITK 33 51 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCCC1 ZINC000880650979 DG On-Demand Mild PANC 57 38 CC[C@@](C)(NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)c1nccs1 ZINC000880650983 GH On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CC3)cn2)cc1 ZINC000880650984 EG On-Demand Mild DPP4 17 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CC3)cn2)cc1 ZINC000880650984 EG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CC3)cn2)cc1 ZINC000880650984 EG On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CC3)cn2)cc1 ZINC000880650985 EG On-Demand Mild DPP4 17 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CC3)cn2)cc1 ZINC000880650985 EG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CC3)cn2)cc1 ZINC000880650985 EG On-Demand Mild PANC 53 38 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1 ZINC000880650990 EE On-Demand Mild ITK 16 49 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1 ZINC000880650990 EE On-Demand Mild PANC 49 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650992 GF On-Demand Mild CCR3 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650992 GF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650992 GF On-Demand Mild MLNR 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650992 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650993 GF On-Demand Mild CCR3 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650993 GF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650993 GF On-Demand Mild MLNR 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCC4)C3)cn2)cc1 ZINC000880650993 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OCC4CC4)CC3)cn2)cc1 ZINC000880650997 GG On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OCC4CC4)CC3)cn2)cc1 ZINC000880650997 GG On-Demand Mild MLNR 20 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OCC4CC4)CC3)cn2)cc1 ZINC000880650997 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3Cn3cccn3)cn2)cc1 ZINC000880651003 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3Cn3cccn3)cn2)cc1 ZINC000880651004 GF On-Demand Mild ITK 15 47 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651005 FD On-Demand Mild ITK 15 47 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651005 FD On-Demand Mild MLNR 22 40 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651005 FD On-Demand Mild PANC 51 36 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651006 FD On-Demand Mild ITK 15 47 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651006 FD On-Demand Mild MLNR 22 40 CC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651006 FD On-Demand Mild PANC 51 36 Cn1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)cn1 ZINC000880651007 GF On-Demand Mild ITK 19 47 Cn1cc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)cn1 ZINC000880651007 GF On-Demand Mild PANC 58 40 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CC4)CC3)cn2)cc1 ZINC000880651016 DF On-Demand Mild ITK 18 51 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CC4)CC3)cn2)cc1 ZINC000880651016 DF On-Demand Mild PANC 54 36 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651017 EE On-Demand Mild ITK 20 49 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651017 EE On-Demand Mild MLNR 19 40 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651017 EE On-Demand Mild PANC 56 39 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651020 EF On-Demand Mild ITK 15 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651020 EF On-Demand Mild PANC 49 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651021 EF On-Demand Mild ITK 15 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651021 EF On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CO)C3)cn2)cc1 ZINC000880651024 ED On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CO)C3)cn2)cc1 ZINC000880651024 ED On-Demand Mild MLNR 23 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CO)C3)cn2)cc1 ZINC000880651024 ED On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CO)C3)cn2)cc1 ZINC000880651025 ED On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CO)C3)cn2)cc1 ZINC000880651025 ED On-Demand Mild MLNR 23 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CO)C3)cn2)cc1 ZINC000880651025 ED On-Demand Mild PANC 53 38 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C[C@H](C)O ZINC000880651026 GE On-Demand Mild ITK 15 44 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C[C@@H](C)O ZINC000880651029 GE On-Demand Mild ITK 15 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC(F)(F)F)C3)cn2)cc1 ZINC000880651030 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC(F)(F)F)C3)cn2)cc1 ZINC000880651030 FG On-Demand Mild PANC 53 37 CN(CCC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651033 DG On-Demand Mild ITK 22 49 CN(CCC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651033 DG On-Demand Mild PANC 60 41 COCCN(CCN(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651040 FD On-Demand Mild ITK 24 50 COCCN(CCN(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651040 FD On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC4(CCOCC4)C3)cn2)cc1 ZINC000880651048 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCCc4sccc4C3)cn2)cc1 ZINC000880651050 GH On-Demand Mild ITK 15 46 CN(CC1(O)CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651052 FF On-Demand Mild ITK 19 49 CN(CC1(O)CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651052 FF On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651055 GF On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651055 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651055 GF On-Demand Mild L3MBTL3 75 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651056 GF On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651056 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCCC4)C3)cn2)cc1 ZINC000880651056 GF On-Demand Mild L3MBTL3 75 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCC4)CC3)cn2)cc1 ZINC000880651062 FF On-Demand Mild HRH3 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCC4)CC3)cn2)cc1 ZINC000880651062 FF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCC4)CC3)cn2)cc1 ZINC000880651062 FF On-Demand Mild PANC 53 37 C[C@@H]1N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1(C)C ZINC000880651063 FF On-Demand Mild ITK 15 47 C[C@@H]1N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1(C)C ZINC000880651063 FF On-Demand Mild PANC 53 37 COCCN(Cc1ccc(C)o1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651068 GG On-Demand Mild ITK 17 45 COCCN(Cc1ccc(C)o1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651068 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880651071 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880651071 GD On-Demand Mild MLNR 15 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880651071 GD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCOC4)CC3)cn2)cc1 ZINC000880651072 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCOC4)CC3)cn2)cc1 ZINC000880651072 GD On-Demand Mild MLNR 15 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCOC4)CC3)cn2)cc1 ZINC000880651072 GD On-Demand Mild PANC 41 36 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880651075 EE On-Demand Mild ITK 19 50 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880651075 EE On-Demand Mild PANC 56 38 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880651077 EE On-Demand Mild ITK 19 50 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880651077 EE On-Demand Mild PANC 56 38 CN(C)C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651080 FD On-Demand Mild ITK 23 47 CN(C)C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651080 FD On-Demand Mild PANC 54 38 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651082 GD On-Demand Mild ITK 15 45 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651082 GD On-Demand Mild MLNR 32 42 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651082 GD On-Demand Mild PANC 40 34 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651083 GD On-Demand Mild ITK 15 45 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651083 GD On-Demand Mild MLNR 32 42 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651083 GD On-Demand Mild PANC 40 34 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C[C@@H](C)O ZINC000880651085 GD On-Demand Mild ITK 15 45 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C[C@@H](C)O ZINC000880651085 GD On-Demand Mild MLNR 32 42 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C[C@@H](C)O ZINC000880651085 GD On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C(F)F)CC3)cn2)cc1 ZINC000880651087 FG On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C(F)F)CC3)cn2)cc1 ZINC000880651087 FG On-Demand Mild PANC 56 39 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651089 GE On-Demand Mild PANC 40 35 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651090 GE On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N(CCCO)C3CC3)cn2)cc1 ZINC000880651093 EE On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N(CCCO)C3CC3)cn2)cc1 ZINC000880651093 EE On-Demand Mild MCHR1 24 40 N#Cc1ccc(Cn2cc(NC(=O)N(CCCO)C3CC3)cn2)cc1 ZINC000880651093 EE On-Demand Mild PANC 53 38 CN(CCC1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651094 FG On-Demand Mild ITK 19 46 CN(CCC1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651094 FG On-Demand Mild PANC 59 40 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCCc2c1cnn2C ZINC000880651095 GG On-Demand Mild ITK 23 46 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCCc2c1cnn2C ZINC000880651095 GG On-Demand Mild PANC 53 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCc2c1cnn2C ZINC000880651096 GG On-Demand Mild ITK 23 46 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCc2c1cnn2C ZINC000880651096 GG On-Demand Mild PANC 53 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880651100 FE On-Demand Mild ITK 19 48 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880651100 FE On-Demand Mild PANC 41 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880651101 FE On-Demand Mild ITK 19 48 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880651101 FE On-Demand Mild PANC 41 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880651102 FE On-Demand Mild ITK 19 48 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880651102 FE On-Demand Mild PANC 41 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880651103 FE On-Demand Mild ITK 19 48 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880651103 FE On-Demand Mild PANC 41 35 CC[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651104 GD On-Demand Mild ITK 17 49 CC[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651104 GD On-Demand Mild MLNR 25 40 CC[C@@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651105 GD On-Demand Mild ITK 17 49 CC[C@@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651105 GD On-Demand Mild MLNR 25 40 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880651108 DG On-Demand Mild ITK 18 50 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880651108 DG On-Demand Mild PANC 56 39 C[C@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651109 DG On-Demand Mild ITK 18 50 C[C@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651109 DG On-Demand Mild PANC 56 39 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651110 DG On-Demand Mild ITK 18 50 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651110 DG On-Demand Mild PANC 56 39 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651111 DG On-Demand Mild ITK 18 50 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651111 DG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](c4ccco4)C3)cn2)cc1 ZINC000880651113 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](c4ccco4)C3)cn2)cc1 ZINC000880651114 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CCOCC4)C3)cn2)cc1 ZINC000880651124 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CCOCC4)C3)cn2)cc1 ZINC000880651124 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CCOCC4)C3)cn2)cc1 ZINC000880651126 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CCOCC4)C3)cn2)cc1 ZINC000880651126 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CC=CC4)C3)cn2)cc1 ZINC000880651127 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CC=CC4)C3)cn2)cc1 ZINC000880651127 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CC=CC4)C3)cn2)cc1 ZINC000880651128 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CC=CC4)C3)cn2)cc1 ZINC000880651128 FE On-Demand Mild PANC 41 36 CC(C)(C)CN(CCCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651131 FG On-Demand Mild ITK 16 49 CC(C)(C)CN(CCCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651131 FG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C3)cn2)cc1 ZINC000880651136 DD On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C3)cn2)cc1 ZINC000880651136 DD On-Demand Mild MLNR 28 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C3)cn2)cc1 ZINC000880651136 DD On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](c4cccs4)C3)cn2)cc1 ZINC000880651143 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](c4cccs4)C3)cn2)cc1 ZINC000880651145 GG On-Demand Mild ITK 15 46 CN(C[C@@H]1CCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651151 FE On-Demand Mild ITK 30 47 CN(C[C@@H]1CCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651151 FE On-Demand Mild PANC 56 39 CN(C[C@@H]1CCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651153 FE On-Demand Mild ITK 30 47 CN(C[C@@H]1CCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651153 FE On-Demand Mild PANC 56 39 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651154 EE On-Demand Mild ITK 19 49 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651154 EE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H](C3)O4)cn2)cc1 ZINC000880651160 EE On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H](C3)O4)cn2)cc1 ZINC000880651160 EE On-Demand Mild PANC 56 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC4(CCCC4)C3)cn2)cc1 ZINC000880651161 FF On-Demand Mild EPHX2 16 50 CN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651166 EE On-Demand Mild ITK 20 54 CN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651166 EE On-Demand Mild PANC 60 40 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)CC3CC3)cn2)cc1 ZINC000880651167 EE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)CC3CC3)cn2)cc1 ZINC000880651167 EE On-Demand Mild PANC 53 35 CC[C@@](C)(NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)c1nc(C)cs1 ZINC000880651172 GI On-Demand Mild ITK 16 47 CC[C@@](C)(NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)c1nc(C)cs1 ZINC000880651172 GI On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C(F)(F)F)CC3)cn2)cc1 ZINC000880651173 GH On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C(F)(F)F)CC3)cn2)cc1 ZINC000880651173 GH On-Demand Mild PANC 58 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(CC(F)F)CC3)cn2)cc1 ZINC000880651174 GF On-Demand Mild ITK 15 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CCCC4=O)CC3)cn2)cc1 ZINC000880651180 GE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@](O)(C(F)(F)F)C3)cn2)cc1 ZINC000880651181 GE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@](O)(C(F)(F)F)C3)cn2)cc1 ZINC000880651182 GE On-Demand Mild ITK 15 47 CN(CCC#N)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651186 DE On-Demand Mild ITK 18 52 CN(CCC#N)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651186 DE On-Demand Mild PANC 49 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCC4)C3)cn2)cc1 ZINC000880651188 EG On-Demand Mild ITK 17 51 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCOC1 ZINC000880651190 EE On-Demand Mild ITK 24 49 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCOC1 ZINC000880651190 EE On-Demand Mild PANC 57 38 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCOC1 ZINC000880651191 EE On-Demand Mild ITK 24 49 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCOC1 ZINC000880651191 EE On-Demand Mild PANC 57 38 CC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651204 CF On-Demand Mild ITK 18 57 CC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651204 CF On-Demand Mild PANC 59 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccccn4)CC3)cn2)cc1 ZINC000880651205 GH On-Demand Mild CACNA1H 31 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccccn4)CC3)cn2)cc1 ZINC000880651205 GH On-Demand Mild ITK 18 53 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccccn4)CC3)cn2)cc1 ZINC000880651205 GH On-Demand Mild PANC 49 36 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651212 GF On-Demand Mild ITK 16 45 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651212 GF On-Demand Mild PANC 41 36 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651213 GF On-Demand Mild ITK 16 45 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880651213 GF On-Demand Mild PANC 41 36 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651214 GF On-Demand Mild ITK 16 45 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651214 GF On-Demand Mild PANC 41 36 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651215 GF On-Demand Mild ITK 16 45 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880651215 GF On-Demand Mild PANC 41 36 C[C@H]1CCCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651221 EH On-Demand Mild ITK 29 49 C[C@H]1CCCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651221 EH On-Demand Mild PANC 55 38 CC(C)(C)CN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651227 FF On-Demand Mild ITK 16 49 CC(C)(C)CN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651227 FF On-Demand Mild PANC 53 35 CN(C[C@@H]1C[C@H](O)C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651229 EE On-Demand Mild ITK 18 49 CN(C[C@@H]1C[C@H](O)C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651229 EE On-Demand Mild PANC 56 39 CN(C[C@@H]1COCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651234 FD On-Demand Mild ITK 19 45 CN(C[C@@H]1COCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651234 FD On-Demand Mild PANC 57 39 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651240 EE On-Demand Mild DPP4 17 42 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651240 EE On-Demand Mild ITK 18 49 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651240 EE On-Demand Mild PANC 55 38 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651241 EE On-Demand Mild DPP4 17 42 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651241 EE On-Demand Mild ITK 18 49 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651241 EE On-Demand Mild PANC 55 38 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651242 EE On-Demand Mild DPP4 17 42 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651242 EE On-Demand Mild ITK 18 49 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651242 EE On-Demand Mild PANC 55 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@](=O)C1 ZINC000880651246 FE On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@](=O)C1 ZINC000880651246 FE On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@](=O)C1 ZINC000880651247 FE On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@](=O)C1 ZINC000880651247 FE On-Demand Mild PANC 41 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@](=O)C1 ZINC000880651248 FE On-Demand Mild ITK 15 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@](=O)C1 ZINC000880651248 FE On-Demand Mild PANC 41 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@](=O)C1 ZINC000880651249 FE On-Demand Mild ITK 15 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@](=O)C1 ZINC000880651249 FE On-Demand Mild PANC 41 36 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651250 FG On-Demand Mild PDGFRB 21 43 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651250 FG On-Demand Mild ITK 19 46 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651250 FG On-Demand Mild PANC 55 38 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCc3cccnc32)c1 ZINC000880651252 DF On-Demand Anodyne G2YM83_BOTF4 72 42 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCc3cccnc32)c1 ZINC000880651253 DF On-Demand Anodyne G2YM83_BOTF4 72 42 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC3(CC3)C4)cn2)cc1 ZINC000880651254 FH On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC3(CC3)C4)cn2)cc1 ZINC000880651254 FH On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C(F)(F)F)CC3)cn2)cc1 ZINC000880651255 GF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C(F)(F)F)CC3)cn2)cc1 ZINC000880651256 GF On-Demand Mild PANC 55 38 CCc1cnc(CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)s1 ZINC000880651258 GG On-Demand Mild ITK 16 47 CCc1cnc(CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)s1 ZINC000880651258 GG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCCC4)C3)cn2)cc1 ZINC000880651261 EH On-Demand Mild ITK 17 51 C[S@@](=O)CCCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651263 ED On-Demand Mild CCR3 22 43 C[S@@](=O)CCCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651263 ED On-Demand Mild ITK 16 54 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCCO4)CC3)cn2)cc1 ZINC000880651267 GE On-Demand Mild ITK 20 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCCO4)CC3)cn2)cc1 ZINC000880651267 GE On-Demand Mild MLNR 16 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@@H]4CCCO4)CC3)cn2)cc1 ZINC000880651267 GE On-Demand Mild PANC 57 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCCO4)CC3)cn2)cc1 ZINC000880651268 GE On-Demand Mild ITK 20 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCCO4)CC3)cn2)cc1 ZINC000880651268 GE On-Demand Mild MLNR 16 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C[C@H]4CCCO4)CC3)cn2)cc1 ZINC000880651268 GE On-Demand Mild PANC 57 39 C[C@@H](O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651271 FE On-Demand Mild ITK 19 51 C[C@@H](O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651271 FE On-Demand Mild MLNR 24 41 C[C@@H](O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651271 FE On-Demand Mild PANC 57 40 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N1CCOCC1 ZINC000880651278 GD On-Demand Mild ITK 15 45 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N1CCOCC1 ZINC000880651278 GD On-Demand Mild PANC 41 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N1CCOCC1 ZINC000880651279 GD On-Demand Mild ITK 15 45 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N1CCOCC1 ZINC000880651279 GD On-Demand Mild PANC 41 36 C[C@]1(C#N)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651280 EF On-Demand Mild ITK 16 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N1CCOCC1 ZINC000880651281 GD On-Demand Mild ITK 15 45 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N1CCOCC1 ZINC000880651281 GD On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N1CCOCC1 ZINC000880651282 GD On-Demand Mild ITK 15 45 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N1CCOCC1 ZINC000880651282 GD On-Demand Mild PANC 41 36 C[C@@]1(C#N)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651284 EF On-Demand Mild ITK 16 51 Cc1nc(C(C)(C)NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)sc1C ZINC000880651289 GH On-Demand Mild ITK 15 47 Cc1nc(C(C)(C)NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)sc1C ZINC000880651289 GH On-Demand Mild PANC 54 37 CNC(C)(C)CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651291 ED On-Demand Mild ITK 17 52 CNC(C)(C)CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651291 ED On-Demand Mild PANC 55 37 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651292 FF On-Demand Mild ITK 19 49 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651292 FF On-Demand Mild PANC 60 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C4CCC4)C3)cn2)cc1 ZINC000880651295 FF On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C4CCC4)C3)cn2)cc1 ZINC000880651295 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(C3)OCCO4)cn2)cc1 ZINC000880651296 FD On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880651297 FF On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880651297 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@]4(CCSC4)C3)cn2)cc1 ZINC000880651299 GH On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(O)C4)cn2)cc1 ZINC000880651300 FE On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(O)C4)cn2)cc1 ZINC000880651300 FE On-Demand Mild PANC 54 38 COCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651301 FF On-Demand Mild PDGFRB 19 43 COCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651301 FF On-Demand Mild ITK 20 49 COCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651301 FF On-Demand Mild MLNR 23 41 COCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651301 FF On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@]4(CCSC4)C3)cn2)cc1 ZINC000880651304 GH On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C(F)(F)F)C3)cn2)cc1 ZINC000880651306 EF On-Demand Mild ITK 15 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C(F)(F)F)C3)cn2)cc1 ZINC000880651306 EF On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O[C@H]4CCOC4)CC3)cn2)cc1 ZINC000880651308 GF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O[C@H]4CCOC4)CC3)cn2)cc1 ZINC000880651308 GF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O[C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880651309 GF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O[C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880651309 GF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccon4)CC3)cn2)cc1 ZINC000880651313 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccon4)CC3)cn2)cc1 ZINC000880651313 GG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CC3)OCCCO4)cn2)cc1 ZINC000880651316 GF On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC(C4CC4)(C4CC4)C3)cn2)cc1 ZINC000880651318 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC(C4CC4)(C4CC4)C3)cn2)cc1 ZINC000880651318 GG On-Demand Mild PANC 49 36 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651321 GF On-Demand Mild ITK 15 45 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651321 GF On-Demand Mild PANC 41 34 CCN1CCC[C@H]1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651322 FF On-Demand Mild ITK 18 45 CCN1CCC[C@H]1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651322 FF On-Demand Mild PANC 57 39 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651323 GF On-Demand Mild ITK 15 45 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651323 GF On-Demand Mild PANC 41 34 CCN1CCC[C@@H]1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651324 FF On-Demand Mild ITK 18 45 CCN1CCC[C@@H]1CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651324 FF On-Demand Mild PANC 57 39 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651325 GF On-Demand Mild ITK 15 45 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651325 GF On-Demand Mild PANC 41 34 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651327 GF On-Demand Mild ITK 15 45 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651327 GF On-Demand Mild PANC 41 34 N#CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651329 EF On-Demand Mild ITK 17 50 N#CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651329 EF On-Demand Mild PANC 54 38 N#CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651330 EF On-Demand Mild ITK 17 50 N#CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651330 EF On-Demand Mild PANC 54 38 C[C@@H](CCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)N(C)C ZINC000880651332 EE On-Demand Mild ITK 15 50 C[C@H](CCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)N(C)C ZINC000880651334 EE On-Demand Mild ITK 15 50 CN(C)CCC[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651338 GE On-Demand Mild ITK 16 45 CN(C)CCC[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651338 GE On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4C=CC[C@H]3CC4)cn2)cc1 ZINC000880651343 EG On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4C=CC[C@H]3CC4)cn2)cc1 ZINC000880651343 EG On-Demand Mild PANC 55 36 CC[C@]1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651346 EG On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(C3)CC4(F)F)cn2)cc1 ZINC000880651351 EF On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(C3)CC4(F)F)cn2)cc1 ZINC000880651351 EF On-Demand Mild PANC 40 35 COCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651352 EE On-Demand Mild ITK 18 51 COCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651352 EE On-Demand Mild PANC 57 39 Cn1cc([C@@H]2N(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC2(C)C)cn1 ZINC000880651354 GG On-Demand Mild ITK 18 47 Cn1cc([C@@H]2N(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC2(C)C)cn1 ZINC000880651354 GG On-Demand Mild PANC 53 35 C[C@@H](C1CC1)N(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880651355 EH On-Demand Mild ITK 20 51 C[C@@H](C1CC1)N(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880651355 EH On-Demand Mild PANC 57 39 N#Cc1ccc(Cn2cc(NC(=O)NCC3CSC3)cn2)cc1 ZINC000880651358 EE On-Demand Mild ITK 19 54 N#Cc1ccc(Cn2cc(NC(=O)NCC3CSC3)cn2)cc1 ZINC000880651358 EE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)NCCCC(F)(F)F)cn2)cc1 ZINC000880651359 FG On-Demand Mild ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)NCCCC(F)(F)F)cn2)cc1 ZINC000880651359 FG On-Demand Mild PANC 40 35 C=CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651360 EG On-Demand Mild ITK 16 49 C=CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651360 EG On-Demand Mild PANC 53 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@]1(C)CO ZINC000880651363 FE On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@]1(C)CO ZINC000880651363 FE On-Demand Mild PANC 41 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@]1(C)CO ZINC000880651365 FE On-Demand Mild ITK 15 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@]1(C)CO ZINC000880651365 FE On-Demand Mild PANC 41 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@]1(C)CO ZINC000880651366 FE On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@]1(C)CO ZINC000880651366 FE On-Demand Mild PANC 41 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@]1(C)CO ZINC000880651367 FE On-Demand Mild ITK 15 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@]1(C)CO ZINC000880651367 FE On-Demand Mild PANC 41 35 CC(=O)[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651368 FF On-Demand Mild ITK 28 48 CC(=O)[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651368 FF On-Demand Mild GPBAR1 21 40 CC(=O)[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651368 FF On-Demand Mild PANC 54 38 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651370 DG On-Demand Mild ITK 17 51 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651370 DG On-Demand Mild PANC 41 36 CCOC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651372 FG On-Demand Mild ITK 16 45 CCOC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651372 FG On-Demand Mild PANC 54 38 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651374 FF On-Demand Mild ITK 28 48 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651374 FF On-Demand Mild GPBAR1 21 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651374 FF On-Demand Mild PANC 54 38 C=CCCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651383 EH On-Demand Mild ITK 16 51 C=CCCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651383 EH On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(O)CCCC[C@H]4C3)cn2)cc1 ZINC000880651384 GF On-Demand Mild ITK 18 45 C#CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651385 EG On-Demand Mild ITK 15 49 C#CC[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651385 EG On-Demand Mild PANC 53 37 C#CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651386 EG On-Demand Mild ITK 15 49 C#CC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651386 EG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5CC[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651387 FG On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5CC[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651387 FG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H]5CC[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651388 FG On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H]5CC[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651388 FG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5CC[C@@H](C5)[C@@H]4C3)cn2)cc1 ZINC000880651389 FG On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5CC[C@@H](C5)[C@@H]4C3)cn2)cc1 ZINC000880651389 FG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5C=C[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651390 FG On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5C=C[C@@H](C5)[C@H]4C3)cn2)cc1 ZINC000880651390 FG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(O)CCCC[C@@H]4C3)cn2)cc1 ZINC000880651391 GF On-Demand Mild ITK 18 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(O)CCCC[C@H]4C3)cn2)cc1 ZINC000880651393 GF On-Demand Mild ITK 18 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(O)CCCC[C@@H]4C3)cn2)cc1 ZINC000880651395 GF On-Demand Mild ITK 18 45 N#Cc1ccc(Cn2cc(NC(=O)NC[C@@H]3CCCN(CC4CC4)C3)cn2)cc1 ZINC000880651401 GG On-Demand Mild CCR3 76 41 N#Cc1ccc(Cn2cc(NC(=O)NC[C@@H]3CCCN(CC4CC4)C3)cn2)cc1 ZINC000880651401 GG On-Demand Mild ITK 15 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651402 DF On-Demand Mild ITK 20 53 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651402 DF On-Demand Mild MLNR 24 40 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651402 DF On-Demand Mild PANC 56 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651403 DF On-Demand Mild ITK 20 53 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651403 DF On-Demand Mild MLNR 24 40 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651403 DF On-Demand Mild PANC 56 38 N#Cc1ccc(Cn2cc(NC(=O)NC[C@H]3CCCN(CC4CC4)C3)cn2)cc1 ZINC000880651404 GG On-Demand Mild CCR3 76 41 N#Cc1ccc(Cn2cc(NC(=O)NC[C@H]3CCCN(CC4CC4)C3)cn2)cc1 ZINC000880651404 GG On-Demand Mild ITK 15 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651405 DF On-Demand Mild ITK 20 53 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651405 DF On-Demand Mild MLNR 24 40 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651405 DF On-Demand Mild PANC 56 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(n4ccnc4)CC3)cn2)cc1 ZINC000880651408 GF On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(n4ccnc4)CC3)cn2)cc1 ZINC000880651408 GF On-Demand Mild MLNR 15 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@](O)(C4CC4)C3)cn2)cc1 ZINC000880651411 FF On-Demand Mild ITK 18 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@](O)(C4CC4)C3)cn2)cc1 ZINC000880651413 FF On-Demand Mild ITK 18 46 N#Cc1ccc(Cn2cc(NC(=O)N(CCCCO)C3CC3)cn2)cc1 ZINC000880651414 FF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N(CCCCO)C3CC3)cn2)cc1 ZINC000880651414 FF On-Demand Mild PANC 53 37 COCCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651415 FE On-Demand Mild ITK 22 51 COCCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651415 FE On-Demand Mild PANC 56 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCCC[C@H]4C3)cn2)cc1 ZINC000880651421 FF On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCCC[C@H]4C3)cn2)cc1 ZINC000880651421 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCCC[C@@H]4C3)cn2)cc1 ZINC000880651423 FF On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCCC[C@@H]4C3)cn2)cc1 ZINC000880651423 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC4(CCOCC4)C3)cn2)cc1 ZINC000880651425 GE On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(c4cccs4)CC3)cn2)cc1 ZINC000880651426 GG On-Demand Mild ITK 15 49 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CCOC ZINC000880651427 GE On-Demand Mild ITK 18 45 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CCOC ZINC000880651427 GE On-Demand Mild PANC 52 36 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3COC4)cn2)cc1 ZINC000880651431 EE On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3COC4)cn2)cc1 ZINC000880651431 EE On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C34CCCC4)cn2)cc1 ZINC000880651432 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C34CCCC4)cn2)cc1 ZINC000880651432 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C34CCCC4)cn2)cc1 ZINC000880651433 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C34CCCC4)cn2)cc1 ZINC000880651433 FF On-Demand Mild PANC 41 36 CCN1CC[C@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651434 FF On-Demand Mild ITK 18 47 CCN1CC[C@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651434 FF On-Demand Mild MLNR 25 41 CCN1CC[C@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651434 FF On-Demand Mild PANC 53 37 CCN1CC[C@@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651435 FF On-Demand Mild ITK 18 47 CCN1CC[C@@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651435 FF On-Demand Mild MLNR 25 41 CCN1CC[C@@H](N(CC)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651435 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880651437 GF On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880651437 GF On-Demand Mild PANC 41 36 CCC(CC)N(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651439 FG On-Demand Mild ITK 21 49 CCC(CC)N(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651439 FG On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@@H]4CCCC[C@H]43)cn2)cc1 ZINC000880651441 GF On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@@H]4CCCC[C@H]43)cn2)cc1 ZINC000880651441 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880651445 GF On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880651445 GF On-Demand Mild PANC 41 36 CC[C@@H]1CN2CCC[C@H]2CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651448 GF On-Demand Mild ITK 15 44 CC[C@@H]1CN2CCC[C@H]2CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651448 GF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@H]4CCCC[C@H]43)cn2)cc1 ZINC000880651449 GF On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)[C@H]4CCCC[C@H]43)cn2)cc1 ZINC000880651449 GF On-Demand Mild PANC 41 36 CC[C@@H]1CN2CCC[C@@H]2CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651451 GF On-Demand Mild ITK 15 44 CC[C@@H]1CN2CCC[C@@H]2CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651451 GF On-Demand Mild PANC 53 37 CCOC[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651455 FG On-Demand Mild ITK 24 45 CCOC[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651455 FG On-Demand Mild PANC 54 38 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651464 FG On-Demand Mild ITK 15 47 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651464 FG On-Demand Mild PANC 54 37 C[C@@]12COC[C@@H]1CN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880651465 FE On-Demand Mild ITK 15 45 C[C@@]12COC[C@@H]1CN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880651465 FE On-Demand Mild PANC 41 34 C[C@@]12COC[C@H]1CN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880651468 FE On-Demand Mild ITK 15 45 C[C@@]12COC[C@H]1CN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880651468 FE On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CN3CCOCC3)cn2)cc1 ZINC000880651469 GE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CN3CCOCC3)cn2)cc1 ZINC000880651470 GE On-Demand Mild PANC 41 36 Cn1cc([C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)cn1 ZINC000880651476 GF On-Demand Mild ITK 24 47 Cn1cc([C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)cn1 ZINC000880651476 GF On-Demand Mild MLNR 19 40 Cn1cc([C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)cn1 ZINC000880651476 GF On-Demand Mild PANC 56 39 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC(CO)CC1 ZINC000880651477 FF On-Demand Mild ITK 19 48 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC(CO)CC1 ZINC000880651477 FF On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCC(O)CC4)CC3)cn2)cc1 ZINC000880651478 GG On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCC(O)CC4)CC3)cn2)cc1 ZINC000880651478 GG On-Demand Mild PANC 54 38 C[C@]1(O)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651480 EE On-Demand Mild ITK 18 49 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880651481 FD On-Demand Mild ITK 16 49 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880651481 FD On-Demand Mild PANC 49 37 CC(C)(C)C1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651483 EG On-Demand Mild ITK 18 51 CC(C)(C)C1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651483 EG On-Demand Mild PANC 68 45 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651487 FF On-Demand Mild PDGFRB 15 42 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651487 FF On-Demand Mild ITK 20 47 COC[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651487 FF On-Demand Mild PANC 56 39 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C(F)(F)F)O1 ZINC000880651489 GF On-Demand Mild PANC 54 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C(F)(F)F)O1 ZINC000880651490 GF On-Demand Mild PANC 54 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C(F)(F)F)O1 ZINC000880651491 GF On-Demand Mild PANC 54 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C(F)(F)F)O1 ZINC000880651492 GF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4CCOCC4)CC3)cn2)cc1 ZINC000880651498 GG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4CCOCC4)CC3)cn2)cc1 ZINC000880651498 GG On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651509 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651509 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651510 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651510 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651511 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651511 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651512 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651512 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CO)cn2)cc1 ZINC000880651515 ED On-Demand Mild DPP4 15 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CO)cn2)cc1 ZINC000880651515 ED On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CO)cn2)cc1 ZINC000880651515 ED On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CO)cn2)cc1 ZINC000880651516 ED On-Demand Mild DPP4 15 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CO)cn2)cc1 ZINC000880651516 ED On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CO)cn2)cc1 ZINC000880651516 ED On-Demand Mild PANC 53 37 CCCCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651517 FG On-Demand Mild ITK 21 50 CCCCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651517 FG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H]([C@H]4CCCO4)C3)cn2)cc1 ZINC000880651523 GE On-Demand Mild ITK 21 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H]([C@H]4CCCO4)C3)cn2)cc1 ZINC000880651523 GE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H]([C@@H]4CCCO4)C3)cn2)cc1 ZINC000880651524 GE On-Demand Mild ITK 21 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H]([C@@H]4CCCO4)C3)cn2)cc1 ZINC000880651524 GE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H]([C@@H]4CCCO4)C3)cn2)cc1 ZINC000880651525 GE On-Demand Mild ITK 21 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H]([C@@H]4CCCO4)C3)cn2)cc1 ZINC000880651525 GE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H]([C@H]4CCCO4)C3)cn2)cc1 ZINC000880651526 GE On-Demand Mild ITK 21 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H]([C@H]4CCCO4)C3)cn2)cc1 ZINC000880651526 GE On-Demand Mild PANC 55 38 C[C@H]1C[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651528 DG On-Demand Mild ITK 18 51 C[C@H]1C[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651528 DG On-Demand Mild PANC 57 38 C[C@H]1C[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651529 DG On-Demand Mild ITK 18 51 C[C@H]1C[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651529 DG On-Demand Mild PANC 57 38 CCC1(CO)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651535 FF On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C(F)(F)F)C3)cn2)cc1 ZINC000880651541 GF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C(F)(F)F)C3)cn2)cc1 ZINC000880651542 GF On-Demand Mild PANC 53 37 CN(CCOC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651544 FG On-Demand Mild ITK 17 49 CN(CCOC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651544 FG On-Demand Mild PANC 57 39 CCC[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651546 FF On-Demand Mild ITK 16 48 CCC[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651546 FF On-Demand Mild PANC 55 38 CCC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651547 FF On-Demand Mild ITK 16 48 CCC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651547 FF On-Demand Mild PANC 55 38 CCOCCN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651551 EF On-Demand Mild ITK 16 49 CCOCCN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651551 EF On-Demand Mild PANC 40 34 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651556 GD On-Demand Mild PDGFRB 22 44 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651556 GD On-Demand Mild ITK 18 49 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651556 GD On-Demand Mild FAAH 15 41 CCOCCN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651556 GD On-Demand Mild PANC 40 35 Cn1ccnc1[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651570 GF On-Demand Mild ITK 20 44 Cn1ccnc1[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651570 GF On-Demand Mild PANC 40 35 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651571 GF On-Demand Mild ITK 20 44 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651571 GF On-Demand Mild PANC 40 35 C[C@H](O)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651573 DD On-Demand Mild ITK 19 52 C[C@H](O)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651573 DD On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651574 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651574 EH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4CCC[C@H]43)cn2)cc1 ZINC000880651575 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4CCC[C@H]43)cn2)cc1 ZINC000880651575 EH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651576 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651576 EH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4CCC[C@H]43)cn2)cc1 ZINC000880651577 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4CCC[C@H]43)cn2)cc1 ZINC000880651577 EH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880651578 GG On-Demand Mild ITK 19 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@H](N4CCCC4)C3)cn2)cc1 ZINC000880651578 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880651579 GG On-Demand Mild ITK 19 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H](N4CCCC4)C3)cn2)cc1 ZINC000880651579 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC4(CCCCC4)C3)cn2)cc1 ZINC000880651580 GG On-Demand Mild EPHX2 15 49 CN(C[C@H](O)C1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651581 EE On-Demand Mild ITK 22 50 CN(C[C@H](O)C1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651581 EE On-Demand Mild PANC 59 40 CC[C@H](C)CN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651588 EH On-Demand Mild ITK 16 50 CC[C@@H](C)CN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651589 EH On-Demand Mild ITK 16 50 C=C(C)CN(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651590 DG On-Demand Mild ITK 15 51 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCSC1 ZINC000880651591 EF On-Demand Mild ITK 19 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCSC1 ZINC000880651591 EF On-Demand Mild PANC 53 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCSC1 ZINC000880651592 EF On-Demand Mild ITK 19 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCSC1 ZINC000880651592 EF On-Demand Mild PANC 53 36 CCCN(C)C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651593 GF On-Demand Mild ITK 18 44 CCCN(C)C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651593 GF On-Demand Mild PANC 55 38 CCCN(C)C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651594 GF On-Demand Mild ITK 18 44 CCCN(C)C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651594 GF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCOCC4)CC3)cn2)cc1 ZINC000880651595 GE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CCOCC4)CC3)cn2)cc1 ZINC000880651595 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(Cn4cccn4)CC3)cn2)cc1 ZINC000880651598 GF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(Cn4cccn4)CC3)cn2)cc1 ZINC000880651598 GF On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](c4ccsc4)C3)cn2)cc1 ZINC000880651599 GG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](c4ccsc4)C3)cn2)cc1 ZINC000880651600 GG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC=CC4)CC3)cn2)cc1 ZINC000880651607 GF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC=CC4)CC3)cn2)cc1 ZINC000880651607 GF On-Demand Mild PANC 49 37 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651609 GG On-Demand Mild ITK 19 45 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651609 GG On-Demand Mild PANC 55 38 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651610 GG On-Demand Mild ITK 19 45 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651610 GG On-Demand Mild PANC 55 38 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651611 GG On-Demand Mild ITK 19 45 CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651611 GG On-Demand Mild PANC 55 38 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651612 GG On-Demand Mild ITK 19 45 CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651612 GG On-Demand Mild PANC 55 38 CC(C)[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651613 EG On-Demand Mild ITK 19 51 CC(C)[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651613 EG On-Demand Mild MLNR 27 41 CC(C)[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651613 EG On-Demand Mild PANC 57 40 Cn1nccc1C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651616 GF On-Demand Mild ITK 20 46 Cn1nccc1C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651616 GF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N(C3CCCC3)C3CC3)cn2)cc1 ZINC000880651621 EH On-Demand Mild ITK 27 52 N#Cc1ccc(Cn2cc(NC(=O)N(C3CCCC3)C3CC3)cn2)cc1 ZINC000880651621 EH On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCO)CC3)cn2)cc1 ZINC000880651633 FE On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCO)CC3)cn2)cc1 ZINC000880651633 FE On-Demand Mild PANC 55 39 CN(C[C@@H]1CCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651634 EE On-Demand Mild ITK 21 47 CN(C[C@@H]1CCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651634 EE On-Demand Mild PANC 58 40 CCCO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651639 GH On-Demand Mild ITK 16 46 CCCO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651639 GH On-Demand Mild PANC 53 37 CCCO[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651640 GH On-Demand Mild ITK 16 46 CCCO[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651640 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)NCCCF)cn2)cc1 ZINC000880651643 DE On-Demand Mild ADRB1 42 33 N#Cc1ccc(Cn2cc(NC(=O)NCCCF)cn2)cc1 ZINC000880651643 DE On-Demand Mild ITK 16 55 N#Cc1ccc(Cn2cc(NC(=O)NCCCF)cn2)cc1 ZINC000880651643 DE On-Demand Mild PANC 42 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)(C(F)(F)F)CC3)cn2)cc1 ZINC000880651647 GF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)(C(F)(F)F)CC3)cn2)cc1 ZINC000880651647 GF On-Demand Mild TRPM8 21 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)(C(F)(F)F)CC3)cn2)cc1 ZINC000880651647 GF On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](c4ccco4)C3)cn2)cc1 ZINC000880651650 FG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](c4ccco4)C3)cn2)cc1 ZINC000880651650 FG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](c4ccco4)C3)cn2)cc1 ZINC000880651651 FG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](c4ccco4)C3)cn2)cc1 ZINC000880651651 FG On-Demand Mild PANC 53 36 C[C@H]1CC[C@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651655 DG On-Demand Mild ITK 20 53 C[C@H]1CC[C@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651655 DG On-Demand Mild PANC 61 41 C[C@H]1CC[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651656 DG On-Demand Mild ITK 20 53 C[C@H]1CC[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651656 DG On-Demand Mild PANC 61 41 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651657 DG On-Demand Mild ITK 20 53 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651657 DG On-Demand Mild PANC 61 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(CCOC4)C3)cn2)cc1 ZINC000880651661 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(CCOC4)C3)cn2)cc1 ZINC000880651662 FE On-Demand Mild ITK 16 48 C[C@@H](N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1(C)CC1 ZINC000880651664 EG On-Demand Mild ITK 19 49 COCCCOC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651665 GF On-Demand Mild PDGFRB 15 43 COCCCOC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651665 GF On-Demand Mild ITK 22 50 COCCCOC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651665 GF On-Demand Mild MLNR 25 41 COCCCOC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651665 GF On-Demand Mild PANC 57 40 C[C@H]1CC[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651666 EG On-Demand Mild ITK 18 49 C[C@H]1CC[C@@H](C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651666 EG On-Demand Mild PANC 60 41 C[C@H]1CC[C@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651667 EG On-Demand Mild ITK 18 49 C[C@H]1CC[C@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651667 EG On-Demand Mild PANC 60 41 C[C@@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651668 EG On-Demand Mild ITK 18 49 C[C@@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651668 EG On-Demand Mild PANC 60 41 C[C@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651669 EG On-Demand Mild ITK 18 49 C[C@H]1CC[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651669 EG On-Demand Mild PANC 60 41 CC[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651673 EE On-Demand Mild ITK 15 47 CC[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651673 EE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CCC[C@H]3CC4)cn2)cc1 ZINC000880651680 EG On-Demand Mild ITK 19 52 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CCC[C@H]3CC4)cn2)cc1 ZINC000880651680 EG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCC[C@@H]4C3)cn2)cc1 ZINC000880651686 FE On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCC[C@@H]4C3)cn2)cc1 ZINC000880651686 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCC[C@H]4C3)cn2)cc1 ZINC000880651687 FE On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4CCC[C@H]4C3)cn2)cc1 ZINC000880651687 FE On-Demand Mild PANC 41 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)S1 ZINC000880651688 FG On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)S1 ZINC000880651688 FG On-Demand Mild PANC 57 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)S1 ZINC000880651689 FG On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)S1 ZINC000880651689 FG On-Demand Mild PANC 57 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)S1 ZINC000880651690 FG On-Demand Mild ITK 17 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)S1 ZINC000880651690 FG On-Demand Mild PANC 57 38 CSC(C)(C)CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651691 EG On-Demand Mild ITK 16 52 CSC(C)(C)CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651691 EG On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCO)C3)cn2)cc1 ZINC000880651692 FE On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCO)C3)cn2)cc1 ZINC000880651692 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCO)C3)cn2)cc1 ZINC000880651693 FE On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCO)C3)cn2)cc1 ZINC000880651693 FE On-Demand Mild PANC 41 36 CCCCCN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651694 FF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CCO)C3)cn2)cc1 ZINC000880651698 EE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CCO)C3)cn2)cc1 ZINC000880651698 EE On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CCO)C3)cn2)cc1 ZINC000880651699 EE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CCO)C3)cn2)cc1 ZINC000880651699 EE On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CCO)CC3)cn2)cc1 ZINC000880651700 FC On-Demand Mild ITK 17 53 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CCO)CC3)cn2)cc1 ZINC000880651700 FC On-Demand Mild MLNR 17 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CCO)CC3)cn2)cc1 ZINC000880651700 FC On-Demand Mild FAAH 20 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(CCO)CC3)cn2)cc1 ZINC000880651700 FC On-Demand Mild KCNJ1 15 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3C3CC3)cn2)cc1 ZINC000880651705 FE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3C3CC3)cn2)cc1 ZINC000880651706 FE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCOCC4)C3)cn2)cc1 ZINC000880651710 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCOCC4)C3)cn2)cc1 ZINC000880651710 GD On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCOCC4)C3)cn2)cc1 ZINC000880651711 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCOCC4)C3)cn2)cc1 ZINC000880651711 GD On-Demand Mild PANC 53 37 CN(CCN1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651736 FD On-Demand Mild CASR 46 43 CN(CCN1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651736 FD On-Demand Mild ITK 18 47 CN(CCN1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651736 FD On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C4OCCO4)C3)cn2)cc1 ZINC000880651739 GE On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C4OCCO4)C3)cn2)cc1 ZINC000880651739 GE On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C4OCCO4)C3)cn2)cc1 ZINC000880651740 GE On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C4OCCO4)C3)cn2)cc1 ZINC000880651740 GE On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N(CCC(F)(F)F)CC3CC3)cn2)cc1 ZINC000880651742 GH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N(CCC(F)(F)F)CC3CC3)cn2)cc1 ZINC000880651742 GH On-Demand Mild PANC 53 37 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1 ZINC000880651743 DG On-Demand Mild ITK 16 50 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1 ZINC000880651743 DG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CC4)C(=O)C3)cn2)cc1 ZINC000880651744 FD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CC4)C(=O)C3)cn2)cc1 ZINC000880651744 FD On-Demand Mild PANC 41 36 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651745 FG On-Demand Mild ITK 15 47 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651745 FG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCOCC4)C3)cn2)cc1 ZINC000880651747 FF On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCOCC4)C3)cn2)cc1 ZINC000880651747 FF On-Demand Mild PANC 41 36 Cc1nn(C)cc1[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651748 GG On-Demand Mild ITK 17 44 Cc1nn(C)cc1[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651748 GG On-Demand Mild PANC 53 37 Cc1nn(C)cc1[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651749 GG On-Demand Mild ITK 17 44 Cc1nn(C)cc1[C@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651749 GG On-Demand Mild PANC 53 37 CCSCC[C@H](C)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651751 FH On-Demand Mild ITK 17 50 CCSCC[C@@H](C)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651752 FH On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CN3CCCC3)cn2)cc1 ZINC000880651754 GF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CN3CCCC3)cn2)cc1 ZINC000880651754 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CN3CCCC3)cn2)cc1 ZINC000880651755 GF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CN3CCCC3)cn2)cc1 ZINC000880651755 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H](O)C(F)(F)F)cn2)cc1 ZINC000880651756 GF On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@H](O)C(F)(F)F)cn2)cc1 ZINC000880651757 GF On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H](O)C(F)(F)F)cn2)cc1 ZINC000880651758 GF On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@@H](O)C(F)(F)F)cn2)cc1 ZINC000880651759 GF On-Demand Mild PANC 49 36 N#CCCN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651761 EF On-Demand Mild ITK 16 49 N#CCCN(CC1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651761 EF On-Demand Mild PANC 48 35 CN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651767 CD On-Demand Mild ITK 19 53 CN(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651767 CD On-Demand Mild PANC 53 36 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651768 FD On-Demand Mild ITK 16 51 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651768 FD On-Demand Mild MLNR 24 43 CN(C)CCCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651770 GG On-Demand Mild ITK 18 47 CN(C)CCCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651770 GG On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C#N)CC3)cn2)cc1 ZINC000880651772 EF On-Demand Mild ITK 17 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C#N)CC3)cn2)cc1 ZINC000880651772 EF On-Demand Mild MLNR 23 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C#N)CC3)cn2)cc1 ZINC000880651772 EF On-Demand Mild PANC 55 38 CN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880651775 FD On-Demand Mild ITK 25 47 CN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880651775 FD On-Demand Mild PANC 54 37 C[C@@H](CC#N)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651778 DF On-Demand Mild ITK 19 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCC[C@H]43)cn2)cc1 ZINC000880651780 DF On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCC[C@H]43)cn2)cc1 ZINC000880651780 DF On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@H]43)cn2)cc1 ZINC000880651781 DF On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@H]43)cn2)cc1 ZINC000880651781 DF On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651782 DF On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651782 DF On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651783 DF On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@@H]43)cn2)cc1 ZINC000880651783 DF On-Demand Mild PANC 53 36 C[C@@H](O)CCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651791 EE On-Demand Mild ITK 18 50 C[C@@H](O)CCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651791 EE On-Demand Mild PANC 40 34 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651796 EG On-Demand Mild DPP4 15 42 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651796 EG On-Demand Mild ITK 18 49 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651796 EG On-Demand Mild PANC 55 38 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651798 EG On-Demand Mild DPP4 15 42 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651798 EG On-Demand Mild ITK 18 49 C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880651798 EG On-Demand Mild PANC 55 38 CC[C@@H](C)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651801 EG On-Demand Mild ITK 17 50 CC[C@@H](C)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651801 EG On-Demand Mild PANC 40 34 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880651803 CE On-Demand Mild ITK 29 52 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880651803 CE On-Demand Mild PANC 58 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC4(CCC4)C3)cn2)cc1 ZINC000880651805 FF On-Demand Mild EPHX2 16 50 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC1 ZINC000880651808 DF On-Demand Mild ITK 32 52 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC1 ZINC000880651808 DF On-Demand Mild PANC 57 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CC4)CC3)cn2)cc1 ZINC000880651812 FE On-Demand Mild ITK 19 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CC4)CC3)cn2)cc1 ZINC000880651812 FE On-Demand Mild MLNR 18 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C4CC4)CC3)cn2)cc1 ZINC000880651812 FE On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C4CCCC4)CC3)cn2)cc1 ZINC000880651814 GG On-Demand Mild HRH3 22 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C4CCCC4)CC3)cn2)cc1 ZINC000880651814 GG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C4CCCC4)CC3)cn2)cc1 ZINC000880651814 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3c3ccco3)cn2)cc1 ZINC000880651816 FH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3c3ccco3)cn2)cc1 ZINC000880651816 FH On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3c3ccco3)cn2)cc1 ZINC000880651817 FH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3c3ccco3)cn2)cc1 ZINC000880651817 FH On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCS(=O)CC3)cn2)cc1 ZINC000880651818 ED On-Demand Mild ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@H]4CCC[C@@H]4O)CC3)cn2)cc1 ZINC000880651823 GD On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@H]4CCC[C@@H]4O)CC3)cn2)cc1 ZINC000880651823 GD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@@H]4CCC[C@@H]4O)CC3)cn2)cc1 ZINC000880651824 GD On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@@H]4CCC[C@@H]4O)CC3)cn2)cc1 ZINC000880651824 GD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@H]4CCC[C@H]4O)CC3)cn2)cc1 ZINC000880651825 GD On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@H]4CCC[C@H]4O)CC3)cn2)cc1 ZINC000880651825 GD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@@H]4CCC[C@H]4O)CC3)cn2)cc1 ZINC000880651826 GD On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@@H]4CCC[C@H]4O)CC3)cn2)cc1 ZINC000880651826 GD On-Demand Mild PANC 41 36 CCC(C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651829 EH On-Demand Mild ITK 16 53 CCC(C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651829 EH On-Demand Mild PANC 59 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CC4)C3)cn2)cc1 ZINC000880651832 EG On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CC4)C3)cn2)cc1 ZINC000880651832 EG On-Demand Mild MLNR 29 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CC4)C3)cn2)cc1 ZINC000880651832 EG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CC4)C3)cn2)cc1 ZINC000880651833 EG On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CC4)C3)cn2)cc1 ZINC000880651833 EG On-Demand Mild MLNR 29 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CC4)C3)cn2)cc1 ZINC000880651833 EG On-Demand Mild PANC 55 38 CC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651834 DG On-Demand Mild ITK 18 49 CC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651834 DG On-Demand Mild MLNR 27 41 CC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651834 DG On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4C(=O)CC[C@H]4C3)cn2)cc1 ZINC000880651841 FD On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4C(=O)CC[C@@H]4C3)cn2)cc1 ZINC000880651842 FD On-Demand Mild PANC 53 37 CCC1(O)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651843 FF On-Demand Mild ITK 15 49 CCC1(O)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651843 FF On-Demand Mild S1PR2 26 45 CCCN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651844 FF On-Demand Mild ITK 15 49 CCCN(CC(C)(C)O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651844 FF On-Demand Mild PANC 48 35 CCOC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651849 FF On-Demand Mild ITK 17 47 CCOC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651849 FF On-Demand Mild PANC 56 39 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651851 EG On-Demand Mild ITK 19 50 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651851 EG On-Demand Mild MLNR 47 44 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651851 EG On-Demand Mild PANC 56 39 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651852 EG On-Demand Mild ITK 19 50 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651852 EG On-Demand Mild MLNR 47 44 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1C ZINC000880651852 EG On-Demand Mild PANC 56 39 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880651853 EG On-Demand Mild ITK 19 50 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880651853 EG On-Demand Mild MLNR 47 44 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880651853 EG On-Demand Mild PANC 56 39 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651854 EG On-Demand Mild ITK 19 50 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651854 EG On-Demand Mild MLNR 47 44 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1C ZINC000880651854 EG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC(OCC(F)F)C3)cn2)cc1 ZINC000880651861 FE On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC(OCC(F)F)C3)cn2)cc1 ZINC000880651861 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4OCC[C@@H]4C3)cn2)cc1 ZINC000880651866 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4OCC[C@@H]4C3)cn2)cc1 ZINC000880651866 FE On-Demand Mild PANC 53 37 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880651867 FF On-Demand Mild ITK 25 51 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880651867 FF On-Demand Mild PANC 60 40 C[C@@H](CO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651868 FF On-Demand Mild ITK 17 49 C[C@@H](CO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651868 FF On-Demand Mild MLNR 20 40 C[C@@H](CO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651868 FF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)NOCCC3CC3)cn2)cc1 ZINC000880651869 EF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)NOCCC3CC3)cn2)cc1 ZINC000880651869 EF On-Demand Mild PANC 58 39 CCCCN(CCCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651871 FF On-Demand Mild ITK 16 50 CCCCN(CCCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651871 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC=CC[C@H]3C(F)(F)F)cn2)cc1 ZINC000880651872 GH On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC=CC[C@H]3C(F)(F)F)cn2)cc1 ZINC000880651872 GH On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880651873 FF On-Demand Mild ITK 23 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880651873 FF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880651875 FF On-Demand Mild ITK 23 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880651875 FF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880651877 FF On-Demand Mild ITK 23 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880651877 FF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880651879 FF On-Demand Mild ITK 23 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880651879 FF On-Demand Mild PANC 56 39 C[C@H]1C[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651881 FE On-Demand Mild ITK 16 47 C[C@H]1C[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651881 FE On-Demand Mild PANC 53 37 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880651885 GF On-Demand Mild ITK 15 47 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880651887 GF On-Demand Mild ITK 15 47 CC1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651891 EH On-Demand Mild ITK 18 50 CC1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651891 EH On-Demand Mild PANC 56 39 C[C@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651895 GF On-Demand Mild ITK 17 47 C[C@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651895 GF On-Demand Mild PANC 53 37 C[C@H]1[C@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651896 GF On-Demand Mild ITK 17 47 C[C@H]1[C@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651896 GF On-Demand Mild PANC 53 37 C[C@@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651900 GF On-Demand Mild ITK 17 47 C[C@@H]1[C@@H](N2CCCC2)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651900 GF On-Demand Mild PANC 53 37 C#C[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651901 EF On-Demand Mild ITK 16 48 C#C[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651901 EF On-Demand Mild PANC 41 36 C[C@]1(CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651902 EE On-Demand Mild ITK 19 48 C[C@@]1(CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651903 EE On-Demand Mild ITK 19 48 C#C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651904 EF On-Demand Mild ITK 16 48 C#C[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880651904 EF On-Demand Mild PANC 41 36 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)CSc3ccncc3)sc2C1 ZINC000880651905 HH On-Demand Anodyne FAS 43 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](CCF)C3)cn2)cc1 ZINC000880651906 FE On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](CCF)C3)cn2)cc1 ZINC000880651906 FE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](CCF)C3)cn2)cc1 ZINC000880651908 FE On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](CCF)C3)cn2)cc1 ZINC000880651908 FE On-Demand Mild PANC 54 37 CON(C)CCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651910 ED On-Demand Mild ITK 20 51 CON(C)CCNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651910 ED On-Demand Mild PANC 41 35 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCC[C@@H]1C#N ZINC000880651919 EF On-Demand Mild ITK 24 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCC[C@@H]1C#N ZINC000880651919 EF On-Demand Mild PANC 53 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCC[C@H]1C#N ZINC000880651921 EF On-Demand Mild ITK 24 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCC[C@H]1C#N ZINC000880651921 EF On-Demand Mild PANC 53 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCC[C@@H]1C#N ZINC000880651922 EF On-Demand Mild ITK 24 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCC[C@@H]1C#N ZINC000880651922 EF On-Demand Mild PANC 53 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCC[C@H]1C#N ZINC000880651923 EF On-Demand Mild ITK 24 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCC[C@H]1C#N ZINC000880651923 EF On-Demand Mild PANC 53 36 CN(C[C@@H]1CCc2nccn2C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651924 GF On-Demand Mild ITK 16 44 CN(C[C@@H]1CCc2nccn2C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651924 GF On-Demand Mild PANC 60 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CC[C@@H](O)[C@@H]43)cn2)cc1 ZINC000880651925 FE On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CC[C@@H](O)[C@@H]43)cn2)cc1 ZINC000880651925 FE On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@]4(CO)C3)cn2)cc1 ZINC000880651926 ED On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@]4(CO)C3)cn2)cc1 ZINC000880651928 ED On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@@]4(CO)C3)cn2)cc1 ZINC000880651929 ED On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@@]4(CO)C3)cn2)cc1 ZINC000880651931 ED On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CCOCC4)C3)cn2)cc1 ZINC000880651933 FF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CCOCC4)C3)cn2)cc1 ZINC000880651933 FF On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCCO4)C3)cn2)cc1 ZINC000880651937 EE On-Demand Mild ITK 16 49 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651939 DF On-Demand Mild ITK 16 52 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880651939 DF On-Demand Mild PANC 41 35 C[C@H]1[C@H](C(F)(F)F)OCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651941 GF On-Demand Mild ITK 15 45 C[C@H]1[C@H](C(F)(F)F)OCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651941 GF On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651942 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC([C@H]4CCOC4)C3)cn2)cc1 ZINC000880651942 FE On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651943 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC([C@@H]4CCOC4)C3)cn2)cc1 ZINC000880651943 FE On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C(F)F)C3)cn2)cc1 ZINC000880651945 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C(F)F)C3)cn2)cc1 ZINC000880651945 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C(F)F)C3)cn2)cc1 ZINC000880651947 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C(F)F)C3)cn2)cc1 ZINC000880651947 FE On-Demand Mild PANC 41 36 C[C@@H]1[C@@H](C(F)(F)F)OCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651948 GF On-Demand Mild ITK 15 45 C[C@@H]1[C@@H](C(F)(F)F)OCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651948 GF On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](F)C3)cn2)cc1 ZINC000880651951 DE On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](F)C3)cn2)cc1 ZINC000880651951 DE On-Demand Mild MLNR 38 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](F)C3)cn2)cc1 ZINC000880651951 DE On-Demand Mild PANC 55 38 C[C@H]1C(=O)N(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651952 FD On-Demand Mild ITK 17 50 C[C@H]1C(=O)N(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651952 FD On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](F)C3)cn2)cc1 ZINC000880651954 DE On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](F)C3)cn2)cc1 ZINC000880651954 DE On-Demand Mild MLNR 38 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](F)C3)cn2)cc1 ZINC000880651954 DE On-Demand Mild PANC 55 38 C[C@H]1CC[C@H](C(F)(F)F)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651955 GH On-Demand Mild PANC 63 43 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(C3)CC4(F)F)cn2)cc1 ZINC000880651956 FG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(C3)CC4(F)F)cn2)cc1 ZINC000880651957 FG On-Demand Mild ITK 15 48 C[C@@H]1CC[C@@H](C(F)(F)F)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651960 GH On-Demand Mild PANC 63 43 C[C@H]1CC[C@@H](C(F)(F)F)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651962 GH On-Demand Mild PANC 63 43 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651964 FG On-Demand Mild ITK 16 47 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651964 FG On-Demand Mild MLNR 32 42 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651964 FG On-Demand Mild PANC 54 37 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651966 FG On-Demand Mild ITK 16 47 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651966 FG On-Demand Mild MLNR 32 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880651966 FG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)NCCN3CC=CCC3)cn2)cc1 ZINC000880651971 FE On-Demand Mild CCR3 18 44 N#Cc1ccc(Cn2cc(NC(=O)NCCN3CC=CCC3)cn2)cc1 ZINC000880651971 FE On-Demand Mild ITK 15 48 COC[C@]1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651972 FE On-Demand Mild ITK 15 44 COC[C@]1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651972 FE On-Demand Mild PANC 41 35 COC[C@@]1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651974 FE On-Demand Mild ITK 15 44 COC[C@@]1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880651974 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)(F)C3)cn2)cc1 ZINC000880651980 EF On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)(F)C3)cn2)cc1 ZINC000880651980 EF On-Demand Mild PANC 41 36 C[C@H](CCO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651981 EE On-Demand Mild ITK 18 52 C[C@@H](CCO)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880651983 EE On-Demand Mild ITK 18 52 CN1CC[C@@]2(CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)C1 ZINC000880651984 FE On-Demand Mild ITK 16 49 CN1CC[C@@]2(CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)C1 ZINC000880651984 FE On-Demand Mild PANC 41 36 C[C@H]1CCOCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652001 EE On-Demand Mild ITK 15 47 C[C@H]1CCOCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652001 EE On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC4CC3(c3ccccc3)C4)cn2)cc1 ZINC000880652002 GH On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC4CC3(c3ccccc3)C4)cn2)cc1 ZINC000880652002 GH On-Demand Mild PANC 48 36 C[C@@H]1CCOCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652003 EE On-Demand Mild ITK 15 47 C[C@@H]1CCOCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652003 EE On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)NC(CF)CF)cn2)cc1 ZINC000880652007 DE On-Demand Mild ITK 16 55 N#Cc1ccc(Cn2cc(NC(=O)NC(CF)CF)cn2)cc1 ZINC000880652007 DE On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C(=O)C4CC4)C3)cn2)cc1 ZINC000880652009 FD On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCN(C(=O)C4CC4)C3)cn2)cc1 ZINC000880652009 FD On-Demand Mild PANC 53 38 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652010 GE On-Demand Mild ITK 15 47 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652010 GE On-Demand Mild PANC 53 37 CC1(CO)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652012 ED On-Demand Mild ITK 18 52 CC1(CO)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652012 ED On-Demand Mild PANC 42 37 Cn1ncc2c1CCCN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880652016 GF On-Demand Mild ITK 15 47 Cn1ncc2c1CCCN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880652016 GF On-Demand Mild PANC 41 36 CN(C)C(=O)CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652025 GF On-Demand Mild ITK 20 47 CN(C)C(=O)CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652025 GF On-Demand Mild PANC 53 37 CO[C@@]1(C)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652026 FF On-Demand Mild ITK 19 46 CO[C@@]1(C)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652026 FF On-Demand Mild PANC 47 35 CCC1(O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652028 ED On-Demand Mild ITK 18 54 CCC1(O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652028 ED On-Demand Mild PANC 41 35 CN(C)CC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1 ZINC000880652029 FE On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(CCCOC4)C3)cn2)cc1 ZINC000880652032 FF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(CCCOC4)C3)cn2)cc1 ZINC000880652033 FF On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652036 EE On-Demand Mild ITK 18 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652036 EE On-Demand Mild MLNR 44 43 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652036 EE On-Demand Mild PANC 56 39 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652037 EE On-Demand Mild ITK 18 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652037 EE On-Demand Mild MLNR 44 43 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652037 EE On-Demand Mild PANC 56 39 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652038 EE On-Demand Mild ITK 18 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652038 EE On-Demand Mild MLNR 44 43 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1O ZINC000880652038 EE On-Demand Mild PANC 56 39 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652039 EE On-Demand Mild ITK 18 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652039 EE On-Demand Mild MLNR 44 43 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1O ZINC000880652039 EE On-Demand Mild PANC 56 39 CCC(CC)N(CC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652042 EH On-Demand Mild ITK 17 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@](F)(C#N)C3)cn2)cc1 ZINC000880652043 EE On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@](F)(C#N)C3)cn2)cc1 ZINC000880652043 EE On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@](F)(C#N)C3)cn2)cc1 ZINC000880652044 EE On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@](F)(C#N)C3)cn2)cc1 ZINC000880652044 EE On-Demand Mild PANC 40 35 C[C@H](O)CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCCCC1 ZINC000880652045 GG On-Demand Mild ITK 31 47 C[C@H](O)CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCCCC1 ZINC000880652045 GG On-Demand Mild PANC 53 35 C[C@H]1C[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652049 DF On-Demand Mild ITK 19 53 C[C@H]1C[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652049 DF On-Demand Mild PANC 56 38 CO[C@@H](C)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652058 EE On-Demand Mild ITK 18 49 CO[C@@H](C)CN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652058 EE On-Demand Mild PANC 53 36 CCC[C@]1(CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652071 FF On-Demand Mild ITK 17 45 CN(CC1(CO)CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652073 EE On-Demand Mild ITK 19 49 CN(CC1(CO)CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652073 EE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N(CC3CC3)CC3CC3)cn2)cc1 ZINC000880652082 EG On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N(CC3CC3)CC3CC3)cn2)cc1 ZINC000880652082 EG On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCCCC3)cn2)cc1 ZINC000880652083 FF On-Demand Mild ITK 26 49 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCCCC3)cn2)cc1 ZINC000880652083 FF On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCCOC4)C3)cn2)cc1 ZINC000880652086 FE On-Demand Mild ITK 15 47 CCOCCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652087 FE On-Demand Mild ITK 16 48 CCOCCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652087 FE On-Demand Mild PANC 45 35 C[C@@H](CF)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652089 DE On-Demand Mild ITK 16 53 C[C@@H](CF)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652089 DE On-Demand Mild PANC 41 36 C[C@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652108 EG On-Demand Mild ITK 27 49 C[C@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652108 EG On-Demand Mild MLNR 32 41 C[C@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652108 EG On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@H]3c3ccco3)cn2)cc1 ZINC000880652115 GI On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@H]3c3ccco3)cn2)cc1 ZINC000880652115 GI On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3c3ccco3)cn2)cc1 ZINC000880652119 GI On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3c3ccco3)cn2)cc1 ZINC000880652119 GI On-Demand Mild PANC 54 37 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652121 FF On-Demand Mild ITK 15 47 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652121 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OCC4CC4)C3)cn2)cc1 ZINC000880652125 GG On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OCC4CC4)C3)cn2)cc1 ZINC000880652125 GG On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OCC4CC4)C3)cn2)cc1 ZINC000880652127 GG On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OCC4CC4)C3)cn2)cc1 ZINC000880652127 GG On-Demand Mild PANC 49 36 CN(C[C@@H]1CCn2ccnc2C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652129 GF On-Demand Mild ITK 16 44 CN(C[C@@H]1CCn2ccnc2C1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652129 GF On-Demand Mild PANC 55 38 C[C@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652155 GH On-Demand Mild ITK 15 45 C[C@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652155 GH On-Demand Mild PANC 47 34 C[C@@H]1C[C@@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652156 GH On-Demand Mild ITK 15 45 C[C@@H]1C[C@@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652156 GH On-Demand Mild PANC 47 34 C[C@@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652157 GH On-Demand Mild ITK 15 45 C[C@@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652157 GH On-Demand Mild PANC 47 34 COCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652177 FD On-Demand Mild ITK 23 52 COCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652177 FD On-Demand Mild PANC 57 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880652205 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880652205 GG On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H](C4CCC4)C3)cn2)cc1 ZINC000880652207 GG On-Demand Mild ITK 15 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H](C4CCC4)C3)cn2)cc1 ZINC000880652207 GG On-Demand Mild PANC 49 36 COc1ccc(CC(=O)NCc2cc(O)nc(SC)n2)cc1F ZINC000880652221 ED On-Demand Anodyne DRTS_TRYCR 43 29 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](O)C[C@H]3C3CC3)cn2)cc1 ZINC000880652224 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](O)C[C@H]3C3CC3)cn2)cc1 ZINC000880652224 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](O)C[C@@H]3C3CC3)cn2)cc1 ZINC000880652225 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](O)C[C@@H]3C3CC3)cn2)cc1 ZINC000880652225 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](O)C[C@H]3C3CC3)cn2)cc1 ZINC000880652226 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](O)C[C@H]3C3CC3)cn2)cc1 ZINC000880652226 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](O)C[C@@H]3C3CC3)cn2)cc1 ZINC000880652227 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](O)C[C@@H]3C3CC3)cn2)cc1 ZINC000880652227 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCSCC4)CC3)cn2)cc1 ZINC000880652228 GH On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCSCC4)CC3)cn2)cc1 ZINC000880652228 GH On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880652229 EG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880652229 EG On-Demand Mild PANC 53 36 CCOC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652231 FE On-Demand Mild ITK 15 47 CCOC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652231 FE On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4C[C@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652234 FD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCN4C[C@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652234 FD On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccco4)CC3)cn2)cc1 ZINC000880652235 GH On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccco4)CC3)cn2)cc1 ZINC000880652235 GH On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3OC4CCC3CC4)cn2)cc1 ZINC000880652240 EF On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3OC4CCC3CC4)cn2)cc1 ZINC000880652240 EF On-Demand Mild PANC 58 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC(F)(F)C3)cn2)cc1 ZINC000880652241 EG On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC(F)(F)C3)cn2)cc1 ZINC000880652241 EG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](CF)C3)cn2)cc1 ZINC000880652244 EE On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](CF)C3)cn2)cc1 ZINC000880652244 EE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](CF)C3)cn2)cc1 ZINC000880652245 EE On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](CF)C3)cn2)cc1 ZINC000880652245 EE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCO)CC3)cn2)cc1 ZINC000880652246 FF On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCO)CC3)cn2)cc1 ZINC000880652246 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCO)CC3)cn2)cc1 ZINC000880652247 FF On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCO)CC3)cn2)cc1 ZINC000880652247 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@]4(C3)CC4(F)F)cn2)cc1 ZINC000880652255 FG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@]4(C3)CC4(F)F)cn2)cc1 ZINC000880652256 FG On-Demand Mild ITK 15 47 CC[C@@](C)(NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652266 EH On-Demand Mild ITK 20 49 CC[C@@](C)(NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652266 EH On-Demand Mild PANC 65 44 C#CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652268 EF On-Demand Mild ITK 16 50 C#CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652268 EF On-Demand Mild MLNR 28 42 C#CC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652268 EF On-Demand Mild PANC 56 39 CN(CCN1CCCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652273 FF On-Demand Mild ITK 28 50 CN(CCN1CCCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652273 FF On-Demand Mild MCHR1 24 43 CN(CCN1CCCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652273 FF On-Demand Mild PANC 41 36 C[C@H]1CCC(C)(C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652275 EH On-Demand Mild ITK 19 51 C[C@H]1CCC(C)(C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652275 EH On-Demand Mild PANC 55 38 C[C@@H]1CC(F)(F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652279 FG On-Demand Mild ITK 15 47 C[C@@H]1CC(F)(F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652279 FG On-Demand Mild PANC 40 35 C[C@H]1CC(F)(F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652280 FG On-Demand Mild ITK 15 47 C[C@H]1CC(F)(F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652280 FG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CC34CCOCC4)cn2)cc1 ZINC000880652292 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CC34CCOCC4)cn2)cc1 ZINC000880652292 FE On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC34CCOCC4)cn2)cc1 ZINC000880652296 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC34CCOCC4)cn2)cc1 ZINC000880652296 FE On-Demand Mild PANC 40 34 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCC[C@H]1O ZINC000880652299 FF On-Demand Mild ITK 29 49 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCC[C@H]1O ZINC000880652299 FF On-Demand Mild PANC 55 37 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCN2CCO[C@H]1C2 ZINC000880652302 GD On-Demand Mild ITK 18 45 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCN2CCO[C@H]1C2 ZINC000880652302 GD On-Demand Mild PANC 49 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCN2CCO[C@H]1C2 ZINC000880652305 GD On-Demand Mild ITK 18 45 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCN2CCO[C@H]1C2 ZINC000880652305 GD On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCCOC3)cn2)cc1 ZINC000880652308 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@H]3CCCOC3)cn2)cc1 ZINC000880652312 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3[C@@H]3CCCOC3)cn2)cc1 ZINC000880652315 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCCOC3)cn2)cc1 ZINC000880652317 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccsc4)CC3)cn2)cc1 ZINC000880652318 GI On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccsc4)CC3)cn2)cc1 ZINC000880652318 GI On-Demand Mild PANC 49 36 CC(C)C1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652320 DG On-Demand Mild ITK 16 51 CC(C)C1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652320 DG On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC(F)F)C3)cn2)cc1 ZINC000880652327 EF On-Demand Mild ITK 15 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC(F)F)C3)cn2)cc1 ZINC000880652327 EF On-Demand Mild PANC 41 36 CN(C)CC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652329 EE On-Demand Mild ITK 17 53 CN(C)CC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652329 EE On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)(C(F)F)CC3)cn2)cc1 ZINC000880652330 GE On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(O)(C(F)F)CC3)cn2)cc1 ZINC000880652330 GE On-Demand Mild S1PR2 22 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC4(CC4)C3)cn2)cc1 ZINC000880652335 EG On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880652337 GE On-Demand Mild ITK 18 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880652337 GE On-Demand Mild PANC 53 37 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1(C)C ZINC000880652338 FF On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880652339 GE On-Demand Mild ITK 18 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880652339 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880652341 GE On-Demand Mild ITK 18 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880652341 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880652343 GE On-Demand Mild ITK 18 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880652343 GE On-Demand Mild PANC 53 37 C[C@@H](N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)O ZINC000880652346 EE On-Demand Mild ITK 17 50 C[C@@H](N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)O ZINC000880652346 EE On-Demand Mild PANC 53 36 CN(CC1(C)COC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652349 EE On-Demand Mild ITK 17 49 CN(CC1(C)COC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652349 EE On-Demand Mild PANC 55 37 COC[C@@]1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652351 FF On-Demand Mild ITK 17 46 COC[C@]1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652353 FF On-Demand Mild ITK 17 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC34CCC4)cn2)cc1 ZINC000880652354 EG On-Demand Mild ITK 17 51 C=CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652356 GE On-Demand Mild ITK 17 45 C=CCN1CC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652356 GE On-Demand Mild PANC 40 35 CC[C@H]1[C@@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652357 FE On-Demand Mild ITK 15 47 CC[C@H]1[C@@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652357 FE On-Demand Mild PANC 53 37 C=CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652358 GE On-Demand Mild ITK 17 45 C=CCN1CC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652358 GE On-Demand Mild PANC 40 35 CC[C@@H]1[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652359 FE On-Demand Mild ITK 15 47 CC[C@@H]1[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652359 FE On-Demand Mild PANC 53 37 CC[C@H]1[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652364 FE On-Demand Mild ITK 15 47 CC[C@H]1[C@H](CO)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652364 FE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C3)cn2)cc1 ZINC000880652365 DD On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C3)cn2)cc1 ZINC000880652365 DD On-Demand Mild MLNR 28 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C3)cn2)cc1 ZINC000880652365 DD On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4COC[C@@H](C3)O4)cn2)cc1 ZINC000880652369 FD On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4COC[C@@H](C3)O4)cn2)cc1 ZINC000880652369 FD On-Demand Mild PANC 53 35 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880652371 GD On-Demand Mild ITK 15 47 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880652371 GD On-Demand Mild MLNR 22 40 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880652372 GD On-Demand Mild ITK 15 47 C[C@H](O)CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)C1 ZINC000880652372 GD On-Demand Mild MLNR 22 40 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652382 ED On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652382 ED On-Demand Mild MLNR 26 41 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652382 ED On-Demand Mild PANC 54 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652383 ED On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652383 ED On-Demand Mild MLNR 26 41 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652383 ED On-Demand Mild PANC 54 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652384 ED On-Demand Mild ITK 17 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652384 ED On-Demand Mild MLNR 26 41 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1O ZINC000880652384 ED On-Demand Mild PANC 54 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652385 ED On-Demand Mild ITK 17 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652385 ED On-Demand Mild MLNR 26 41 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1O ZINC000880652385 ED On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC(F)F)C3)cn2)cc1 ZINC000880652391 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC(F)F)C3)cn2)cc1 ZINC000880652391 GG On-Demand Mild PANC 42 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC(F)F)C3)cn2)cc1 ZINC000880652392 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC(F)F)C3)cn2)cc1 ZINC000880652392 GG On-Demand Mild PANC 42 36 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(=O)C4)cn2)cc1 ZINC000880652407 EF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(=O)C4)cn2)cc1 ZINC000880652407 EF On-Demand Mild PANC 57 40 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652408 FE On-Demand Mild ITK 15 49 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652408 FE On-Demand Mild MLNR 40 41 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652408 FE On-Demand Mild PANC 54 37 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652409 FE On-Demand Mild ITK 15 49 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652409 FE On-Demand Mild MLNR 40 41 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652409 FE On-Demand Mild PANC 54 37 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652410 FE On-Demand Mild ITK 15 49 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652410 FE On-Demand Mild MLNR 40 41 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880652410 FE On-Demand Mild PANC 54 37 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652411 FE On-Demand Mild ITK 15 49 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652411 FE On-Demand Mild MLNR 40 41 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880652411 FE On-Demand Mild PANC 54 37 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOCC1 ZINC000880652418 FF On-Demand Mild ITK 15 48 CCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOCC1 ZINC000880652418 FF On-Demand Mild PANC 41 35 C[C@H]1[C@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652421 GH On-Demand Mild ITK 15 47 C[C@H]1[C@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652421 GH On-Demand Mild PANC 56 39 C[C@@H]1[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652428 GH On-Demand Mild ITK 15 47 C[C@@H]1[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652428 GH On-Demand Mild PANC 56 39 C[C@]1(O)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652429 FF On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3C3CCOCC3)cn2)cc1 ZINC000880652437 GG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3C3CCOCC3)cn2)cc1 ZINC000880652439 GG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCO4)CC3)cn2)cc1 ZINC000880652445 FF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCO4)CC3)cn2)cc1 ZINC000880652445 FF On-Demand Mild TRPM8 16 47 C[C@@]1(C#N)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652446 EF On-Demand Mild ITK 16 49 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1CO ZINC000880652451 EE On-Demand Mild ITK 18 48 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1CO ZINC000880652451 EE On-Demand Mild PANC 57 40 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1CO ZINC000880652453 EE On-Demand Mild ITK 18 48 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1CO ZINC000880652453 EE On-Demand Mild PANC 57 40 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1CO ZINC000880652456 EE On-Demand Mild ITK 18 48 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1CO ZINC000880652456 EE On-Demand Mild PANC 57 40 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1CO ZINC000880652458 EE On-Demand Mild ITK 18 48 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1CO ZINC000880652458 EE On-Demand Mild PANC 57 40 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](CC)O1 ZINC000880652486 FG On-Demand Mild ITK 15 51 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](CC)O1 ZINC000880652486 FG On-Demand Mild PANC 56 37 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](CC)O1 ZINC000880652487 FG On-Demand Mild ITK 15 51 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](CC)O1 ZINC000880652487 FG On-Demand Mild PANC 56 37 C[C@H]1[C@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652489 FF On-Demand Mild ITK 16 48 C[C@H]1[C@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652489 FF On-Demand Mild PANC 54 36 C[C@@H]1[C@@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652490 FF On-Demand Mild ITK 16 48 C[C@@H]1[C@@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652490 FF On-Demand Mild PANC 54 36 C[C@H]1[C@@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652492 FF On-Demand Mild ITK 16 48 C[C@H]1[C@@H](O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652492 FF On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)NC34CCC(CC3)CC4)cn2)cc1 ZINC000880652493 EH On-Demand Mild ITK 19 51 N#Cc1ccc(Cn2cc(NC(=O)NC34CCC(CC3)CC4)cn2)cc1 ZINC000880652493 EH On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3C3CCC3)cn2)cc1 ZINC000880652494 FF On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@H]3C3CCC3)cn2)cc1 ZINC000880652494 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3C3CCC3)cn2)cc1 ZINC000880652495 FF On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC[C@@H]3C3CCC3)cn2)cc1 ZINC000880652495 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)CC3)cn2)cc1 ZINC000880652496 EF On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)CC3)cn2)cc1 ZINC000880652496 EF On-Demand Mild MLNR 34 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)CC3)cn2)cc1 ZINC000880652496 EF On-Demand Mild PANC 56 39 CN(CC1=CCSC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652497 FF On-Demand Mild ITK 17 47 CN(CC1=CCSC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652497 FF On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4COC[C@H]4C3)cn2)cc1 ZINC000880652500 ED On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4COC[C@H]4C3)cn2)cc1 ZINC000880652500 ED On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC4CCC4)C3)cn2)cc1 ZINC000880652501 GG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC4CCC4)C3)cn2)cc1 ZINC000880652501 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC4CCC4)C3)cn2)cc1 ZINC000880652502 GG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC4CCC4)C3)cn2)cc1 ZINC000880652502 GG On-Demand Mild PANC 54 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCC2)O1 ZINC000880652503 FF On-Demand Mild ITK 15 45 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCC2)O1 ZINC000880652503 FF On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCC2)O1 ZINC000880652504 FF On-Demand Mild ITK 15 45 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCC2)O1 ZINC000880652504 FF On-Demand Mild PANC 41 36 CN(CC1=CCCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652505 FF On-Demand Mild ITK 17 47 CN(CC1=CCCOC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652505 FF On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3O[C@H]4C=C[C@H]3CC4)cn2)cc1 ZINC000880652506 EF On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3O[C@H]4C=C[C@H]3CC4)cn2)cc1 ZINC000880652506 EF On-Demand Mild PANC 57 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4ccncn4)CC3)cn2)cc1 ZINC000880652511 GG On-Demand Mild ITK 17 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCc2cccnc21 ZINC000880652513 FE On-Demand Anodyne PAPA1_CARPA 36 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCc2cccnc21 ZINC000880652513 FE On-Demand Anodyne REN 53 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCc2cccnc21 ZINC000880652514 FE On-Demand Anodyne PAPA1_CARPA 36 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCc2cccnc21 ZINC000880652514 FE On-Demand Anodyne REN 53 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCc2cccnc21 ZINC000880652515 FE On-Demand Anodyne PAPA1_CARPA 36 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCc2cccnc21 ZINC000880652515 FE On-Demand Anodyne REN 53 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCc2cccnc21 ZINC000880652516 FE On-Demand Anodyne PAPA1_CARPA 36 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCc2cccnc21 ZINC000880652516 FE On-Demand Anodyne REN 53 36 CC(C)[C@H]1CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652519 DG On-Demand Mild ITK 19 51 CC(C)[C@H]1CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652519 DG On-Demand Mild PANC 57 40 CN1CCCC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652521 GE On-Demand Mild ITK 28 45 CN1CCCC[C@@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652521 GE On-Demand Mild PANC 41 36 CN1CCCC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652522 GE On-Demand Mild ITK 28 45 CN1CCCC[C@H](N(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1=O ZINC000880652522 GE On-Demand Mild PANC 41 36 C#C[C@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)C ZINC000880652523 EF On-Demand Mild ITK 15 50 C#C[C@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)C ZINC000880652523 EF On-Demand Mild PANC 53 36 C#C[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)C ZINC000880652524 EF On-Demand Mild ITK 15 50 C#C[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(C)(C)C ZINC000880652524 EF On-Demand Mild PANC 53 36 COC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652527 EE On-Demand Mild DPP4 15 41 COC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652527 EE On-Demand Mild ITK 20 47 COC[C@@H]1CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652527 EE On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCCC[C@@H]3C4)cn2)cc1 ZINC000880652530 EG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCCC[C@@H]3C4)cn2)cc1 ZINC000880652530 EG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCCC[C@H]3C4)cn2)cc1 ZINC000880652531 EG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCCC[C@H]3C4)cn2)cc1 ZINC000880652531 EG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@@]34CCCC[C@H]3C4)cn2)cc1 ZINC000880652532 EG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@@]34CCCC[C@H]3C4)cn2)cc1 ZINC000880652532 EG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@@]34CCCC[C@@H]3C4)cn2)cc1 ZINC000880652533 EG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N[C@@]34CCCC[C@@H]3C4)cn2)cc1 ZINC000880652533 EG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCC4)CC3)cn2)cc1 ZINC000880652534 GG On-Demand Mild ITK 19 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCC4)CC3)cn2)cc1 ZINC000880652534 GG On-Demand Mild MLNR 25 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(OC4CCC4)CC3)cn2)cc1 ZINC000880652534 GG On-Demand Mild PANC 55 39 CN1CCO[C@H](CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652536 FD On-Demand Mild ITK 27 44 CN1CCO[C@H](CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652536 FD On-Demand Mild PANC 56 38 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@@H]21 ZINC000880652540 FE On-Demand Mild ITK 20 49 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@@H]21 ZINC000880652540 FE On-Demand Mild MLNR 20 40 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@@H]21 ZINC000880652540 FE On-Demand Mild PANC 56 39 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@H]21 ZINC000880652543 FE On-Demand Mild ITK 20 49 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@H]21 ZINC000880652543 FE On-Demand Mild MLNR 20 40 CN1CC[C@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)CC[C@H]21 ZINC000880652543 FE On-Demand Mild PANC 56 39 COC[C@@H]1CCCN1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652546 FD On-Demand Mild ITK 19 47 COC[C@@H]1CCCN1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652546 FD On-Demand Mild PANC 55 39 C#C[C@](C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652548 DF On-Demand Mild ITK 15 51 C#C[C@](C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652548 DF On-Demand Mild PANC 59 40 C#C[C@@](C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652549 DF On-Demand Mild ITK 15 51 C#C[C@@](C)(CC)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652549 DF On-Demand Mild PANC 59 40 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](CO)[C@H](C(F)(F)F)C3)cn2)cc1 ZINC000880652553 GE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5C=C[C@@H](O5)[C@H]4C3)cn2)cc1 ZINC000880652554 FE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H]5C=C[C@@H](O5)[C@H]4C3)cn2)cc1 ZINC000880652554 FE On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H]5C=C[C@@H](O5)[C@H]4C3)cn2)cc1 ZINC000880652555 FE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H]5C=C[C@@H](O5)[C@H]4C3)cn2)cc1 ZINC000880652555 FE On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C3)[C@H]3C=C[C@H]4O3)cn2)cc1 ZINC000880652556 FE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C3)[C@H]3C=C[C@H]4O3)cn2)cc1 ZINC000880652556 FE On-Demand Mild PANC 53 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@](C)(C(F)F)O1 ZINC000880652559 GG On-Demand Mild PANC 40 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@](C)(C(F)F)O1 ZINC000880652560 GG On-Demand Mild PANC 40 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@](C)(C(F)F)O1 ZINC000880652561 GG On-Demand Mild PANC 40 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@](C)(C(F)F)O1 ZINC000880652562 GG On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CO)CC3)cn2)cc1 ZINC000880652564 FE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CO)CC3)cn2)cc1 ZINC000880652564 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CO)CC3)cn2)cc1 ZINC000880652567 FE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CO)CC3)cn2)cc1 ZINC000880652567 FE On-Demand Mild PANC 41 36 CCNc1nc(C)c(C(=O)NCc2cc(O)nc(SC)n2)s1 ZINC000880652572 EE On-Demand Anodyne SCD1 26 43 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC(F)(F)CC3)cn2)cc1 ZINC000880652577 FG On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](C4CC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880652578 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](C4CC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880652578 FG On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](C4CC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880652579 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](C4CC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880652579 FG On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](C4CC4)[C@H]3C3CC3)cn2)cc1 ZINC000880652580 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](C4CC4)[C@H]3C3CC3)cn2)cc1 ZINC000880652580 FG On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](C4CC4)[C@H]3C3CC3)cn2)cc1 ZINC000880652581 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](C4CC4)[C@H]3C3CC3)cn2)cc1 ZINC000880652581 FG On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC34CCCC4)cn2)cc1 ZINC000880652582 EG On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(COC4)C3)cn2)cc1 ZINC000880652586 EE On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(COC4)C3)cn2)cc1 ZINC000880652586 EE On-Demand Mild PANC 41 36 CN(C[C@H]1CCCN1C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652587 FE On-Demand Mild ITK 31 48 CN(C[C@H]1CCCN1C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652587 FE On-Demand Mild PANC 58 40 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652588 FE On-Demand Mild ITK 31 48 CN(C[C@@H]1CCCN1C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652588 FE On-Demand Mild PANC 58 40 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC(O)C1 ZINC000880652590 ED On-Demand Mild ITK 18 50 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC(O)C1 ZINC000880652590 ED On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CC(F)(F)F)CC3)cn2)cc1 ZINC000880652593 GH On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CC(F)(F)F)CC3)cn2)cc1 ZINC000880652593 GH On-Demand Mild PANC 54 38 CC[C@H](C)N(CCO)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652596 EE On-Demand Mild ITK 16 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CC(C)(C)O ZINC000880652598 GE On-Demand Mild PANC 54 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CC(C)(C)O ZINC000880652599 GE On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CO)C3)cn2)cc1 ZINC000880652600 DD On-Demand Mild ITK 17 53 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CO)C3)cn2)cc1 ZINC000880652600 DD On-Demand Mild PANC 53 36 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652601 GF On-Demand Mild ITK 15 44 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652602 GF On-Demand Mild ITK 15 44 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO[C@H]1C1CC1 ZINC000880652604 FF On-Demand Mild ITK 16 45 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO[C@H]1C1CC1 ZINC000880652604 FF On-Demand Mild PANC 54 36 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO[C@@H]1C1CC1 ZINC000880652605 FF On-Demand Mild ITK 16 45 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO[C@@H]1C1CC1 ZINC000880652605 FF On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CC34CCCC4)cn2)cc1 ZINC000880652608 EG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC34CCCC4)cn2)cc1 ZINC000880652609 EG On-Demand Mild ITK 15 49 COc1cccc(OC)c1C(=O)NCc1cc(O)nc(SC)n1 ZINC000880652616 ED On-Demand Anodyne ALS 81 41 CCCC[C@H](C)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652624 EH On-Demand Mild ITK 18 51 CCCC[C@@H](C)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652625 EH On-Demand Mild ITK 18 51 CCN(CC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652629 EH On-Demand Mild ITK 17 51 CCN(CC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652629 EH On-Demand Mild PANC 54 36 Cn1cc([C@@H]2CCCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)cn1 ZINC000880652632 GF On-Demand Mild ITK 19 47 Cn1cc([C@@H]2CCCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)cn1 ZINC000880652632 GF On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)NC34CCC(CC3)C4)cn2)cc1 ZINC000880652634 EG On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)NC34CCC(CC3)C4)cn2)cc1 ZINC000880652634 EG On-Demand Mild EPHX2 35 45 N#Cc1ccc(Cn2cc(NC(=O)NC34CCC(CC3)C4)cn2)cc1 ZINC000880652634 EG On-Demand Mild PANC 53 35 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652636 GH On-Demand Mild DPP4 15 42 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652636 GH On-Demand Mild ITK 16 46 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652636 GH On-Demand Mild PANC 55 38 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652638 GH On-Demand Mild DPP4 15 42 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652638 GH On-Demand Mild ITK 16 46 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652638 GH On-Demand Mild PANC 55 38 COCC[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652657 FE On-Demand Mild ITK 18 45 COCC[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652657 FE On-Demand Mild PANC 55 38 COCC[C@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652658 FE On-Demand Mild ITK 18 45 COCC[C@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652658 FE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C(=O)C4CC4)CC3)cn2)cc1 ZINC000880652659 GE On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C(=O)C4CC4)CC3)cn2)cc1 ZINC000880652659 GE On-Demand Mild PANC 53 37 CCC[C@]1(CO)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652663 FF On-Demand Mild ITK 15 46 CN1CC=C(CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652665 FE On-Demand Mild ITK 17 49 CN1CC=C(CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652665 FE On-Demand Mild PANC 53 37 CN(C[C@H]1CC=CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652671 EH On-Demand Mild ITK 18 47 CN(C[C@H]1CC=CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652671 EH On-Demand Mild PANC 56 39 CN(C[C@@H]1CC=CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652672 EH On-Demand Mild ITK 18 47 CN(C[C@@H]1CC=CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652672 EH On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CCC4)CCC3)cn2)cc1 ZINC000880652675 EH On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CCC4)CCC3)cn2)cc1 ZINC000880652675 EH On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C#N)C3)cn2)cc1 ZINC000880652676 DD On-Demand Mild ITK 16 53 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C#N)C3)cn2)cc1 ZINC000880652676 DD On-Demand Mild PANC 53 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)N1CCO ZINC000880652677 GD On-Demand Mild ITK 19 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)N1CCO ZINC000880652677 GD On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C[C@H]3CO)cn2)cc1 ZINC000880652679 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C[C@H]3CO)cn2)cc1 ZINC000880652679 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCCC4=O)CC3)cn2)cc1 ZINC000880652681 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C[C@@H]3CO)cn2)cc1 ZINC000880652682 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C[C@@H]3CO)cn2)cc1 ZINC000880652682 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCC4(CCOCC4)C3)cn2)cc1 ZINC000880652683 GE On-Demand Mild ITK 15 45 Cc1csc([C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)n1 ZINC000880652688 GH On-Demand Mild ITK 20 44 Cc1csc([C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C2)n1 ZINC000880652688 GH On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C3CC3)cn2)cc1 ZINC000880652690 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C3CC3)cn2)cc1 ZINC000880652690 DF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C3CC3)cn2)cc1 ZINC000880652691 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C3CC3)cn2)cc1 ZINC000880652691 DF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](CC(F)(F)F)C3)cn2)cc1 ZINC000880652692 GF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](CC(F)(F)F)C3)cn2)cc1 ZINC000880652693 GF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@H]4C3)cn2)cc1 ZINC000880652694 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@H]4C3)cn2)cc1 ZINC000880652694 DF On-Demand Mild MLNR 20 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@H]4C3)cn2)cc1 ZINC000880652694 DF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@H]4C3)cn2)cc1 ZINC000880652695 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@H]4C3)cn2)cc1 ZINC000880652695 DF On-Demand Mild MLNR 20 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@H]4C3)cn2)cc1 ZINC000880652695 DF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652696 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652696 DF On-Demand Mild MLNR 20 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652696 DF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652697 DF On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652697 DF On-Demand Mild MLNR 20 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4C[C@@H]4C3)cn2)cc1 ZINC000880652697 DF On-Demand Mild PANC 54 38 C=CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H](C)COC ZINC000880652702 FF On-Demand Mild ITK 17 46 C=CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H](C)COC ZINC000880652703 FF On-Demand Mild ITK 17 46 CC1(C)CC[C@@H](CC(=O)NC[C@H]2CCc3cccnc32)OC1 ZINC000880652704 DF On-Demand Anodyne G2YM83_BOTF4 44 32 CC1(C)CC[C@@H](CC(=O)NC[C@@H]2CCc3cccnc32)OC1 ZINC000880652705 DF On-Demand Anodyne G2YM83_BOTF4 44 32 O=C(CC[C@H]1CCc2ccccc21)NC[C@@H]1CCc2cccnc21 ZINC000880652708 DH On-Demand Anodyne MTNR1A 20 47 O=C(CC[C@H]1CCc2ccccc21)NC[C@@H]1CCc2cccnc21 ZINC000880652708 DH On-Demand Anodyne MTNR1B 23 47 O=C(CC[C@@H]1CCc2ccccc21)NC[C@H]1CCc2cccnc21 ZINC000880652709 DH On-Demand Anodyne MTNR1A 20 47 O=C(CC[C@@H]1CCc2ccccc21)NC[C@H]1CCc2cccnc21 ZINC000880652709 DH On-Demand Anodyne MTNR1B 23 47 O=C(CC[C@H]1CCc2ccccc21)NC[C@H]1CCc2cccnc21 ZINC000880652710 DH On-Demand Anodyne MTNR1A 20 47 O=C(CC[C@H]1CCc2ccccc21)NC[C@H]1CCc2cccnc21 ZINC000880652710 DH On-Demand Anodyne MTNR1B 23 47 O=C(CC[C@@H]1CCc2ccccc21)NC[C@@H]1CCc2cccnc21 ZINC000880652711 DH On-Demand Anodyne MTNR1A 20 47 O=C(CC[C@@H]1CCc2ccccc21)NC[C@@H]1CCc2cccnc21 ZINC000880652711 DH On-Demand Anodyne MTNR1B 23 47 COCCCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652712 EF On-Demand Mild ITK 24 51 COCCCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652712 EF On-Demand Mild PANC 55 38 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652713 ED On-Demand Mild ITK 19 47 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652713 ED On-Demand Mild PANC 58 40 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652714 ED On-Demand Mild ITK 19 47 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880652714 ED On-Demand Mild PANC 58 40 N#Cc1ccc(Cn2cc(NC(=O)NN3CCCCC3)cn2)cc1 ZINC000880652715 DE On-Demand Mild ITK 18 53 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880652717 EH On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880652717 EH On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(O)C[C@H]4C3)cn2)cc1 ZINC000880652719 ED On-Demand Mild ITK 15 48 C[C@@H]1CC[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652722 EE On-Demand Mild ITK 19 49 C[C@@H]1CC[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652722 EE On-Demand Mild PANC 60 40 C[C@H]1CC[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652723 EE On-Demand Mild ITK 19 49 C[C@H]1CC[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652723 EE On-Demand Mild PANC 60 40 C[C@H]1CC[C@@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652724 EE On-Demand Mild ITK 19 49 C[C@H]1CC[C@@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652724 EE On-Demand Mild PANC 60 40 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652728 EE On-Demand Mild ITK 18 49 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652728 EE On-Demand Mild PANC 49 37 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652729 EE On-Demand Mild ITK 18 49 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652729 EE On-Demand Mild PANC 49 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)C1(F)F ZINC000880652734 FH On-Demand Mild ITK 16 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)C1(F)F ZINC000880652734 FH On-Demand Mild PANC 53 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1(F)F ZINC000880652735 FH On-Demand Mild ITK 16 49 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1(F)F ZINC000880652735 FH On-Demand Mild PANC 53 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1(F)F ZINC000880652736 FH On-Demand Mild ITK 16 49 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1(F)F ZINC000880652736 FH On-Demand Mild PANC 53 37 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652738 FE On-Demand Mild ITK 17 47 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652738 FE On-Demand Mild PANC 53 37 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652740 FE On-Demand Mild ITK 17 47 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652740 FE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4COC[C@@H]43)cn2)cc1 ZINC000880652743 FE On-Demand Mild PANC 53 37 C[C@H]1CC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652746 EG On-Demand Mild ITK 15 49 C[C@H]1CC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652746 EG On-Demand Mild PANC 49 35 C[C@@H]1CC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652747 EG On-Demand Mild ITK 15 49 C[C@@H]1CC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652747 EG On-Demand Mild PANC 49 35 N#Cc1ccc(Cn2cc(NC(=O)N(C3CC3)C3CC3)cn2)cc1 ZINC000880652748 DF On-Demand Mild ITK 20 54 N#Cc1ccc(Cn2cc(NC(=O)N(C3CC3)C3CC3)cn2)cc1 ZINC000880652748 DF On-Demand Mild PANC 57 38 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H](CO)CC(C)(C)C ZINC000880652751 FG On-Demand Mild ITK 17 48 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H](CO)CC(C)(C)C ZINC000880652751 FG On-Demand Mild PANC 41 35 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H](CO)CC(C)(C)C ZINC000880652752 FG On-Demand Mild ITK 17 48 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H](CO)CC(C)(C)C ZINC000880652752 FG On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C(F)(F)C3)cn2)cc1 ZINC000880652756 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](O)C(F)(F)C3)cn2)cc1 ZINC000880652756 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C(F)(F)C3)cn2)cc1 ZINC000880652757 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)C(F)(F)C3)cn2)cc1 ZINC000880652757 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)[S@@]4=O)cn2)cc1 ZINC000880652758 GE On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)[S@@]4=O)cn2)cc1 ZINC000880652758 GE On-Demand Mild PANC 42 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)[S@]4=O)cn2)cc1 ZINC000880652759 GE On-Demand Mild ITK 18 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)[S@]4=O)cn2)cc1 ZINC000880652759 GE On-Demand Mild PANC 42 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@@H](C4)C3)cn2)cc1 ZINC000880652760 EG On-Demand Mild ITK 17 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@@H](C4)C3)cn2)cc1 ZINC000880652760 EG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC3(C4)CC3(F)F)cn2)cc1 ZINC000880652761 GH On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC3(C4)CC3(F)F)cn2)cc1 ZINC000880652761 GH On-Demand Mild PANC 41 36 CC[C@@H]1COC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652762 FG On-Demand Mild ITK 15 46 CC[C@@H]1COC(C)(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652762 FG On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC[C@H](O)C4)CC3)cn2)cc1 ZINC000880652764 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC[C@H](O)C4)CC3)cn2)cc1 ZINC000880652764 GD On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC[C@@H](O)C4)CC3)cn2)cc1 ZINC000880652765 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(N4CC[C@@H](O)C4)CC3)cn2)cc1 ZINC000880652765 GD On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@H]3C(F)(F)F)cn2)cc1 ZINC000880652767 EF On-Demand Mild ITK 15 50 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@H]3C(F)(F)F)cn2)cc1 ZINC000880652767 EF On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(CCO)C4)cn2)cc1 ZINC000880652768 GF On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(CCO)C4)cn2)cc1 ZINC000880652768 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCCN3)cn2)cc1 ZINC000880652769 ED On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCCN3)cn2)cc1 ZINC000880652769 ED On-Demand Mild PANC 41 36 CCCOc1ccc(OCC(=O)NCc2cc(O)nc(SC)n2)cc1 ZINC000880652770 FE On-Demand Anodyne MTNR1A 21 40 CCCOc1ccc(OCC(=O)NCc2cc(O)nc(SC)n2)cc1 ZINC000880652770 FE On-Demand Anodyne PLA2G4B 68 32 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652772 EH On-Demand Mild ITK 16 50 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652772 EH On-Demand Mild PANC 56 39 C[C@H](O)CN(CC(F)F)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652778 FE On-Demand Mild ITK 15 49 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652782 FE On-Demand Mild ITK 16 47 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652782 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3[C@@H](CO)C4)cn2)cc1 ZINC000880652792 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3[C@@H](CO)C4)cn2)cc1 ZINC000880652792 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3[C@H](CO)C4)cn2)cc1 ZINC000880652793 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3[C@H](CO)C4)cn2)cc1 ZINC000880652793 FE On-Demand Mild PANC 41 35 CN(CC1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652797 FF On-Demand Mild ITK 25 48 CN(CC1CCOCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652797 FF On-Demand Mild PANC 59 41 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CCO ZINC000880652799 FD On-Demand Mild ITK 19 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1CCO ZINC000880652800 FD On-Demand Mild ITK 19 47 CO[C@@H]1[C@@H]2C[C@@H]3[C@@H]1N(C(=O)Nc1cnn(Cc4ccc(C#N)cc4)c1)C[C@@H]3C2 ZINC000880652806 GF On-Demand Mild ITK 15 45 CO[C@@H]1[C@@H]2C[C@@H]3[C@@H]1N(C(=O)Nc1cnn(Cc4ccc(C#N)cc4)c1)C[C@@H]3C2 ZINC000880652806 GF On-Demand Mild PANC 44 35 CO[C@@H]1[C@@H]2C[C@H]3[C@@H](C2)CN(C(=O)Nc2cnn(Cc4ccc(C#N)cc4)c2)[C@H]31 ZINC000880652807 GF On-Demand Mild ITK 15 45 CO[C@@H]1[C@@H]2C[C@H]3[C@@H](C2)CN(C(=O)Nc2cnn(Cc4ccc(C#N)cc4)c2)[C@H]31 ZINC000880652807 GF On-Demand Mild PANC 44 35 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnn(Cc5ccc(C#N)cc5)c4)[C@H]1[C@H]3C2 ZINC000880652808 GF On-Demand Mild ITK 15 45 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnn(Cc5ccc(C#N)cc5)c4)[C@H]1[C@H]3C2 ZINC000880652808 GF On-Demand Mild PANC 44 35 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnn(Cc5ccc(C#N)cc5)c4)[C@@H]1[C@H]3C2 ZINC000880652809 GF On-Demand Mild ITK 15 45 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnn(Cc5ccc(C#N)cc5)c4)[C@@H]1[C@H]3C2 ZINC000880652809 GF On-Demand Mild PANC 44 35 CN1CCC(C)(CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652811 FF On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCOCC4)C3)cn2)cc1 ZINC000880652812 GD On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCOCC4)C3)cn2)cc1 ZINC000880652812 GD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCOCC4)C3)cn2)cc1 ZINC000880652813 GD On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCOCC4)C3)cn2)cc1 ZINC000880652813 GD On-Demand Mild PANC 41 36 CN1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652817 ED On-Demand Mild CCR3 55 46 CN1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652817 ED On-Demand Mild ITK 18 51 CN1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652817 ED On-Demand Mild PANC 55 38 CN1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652818 ED On-Demand Mild CCR3 55 46 CN1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652818 ED On-Demand Mild ITK 18 51 CN1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652818 ED On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@](F)(CO)C3)cn2)cc1 ZINC000880652819 ED On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@](F)(CO)C3)cn2)cc1 ZINC000880652820 ED On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCOC4(CCOCC4)CC3)cn2)cc1 ZINC000880652821 GF On-Demand Mild ITK 15 46 CCC1(CC)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652822 EG On-Demand Mild ITK 17 52 CCC1(CC)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652822 EG On-Demand Mild PANC 49 36 C[C@H]1CCSCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652823 FG On-Demand Mild ITK 15 47 C[C@H]1CCSCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652823 FG On-Demand Mild PANC 53 37 C[C@@H]1CCSCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652824 FG On-Demand Mild ITK 15 47 C[C@@H]1CCSCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652824 FG On-Demand Mild PANC 53 37 CN(C)C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652832 FE On-Demand Mild ITK 20 48 CN(C)C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652832 FE On-Demand Mild MLNR 34 40 CN(C)C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652832 FE On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCO3)cn2)cc1 ZINC000880652834 DE On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCO3)cn2)cc1 ZINC000880652834 DE On-Demand Mild PANC 54 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C2CC2)O1 ZINC000880652835 FF On-Demand Mild ITK 16 46 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C2CC2)O1 ZINC000880652835 FF On-Demand Mild PANC 55 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C2CC2)O1 ZINC000880652836 FF On-Demand Mild ITK 16 46 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C2CC2)O1 ZINC000880652836 FF On-Demand Mild PANC 55 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C2CC2)O1 ZINC000880652837 FF On-Demand Mild ITK 16 46 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C2CC2)O1 ZINC000880652837 FF On-Demand Mild PANC 55 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C2CC2)O1 ZINC000880652838 FF On-Demand Mild ITK 16 46 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C2CC2)O1 ZINC000880652838 FF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC34CCOCC4)cn2)cc1 ZINC000880652843 FF On-Demand Mild ITK 15 49 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652844 GG On-Demand Mild ITK 24 44 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652844 GG On-Demand Mild PANC 58 40 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652845 GG On-Demand Mild ITK 24 44 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652845 GG On-Demand Mild PANC 58 40 C[C@@H]1CSCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652846 FG On-Demand Mild ITK 15 48 C[C@@H]1CSCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652846 FG On-Demand Mild PANC 41 36 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1OC ZINC000880652854 FD On-Demand Mild ITK 20 53 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1OC ZINC000880652854 FD On-Demand Mild PANC 57 39 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CC[C@@H](O)CC1 ZINC000880652855 FF On-Demand Mild ITK 27 49 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CC[C@@H](O)CC1 ZINC000880652855 FF On-Demand Mild PANC 55 37 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC=CCC1 ZINC000880652858 EG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CF)C3)cn2)cc1 ZINC000880652860 EG On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CF)C3)cn2)cc1 ZINC000880652860 EG On-Demand Mild PANC 41 36 COC[C@@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652861 FG On-Demand Mild PDGFRB 18 42 COC[C@@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652861 FG On-Demand Mild ITK 23 47 COC[C@@H]1CCCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652861 FG On-Demand Mild PANC 55 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CF)C3)cn2)cc1 ZINC000880652862 EG On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CF)C3)cn2)cc1 ZINC000880652862 EG On-Demand Mild PANC 41 36 CN(CCC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652866 EH On-Demand Mild ITK 19 51 CN(CCC(C)(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652866 EH On-Demand Mild PANC 56 38 C=CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652867 DF On-Demand Mild ITK 19 51 C=CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652867 DF On-Demand Mild PANC 54 36 CC[C@H](C)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880652868 FF On-Demand Mild ITK 16 49 C[C@H](O)CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652877 EE On-Demand Mild ITK 23 49 C[C@H](O)CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652877 EE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C(=O)N4CCCC4)C3)cn2)cc1 ZINC000880652878 GE On-Demand Mild ITK 22 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C(=O)N4CCCC4)C3)cn2)cc1 ZINC000880652878 GE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@](O)(C(F)F)C3)cn2)cc1 ZINC000880652880 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C(=O)N4CCCC4)C3)cn2)cc1 ZINC000880652881 GE On-Demand Mild ITK 22 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C(=O)N4CCCC4)C3)cn2)cc1 ZINC000880652881 GE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@](O)(C(F)F)C3)cn2)cc1 ZINC000880652882 FE On-Demand Mild ITK 15 47 Cc1c(CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)cnn1C ZINC000880652884 FF On-Demand Mild ITK 17 48 Cc1c(CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)cnn1C ZINC000880652884 FF On-Demand Mild PANC 43 33 COC[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652886 FF On-Demand Mild ITK 27 47 COC[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652886 FF On-Demand Mild PANC 55 39 Cn1cnc2c1CCN(C(=O)Nc1cnn(Cc3ccc(C#N)cc3)c1)C2 ZINC000880652887 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CCO)cn2)cc1 ZINC000880652889 EE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]3CCO)cn2)cc1 ZINC000880652889 EE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CCO)cn2)cc1 ZINC000880652890 EE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3CCO)cn2)cc1 ZINC000880652890 EE On-Demand Mild PANC 41 36 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652907 GF On-Demand Mild ITK 17 45 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652907 GF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCF)CC3)cn2)cc1 ZINC000880652908 FG On-Demand Mild CCR3 17 41 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCF)CC3)cn2)cc1 ZINC000880652908 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCF)CC3)cn2)cc1 ZINC000880652908 FG On-Demand Mild PANC 56 39 Cn1nccc1[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652910 GF On-Demand Mild ITK 17 45 Cn1nccc1[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652910 GF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CCC4)CC3)cn2)cc1 ZINC000880652912 EG On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)NC3(C4CCC4)CC3)cn2)cc1 ZINC000880652912 EG On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)NNCC(F)(F)C(F)(F)F)cn2)cc1 ZINC000880652914 GF On-Demand Reactive ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)NNCC(F)(F)C(F)(F)F)cn2)cc1 ZINC000880652914 GF On-Demand Reactive PANC 40 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H](C)O1 ZINC000880652917 FF On-Demand Mild ITK 16 48 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H](C)O1 ZINC000880652917 FF On-Demand Mild MLNR 37 42 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H](C)O1 ZINC000880652917 FF On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCOC4)CC3)cn2)cc1 ZINC000880652923 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCOC4)CC3)cn2)cc1 ZINC000880652923 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880652925 GG On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880652925 GG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCN(C=O)CC3)cn2)cc1 ZINC000880652926 FD On-Demand Mild ITK 15 51 C#C[C@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652929 ED On-Demand Mild ITK 15 47 C#C[C@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652929 ED On-Demand Mild PANC 53 37 C#C[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652930 ED On-Demand Mild ITK 15 47 C#C[C@@H]1COCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652930 ED On-Demand Mild PANC 53 37 CC[C@@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652931 FE On-Demand Mild ITK 17 47 CC[C@@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652931 FE On-Demand Mild PANC 41 36 CC[C@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652933 FE On-Demand Mild ITK 17 47 CC[C@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652933 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880652934 EG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880652934 EG On-Demand Mild MLNR 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](C4CCC4)C3)cn2)cc1 ZINC000880652934 EG On-Demand Mild PANC 53 38 COC1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652935 EE On-Demand Mild ITK 19 51 COC1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880652935 EE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CCC4)C3)cn2)cc1 ZINC000880652936 EG On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CCC4)C3)cn2)cc1 ZINC000880652936 EG On-Demand Mild MLNR 19 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](C4CCC4)C3)cn2)cc1 ZINC000880652936 EG On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)C3)cn2)cc1 ZINC000880652937 FE On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)C3)cn2)cc1 ZINC000880652937 FE On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CC4)C3)cn2)cc1 ZINC000880652941 DE On-Demand Mild ITK 17 54 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CC4)C3)cn2)cc1 ZINC000880652941 DE On-Demand Mild PANC 41 35 C[C@H]1C(=O)N(CCN(C)C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652942 GD On-Demand Mild ITK 18 47 C[C@H]1C(=O)N(CCN(C)C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880652942 GD On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](F)C3)cn2)cc1 ZINC000880652945 EF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](F)C3)cn2)cc1 ZINC000880652945 EF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](F)C3)cn2)cc1 ZINC000880652946 EF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](F)C3)cn2)cc1 ZINC000880652946 EF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@H]4CCOC4)CC3)cn2)cc1 ZINC000880652949 GD On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCN([C@@H]4CCOC4)CC3)cn2)cc1 ZINC000880652950 GD On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@H]3C3CCC3)cn2)cc1 ZINC000880652953 EG On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@H]3C3CCC3)cn2)cc1 ZINC000880652953 EG On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3[C@@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880652954 GG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3[C@H]3CCC[C@H]3O)cn2)cc1 ZINC000880652955 GG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3[C@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880652956 GG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC[C@@H]3[C@@H]3CCC[C@H]3O)cn2)cc1 ZINC000880652957 GG On-Demand Mild ITK 17 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C(F)(F)C3)cn2)cc1 ZINC000880652966 FF On-Demand Mild ITK 20 54 N#Cc1ccc(Cn2cc(NC(=O)N3CC(F)(F)C(F)(F)C3)cn2)cc1 ZINC000880652966 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652967 GH On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652967 GH On-Demand Mild MLNR 22 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652967 GH On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652968 GH On-Demand Mild ITK 18 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652968 GH On-Demand Mild MLNR 22 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](OC4CCC4)CC3)cn2)cc1 ZINC000880652968 GH On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C[C@H]4c4ccccc4)C3)cn2)cc1 ZINC000880652970 GI On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C[C@H]4c4ccccc4)C3)cn2)cc1 ZINC000880652970 GI On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CCCO)C3)cn2)cc1 ZINC000880652971 FE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CCCO)C3)cn2)cc1 ZINC000880652971 FE On-Demand Mild PANC 41 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CCCO)C3)cn2)cc1 ZINC000880652972 FE On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CCCO)C3)cn2)cc1 ZINC000880652972 FE On-Demand Mild PANC 41 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652973 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652973 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652974 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652974 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@@H](O)CC[C@H]4C3)cn2)cc1 ZINC000880652975 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@@H](O)CC[C@H]4C3)cn2)cc1 ZINC000880652975 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@H](O)CC[C@H]4C3)cn2)cc1 ZINC000880652976 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@H](O)CC[C@H]4C3)cn2)cc1 ZINC000880652976 FE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652977 FE On-Demand Mild ITK 16 48 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC[C@@H](O)C[C@H]4C3)cn2)cc1 ZINC000880652977 FE On-Demand Mild PANC 41 35 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)CN1CCO ZINC000880652979 GD On-Demand Mild ITK 18 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)CN1CCO ZINC000880652979 GD On-Demand Mild PANC 53 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CN1CCO ZINC000880652980 GD On-Demand Mild ITK 18 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CN1CCO ZINC000880652980 GD On-Demand Mild PANC 53 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CN1CCO ZINC000880652981 GD On-Demand Mild ITK 18 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CN1CCO ZINC000880652981 GD On-Demand Mild PANC 53 36 C#CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652982 DE On-Demand Mild ITK 19 50 C#CCN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC1 ZINC000880652982 DE On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC(Cc4ccco4)C3)cn2)cc1 ZINC000880653060 FG On-Demand Mild PANC 44 34 CN1C[C@@H]2CCCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)[C@@H]2C1 ZINC000880653064 FE On-Demand Mild ITK 20 46 CN1C[C@@H]2CCCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)[C@@H]2C1 ZINC000880653064 FE On-Demand Mild PANC 49 36 CC[C@@H]1CN(CC)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653070 FF On-Demand Mild ITK 15 49 CC[C@@H]1CN(CC)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653070 FF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCC4=O)C3)cn2)cc1 ZINC000880653073 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCC4=O)C3)cn2)cc1 ZINC000880653075 GE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCCCO4)CC3)cn2)cc1 ZINC000880653078 GH On-Demand Mild ITK 25 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCCCO4)CC3)cn2)cc1 ZINC000880653078 GH On-Demand Mild PANC 55 38 C[C@@H]1O[C@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880653079 FF On-Demand Mild ITK 15 48 C[C@@H]1O[C@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H]1C ZINC000880653079 FF On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCCCO4)CC3)cn2)cc1 ZINC000880653080 GH On-Demand Mild ITK 25 46 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCCCO4)CC3)cn2)cc1 ZINC000880653080 GH On-Demand Mild PANC 55 38 C[C@@H]1O[C@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880653081 FF On-Demand Mild ITK 15 48 C[C@@H]1O[C@H](C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H]1C ZINC000880653081 FF On-Demand Mild PANC 54 36 C[C@]1(C(F)(F)F)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880653084 GF On-Demand Mild ITK 15 45 C[C@]1(C(F)(F)F)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880653084 GF On-Demand Mild EPHX2 15 44 C[C@]1(C(F)(F)F)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880653084 GF On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@@H](C)O1 ZINC000880653085 FF On-Demand Mild ITK 15 48 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@@H](C)O1 ZINC000880653085 FF On-Demand Mild PANC 54 36 CCO[C@@]1(C)C[C@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653086 EE On-Demand Mild ITK 17 47 CCO[C@@]1(C)C[C@H]1NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653086 EE On-Demand Mild PANC 53 35 CCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653087 EE On-Demand Mild ITK 17 49 CCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653087 EE On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H](C3)C4(F)F)cn2)cc1 ZINC000880653088 EF On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@H](C3)C4(F)F)cn2)cc1 ZINC000880653088 EF On-Demand Mild PANC 42 37 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H](C3)C4(F)F)cn2)cc1 ZINC000880653090 EF On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4[C@H](C3)C4(F)F)cn2)cc1 ZINC000880653090 EF On-Demand Mild PANC 42 37 N#CCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653091 EF On-Demand Mild ITK 17 50 N#CCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653091 EF On-Demand Mild MLNR 22 42 N#CCC1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653091 EF On-Demand Mild PANC 53 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880653092 EE On-Demand Mild ITK 18 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880653092 EE On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C3)C4(F)F)cn2)cc1 ZINC000880653093 EF On-Demand Mild ITK 16 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](C3)C4(F)F)cn2)cc1 ZINC000880653093 EF On-Demand Mild PANC 42 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880653094 EE On-Demand Mild ITK 18 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1=O ZINC000880653094 EE On-Demand Mild PANC 55 38 Cc1cncc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)c1 ZINC000880653095 GH On-Demand Mild ITK 17 45 Cc1cncc([C@@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)c1 ZINC000880653095 GH On-Demand Mild PANC 56 39 Cc1cncc([C@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)c1 ZINC000880653097 GH On-Demand Mild ITK 17 45 Cc1cncc([C@H]2CCCN2C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)c1 ZINC000880653097 GH On-Demand Mild PANC 56 39 CN(C)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653098 FF On-Demand Mild ITK 25 47 CN(C)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653098 FF On-Demand Mild MLNR 30 40 CN(C)[C@@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653098 FF On-Demand Mild PANC 53 37 COCC(C)(C)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653101 GE On-Demand Mild PDGFRB 15 42 COCC(C)(C)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653101 GE On-Demand Mild ITK 17 47 COCC(C)(C)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653101 GE On-Demand Mild PANC 56 39 C[C@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653107 GH On-Demand Mild ITK 15 46 C[C@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653107 GH On-Demand Mild PANC 58 40 C[C@@H]1CC2(CCC2)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653108 EH On-Demand Mild ITK 15 47 C[C@@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653109 GH On-Demand Mild ITK 15 46 C[C@@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653109 GH On-Demand Mild PANC 58 40 COC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653110 FF On-Demand Mild ITK 19 49 COC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653110 FF On-Demand Mild PANC 49 37 C[C@H]1[C@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653114 FE On-Demand Mild ITK 20 51 C[C@H]1[C@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653114 FE On-Demand Mild PANC 56 39 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653115 FE On-Demand Mild ITK 20 51 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653115 FE On-Demand Mild PANC 56 39 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880653116 EG On-Demand Mild ITK 18 49 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C1 ZINC000880653116 EG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cccn4)C3)cn2)cc1 ZINC000880653119 FE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cccn4)C3)cn2)cc1 ZINC000880653119 FE On-Demand Mild MLNR 25 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cccn4)C3)cn2)cc1 ZINC000880653119 FE On-Demand Mild PANC 52 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cccn4)C3)cn2)cc1 ZINC000880653121 FE On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cccn4)C3)cn2)cc1 ZINC000880653121 FE On-Demand Mild MLNR 25 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cccn4)C3)cn2)cc1 ZINC000880653121 FE On-Demand Mild PANC 52 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1=O ZINC000880653122 FE On-Demand Mild ITK 17 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1=O ZINC000880653122 FE On-Demand Mild PANC 54 36 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC(C)(C)C1 ZINC000880653124 EG On-Demand Mild ITK 24 51 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CC(C)(C)C1 ZINC000880653124 EG On-Demand Mild PANC 54 36 CC(C)[C@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653125 FF On-Demand Mild ITK 17 47 CC(C)[C@H]1CN(C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653125 FF On-Demand Mild PANC 41 36 C#CCCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653126 FE On-Demand Mild ITK 19 49 CN1CCO[C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@H]21 ZINC000880653127 GD On-Demand Mild ITK 25 47 CN1CCO[C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@H]21 ZINC000880653127 GD On-Demand Mild PANC 56 39 CN1CCO[C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653128 GD On-Demand Mild ITK 25 47 CN1CCO[C@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653128 GD On-Demand Mild PANC 56 39 CN1CCO[C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653129 GD On-Demand Mild ITK 25 47 CN1CCO[C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653129 GD On-Demand Mild PANC 56 39 CN1CCO[C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@H]21 ZINC000880653131 GD On-Demand Mild ITK 25 47 CN1CCO[C@@H]2CCN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@H]21 ZINC000880653131 GD On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CSC[C@H]4C3)cn2)cc1 ZINC000880653133 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CSC[C@H]4C3)cn2)cc1 ZINC000880653133 FG On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CSC[C@H]4C3)cn2)cc1 ZINC000880653135 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CSC[C@H]4C3)cn2)cc1 ZINC000880653135 FG On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CSC[C@@H]4C3)cn2)cc1 ZINC000880653138 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CSC[C@@H]4C3)cn2)cc1 ZINC000880653138 FG On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CSC[C@@H]4C3)cn2)cc1 ZINC000880653140 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]4CSC[C@@H]4C3)cn2)cc1 ZINC000880653140 FG On-Demand Mild PANC 49 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCC4)CC3)cn2)cc1 ZINC000880653141 EH On-Demand Mild ITK 17 53 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCC4)CC3)cn2)cc1 ZINC000880653141 EH On-Demand Mild PANC 41 36 CC[C@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653145 EG On-Demand Mild ITK 16 48 CC[C@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653145 EG On-Demand Mild PANC 54 38 CC[C@H]1[C@@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653147 EG On-Demand Mild ITK 16 48 CC[C@H]1[C@@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653147 EG On-Demand Mild PANC 54 38 CC[C@@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653149 EG On-Demand Mild ITK 16 48 CC[C@@H]1[C@H](C)CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653149 EG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCO3)cn2)cc1 ZINC000880653151 EF On-Demand Mild ITK 17 50 N#Cc1ccc(Cn2cc(NC(=O)N3CCCCCO3)cn2)cc1 ZINC000880653151 EF On-Demand Mild PANC 53 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880653155 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880653155 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCC[C@H]3O)cn2)cc1 ZINC000880653157 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@H]3CCC[C@H]3O)cn2)cc1 ZINC000880653157 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCC[C@H]3O)cn2)cc1 ZINC000880653159 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCC[C@H]3O)cn2)cc1 ZINC000880653159 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880653161 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]3[C@@H]3CCC[C@@H]3O)cn2)cc1 ZINC000880653161 GF On-Demand Mild PANC 41 36 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653163 GH On-Demand Mild ITK 15 47 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653163 GH On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CC34CC4)cn2)cc1 ZINC000880653167 DE On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CC34CC4)cn2)cc1 ZINC000880653167 DE On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC34CC4)cn2)cc1 ZINC000880653170 DE On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CC34CC4)cn2)cc1 ZINC000880653170 DE On-Demand Mild PANC 41 35 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653178 GD On-Demand Mild CCR3 46 38 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653178 GD On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@]4(CCCO4)[C@H]3C3CC3)cn2)cc1 ZINC000880653194 GF On-Demand Mild ITK 17 44 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@]4(CCCO4)[C@@H]3C3CC3)cn2)cc1 ZINC000880653196 GF On-Demand Mild ITK 17 44 COCCO[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653197 FE On-Demand Mild ITK 22 50 COCCO[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653197 FE On-Demand Mild MLNR 32 42 COCCO[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653197 FE On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]4(CCCO4)[C@@H]3C3CC3)cn2)cc1 ZINC000880653198 GF On-Demand Mild ITK 17 44 COCCO[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653199 FE On-Demand Mild ITK 22 50 COCCO[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653199 FE On-Demand Mild MLNR 32 42 COCCO[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653199 FE On-Demand Mild PANC 57 40 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]4(CCCO4)[C@H]3C3CC3)cn2)cc1 ZINC000880653200 GF On-Demand Mild ITK 17 44 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880653204 FG On-Demand Mild ITK 20 47 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCO1 ZINC000880653204 FG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)NCCN3C[C@@H]4CC[C@H](C3)O4)cn2)cc1 ZINC000880653206 GD On-Demand Mild CCR3 25 45 N#Cc1ccc(Cn2cc(NC(=O)NCCN3C[C@@H]4CC[C@H](C3)O4)cn2)cc1 ZINC000880653206 GD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)NCCN3C[C@@H]4CC[C@H](C3)O4)cn2)cc1 ZINC000880653206 GD On-Demand Mild PANC 56 37 CC1(C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCS1 ZINC000880653208 FH On-Demand Mild ITK 15 47 CN(CC(=O)N1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653210 FD On-Demand Mild ITK 28 49 CN(CC(=O)N1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653210 FD On-Demand Mild PANC 53 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)C1O ZINC000880653212 FE On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H](C)C1O ZINC000880653212 FE On-Demand Mild PANC 54 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)[C@@H]1O ZINC000880653214 FE On-Demand Mild ITK 17 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)[C@@H]1O ZINC000880653214 FE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](N4CCCC4=O)C3)cn2)cc1 ZINC000880653215 GE On-Demand Mild PANC 54 38 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1O ZINC000880653216 FE On-Demand Mild ITK 17 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)C1O ZINC000880653216 FE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](N4CCCC4=O)C3)cn2)cc1 ZINC000880653218 GE On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](CO)[C@@H]4C3)cn2)cc1 ZINC000880653220 ED On-Demand Mild ITK 17 51 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4[C@@H](CO)[C@@H]4C3)cn2)cc1 ZINC000880653220 ED On-Demand Mild PANC 41 35 CCCN(C[C@@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653222 GH On-Demand Mild ITK 28 44 CCCN(C[C@@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653222 GH On-Demand Mild PANC 59 40 CCCN(C[C@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653224 GH On-Demand Mild ITK 28 44 CCCN(C[C@H]1CCCCO1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653224 GH On-Demand Mild PANC 59 40 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653225 FE On-Demand Mild ITK 15 47 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653225 FE On-Demand Mild MLNR 37 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653225 FE On-Demand Mild PANC 54 37 CN(CC1(O)CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653226 EE On-Demand Mild ITK 19 49 CN(CC1(O)CCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653226 EE On-Demand Mild PANC 53 35 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653227 FE On-Demand Mild ITK 15 47 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653227 FE On-Demand Mild MLNR 37 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653227 FE On-Demand Mild PANC 54 37 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653229 FE On-Demand Mild ITK 15 47 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653229 FE On-Demand Mild MLNR 37 42 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1CO ZINC000880653229 FE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@H]43)cn2)cc1 ZINC000880653230 DF On-Demand Mild DPP4 17 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@H]43)cn2)cc1 ZINC000880653230 DF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@H]43)cn2)cc1 ZINC000880653230 DF On-Demand Mild PANC 55 38 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653231 FE On-Demand Mild ITK 15 47 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653231 FE On-Demand Mild MLNR 37 42 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1CO ZINC000880653231 FE On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@H]43)cn2)cc1 ZINC000880653232 DF On-Demand Mild DPP4 17 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@H]43)cn2)cc1 ZINC000880653232 DF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@H]43)cn2)cc1 ZINC000880653232 DF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC4CC4)C3)cn2)cc1 ZINC000880653233 EG On-Demand Mild ITK 18 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC4CC4)C3)cn2)cc1 ZINC000880653233 EG On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@@H]43)cn2)cc1 ZINC000880653234 DF On-Demand Mild DPP4 17 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@@H]43)cn2)cc1 ZINC000880653234 DF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]4C[C@@H]43)cn2)cc1 ZINC000880653234 DF On-Demand Mild PANC 55 38 C=CC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653235 EG On-Demand Mild ITK 15 47 C=CC[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653235 EG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@@H]43)cn2)cc1 ZINC000880653236 DF On-Demand Mild DPP4 17 42 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@@H]43)cn2)cc1 ZINC000880653236 DF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]4C[C@@H]43)cn2)cc1 ZINC000880653236 DF On-Demand Mild PANC 55 38 C=CC[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653237 EG On-Demand Mild ITK 15 47 C=CC[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653237 EG On-Demand Mild PANC 41 36 CN1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1=O ZINC000880653238 DD On-Demand Mild ITK 16 50 CN1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1=O ZINC000880653238 DD On-Demand Mild PANC 44 34 CCC1(N(C)C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653239 GG On-Demand Mild ITK 18 50 CCC1(N(C)C)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653239 GG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(C3)OCc3ccccc34)cn2)cc1 ZINC000880653241 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@]4(C3)OCc3ccccc34)cn2)cc1 ZINC000880653241 GG On-Demand Mild NPY5R 16 40 CN(C)CCCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653242 FG On-Demand Mild ITK 17 51 CN(C)CCCC(C)(C)NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653242 FG On-Demand Mild PANC 48 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(C3)OCc3ccccc34)cn2)cc1 ZINC000880653243 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@]4(C3)OCc3ccccc34)cn2)cc1 ZINC000880653243 GG On-Demand Mild NPY5R 16 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)S4)cn2)cc1 ZINC000880653245 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]4CC[C@@H](C3)S4)cn2)cc1 ZINC000880653245 FG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCC[C@H]3OCC4)cn2)cc1 ZINC000880653247 FF On-Demand Mild ITK 18 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@]34CCC[C@H]3OCC4)cn2)cc1 ZINC000880653247 FF On-Demand Mild PANC 41 35 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653249 EG On-Demand Mild ITK 16 48 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653249 EG On-Demand Mild MLNR 47 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653249 EG On-Demand Mild PANC 55 38 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCc3cccnc32)CC1 ZINC000880653250 ED On-Demand Anodyne MTNR1A 27 42 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCc3cccnc32)CC1 ZINC000880653250 ED On-Demand Anodyne MTNR1B 22 42 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCc3cccnc32)CC1 ZINC000880653251 ED On-Demand Anodyne MTNR1A 27 42 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCc3cccnc32)CC1 ZINC000880653251 ED On-Demand Anodyne MTNR1B 22 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653253 EG On-Demand Mild ITK 16 48 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653253 EG On-Demand Mild MLNR 47 42 C[C@@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653253 EG On-Demand Mild PANC 55 38 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653255 EG On-Demand Mild ITK 16 48 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653255 EG On-Demand Mild MLNR 47 42 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1F ZINC000880653255 EG On-Demand Mild PANC 55 38 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653257 EG On-Demand Mild ITK 16 48 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653257 EG On-Demand Mild MLNR 47 42 C[C@H]1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1F ZINC000880653257 EG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)(F)CC3)cn2)cc1 ZINC000880653258 EG On-Demand Mild ITK 17 52 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(F)(F)CC3)cn2)cc1 ZINC000880653258 EG On-Demand Mild PANC 40 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)[C@H]1C ZINC000880653262 EG On-Demand Mild ITK 19 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)[C@H]1C ZINC000880653262 EG On-Demand Mild PANC 54 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)[C@@H]1C ZINC000880653263 EG On-Demand Mild ITK 19 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](C)[C@@H]1C ZINC000880653263 EG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCCO)CC3)cn2)cc1 ZINC000880653265 FF On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(CCCO)CC3)cn2)cc1 ZINC000880653265 FF On-Demand Mild PANC 55 40 CN(C[C@@H]1CCCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653266 FF On-Demand Mild ITK 31 47 CN(C[C@@H]1CCCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653266 FF On-Demand Mild PANC 56 39 CN(C[C@H]1CCCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653267 FF On-Demand Mild ITK 31 47 CN(C[C@H]1CCCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653267 FF On-Demand Mild PANC 56 39 CN(C[C@H]1CCCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653268 FF On-Demand Mild ITK 31 47 CN(C[C@H]1CCCC[C@@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653268 FF On-Demand Mild PANC 56 39 CN(C[C@@H]1CCCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653269 FF On-Demand Mild ITK 31 47 CN(C[C@@H]1CCCC[C@H]1O)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653269 FF On-Demand Mild PANC 56 39 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1(F)F ZINC000880653275 FG On-Demand Mild ITK 16 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1(F)F ZINC000880653275 FG On-Demand Mild PANC 41 36 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1(F)F ZINC000880653276 FG On-Demand Mild ITK 16 47 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1(F)F ZINC000880653276 FG On-Demand Mild PANC 41 36 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653280 FF On-Demand Mild ITK 20 49 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653280 FF On-Demand Mild MLNR 27 41 CO[C@H]1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653280 FF On-Demand Mild PANC 55 39 COCCCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653283 FE On-Demand Mild ITK 22 49 COCCCOCCN(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653283 FE On-Demand Mild PANC 56 40 C=CCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653289 EE On-Demand Mild ITK 21 49 C=CCN(CCOC)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653289 EE On-Demand Mild PANC 41 35 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@H]1C ZINC000880653290 EG On-Demand Mild ITK 19 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@H]1C ZINC000880653290 EG On-Demand Mild PANC 54 37 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@@H]1C ZINC000880653292 EG On-Demand Mild ITK 19 51 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)[C@@H]1C ZINC000880653292 EG On-Demand Mild PANC 54 37 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653293 GF On-Demand Mild ITK 25 48 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653293 GF On-Demand Mild PANC 55 38 CC(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653294 FF On-Demand Mild ITK 26 50 CC(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653294 FF On-Demand Mild MLNR 28 42 CC(=O)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653294 FF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C(F)(F)F)cn2)cc1 ZINC000880653296 EF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C(F)(F)F)cn2)cc1 ZINC000880653296 EF On-Demand Mild PANC 56 39 CCCN(CCN1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653297 GG On-Demand Mild ITK 19 49 CCCN(CCN1CCCC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653297 GG On-Demand Mild MCHR1 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880653299 GG On-Demand Mild ITK 16 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880653299 GG On-Demand Mild PANC 52 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880653300 GG On-Demand Mild ITK 16 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880653300 GG On-Demand Mild PANC 52 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C(F)(F)F)cn2)cc1 ZINC000880653301 EF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C(F)(F)F)cn2)cc1 ZINC000880653301 EF On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880653302 GG On-Demand Mild ITK 16 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@H]3[C@@H]3CCCO3)cn2)cc1 ZINC000880653302 GG On-Demand Mild PANC 52 35 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880653304 GG On-Demand Mild ITK 16 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCC4)[C@H]3[C@H]3CCCO3)cn2)cc1 ZINC000880653304 GG On-Demand Mild PANC 52 35 C[C@H]1C(=O)N(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653310 ED On-Demand Mild ITK 18 51 C[C@H]1C(=O)N(C)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653310 ED On-Demand Mild PANC 57 39 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)N1C ZINC000880653318 FE On-Demand Mild ITK 19 51 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H](C)N1C ZINC000880653318 FE On-Demand Mild PANC 54 36 C=C[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653319 EG On-Demand Mild ITK 17 47 C=C[C@@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653319 EG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880653322 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)[C@@H]3C3CC3)cn2)cc1 ZINC000880653322 GG On-Demand Mild PANC 41 34 C=C[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653323 EG On-Demand Mild ITK 17 47 C=C[C@H]1CCCCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653323 EG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)[C@H]3C3CC3)cn2)cc1 ZINC000880653324 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOCC4)[C@H]3C3CC3)cn2)cc1 ZINC000880653324 GG On-Demand Mild PANC 41 34 CN(CCN(C)C1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653350 FE On-Demand Mild ITK 23 49 CN(CCN(C)C1CC1)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653350 FE On-Demand Mild PANC 58 39 N#Cc1ccc(Cn2cc(NC(=O)NC3([C@@H]4CCCCO4)CCC3)cn2)cc1 ZINC000880653351 GG On-Demand Mild ITK 23 45 N#Cc1ccc(Cn2cc(NC(=O)NC3([C@@H]4CCCCO4)CCC3)cn2)cc1 ZINC000880653351 GG On-Demand Mild PANC 53 36 CN(CCO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653353 GD On-Demand Mild ITK 19 47 CN(CCO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653353 GD On-Demand Mild MLNR 31 40 CN(CCO)C1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653353 GD On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)NC3([C@H]4CCCCO4)CCC3)cn2)cc1 ZINC000880653355 GG On-Demand Mild ITK 23 45 N#Cc1ccc(Cn2cc(NC(=O)NC3([C@H]4CCCCO4)CCC3)cn2)cc1 ZINC000880653355 GG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC=CC[C@H]4C3)cn2)cc1 ZINC000880653372 EG On-Demand Mild ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CC=CC[C@H]4C3)cn2)cc1 ZINC000880653372 EG On-Demand Mild PANC 41 35 N#Cc1ccc(Cn2cc(NC(=O)NC3CC4(CSC4)C3)cn2)cc1 ZINC000880653376 FF On-Demand Mild ITK 16 49 N#Cc1ccc(Cn2cc(NC(=O)NC3CC4(CSC4)C3)cn2)cc1 ZINC000880653376 FF On-Demand Mild PANC 40 33 C[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCOC1 ZINC000880653380 EE On-Demand Mild ITK 15 47 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653384 GG On-Demand Mild ITK 18 46 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653384 GG On-Demand Mild MLNR 25 41 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653384 GG On-Demand Mild PANC 55 38 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653385 GG On-Demand Mild ITK 18 46 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653385 GG On-Demand Mild MLNR 25 41 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN(C2CCC2)C1 ZINC000880653385 GG On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(F)(F)C4)cn2)cc1 ZINC000880653386 FH On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3[C@H]4CC[C@H]3CC(F)(F)C4)cn2)cc1 ZINC000880653386 FH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CCCC4)C3)cn2)cc1 ZINC000880653387 EG On-Demand Mild ITK 19 51 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CCCC4)C3)cn2)cc1 ZINC000880653387 EG On-Demand Mild PANC 54 36 COCC1=CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653388 FF On-Demand Mild ITK 17 47 COCC1=CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653388 FF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCC(F)(F)C3)cn2)cc1 ZINC000880653390 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCC(F)(F)C3)cn2)cc1 ZINC000880653390 FE On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)NC3(C(F)F)CC3)cn2)cc1 ZINC000880653392 EF On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)NC3(CF)CCOCC3)cn2)cc1 ZINC000880653393 FE On-Demand Mild ITK 15 48 CC1(CO)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653394 FE On-Demand Mild ITK 17 49 CN(C[C@@H]1CC1(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653395 EG On-Demand Mild ITK 18 49 CN(C[C@@H]1CC1(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653395 EG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCCc4occc4C3)cn2)cc1 ZINC000880653399 FG On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CC(Cc4cccs4)C3)cn2)cc1 ZINC000880653401 GH On-Demand Mild PANC 44 34 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C(F)F)cn2)cc1 ZINC000880653403 EF On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H]3C(F)F)cn2)cc1 ZINC000880653403 EF On-Demand Mild PANC 54 38 CCC[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1 ZINC000880653407 FF On-Demand Mild ITK 15 45 CCC[C@]1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCOC1 ZINC000880653407 FF On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C(F)F)cn2)cc1 ZINC000880653410 EF On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H]3C(F)F)cn2)cc1 ZINC000880653410 EF On-Demand Mild PANC 54 38 CCn1nc(C)c(CN(C)C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)c1C ZINC000880653417 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3CCCC4(CC3)CC4)cn2)cc1 ZINC000880653419 EH On-Demand Mild ITK 16 51 C[C@H]1C(=O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653421 FF On-Demand Mild ITK 17 47 C[C@H]1C(=O)C[C@H]2CC[C@H]1N2C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653421 FF On-Demand Mild PANC 55 37 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCC1 ZINC000880653423 FF On-Demand Mild ITK 19 48 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCC1 ZINC000880653423 FF On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCCC[C@H]4C3)cn2)cc1 ZINC000880653426 EG On-Demand Mild ITK 19 52 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCCC[C@H]4C3)cn2)cc1 ZINC000880653426 EG On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC(N4CC[C@@H](O)C4)C3)cn2)cc1 ZINC000880653427 FD On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(N4CC[C@@H](O)C4)C3)cn2)cc1 ZINC000880653427 FD On-Demand Mild PANC 56 39 N#CCC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653428 DE On-Demand Mild ITK 15 52 N#CCC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653428 DE On-Demand Mild PANC 41 35 CCC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653429 FD On-Demand Mild ITK 15 50 CCC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653429 FD On-Demand Mild MLNR 17 40 CCC(=O)N1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653429 FD On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCF)C3)cn2)cc1 ZINC000880653431 FG On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CCF)C3)cn2)cc1 ZINC000880653431 FG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCF)C3)cn2)cc1 ZINC000880653432 FG On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CCF)C3)cn2)cc1 ZINC000880653432 FG On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]([C@@H]4CCCCO4)C3)cn2)cc1 ZINC000880653437 GH On-Demand Mild ITK 22 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]([C@@H]4CCCCO4)C3)cn2)cc1 ZINC000880653437 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]([C@@H]4CCCCO4)C3)cn2)cc1 ZINC000880653438 GH On-Demand Mild ITK 22 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]([C@@H]4CCCCO4)C3)cn2)cc1 ZINC000880653438 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]([C@H]4CCCCO4)C3)cn2)cc1 ZINC000880653439 GH On-Demand Mild ITK 22 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H]([C@H]4CCCCO4)C3)cn2)cc1 ZINC000880653439 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]([C@H]4CCCCO4)C3)cn2)cc1 ZINC000880653440 GH On-Demand Mild ITK 22 44 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H]([C@H]4CCCCO4)C3)cn2)cc1 ZINC000880653440 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](CC(F)(F)F)C3)cn2)cc1 ZINC000880653443 GH On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](CC(F)(F)F)C3)cn2)cc1 ZINC000880653444 GH On-Demand Mild PANC 53 37 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653449 FF On-Demand Mild ITK 21 51 CC(C)[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCN1C ZINC000880653449 FF On-Demand Mild PANC 55 38 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@H]3CN4c3ccccc3)cn2)cc1 ZINC000880653453 GG On-Demand Mild ITK 15 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@H]3CN4c3ccccc3)cn2)cc1 ZINC000880653453 GG On-Demand Mild PANC 44 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@]45CCCC[C@]4(COC5)C3)cn2)cc1 ZINC000880653454 GG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@]45CCCC[C@]4(COC5)C3)cn2)cc1 ZINC000880653454 GG On-Demand Mild PANC 40 33 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]45CCCC[C@]4(COC5)C3)cn2)cc1 ZINC000880653455 GG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]45CCCC[C@]4(COC5)C3)cn2)cc1 ZINC000880653455 GG On-Demand Mild PANC 40 33 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]45CCCC[C@@]4(COC5)C3)cn2)cc1 ZINC000880653456 GG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@]45CCCC[C@@]4(COC5)C3)cn2)cc1 ZINC000880653456 GG On-Demand Mild PANC 40 33 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4(O)CC4)CC3)cn2)cc1 ZINC000880653457 FF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(C4(O)CC4)CC3)cn2)cc1 ZINC000880653457 FF On-Demand Mild PANC 49 37 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCCC2)O1 ZINC000880653461 GG On-Demand Mild ITK 15 45 C[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCCC2)O1 ZINC000880653461 GG On-Demand Mild PANC 41 36 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCCC2)O1 ZINC000880653462 GG On-Demand Mild ITK 15 45 C[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC2(CCCC2)O1 ZINC000880653462 GG On-Demand Mild PANC 41 36 CN1CCO[C@@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653482 FD On-Demand Mild ITK 21 47 CN1CCO[C@@H]2CN(C(=O)Nc3cnn(Cc4ccc(C#N)cc4)c3)C[C@@H]21 ZINC000880653482 FD On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CCC[C@]4(CO)C3)cn2)cc1 ZINC000880653488 FE On-Demand Mild PANC 54 37 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](CC)CO1 ZINC000880653490 FG On-Demand Mild ITK 16 48 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](CC)CO1 ZINC000880653490 FG On-Demand Mild PANC 54 36 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](CC)CO1 ZINC000880653491 FG On-Demand Mild ITK 16 48 CC[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@@H](CC)CO1 ZINC000880653491 FG On-Demand Mild PANC 54 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CC3)CC4(F)F)cn2)cc1 ZINC000880653497 FG On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](O)CC3)cn2)cc1 ZINC000880653498 EE On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](O)CC3)cn2)cc1 ZINC000880653498 EE On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](O)CC3)cn2)cc1 ZINC000880653500 EE On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](O)CC3)cn2)cc1 ZINC000880653500 EE On-Demand Mild PANC 53 37 C[C@@H]1CN(CCNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CO1 ZINC000880653505 GE On-Demand Mild ITK 15 45 C[C@@H]1CN(CCNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)CO1 ZINC000880653505 GE On-Demand Mild PANC 41 36 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCc3cccnc31)C2 ZINC000880653515 EG On-Demand Anodyne NQO2 30 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCc3cccnc31)C2 ZINC000880653515 EG On-Demand Anodyne MTNR1A 54 48 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCc3cccnc31)C2 ZINC000880653515 EG On-Demand Anodyne MTNR1B 51 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCc3cccnc31)C2 ZINC000880653515 EG On-Demand Anodyne FAAH 15 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCc3cccnc31)C2 ZINC000880653517 EG On-Demand Anodyne NQO2 30 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCc3cccnc31)C2 ZINC000880653517 EG On-Demand Anodyne MTNR1A 54 48 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCc3cccnc31)C2 ZINC000880653517 EG On-Demand Anodyne MTNR1B 51 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCc3cccnc31)C2 ZINC000880653517 EG On-Demand Anodyne FAAH 15 43 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCOC4)C3)cn2)cc1 ZINC000880653522 EE On-Demand Mild ITK 15 49 CCc1nc2ccccc2n1CC(=O)NCc1cc(O)nc(SC)n1 ZINC000880653524 FE On-Demand Anodyne IMDH_CRYPV 33 44 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)[C@H](C4CCCC4)C3)cn2)cc1 ZINC000880653526 GG On-Demand Mild ITK 18 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](O)[C@H](C4CCCC4)C3)cn2)cc1 ZINC000880653526 GG On-Demand Mild PANC 41 36 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653528 GG On-Demand Mild CCR3 36 42 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653528 GG On-Demand Mild ITK 16 48 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653528 GG On-Demand Mild PANC 58 40 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653530 GG On-Demand Mild CCR3 36 42 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653530 GG On-Demand Mild ITK 16 48 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653530 GG On-Demand Mild PANC 58 40 CC(C)(CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)CC(F)F ZINC000880653539 FH On-Demand Mild ITK 16 52 CC(C)(CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)CC(F)F ZINC000880653539 FH On-Demand Mild PANC 54 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@H](C(F)F)CC3)cn2)cc1 ZINC000880653562 GF On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@H](C(F)F)CC3)cn2)cc1 ZINC000880653564 GF On-Demand Mild PANC 41 36 CC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653570 CE On-Demand Mild ITK 20 53 CC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653570 CE On-Demand Mild MLNR 42 42 CC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653570 CE On-Demand Mild PANC 56 39 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653572 FF On-Demand Mild ITK 17 47 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653572 FF On-Demand Mild MLNR 32 41 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653572 FF On-Demand Mild PANC 56 39 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653573 FF On-Demand Mild ITK 17 47 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653573 FF On-Demand Mild MLNR 32 41 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653573 FF On-Demand Mild PANC 56 39 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653574 FF On-Demand Mild ITK 17 47 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653574 FF On-Demand Mild MLNR 32 41 CO[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@@H]1C ZINC000880653574 FF On-Demand Mild PANC 56 39 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653575 FF On-Demand Mild ITK 17 47 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653575 FF On-Demand Mild MLNR 32 41 CO[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[C@H]1C ZINC000880653575 FF On-Demand Mild PANC 56 39 CCOCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653578 FE On-Demand Mild ITK 17 48 CCOCCOC1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653578 FE On-Demand Mild PANC 52 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCCO4)CC3)cn2)cc1 ZINC000880653583 GG On-Demand Mild ITK 24 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@@H]4CCCO4)CC3)cn2)cc1 ZINC000880653583 GG On-Demand Mild PANC 56 39 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCCO4)CC3)cn2)cc1 ZINC000880653584 GG On-Demand Mild ITK 24 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCC([C@H]4CCCO4)CC3)cn2)cc1 ZINC000880653584 GG On-Demand Mild PANC 56 39 CCC1(CC)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@]1=O ZINC000880653586 GF On-Demand Mild ITK 15 47 CCC1(CC)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC[S@@]1=O ZINC000880653587 GF On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CC4)C3)cn2)cc1 ZINC000880653588 DF On-Demand Mild ITK 18 52 N#Cc1ccc(Cn2cc(NC(=O)N3CC(C4CC4)C3)cn2)cc1 ZINC000880653588 DF On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCOCC4)CC3)cn2)cc1 ZINC000880653594 GG On-Demand Mild ITK 16 51 N#Cc1ccc(Cn2cc(NC(=O)N3CCC4(CCOCC4)CC3)cn2)cc1 ZINC000880653594 GG On-Demand Mild PANC 49 37 C[C@H]1C[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653600 ED On-Demand Mild ITK 19 50 C[C@H]1C[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653600 ED On-Demand Mild PANC 56 38 C[C@@H]1C[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653602 ED On-Demand Mild ITK 19 50 C[C@@H]1C[C@H](O)CN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653602 ED On-Demand Mild PANC 56 38 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@@]4(CCOC4)C3)cn2)cc1 ZINC000880653612 FD On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CCO[C@]4(CCOC4)C3)cn2)cc1 ZINC000880653613 FD On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653614 GG On-Demand Mild CCR3 35 43 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653614 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653614 GG On-Demand Mild RPS6KA3 17 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653615 GG On-Demand Mild CCR3 35 43 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653615 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](Cc4ccncc4)C3)cn2)cc1 ZINC000880653615 GG On-Demand Mild RPS6KA3 17 41 CO[C@@]1(C)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653616 FG On-Demand Mild ITK 20 46 CO[C@@]1(C)CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653616 FG On-Demand Mild PANC 47 35 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4cccnc4)CC3)cn2)cc1 ZINC000880653618 GH On-Demand Mild ITK 19 48 N#Cc1ccc(Cn2cc(NC(=O)N3CCC(c4cccnc4)CC3)cn2)cc1 ZINC000880653618 GH On-Demand Mild PANC 53 36 CC(C)C1(O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653619 EE On-Demand Mild ITK 16 51 CC(C)C1(O)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880653619 EE On-Demand Mild PANC 41 35 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC(F)(F)CC1 ZINC000880653620 FH On-Demand Mild ITK 22 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1CCC(F)(F)CC1 ZINC000880653620 FH On-Demand Mild PANC 54 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCCC4)C3)cn2)cc1 ZINC000880653621 GG On-Demand Mild CCR3 18 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CN4CCCCC4)C3)cn2)cc1 ZINC000880653621 GG On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCCC4)C3)cn2)cc1 ZINC000880653622 GG On-Demand Mild CCR3 18 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CN4CCCCC4)C3)cn2)cc1 ZINC000880653622 GG On-Demand Mild ITK 19 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@@H](C4)C3)cn2)cc1 ZINC000880653629 EG On-Demand Mild ITK 19 50 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4CCC[C@@H](C4)C3)cn2)cc1 ZINC000880653629 EG On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC(=O)N(C4CC4)C3)cn2)cc1 ZINC000880653633 FD On-Demand Mild PANC 41 35 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880653646 GF On-Demand Mild ITK 23 47 CN(C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880653646 GF On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCSCC3)cn2)cc1 ZINC000880653647 GF On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCSCC3)cn2)cc1 ZINC000880653647 GF On-Demand Mild PANC 40 34 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1 ZINC000880653648 EE On-Demand Mild ITK 19 48 COCC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCC1 ZINC000880653648 EE On-Demand Mild PANC 54 37 CCCN(CCCN(C)C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880653653 FF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C4CC4)C3)cn2)cc1 ZINC000880653657 EG On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@@H](C4CC4)C3)cn2)cc1 ZINC000880653657 EG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C4CC4)C3)cn2)cc1 ZINC000880653658 EG On-Demand Mild ITK 17 49 N#Cc1ccc(Cn2cc(NC(=O)N3CCC[C@H](C4CC4)C3)cn2)cc1 ZINC000880653658 EG On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCC4(CC4)C3)cn2)cc1 ZINC000880653659 FE On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CCOCC4(CC4)C3)cn2)cc1 ZINC000880653659 FE On-Demand Mild EPHX2 15 41 N#Cc1ccc(Cn2cc(NC(=O)NCC(F)(F)C(F)F)cn2)cc1 ZINC000880653660 FF On-Demand Mild ITK 15 52 N#Cc1ccc(Cn2cc(NC(=O)NCC(F)(F)C(F)F)cn2)cc1 ZINC000880653660 FF On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H](O)CC(F)(F)C3)cn2)cc1 ZINC000880653663 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H](O)CC(F)(F)C3)cn2)cc1 ZINC000880653664 FE On-Demand Mild PANC 41 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653665 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653665 GG On-Demand Mild CXCR3 23 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653665 GG On-Demand Mild PANC 41 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653666 GG On-Demand Mild ITK 15 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653666 GG On-Demand Mild CXCR3 23 40 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](n4cc(Cl)cn4)C3)cn2)cc1 ZINC000880653666 GG On-Demand Mild PANC 41 37 CN1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653668 ED On-Demand Mild ITK 20 50 CN1CCCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880653668 ED On-Demand Mild PANC 41 36 CS[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880653670 GE On-Demand Mild ITK 16 47 CS[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@H]1N(C)C ZINC000880653671 GE On-Demand Mild ITK 16 47 CS[C@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880653672 GE On-Demand Mild ITK 16 47 CS[C@@H]1CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C[C@@H]1N(C)C ZINC000880653673 GE On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCC3)cn2)cc1 ZINC000880653675 EE On-Demand Mild ITK 20 50 N#Cc1ccc(Cn2cc(NC(=O)N(CCO)C3CCC3)cn2)cc1 ZINC000880653675 EE On-Demand Mild PANC 53 36 N#Cc1ccc(Cn2cc(NC(=O)N3CC4(CCCCC4)C3)cn2)cc1 ZINC000880653676 EH On-Demand Mild ITK 18 52 CC[C@]1(C)CN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCO1 ZINC000880653684 FF On-Demand Mild ITK 15 46 O=C(NOCc1ccc(F)cc1)Nc1ccnn1CC1CCC1 ZINC000880653693 DG On-Demand Anodyne CCR3 91 34 O=C(CCCc1ccccc1)NNC(=O)Nc1ccnn1CC1CCC1 ZINC000880653701 FF On-Demand Reactive PREP 43 37 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(N=S(C)(C)=O)cc2)C1 ZINC000880653708 GG On-Demand Mild L3MBTL3 55 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(N=S(C)(C)=O)cc2)C1 ZINC000880653709 GG On-Demand Mild L3MBTL3 55 38 O=C(NNc1ccc(F)cc1)Nc1ccnn1CC1CCC1 ZINC000880653761 DF On-Demand Reactive CCR3 54 36 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)Cn3nnc(-c4ccccc4)n3)sc2C1 ZINC000880653771 IF On-Demand Anodyne SLC27A1 36 42 O=C(NCc1cc(F)cnc1Cl)Nc1ccnn1CC1CCC1 ZINC000880653840 EG On-Demand Anodyne P2RX7 57 45 COC(=O)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880653869 EE On-Demand Anodyne EPHX2 49 42 COC(=O)c1ccc(CC(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cn1 ZINC000880653903 GE On-Demand Mild MLNR 29 42 COC(=O)c1ccc(CC(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cn1 ZINC000880653904 GE On-Demand Mild MLNR 29 42 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880653985 EH On-Demand Mild ITK 17 48 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3C[C@@H]4CCCC[C@@H]43)cn2)cc1 ZINC000880653985 EH On-Demand Mild PANC 41 35 O=C(NOCc1cccnc1)Nc1ccnn1CC1CCC1 ZINC000880654107 DE On-Demand Anodyne CHRNA7 45 38 Cc1nc(NC2CC2)sc1C(=O)NCCCc1nc(-c2ccccn2)cs1 ZINC000880654172 GH On-Demand Anodyne NPY5R 15 40 CN1CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1(C)C ZINC000880654214 FE On-Demand Mild ITK 16 49 CC[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCOC1 ZINC000880654222 FG On-Demand Mild ITK 15 45 CC[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@@H]1CCCOC1 ZINC000880654222 FG On-Demand Mild PANC 54 36 CC[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCCOC1 ZINC000880654224 FG On-Demand Mild ITK 15 45 CC[C@@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)[C@H]1CCCOC1 ZINC000880654224 FG On-Demand Mild PANC 54 36 O=C(COC1CC1)NCCCc1nc(-c2ccccn2)cs1 ZINC000880654326 DE On-Demand Anodyne NPY5R 15 44 O=C(Cc1ccc(F)cc1)NNC(=O)Nc1ccnn1CC1CCC1 ZINC000880654331 EE On-Demand Reactive CCR3 92 35 CNc1nc(C(=O)NCCCc2nc(-c3ccccn3)cs2)cs1 ZINC000880654345 FG On-Demand Anodyne NPY5R 16 43 CNc1nc(C(=O)NCCCc2nc(-c3ccccn3)cs2)cs1 ZINC000880654345 FG On-Demand Anodyne KCNN1 26 40 CC[C@@H](C(=O)NNC(=O)Nc1ccnn1CC1CCC1)c1ccccc1 ZINC000880654421 FG On-Demand Reactive KCNQ2 48 41 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H]3c3ccccc34)cn2)cc1 ZINC000880654444 GI On-Demand Mild ITK 15 51 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4CC[C@H]3c3ccccc34)cn2)cc1 ZINC000880654444 GI On-Demand Mild PANC 56 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc(Cl)cn2)C1 ZINC000880654445 FF On-Demand Mild MLNR 24 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc(Cl)cn2)C1 ZINC000880654450 FF On-Demand Mild MLNR 24 40 O=C(NNc1ccc(F)c(Cl)c1)Nc1ccnn1CC1CCC1 ZINC000880654467 EH On-Demand Reactive ERBB4 46 31 CCN1CC[C@@H]1CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654482 EE On-Demand Mild CCR3 35 41 CCN1CC[C@@H]1CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654482 EE On-Demand Mild ITK 18 51 CCN1CC[C@@H]1CNC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654482 EE On-Demand Mild PANC 55 38 C[C@H]1C(=O)N(C)[C@H](C)[C@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654504 GE On-Demand Mild ITK 16 51 C[C@H]1C(=O)N(C)[C@H](C)[C@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654504 GE On-Demand Mild PANC 49 35 C[C@H]1C(=O)N(C)[C@H](C)[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654506 GE On-Demand Mild ITK 16 51 C[C@H]1C(=O)N(C)[C@H](C)[C@@H](C)N1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654506 GE On-Demand Mild PANC 49 35 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C(=O)N1C ZINC000880654510 GE On-Demand Mild ITK 16 51 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)[C@H](C)C(=O)N1C ZINC000880654510 GE On-Demand Mild PANC 49 35 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@@]34CCCO4)cn2)cc1 ZINC000880654544 FG On-Demand Mild ITK 16 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@@]34CCCO4)cn2)cc1 ZINC000880654544 FG On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@]34CCCO4)cn2)cc1 ZINC000880654546 FG On-Demand Mild ITK 16 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@]34CCCO4)cn2)cc1 ZINC000880654546 FG On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@]34CCCO4)cn2)cc1 ZINC000880654548 FG On-Demand Mild ITK 16 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@]34CCCO4)cn2)cc1 ZINC000880654548 FG On-Demand Mild PANC 41 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@@]34CCCO4)cn2)cc1 ZINC000880654550 FG On-Demand Mild ITK 16 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@@]34CCCO4)cn2)cc1 ZINC000880654550 FG On-Demand Mild PANC 41 34 C[C@@H](Cc1ccc(O)c(O)c1)NC(=O)Nc1ccnn1CC1CCC1 ZINC000880654553 EF On-Demand Clean CCR3 50 38 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)c3cccnc3N3CCOCC3)sc2C1 ZINC000880654562 IF On-Demand Anodyne MTOR 19 46 C[C@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(F)F ZINC000880654565 DF On-Demand Mild ITK 16 52 C[C@H](NC(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1)C(F)F ZINC000880654565 DF On-Demand Mild PANC 40 35 N#Cc1ccc(Cn2cc(NC(=O)NC[C@H]3C=CCC3)cn2)cc1 ZINC000880654579 DF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)NC[C@H]3C=CCC3)cn2)cc1 ZINC000880654579 DF On-Demand Mild PANC 53 35 N#Cc1ccc(Cn2cc(NC(=O)NC[C@@H]3C=CCC3)cn2)cc1 ZINC000880654580 DF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)NC[C@@H]3C=CCC3)cn2)cc1 ZINC000880654580 DF On-Demand Mild PANC 53 35 O=C(NNc1ccccc1Cl)Nc1ccnn1CC1CCC1 ZINC000880654632 DG On-Demand Reactive EPHB3 45 32 C#CCC1(O)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CC1 ZINC000880654686 FE On-Demand Mild ITK 15 48 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](c4nccs4)C3)cn2)cc1 ZINC000880654718 GG On-Demand Mild ITK 17 45 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](c4nccs4)C3)cn2)cc1 ZINC000880654719 GG On-Demand Mild ITK 17 45 COc1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)c(OC)c1 ZINC000880654731 GG On-Demand Clean HTR1A 27 41 COc1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)c(OC)c1 ZINC000880654731 GG On-Demand Clean PDGFRB 64 42 COc1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)c(OC)c1 ZINC000880654731 GG On-Demand Clean RBP4 18 40 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C=C[C@H]3C4)cn2)cc1 ZINC000880654788 DF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C=C[C@H]3C4)cn2)cc1 ZINC000880654788 DF On-Demand Mild PANC 53 35 CCNc1nc(C)c(C(=O)NCCCc2nc(-c3ccccn3)cs2)s1 ZINC000880654791 GH On-Demand Anodyne NPY5R 15 44 CCNc1nc(C)c(C(=O)NCCCc2nc(-c3ccccn3)cs2)s1 ZINC000880654791 GH On-Demand Anodyne SCD1 19 40 COC(=O)Nc1cccc(CNC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880654796 FG On-Demand Anodyne CCR3 44 38 COC(=O)Nc1cccc(CNC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880654796 FG On-Demand Anodyne ROCK2 25 42 CNc1ncc(C(=O)NCCCc2nc(-c3ccccn3)cs2)s1 ZINC000880654801 FG On-Demand Anodyne NPY5R 17 42 C[C@H](NC(=O)OC(C)(C)C)[C@H]1CCN(C(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880654805 GG On-Demand Anodyne REN 44 36 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880654815 GG On-Demand Anodyne CACNA1I 44 36 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880654815 GG On-Demand Anodyne GPR119 40 38 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880654816 GG On-Demand Anodyne CACNA1I 44 36 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880654816 GG On-Demand Anodyne GPR119 40 38 N#Cc1ccc(Cn2cc(NC(=O)NN3C[C@H]4CCC[C@@H](C4)C3)cn2)cc1 ZINC000880654842 FF On-Demand Mild ITK 18 49 N#Cc1ccc(Cn2cc(NC(=O)NN3C[C@H]4CCC[C@@H](C4)C3)cn2)cc1 ZINC000880654842 FF On-Demand Mild PANC 48 35 C[C@H]1c2sccc2CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654858 GI On-Demand Mild ITK 15 47 C[C@H]1c2sccc2CCN1C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880654858 GI On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)NC[C@H]3CCC4(CCC4)O3)cn2)cc1 ZINC000880654860 FG On-Demand Mild PANC 49 36 N#Cc1ccc(Cn2cc(NC(=O)NC[C@@H]3CCC4(CCC4)O3)cn2)cc1 ZINC000880654861 FG On-Demand Mild PANC 49 36 O=C(NCc1nc(-c2ccncc2)cs1)Nc1ccnn1CC1CCC1 ZINC000880654896 FH On-Demand Anodyne ROCK1 23 44 O=C(NCc1nc(-c2ccncc2)cs1)Nc1ccnn1CC1CCC1 ZINC000880654896 FH On-Demand Anodyne ROCK2 17 44 O=C(NCc1cc(O)ccc1Cl)Nc1ccnn1CC1CCC1 ZINC000880654908 EG On-Demand Anodyne P2RX7 22 40 O=C(NCCn1ccnn1)c1cccc(S(=O)(=O)C(F)F)c1 ZINC000880654912 EC On-Demand Anodyne DRD4 40 31 CN1CCN(C2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)CC1 ZINC000880654921 FD On-Demand Anodyne L3MBTL3 73 42 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@@](C)(O)c1ccccc1 ZINC000880654955 EG On-Demand Anodyne AMY2 43 30 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@](C)(O)c1ccccc1 ZINC000880654957 EG On-Demand Anodyne AMY2 43 30 N#Cc1ccc(Cn2cc(NC(=O)NC3CCC4(CC3)COC4)cn2)cc1 ZINC000880655023 FF On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)NC3CCC4(CC3)COC4)cn2)cc1 ZINC000880655023 FF On-Demand Mild PANC 54 36 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880655034 GF On-Demand Mild ITK 15 45 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)C1 ZINC000880655034 GF On-Demand Mild PANC 42 36 C#CC1(NC(=O)Nc2cnn(Cc3ccc(C#N)cc3)c2)CCCC1 ZINC000880655038 EF On-Demand Mild ITK 16 50 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@@]34CCCCO4)cn2)cc1 ZINC000880655050 GG On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@@]34CCCCO4)cn2)cc1 ZINC000880655050 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@@]34CCCCO4)cn2)cc1 ZINC000880655051 GG On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@@]34CCCCO4)cn2)cc1 ZINC000880655051 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@]34CCCCO4)cn2)cc1 ZINC000880655052 GG On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@H]3CCC[C@]34CCCCO4)cn2)cc1 ZINC000880655052 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@]34CCCCO4)cn2)cc1 ZINC000880655053 GG On-Demand Mild ITK 15 45 N#Cc1ccc(Cn2cc(NC(=O)N[C@@H]3CCC[C@]34CCCCO4)cn2)cc1 ZINC000880655053 GG On-Demand Mild PANC 40 34 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@]4(O)C3)cn2)cc1 ZINC000880655058 DD On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@H]4C[C@@]4(O)C3)cn2)cc1 ZINC000880655059 DD On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@@]4(O)C3)cn2)cc1 ZINC000880655060 DD On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3C[C@@H]4C[C@]4(O)C3)cn2)cc1 ZINC000880655061 DD On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CF)C3)cn2)cc1 ZINC000880655065 EF On-Demand Mild CCR3 17 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CF)C3)cn2)cc1 ZINC000880655065 EF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@@H](CF)C3)cn2)cc1 ZINC000880655065 EF On-Demand Mild PANC 53 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CF)C3)cn2)cc1 ZINC000880655066 EF On-Demand Mild CCR3 17 41 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CF)C3)cn2)cc1 ZINC000880655066 EF On-Demand Mild ITK 15 49 N#Cc1ccc(Cn2cc(NC(=O)N3CC[C@H](CF)C3)cn2)cc1 ZINC000880655066 EF On-Demand Mild PANC 53 37 CO[C@H]1COCC[C@@H]1N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880655077 FE On-Demand Mild ITK 18 44 CO[C@H]1COCC[C@@H]1N(C)C(=O)Nc1cnn(Cc2ccc(C#N)cc2)c1 ZINC000880655077 FE On-Demand Mild PANC 55 37 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC4CCOCC4)C3)cn2)cc1 ZINC000880655081 GG On-Demand Mild ITK 16 47 N#Cc1ccc(Cn2cc(NC(=O)N3CC(CC4CCOCC4)C3)cn2)cc1 ZINC000880655081 GG On-Demand Mild PANC 53 36 N#Cc1cccc(NNC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880655120 DF On-Demand Reactive CCR3 18 41 CN(C(=O)Nc1ccnn1CC1CCC1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880655211 GH On-Demand Anodyne GPR119 43 39 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880655220 GG On-Demand Anodyne EPHX2 51 39 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880655220 GG On-Demand Anodyne GPR119 46 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cnccc2Cl)C1 ZINC000880655232 FF On-Demand Mild PGR 17 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cnccc2Cl)C1 ZINC000880655232 FF On-Demand Mild ITGA4 40 30 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cnccc2Cl)C1 ZINC000880655233 FF On-Demand Mild PGR 17 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cnccc2Cl)C1 ZINC000880655233 FF On-Demand Mild ITGA4 40 30 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H](F)C(F)(F)F)C1 ZINC000880655234 EE On-Demand Mild MCHR1 35 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H](F)C(F)(F)F)C1 ZINC000880655235 EE On-Demand Mild MCHR1 35 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H](F)C(F)(F)F)C1 ZINC000880655236 EE On-Demand Mild MCHR1 35 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H](F)C(F)(F)F)C1 ZINC000880655237 EE On-Demand Mild MCHR1 35 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H](O)c2cccnc2)C1 ZINC000880655253 ED On-Demand Mild PTAFR 15 43 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H](O)c2cccnc2)C1 ZINC000880655254 ED On-Demand Mild PTAFR 15 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H](O)c2cccnc2)C1 ZINC000880655255 ED On-Demand Mild PTAFR 15 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H](O)c2cccnc2)C1 ZINC000880655256 ED On-Demand Mild PTAFR 15 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(CF)cc2)C1 ZINC000880655275 EG On-Demand Mild L3MBTL3 59 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(CF)cc2)C1 ZINC000880655276 EG On-Demand Mild L3MBTL3 59 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc(F)cn2)C1 ZINC000880655346 EE On-Demand Mild MLNR 46 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc(F)cn2)C1 ZINC000880655347 EE On-Demand Mild MLNR 46 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc(C#N)nc2)C1 ZINC000880655350 EE On-Demand Mild MLNR 34 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc(C#N)nc2)C1 ZINC000880655351 EE On-Demand Mild MLNR 34 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655365 GE On-Demand Mild PGR 15 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655365 GE On-Demand Mild CACNA1B 22 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655365 GE On-Demand Mild CCR5 24 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655366 GE On-Demand Mild PGR 15 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655366 GE On-Demand Mild CACNA1B 22 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccccc2S(C)(=O)=O)C1 ZINC000880655366 GE On-Demand Mild CCR5 24 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccccc2CC#N)C1 ZINC000880655374 FF On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccccc2CC#N)C1 ZINC000880655375 FF On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655405 FG On-Demand Mild CACNA1B 27 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655405 FG On-Demand Mild SLC9A1 16 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655405 FG On-Demand Mild PKNB 16 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655405 FG On-Demand Mild MAP3K12 25 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655406 FG On-Demand Mild CACNA1B 27 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655406 FG On-Demand Mild SLC9A1 16 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655406 FG On-Demand Mild PKNB 16 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(C(F)(F)F)c2)C1 ZINC000880655406 FG On-Demand Mild MAP3K12 25 40 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880655420 GG On-Demand Anodyne GPR119 46 39 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCc3cncn3C2)C1 ZINC000880655421 EE On-Demand Mild CYP11B1 16 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCc3cncn3C2)C1 ZINC000880655422 EE On-Demand Mild CYP11B1 16 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCc3cncn3C2)C1 ZINC000880655423 EE On-Demand Mild CYP11B1 16 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCc3cncn3C2)C1 ZINC000880655424 EE On-Demand Mild CYP11B1 16 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCc3nc[nH]c3C2)C1 ZINC000880655426 EE On-Demand Mild HTR3A 15 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCc3nc[nH]c3C2)C1 ZINC000880655427 EE On-Demand Mild HTR3A 15 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCc3nc[nH]c3C2)C1 ZINC000880655428 EE On-Demand Mild HTR3A 15 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCc3nc[nH]c3C2)C1 ZINC000880655429 EE On-Demand Mild HTR3A 15 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cncnc2)C1 ZINC000880655438 DD On-Demand Mild MLNR 23 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cncnc2)C1 ZINC000880655439 DD On-Demand Mild MLNR 23 42 Cc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cc1C#N ZINC000880655440 EG On-Demand Mild L3MBTL3 52 36 Cc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cc1C#N ZINC000880655441 EG On-Demand Mild L3MBTL3 52 36 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@H](O)c1cccc(F)c1 ZINC000880655532 EG On-Demand Anodyne CCR3 42 36 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@@H](O)c1cccc(F)c1 ZINC000880655534 EG On-Demand Anodyne CCR3 42 36 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655539 CE On-Demand Mild PGR 15 45 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655539 CE On-Demand Mild CACNA1B 23 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655539 CE On-Demand Mild MCHR1 40 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655540 CE On-Demand Mild PGR 15 45 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655540 CE On-Demand Mild CACNA1B 23 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(C)F)C1 ZINC000880655540 CE On-Demand Mild MCHR1 40 38 O=C(NCc1ccccc1N1CCOCC1)Nc1ccnn1CC1CCC1 ZINC000880655558 FF On-Demand Anodyne SCN10A 15 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc3c(c2)NC(=O)C3)C1 ZINC000880655561 FE On-Demand Mild MLNR 26 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc3c(c2)NC(=O)C3)C1 ZINC000880655562 FE On-Demand Mild MLNR 26 41 COc1ccc(N2CCC(NC(=O)Nc3ccnn3CC3CCC3)CC2)cc1 ZINC000880655572 GG On-Demand Clean EPHX2 45 36 COc1ccc(N2CCC(NC(=O)Nc3ccnn3CC3CCC3)CC2)cc1 ZINC000880655572 GG On-Demand Clean PDK1 48 37 O=C(NCc1ccc(-n2ccnc2)cc1)Nc1ccnn1CC1CCC1 ZINC000880655618 FG On-Demand Anodyne NOS2 92 36 O=C(NC[C@H](O)c1cccc(Cl)c1)Nc1ccnn1CC1CCC1 ZINC000880655631 EG On-Demand Anodyne ADRB3 38 40 O=C(NC[C@@H](O)c1cccc(Cl)c1)Nc1ccnn1CC1CCC1 ZINC000880655632 EG On-Demand Anodyne ADRB3 38 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(Cl)Cl)C1 ZINC000880655637 EF On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(Cl)Cl)C1 ZINC000880655637 EF On-Demand Mild MLNR 17 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(Cl)Cl)C1 ZINC000880655638 EF On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(Cl)Cl)C1 ZINC000880655638 EF On-Demand Mild MLNR 17 40 COc1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)cc1 ZINC000880655647 FG On-Demand Clean PDGFRB 48 36 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C2CCC(O)CC2)C1 ZINC000880655670 EE On-Demand Mild MCHR1 15 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C2CCC(O)CC2)C1 ZINC000880655671 EE On-Demand Mild MCHR1 15 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(F)F)C1 ZINC000880655694 CE On-Demand Mild CACNA1B 27 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(F)F)C1 ZINC000880655695 CE On-Demand Mild CACNA1B 27 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccccc2N2CCOCC2)C1 ZINC000880655755 GF On-Demand Mild SLC6A9 17 43 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccccc2N2CCOCC2)C1 ZINC000880655756 GF On-Demand Mild SLC6A9 17 43 O=C(/C=C\c1cccnc1)N1CCN(S(=O)(=O)c2ccc3nc(O)[nH]c3c2)CC1 ZINC000880655762 HD On-Demand Anodyne TGM2 42 31 O=C(/C=C/c1cccnc1)N1CCN(S(=O)(=O)c2ccc3nc(O)[nH]c3c2)CC1 ZINC000880655763 HD On-Demand Anodyne TGM2 42 31 N#Cc1ccc(F)c(CNC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880655764 EG On-Demand Mild P2RX7 22 40 Cc1cccc2c1CCN(C(=O)Nc1ccnn1CC1CCC1)C2 ZINC000880655776 DH On-Demand Anodyne P2RY14 49 35 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccnn1CC1CCC1 ZINC000880655779 GF On-Demand Anodyne EPHX2 15 46 CCC(F)(F)C(=O)N1CC[C@H](N(C)c2cccc(C#N)c2)C1 ZINC000880655794 DF On-Demand Mild PGR 15 42 CCC(F)(F)C(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1 ZINC000880655795 DF On-Demand Mild PGR 15 42 CN(C)CCc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880655801 GG On-Demand Mild MCHR1 28 41 CN(C)CCc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880655801 GG On-Demand Mild L3MBTL3 53 38 CN(C)CCc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880655802 GG On-Demand Mild MCHR1 28 41 CN(C)CCc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880655802 GG On-Demand Mild L3MBTL3 53 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2nc(Cl)ccc2F)C1 ZINC000880655803 FG On-Demand Mild MCHR1 40 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2nc(Cl)ccc2F)C1 ZINC000880655804 FG On-Demand Mild MCHR1 40 38 COC(=O)Nc1cccc(NC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880655822 EH On-Demand Anodyne CCR3 42 38 COC(=O)Nc1cccc(NC(=O)Nc2ccnn2CC2CCC2)c1 ZINC000880655822 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@@H]1CCn2ccnc21 ZINC000880655912 EF On-Demand Anodyne CCR3 51 37 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@H]1CCn2ccnc21 ZINC000880655913 EF On-Demand Anodyne CCR3 51 37 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc(O)cc1Cl)C2 ZINC000880655938 EH On-Demand Anodyne ROCK2 21 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@](O)(C(F)F)C1 ZINC000880655940 EF On-Demand Anodyne CACNA1H 32 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@](O)(C(F)F)C1 ZINC000880655940 EF On-Demand Anodyne S1PR2 31 45 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@](O)(C(F)F)C1 ZINC000880655941 EF On-Demand Anodyne CACNA1H 32 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@](O)(C(F)F)C1 ZINC000880655941 EF On-Demand Anodyne S1PR2 31 45 CN(C(=O)C[C@@H]1CCNC1=O)[C@H](CO)Cc1ccccc1 ZINC000880655959 CC On-Demand Anodyne GALR1 44 32 CN(C(=O)C[C@H]1CCNC1=O)[C@H](CO)Cc1ccccc1 ZINC000880655960 CC On-Demand Anodyne GALR1 44 32 CN(C(=O)C[C@@H]1CCNC1=O)[C@@H](CO)Cc1ccccc1 ZINC000880655961 CC On-Demand Anodyne GALR1 44 32 CN(C(=O)C[C@H]1CCNC1=O)[C@@H](CO)Cc1ccccc1 ZINC000880655962 CC On-Demand Anodyne GALR1 44 32 CS(=O)(=O)C1CCC(C(=O)Nc2ccc(O)cc2Cl)CC1 ZINC000880655993 EF On-Demand Anodyne EPHX2 15 42 CS(=O)(=O)C1CCC(C(=O)Nc2ccc(O)cc2Cl)CC1 ZINC000880655993 EF On-Demand Anodyne TYK2 38 41 O=C(N[C@@H]1CCNC1=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880656003 DD On-Demand Anodyne PDE4D 20 42 O=C(N[C@H]1CCNC1=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880656005 DD On-Demand Anodyne PDE4D 20 42 CC(C)(C)OC(=O)N1CCC[C@@H](C2CCN(C(=O)C[C@@H]3CCNC3=O)CC2)C1 ZINC000880656043 GE On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CCC[C@@H](C2CCN(C(=O)C[C@H]3CCNC3=O)CC2)C1 ZINC000880656045 GE On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CCC[C@H](C2CCN(C(=O)C[C@@H]3CCNC3=O)CC2)C1 ZINC000880656047 GE On-Demand Anodyne GPR119 21 41 CC(C)(C)OC(=O)N1CCC[C@H](C2CCN(C(=O)C[C@H]3CCNC3=O)CC2)C1 ZINC000880656049 GE On-Demand Anodyne GPR119 21 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CC(=O)NCC(F)(F)F)C1 ZINC000880656077 FD On-Demand Mild MCHR1 40 37 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CC(=O)NCC(F)(F)F)C1 ZINC000880656078 FD On-Demand Mild MCHR1 40 37 CCn1cc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)c(C(F)(F)F)n1 ZINC000880656094 GG On-Demand Mild CACNA1B 22 40 CCn1cc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)c(C(F)(F)F)n1 ZINC000880656095 GG On-Demand Mild CACNA1B 22 40 O=C(NCc1ccc(Cl)nc1)Nc1ccnn1CC1CCC1 ZINC000880656109 DG On-Demand Anodyne NAMPT 37 44 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1ccnn1CC1CCC1 ZINC000880656135 FG On-Demand Anodyne CCR3 60 44 C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)Nc1ccnn1CC1CCC1 ZINC000880656137 FG On-Demand Anodyne CCR3 60 44 C#CC[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880656175 EH On-Demand Mild CCR3 59 33 C#CC[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880656177 EH On-Demand Mild CCR3 59 33 O=C(NOCC1CCC1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880656194 DG On-Demand Anodyne CCR3 47 37 Cc1ncc(CC(=O)N2CCC([C@H]3CCCN(C(=O)OC(C)(C)C)C3)CC2)o1 ZINC000880656227 GG On-Demand Anodyne GPR119 44 44 Cc1ncc(CC(=O)N2CCC([C@@H]3CCCN(C(=O)OC(C)(C)C)C3)CC2)o1 ZINC000880656228 GG On-Demand Anodyne GPR119 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656234 ED On-Demand Anodyne PAPA1_CARPA 41 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656234 ED On-Demand Anodyne CTSK 18 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656234 ED On-Demand Anodyne CTSL 16 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656234 ED On-Demand Anodyne FPR1 44 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656235 ED On-Demand Anodyne PAPA1_CARPA 41 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656235 ED On-Demand Anodyne CTSK 18 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656235 ED On-Demand Anodyne CTSL 16 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)n1 ZINC000880656235 ED On-Demand Anodyne FPR1 44 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(O)cc1Cl ZINC000880656237 FF On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(O)cc1Cl ZINC000880656238 FF On-Demand Anodyne PAPA1_CARPA 38 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cccs2)C1 ZINC000880656245 EF On-Demand Mild ETHR 33 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cccs2)C1 ZINC000880656246 EF On-Demand Mild ETHR 33 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656270 GG On-Demand Mild CYP11B1 18 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656270 GG On-Demand Mild CCR5 18 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656270 GG On-Demand Mild CYP11B2 17 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656270 GG On-Demand Mild MLNR 21 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656271 GG On-Demand Mild CYP11B1 18 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656271 GG On-Demand Mild CCR5 18 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656271 GG On-Demand Mild CYP11B2 17 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2cncn2Cc2ccccc2)C1 ZINC000880656271 GG On-Demand Mild MLNR 21 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(C(N)=S)cc2)C1 ZINC000880656296 FF On-Demand Mild SLC9A1 19 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(C(N)=S)cc2)C1 ZINC000880656296 FF On-Demand Mild L3MBTL3 56 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(C(N)=S)cc2)C1 ZINC000880656297 FF On-Demand Mild SLC9A1 19 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(C(N)=S)cc2)C1 ZINC000880656297 FF On-Demand Mild L3MBTL3 56 38 O=C(Nc1ccc(O)cc1Cl)c1ccc(CN2CCOCC2)o1 ZINC000880656356 EF On-Demand Anodyne CSF1R 21 40 O=C(Nc1cccc(CN2CCOC2=O)c1)Nc1ccnn1CC1CCC1 ZINC000880656359 FG On-Demand Anodyne CCR3 50 38 O=C(CCc1cc(Br)c(Br)s1)N[C@@H]1CCNC1=O ZINC000880656386 GE On-Demand Anodyne LUXR 53 38 O=C(CCc1cc(Br)c(Br)s1)N[C@H]1CCNC1=O ZINC000880656387 GE On-Demand Anodyne LUXR 53 38 CN(C(=O)C[C@H]1CCC(C)(C)CO1)[C@H](CO)Cc1ccccc1 ZINC000880656390 DF On-Demand Anodyne TIMP3 47 33 CN(C(=O)C[C@H]1CCC(C)(C)CO1)[C@@H](CO)Cc1ccccc1 ZINC000880656391 DF On-Demand Anodyne TIMP3 47 33 CN(C(=O)C[C@@H]1CCC(C)(C)CO1)[C@H](CO)Cc1ccccc1 ZINC000880656392 DF On-Demand Anodyne TIMP3 47 33 CN(C(=O)C[C@@H]1CCC(C)(C)CO1)[C@@H](CO)Cc1ccccc1 ZINC000880656393 DF On-Demand Anodyne TIMP3 47 33 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCN(c2ccnc(F)c2)CC1 ZINC000880656419 GG On-Demand Anodyne PDGFRB 42 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cccc(F)c2C#N)C1 ZINC000880656470 EF On-Demand Mild CACNA1B 18 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cccc(F)c2C#N)C1 ZINC000880656471 EF On-Demand Mild CACNA1B 18 40 O=C(NCc1cccnc1-n1ccnc1)Nc1ccnn1CC1CCC1 ZINC000880656488 FF On-Demand Anodyne NOS2 91 34 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656493 GE On-Demand Mild PREP 54 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656493 GE On-Demand Mild SFRP1 50 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656493 GE On-Demand Mild WNT3 59 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656494 GE On-Demand Mild PREP 54 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656494 GE On-Demand Mild SFRP1 50 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656494 GE On-Demand Mild WNT3 59 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656495 GE On-Demand Mild PREP 54 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656495 GE On-Demand Mild SFRP1 50 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656495 GE On-Demand Mild WNT3 59 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656496 GE On-Demand Mild PREP 54 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656496 GE On-Demand Mild SFRP1 50 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCCN2C(=O)C(F)(F)F)C1 ZINC000880656496 GE On-Demand Mild WNT3 59 38 CCN(CCNC(=O)Nc1ccnn1CC1CCC1)C(C)C ZINC000880656506 DF On-Demand Anodyne DOT1L 40 31 COc1ccc(N2CCCN(C(=O)Nc3ccnn3CC3CCC3)CC2)cc1 ZINC000880656522 GG On-Demand Clean PDGFRB 42 35 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880656529 GG On-Demand Anodyne ACACB 15 41 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccnn2CC2CCC2)C1 ZINC000880656530 GG On-Demand Anodyne ACACB 15 41 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@H](O)c1ccc(F)cc1 ZINC000880656545 EG On-Demand Anodyne CCR3 57 39 C[C@H](NC(=O)Nc1ccnn1CC1CCC1)[C@@H](O)c1ccc(F)cc1 ZINC000880656547 EG On-Demand Anodyne CCR3 57 39 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(C#N)c2)C1 ZINC000880656552 EE On-Demand Mild MAP3K12 29 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(C#N)c2)C1 ZINC000880656553 EE On-Demand Mild MAP3K12 29 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(F)F)C1 ZINC000880656563 CD On-Demand Mild MCHR1 28 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(F)F)C1 ZINC000880656565 CD On-Demand Mild MCHR1 28 40 CC[C@H](C)N(CC)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880656577 CG On-Demand Anodyne MPO 71 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@H]1CCCN(O)C1=O ZINC000880656619 ED On-Demand Mild CCR3 44 33 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@@H]1CCCN(O)C1=O ZINC000880656620 ED On-Demand Mild CCR3 44 33 O=C1NCC[C@@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656662 EC On-Demand Anodyne GRIN2B 19 40 O=C1NCC[C@@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656662 EC On-Demand Anodyne PREP 25 40 O=C1NCC[C@@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656662 EC On-Demand Anodyne LGMN 66 40 O=C1NCC[C@@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656662 EC On-Demand Anodyne Q9NAW4_PLAFA 38 44 O=C1NCC[C@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656663 EC On-Demand Anodyne GRIN2B 19 40 O=C1NCC[C@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656663 EC On-Demand Anodyne PREP 25 40 O=C1NCC[C@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656663 EC On-Demand Anodyne LGMN 66 40 O=C1NCC[C@H]1NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656663 EC On-Demand Anodyne Q9NAW4_PLAFA 38 44 COC(=O)NCc1ccc(NC(=O)Nc2ccnn2CC2CCC2)cc1 ZINC000880656705 FG On-Demand Anodyne MTOR 41 31 C[C@@H](C(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1)C(C)(F)F ZINC000880656710 DF On-Demand Mild MCHR1 26 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C2CCN(C3CC3)CC2)C1 ZINC000880656725 FE On-Demand Mild MCHR1 18 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C2CCN(C3CC3)CC2)C1 ZINC000880656725 FE On-Demand Mild L3MBTL3 62 37 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C2CCN(C3CC3)CC2)C1 ZINC000880656726 FE On-Demand Mild MCHR1 18 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C2CCN(C3CC3)CC2)C1 ZINC000880656726 FE On-Demand Mild L3MBTL3 62 37 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(C)C(C)(F)F)C1 ZINC000880656748 EG On-Demand Mild CACNA1B 17 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(C)C(C)(F)F)C1 ZINC000880656749 EG On-Demand Mild CACNA1B 17 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 ZINC000880656767 FF On-Demand Mild CCR5 17 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 ZINC000880656767 FF On-Demand Mild MLNR 33 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 ZINC000880656768 FF On-Demand Mild CCR5 17 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 ZINC000880656768 FF On-Demand Mild MLNR 33 44 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880656778 GH On-Demand Anodyne EPHX2 30 52 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880656779 GH On-Demand Anodyne EPHX2 30 52 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880656784 FF On-Demand Anodyne CACNA1H 31 41 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880656784 FF On-Demand Anodyne S1PR2 28 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CCNC2=O)CC1 ZINC000880656792 FF On-Demand Anodyne CACNA1H 60 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CCNC2=O)CC1 ZINC000880656792 FF On-Demand Anodyne S1PR2 30 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCN(c2cccc(F)n2)CC1 ZINC000880656803 GG On-Demand Anodyne PDGFRB 36 40 CCOC(=O)N1CCN(C(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880656814 ED On-Demand Anodyne P2RY12 52 38 CC[C@H](C)N(CC)C(=O)Cc1ccccc1N1CCCC1=O ZINC000880656835 DG On-Demand Anodyne KCNQ2 57 37 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)COc2cccnc2)C1 ZINC000880656838 EE On-Demand Mild CPT1A 93 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)COc2cccnc2)C1 ZINC000880656841 EE On-Demand Mild CPT1A 93 42 CCOC(=O)N1CCCN(C(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880656863 EE On-Demand Anodyne P2RY12 41 37 CCS(=O)(=O)NCC(=O)N1CC[C@H](N(C)c2cccc(C#N)c2)C1 ZINC000880656882 FC On-Demand Mild CCR5 19 43 CN(C(=O)Cc1ccccc1N1CCCC1=O)[C@H](CO)Cc1ccccc1 ZINC000880656883 FE On-Demand Anodyne OPRK1 17 41 CN(C(=O)Cc1ccccc1N1CCCC1=O)[C@@H](CO)Cc1ccccc1 ZINC000880656884 FE On-Demand Anodyne OPRK1 17 41 CCS(=O)(=O)NCC(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1 ZINC000880656890 FC On-Demand Mild CCR5 19 43 C[S@](=N)(=O)N1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880656922 FE On-Demand Anodyne S1PR2 27 40 CN(Cc1cnc[nH]1)C(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880656937 FE On-Demand Anodyne PREP 23 41 C[C@@H]1[C@H](C(=O)NNC(=O)Nc2cc(F)cc(OC(F)F)c2)CCCN1C ZINC000880656965 FE On-Demand Reactive CCR3 59 34 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(NC=O)cc2)C1 ZINC000880656969 EE On-Demand Mild L3MBTL3 57 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(NC=O)cc2)C1 ZINC000880656970 EE On-Demand Mild L3MBTL3 57 38 CN(C(=O)COC1CC1)[C@@H](CO)Cc1ccccc1 ZINC000880656987 CD On-Demand Anodyne TIMP3 85 40 CN(C(=O)COC1CC1)[C@H](CO)Cc1ccccc1 ZINC000880656989 CD On-Demand Anodyne TIMP3 85 40 Cn1nnnc1C1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880657000 FE On-Demand Anodyne CCR3 56 35 COC[C@@H]1CCCN1NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880657028 EF On-Demand Anodyne CCR3 62 33 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CC(N)=O)C1 ZINC000880657032 CC On-Demand Mild MLNR 17 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CC(N)=O)C1 ZINC000880657038 CC On-Demand Mild MLNR 17 41 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CC2(CSC2)C1 ZINC000880657039 EG On-Demand Anodyne EPHX2 15 45 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880657091 GE On-Demand Mild MLNR 15 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880657092 GE On-Demand Mild MLNR 15 40 CN(Cc1cnc[nH]1)C(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880657093 CE On-Demand Anodyne TAAR1 23 41 C#CCC1(O)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880657096 EF On-Demand Mild CACNA1H 33 41 C#CCC1(O)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880657096 EF On-Demand Mild S1PR2 34 49 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCCN2C)C1 ZINC000880657098 DD On-Demand Mild CHRNA10 18 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)OCCCO2 ZINC000880657120 FG On-Demand Anodyne CACNA1H 32 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)OCCCO2 ZINC000880657120 FG On-Demand Anodyne S1PR2 29 42 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccnn1CC1CCC1 ZINC000880657131 GG On-Demand Anodyne L3MBTL3 64 37 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccnn1CC1CCC1 ZINC000880657131 GG On-Demand Anodyne NAMPT 37 49 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC2(CC2)C1 ZINC000880657142 CG On-Demand Anodyne CACNA1H 31 42 O=C(COC1CC1)NCc1cc(Cl)cc(Cl)c1 ZINC000880657152 CF On-Demand Anodyne CACNA1I 50 34 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)c(F)c1 ZINC000880657170 GG On-Demand Anodyne NPY2R 83 36 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccnn3CC3CCC3)CC2)c(F)c1 ZINC000880657170 GG On-Demand Anodyne SLC6A9 18 45 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C1 ZINC000880657176 GE On-Demand Mild ADK 29 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C1 ZINC000880657176 GE On-Demand Mild FASN 32 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C1 ZINC000880657177 GE On-Demand Mild ADK 29 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc(N3CCOCC3)nc2)C1 ZINC000880657177 GE On-Demand Mild FASN 32 42 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880657183 FF On-Demand Anodyne SLC6A3 42 41 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880657184 FF On-Demand Anodyne SLC6A3 42 41 COC(=O)Nc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880657200 GG On-Demand Mild MCHR1 38 43 COC(=O)Nc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880657200 GG On-Demand Mild L3MBTL3 48 36 COC(=O)Nc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880657201 GG On-Demand Mild MCHR1 38 43 COC(=O)Nc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cc1 ZINC000880657201 GG On-Demand Mild L3MBTL3 48 36 Cn1ccnc1[C@@H]1OCCC[C@H]1CNC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880657202 GG On-Demand Anodyne CCR3 62 35 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccncc2)C1 ZINC000880657218 DE On-Demand Mild CCR5 18 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)Cc2ccncc2)C1 ZINC000880657218 DE On-Demand Mild MLNR 30 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccncc2)C1 ZINC000880657219 DE On-Demand Mild CCR5 18 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)Cc2ccncc2)C1 ZINC000880657219 DE On-Demand Mild MLNR 30 44 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)OCCO2 ZINC000880657261 EF On-Demand Anodyne CACNA1H 33 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CC1)OCCO2 ZINC000880657261 EF On-Demand Anodyne S1PR2 30 43 Cc1cc(OCC(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)no1 ZINC000880657269 ED On-Demand Mild CPT1A 37 40 Cc1cc(OCC(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)no1 ZINC000880657271 ED On-Demand Mild CPT1A 37 40 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880657311 GG On-Demand Anodyne CACNA1I 41 33 Cn1nnc(C(=O)N2CCC([C@H]3CCCN(C(=O)OC(C)(C)C)C3)CC2)n1 ZINC000880657341 GD On-Demand Anodyne GPR119 22 43 Cn1nnc(C(=O)N2CCC([C@@H]3CCCN(C(=O)OC(C)(C)C)C3)CC2)n1 ZINC000880657342 GD On-Demand Anodyne GPR119 22 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@H]1CCOC1=O ZINC000880657360 DD On-Demand Anodyne LUXR 70 39 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@H]1CCOC1=O ZINC000880657360 DD On-Demand Anodyne TRAR 85 39 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@H]1CCOC1=O ZINC000880657360 DD On-Demand Anodyne LASR 56 34 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(Cl)c2)C1 ZINC000880657368 EF On-Demand Mild MAP3K12 26 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(Cl)c2)C1 ZINC000880657369 EF On-Demand Mild MAP3K12 26 41 CN1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CCC1(C)C ZINC000880657372 EG On-Demand Anodyne CACNA1H 33 46 CN1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CCC1(C)C ZINC000880657372 EG On-Demand Anodyne S1PR2 30 43 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CNC(=O)c2ccncc2)C1 ZINC000880657381 FD On-Demand Mild PREP 18 43 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CNC(=O)c2ccncc2)C1 ZINC000880657381 FD On-Demand Mild CCR2 23 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CNC(=O)c2ccncc2)C1 ZINC000880657382 FD On-Demand Mild PREP 18 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CNC(=O)c2ccncc2)C1 ZINC000880657382 FD On-Demand Mild CCR2 23 44 CN1CC[C@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC[C@@H]21 ZINC000880657385 EF On-Demand Anodyne CACNA1H 17 41 CN1CC[C@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC[C@H]21 ZINC000880657386 EF On-Demand Anodyne CACNA1H 17 41 CN1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)Cc2cccnc21 ZINC000880657389 FG On-Demand Anodyne PDGFRB 40 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CNC(=O)c2cccnc2)C1 ZINC000880657392 FD On-Demand Mild CCR2 30 45 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CNC(=O)c2cccnc2)C1 ZINC000880657393 FD On-Demand Mild CCR2 30 45 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CCCC(N)=O)C1 ZINC000880657394 DD On-Demand Mild ITK 27 43 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CCCC(N)=O)C1 ZINC000880657394 DD On-Demand Mild MLNR 15 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CCCC(N)=O)C1 ZINC000880657395 DD On-Demand Mild ITK 27 43 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CCCC(N)=O)C1 ZINC000880657395 DD On-Demand Mild MLNR 15 40 CNc1nc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cs1 ZINC000880657402 EE On-Demand Mild TRPC6 61 40 CNc1nc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cs1 ZINC000880657402 EE On-Demand Mild TRPC3 54 40 CNc1nc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cs1 ZINC000880657403 EE On-Demand Mild TRPC6 61 40 CNc1nc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cs1 ZINC000880657403 EE On-Demand Mild TRPC3 54 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(CO)(CO)CC1 ZINC000880657404 EE On-Demand Anodyne CACNA1H 37 44 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(CO)(CO)CC1 ZINC000880657404 EE On-Demand Anodyne S1PR2 32 45 O=C(NCc1ccc(-n2ccnc2)nc1)Nc1ccnn1CC1CCC1 ZINC000880657435 FF On-Demand Anodyne NOS2 98 37 O=C(NCc1ccc(-n2ccnc2)nc1)Nc1ccnn1CC1CCC1 ZINC000880657435 FF On-Demand Anodyne NAMPT 35 54 COC(=O)c1cc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)ccn1 ZINC000880657458 FE On-Demand Mild MAP3K12 31 42 COC(=O)c1cc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)ccn1 ZINC000880657459 FE On-Demand Mild MAP3K12 31 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@H](CO)CC1 ZINC000880657463 EG On-Demand Anodyne CCR3 54 46 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@@H](CO)CC1 ZINC000880657464 EG On-Demand Anodyne CCR3 54 46 CC(C)(C)OC(=O)N1CCC[C@H](C2CCN(C(=O)COC3CC3)CC2)C1 ZINC000880657480 FG On-Demand Anodyne GPR119 24 41 CC(C)(C)OC(=O)N1CCC[C@@H](C2CCN(C(=O)COC3CC3)CC2)C1 ZINC000880657481 FG On-Demand Anodyne GPR119 24 41 C=CCCC[C@H](C(=O)N(C)Cc1cnc[nH]1)c1ccccc1 ZINC000880657558 CH On-Demand Mild TAAR1 23 40 CN(Cc1cnc[nH]1)C(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1 ZINC000880657560 EG On-Demand Anodyne TAAR1 27 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cccc(-n3cnnn3)c2)C1 ZINC000880657561 FD On-Demand Mild KCNJ1 18 43 C[C@@H](CNC(=O)c1ccc(OC(F)F)c(Cl)c1)c1ccccn1 ZINC000880657562 EH On-Demand Anodyne PDE4D 21 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)c1ccccn1)C2 ZINC000880657564 DG On-Demand Anodyne MTNR1A 42 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)c1ccccn1)C2 ZINC000880657564 DG On-Demand Anodyne MTNR1B 38 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](C)c1ccccn1)C2 ZINC000880657564 DG On-Demand Anodyne FAAH 18 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)c1ccccn1)C2 ZINC000880657567 DG On-Demand Anodyne MTNR1A 42 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)c1ccccn1)C2 ZINC000880657567 DG On-Demand Anodyne MTNR1B 38 47 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](C)c1ccccn1)C2 ZINC000880657567 DG On-Demand Anodyne FAAH 18 45 Cn1nnc(C(=O)N2CCC[C@H](C3CCN(C(=O)OC(C)(C)C)CC3)C2)n1 ZINC000880657586 GD On-Demand Anodyne GPR119 30 46 Cn1nnc(C(=O)N2CCC[C@@H](C3CCN(C(=O)OC(C)(C)C)CC3)C2)n1 ZINC000880657588 GD On-Demand Anodyne GPR119 30 46 CC(C)(C)OC(=O)N1CCC([C@@H]2CCCN(C(=O)C[C@@H]3CCNC3=O)C2)CC1 ZINC000880657590 GE On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CCC([C@@H]2CCCN(C(=O)C[C@H]3CCNC3=O)C2)CC1 ZINC000880657591 GE On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CCC([C@H]2CCCN(C(=O)C[C@@H]3CCNC3=O)C2)CC1 ZINC000880657592 GE On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CCC([C@H]2CCCN(C(=O)C[C@H]3CCNC3=O)C2)CC1 ZINC000880657593 GE On-Demand Anodyne GPR119 25 43 C[C@@H](CNC(=O)c1ncsc1C1CC1)c1ccccn1 ZINC000880657607 CF On-Demand Anodyne MAP1 105 37 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(F)c2)C1 ZINC000880657653 DE On-Demand Mild MAP3K12 27 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(F)c2)C1 ZINC000880657655 DE On-Demand Mild MAP3K12 27 41 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657672 GF On-Demand Anodyne ADRB2 36 51 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657672 GF On-Demand Anodyne ADRB1 68 51 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657672 GF On-Demand Anodyne ADRB3 46 41 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657676 GF On-Demand Anodyne ADRB2 36 51 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657676 GF On-Demand Anodyne ADRB1 68 51 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)cc1 ZINC000880657676 GF On-Demand Anodyne ADRB3 46 41 Cn1ncc(Br)c1CC(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880657679 FD On-Demand Anodyne CACNA1I 58 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(C)(C)NS(C)(=O)=O)C1 ZINC000880657680 FC On-Demand Mild CACNA1B 19 42 Cn1ncc(Br)c1CC(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880657681 FD On-Demand Anodyne CACNA1I 58 40 COC1CC(CCNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880657683 CF On-Demand Anodyne SIRT3 46 37 COC1CC(CCNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880657683 CF On-Demand Anodyne SIRT2 55 37 COC1CC(CCNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880657683 CF On-Demand Anodyne SIRT1 47 37 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(C)(C)NS(C)(=O)=O)C1 ZINC000880657688 FC On-Demand Mild CACNA1B 19 42 CC(C)(C)OC(=O)N1CCC([C@H]2CCCN(C(=O)COC3CC3)C2)CC1 ZINC000880657692 FG On-Demand Anodyne GPR119 29 44 CC(C)(C)OC(=O)N1CCC([C@@H]2CCCN(C(=O)COC3CC3)C2)CC1 ZINC000880657693 FG On-Demand Anodyne GPR119 29 44 C=CC[C@@H]1CCCC[C@@H]1NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880657701 EH On-Demand Mild SSTR3 31 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cccc(-n3cnnn3)c2)C1 ZINC000880657702 FD On-Demand Mild KCNJ1 18 43 C=CC[C@@H]1CCCC[C@@H]1NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880657704 EH On-Demand Mild SSTR3 31 44 C=CC[C@@H]1CCCC[C@H]1NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880657706 EH On-Demand Mild SSTR3 31 44 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)COC2CC2)C1 ZINC000880657707 CD On-Demand Mild MLNR 17 41 C=CC[C@@H]1CCCC[C@H]1NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880657708 EH On-Demand Mild SSTR3 31 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)COC2CC2)C1 ZINC000880657709 CD On-Demand Mild MLNR 17 41 CN1CC[C@@H](CNC(=O)Nc2cc(F)cc(OC(F)F)c2)[C@@H]1c1cccnc1 ZINC000880657726 GH On-Demand Anodyne CCR3 56 38 CN(Cc1cnc[nH]1)C(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880657752 CE On-Demand Anodyne TAAR1 22 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccnc(Br)c2)C1 ZINC000880657786 GG On-Demand Mild MAP3K12 26 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccnc(Br)c2)C1 ZINC000880657788 GG On-Demand Mild MAP3K12 26 41 CC[C@H](C)N(CC)C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880657796 DF On-Demand Anodyne PAPA1_CARPA 36 42 CC[C@H](C)N(CC)C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880657796 DF On-Demand Anodyne CTSK 18 49 CC[C@H](C)N(CC)C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880657797 DF On-Demand Anodyne PAPA1_CARPA 36 42 CC[C@H](C)N(CC)C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880657797 DF On-Demand Anodyne CTSK 18 49 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880657804 ED On-Demand Anodyne CACNA1H 36 44 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880657804 ED On-Demand Anodyne S1PR2 30 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@H](CF)C1 ZINC000880657807 DH On-Demand Anodyne CCR3 81 35 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@@H](CF)C1 ZINC000880657808 DH On-Demand Anodyne CCR3 81 35 CCCS(=O)(=O)CC(=O)N1CC[C@H](N(C)c2cccc(C#N)c2)C1 ZINC000880657822 ED On-Demand Mild CCR8 48 33 CCCS(=O)(=O)CC(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1 ZINC000880657823 ED On-Demand Mild CCR8 48 33 CC(=O)[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880657826 EG On-Demand Anodyne CACNA1H 29 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880657827 EG On-Demand Anodyne CACNA1H 29 40 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880657830 FF On-Demand Anodyne GPR119 48 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H](NS(C)(=O)=O)C(C)(C)C)C1 ZINC000880657833 GD On-Demand Mild CACNA1B 18 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H](NS(C)(=O)=O)C(C)(C)C)C1 ZINC000880657834 GD On-Demand Mild CACNA1B 18 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H](NS(C)(=O)=O)C(C)(C)C)C1 ZINC000880657835 GD On-Demand Mild CACNA1B 18 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H](NS(C)(=O)=O)C(C)(C)C)C1 ZINC000880657836 GD On-Demand Mild CACNA1B 18 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cc(C3CC3)[nH]n2)C1 ZINC000880657839 EF On-Demand Mild PKNB 27 44 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cc(C3CC3)[nH]n2)C1 ZINC000880657840 EF On-Demand Mild PKNB 27 44 C#CCN1CCC(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)CC1 ZINC000880657844 FD On-Demand Mild MLNR 15 42 C#CCN1CCC(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)CC1 ZINC000880657845 FD On-Demand Mild MLNR 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880657848 FE On-Demand Anodyne PAPA1_CARPA 36 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880657850 FE On-Demand Anodyne PAPA1_CARPA 36 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880657852 FE On-Demand Anodyne PAPA1_CARPA 36 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880657853 FE On-Demand Anodyne PAPA1_CARPA 36 46 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccnn1CC1CCC1 ZINC000880657856 FF On-Demand Clean NAMPT 44 38 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657866 EG On-Demand Anodyne NQO2 29 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657866 EG On-Demand Anodyne MTNR1A 41 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657866 EG On-Demand Anodyne NPY5R 18 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657866 EG On-Demand Anodyne CACNA1I 45 31 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657869 EG On-Demand Anodyne NQO2 29 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657869 EG On-Demand Anodyne MTNR1A 41 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657869 EG On-Demand Anodyne NPY5R 18 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880657869 EG On-Demand Anodyne CACNA1I 45 31 O=C(NCCS(=O)(=O)Cc1ccccc1)Nc1ccnn1CC1CCC1 ZINC000880657870 GE On-Demand Anodyne CCR3 25 41 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@H](CF)C1 ZINC000880657872 DG On-Demand Anodyne CCR3 44 48 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@H](CF)C1 ZINC000880657874 DG On-Demand Anodyne CCR3 44 48 Cc1ncc(CC(=O)N2CCC[C@H](C3CCN(C(=O)OC(C)(C)C)CC3)C2)o1 ZINC000880657912 GG On-Demand Anodyne GPR119 48 46 Cc1ncc(CC(=O)N2CCC[C@@H](C3CCN(C(=O)OC(C)(C)C)CC3)C2)o1 ZINC000880657914 GG On-Demand Anodyne GPR119 48 46 COC1CC(CCNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880657929 FD On-Demand Anodyne ACHE 23 42 CC(C)(C)N1CC[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880657939 EH On-Demand Anodyne MTNR1A 18 45 CC(C)(C)N1CC[C@@H](CNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880657941 EH On-Demand Anodyne MTNR1A 18 45 CC(C)(C)N1CC[C@H](CNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880657943 EH On-Demand Anodyne MTNR1A 18 45 CC(C)(C)N1CC[C@@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880657945 EH On-Demand Anodyne MTNR1A 18 45 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1ccnn1CC1CCC1 ZINC000880657950 FE On-Demand Anodyne ADRB1 34 44 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1ccnn1CC1CCC1 ZINC000880657952 FE On-Demand Anodyne ADRB1 34 44 CN(C)C(=O)Nc1cccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)c1 ZINC000880657954 GG On-Demand Mild MCHR1 40 43 CN(C)C(=O)Nc1cccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)c1 ZINC000880657956 GG On-Demand Mild MCHR1 40 43 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c1 ZINC000880657962 DF On-Demand Anodyne CACNA1I 79 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CCN2CCOCC2)C1 ZINC000880657964 ED On-Demand Mild CASR 23 43 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c1 ZINC000880657965 DF On-Demand Anodyne CACNA1I 79 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CCN2CCOCC2)C1 ZINC000880657968 ED On-Demand Mild CASR 23 43 COCCc1ccc(OC[C@@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657972 GD On-Demand Anodyne ADRB2 39 56 COCCc1ccc(OC[C@@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657972 GD On-Demand Anodyne ADRB1 68 56 COCCc1ccc(OC[C@@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657972 GD On-Demand Anodyne ADRB3 43 41 COCCc1ccc(OC[C@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657973 GD On-Demand Anodyne ADRB2 39 56 COCCc1ccc(OC[C@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657973 GD On-Demand Anodyne ADRB1 68 56 COCCc1ccc(OC[C@H](O)CNC(=O)c2nccnc2SC)cc1 ZINC000880657973 GD On-Demand Anodyne ADRB3 43 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cccc(C3OCCO3)c2)C1 ZINC000880657974 GF On-Demand Mild HRH3 18 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cccc(C3OCCO3)c2)C1 ZINC000880657974 GF On-Demand Mild L3MBTL3 52 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cccc(C3OCCO3)c2)C1 ZINC000880657976 GF On-Demand Mild HRH3 18 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cccc(C3OCCO3)c2)C1 ZINC000880657976 GF On-Demand Mild L3MBTL3 52 40 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880657995 DE On-Demand Anodyne HTR4 42 35 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880657995 DE On-Demand Anodyne CACNA1I 73 39 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880657997 DE On-Demand Anodyne HTR4 42 35 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880657997 DE On-Demand Anodyne CACNA1I 73 39 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880657999 GE On-Demand Anodyne ADRB2 41 53 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880657999 GE On-Demand Anodyne ADRB1 70 53 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880657999 GE On-Demand Anodyne ADRB3 47 39 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880658000 GE On-Demand Anodyne ADRB2 41 53 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880658000 GE On-Demand Anodyne ADRB1 70 53 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)cnc2Cl)cc1 ZINC000880658000 GE On-Demand Anodyne ADRB3 47 39 CC(C)C1(O)CN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658011 DF On-Demand Anodyne CACNA1H 24 42 CC(C)C1(O)CN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658011 DF On-Demand Anodyne S1PR2 29 42 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)Cn3cnc4ccccc43)sc2C1 ZINC000880658013 HG On-Demand Anodyne SLC27A1 36 40 CC(C)(C)N1CC[C@@H](CNC(=O)[C@H]2CCc3nncn3CC2)C1 ZINC000880658018 DD On-Demand Anodyne CACNA1I 41 32 CC(C)(C)N1CC[C@H](CNC(=O)[C@H]2CCc3nncn3CC2)C1 ZINC000880658019 DD On-Demand Anodyne CACNA1I 41 32 CC(C)(C)N1CC[C@@H](CNC(=O)[C@@H]2CCc3nncn3CC2)C1 ZINC000880658020 DD On-Demand Anodyne CACNA1I 41 32 CC(C)(C)N1CC[C@H](CNC(=O)[C@@H]2CCc3nncn3CC2)C1 ZINC000880658021 DD On-Demand Anodyne CACNA1I 41 32 C#Cc1ccc(C(=O)N2CC[C@H](N(C)c3cccc(C#N)c3)C2)cn1 ZINC000880658031 EE On-Demand Mild L3MBTL3 46 37 C#Cc1ccc(C(=O)N2CC[C@@H](N(C)c3cccc(C#N)c3)C2)cn1 ZINC000880658032 EE On-Demand Mild L3MBTL3 46 37 CC(C)(C)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880658033 EG On-Demand Anodyne EPHX2 44 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2cccnc2Cl)C1 ZINC000880658056 EF On-Demand Mild G2YM83_BOTF4 52 34 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2cccnc2Cl)C1 ZINC000880658057 EF On-Demand Mild G2YM83_BOTF4 52 34 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CNCC(F)(F)F)C1 ZINC000880658060 ED On-Demand Mild MCHR1 44 38 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CNCC(F)(F)F)C1 ZINC000880658061 ED On-Demand Mild MCHR1 44 38 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658066 GG On-Demand Anodyne CACNA1H 30 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N[C@@H]1CC[C@H](O)CC1 ZINC000880658070 DF On-Demand Anodyne EPHX2 48 44 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(F)CC1 ZINC000880658071 DG On-Demand Anodyne CACNA1H 32 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CCCCO2)CC1 ZINC000880658078 FH On-Demand Anodyne CACNA1H 31 41 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(CCCCO2)CC1 ZINC000880658078 FH On-Demand Anodyne S1PR2 28 40 Cc1n[nH]c(C)c1CCC(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1 ZINC000880658079 FF On-Demand Mild HAO2 42 44 Cc1n[nH]c(C)c1CCC(=O)N1CC[C@H](N(C)c2cccc(C#N)c2)C1 ZINC000880658080 FF On-Demand Mild HAO2 42 44 COCC1CC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658094 DF On-Demand Anodyne CCR3 40 42 CN1CCN(C2CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)CC1 ZINC000880658097 GF On-Demand Anodyne CACNA1H 28 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc3n[nH]cc3c2)C1 ZINC000880658101 EF On-Demand Mild FASN 39 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)c2ccc3n[nH]cc3c2)C1 ZINC000880658101 EF On-Demand Mild MAP3K12 29 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc3n[nH]cc3c2)C1 ZINC000880658102 EF On-Demand Mild FASN 39 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)c2ccc3n[nH]cc3c2)C1 ZINC000880658102 EF On-Demand Mild MAP3K12 29 42 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3c(cc2[N+](=O)[O-])OCCCO3)C1 ZINC000880658124 GF On-Demand Bother CACNA1I 43 34 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3c(cc2[N+](=O)[O-])OCCCO3)C1 ZINC000880658125 GF On-Demand Bother CACNA1I 43 34 CC(C)(C)N1CC[C@@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658133 EE On-Demand Anodyne GABRA1 18 46 CC(C)(C)N1CC[C@@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658133 EE On-Demand Anodyne MPO 41 34 CC(C)(C)N1CC[C@@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658133 EE On-Demand Anodyne GABRA2 15 46 CC(C)(C)N1CC[C@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658134 EE On-Demand Anodyne GABRA1 18 46 CC(C)(C)N1CC[C@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658134 EE On-Demand Anodyne MPO 41 34 CC(C)(C)N1CC[C@H]1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880658134 EE On-Demand Anodyne GABRA2 15 46 O=C(CC1CCCC1)NNC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880658135 EG On-Demand Reactive CCR3 50 33 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880658136 GH On-Demand Anodyne PDGFRB 51 44 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880658136 GH On-Demand Anodyne TRPV1 15 47 N#CCCNC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880658138 CE On-Demand Mild ADRB1 42 36 Cn1nc2c(c1C(=O)NC[C@H]1CCN(C(C)(C)C)C1)CSCC2 ZINC000880658140 EE On-Demand Anodyne CACNA1I 44 34 Cn1nc2c(c1C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)CSCC2 ZINC000880658141 EE On-Demand Anodyne CACNA1I 44 34 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658156 FH On-Demand Anodyne CCR3 65 38 Cn1nccc1[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658157 FH On-Demand Anodyne CCR3 65 38 CC(C)(C)N1CC[C@@H]1CNC(=O)c1cnc2cc[nH]c2c1 ZINC000880658160 CE On-Demand Anodyne CACNA1I 62 35 CC(C)(C)N1CC[C@H]1CNC(=O)c1cnc2cc[nH]c2c1 ZINC000880658161 CE On-Demand Anodyne CACNA1I 62 35 CC(C)(C(=O)NC[C@H]1CCN(C(C)(C)C)C1)c1ccc(F)cc1F ZINC000880658169 EG On-Demand Anodyne CACNA1I 50 35 CC(C)(C(=O)NC[C@@H]1CCN(C(C)(C)C)C1)c1ccc(F)cc1F ZINC000880658170 EG On-Demand Anodyne CACNA1I 50 35 COC1CC(CCNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880658185 EG On-Demand Anodyne PDE4D 22 43 COC1CC(CCNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880658185 EG On-Demand Anodyne CACNA1I 42 35 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880658209 GI On-Demand Anodyne EPHX2 24 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880658209 GI On-Demand Anodyne SCD1 23 42 Cn1nccc1CCNC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880658217 EF On-Demand Anodyne CCR3 51 39 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@H](OC2CCC2)CC1 ZINC000880658227 FI On-Demand Anodyne CACNA1H 28 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880658228 FI On-Demand Anodyne CACNA1H 28 40 CC(=O)N(C)CC(=O)N1CC[C@H](N(C)c2cccc(C#N)c2)C1 ZINC000880658230 DD On-Demand Mild MLNR 18 41 CC(=O)N(C)CC(=O)N1CC[C@@H](N(C)c2cccc(C#N)c2)C1 ZINC000880658231 DD On-Demand Mild MLNR 18 41 N#Cc1ccc(N2CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)cn1 ZINC000880658232 GG On-Demand Mild PDGFRB 46 39 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CC(F)(F)F)C1 ZINC000880658261 DF On-Demand Mild MCHR1 44 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CC(F)(F)F)C1 ZINC000880658262 DF On-Demand Mild MCHR1 44 38 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)CSCC(N)=O)C1 ZINC000880658272 EC On-Demand Mild MLNR 15 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)CSCC(N)=O)C1 ZINC000880658273 EC On-Demand Mild MLNR 15 41 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658292 FH On-Demand Anodyne CACNA1H 35 42 CC(=O)C1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658293 EG On-Demand Anodyne CACNA1H 31 44 CC(=O)C1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658293 EG On-Demand Anodyne CCR3 17 41 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658305 CE On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658305 CE On-Demand Mild CACNA1B 19 40 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658305 CE On-Demand Mild SLC9A1 16 41 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658306 CE On-Demand Mild PGR 15 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658306 CE On-Demand Mild CACNA1B 19 40 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)C(F)(F)F)C1 ZINC000880658306 CE On-Demand Mild SLC9A1 16 41 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)c1cn(C)nn1)C2 ZINC000880658330 EC On-Demand Reactive DRD4 40 32 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)cc1 ZINC000880658335 GD On-Demand Anodyne ADRB2 20 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)cc1 ZINC000880658335 GD On-Demand Anodyne ADRB1 47 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)cc1 ZINC000880658336 GD On-Demand Anodyne ADRB2 20 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)cc1 ZINC000880658336 GD On-Demand Anodyne ADRB1 47 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)cc1 ZINC000880658337 GD On-Demand Anodyne ADRB2 20 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)cc1 ZINC000880658337 GD On-Demand Anodyne ADRB1 47 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)cc1 ZINC000880658338 GD On-Demand Anodyne ADRB2 20 46 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)cc1 ZINC000880658338 GD On-Demand Anodyne ADRB1 47 46 CC(C)(C)N1CC[C@@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880658351 ED On-Demand Anodyne HTR4 47 41 CC(C)(C)N1CC[C@@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880658351 ED On-Demand Anodyne CACNA1I 66 39 CC(C)(C)N1CC[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880658352 ED On-Demand Anodyne HTR4 47 41 CC(C)(C)N1CC[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880658352 ED On-Demand Anodyne CACNA1I 66 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1COC(C)(C)C1 ZINC000880658358 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1COC(C)(C)C1 ZINC000880658359 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1COC(C)(C)C1 ZINC000880658360 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1COC(C)(C)C1 ZINC000880658361 ED On-Demand Anodyne PAPA1_CARPA 33 40 O=C(CC[C@@H]1CCc2ccccc21)NCCc1noc2ccccc12 ZINC000880658377 EH On-Demand Anodyne NQO2 16 40 O=C(CC[C@H]1CCc2ccccc21)NCCc1noc2ccccc12 ZINC000880658378 EH On-Demand Anodyne NQO2 16 40 CC(C)(C)N1CC[C@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880658379 ED On-Demand Anodyne CACNA1I 44 34 CC(C)(C)N1CC[C@@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880658380 ED On-Demand Anodyne CACNA1I 44 34 CCOC(=O)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880658432 EE On-Demand Anodyne EPHX2 48 43 CCOC(=O)N1CCC(NC(=O)Nc2ccnn2CC2CCC2)CC1 ZINC000880658432 EE On-Demand Anodyne CCR8 28 42 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@H]2CCCN2S(C)(=O)=O)C1 ZINC000880658456 GD On-Demand Mild WNT3 40 32 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@H]2CCCN2S(C)(=O)=O)C1 ZINC000880658457 GD On-Demand Mild WNT3 40 32 CN(c1cccc(C#N)c1)[C@H]1CCN(C(=O)[C@@H]2CCCN2S(C)(=O)=O)C1 ZINC000880658458 GD On-Demand Mild WNT3 40 32 CN(c1cccc(C#N)c1)[C@@H]1CCN(C(=O)[C@@H]2CCCN2S(C)(=O)=O)C1 ZINC000880658459 GD On-Demand Mild WNT3 40 32 NC(=O)[C@H](F)C1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658488 FE On-Demand Anodyne S1PR2 27 40 NC(=O)[C@@H](F)C1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658489 FE On-Demand Anodyne S1PR2 27 40 O=C(NCCc1cccnc1)Nc1ccnn1CC1CCC1 ZINC000880658496 CE On-Demand Anodyne CHRNA7 45 38 O=C(NCCc1cccnc1)Nc1ccnn1CC1CCC1 ZINC000880658496 CE On-Demand Anodyne NAMPT 46 52 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(F)(F)CC1 ZINC000880658515 DH On-Demand Anodyne CACNA1H 44 48 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(F)(F)CC1 ZINC000880658515 DH On-Demand Anodyne S1PR2 31 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne CTSK 24 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne CTSL 19 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne REN 50 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne CTSS 16 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658598 FE On-Demand Anodyne FPR1 50 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne CTSK 24 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne CTSL 19 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne REN 50 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne CTSS 16 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658599 FE On-Demand Anodyne FPR1 50 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne CTSK 24 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne CTSL 19 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne REN 50 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne CTSS 16 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H](C)c1ccccn1 ZINC000880658600 FE On-Demand Anodyne FPR1 50 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne PAPA1_CARPA 45 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne CTSK 24 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne CTSL 19 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne REN 50 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne CTSS 16 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H](C)c1ccccn1 ZINC000880658601 FE On-Demand Anodyne FPR1 50 39 CC(C)(C)N1CC[C@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880658604 EE On-Demand Anodyne CACNA1I 75 39 CC(C)(C)N1CC[C@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880658605 EE On-Demand Anodyne CACNA1I 75 39 CC(C)(C)N1CC[C@@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880658606 EE On-Demand Anodyne CACNA1I 75 39 CC(C)(C)N1CC[C@@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880658607 EE On-Demand Anodyne CACNA1I 75 39 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(c2cn[nH]c2)CC1 ZINC000880658608 FH On-Demand Anodyne CACNA1H 30 41 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2C(C)(C)C)c1 ZINC000880658620 CF On-Demand Anodyne CACNA1I 66 36 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2C(C)(C)C)c1 ZINC000880658621 CF On-Demand Anodyne CACNA1I 66 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880658630 DE On-Demand Anodyne CACNA1I 40 31 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880658631 DE On-Demand Anodyne CACNA1I 40 31 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880658632 DE On-Demand Anodyne CACNA1I 40 31 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880658633 DE On-Demand Anodyne CACNA1I 40 31 COC1CC(CCNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880658636 GF On-Demand Anodyne Q9NAW4_PLAFA 30 46 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658638 EH On-Demand Anodyne HTR4 55 36 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658638 EH On-Demand Anodyne ACACB 15 42 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658638 EH On-Demand Anodyne CACNA1I 75 38 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658639 EH On-Demand Anodyne HTR4 55 36 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658639 EH On-Demand Anodyne ACACB 15 42 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880658639 EH On-Demand Anodyne CACNA1I 75 38 CS(=O)(=O)C1CCC(C(=O)NCCc2noc3ccccc23)CC1 ZINC000880658640 FE On-Demand Anodyne MTNR1A 22 41 Cn1nnc(C(=O)NC[C@H]2CCN2C(C)(C)C)n1 ZINC000880658643 CB On-Demand Anodyne CACNA1I 45 33 Cn1nnc(C(=O)NC[C@@H]2CCN2C(C)(C)C)n1 ZINC000880658644 CB On-Demand Anodyne CACNA1I 45 33 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880658645 GH On-Demand Anodyne CACNA1H 48 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880658645 GH On-Demand Anodyne OPRL1 17 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880658645 GH On-Demand Anodyne S1PR2 32 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN1C(C)(C)C)C2 ZINC000880658661 EF On-Demand Anodyne NQO2 27 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN1C(C)(C)C)C2 ZINC000880658661 EF On-Demand Anodyne MTNR1A 41 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN1C(C)(C)C)C2 ZINC000880658661 EF On-Demand Anodyne MTNR1B 41 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN1C(C)(C)C)C2 ZINC000880658663 EF On-Demand Anodyne NQO2 27 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN1C(C)(C)C)C2 ZINC000880658663 EF On-Demand Anodyne MTNR1A 41 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN1C(C)(C)C)C2 ZINC000880658663 EF On-Demand Anodyne MTNR1B 41 41 CC(C)(C)N1CC[C@H]1CNC(=O)c1ncccc1-c1ccccn1 ZINC000880658665 DF On-Demand Anodyne HCRTR1 17 40 CC(C)(C)N1CC[C@@H]1CNC(=O)c1ncccc1-c1ccccn1 ZINC000880658666 DF On-Demand Anodyne HCRTR1 17 40 CC(C)(C)N1CC[C@@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880658675 GD On-Demand Anodyne F2 32 42 CC(C)(C)N1CC[C@@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880658675 GD On-Demand Anodyne CACNA1I 41 32 CC(C)(C)N1CC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880658676 GD On-Demand Anodyne F2 32 42 CC(C)(C)N1CC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880658676 GD On-Demand Anodyne CACNA1I 41 32 COC1CC(CCNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880658689 DE On-Demand Anodyne GABRA1 18 47 COC1CC(CCNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880658689 DE On-Demand Anodyne MPO 46 35 COC1CC(CCNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880658689 DE On-Demand Anodyne GABRA2 16 47 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1noc3ccccc13)C2 ZINC000880658701 FG On-Demand Anodyne NQO2 39 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1noc3ccccc13)C2 ZINC000880658701 FG On-Demand Anodyne MTNR1A 93 46 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1noc3ccccc13)C2 ZINC000880658701 FG On-Demand Anodyne MTNR1B 77 43 CC(C)(C)N1CC[C@@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658708 EF On-Demand Anodyne HTR4 36 40 CC(C)(C)N1CC[C@@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658708 EF On-Demand Anodyne CACNA1I 54 36 CC(C)(C)N1CC[C@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658709 EF On-Demand Anodyne HTR4 36 40 CC(C)(C)N1CC[C@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658709 EF On-Demand Anodyne CACNA1I 54 36 COC1CC(CCNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880658710 CE On-Demand Anodyne SIRT3 40 33 COC1CC(CCNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880658710 CE On-Demand Anodyne SIRT1 40 33 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658723 GG On-Demand Anodyne DRD2 26 45 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658723 GG On-Demand Anodyne DRD4 17 45 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658723 GG On-Demand Anodyne DRD3 27 41 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658723 GG On-Demand Anodyne HTR4 51 37 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658723 GG On-Demand Anodyne CACNA1I 49 33 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658724 GG On-Demand Anodyne DRD2 26 45 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658724 GG On-Demand Anodyne DRD4 17 45 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658724 GG On-Demand Anodyne DRD3 27 41 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658724 GG On-Demand Anodyne HTR4 51 37 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880658724 GG On-Demand Anodyne CACNA1I 49 33 CC(C)(C)N1CC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880658732 DE On-Demand Anodyne HTR4 55 38 CC(C)(C)N1CC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880658732 DE On-Demand Anodyne CACNA1I 58 37 CC(C)(C)N1CC[C@@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880658733 DE On-Demand Anodyne HTR4 55 38 CC(C)(C)N1CC[C@@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880658733 DE On-Demand Anodyne CACNA1I 58 37 COC1CC(CCNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880658737 DG On-Demand Anodyne NQO2 24 51 COC1CC(CCNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880658737 DG On-Demand Anodyne MTNR1A 30 43 COC1CC(CCNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880658737 DG On-Demand Anodyne MTNR1B 32 41 COC1CC(CCNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880658738 DG On-Demand Anodyne NQO2 24 51 COC1CC(CCNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880658738 DG On-Demand Anodyne MTNR1A 30 43 COC1CC(CCNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880658738 DG On-Demand Anodyne MTNR1B 32 41 Cc1nc(C(C)C)ncc1C(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880658740 DF On-Demand Anodyne CACNA1I 59 37 Cc1nc(C(C)C)ncc1C(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880658741 DF On-Demand Anodyne CACNA1I 59 37 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880658754 FH On-Demand Anodyne CACNA1H 39 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880658754 FH On-Demand Anodyne CCR3 25 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880658754 FH On-Demand Anodyne S1PR2 24 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880658755 FH On-Demand Anodyne CACNA1H 39 43 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880658755 FH On-Demand Anodyne CCR3 25 40 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880658755 FH On-Demand Anodyne S1PR2 24 40 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658764 FH On-Demand Anodyne CCR3 50 34 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880658765 FH On-Demand Anodyne CCR3 50 34 CC(C)(C)N1CC[C@@H]1CNC(=O)c1cnc(CC2CC2)s1 ZINC000880658767 DF On-Demand Anodyne CACNA1I 42 32 CC(C)(C)N1CC[C@@H]1CNC(=O)c1cnc(CC2CC2)s1 ZINC000880658767 DF On-Demand Anodyne SIRT2 43 32 CC(C)(C)N1CC[C@H]1CNC(=O)c1cnc(CC2CC2)s1 ZINC000880658768 DF On-Demand Anodyne CACNA1I 42 32 CC(C)(C)N1CC[C@H]1CNC(=O)c1cnc(CC2CC2)s1 ZINC000880658768 DF On-Demand Anodyne SIRT2 43 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C(C)(C)C ZINC000880658782 FD On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C(C)(C)C ZINC000880658783 FD On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C(C)(C)C ZINC000880658784 FD On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C(C)(C)C ZINC000880658785 FD On-Demand Anodyne PAPA1_CARPA 37 45 COC1CC(CCNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658786 DF On-Demand Anodyne SIRT3 40 31 COC1CC(CCNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880658786 DF On-Demand Anodyne SIRT1 40 31 CC(C)(C)N1CC[C@H](CNC(=O)C[C@@H]2CCNC2=O)C1 ZINC000880658787 CC On-Demand Anodyne CACNA1I 40 33 CC(C)(C)N1CC[C@@H](CNC(=O)C[C@H]2CCNC2=O)C1 ZINC000880658788 CC On-Demand Anodyne CACNA1I 40 33 CC(C)(C)N1CC[C@@H](CNC(=O)C[C@@H]2CCNC2=O)C1 ZINC000880658789 CC On-Demand Anodyne CACNA1I 40 33 CC(C)(C)N1CC[C@H](CNC(=O)C[C@H]2CCNC2=O)C1 ZINC000880658790 CC On-Demand Anodyne CACNA1I 40 33 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658798 GE On-Demand Anodyne ADRB2 43 51 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658798 GE On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658798 GE On-Demand Anodyne ADRB3 50 42 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658799 GE On-Demand Anodyne ADRB2 43 51 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658799 GE On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccc3nsnc23)cc1 ZINC000880658799 GE On-Demand Anodyne ADRB3 50 42 CC(C)(C)N1CC[C@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658801 DF On-Demand Anodyne HTR4 53 38 CC(C)(C)N1CC[C@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658801 DF On-Demand Anodyne ACACB 15 41 CC(C)(C)N1CC[C@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658801 DF On-Demand Anodyne CACNA1I 54 36 CC(C)(C)N1CC[C@@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658802 DF On-Demand Anodyne HTR4 53 38 CC(C)(C)N1CC[C@@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658802 DF On-Demand Anodyne ACACB 15 41 CC(C)(C)N1CC[C@@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880658802 DF On-Demand Anodyne CACNA1I 54 36 Cn1nnc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)n1 ZINC000880658813 CC On-Demand Anodyne HTR4 41 36 Cn1nnc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)n1 ZINC000880658813 CC On-Demand Anodyne CACNA1I 70 38 Cn1nnc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)n1 ZINC000880658814 CC On-Demand Anodyne HTR4 41 36 Cn1nnc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)n1 ZINC000880658814 CC On-Demand Anodyne CACNA1I 70 38 Cc1coc(C(=O)NC[C@H]2CCN2C(C)(C)C)c1 ZINC000880658828 CE On-Demand Anodyne CACNA1I 57 34 Cc1coc(C(=O)NC[C@@H]2CCN2C(C)(C)C)c1 ZINC000880658829 CE On-Demand Anodyne CACNA1I 57 34 Cc1coc(C(=O)NC[C@H]2CCN(C(C)(C)C)C2)c1 ZINC000880658830 CE On-Demand Anodyne CACNA1I 73 39 Cc1coc(C(=O)NC[C@@H]2CCN(C(C)(C)C)C2)c1 ZINC000880658831 CE On-Demand Anodyne CACNA1I 73 39 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658844 FD On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658844 FD On-Demand Anodyne ADRB1 64 51 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658844 FD On-Demand Anodyne ADRB3 46 38 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658845 FD On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658845 FD On-Demand Anodyne ADRB1 64 51 COCCc1ccc(OC[C@H](O)CNC(=O)c2cccn3nccc23)cc1 ZINC000880658845 FD On-Demand Anodyne ADRB3 46 38 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880658853 GH On-Demand Anodyne HTR4 41 38 CC(C)(C)N1CC[C@H](CNC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880658853 GH On-Demand Anodyne CACNA1I 68 39 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880658854 GH On-Demand Anodyne HTR4 41 38 CC(C)(C)N1CC[C@@H](CNC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880658854 GH On-Demand Anodyne CACNA1I 68 39 CC(C)(C)N1CC[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880658862 EF On-Demand Anodyne GABRA1 16 46 CC(C)(C)N1CC[C@@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880658863 EF On-Demand Anodyne GABRA1 16 46 CC(C)(C)N1CC[C@H](CNC(=O)c2ncsc2C2CC2)C1 ZINC000880658868 DF On-Demand Anodyne CACNA1I 55 34 CC(C)(C)N1CC[C@@H](CNC(=O)c2ncsc2C2CC2)C1 ZINC000880658869 DF On-Demand Anodyne CACNA1I 55 34 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658900 DF On-Demand Anodyne CACNA1I 57 36 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658900 DF On-Demand Anodyne SIRT3 46 35 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658900 DF On-Demand Anodyne SIRT2 45 34 CC(C)(C)N1CC[C@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658900 DF On-Demand Anodyne SIRT1 45 34 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658901 DF On-Demand Anodyne CACNA1I 57 36 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658901 DF On-Demand Anodyne SIRT3 46 35 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658901 DF On-Demand Anodyne SIRT2 45 34 CC(C)(C)N1CC[C@@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880658901 DF On-Demand Anodyne SIRT1 45 34 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C(C)(C)C)c(O)n1 ZINC000880658904 FG On-Demand Anodyne DRD2 33 43 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C(C)(C)C)c(O)n1 ZINC000880658904 FG On-Demand Anodyne KCNA3 40 35 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C(C)(C)C)c(O)n1 ZINC000880658905 FG On-Demand Anodyne DRD2 33 43 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C(C)(C)C)c(O)n1 ZINC000880658905 FG On-Demand Anodyne KCNA3 40 35 O=C1NCC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)O1 ZINC000880658910 FF On-Demand Anodyne CACNA1H 34 43 O=C1NCC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)O1 ZINC000880658910 FF On-Demand Anodyne S1PR2 30 43 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658947 GE On-Demand Anodyne ADRB2 38 54 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658947 GE On-Demand Anodyne ADRB1 58 54 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658947 GE On-Demand Anodyne ADRB3 40 41 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658948 GE On-Demand Anodyne ADRB2 38 54 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658948 GE On-Demand Anodyne ADRB1 58 54 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc(C(C)C)nc2C)cc1 ZINC000880658948 GE On-Demand Anodyne ADRB3 40 41 COC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658967 FF On-Demand Anodyne CCR3 48 40 COC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658967 FF On-Demand Anodyne EPHX2 57 46 COC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880658967 FF On-Demand Anodyne CXCR3 19 48 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658974 GE On-Demand Anodyne ADRB2 30 48 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658974 GE On-Demand Anodyne ADRB1 66 48 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658974 GE On-Demand Anodyne ADRB3 41 38 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658975 GE On-Demand Anodyne ADRB2 30 48 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658975 GE On-Demand Anodyne ADRB1 66 48 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658975 GE On-Demand Anodyne ADRB3 41 38 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658976 GE On-Demand Anodyne ADRB2 30 48 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658976 GE On-Demand Anodyne ADRB1 66 48 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCC(C)(C)CO2)cc1 ZINC000880658976 GE On-Demand Anodyne ADRB3 41 38 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658977 GE On-Demand Anodyne ADRB2 30 48 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658977 GE On-Demand Anodyne ADRB1 66 48 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCC(C)(C)CO2)cc1 ZINC000880658977 GE On-Demand Anodyne ADRB3 41 38 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659003 FD On-Demand Anodyne ADRB2 40 50 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659003 FD On-Demand Anodyne ADRB1 72 50 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659003 FD On-Demand Anodyne ADRB3 50 38 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659004 FD On-Demand Anodyne ADRB2 40 50 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659004 FD On-Demand Anodyne ADRB1 72 50 COCCc1ccc(OC[C@H](O)CNC(=O)c2cnc3cc[nH]c3c2)cc1 ZINC000880659004 FD On-Demand Anodyne ADRB3 50 38 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659028 FC On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659028 FC On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659028 FC On-Demand Anodyne ADRB3 48 40 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659029 FC On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659029 FC On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659029 FC On-Demand Anodyne ADRB3 48 40 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659030 FC On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659030 FC On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@H]2CCNC2=O)cc1 ZINC000880659030 FC On-Demand Anodyne ADRB3 48 40 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659031 FC On-Demand Anodyne ADRB2 38 51 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659031 FC On-Demand Anodyne ADRB1 74 51 COCCc1ccc(OC[C@H](O)CNC(=O)C[C@@H]2CCNC2=O)cc1 ZINC000880659031 FC On-Demand Anodyne ADRB3 48 40 CC(C)(C)N1CC[C@@H](CNC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880659034 EG On-Demand Anodyne CACNA1I 52 45 CC(C)(C)N1CC[C@H](CNC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880659035 EG On-Demand Anodyne CACNA1I 52 45 COC1CC(CCNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880659036 DE On-Demand Anodyne PLD1 45 38 COC1CC(CCNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880659037 DE On-Demand Anodyne PLD1 45 38 CC(C)(C)N1CC[C@H](CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)C1 ZINC000880659043 DG On-Demand Anodyne CACNA1I 41 32 CC(C)(C)N1CC[C@@H](CNC(=O)[C@@H]2C[C@]2(C)c2ccccc2)C1 ZINC000880659044 DG On-Demand Anodyne CACNA1I 41 32 O=C1NC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)CO1 ZINC000880659065 FF On-Demand Anodyne CACNA1H 35 41 O=C1NC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)CO1 ZINC000880659065 FF On-Demand Anodyne S1PR2 29 41 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659070 ED On-Demand Anodyne ADRB2 44 58 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659070 ED On-Demand Anodyne ADRB1 72 58 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659070 ED On-Demand Anodyne ADRB3 46 42 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659071 ED On-Demand Anodyne ADRB2 44 58 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659071 ED On-Demand Anodyne ADRB1 72 58 COCCc1ccc(OC[C@H](O)CNC(=O)c2cc(C)co2)cc1 ZINC000880659071 ED On-Demand Anodyne ADRB3 46 42 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1 ZINC000880659083 FD On-Demand Anodyne ADRB2 26 52 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1 ZINC000880659083 FD On-Demand Anodyne ADRB1 58 52 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1 ZINC000880659084 FD On-Demand Anodyne ADRB2 26 52 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1 ZINC000880659084 FD On-Demand Anodyne ADRB1 58 52 CC(C)(C)N1CC[C@H](CNC(=O)COC2CC2)C1 ZINC000880659085 CD On-Demand Anodyne CACNA1I 47 37 CC(C)(C)N1CC[C@@H](CNC(=O)COC2CC2)C1 ZINC000880659086 CD On-Demand Anodyne CACNA1I 47 37 CC(C)(C)N1CC[C@H](CNC(=O)c2cncc3[nH]ccc23)C1 ZINC000880659088 DE On-Demand Anodyne HTR4 45 36 CC(C)(C)N1CC[C@H](CNC(=O)c2cncc3[nH]ccc23)C1 ZINC000880659088 DE On-Demand Anodyne CACNA1I 53 34 CC(C)(C)N1CC[C@@H](CNC(=O)c2cncc3[nH]ccc23)C1 ZINC000880659089 DE On-Demand Anodyne HTR4 45 36 CC(C)(C)N1CC[C@@H](CNC(=O)c2cncc3[nH]ccc23)C1 ZINC000880659089 DE On-Demand Anodyne CACNA1I 53 34 CC(C)(C)N1CC[C@@H](CNC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880659123 FF On-Demand Anodyne CACNA1I 43 38 CC(C)(C)N1CC[C@H](CNC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880659124 FF On-Demand Anodyne CACNA1I 43 38 O=C(NCCCCCCO)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659148 DG On-Demand Anodyne CCR3 28 40 CC(C)(C)N1CC[C@@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880659169 EE On-Demand Anodyne CACNA1I 52 34 CC(C)(C)N1CC[C@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880659170 EE On-Demand Anodyne CACNA1I 52 34 CC(C)(C)N1CC[C@@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880659171 EE On-Demand Anodyne CACNA1I 52 34 CC(C)(C)N1CC[C@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880659172 EE On-Demand Anodyne CACNA1I 52 34 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC(CCCO)CC1 ZINC000880659179 EG On-Demand Anodyne CCR3 33 42 COCCc1ccc(OC[C@@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659180 GE On-Demand Anodyne ADRB2 42 52 COCCc1ccc(OC[C@@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659180 GE On-Demand Anodyne ADRB1 75 52 COCCc1ccc(OC[C@@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659180 GE On-Demand Anodyne ADRB3 50 41 COCCc1ccc(OC[C@@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659180 GE On-Demand Anodyne MAP1 51 36 COCCc1ccc(OC[C@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659181 GE On-Demand Anodyne ADRB2 42 52 COCCc1ccc(OC[C@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659181 GE On-Demand Anodyne ADRB1 75 52 COCCc1ccc(OC[C@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659181 GE On-Demand Anodyne ADRB3 50 41 COCCc1ccc(OC[C@H](O)CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880659181 GE On-Demand Anodyne MAP1 51 36 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cncc3[nH]ccc23)cc1 ZINC000880659188 FD On-Demand Anodyne ADRB2 33 50 COCCc1ccc(OC[C@@H](O)CNC(=O)c2cncc3[nH]ccc23)cc1 ZINC000880659188 FD On-Demand Anodyne ADRB1 60 50 COCCc1ccc(OC[C@H](O)CNC(=O)c2cncc3[nH]ccc23)cc1 ZINC000880659189 FD On-Demand Anodyne ADRB2 33 50 COCCc1ccc(OC[C@H](O)CNC(=O)c2cncc3[nH]ccc23)cc1 ZINC000880659189 FD On-Demand Anodyne ADRB1 60 50 COc1ccccc1-c1ccc(C(=O)NCCC2CC(OC)C2)c(O)n1 ZINC000880659192 FG On-Demand Anodyne DRD2 18 40 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2CCc3nncn3CC2)cc1 ZINC000880659198 GC On-Demand Anodyne ADRB2 25 47 COCCc1ccc(OC[C@H](O)CNC(=O)[C@H]2CCc3nncn3CC2)cc1 ZINC000880659198 GC On-Demand Anodyne ADRB1 61 47 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2CCc3nncn3CC2)cc1 ZINC000880659199 GC On-Demand Anodyne ADRB2 25 47 COCCc1ccc(OC[C@H](O)CNC(=O)[C@@H]2CCc3nncn3CC2)cc1 ZINC000880659199 GC On-Demand Anodyne ADRB1 61 47 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@H]2CCc3nncn3CC2)cc1 ZINC000880659200 GC On-Demand Anodyne ADRB2 25 47 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@H]2CCc3nncn3CC2)cc1 ZINC000880659200 GC On-Demand Anodyne ADRB1 61 47 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2CCc3nncn3CC2)cc1 ZINC000880659201 GC On-Demand Anodyne ADRB2 25 47 COCCc1ccc(OC[C@@H](O)CNC(=O)[C@@H]2CCc3nncn3CC2)cc1 ZINC000880659201 GC On-Demand Anodyne ADRB1 61 47 O=C(NC[C@@H]1CN2CCC[C@H]2CO1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659216 FE On-Demand Anodyne CCR3 44 35 O=C(NC[C@H]1CN2CCC[C@H]2CO1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659217 FE On-Demand Anodyne CCR3 44 35 O=C(NC[C@H]1CN2CCC[C@@H]2CO1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659218 FE On-Demand Anodyne CCR3 44 35 O=C(NC[C@@H]1CN2CCC[C@@H]2CO1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659219 FE On-Demand Anodyne CCR3 44 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](OC)[C@H]1CCOC1)C2 ZINC000880659234 ED On-Demand Anodyne MTNR1A 34 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](OC)[C@H]1CCOC1)C2 ZINC000880659234 ED On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](OC)[C@@H]1CCOC1)C2 ZINC000880659235 ED On-Demand Anodyne MTNR1A 34 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](OC)[C@@H]1CCOC1)C2 ZINC000880659235 ED On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](OC)[C@@H]1CCOC1)C2 ZINC000880659236 ED On-Demand Anodyne MTNR1A 34 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](OC)[C@@H]1CCOC1)C2 ZINC000880659236 ED On-Demand Anodyne MTNR1B 30 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](OC)[C@H]1CCOC1)C2 ZINC000880659237 ED On-Demand Anodyne MTNR1A 34 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](OC)[C@H]1CCOC1)C2 ZINC000880659237 ED On-Demand Anodyne MTNR1B 30 42 O=C(NCC1CCN(C2CCOCC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880659287 EE On-Demand Anodyne HTR4 55 39 O=C(NCC1CCN(C2CCOCC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880659287 EE On-Demand Anodyne CACNA1I 63 38 O=C(NCC1CCN(C2CCOCC2)CC1)c1coc(-c2ccccn2)n1 ZINC000880659308 FE On-Demand Anodyne HTR4 44 39 O=C(NCC1CCN(C2CCOCC2)CC1)c1cncc2[nH]ccc12 ZINC000880659321 EE On-Demand Anodyne HTR4 62 40 O=C(NCC1CCN(C2CCOCC2)CC1)c1cncc2[nH]ccc12 ZINC000880659321 EE On-Demand Anodyne CACNA1I 44 32 Cc1cnc(Cl)c(C(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880659350 FF On-Demand Anodyne HTR4 55 41 Cc1cnc(Cl)c(C(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880659350 FF On-Demand Anodyne CCR3 17 41 Cc1cnc(Cl)c(C(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880659350 FF On-Demand Anodyne CACNA1I 78 44 C=CC(C)(C)CC(=O)NC[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880659372 DH On-Demand Mild CACNA1I 59 37 C=CC(C)(C)CC(=O)NC[C@H]1CCN(c2ccccc2Cl)C1 ZINC000880659373 DH On-Demand Mild CACNA1I 59 37 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880659383 FF On-Demand Anodyne HTR4 52 42 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880659383 FF On-Demand Anodyne CACNA1I 55 34 O=C(NCC1CCN(C2CCOCC2)CC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880659392 GG On-Demand Anodyne NAMPT 32 40 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@@H]1CCOC1 ZINC000880659400 ED On-Demand Anodyne GABRA1 17 42 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@@H]1CCOC1 ZINC000880659400 ED On-Demand Anodyne GABRA2 15 42 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@H]1CCOC1 ZINC000880659401 ED On-Demand Anodyne GABRA1 17 42 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@H]1CCOC1 ZINC000880659401 ED On-Demand Anodyne GABRA2 15 42 CSCC[C@@H](C)NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659411 DH On-Demand Anodyne CCR3 42 35 CSCC[C@H](C)NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659412 DH On-Demand Anodyne CCR3 42 35 Cn1ccnc1[C@@H](O)[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659413 GG On-Demand Anodyne CCR3 44 33 Cn1ccnc1[C@H](O)[C@@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659414 GG On-Demand Anodyne CCR3 44 33 Cn1ccnc1[C@@H](O)[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659415 GG On-Demand Anodyne CCR3 44 33 Cn1ccnc1[C@H](O)[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659416 GG On-Demand Anodyne CCR3 44 33 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(C4CCOCC4)CC3)cc2)N1 ZINC000880659446 GE On-Demand Anodyne PLD1 40 33 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(C4CCOCC4)CC3)cc2)N1 ZINC000880659446 GE On-Demand Anodyne CACNA1I 62 36 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(C4CCOCC4)CC3)cc2)N1 ZINC000880659447 GE On-Demand Anodyne PLD1 40 33 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(C4CCOCC4)CC3)cc2)N1 ZINC000880659447 GE On-Demand Anodyne CACNA1I 62 36 Cn1nc2c(c1C(=O)NCC1CCN(C3CCOCC3)CC1)CSCC2 ZINC000880659448 GD On-Demand Anodyne CACNA1I 50 33 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(C1)OCCO2 ZINC000880659466 EE On-Demand Anodyne CACNA1H 31 42 O=C(Nc1cc(F)cc(OC(F)F)c1)N1CCC2(C1)OCCO2 ZINC000880659466 EE On-Demand Anodyne S1PR2 27 40 CS(=O)(=O)CC1(CCNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1 ZINC000880659467 FD On-Demand Anodyne PLD1 29 40 CS(=O)(=O)CC1(CCNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1 ZINC000880659467 FD On-Demand Anodyne PLD2 58 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CNC(C)=O)cc1)C2 ZINC000880659468 FF On-Demand Anodyne NQO2 41 49 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CNC(C)=O)cc1)C2 ZINC000880659468 FF On-Demand Anodyne MTNR1A 97 51 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CNC(C)=O)cc1)C2 ZINC000880659468 FF On-Demand Anodyne MTNR1B 92 44 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CNC(C)=O)cc1)C2 ZINC000880659468 FF On-Demand Anodyne CA9 15 40 O=C(Cc1ccccc1N1CCCC1=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880659477 GE On-Demand Anodyne CACNA1I 46 37 C[S@@](=O)CCCNC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659483 DE On-Demand Anodyne CCR3 39 43 O=C(Nc1cccc(CN2CCCS2(=O)=O)c1)c1cnc(CC2CC2)s1 ZINC000880659508 GF On-Demand Anodyne CCR3 23 43 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659514 GH On-Demand Anodyne DRD2 24 45 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659514 GH On-Demand Anodyne DRD3 48 41 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659514 GH On-Demand Anodyne CACNA1I 53 37 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659515 GH On-Demand Anodyne DRD2 24 45 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659515 GH On-Demand Anodyne DRD3 48 41 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659515 GH On-Demand Anodyne CACNA1I 53 37 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659516 GH On-Demand Anodyne DRD2 24 45 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659516 GH On-Demand Anodyne DRD3 48 41 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659516 GH On-Demand Anodyne CACNA1I 53 37 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659517 GH On-Demand Anodyne DRD2 24 45 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659517 GH On-Demand Anodyne DRD3 48 41 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN(c4ccccc4Cl)C3)cc2)N1 ZINC000880659517 GH On-Demand Anodyne CACNA1I 53 37 CCOC(=O)N1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880659524 GG On-Demand Anodyne S1PR2 29 41 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880659525 GG On-Demand Anodyne CCR3 56 42 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880659525 GG On-Demand Anodyne EPHX2 41 37 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880659525 GG On-Demand Anodyne CXCR3 20 48 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880659526 GG On-Demand Anodyne CCR3 56 42 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880659526 GG On-Demand Anodyne EPHX2 41 37 O=C(Nc1cc(F)cc(OC(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880659526 GG On-Demand Anodyne CXCR3 20 48 C=CC(C)(C)CC(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880659540 DF On-Demand Mild CACNA1I 47 36 O=C(NCC1CCN(C2CCOCC2)CC1)c1cnc(CC2CC2)s1 ZINC000880659553 FF On-Demand Anodyne HTR4 36 40 O=C(NCC1CCN(C2CCOCC2)CC1)c1cnc(CC2CC2)s1 ZINC000880659553 FF On-Demand Anodyne CACNA1I 55 37 CC(=O)OC1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880659564 EF On-Demand Anodyne CACNA1H 30 41 CC(C)(C(=O)NCC1CCN(C2CCOCC2)CC1)c1ccc(F)cc1F ZINC000880659574 GG On-Demand Anodyne CACNA1I 64 37 Cc1coc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659580 DG On-Demand Anodyne DRD2 22 42 Cc1coc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659580 DG On-Demand Anodyne DRD4 23 42 Cc1coc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659580 DG On-Demand Anodyne HTR4 44 36 Cc1coc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659580 DG On-Demand Anodyne CACNA1I 64 42 Cc1coc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659581 DG On-Demand Anodyne DRD2 22 42 Cc1coc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659581 DG On-Demand Anodyne DRD4 23 42 Cc1coc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659581 DG On-Demand Anodyne HTR4 44 36 Cc1coc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)c1 ZINC000880659581 DG On-Demand Anodyne CACNA1I 64 42 O=C(NCC1CCN(C2CCOCC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880659597 GE On-Demand Anodyne HTR4 20 42 CS(=O)(=O)CC1(CCNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CC1 ZINC000880659605 FD On-Demand Anodyne MPO 41 34 O=C(NCC1CCN(C2CCOCC2)CC1)c1ncccc1-c1ccccn1 ZINC000880659606 GF On-Demand Anodyne HTR4 54 42 O=C(NCC1CCN(C2CCOCC2)CC1)c1ncccc1-c1ccccn1 ZINC000880659606 GF On-Demand Anodyne CACNA1I 52 33 O=C(NCC1CCN(C2CCOCC2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880659626 GD On-Demand Anodyne HTR4 54 43 O=C(NCC1CCN(C2CCOCC2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880659626 GD On-Demand Anodyne CACNA1I 68 44 Cc1coc(C(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)c1 ZINC000880659634 EH On-Demand Anodyne KCNK3 62 37 Cc1coc(C(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)c1 ZINC000880659634 EH On-Demand Anodyne KCNK9 51 33 N#Cc1cccc([C@@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CCO2)c1 ZINC000880659635 GH On-Demand Mild CACNA1H 25 41 N#Cc1cccc([C@@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CCO2)c1 ZINC000880659635 GH On-Demand Mild CCR3 15 42 N#Cc1cccc([C@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CCO2)c1 ZINC000880659636 GH On-Demand Mild CACNA1H 25 41 N#Cc1cccc([C@H]2CN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CCO2)c1 ZINC000880659636 GH On-Demand Mild CCR3 15 42 C[C@H](C[C@@H](O)c1ccco1)NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659637 FH On-Demand Anodyne CCR3 43 36 C[C@@H](C[C@@H](O)c1ccco1)NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659639 FH On-Demand Anodyne CCR3 43 36 C[C@@H](C[C@H](O)c1ccco1)NC(=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659640 FH On-Demand Anodyne CCR3 43 36 Cc1coc(C(=O)Nc2cccc(CN3CCCS3(=O)=O)c2)c1 ZINC000880659650 EE On-Demand Anodyne CDK1 15 40 Cc1coc(C(=O)Nc2cccc(CN3CCCS3(=O)=O)c2)c1 ZINC000880659650 EE On-Demand Anodyne KCNK3 63 40 Cc1coc(C(=O)Nc2cccc(CN3CCCS3(=O)=O)c2)c1 ZINC000880659650 EE On-Demand Anodyne KCNK9 44 35 O=C(NCC1CCN(C2CCOCC2)CC1)c1cc2ccccc2cc1F ZINC000880659657 FH On-Demand Anodyne HTR4 67 42 O=C(NCC1CCN(C2CCOCC2)CC1)c1cc2ccccc2cc1F ZINC000880659657 FH On-Demand Anodyne CCR3 40 42 O=C(NCC1CCN(C2CCOCC2)CC1)c1cc2ccccc2cc1F ZINC000880659657 FH On-Demand Anodyne CACNA1I 64 35 CS(=O)(=O)CC1(CCNC(=O)CC[C@@H]2CCc3ccccc32)CC1 ZINC000880659697 EF On-Demand Anodyne NQO2 19 42 CS(=O)(=O)CC1(CCNC(=O)CC[C@H]2CCc3ccccc32)CC1 ZINC000880659698 EF On-Demand Anodyne NQO2 19 42 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659725 FF On-Demand Anodyne CACNA1H 36 43 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880659725 FF On-Demand Anodyne S1PR2 29 41 O=C(NCC1CCN(C2CCOCC2)CC1)c1cccc2nsnc12 ZINC000880659750 FE On-Demand Anodyne HTR4 65 40 O=C(NCC1CCN(C2CCOCC2)CC1)c1cccc2nsnc12 ZINC000880659750 FE On-Demand Anodyne CACNA1I 53 33 O=C(NCCS(=O)(=O)CC1CC1)Nc1cc(F)cc(OC(F)F)c1 ZINC000880659770 FE On-Demand Anodyne CCR3 43 42 O=C1CC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)CN1 ZINC000880659780 FF On-Demand Anodyne CACNA1H 34 42 O=C1CC2(CCN(C(=O)Nc3cc(F)cc(OC(F)F)c3)CC2)CN1 ZINC000880659780 FF On-Demand Anodyne S1PR2 29 41 CSc1nccnc1C(=O)Nc1nnc(CCC(C)C)s1 ZINC000880659790 DF On-Demand Anodyne MAP1 85 38 CO[C@H](CNC(=O)CC[C@H]1CCc2ccccc21)[C@@H]1CCOC1 ZINC000880659899 DF On-Demand Anodyne NQO2 19 41 CO[C@H](CNC(=O)CC[C@@H]1CCc2ccccc21)[C@@H]1CCOC1 ZINC000880659900 DF On-Demand Anodyne NQO2 19 41 CO[C@H](CNC(=O)CC[C@H]1CCc2ccccc21)[C@H]1CCOC1 ZINC000880659901 DF On-Demand Anodyne NQO2 19 41 CO[C@H](CNC(=O)CC[C@@H]1CCc2ccccc21)[C@H]1CCOC1 ZINC000880659902 DF On-Demand Anodyne NQO2 19 41 COC[C@@H](CCNC(=O)c1ccc(OC(F)F)c(Cl)c1)OC ZINC000880659943 EF On-Demand Anodyne PDE4D 15 43 COc1ccc(N2CC[C@H](NC(=O)COC3CC3)C2)cc1 ZINC000880659955 CD On-Demand Clean MTNR1A 15 55 COc1ccc(N2CC[C@H](NC(=O)COC3CC3)C2)cc1 ZINC000880659955 CD On-Demand Clean MTNR1B 17 55 COc1ccc(N2CC[C@H](NC(=O)COC3CC3)C2)cc1 ZINC000880659955 CD On-Demand Clean MCHR1 21 44 N#Cc1ccc(CCNC(=O)[C@H]2CCc3nncn3CC2)cc1 ZINC000880659959 DD On-Demand Mild GPBAR1 38 46 N#Cc1ccc(CCNC(=O)[C@@H]2CCc3nncn3CC2)cc1 ZINC000880659960 DD On-Demand Mild GPBAR1 38 46 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean DRD4 20 41 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean EDNRA 22 40 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean SIGMAR1 22 49 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean MTNR1A 15 54 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean MTNR1B 15 54 COc1ccc(N2CC[C@H](NC(=O)CN(C(C)=O)c3ccccc3)C2)cc1 ZINC000880659969 FE On-Demand Clean MCHR1 20 40 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)co3)C2)cc1 ZINC000880659976 DF On-Demand Clean MTNR1A 16 48 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)co3)C2)cc1 ZINC000880659976 DF On-Demand Clean PDK1 41 35 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)co3)C2)cc1 ZINC000880659976 DF On-Demand Clean MCHR1 21 42 CN1CCN(C2CCN(C(=O)Nc3c(F)ccc4c3OCO4)CC2)CC1 ZINC000880659978 FD On-Demand Anodyne L3MBTL3 48 39 O=C(COC1CC1)NC[C@H]1CCN(c2ccccc2Cl)C1 ZINC000880660028 DE On-Demand Anodyne CACNA1I 54 35 O=C(COC1CC1)NC[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880660029 DE On-Demand Anodyne CACNA1I 54 35 O=C(NCC1CCN(C2CCOCC2)CC1)c1cccn2nccc12 ZINC000880660034 ED On-Demand Anodyne HTR4 64 43 O=C(NCC1CCN(C2CCOCC2)CC1)c1cccn2nccc12 ZINC000880660034 ED On-Demand Anodyne CACNA1I 54 35 O=C(NCC1CCN(C2CCOCC2)CC1)c1ncsc1C1CC1 ZINC000880660039 EF On-Demand Anodyne HTR4 33 41 O=C(NCC1CCN(C2CCOCC2)CC1)c1ncsc1C1CC1 ZINC000880660039 EF On-Demand Anodyne CACNA1I 53 33 Cn1nnc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660062 DD On-Demand Anodyne DRD2 27 41 Cn1nnc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660062 DD On-Demand Anodyne DRD3 49 39 Cn1nnc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660062 DD On-Demand Anodyne HTR4 62 39 Cn1nnc(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660062 DD On-Demand Anodyne CACNA1I 73 40 Cn1nnc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660063 DD On-Demand Anodyne DRD2 27 41 Cn1nnc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660063 DD On-Demand Anodyne DRD3 49 39 Cn1nnc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660063 DD On-Demand Anodyne HTR4 62 39 Cn1nnc(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)n1 ZINC000880660063 DD On-Demand Anodyne CACNA1I 73 40 Cn1ncc(Br)c1CC(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880660067 GD On-Demand Anodyne CACNA1I 55 38 O=C(NCC1CCN(C2CCOCC2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880660075 FG On-Demand Anodyne CACNA1I 22 42 Cc1coc(C(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880660092 DE On-Demand Anodyne HTR4 49 38 Cc1coc(C(=O)NCC2CCN(C3CCOCC3)CC2)c1 ZINC000880660092 DE On-Demand Anodyne CACNA1I 67 43 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)CC1 ZINC000880660103 GF On-Demand Anodyne EPHX2 28 40 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCN(c3ccccc3Cl)C2)CC1 ZINC000880660103 GF On-Demand Anodyne CACNA1I 41 32 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)CC1 ZINC000880660104 GF On-Demand Anodyne EPHX2 28 40 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCN(c3ccccc3Cl)C2)CC1 ZINC000880660104 GF On-Demand Anodyne CACNA1I 41 32 O=C(NCCCN1CCOC1=O)Nc1cc(F)cc(OC(F)F)c1 ZINC000880660105 EE On-Demand Anodyne CCR3 38 42 O=C(NCc1cnc(C(F)(F)F)nc1)c1ccc(CN2CCOCC2)o1 ZINC000880660126 FD On-Demand Anodyne NAMPT 38 41 CCOC(=O)N1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880660128 FF On-Demand Anodyne S1PR2 31 43 COc1ccc(N2CC[C@H](NC(=O)Cc3cnc(C)o3)C2)cc1 ZINC000880660146 DD On-Demand Clean MCHR1 20 40 COCC1(NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CCCC1 ZINC000880660154 DF On-Demand Anodyne GABRA1 15 45 COCC1(NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CCCC1 ZINC000880660154 DF On-Demand Anodyne MPO 49 36 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880660171 GD On-Demand Anodyne S1PR2 30 42 Cn1nc2c(c1C(=O)NC[C@H]1CCN(c3ccccc3Cl)C1)CSCC2 ZINC000880660208 GG On-Demand Anodyne CACNA1I 50 36 Cn1nc2c(c1C(=O)NC[C@@H]1CCN(c3ccccc3Cl)C1)CSCC2 ZINC000880660210 GG On-Demand Anodyne CACNA1I 50 36 N#Cc1ccc(CCNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1 ZINC000880660224 CE On-Demand Mild GPBAR1 33 40 CC[C@H]1CCC[C@@]1(C)C(=O)NCCc1ccc(C#N)cc1 ZINC000880660228 CG On-Demand Mild GPBAR1 28 41 CC[C@@H]1CCC[C@@]1(C)C(=O)NCCc1ccc(C#N)cc1 ZINC000880660229 CG On-Demand Mild GPBAR1 28 41 CC[C@H]1CCC[C@]1(C)C(=O)NCCc1ccc(C#N)cc1 ZINC000880660230 CG On-Demand Mild GPBAR1 28 41 CS(=O)(=O)C1CCC(C(=O)NCCc2ccc(C#N)cc2)CC1 ZINC000880660253 ED On-Demand Mild MTNR1A 18 40 CS(=O)(=O)C1CCC(C(=O)NCCc2ccc(C#N)cc2)CC1 ZINC000880660253 ED On-Demand Mild GPBAR1 36 44 O=C(Nc1c(F)ccc2c1OCO2)N[C@@H]1CC[C@H](O)CC1 ZINC000880660282 CD On-Demand Anodyne EPHX2 18 40 COc1ccc(N2CC[C@H](NC(=O)C3CCC(S(C)(=O)=O)CC3)C2)cc1 ZINC000880660314 GD On-Demand Clean MTNR1A 25 46 COc1ccc(N2CC[C@H](NC(=O)C3CCC(S(C)(=O)=O)CC3)C2)cc1 ZINC000880660314 GD On-Demand Clean MTNR1B 22 46 COc1ccc(N2CC[C@H](NC(=O)C3CCC(S(C)(=O)=O)CC3)C2)cc1 ZINC000880660314 GD On-Demand Clean MMP3 40 39 COc1ccc(N2CC[C@H](NC(=O)C3CCC(S(C)(=O)=O)CC3)C2)cc1 ZINC000880660314 GD On-Demand Clean EPHX2 23 49 N#Cc1ccc(CCNC(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)cc1 ZINC000880660325 GD On-Demand Mild GPBAR1 34 43 O=C(Nc1c(F)ccc2c1OCO2)N1CCC2(CCNC2=O)CC1 ZINC000880660329 ED On-Demand Anodyne CACNA1H 45 35 COC[C@@H](CCNC(=O)CC[C@H]1CCc2ccccc21)OC ZINC000880660359 DF On-Demand Anodyne NQO2 22 46 COC[C@@H](CCNC(=O)CC[C@@H]1CCc2ccccc21)OC ZINC000880660360 DF On-Demand Anodyne NQO2 22 46 COc1ccc([C@@H]2CN(C(=O)Nc3c(F)ccc4c3OCO4)CCO2)cc1 ZINC000880660384 FG On-Demand Anodyne EDNRB 50 38 COc1ccc([C@@H]2CN(C(=O)Nc3c(F)ccc4c3OCO4)CCO2)cc1 ZINC000880660384 FG On-Demand Anodyne EDNRA 41 39 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean DRD4 32 46 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean KCNH2 17 46 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean SIGMAR1 22 45 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean SSTR5 45 35 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean MMP13 27 41 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean CCR3 24 41 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean MMP9 17 41 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean PDK1 53 40 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean MMP1 21 41 COc1ccc(N2CC[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)C2)cc1 ZINC000880660397 GE On-Demand Clean MCHR1 39 46 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild NQO2 39 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild CTSK 20 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild CTSL 15 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild MTNR1A 78 45 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild MTNR1B 70 40 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccc(C#N)cc1)C2 ZINC000880660413 EG On-Demand Mild GPBAR1 39 45 Cc1nc(C(C)C)ncc1C(=O)NCCc1ccc(C#N)cc1 ZINC000880660447 DF On-Demand Mild CTSK 34 44 Cc1nc(C(C)C)ncc1C(=O)NCCc1ccc(C#N)cc1 ZINC000880660447 DF On-Demand Mild CTSL 27 48 COCC1(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)CCCC1 ZINC000880660452 DF On-Demand Anodyne MTNR1A 33 41 COCC1(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)CCCC1 ZINC000880660452 DF On-Demand Anodyne MTNR1B 32 41 COCC1(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)CCCC1 ZINC000880660453 DF On-Demand Anodyne MTNR1A 33 41 COCC1(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)CCCC1 ZINC000880660453 DF On-Demand Anodyne MTNR1B 32 41 COc1ccc(N2CC[C@H](NC(=O)CN3CCCCS3(=O)=O)C2)cc1 ZINC000880660489 FC On-Demand Clean MTNR1B 17 49 COC[C@@H](CCNC(=O)c1ncsc1C1CC1)OC ZINC000880660506 CD On-Demand Anodyne MAP1 50 39 Cc1sc(NC(=O)c2ncsc2C2CC2)nc1C(C)C ZINC000880660525 DI On-Demand Anodyne MAP1 89 40 N#Cc1ccc(CCNC(=O)COC2CC2)cc1 ZINC000880660539 BD On-Demand Mild GPBAR1 31 40 COCC1(NC(=O)c2cc(-c3ccc(OC)cc3)on2)CCCC1 ZINC000880660551 EG On-Demand Anodyne PDK1 42 32 COC[C@@H](CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660556 DD On-Demand Anodyne NQO2 33 41 COC[C@@H](CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660556 DD On-Demand Anodyne MTNR1A 51 42 COC[C@@H](CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660556 DD On-Demand Anodyne MTNR1B 44 40 COC[C@@H](CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660557 DD On-Demand Anodyne NQO2 33 41 COC[C@@H](CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660557 DD On-Demand Anodyne MTNR1A 51 42 COC[C@@H](CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1)OC ZINC000880660557 DD On-Demand Anodyne MTNR1B 44 40 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660571 GF On-Demand Clean DRD4 41 33 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660571 GF On-Demand Clean F10 15 45 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660571 GF On-Demand Clean MCHR1 15 41 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660572 GF On-Demand Clean DRD4 41 33 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660572 GF On-Demand Clean F10 15 45 COc1ccc(N2CC[C@H](NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)C2)cc1 ZINC000880660572 GF On-Demand Clean MCHR1 15 41 COC[C@@H](CCNC(=O)c1cc2cc(F)ccc2[nH]c1=O)OC ZINC000880660576 DD On-Demand Anodyne CNR2 36 42 N#Cc1ccc(CCNC(=O)CC[C@@H]2CCc3ccccc32)cc1 ZINC000880660578 DH On-Demand Mild NQO2 16 40 N#Cc1ccc(CCNC(=O)CC[C@H]2CCc3ccccc32)cc1 ZINC000880660579 DH On-Demand Mild NQO2 16 40 N#Cc1ccc(CCNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)cc1 ZINC000880660633 ED On-Demand Mild GPBAR1 37 47 COC[C@@H](CCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)OC ZINC000880660636 GD On-Demand Anodyne PREP 24 41 COC[C@@H](CCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)OC ZINC000880660636 GD On-Demand Anodyne LGMN 56 37 COC[C@@H](CCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)OC ZINC000880660636 GD On-Demand Anodyne GHSR 21 40 COC[C@@H](CCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)OC ZINC000880660636 GD On-Demand Anodyne KLK5 40 36 COC[C@@H](CCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)OC ZINC000880660636 GD On-Demand Anodyne Q9NAW4_PLAFA 40 46 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)cnc3Cl)C2)cc1 ZINC000880660644 EG On-Demand Clean CNR1 15 42 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)cnc3Cl)C2)cc1 ZINC000880660644 EG On-Demand Clean DRD4 44 36 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)cnc3Cl)C2)cc1 ZINC000880660644 EG On-Demand Clean PDK1 41 35 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)cnc3Cl)C2)cc1 ZINC000880660644 EG On-Demand Clean MCHR1 22 43 COc1ccc(N2CC[C@H](NC(=O)c3cc(C)cnc3Cl)C2)cc1 ZINC000880660644 EG On-Demand Clean PARE 57 31 COc1ccc(CN(CCO)C(=O)Nc2c(F)ccc3c2OCO3)cc1 ZINC000880660652 FF On-Demand Anodyne BMP1 80 37 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cc(F)cc(OC(F)F)c2)C1 ZINC000880660670 GG On-Demand Anodyne CCR3 57 41 COC[C@@H](CCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)OC ZINC000880660743 DD On-Demand Anodyne GABRA1 15 47 COc1ccc(N2CC[C@H](NC(=O)Cc3ccccc3N3CCCC3=O)C2)cc1 ZINC000880660754 GF On-Demand Clean F10 22 40 COc1ccc(N2CC[C@H](NC(=O)Cc3ccccc3N3CCCC3=O)C2)cc1 ZINC000880660754 GF On-Demand Clean EDNRA 21 40 COc1ccc(N2CC[C@H](NC(=O)Cc3ccccc3N3CCCC3=O)C2)cc1 ZINC000880660754 GF On-Demand Clean SIGMAR1 19 45 COc1ccc(N2CC[C@H](NC(=O)Cc3ccccc3N3CCCC3=O)C2)cc1 ZINC000880660754 GF On-Demand Clean MTNR1A 15 49 COc1ccc(N2CC[C@H](NC(=O)Cc3ccccc3N3CCCC3=O)C2)cc1 ZINC000880660754 GF On-Demand Clean MTNR1B 15 49 O=C(C(=O)N1CC[C@@H](Cn2ccnn2)C1)c1c[nH]c2cc(F)ccc12 ZINC000880660757 ED On-Demand Anodyne GRIN2B 16 54 O=C(C(=O)N1CC[C@H](Cn2ccnn2)C1)c1c[nH]c2cc(F)ccc12 ZINC000880660758 ED On-Demand Anodyne GRIN2B 16 54 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cnc(C(F)(F)F)nc1)C2 ZINC000880660761 FF On-Demand Anodyne NQO2 31 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cnc(C(F)(F)F)nc1)C2 ZINC000880660761 FF On-Demand Anodyne RAF1 16 41 COc1ccc(N2CC[C@H](NC(=O)c3c[nH]cc3C3CC3)C2)cc1 ZINC000880660787 EF On-Demand Clean HTR1F 44 36 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2c(F)ccc4c2OCO4)C3)c1 ZINC000880660789 GD On-Demand Anodyne P2RX7 21 40 O=C(Nc1c(F)ccc2c1OCO2)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880660790 GE On-Demand Anodyne ETHR 50 35 O=C(Nc1c(F)ccc2c1OCO2)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880660791 GE On-Demand Anodyne ETHR 50 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(COC)CCCC1 ZINC000880660829 ED On-Demand Anodyne PAPA1_CARPA 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(COC)CCCC1 ZINC000880660830 ED On-Demand Anodyne PAPA1_CARPA 34 43 COc1ccc(N2CC[C@H](NC(=O)c3ccc4c(O)ncnc4c3)C2)cc1 ZINC000880660842 FE On-Demand Clean PDE3A 41 38 COc1ccc(N2CC[C@H](NC(=O)c3ccc4c(O)ncnc4c3)C2)cc1 ZINC000880660842 FE On-Demand Clean UTS2R 22 40 COc1ccc(N2CC[C@H](NC(=O)c3ccc4c(O)ncnc4c3)C2)cc1 ZINC000880660842 FE On-Demand Clean PDE3B 45 38 COc1ccc(N2CC[C@H](NC(=O)c3ccc4c(O)ncnc4c3)C2)cc1 ZINC000880660842 FE On-Demand Clean MCHR1 20 42 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880660848 GG On-Demand Anodyne CCR3 61 40 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880660848 GG On-Demand Anodyne EPHX2 57 48 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)cc(OC(F)F)c2)CC1 ZINC000880660848 GG On-Demand Anodyne CXCR3 20 48 COC[C@@H](CCNC(=O)c1cc(-c2ccc(OC)cc2)on1)OC ZINC000880660880 EE On-Demand Anodyne HDAC10 15 44 COC[C@@H](CCNC(=O)c1cc(-c2ccc(OC)cc2)on1)OC ZINC000880660880 EE On-Demand Anodyne PDK1 42 32 N#Cc1ccc(CCNC(=O)c2cnc(CC3CC3)s2)cc1 ZINC000880660910 DF On-Demand Mild CTSK 26 40 N#Cc1ccc(CCNC(=O)c2cnc(CC3CC3)s2)cc1 ZINC000880660910 DF On-Demand Mild CTSL 18 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1c(F)ccc2c1OCO2 ZINC000880660924 GF On-Demand Clean NOS2 46 32 C=CC(C)(C)CC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880660956 EF On-Demand Mild CA1 15 40 COc1ccc(N2CC[C@H](NC(=O)Nc3c(F)ccc4c3OCO4)C2)cc1 ZINC000880660960 FF On-Demand Clean EDNRB 48 41 COc1ccc(N2CC[C@H](NC(=O)Nc3c(F)ccc4c3OCO4)C2)cc1 ZINC000880660960 FF On-Demand Clean EDNRA 37 41 O=C(Nc1c(F)ccc2c1OCO2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880660998 GH On-Demand Anodyne SMO 37 41 O=C(Nc1c(F)ccc2c1OCO2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880660998 GH On-Demand Anodyne ETHR 61 45 O=C(Nc1c(F)ccc2c1OCO2)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880661034 FG On-Demand Anodyne EPHX2 19 44 O=C(Nc1c(F)ccc2c1OCO2)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880661035 FG On-Demand Anodyne EPHX2 19 44 CC(C)(C(=O)N1CCC[C@H](CC#N)C1)c1ccc(C(F)(F)F)cc1 ZINC000880661134 EI On-Demand Mild DPP4 15 42 CC(C)(C(=O)N1CCC[C@@H](CC#N)C1)c1ccc(C(F)(F)F)cc1 ZINC000880661135 EI On-Demand Mild DPP4 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](CC#N)C1 ZINC000880661145 EE On-Demand Mild PAPA1_CARPA 32 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](CC#N)C1 ZINC000880661146 EE On-Demand Mild PAPA1_CARPA 32 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](CC#N)C1 ZINC000880661147 EE On-Demand Mild PAPA1_CARPA 32 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](CC#N)C1 ZINC000880661148 EE On-Demand Mild PAPA1_CARPA 32 42 N#CC[C@@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661150 FF On-Demand Mild CELA1 20 45 N#CC[C@@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661150 FF On-Demand Mild PREP 104 54 N#CC[C@@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661150 FF On-Demand Mild LGMN 77 44 N#CC[C@@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661150 FF On-Demand Mild KLK5 22 41 N#CC[C@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661151 FF On-Demand Mild CELA1 20 45 N#CC[C@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661151 FF On-Demand Mild PREP 104 54 N#CC[C@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661151 FF On-Demand Mild LGMN 77 44 N#CC[C@H]1CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880661151 FF On-Demand Mild KLK5 22 41 CNc1ncc(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661161 FD On-Demand Anodyne USP7 45 38 CNc1ncc(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661161 FD On-Demand Anodyne USP47 57 38 CCNc1nc(C)c(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661182 GF On-Demand Anodyne S1PR4 37 40 CCNc1nc(C)c(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661182 GF On-Demand Anodyne S1PR3 18 40 O=C(Nc1c(F)ccc2c1OCO2)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880661206 FG On-Demand Anodyne EPHX2 23 53 O=C(Nc1c(F)ccc2c1OCO2)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880661207 FG On-Demand Anodyne EPHX2 23 53 O=C(Nc1c(F)ccc2c1OCO2)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880661219 FH On-Demand Anodyne SMO 25 43 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)[C@@H](NC(=O)c3ccccc3)c3ccccc3)sc2C1 ZINC000880661331 JJ On-Demand Anodyne MTTP 47 36 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)[C@H](NC(=O)c3ccccc3)c3ccccc3)sc2C1 ZINC000880661332 JJ On-Demand Anodyne MTTP 47 36 N#CC[C@H]1CCCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880661354 CE On-Demand Mild JAK1 18 41 N#CC[C@@H]1CCCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880661355 CE On-Demand Mild JAK1 18 41 CC(=O)N(CC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1)c1ccccc1 ZINC000880661378 GE On-Demand Anodyne LTA4H 53 40 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880661390 FF On-Demand Anodyne GPR119 32 41 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880661391 FF On-Demand Anodyne GPR119 32 41 O=C(NCc1ccccc1N1CCOCC1)Nc1c(F)ccc2c1OCO2 ZINC000880661451 FF On-Demand Anodyne SCN10A 15 47 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1C[C@H]2C(=O)N(Cc3ccccc3)C(=O)[C@H]2C1 ZINC000880661499 FD On-Demand Anodyne SAP2 35 44 CC(C)(C)OC(=O)CN1CCC(NC(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880661578 GE On-Demand Anodyne MCHR1 16 43 COc1ccc(N2CCN(C(=O)Nc3c(F)ccc4c3OCO4)CC2)cc1F ZINC000880661655 GG On-Demand Clean RBP4 17 41 CN(C(=O)Nc1c(F)ccc2c1OCO2)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880661702 GG On-Demand Anodyne GPR119 42 43 Cc1ccc(-c2nc(C)c(C(=O)N3CCC[C@@H](CC#N)C3)s2)c(F)c1 ZINC000880661756 FI On-Demand Mild HCRTR1 16 41 Cc1ccc(-c2nc(C)c(C(=O)N3CCC[C@H](CC#N)C3)s2)c(F)c1 ZINC000880661757 FI On-Demand Mild HCRTR1 16 41 N#CC[C@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880661782 FD On-Demand Mild PREP 71 40 N#CC[C@@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880661783 FD On-Demand Mild PREP 71 40 O=C(Nc1c(F)ccc2c1OCO2)N[C@H]1CCOC1=O ZINC000880661795 CC On-Demand Anodyne LUXR 78 47 O=C(Nc1c(F)ccc2c1OCO2)N[C@H]1CCOC1=O ZINC000880661795 CC On-Demand Anodyne TRAR 90 43 O=C(Nc1c(F)ccc2c1OCO2)N[C@H]1CCOC1=O ZINC000880661795 CC On-Demand Anodyne LASR 59 40 O=C(Nc1c(F)ccc2c1OCO2)NC12CCC(CC1)C2 ZINC000880661815 CG On-Demand Anodyne EPHX2 25 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)C1CCC1 ZINC000880661816 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)C1CCC1 ZINC000880661816 ED On-Demand Anodyne REN 30 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)C1CCC1 ZINC000880661817 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)C1CCC1 ZINC000880661817 ED On-Demand Anodyne REN 30 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)C1CCC1 ZINC000880661818 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)C1CCC1 ZINC000880661818 ED On-Demand Anodyne REN 30 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)C1CCC1 ZINC000880661819 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)C1CCC1 ZINC000880661819 ED On-Demand Anodyne REN 30 41 O=C(COC1CC1)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880661834 DE On-Demand Anodyne F10 35 55 C=CCNc1ncc(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661839 GE On-Demand Mild USP7 44 38 C=CCNc1ncc(C(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)s1 ZINC000880661839 GE On-Demand Mild USP47 55 38 O=C(Nc1c(F)ccc2c1OCO2)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880661898 GG On-Demand Anodyne TRPM8 29 43 Cc1cc(F)ccc1C[C@@H](C)NC(=O)Cc1c(Br)cnn1C ZINC000880661934 FF On-Demand Anodyne P2RX7 18 45 Cc1cc(F)ccc1C[C@H](C)NC(=O)Cc1c(Br)cnn1C ZINC000880661937 FF On-Demand Anodyne P2RX7 18 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880662031 FH On-Demand Anodyne EPHX2 25 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880662031 FH On-Demand Anodyne TRPM8 31 52 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880662032 FH On-Demand Anodyne EPHX2 25 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880662032 FH On-Demand Anodyne TRPM8 31 52 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880662049 GG On-Demand Anodyne TRPM8 29 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880662050 GG On-Demand Anodyne TRPM8 29 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880662051 GG On-Demand Anodyne TRPM8 29 45 O=C(Nc1c(F)ccc2c1OCO2)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880662052 GG On-Demand Anodyne TRPM8 29 45 O=C(Nc1c(F)ccc2c1OCO2)N1CCc2cc(Cl)nnc2C1 ZINC000880662170 FF On-Demand Anodyne MAPK1 41 36 O=C(Nc1c(F)ccc2c1OCO2)N1CCC2(CCCC2)C1 ZINC000880662211 DG On-Demand Anodyne EPHX2 29 40 CN(C(=O)Nc1c(F)ccc2c1OCO2)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880662232 GG On-Demand Anodyne GPR119 32 42 CN(C(=O)Nc1c(F)ccc2c1OCO2)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880662233 GG On-Demand Anodyne GPR119 32 42 O=C(Nc1c(F)ccc2c1OCO2)N1CCCC[C@H]1c1ccccc1 ZINC000880662246 EI On-Demand Anodyne CPT1A 42 36 O=C(Nc1c(F)ccc2c1OCO2)N1CCCC[C@@H]1c1ccccc1 ZINC000880662247 EI On-Demand Anodyne CPT1A 42 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880662270 FG On-Demand Anodyne F10 29 53 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880662271 FG On-Demand Anodyne F10 29 53 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880662272 FG On-Demand Anodyne F10 29 53 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880662273 FG On-Demand Anodyne F10 29 53 O=C(Nc1ccc(-n2ccccc2=O)cc1F)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880662276 EF On-Demand Anodyne F10 25 51 CC(C)(C)N1CC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880662286 EE On-Demand Anodyne GABRA1 18 42 CC(C)(C)N1CC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880662286 EE On-Demand Anodyne GABRA2 16 42 CC(C)(C)N1CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880662287 EE On-Demand Anodyne GABRA1 18 42 CC(C)(C)N1CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880662287 EE On-Demand Anodyne GABRA2 16 42 COC[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1CCOCC1 ZINC000880662295 FG On-Demand Anodyne PDE4D 25 44 COC[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1CCOCC1 ZINC000880662296 FG On-Demand Anodyne PDE4D 25 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880662328 EF On-Demand Anodyne MMP3 31 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)(C)C)C1)C2 ZINC000880662328 EF On-Demand Anodyne MMP8 18 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880662330 EF On-Demand Anodyne MMP3 31 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(C(C)(C)C)C1)C2 ZINC000880662330 EF On-Demand Anodyne MMP8 18 41 O=C(CC[C@H]1CCc2ccccc21)NCC[S@@](=O)CC(F)(F)F ZINC000880662339 EF On-Demand Anodyne NQO2 20 40 O=C(CC[C@H]1CCc2ccccc21)NCC[S@@](=O)CC(F)(F)F ZINC000880662339 EF On-Demand Anodyne MTNR1B 15 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[S@](=O)CC(F)(F)F ZINC000880662340 EF On-Demand Anodyne NQO2 20 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[S@](=O)CC(F)(F)F ZINC000880662340 EF On-Demand Anodyne MTNR1B 15 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[S@@](=O)CC(F)(F)F ZINC000880662341 EF On-Demand Anodyne NQO2 20 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[S@@](=O)CC(F)(F)F ZINC000880662341 EF On-Demand Anodyne MTNR1B 15 40 O=C(NCCc1ccc(C2CCCCC2)cc1)[C@H]1CCc2nncn2CC1 ZINC000880662357 FH On-Demand Anodyne GPBAR1 23 40 O=C(NCCc1ccc(C2CCCCC2)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880662358 FH On-Demand Anodyne GPBAR1 23 40 O=C(CC[C@H]1CCc2ccccc21)NCC[S@](=O)CC(F)(F)F ZINC000880662442 EF On-Demand Anodyne NQO2 20 40 O=C(CC[C@H]1CCc2ccccc21)NCC[S@](=O)CC(F)(F)F ZINC000880662442 EF On-Demand Anodyne MTNR1B 15 40 O=C(NCC[S@](=O)CC(F)(F)F)c1cc2cc(F)ccc2[nH]c1=O ZINC000880662472 FD On-Demand Anodyne PLD1 27 40 O=C(NCC[S@](=O)CC(F)(F)F)c1cc2cc(F)ccc2[nH]c1=O ZINC000880662472 FD On-Demand Anodyne PLD2 55 40 O=C(NCC[S@@](=O)CC(F)(F)F)c1cc2cc(F)ccc2[nH]c1=O ZINC000880662473 FD On-Demand Anodyne PLD1 27 40 O=C(NCC[S@@](=O)CC(F)(F)F)c1cc2cc(F)ccc2[nH]c1=O ZINC000880662473 FD On-Demand Anodyne PLD2 55 40 COc1ccc2c(c1)CC[C@H](C(=O)NCC[S@@](=O)CC(F)(F)F)C2 ZINC000880662475 FE On-Demand Anodyne NQO2 33 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[S@@](=O)CC(F)(F)F)C2 ZINC000880662475 FE On-Demand Anodyne MTNR1A 42 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[S@](=O)CC(F)(F)F)C2 ZINC000880662476 FE On-Demand Anodyne NQO2 33 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[S@](=O)CC(F)(F)F)C2 ZINC000880662476 FE On-Demand Anodyne MTNR1A 42 41 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CCC(c2ccco2)CC1 ZINC000880662565 FG On-Demand Bother L3MBTL3 15 42 CC(C)(C)N1CC[C@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880662567 FD On-Demand Anodyne DRD4 23 42 CC(C)(C)N1CC[C@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880662567 FD On-Demand Anodyne SIGMAR1 21 42 CC(C)(C)N1CC[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880662569 FD On-Demand Anodyne DRD4 23 42 CC(C)(C)N1CC[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880662569 FD On-Demand Anodyne SIGMAR1 21 42 CC(C)(C)N1CC[C@H](NC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880662577 ED On-Demand Anodyne DRD4 21 40 CC(C)(C)N1CC[C@H](NC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880662577 ED On-Demand Anodyne MCHR1 33 40 CC(C)(C)N1CC[C@@H](NC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880662579 ED On-Demand Anodyne DRD4 21 40 CC(C)(C)N1CC[C@@H](NC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880662579 ED On-Demand Anodyne MCHR1 33 40 Cc1cc(F)ccc1C[C@@H](C)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880662727 FG On-Demand Anodyne PLD1 57 42 Cc1cc(F)ccc1C[C@H](C)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880662728 FG On-Demand Anodyne PLD1 57 42 Cc1cc(F)ccc1C[C@@H](C)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880662729 FG On-Demand Anodyne PLD1 57 42 Cc1cc(F)ccc1C[C@H](C)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880662731 FG On-Demand Anodyne PLD1 57 42 O=C(Nc1ccc(-n2ccccc2=O)cc1F)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880662807 GE On-Demand Anodyne F10 30 54 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(c4ccco4)CC3)cc2)N1 ZINC000880662811 EG On-Demand Anodyne L3MBTL3 54 36 O=C1CC[C@H](c2ccc(C(=O)N3CCC(c4ccco4)CC3)cc2)N1 ZINC000880662812 EG On-Demand Anodyne L3MBTL3 54 36 O=C(Nc1c(F)ccc2c1OCO2)N1CCCC2(CCCC2)C1 ZINC000880662832 DH On-Demand Anodyne EPHX2 25 40 O=C(Nc1ccc(-n2ccccc2=O)cc1F)[C@@H]1CCc2nncn2CC1 ZINC000880662835 FE On-Demand Anodyne F10 29 53 O=C(Nc1ccc(-n2ccccc2=O)cc1F)[C@H]1CCc2nncn2CC1 ZINC000880662836 FE On-Demand Anodyne F10 29 53 CC(C)(C)N1CC[C@H](NC(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880662955 ED On-Demand Anodyne EPHX2 19 42 CC(C)(C)N1CC[C@@H](NC(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880662956 ED On-Demand Anodyne EPHX2 19 42 O=C(NCC[S@](=O)CC(F)(F)F)c1ccc(CN2CCOCC2)o1 ZINC000880662997 FD On-Demand Anodyne EPHX2 15 42 O=C(NCC[S@@](=O)CC(F)(F)F)c1ccc(CN2CCOCC2)o1 ZINC000880662998 FD On-Demand Anodyne EPHX2 15 42 CC(C)(C)N1CC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880663005 CD On-Demand Anodyne DRD4 16 41 CC(C)(C)N1CC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880663006 CD On-Demand Anodyne DRD4 16 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H](CO)C1CCC1 ZINC000880663041 DD On-Demand Anodyne KCNQ2 52 34 C[C@@H]1C[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)c2ncnn21 ZINC000880663063 EF On-Demand Anodyne PDE4D 18 42 C[C@H]1C[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)c2ncnn21 ZINC000880663064 EF On-Demand Anodyne PDE4D 18 42 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1c(F)ccc2c1OCO2 ZINC000880663084 GE On-Demand Anodyne EPHX2 15 45 O=C(Cc1ccccc1N1CCCC1=O)N[C@H](CO)C1CCC1 ZINC000880663104 DD On-Demand Anodyne KCNQ2 52 34 COc1ccccc1-c1ccc(C(=O)N[C@@H](CO)C2CCC2)c(O)n1 ZINC000880663105 EE On-Demand Anodyne NTSR2 18 42 COc1ccccc1-c1ccc(C(=O)N[C@H](CO)C2CCC2)c(O)n1 ZINC000880663106 EE On-Demand Anodyne NTSR2 18 42 COC[C@@H](NC(=O)c1cc2ccccc2cc1F)C1CCOCC1 ZINC000880663206 EG On-Demand Anodyne PYGL 29 43 COC[C@H](NC(=O)c1cc2ccccc2cc1F)C1CCOCC1 ZINC000880663207 EG On-Demand Anodyne PYGL 29 43 COC(=O)N1CCC(NC(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880663210 ED On-Demand Anodyne EPHX2 41 40 O=C(c1cnc(CC2CC2)s1)N1CCC(c2ccco2)CC1 ZINC000880663227 DH On-Demand Anodyne RBP4 18 40 O=C(N[C@H](CO)C1CCC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880663228 DF On-Demand Anodyne PDE4D 22 45 O=C(N[C@@H](CO)C1CCC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880663229 DF On-Demand Anodyne PDE4D 22 45 CC[C@@H](C(=O)Nc1ccc(OCCS(C)(=O)=O)cc1)[C@@H](C)O ZINC000880663230 ED On-Demand Anodyne CA12 16 43 CC[C@@H](C(=O)Nc1ccc(OCCS(C)(=O)=O)cc1)[C@@H](C)O ZINC000880663230 ED On-Demand Anodyne CA9 16 43 CC[C@@H](C(=O)Nc1ccc(OCCS(C)(=O)=O)cc1)[C@H](C)O ZINC000880663233 ED On-Demand Anodyne CA12 16 43 CC[C@@H](C(=O)Nc1ccc(OCCS(C)(=O)=O)cc1)[C@H](C)O ZINC000880663233 ED On-Demand Anodyne CA9 16 43 CN1CCCC[C@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663238 FE On-Demand Anodyne HRH3 22 41 CN1CCCC[C@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663238 FE On-Demand Anodyne EPHX2 21 41 CN1CCCC[C@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663238 FE On-Demand Anodyne CHRNA10 57 37 CN1CCCC[C@@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663239 FE On-Demand Anodyne HRH3 22 41 CN1CCCC[C@@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663239 FE On-Demand Anodyne EPHX2 21 41 CN1CCCC[C@@H]1CCC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663239 FE On-Demand Anodyne CHRNA10 57 37 O=C(N[C@@H](CO)C1CCC1)c1cc2ccccc2cc1F ZINC000880663241 CF On-Demand Anodyne PYGL 26 42 O=C(N[C@H](CO)C1CCC1)c1cc2ccccc2cc1F ZINC000880663242 CF On-Demand Anodyne PYGL 26 42 CS(=O)(=O)C1CCC(C(=O)Nc2ccc(-n3ccccc3=O)cc2F)CC1 ZINC000880663252 GF On-Demand Anodyne F10 39 59 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(c2ccco2)CC1 ZINC000880663264 GJ On-Demand Anodyne RBP4 47 48 O=C(CN1CCCCS1(=O)=O)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880663268 GD On-Demand Anodyne F10 28 51 O=C(C[C@@H]1C[C@H]1C1CC1)Nc1ccc(-n2ccccc2=O)cc1F ZINC000880663304 EG On-Demand Anodyne F10 27 55 CC(C)(C)N1CC[C@@H](NC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880663328 GH On-Demand Anodyne DRD4 17 42 CC(C)(C)N1CC[C@@H](NC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880663328 GH On-Demand Anodyne SFRP1 72 32 CC(C)(C)N1CC[C@H](NC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880663329 GH On-Demand Anodyne DRD4 17 42 CC(C)(C)N1CC[C@H](NC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880663329 GH On-Demand Anodyne SFRP1 72 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccco2)CC1 ZINC000880663330 FF On-Demand Anodyne P2RY12 97 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccco2)CC1 ZINC000880663331 FF On-Demand Anodyne P2RY12 97 35 O=C(Nc1c(F)ccc2c1OCO2)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880663339 GG On-Demand Anodyne CACNA1H 48 35 CC(C)(C)N1CC[C@@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880663359 CE On-Demand Anodyne SSTR5 45 36 CC(C)(C)N1CC[C@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880663360 CE On-Demand Anodyne SSTR5 45 36 Cc1cc([C@@H]2CCCN2C(=O)Nc2c(F)ccc3c2OCO3)no1 ZINC000880663384 EG On-Demand Anodyne TRPC6 47 36 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880663385 FG On-Demand Anodyne DRD2 23 40 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C(C)(C)C)C2)c(O)n1 ZINC000880663386 FG On-Demand Anodyne DRD2 23 40 COC[C@H](NC(=O)c1cc(-c2ccc(OC)cc2)on1)C1CCOCC1 ZINC000880663397 FF On-Demand Anodyne PDK1 43 32 COC[C@@H](NC(=O)c1cc(-c2ccc(OC)cc2)on1)C1CCOCC1 ZINC000880663398 FF On-Demand Anodyne PDK1 43 32 C#CCC(CC#C)C(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880663399 ED On-Demand Mild CA1 18 40 O=C(c1cccn2nccc12)N1CCC(c2ccco2)CC1 ZINC000880663404 CF On-Demand Anodyne RBP4 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCN(C(C)(C)C)C1 ZINC000880663408 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCN(C(C)(C)C)C1 ZINC000880663409 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCN(C(C)(C)C)C1 ZINC000880663410 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCN(C(C)(C)C)C1 ZINC000880663411 FD On-Demand Anodyne PAPA1_CARPA 35 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H](CO)C2CCC2)N1Cc1ccccc1 ZINC000880663426 EC On-Demand Anodyne XIAP 49 34 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H](CO)C2CCC2)N1Cc1ccccc1 ZINC000880663427 EC On-Demand Anodyne XIAP 49 34 O=C(N[C@@H](CO)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663440 DD On-Demand Anodyne GABRA1 16 43 O=C(N[C@@H](CO)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663440 DD On-Demand Anodyne GABRA2 15 43 O=C(N[C@H](CO)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663441 DD On-Demand Anodyne GABRA1 16 43 O=C(N[C@H](CO)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663441 DD On-Demand Anodyne GABRA2 15 43 O=C1CC[C@@H](c2ccc(C(=O)NCC[S@@](=O)CC(F)(F)F)cc2)N1 ZINC000880663467 FD On-Demand Anodyne PLD1 40 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[S@@](=O)CC(F)(F)F)cc2)N1 ZINC000880663467 FD On-Demand Anodyne PLD2 50 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[S@](=O)CC(F)(F)F)cc2)N1 ZINC000880663468 FD On-Demand Anodyne PLD1 40 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[S@](=O)CC(F)(F)F)cc2)N1 ZINC000880663468 FD On-Demand Anodyne PLD2 50 33 O=C1CC[C@H](c2ccc(C(=O)NCC[S@@](=O)CC(F)(F)F)cc2)N1 ZINC000880663469 FD On-Demand Anodyne PLD1 40 33 O=C1CC[C@H](c2ccc(C(=O)NCC[S@@](=O)CC(F)(F)F)cc2)N1 ZINC000880663469 FD On-Demand Anodyne PLD2 50 33 O=C1CC[C@H](c2ccc(C(=O)NCC[S@](=O)CC(F)(F)F)cc2)N1 ZINC000880663470 FD On-Demand Anodyne PLD1 40 33 O=C1CC[C@H](c2ccc(C(=O)NCC[S@](=O)CC(F)(F)F)cc2)N1 ZINC000880663470 FD On-Demand Anodyne PLD2 50 33 O=C(Nc1c(F)ccc2c1OCO2)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880663495 GG On-Demand Anodyne EPHX2 16 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663527 GG On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663527 GG On-Demand Anodyne CTSK 15 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663527 GG On-Demand Anodyne CTSL 16 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663527 GG On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663527 GG On-Demand Anodyne FPR1 51 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663528 GG On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663528 GG On-Demand Anodyne CTSK 15 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663528 GG On-Demand Anodyne CTSL 16 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663528 GG On-Demand Anodyne POLG_HCV1 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)Cc1ccc(F)cc1C ZINC000880663528 GG On-Demand Anodyne FPR1 51 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663529 GG On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663529 GG On-Demand Anodyne CTSK 15 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663529 GG On-Demand Anodyne CTSL 16 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663529 GG On-Demand Anodyne POLG_HCV1 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663529 GG On-Demand Anodyne FPR1 51 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663530 GG On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663530 GG On-Demand Anodyne CTSK 15 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663530 GG On-Demand Anodyne CTSL 16 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663530 GG On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)Cc1ccc(F)cc1C ZINC000880663530 GG On-Demand Anodyne FPR1 51 39 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663550 GF On-Demand Anodyne CACNA1I 57 35 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663550 GF On-Demand Anodyne GPR119 38 43 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663551 GF On-Demand Anodyne CACNA1I 57 35 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663551 GF On-Demand Anodyne GPR119 38 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne ACE 26 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne PGC 46 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne CCKAR 26 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne CTSL 19 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne PYGL 34 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne PYGM 29 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663606 GD On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne ACE 26 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne PGC 46 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne CCKAR 26 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne CTSL 19 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne PYGL 34 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne PYGM 29 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663607 GD On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne ACE 26 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne PGC 46 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne CCKAR 26 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne CTSL 19 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne PYGL 34 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne PYGM 29 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663608 GD On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne ACE 26 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne PGC 46 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne CCKAR 26 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne CTSL 19 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne PYGL 34 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne PYGM 29 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663609 GD On-Demand Anodyne FPR1 45 36 O=C(NCc1cccnc1N1CCCC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880663611 GH On-Demand Anodyne SCN2A 19 45 O=C(NCc1cccnc1N1CCCC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880663611 GH On-Demand Anodyne SCN10A 20 45 C=CC(C)(C)CC(=O)NCc1cccnc1N1CCCC1 ZINC000880663613 CF On-Demand Mild TRPV1 18 40 C=CC(C)(C)CC(=O)NCc1cccnc1N1CCCC1 ZINC000880663613 CF On-Demand Mild SCN2A 18 45 C=CC(C)(C)CC(=O)NCc1cccnc1N1CCCC1 ZINC000880663613 CF On-Demand Mild SCN10A 20 45 O=C(NCc1cccnc1N1CCCC1)c1cccn2nccc12 ZINC000880663619 DE On-Demand Anodyne SCN2A 21 51 O=C(NCc1cccnc1N1CCCC1)c1cccn2nccc12 ZINC000880663619 DE On-Demand Anodyne SCN10A 33 51 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1cccnc1N1CCCC1 ZINC000880663628 EE On-Demand Anodyne SCN10A 18 43 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1cccnc1N1CCCC1 ZINC000880663629 EE On-Demand Anodyne SCN10A 18 43 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1cccnc1N1CCCC1 ZINC000880663630 EE On-Demand Anodyne SCN10A 18 43 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1cccnc1N1CCCC1 ZINC000880663631 EE On-Demand Anodyne SCN10A 18 43 O=C(NCc1cccnc1N1CCCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663637 FF On-Demand Anodyne SCN2A 18 43 O=C(NCc1cccnc1N1CCCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880663637 FF On-Demand Anodyne SCN10A 19 43 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2c(F)ccc3c2OCO3)c1 ZINC000880663640 FH On-Demand Mild PDS 40 35 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2c(F)ccc3c2OCO3)c1 ZINC000880663641 FH On-Demand Mild PDS 40 35 O=C(NCc1cccnc1N1CCCC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880663651 FG On-Demand Anodyne SCN2A 18 43 O=C(NCc1cccnc1N1CCCC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880663651 FG On-Demand Anodyne SCN10A 23 43 COc1ccc(N2CCC(NC(=O)Nc3c(F)ccc4c3OCO4)CC2)cc1 ZINC000880663655 GG On-Demand Clean EDNRB 48 39 COc1ccc(N2CCC(NC(=O)Nc3c(F)ccc4c3OCO4)CC2)cc1 ZINC000880663655 GG On-Demand Clean EPHX2 40 37 COc1ccc(N2CCC(NC(=O)Nc3c(F)ccc4c3OCO4)CC2)cc1 ZINC000880663655 GG On-Demand Clean MCHR1 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne PGC 52 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne PAPA1_CARPA 42 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne CTSK 15 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne CTSL 16 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne SCN2A 18 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne REN 69 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne SCN10A 40 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663666 GE On-Demand Anodyne FPR1 49 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne PGC 52 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne PAPA1_CARPA 42 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne CTSK 15 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne CTSL 16 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne SCN2A 18 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne REN 69 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne SCN10A 40 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663667 GE On-Demand Anodyne FPR1 49 38 O=C(NCc1cccnc1N1CCCC1)c1ccc(CN2CCOCC2)o1 ZINC000880663789 FE On-Demand Anodyne SCN2A 19 46 O=C(NCc1cccnc1N1CCCC1)c1ccc(CN2CCOCC2)o1 ZINC000880663789 FE On-Demand Anodyne SCN10A 26 49 O=C(NCc1cccnc1N1CCCC1)c1ccc(CN2CCOCC2)o1 ZINC000880663789 FE On-Demand Anodyne NAMPT 28 40 CC1(C)CC[C@@H](CC(=O)NCc2cccnc2N2CCCC2)OC1 ZINC000880663796 EF On-Demand Anodyne SCN2A 17 42 CC1(C)CC[C@@H](CC(=O)NCc2cccnc2N2CCCC2)OC1 ZINC000880663796 EF On-Demand Anodyne SCN10A 19 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc2c1ccn2C(F)F ZINC000880663831 GH On-Demand Anodyne FPR1 40 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc2c1ccn2C(F)F ZINC000880663832 GH On-Demand Anodyne FPR1 40 33 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne SCN2A 20 49 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne SCN10A 27 49 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne SIRT3 57 35 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne SIRT2 54 35 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne SIRT1 46 35 O=C(NCc1cccnc1N1CCCC1)c1cnc(CC2CC2)s1 ZINC000880663837 EG On-Demand Anodyne NAMPT 24 43 O=C(NCc1cccnc1N1CCCC1)[C@H]1CCc2nncn2CC1 ZINC000880663838 ED On-Demand Anodyne P2RX7 27 44 O=C(NCc1cccnc1N1CCCC1)[C@H]1CCc2nncn2CC1 ZINC000880663838 ED On-Demand Anodyne SCN2A 19 45 O=C(NCc1cccnc1N1CCCC1)[C@H]1CCc2nncn2CC1 ZINC000880663838 ED On-Demand Anodyne EPHX2 17 41 O=C(NCc1cccnc1N1CCCC1)[C@H]1CCc2nncn2CC1 ZINC000880663838 ED On-Demand Anodyne SCN10A 20 45 O=C(NCc1cccnc1N1CCCC1)[C@@H]1CCc2nncn2CC1 ZINC000880663839 ED On-Demand Anodyne P2RX7 27 44 O=C(NCc1cccnc1N1CCCC1)[C@@H]1CCc2nncn2CC1 ZINC000880663839 ED On-Demand Anodyne SCN2A 19 45 O=C(NCc1cccnc1N1CCCC1)[C@@H]1CCc2nncn2CC1 ZINC000880663839 ED On-Demand Anodyne EPHX2 17 41 O=C(NCc1cccnc1N1CCCC1)[C@@H]1CCc2nncn2CC1 ZINC000880663839 ED On-Demand Anodyne SCN10A 20 45 O=C(Nc1c(F)ccc2c1OCO2)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880663855 FE On-Demand Anodyne MCHR1 15 41 O=C(Nc1c(F)ccc2c1OCO2)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880663856 FE On-Demand Anodyne MCHR1 15 41 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663877 GF On-Demand Anodyne CACNA1I 45 34 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2c(F)ccc3c2OCO3)C1 ZINC000880663878 GF On-Demand Anodyne CACNA1I 45 34 O=C(COC1CC1)NCc1cccnc1N1CCCC1 ZINC000880663886 CD On-Demand Anodyne SCN2A 19 46 O=C(COC1CC1)NCc1cccnc1N1CCCC1 ZINC000880663886 CD On-Demand Anodyne SCN10A 23 48 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1c(F)ccc2c1OCO2 ZINC000880663891 FF On-Demand Clean STAT6 50 34 C=CC(C)(C)CC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663893 CE On-Demand Mild PYGL 35 49 C=CC(C)(C)CC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880663893 CE On-Demand Mild PYGM 31 49 C=CC(C)(C)CC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663894 CE On-Demand Mild PYGL 35 49 C=CC(C)(C)CC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880663894 CE On-Demand Mild PYGM 31 49 CC[C@H]1CCC[C@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663911 DH On-Demand Anodyne SCN2A 18 44 CC[C@H]1CCC[C@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663911 DH On-Demand Anodyne SCN10A 21 44 CC[C@H]1CCC[C@@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663912 DH On-Demand Anodyne SCN2A 18 44 CC[C@H]1CCC[C@@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663912 DH On-Demand Anodyne SCN10A 21 44 CC[C@@H]1CCC[C@@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663913 DH On-Demand Anodyne SCN2A 18 44 CC[C@@H]1CCC[C@@]1(C)C(=O)NCc1cccnc1N1CCCC1 ZINC000880663913 DH On-Demand Anodyne SCN10A 21 44 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880663941 GG On-Demand Anodyne RBP4 73 35 O=C(NCc1cccnc1N1CCCC1)c1ncsc1C1CC1 ZINC000880663947 EF On-Demand Anodyne SCN2A 20 48 O=C(NCc1cccnc1N1CCCC1)c1ncsc1C1CC1 ZINC000880663947 EF On-Demand Anodyne SCN10A 21 48 CCN(C(=O)c1ccc(-c2ccccc2OC)nc1O)[C@H]1CCN(C)C1 ZINC000880664036 FF On-Demand Anodyne MBTPS1 43 32 CCN(C(=O)c1ccc(-c2ccccc2OC)nc1O)[C@@H]1CCN(C)C1 ZINC000880664037 FF On-Demand Anodyne MBTPS1 43 32 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880664038 GE On-Demand Clean CASR 15 40 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880664038 GE On-Demand Clean CCR3 58 46 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880664038 GE On-Demand Clean MTOR 40 36 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880664038 GE On-Demand Clean STAT6 51 37 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664051 FG On-Demand Anodyne PDE4D 20 41 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664051 FG On-Demand Anodyne EZH2 42 38 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664052 FG On-Demand Anodyne PDE4D 20 41 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664052 FG On-Demand Anodyne EZH2 42 38 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664053 FG On-Demand Anodyne PDE4D 20 41 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664053 FG On-Demand Anodyne EZH2 42 38 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664054 FG On-Demand Anodyne PDE4D 20 41 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880664054 FG On-Demand Anodyne EZH2 42 38 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664055 DD On-Demand Anodyne JAK3 17 40 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664055 DD On-Demand Anodyne TYK2 20 40 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664056 DD On-Demand Anodyne JAK3 17 40 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664056 DD On-Demand Anodyne TYK2 20 40 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664057 DD On-Demand Anodyne JAK3 17 40 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664057 DD On-Demand Anodyne TYK2 20 40 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664058 DD On-Demand Anodyne JAK3 17 40 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880664058 DD On-Demand Anodyne TYK2 20 40 O=C(NCc1cccnc1N1CCCC1)c1cnc2cc[nH]c2c1 ZINC000880664073 DE On-Demand Anodyne SCN2A 25 60 O=C(NCc1cccnc1N1CCCC1)c1cnc2cc[nH]c2c1 ZINC000880664073 DE On-Demand Anodyne SCN10A 47 60 O=C(NCc1cccnc1N1CCCC1)c1cnc2cc[nH]c2c1 ZINC000880664073 DE On-Demand Anodyne NAMPT 49 40 O=C(CC[C@H]1CCc2ccccc21)NCc1cccnc1N1CCCC1 ZINC000880664089 EH On-Demand Anodyne SCN2A 17 41 O=C(CC[C@H]1CCc2ccccc21)NCc1cccnc1N1CCCC1 ZINC000880664089 EH On-Demand Anodyne SCN10A 18 41 O=C(CC[C@@H]1CCc2ccccc21)NCc1cccnc1N1CCCC1 ZINC000880664090 EH On-Demand Anodyne SCN2A 17 41 O=C(CC[C@@H]1CCc2ccccc21)NCc1cccnc1N1CCCC1 ZINC000880664090 EH On-Demand Anodyne SCN10A 18 41 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1cccnc1N1CCCC1 ZINC000880664103 CF On-Demand Anodyne SCN2A 18 44 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1cccnc1N1CCCC1 ZINC000880664103 CF On-Demand Anodyne SCN10A 19 44 O=C1CC[C@H](c2ccc(C(=O)NCc3cccnc3N3CCCC3)cc2)N1 ZINC000880664105 FF On-Demand Anodyne SCN2A 22 52 O=C1CC[C@H](c2ccc(C(=O)NCc3cccnc3N3CCCC3)cc2)N1 ZINC000880664105 FF On-Demand Anodyne SCN10A 33 52 O=C1CC[C@@H](c2ccc(C(=O)NCc3cccnc3N3CCCC3)cc2)N1 ZINC000880664106 FF On-Demand Anodyne SCN2A 22 52 O=C1CC[C@@H](c2ccc(C(=O)NCc3cccnc3N3CCCC3)cc2)N1 ZINC000880664106 FF On-Demand Anodyne SCN10A 33 52 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880664107 GG On-Demand Anodyne EPHX2 43 39 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880664107 GG On-Demand Anodyne GPR119 40 42 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664112 ED On-Demand Anodyne PYGL 32 46 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664112 ED On-Demand Anodyne PYGM 29 46 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664113 ED On-Demand Anodyne PYGL 32 46 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664113 ED On-Demand Anodyne PYGM 29 46 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664114 ED On-Demand Anodyne PYGL 32 46 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664114 ED On-Demand Anodyne PYGM 29 46 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664115 ED On-Demand Anodyne PYGL 32 46 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664115 ED On-Demand Anodyne PYGM 29 46 CCOC(=O)N1CCC(NC(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880664124 FE On-Demand Anodyne EPHX2 43 43 O=C(N1C[C@H]2CC[C@@H](O)C[C@H]2C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880664128 DF On-Demand Anodyne RBP4 42 32 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880664130 GE On-Demand Anodyne CELA1 19 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880664130 GE On-Demand Anodyne PREP 49 48 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880664130 GE On-Demand Anodyne SLC12A5 58 37 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880664130 GE On-Demand Anodyne Q9NAW4_PLAFA 37 43 O=C1CC[C@@H](c2ccc(C(=O)N3C[C@H]4CC[C@@H](O)C[C@H]4C3)cc2)N1 ZINC000880664137 ED On-Demand Anodyne L3MBTL3 29 41 O=C1CC[C@H](c2ccc(C(=O)N3C[C@H]4CC[C@@H](O)C[C@H]4C3)cc2)N1 ZINC000880664138 ED On-Demand Anodyne L3MBTL3 29 41 O=C(NCc1cccnc1N1CCCC1)c1csc(-c2ncc[nH]2)n1 ZINC000880664153 FE On-Demand Anodyne SCN2A 19 46 O=C(NCc1cccnc1N1CCCC1)c1csc(-c2ncc[nH]2)n1 ZINC000880664153 FE On-Demand Anodyne SCN10A 29 51 O=C(Nc1c(F)ccc2c1OCO2)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880664160 GF On-Demand Anodyne FAAH 21 45 O=C(Nc1c(F)ccc2c1OCO2)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880664160 GF On-Demand Anodyne MCHR1 18 41 O=C(Nc1c(F)ccc2c1OCO2)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880664165 GF On-Demand Bother SSTR1 41 41 CCN(C(=O)[C@H]1CCc2cc(OC)ccc2C1)[C@@H]1CCN(C)C1 ZINC000880664185 DE On-Demand Anodyne DRD5 17 41 CCN(C(=O)[C@H]1CCc2cc(OC)ccc2C1)[C@@H]1CCN(C)C1 ZINC000880664185 DE On-Demand Anodyne MTNR1A 15 40 CCN(C(=O)[C@H]1CCc2cc(OC)ccc2C1)[C@H]1CCN(C)C1 ZINC000880664187 DE On-Demand Anodyne DRD5 17 41 CCN(C(=O)[C@H]1CCc2cc(OC)ccc2C1)[C@H]1CCN(C)C1 ZINC000880664187 DE On-Demand Anodyne MTNR1A 15 40 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCC[C@H]([S@@](C)=O)C2)c(O)n1 ZINC000880664236 GF On-Demand Anodyne HTR3A 20 44 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCC[C@@H]([S@@](C)=O)C2)c(O)n1 ZINC000880664237 GF On-Demand Anodyne HTR3A 20 44 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCC[C@H]([S@](C)=O)C2)c(O)n1 ZINC000880664238 GF On-Demand Anodyne HTR3A 20 44 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCC[C@@H]([S@](C)=O)C2)c(O)n1 ZINC000880664239 GF On-Demand Anodyne HTR3A 20 44 Cc1nc(C(C)C)ncc1C(=O)NCc1cccnc1N1CCCC1 ZINC000880664310 EF On-Demand Anodyne SCN2A 20 52 Cc1nc(C(C)C)ncc1C(=O)NCc1cccnc1N1CCCC1 ZINC000880664310 EF On-Demand Anodyne SCN10A 41 52 O=C(NCc1cccnc1N1CCCC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880664325 DE On-Demand Anodyne SCN2A 17 42 O=C(NCc1cccnc1N1CCCC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880664325 DE On-Demand Anodyne SCN10A 19 42 O=C(NCc1cccnc1N1CCCC1)c1cccc2nsnc12 ZINC000880664352 EF On-Demand Anodyne SCN2A 19 47 O=C(NCc1cccnc1N1CCCC1)c1cccc2nsnc12 ZINC000880664352 EF On-Demand Anodyne LIPA 44 31 O=C(NCc1cccnc1N1CCCC1)c1cccc2nsnc12 ZINC000880664352 EF On-Demand Anodyne SCN10A 21 47 Cn1ncc(Br)c1CC(=O)NCc1cccnc1N1CCCC1 ZINC000880664354 GE On-Demand Anodyne P2RX7 24 42 Cn1ncc(Br)c1CC(=O)NCc1cccnc1N1CCCC1 ZINC000880664354 GE On-Demand Anodyne SCN2A 19 47 Cn1ncc(Br)c1CC(=O)NCc1cccnc1N1CCCC1 ZINC000880664354 GE On-Demand Anodyne SCN10A 24 49 O=C(NCc1cccnc1N1CCCC1)c1coc(-c2ccccn2)n1 ZINC000880664367 EF On-Demand Anodyne SCN2A 19 46 O=C(NCc1cccnc1N1CCCC1)c1coc(-c2ccccn2)n1 ZINC000880664367 EF On-Demand Anodyne SCN10A 36 55 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)c(C)cc1OC ZINC000880664437 FG On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)c(C)cc1OC ZINC000880664440 FG On-Demand Anodyne PAPA1_CARPA 37 41 CCN(C(=O)c1cc2cc(F)ccc2[nH]c1=O)[C@@H]1CCN(C)C1 ZINC000880664452 DD On-Demand Anodyne PLD1 43 37 CCN(C(=O)c1cc2cc(F)ccc2[nH]c1=O)[C@@H]1CCN(C)C1 ZINC000880664452 DD On-Demand Anodyne PLD2 40 37 CCN(C(=O)c1cc2cc(F)ccc2[nH]c1=O)[C@H]1CCN(C)C1 ZINC000880664454 DD On-Demand Anodyne PLD1 43 37 CCN(C(=O)c1cc2cc(F)ccc2[nH]c1=O)[C@H]1CCN(C)C1 ZINC000880664454 DD On-Demand Anodyne PLD2 40 37 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne DRD4 40 32 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne NQO2 30 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne SCN2A 18 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne MTNR1A 47 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne MTNR1B 42 39 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne EBP 42 44 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne FAAH 16 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne EPHX2 17 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1N1CCCC1)C2 ZINC000880664473 FG On-Demand Anodyne SCN10A 21 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCCCCCC1 ZINC000880664476 DF On-Demand Anodyne CCR3 24 43 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2cccc(Oc3ccccn3)c2)C1 ZINC000880664481 FG On-Demand Anodyne CFTR 17 41 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2cccc(Oc3ccccn3)c2)C1 ZINC000880664482 FG On-Demand Anodyne CFTR 17 41 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2cccc(Oc3ccccn3)c2)C1 ZINC000880664483 FG On-Demand Anodyne CFTR 17 41 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2cccc(Oc3ccccn3)c2)C1 ZINC000880664484 FG On-Demand Anodyne CFTR 17 41 Cn1nnc(C(=O)NCc2cccnc2N2CCCC2)n1 ZINC000880664493 CC On-Demand Anodyne SCN2A 20 49 Cn1nnc(C(=O)NCc2cccnc2N2CCCC2)n1 ZINC000880664493 CC On-Demand Anodyne SCN10A 24 49 Cn1nnnc1-c1ccccc1NC(=O)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880664516 GF On-Demand Anodyne CCR3 35 40 Cn1nnnc1-c1ccccc1NC(=O)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880664518 GF On-Demand Anodyne CCR3 35 40 COc1cc(C)c(C)cc1NC(=O)Cc1c(Br)cnn1C ZINC000880664564 FF On-Demand Anodyne HTR2A 23 40 Cc1nc(C(C)C)ncc1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664572 EE On-Demand Anodyne PYGL 39 52 Cc1nc(C(C)C)ncc1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664572 EE On-Demand Anodyne PYGM 33 52 Cc1nc(C(C)C)ncc1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664573 EE On-Demand Anodyne PYGL 39 52 Cc1nc(C(C)C)ncc1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664573 EE On-Demand Anodyne PYGM 33 52 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2c(F)ccc3c2OCO3)CC1 ZINC000880664577 GG On-Demand Anodyne CACNA1I 41 33 CSc1nccnc1C(=O)NCc1cccnc1N1CCCC1 ZINC000880664585 EE On-Demand Anodyne SCN2A 21 50 CSc1nccnc1C(=O)NCc1cccnc1N1CCCC1 ZINC000880664585 EE On-Demand Anodyne SCN10A 27 50 Cc1coc(C(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)c1 ZINC000880664597 CD On-Demand Anodyne PYGL 44 62 Cc1coc(C(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)c1 ZINC000880664597 CD On-Demand Anodyne PYGM 43 62 Cc1coc(C(=O)N[C@H]2Cc3ccccc3N(C)C2=O)c1 ZINC000880664598 CD On-Demand Anodyne PYGL 44 62 Cc1coc(C(=O)N[C@H]2Cc3ccccc3N(C)C2=O)c1 ZINC000880664598 CD On-Demand Anodyne PYGM 43 62 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1Cc3ccccc3N(C)C1=O)C2 ZINC000880664610 FF On-Demand Anodyne PYGL 34 49 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1Cc3ccccc3N(C)C1=O)C2 ZINC000880664610 FF On-Demand Anodyne PYGM 31 49 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1Cc3ccccc3N(C)C1=O)C2 ZINC000880664613 FF On-Demand Anodyne PYGL 34 49 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1Cc3ccccc3N(C)C1=O)C2 ZINC000880664613 FF On-Demand Anodyne PYGM 31 49 CS(=O)(=O)C1CCC(C(=O)NCc2cccnc2N2CCCC2)CC1 ZINC000880664626 FD On-Demand Anodyne SCN2A 18 44 CS(=O)(=O)C1CCC(C(=O)NCc2cccnc2N2CCCC2)CC1 ZINC000880664626 FD On-Demand Anodyne EPHX2 27 42 CS(=O)(=O)C1CCC(C(=O)NCc2cccnc2N2CCCC2)CC1 ZINC000880664626 FD On-Demand Anodyne SCN10A 20 44 O=C(C[C@H]1CCNC1=O)NCc1cccnc1N1CCCC1 ZINC000880664631 DC On-Demand Anodyne SCN2A 18 44 O=C(C[C@H]1CCNC1=O)NCc1cccnc1N1CCCC1 ZINC000880664631 DC On-Demand Anodyne SCN10A 19 44 CCN(C(=O)c1ccc(Oc2ccc(C)cn2)cc1)[C@H]1CCN(C)C1 ZINC000880664632 EG On-Demand Anodyne MLNR 21 42 CCN(C(=O)c1ccc(Oc2ccc(C)cn2)cc1)[C@H]1CCN(C)C1 ZINC000880664632 EG On-Demand Anodyne LIPE 19 40 O=C(C[C@@H]1CCNC1=O)NCc1cccnc1N1CCCC1 ZINC000880664633 DC On-Demand Anodyne SCN2A 18 44 O=C(C[C@@H]1CCNC1=O)NCc1cccnc1N1CCCC1 ZINC000880664633 DC On-Demand Anodyne SCN10A 19 44 CCN(C(=O)c1ccc(Oc2ccc(C)cn2)cc1)[C@@H]1CCN(C)C1 ZINC000880664634 EG On-Demand Anodyne MLNR 21 42 CCN(C(=O)c1ccc(Oc2ccc(C)cn2)cc1)[C@@H]1CCN(C)C1 ZINC000880664634 EG On-Demand Anodyne LIPE 19 40 COc1cc(C)c(C)cc1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880664657 FH On-Demand Anodyne KCNQ2 70 42 COc1cc(C)c(C)cc1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880664657 FH On-Demand Anodyne P2RX7 23 42 CCN(C(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1)[C@H]1CCN(C)C1 ZINC000880664662 FG On-Demand Anodyne OPRD1 16 41 CCN(C(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1)[C@@H]1CCN(C)C1 ZINC000880664664 FG On-Demand Anodyne OPRD1 16 41 CSc1nccnc1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664683 ED On-Demand Anodyne PYGL 38 52 CSc1nccnc1C(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880664683 ED On-Demand Anodyne PYGM 34 52 CSc1nccnc1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664685 ED On-Demand Anodyne PYGL 38 52 CSc1nccnc1C(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880664685 ED On-Demand Anodyne PYGM 34 52 Cn1nnnc1-c1ccccc1NC(=O)NCCSC(C)(C)C ZINC000880664689 EF On-Demand Anodyne CCR3 23 40 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2cccn(C3CC3)c2=O)C1 ZINC000880664691 DD On-Demand Anodyne CNR2 16 45 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2cccn(C3CC3)c2=O)C1 ZINC000880664693 DD On-Demand Anodyne CNR2 16 45 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2cccn(C3CC3)c2=O)C1 ZINC000880664695 DD On-Demand Anodyne CNR2 16 45 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2cccn(C3CC3)c2=O)C1 ZINC000880664697 DD On-Demand Anodyne CNR2 16 45 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C#N)CC1 ZINC000880664757 DD On-Demand Mild CCR3 18 41 C[C@H](CCc1ccc(F)cc1)C(=O)N[C@@H]1CCC[C@@H]([S@](C)=O)C1 ZINC000880664762 EG On-Demand Anodyne BIRC2 39 43 C[C@H](CCc1ccc(F)cc1)C(=O)N[C@@H]1CCC[C@@H]([S@@](C)=O)C1 ZINC000880664763 EG On-Demand Anodyne BIRC2 39 43 C[C@H](CCc1ccc(F)cc1)C(=O)N[C@@H]1CCC[C@H]([S@@](C)=O)C1 ZINC000880664764 EG On-Demand Anodyne BIRC2 39 43 C[C@H](CCc1ccc(F)cc1)C(=O)N[C@@H]1CCC[C@H]([S@](C)=O)C1 ZINC000880664765 EG On-Demand Anodyne BIRC2 39 43 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccnc1N1CCCC1 ZINC000880664785 GF On-Demand Anodyne KCNQ2 69 41 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccnc1N1CCCC1 ZINC000880664785 GF On-Demand Anodyne P2RX7 24 41 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccnc1N1CCCC1 ZINC000880664785 GF On-Demand Anodyne SCN2A 20 46 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccnc1N1CCCC1 ZINC000880664785 GF On-Demand Anodyne SCN10A 23 46 Cc1coc(C(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880664789 CF On-Demand Anodyne SCN2A 22 53 Cc1coc(C(=O)NCc2cccnc2N2CCCC2)c1 ZINC000880664789 CF On-Demand Anodyne SCN10A 40 53 O=C(NCc1cccnc1N1CCCC1)c1cncc2[nH]ccc12 ZINC000880664804 DE On-Demand Anodyne SCN2A 25 57 O=C(NCc1cccnc1N1CCCC1)c1cncc2[nH]ccc12 ZINC000880664804 DE On-Demand Anodyne SCN10A 51 57 Cn1nc2c(c1C(=O)NCc1cccnc1N1CCCC1)CSCC2 ZINC000880664833 FE On-Demand Anodyne SCN2A 19 45 Cn1nc2c(c1C(=O)NCc1cccnc1N1CCCC1)CSCC2 ZINC000880664833 FE On-Demand Anodyne SCN10A 22 45 O=C(CN1CCCCS1(=O)=O)NCc1cccnc1N1CCCC1 ZINC000880664834 FC On-Demand Anodyne SCN2A 18 45 O=C(CN1CCCCS1(=O)=O)NCc1cccnc1N1CCCC1 ZINC000880664834 FC On-Demand Anodyne SCN10A 20 45 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880664852 FD On-Demand Anodyne CCR3 26 40 CCN(C(=O)c1cc(-c2ccc(OC)cc2)on1)[C@H]1CCN(C)C1 ZINC000880664927 EF On-Demand Anodyne PDK1 49 37 CCN(C(=O)c1cc(-c2ccc(OC)cc2)on1)[C@H]1CCN(C)C1 ZINC000880664927 EF On-Demand Anodyne MCHR1 15 48 CCN(C(=O)c1cc(-c2ccc(OC)cc2)on1)[C@@H]1CCN(C)C1 ZINC000880664928 EF On-Demand Anodyne PDK1 49 37 CCN(C(=O)c1cc(-c2ccc(OC)cc2)on1)[C@@H]1CCN(C)C1 ZINC000880664928 EF On-Demand Anodyne MCHR1 15 48 CN(C)C[C@@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)C[C@H]1CN(C)C ZINC000880664938 GD On-Demand Anodyne CCR3 26 43 Cn1nnnc1-c1ccccc1NC(=O)NCCSCCC(F)(F)F ZINC000880664939 FF On-Demand Anodyne CCR3 19 40 COCc1cc(NC(=O)N2C[C@H](C)CC2(C)C)ccc1OC ZINC000880664940 DG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2C[C@H](C)CC2(C)C)ccc1OC ZINC000880664940 DG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@@H](C)CC2(C)C)ccc1OC ZINC000880664941 DG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2C[C@@H](C)CC2(C)C)ccc1OC ZINC000880664941 DG On-Demand Anodyne QRFPR 44 36 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CSCCS1 ZINC000880664942 FD On-Demand Anodyne CCR3 23 41 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CSCCS1 ZINC000880664943 FD On-Demand Anodyne CCR3 23 41 COCc1cc(NC(=O)N(C)C[C@@H]2CN(c3ccccc3)C(=O)O2)ccc1OC ZINC000880664944 GG On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)N(C)C[C@H]2CN(c3ccccc3)C(=O)O2)ccc1OC ZINC000880664945 GG On-Demand Anodyne TSHR 67 32 Cn1nnnc1-c1ccccc1NC(=O)N[C@]12CCC[C@H]1OCC2 ZINC000880664948 ED On-Demand Anodyne CCR3 19 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880664949 FG On-Demand Anodyne CCR3 17 41 COCc1cc(NC(=O)N2CCC(C)(N3CCCCC3)CC2)ccc1OC ZINC000880664951 GH On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC(C)(N3CCCCC3)CC2)ccc1OC ZINC000880664951 GH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCC[C@@H]2CCOC2=O)ccc1OC ZINC000880664952 EE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCCC[C@@H]2CCOC2=O)ccc1OC ZINC000880664952 EE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCCC[C@H]2CCOC2=O)ccc1OC ZINC000880664953 EE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCCC[C@H]2CCOC2=O)ccc1OC ZINC000880664953 EE On-Demand Anodyne QRFPR 41 34 Cn1nnnc1-c1ccccc1NC(=O)NN1C[C@H]2CCC[C@@H](C2)C1 ZINC000880664955 EE On-Demand Anodyne CCR3 52 47 COCc1cc(NC(=O)NCCC2CCC2)ccc1OC ZINC000880664956 CG On-Demand Anodyne TSHR 57 34 COCc1cc(NC(=O)NCCC2CCC2)ccc1OC ZINC000880664956 CG On-Demand Anodyne PDE4A 16 41 COCc1cc(NC(=O)NCCC2CCC2)ccc1OC ZINC000880664956 CG On-Demand Anodyne EPHX2 15 40 COCc1cc(NC(=O)NCCC2CCC2)ccc1OC ZINC000880664956 CG On-Demand Anodyne QRFPR 48 39 COCc1cc(NC(=O)NCCC2CCC2)ccc1OC ZINC000880664956 CG On-Demand Anodyne PRMT3 35 50 COCc1cc(NC(=O)NCC(C)(C)CC(F)F)ccc1OC ZINC000880664961 EH On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@H](C)c2ccnn2C)ccc1OC ZINC000880664964 DE On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)N[C@H](C)c2ccnn2C)ccc1OC ZINC000880664964 DE On-Demand Anodyne HTR2A 42 48 COCc1cc(NC(=O)N[C@H](C)c2ccnn2C)ccc1OC ZINC000880664964 DE On-Demand Anodyne HTR2C 15 48 COCc1cc(NC(=O)N[C@H](C)c2ccnn2C)ccc1OC ZINC000880664964 DE On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)N[C@@H](C)c2ccnn2C)ccc1OC ZINC000880664965 DE On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)N[C@@H](C)c2ccnn2C)ccc1OC ZINC000880664965 DE On-Demand Anodyne HTR2A 42 48 COCc1cc(NC(=O)N[C@@H](C)c2ccnn2C)ccc1OC ZINC000880664965 DE On-Demand Anodyne HTR2C 15 48 COCc1cc(NC(=O)N[C@@H](C)c2ccnn2C)ccc1OC ZINC000880664965 DE On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)Nc2cccc3c2N(C)C(=O)CO3)ccc1OC ZINC000880664966 FF On-Demand Anodyne TSHR 48 34 CC[C@H](C)CONC(=O)Nc1ccccc1-c1nnnn1C ZINC000880664967 DD On-Demand Anodyne CCR3 30 40 CC[C@@H](C)CONC(=O)Nc1ccccc1-c1nnnn1C ZINC000880664968 DD On-Demand Anodyne CCR3 30 40 Cn1nnnc1-c1ccccc1NC(=O)NCC1(C)CC(F)(F)C1 ZINC000880664969 EE On-Demand Anodyne CCR3 59 45 COCc1cc(NC(=O)N2CCO[C@H]([C@@H]3COC(C)(C)O3)C2)ccc1OC ZINC000880664970 GE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)ccc1OC ZINC000880664971 GH On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(c2cnn(C)c2)C3)ccc1OC ZINC000880664971 GH On-Demand Anodyne ENPP1 61 33 COCc1cc(NC(=O)NCC2(CC3CC3)CC2)ccc1OC ZINC000880664972 DH On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NCC2(CC3CC3)CC2)ccc1OC ZINC000880664972 DH On-Demand Anodyne QRFPR 44 36 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@]1(C)CC1(Cl)Cl ZINC000880664973 FF On-Demand Anodyne CCR3 35 44 Cn1nnnc1-c1ccccc1NC(=O)NC[C@]1(C)CC1(Cl)Cl ZINC000880664974 FF On-Demand Anodyne CCR3 35 44 COCc1cc(NC(=O)N2C[C@@H]3C[C@H]2CN3c2ccccc2)ccc1OC ZINC000880664977 FG On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2C[C@@H]3C[C@H]2CN3c2ccccc2)ccc1OC ZINC000880664977 FG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)N2CC[C@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664980 EE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CC[C@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664980 EE On-Demand Anodyne HTR1D 22 44 COCc1cc(NC(=O)N2CC[C@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664980 EE On-Demand Anodyne HTR1B 24 44 COCc1cc(NC(=O)N2CC[C@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664980 EE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664981 EE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CC[C@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664981 EE On-Demand Anodyne HTR1D 22 44 COCc1cc(NC(=O)N2CC[C@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664981 EE On-Demand Anodyne HTR1B 24 44 COCc1cc(NC(=O)N2CC[C@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664981 EE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664982 EE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CC[C@@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664982 EE On-Demand Anodyne HTR1D 22 44 COCc1cc(NC(=O)N2CC[C@@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664982 EE On-Demand Anodyne HTR1B 24 44 COCc1cc(NC(=O)N2CC[C@@H]3[C@H](CCN3C)C2)ccc1OC ZINC000880664982 EE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664983 EE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664983 EE On-Demand Anodyne HTR1D 22 44 COCc1cc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664983 EE On-Demand Anodyne HTR1B 24 44 COCc1cc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C)C2)ccc1OC ZINC000880664983 EE On-Demand Anodyne QRFPR 43 35 Cn1nnnc1-c1ccccc1NC(=O)NOCCC1CC1 ZINC000880664984 DD On-Demand Anodyne CCR3 60 46 Cn1nnnc1-c1ccccc1NC(=O)NCC1(CC2CC2)CC1 ZINC000880664985 EF On-Demand Anodyne CCR3 62 48 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H]1CC12CCC2 ZINC000880664986 CD On-Demand Anodyne CCR3 17 47 Cn1nnnc1-c1ccccc1NC(=O)N[C@H]1CC12CCC2 ZINC000880664987 CD On-Demand Anodyne CCR3 17 47 COCc1cc(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)ccc1OC ZINC000880664989 GI On-Demand Mild HTR2A 15 44 COCc1cc(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)ccc1OC ZINC000880664989 GI On-Demand Mild MCHR1 15 40 COCc1cc(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)ccc1OC ZINC000880664990 GI On-Demand Mild HTR2A 15 44 COCc1cc(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)ccc1OC ZINC000880664990 GI On-Demand Mild MCHR1 15 40 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](O)C1(C)C ZINC000880664995 DD On-Demand Anodyne CCR3 23 41 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](O)C1(C)C ZINC000880664996 DD On-Demand Anodyne CCR3 23 41 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C[C@@H]2CCC[C@@H]2O1 ZINC000880664997 ED On-Demand Anodyne CCR3 31 43 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C[C@@H]2CCC[C@H]2O1 ZINC000880664998 ED On-Demand Anodyne CCR3 31 43 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C[C@H]2CCC[C@H]2O1 ZINC000880664999 ED On-Demand Anodyne CCR3 31 43 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C[C@H]2CCC[C@@H]2O1 ZINC000880665000 ED On-Demand Anodyne CCR3 31 43 COCc1cc(NC(=O)N2CCC[C@@H]2c2cncc(C)c2)ccc1OC ZINC000880665001 FH On-Demand Anodyne TSHR 65 31 COCc1cc(NC(=O)N2CCC[C@@H]2c2cncc(C)c2)ccc1OC ZINC000880665001 FH On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@H]2c2cncc(C)c2)ccc1OC ZINC000880665002 FH On-Demand Anodyne TSHR 65 31 COCc1cc(NC(=O)N2CCC[C@H]2c2cncc(C)c2)ccc1OC ZINC000880665002 FH On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@@H]2C[C@H](C(=O)OC)c3ccccc32)ccc1OC ZINC000880665003 GG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@@H]2C[C@H](C(=O)OC)c3ccccc32)ccc1OC ZINC000880665003 GG On-Demand Anodyne QRFPR 44 39 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665004 FE On-Demand Anodyne CCR3 51 44 Cn1nccc1[C@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665005 FE On-Demand Anodyne CCR3 51 44 COCc1cc(NC(=O)N2CC[C@]3(C(=O)OC)CCC[C@H]23)ccc1OC ZINC000880665006 FF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC[C@]3(C(=O)OC)CCC[C@H]23)ccc1OC ZINC000880665006 FF On-Demand Anodyne QRFPR 43 35 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(NC2CCOCC2)CC1 ZINC000880665009 GD On-Demand Anodyne CCR3 21 42 COCc1cc(NC(=O)N2CC[C@@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665010 FH On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CC[C@@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665010 FH On-Demand Anodyne QRFPR 45 39 COCc1cc(NC(=O)N2CC[C@@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665010 FH On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)N2CC[C@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665011 FH On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CC[C@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665011 FH On-Demand Anodyne QRFPR 45 39 COCc1cc(NC(=O)N2CC[C@H](c3nc(C)cs3)C2)ccc1OC ZINC000880665011 FH On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)NCc2ccc(C)nc2Cl)ccc1OC ZINC000880665012 EH On-Demand Anodyne TSHR 68 36 COCc1cc(NC(=O)NCc2ccc(C)nc2Cl)ccc1OC ZINC000880665012 EH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NCc2ccc(C)nc2Cl)ccc1OC ZINC000880665012 EH On-Demand Anodyne ENPP1 71 36 COCc1cc(NC(=O)N2CCc3ccc(NC(C)=O)cc3C2)ccc1OC ZINC000880665015 GG On-Demand Anodyne TSHR 62 34 COCc1cc(NC(=O)N2CCc3ccc(NC(C)=O)cc3C2)ccc1OC ZINC000880665015 GG On-Demand Anodyne HTR1B 15 41 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H]1CCCC[C@@H]1F ZINC000880665018 DE On-Demand Anodyne CCR3 65 60 COCc1cc(NC(=O)NCCOC(F)(F)C(F)(F)F)ccc1OC ZINC000880665020 FG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N[C@H](C)CC(=O)OC)ccc1OC ZINC000880665022 DD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)CC(=O)OC)ccc1OC ZINC000880665022 DD On-Demand Anodyne ENPP1 63 32 CCCONC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665023 CD On-Demand Anodyne CCR3 21 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCCCCCCC1 ZINC000880665024 EG On-Demand Anodyne CCR3 24 43 CN1CC[C@H]2CN(C(=O)Nc3ccccc3-c3nnnn3C)CC[C@H]21 ZINC000880665027 ED On-Demand Anodyne CCR3 46 42 CN1CC[C@H]2CN(C(=O)Nc3ccccc3-c3nnnn3C)CC[C@H]21 ZINC000880665027 ED On-Demand Anodyne RBP4 46 33 CN1CC[C@H]2CN(C(=O)Nc3ccccc3-c3nnnn3C)CC[C@@H]21 ZINC000880665028 ED On-Demand Anodyne CCR3 46 42 CN1CC[C@H]2CN(C(=O)Nc3ccccc3-c3nnnn3C)CC[C@@H]21 ZINC000880665028 ED On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C=CCC1 ZINC000880665029 CD On-Demand Anodyne CCR3 37 44 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1C=CCC1 ZINC000880665030 CD On-Demand Anodyne CCR3 37 44 COCc1cc(NC(=O)N(C)Cc2ccc3cc[nH]c3c2)ccc1OC ZINC000880665031 FH On-Demand Anodyne ENPP1 62 32 CCN(CC)C(=O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665032 DD On-Demand Anodyne TSHR 47 31 CCN(CC)C(=O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665032 DD On-Demand Anodyne QRFPR 41 34 CCN(CC)C(=O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665032 DD On-Demand Anodyne ENPP1 63 33 Cn1nnnc1-c1ccccc1NC(=O)NCCC1CCC1 ZINC000880665033 DE On-Demand Anodyne CCR3 68 51 COCc1cc(NC(=O)N2C[C@@]3(C)CS(=O)(=O)C[C@@]3(C)C2)ccc1OC ZINC000880665034 GE On-Demand Anodyne ENPP1 51 33 COCc1cc(NC(=O)N2CCC[C@@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665035 GF On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N2CCC[C@@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665035 GF On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N2CCC[C@@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665035 GF On-Demand Anodyne ENPP1 45 31 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@@H]1CCN(C)C1 ZINC000880665096 DE On-Demand Anodyne SLC6A4 16 43 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@@H]1CCN(C)C1 ZINC000880665096 DE On-Demand Anodyne HTR1F 46 38 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@@H]1CCN(C)C1 ZINC000880665096 DE On-Demand Anodyne MPO 47 37 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@H]1CCN(C)C1 ZINC000880665097 DE On-Demand Anodyne SLC6A4 16 43 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@H]1CCN(C)C1 ZINC000880665097 DE On-Demand Anodyne HTR1F 46 38 CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)[C@H]1CCN(C)C1 ZINC000880665097 DE On-Demand Anodyne MPO 47 37 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1COc2ccccc2C1 ZINC000880665119 FE On-Demand Anodyne CCR3 25 41 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1COc2ccccc2C1 ZINC000880665120 FE On-Demand Anodyne CCR3 25 41 CCC(C)(C)[C@@H](C)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665125 EF On-Demand Anodyne PAPA1_CARPA 39 50 CCC(C)(C)[C@@H](C)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665125 EF On-Demand Anodyne CTSK 18 51 CCC(C)(C)[C@@H](C)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665125 EF On-Demand Anodyne POLG_HCV1 24 41 CCC(C)(C)[C@@H](C)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665125 EF On-Demand Anodyne FPR1 49 40 CCC(C)(C)[C@@H](C)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665126 EF On-Demand Anodyne PAPA1_CARPA 39 50 CCC(C)(C)[C@@H](C)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665126 EF On-Demand Anodyne CTSK 18 51 CCC(C)(C)[C@@H](C)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665126 EF On-Demand Anodyne POLG_HCV1 24 41 CCC(C)(C)[C@@H](C)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880665126 EF On-Demand Anodyne FPR1 49 40 COCc1cc(NC(=O)N2CCC[C@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665136 GF On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N2CCC[C@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665136 GF On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N2CCC[C@H](c3nnc(S)n3C)C2)ccc1OC ZINC000880665136 GF On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CCC[C@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665139 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665139 GI On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665139 GI On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2CCC[C@@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665140 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665140 GI On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@@H](c3cc(C(C)C)[nH]n3)C2)ccc1OC ZINC000880665140 GI On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NC[C@@H](O)C(F)(F)C(F)(F)F)ccc1OC ZINC000880665142 FF On-Demand Anodyne PRMT3 43 33 COCc1cc(NC(=O)NC[C@H](O)C(F)(F)C(F)(F)F)ccc1OC ZINC000880665143 FF On-Demand Anodyne PRMT3 43 33 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(F)CC1 ZINC000880665146 DD On-Demand Anodyne CCR3 53 45 COCc1cc(NC(=O)N2C[C@@H](CO)[C@@H](CO)C2)ccc1OC ZINC000880665147 DC On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2C[C@@H](CO)[C@@H](CO)C2)ccc1OC ZINC000880665147 DC On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@@H](CO)[C@@H](CO)C2)ccc1OC ZINC000880665147 DC On-Demand Anodyne ENPP1 57 33 COCc1cc(NC(=O)NC[C@@H]2C=CCC2)ccc1OC ZINC000880665148 CF On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@@H]2C=CCC2)ccc1OC ZINC000880665148 CF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)NC[C@H]2C=CCC2)ccc1OC ZINC000880665149 CF On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@H]2C=CCC2)ccc1OC ZINC000880665149 CF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne HTR1D 15 44 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne HTR1B 18 41 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne CCR3 17 46 COCc1cc(NC(=O)N2CCC[C@H](CF)C2)ccc1OC ZINC000880665150 DG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne HTR1D 15 44 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne HTR1B 18 41 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne CCR3 17 46 COCc1cc(NC(=O)N2CCC[C@@H](CF)C2)ccc1OC ZINC000880665151 DG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CCC[C@@H](C(C)=O)C2)ccc1OC ZINC000880665152 DF On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)N2CCC[C@@H](C(C)=O)C2)ccc1OC ZINC000880665152 DF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@@H](C(C)=O)C2)ccc1OC ZINC000880665152 DF On-Demand Anodyne HTR1B 17 40 COCc1cc(NC(=O)N2CCC[C@@H](C(C)=O)C2)ccc1OC ZINC000880665152 DF On-Demand Anodyne QRFPR 47 38 COCc1cc(NC(=O)N2CCC[C@H](C(C)=O)C2)ccc1OC ZINC000880665153 DF On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)N2CCC[C@H](C(C)=O)C2)ccc1OC ZINC000880665153 DF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@H](C(C)=O)C2)ccc1OC ZINC000880665153 DF On-Demand Anodyne HTR1B 17 40 COCc1cc(NC(=O)N2CCC[C@H](C(C)=O)C2)ccc1OC ZINC000880665153 DF On-Demand Anodyne QRFPR 47 38 Cn1nnnc1-c1ccccc1NC(=O)N1CCCN(c2ncccc2F)CC1 ZINC000880665158 GE On-Demand Anodyne CCR3 21 41 COCc1cc(NC(=O)N[C@]23CCC[C@H]2OCC3)ccc1OC ZINC000880665159 DF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@]23CCC[C@H]2OCC3)ccc1OC ZINC000880665159 DF On-Demand Anodyne QRFPR 44 36 Cn1nnnc1-c1ccccc1NC(=O)NC1([C@@H]2CCCCO2)CCC1 ZINC000880665160 FE On-Demand Anodyne CCR3 20 44 Cn1nnnc1-c1ccccc1NC(=O)NC1([C@H]2CCCCO2)CCC1 ZINC000880665161 FE On-Demand Anodyne CCR3 20 44 COCc1cc(NC(=O)N2C[C@@H]3CN(C(C)=O)C[C@@H]3C2)ccc1OC ZINC000880665163 ED On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2C[C@@H]3CN(C(C)=O)C[C@@H]3C2)ccc1OC ZINC000880665163 ED On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@@H]3CN(C(C)=O)C[C@@H]3C2)ccc1OC ZINC000880665163 ED On-Demand Anodyne ENPP1 56 33 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1OCCc2sccc21 ZINC000880665166 FE On-Demand Anodyne CCR3 19 40 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1OCCc2sccc21 ZINC000880665167 FE On-Demand Anodyne CCR3 19 40 CC[C@@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@H]1CCCOC1 ZINC000880665168 EE On-Demand Anodyne CCR3 58 42 CC[C@@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@@H]1CCCOC1 ZINC000880665171 EE On-Demand Anodyne CCR3 58 42 COCc1cc(NC(=O)NN2C[C@H]3CCC[C@@H](C3)C2)ccc1OC ZINC000880665172 EG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NN2C[C@H]3CCC[C@@H](C3)C2)ccc1OC ZINC000880665172 EG On-Demand Anodyne QRFPR 46 38 Cn1nnnc1-c1ccccc1NC(=O)N1[C@H]2CC[C@H]1CC(CCO)C2 ZINC000880665174 FE On-Demand Anodyne CCR3 31 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](C2(C)OCCO2)C1 ZINC000880665176 FD On-Demand Anodyne CCR3 38 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](C2(C)OCCO2)C1 ZINC000880665177 FD On-Demand Anodyne CCR3 38 43 COCc1cc(NC(=O)N2C[C@@H]3CCC[C@]3(C(=O)OC)C2)ccc1OC ZINC000880665178 FF On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2C[C@@H]3CCC[C@]3(C(=O)OC)C2)ccc1OC ZINC000880665178 FF On-Demand Anodyne QRFPR 42 35 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](c2nccs2)C1 ZINC000880665179 FE On-Demand Anodyne CCR3 21 41 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](c2nccs2)C1 ZINC000880665180 FE On-Demand Anodyne CCR3 21 41 COCc1cc(NC(=O)N2CCO[C@H](c3noc(C4CC4)n3)C2)ccc1OC ZINC000880665183 GF On-Demand Anodyne SMO 24 41 COCc1cc(NC(=O)N2CCO[C@@H](c3noc(C4CC4)n3)C2)ccc1OC ZINC000880665184 GF On-Demand Anodyne SMO 24 41 COCc1cc(NC(=O)N2CC[C@](C)(C(F)(F)F)C2)ccc1OC ZINC000880665186 EH On-Demand Anodyne EPHX2 37 44 COCc1cc(NC(=O)N2CC[C@](C)(C(F)(F)F)C2)ccc1OC ZINC000880665186 EH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@](C)(C(F)(F)F)C2)ccc1OC ZINC000880665187 EH On-Demand Anodyne EPHX2 37 44 COCc1cc(NC(=O)N2CC[C@@](C)(C(F)(F)F)C2)ccc1OC ZINC000880665187 EH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCc2cc(C(=O)OC)c(C)n2C)ccc1OC ZINC000880665188 GF On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NC[C@@H]2CC(C)(C)CO2)ccc1OC ZINC000880665191 DF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NC[C@@H]2CC(C)(C)CO2)ccc1OC ZINC000880665191 DF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@H]2CC(C)(C)CO2)ccc1OC ZINC000880665192 DF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NC[C@H]2CC(C)(C)CO2)ccc1OC ZINC000880665192 DF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccc1OC ZINC000880665194 ED On-Demand Anodyne CACNA1H 40 34 COCc1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccc1OC ZINC000880665194 ED On-Demand Anodyne TSHR 59 31 COCc1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccc1OC ZINC000880665194 ED On-Demand Anodyne ENPP1 41 33 COCc1cc(NC(=O)N2CC(O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880665195 FF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2CC(O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880665195 FF On-Demand Anodyne ENPP1 62 34 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](C(C)(C)O)C1 ZINC000880665196 ED On-Demand Anodyne CCR3 59 46 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](C(C)(C)O)C1 ZINC000880665197 ED On-Demand Anodyne CCR3 59 46 COCc1cc(NC(=O)N2CCC[C@@H](CCC(=O)OC)C2)ccc1OC ZINC000880665201 FG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC[C@@H](CCC(=O)OC)C2)ccc1OC ZINC000880665201 FG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC[C@@H](CCC(=O)OC)C2)ccc1OC ZINC000880665201 FG On-Demand Anodyne HTR1B 17 41 COCc1cc(NC(=O)N2CCC[C@@H](CCC(=O)OC)C2)ccc1OC ZINC000880665201 FG On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC[C@@H](CCC(=O)OC)C2)ccc1OC ZINC000880665201 FG On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N2CCC[C@H](CCC(=O)OC)C2)ccc1OC ZINC000880665202 FG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC[C@H](CCC(=O)OC)C2)ccc1OC ZINC000880665202 FG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC[C@H](CCC(=O)OC)C2)ccc1OC ZINC000880665202 FG On-Demand Anodyne HTR1B 17 41 COCc1cc(NC(=O)N2CCC[C@H](CCC(=O)OC)C2)ccc1OC ZINC000880665202 FG On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC[C@H](CCC(=O)OC)C2)ccc1OC ZINC000880665202 FG On-Demand Anodyne QRFPR 44 38 CNC(=O)N(C)c1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880665203 FG On-Demand Anodyne TSHR 41 31 Cn1nnnc1-c1ccccc1NC(=O)NC12CCC(CC1)C2 ZINC000880665206 DE On-Demand Anodyne CCR3 24 43 Cn1nnnc1-c1ccccc1NC(=O)NC12CCC(CC1)C2 ZINC000880665206 DE On-Demand Anodyne EPHX2 34 43 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665207 DG On-Demand Mild TSHR 42 32 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665207 DG On-Demand Mild EPHX2 44 38 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665207 DG On-Demand Mild QRFPR 44 36 Cc1csc([C@H]2CCN(C(=O)Nc3ccccc3-c3nnnn3C)C2)n1 ZINC000880665211 FF On-Demand Anodyne CCR3 24 41 CON(C)CCNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665213 DC On-Demand Anodyne CCR3 30 40 COCc1cc(NC(=O)N2CC[C@](C)(NC(=O)C(F)(F)F)C2)ccc1OC ZINC000880665214 GF On-Demand Anodyne EPHX2 34 42 COCc1cc(NC(=O)N2CC[C@@](C)(NC(=O)C(F)(F)F)C2)ccc1OC ZINC000880665215 GF On-Demand Anodyne EPHX2 34 42 COCc1cc(NC(=O)NC2(CCO)CCCCC2)ccc1OC ZINC000880665218 EG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne HTR1D 15 45 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne HTR1B 17 45 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne ABCB1 15 42 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne ABCG2 25 40 COCc1cc(NC(=O)N2CCc3cc(F)c(F)cc3C2)ccc1OC ZINC000880665220 FH On-Demand Anodyne QRFPR 45 32 COCc1cc(NC(=O)N2CCn3cnc(C(F)(F)F)c3C2)ccc1OC ZINC000880665223 GG On-Demand Anodyne PDGFRB 41 36 COCc1cc(NC(=O)N2CC[C@@](O)(C(=O)OC)C2)ccc1OC ZINC000880665225 EC On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CC[C@@](O)(C(=O)OC)C2)ccc1OC ZINC000880665225 EC On-Demand Anodyne PDGFRB 41 36 COCc1cc(NC(=O)N2CC[C@@](O)(C(=O)OC)C2)ccc1OC ZINC000880665225 EC On-Demand Anodyne EPHX2 29 40 COCc1cc(NC(=O)N2CC[C@@](O)(C(=O)OC)C2)ccc1OC ZINC000880665225 EC On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC[C@@](O)(C(=O)OC)C2)ccc1OC ZINC000880665225 EC On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2CC[C@](O)(C(=O)OC)C2)ccc1OC ZINC000880665227 EC On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CC[C@](O)(C(=O)OC)C2)ccc1OC ZINC000880665227 EC On-Demand Anodyne PDGFRB 41 36 COCc1cc(NC(=O)N2CC[C@](O)(C(=O)OC)C2)ccc1OC ZINC000880665227 EC On-Demand Anodyne EPHX2 29 40 COCc1cc(NC(=O)N2CC[C@](O)(C(=O)OC)C2)ccc1OC ZINC000880665227 EC On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC[C@](O)(C(=O)OC)C2)ccc1OC ZINC000880665227 EC On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1OC ZINC000880665229 ED On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1OC ZINC000880665229 ED On-Demand Anodyne PDGFRB 45 38 COCc1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1OC ZINC000880665229 ED On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1OC ZINC000880665229 ED On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N[C@H]2CCC[C@@]23CCCCO3)ccc1OC ZINC000880665230 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H]2CCC[C@]23CCCCO3)ccc1OC ZINC000880665231 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H]2CCC[C@@]23CCCCO3)ccc1OC ZINC000880665232 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@H]2CCC[C@]23CCCCO3)ccc1OC ZINC000880665233 EG On-Demand Anodyne QRFPR 43 35 Cn1nnnc1-c1ccccc1NC(=O)NC1CCC2(CC1)COC2 ZINC000880665234 ED On-Demand Anodyne CCR3 15 46 Cn1nnnc1-c1ccccc1NC(=O)NOCC(F)F ZINC000880665236 CD On-Demand Anodyne CCR3 31 43 COCc1cc(NC(=O)NCC(Cl)Cl)ccc1OC ZINC000880665237 DF On-Demand Reactive TSHR 71 35 COCc1cc(NC(=O)NCC(Cl)Cl)ccc1OC ZINC000880665237 DF On-Demand Reactive HTR2A 26 41 COCc1cc(NC(=O)NCC(Cl)Cl)ccc1OC ZINC000880665237 DF On-Demand Reactive QRFPR 42 35 COCc1cc(NC(=O)NCC(Cl)Cl)ccc1OC ZINC000880665237 DF On-Demand Reactive ENPP1 57 33 COCc1cc(NC(=O)N2CCN(c3cccc(F)n3)CC2)ccc1OC ZINC000880665238 FF On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)N2CCN(c3cccc(F)n3)CC2)ccc1OC ZINC000880665238 FF On-Demand Anodyne HTR1D 17 49 COCc1cc(NC(=O)N2CCN(c3cccc(F)n3)CC2)ccc1OC ZINC000880665238 FF On-Demand Anodyne HTR1B 20 49 COCc1cc(NC(=O)N2CCN(c3cccc(F)n3)CC2)ccc1OC ZINC000880665238 FF On-Demand Anodyne PDGFRB 61 41 COCc1cc(NC(=O)N2CCN(c3cccc(F)n3)CC2)ccc1OC ZINC000880665238 FF On-Demand Anodyne ENPP1 66 34 COCc1cc(NC(=O)N2CC[C@H](O)C2(C)C)ccc1OC ZINC000880665240 DE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@H](O)C2(C)C)ccc1OC ZINC000880665240 DE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CC[C@@H](O)C2(C)C)ccc1OC ZINC000880665241 DE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@@H](O)C2(C)C)ccc1OC ZINC000880665241 DE On-Demand Anodyne QRFPR 44 36 CC(=O)C1CCN(C(=O)Nc2ccccc2-c2nnnn2C)CC1 ZINC000880665244 ED On-Demand Anodyne CCR3 28 43 COCc1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)ccc1OC ZINC000880665246 DE On-Demand Anodyne TSHR 59 32 COCc1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)ccc1OC ZINC000880665246 DE On-Demand Anodyne EPHX2 54 45 COCc1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)ccc1OC ZINC000880665246 DE On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)ccc1OC ZINC000880665246 DE On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665248 GF On-Demand Anodyne EPHX2 47 42 COCc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665248 GF On-Demand Anodyne F13A1 20 40 COCc1cc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665248 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@]2(CO)CCc3c(OC)cccc32)ccc1OC ZINC000880665249 GF On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665251 GF On-Demand Anodyne EPHX2 47 42 COCc1cc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665251 GF On-Demand Anodyne F13A1 20 40 COCc1cc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880665251 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@@]2(CO)CCc3c(OC)cccc32)ccc1OC ZINC000880665253 GF On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)N[C@@H]2CCC(=O)N[C@H]2c2ccccc2)ccc1OC ZINC000880665254 GF On-Demand Anodyne TSHR 75 37 COCc1cc(NC(=O)N[C@@H]2CCC(=O)N[C@H]2c2ccccc2)ccc1OC ZINC000880665254 GF On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)NC2CCC(C)(N(C)C)CC2)ccc1OC ZINC000880665261 EG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC2CCC(C)(N(C)C)CC2)ccc1OC ZINC000880665261 EG On-Demand Anodyne EPHX2 45 40 COCc1cc(NC(=O)NC2CCC(C)(N(C)C)CC2)ccc1OC ZINC000880665261 EG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC3(CCCC3)CC2)ccc1OC ZINC000880665263 EI On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC3(CCCC3)CC2)ccc1OC ZINC000880665263 EI On-Demand Anodyne HTR1B 15 44 COCc1cc(NC(=O)N2CCC3(CCCC3)CC2)ccc1OC ZINC000880665263 EI On-Demand Anodyne PDGFRB 44 37 COCc1cc(NC(=O)N2CCC3(CCCC3)CC2)ccc1OC ZINC000880665263 EI On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCC3(CCCC3)CC2)ccc1OC ZINC000880665263 EI On-Demand Anodyne ENPP1 69 35 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne FKBP1A 53 35 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne TACR1 16 44 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne PDE4A 23 43 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne CPT1A 45 38 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665265 GH On-Demand Anodyne QRFPR 45 41 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne FKBP1A 53 35 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne TACR1 16 44 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne PDE4A 23 43 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne CPT1A 45 38 COCc1cc(NC(=O)N2CCCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880665267 GH On-Demand Anodyne QRFPR 45 41 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne FKBP1A 53 35 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne TACR1 16 44 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne PDE4A 23 43 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne CPT1A 45 38 COCc1cc(NC(=O)N2CCCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665269 GH On-Demand Anodyne QRFPR 45 41 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne FKBP1A 53 35 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne TACR1 16 44 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne PDE4A 23 43 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne CPT1A 45 38 COCc1cc(NC(=O)N2CCCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880665271 GH On-Demand Anodyne QRFPR 45 41 COCc1cc(NC(=O)NC[C@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665272 GF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC[C@@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665274 GF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC[C@@H]2CCO[C@@H]2C(=O)OC)ccc1OC ZINC000880665282 FD On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NC[C@@H]2CCO[C@@H]2C(=O)OC)ccc1OC ZINC000880665282 FD On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)ccc1OC ZINC000880665284 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)ccc1OC ZINC000880665284 FG On-Demand Anodyne EPHX2 27 49 COCc1cc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)ccc1OC ZINC000880665284 FG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)ccc1OC ZINC000880665285 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)ccc1OC ZINC000880665285 FG On-Demand Anodyne EPHX2 27 49 COCc1cc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)ccc1OC ZINC000880665285 FG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)NNc2ccc(CC(=O)OC)cc2)ccc1OC ZINC000880665286 FF On-Demand Reactive TSHR 47 32 COCc1cc(NC(=O)NNc2ccc(CC(=O)OC)cc2)ccc1OC ZINC000880665286 FF On-Demand Reactive QRFPR 42 35 COCc1cc(NC(=O)NNc2ccc(CC(=O)OC)cc2)ccc1OC ZINC000880665286 FF On-Demand Reactive ENPP1 44 30 COCc1cc(NC(=O)NCc2cccc(C3(C)OCCO3)c2)ccc1OC ZINC000880665287 GG On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NCc2cccc(C3(C)OCCO3)c2)ccc1OC ZINC000880665287 GG On-Demand Anodyne ROCK2 28 43 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(O)(c2ccccc2)C3)ccc1OC ZINC000880665288 GH On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(O)(c2ccccc2)C3)ccc1OC ZINC000880665288 GH On-Demand Anodyne QRFPR 43 40 COCc1cc(NC(=O)N2CCCN(C=O)CC2)ccc1OC ZINC000880665292 DD On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CCCN(C=O)CC2)ccc1OC ZINC000880665292 DD On-Demand Anodyne PDGFRB 50 39 COCc1cc(NC(=O)N2CCCN(C=O)CC2)ccc1OC ZINC000880665292 DD On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N2CCCN(C=O)CC2)ccc1OC ZINC000880665292 DD On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N2CCC(N3CCOC3=O)CC2)ccc1OC ZINC000880665299 FE On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CCC(N3CCOC3=O)CC2)ccc1OC ZINC000880665299 FE On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NCc2ccc(Cl)c(C(=O)OC)n2)ccc1OC ZINC000880665300 GF On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)NCc2ccc(Cl)c(C(=O)OC)n2)ccc1OC ZINC000880665300 GF On-Demand Anodyne ENPP1 55 33 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880665303 FE On-Demand Anodyne GABRA1 16 41 COCc1cc(NC(=O)NNC(=O)c2cc(C)cs2)ccc1OC ZINC000880665308 EF On-Demand Reactive QRFPR 45 48 C[S@](=O)[C@H]1CCC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880665309 FE On-Demand Anodyne GABRA1 16 41 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880665310 FE On-Demand Anodyne GABRA1 16 41 COCc1cc(NC(=O)NCc2ccc(Br)cn2)ccc1OC ZINC000880665313 GG On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NCc2ccc(Br)cn2)ccc1OC ZINC000880665313 GG On-Demand Anodyne HTR2A 22 41 COCc1cc(NC(=O)NCc2ccc(Br)cn2)ccc1OC ZINC000880665313 GG On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NCc2ccc(Br)cn2)ccc1OC ZINC000880665313 GG On-Demand Anodyne ENPP1 48 39 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880665315 FE On-Demand Anodyne GABRA1 16 41 CC[C@@H](C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665319 CF On-Demand Anodyne TSHR 47 32 CC[C@@H](C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665319 CF On-Demand Anodyne ENPP1 59 31 CC[C@H](C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665320 CF On-Demand Anodyne TSHR 47 32 CC[C@H](C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665320 CF On-Demand Anodyne ENPP1 59 31 COCc1cc(NC(=O)NCC[C@@H]2CCCS2)ccc1OC ZINC000880665322 DG On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)NCC[C@@H]2CCCS2)ccc1OC ZINC000880665322 DG On-Demand Anodyne QRFPR 46 39 COCc1cc(NC(=O)NCC[C@@H]2CCCS2)ccc1OC ZINC000880665322 DG On-Demand Anodyne PRMT3 33 42 COCc1cc(NC(=O)NCC[C@H]2CCCS2)ccc1OC ZINC000880665323 DG On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)NCC[C@H]2CCCS2)ccc1OC ZINC000880665323 DG On-Demand Anodyne QRFPR 46 39 COCc1cc(NC(=O)NCC[C@H]2CCCS2)ccc1OC ZINC000880665323 DG On-Demand Anodyne PRMT3 33 42 COCc1cc(NC(=O)N2CC3(CCOC3)C2)ccc1OC ZINC000880665324 DE On-Demand Anodyne ENPP1 62 34 C=C(C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665333 CE On-Demand Mild TSHR 55 32 C=C(C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665333 CE On-Demand Mild QRFPR 40 33 C=C(C)CONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665333 CE On-Demand Mild ENPP1 61 32 C=C[C@H](C)ONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665335 CE On-Demand Mild TSHR 41 30 C=C[C@H](C)ONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665335 CE On-Demand Mild ENPP1 49 31 C=C[C@@H](C)ONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665336 CE On-Demand Mild TSHR 41 30 C=C[C@@H](C)ONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665336 CE On-Demand Mild ENPP1 49 31 COCc1cc(NC(=O)N2CCc3cccc(NC(C)=O)c3C2)ccc1OC ZINC000880665346 GG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)N2CCc3cccc(NC(C)=O)c3C2)ccc1OC ZINC000880665346 GG On-Demand Anodyne P2RY14 47 33 COCc1cc(NC(=O)N2CCc3cccc(NC(C)=O)c3C2)ccc1OC ZINC000880665346 GG On-Demand Anodyne ABCG2 22 40 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880665351 FE On-Demand Anodyne QRFPR 40 32 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880665351 FE On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NOCCOC(C)C)ccc1OC ZINC000880665353 DE On-Demand Anodyne ENPP1 67 33 COCc1cc(NC(=O)N2C[C@H]3C[C@H]2C(=O)O3)ccc1OC ZINC000880665378 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2C[C@H]3C[C@H]2C(=O)O3)ccc1OC ZINC000880665378 DD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H]2C[C@H]3C[C@@]3(C(=O)OC)C2)ccc1OC ZINC000880665380 EE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N(C)C[C@](C)(O)c2ccccc2)ccc1OC ZINC000880665383 FG On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)N(C)C[C@@](C)(O)c2ccccc2)ccc1OC ZINC000880665385 FG On-Demand Anodyne TSHR 55 33 C[C@@H](CNC(=O)Nc1ccccc1-c1nnnn1C)N1CCCCC1 ZINC000880665397 ED On-Demand Anodyne CCR3 61 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(CCN2CCOCC2)CC1 ZINC000880665424 GD On-Demand Anodyne CASR 42 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(CCN2CCOCC2)CC1 ZINC000880665424 GD On-Demand Anodyne CCR3 57 45 CC(C)(C)OC(=O)N1CCc2nc(NC(=O)C3(c4ccc(F)cc4)CCC3)sc2C1 ZINC000880665425 IJ On-Demand Anodyne SLC27A1 50 44 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@@H]1CC1(Cl)Cl ZINC000880665436 FF On-Demand Anodyne CCR3 28 42 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@H]1CC1(Cl)Cl ZINC000880665437 FF On-Demand Anodyne CCR3 28 42 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)ccc1OC ZINC000880665438 GE On-Demand Mild PDGFRB 63 46 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)ccc1OC ZINC000880665438 GE On-Demand Mild CHEK1 15 40 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)ccc1OC ZINC000880665438 GE On-Demand Mild ENPP1 40 31 COCc1cc(NC(=O)N[C@@H]2C[C@@H](S(C)(=O)=O)C2)ccc1OC ZINC000880665440 ED On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N[C@@H]2C[C@@H](S(C)(=O)=O)C2)ccc1OC ZINC000880665440 ED On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@@H]2C[C@@H](S(C)(=O)=O)C2)ccc1OC ZINC000880665440 ED On-Demand Anodyne ENPP1 45 30 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880665444 GF On-Demand Anodyne CCR3 53 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880665445 GF On-Demand Anodyne CCR3 53 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880665446 GF On-Demand Anodyne CCR3 53 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1[C@H](O)c1ccccc1 ZINC000880665447 GF On-Demand Anodyne CCR3 53 42 COCc1cc(NC(=O)NC2([C@@H]3CCCCO3)CCC2)ccc1OC ZINC000880665448 EG On-Demand Anodyne QRFPR 49 41 COCc1cc(NC(=O)NC2([C@H]3CCCCO3)CCC2)ccc1OC ZINC000880665449 EG On-Demand Anodyne QRFPR 49 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880665455 ED On-Demand Anodyne CCR3 59 49 COCc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2nccn2C)ccc1OC ZINC000880665456 GF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2nccn2C)ccc1OC ZINC000880665456 GF On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2nccn2C)ccc1OC ZINC000880665456 GF On-Demand Anodyne ENPP1 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880665457 ED On-Demand Anodyne CCR3 59 49 COCc1cc(NC(=O)NCc2cc(C(=O)OC)co2)ccc1OC ZINC000880665458 EF On-Demand Anodyne TSHR 47 31 Cn1nnnc1-c1ccccc1NC(=O)N1CCN(c2cccc(F)n2)CC1 ZINC000880665459 GD On-Demand Anodyne CCR3 25 41 COCc1cc(NC(=O)NNC(=O)[C@]2(C)CCCO2)ccc1OC ZINC000880665460 ED On-Demand Reactive QRFPR 41 33 COCc1cc(NC(=O)NNC(=O)[C@@]2(C)CCCO2)ccc1OC ZINC000880665461 ED On-Demand Reactive QRFPR 41 33 C#C[C@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665462 CC On-Demand Mild ENPP1 56 32 C#C[C@@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665464 CC On-Demand Mild ENPP1 56 32 C#C[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)C1CCOCC1 ZINC000880665466 EE On-Demand Mild QRFPR 41 34 C#C[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)C1CCOCC1 ZINC000880665468 EE On-Demand Mild QRFPR 41 34 C#CC1CCN(C(=O)Nc2ccccc2-c2nnnn2C)CC1 ZINC000880665473 DD On-Demand Mild CCR3 19 41 COCc1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1OC ZINC000880665477 EE On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1OC ZINC000880665477 EE On-Demand Anodyne PDGFRB 46 44 COCc1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1OC ZINC000880665477 EE On-Demand Anodyne EPHX2 29 42 COCc1cc(NC(=O)N2CCCc3n[nH]cc32)ccc1OC ZINC000880665479 DF On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)N2CCCc3n[nH]cc32)ccc1OC ZINC000880665479 DF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCCc3n[nH]cc32)ccc1OC ZINC000880665479 DF On-Demand Anodyne ENPP1 62 33 Cn1nnnc1-c1ccccc1NC(=O)NC(C)(C)[C@@H]1CCCCO1 ZINC000880665480 EE On-Demand Anodyne CCR3 22 44 Cn1nnnc1-c1ccccc1NC(=O)NC(C)(C)[C@H]1CCCCO1 ZINC000880665482 EE On-Demand Anodyne CCR3 22 44 COCc1cc(NC(=O)N[C@@H]2C[C@@H](SC)C2)ccc1OC ZINC000880665485 DF On-Demand Anodyne TSHR 59 31 COCc1cc(NC(=O)N[C@@H]2C[C@@H](SC)C2)ccc1OC ZINC000880665485 DF On-Demand Anodyne QRFPR 48 39 COCc1cc(NC(=O)N[C@@H]2C[C@@H](SC)C2)ccc1OC ZINC000880665485 DF On-Demand Anodyne ENPP1 60 31 Cn1nnnc1-c1ccccc1NC(=O)NOCC1CC1 ZINC000880665486 CD On-Demand Anodyne CCR3 64 47 COCc1cc(NC(=O)N[C@@H]2C[C@H]3C[C@H]2[C@@H]2C[C@@H]32)ccc1OC ZINC000880665487 DG On-Demand Anodyne QRFPR 43 34 Cn1nnnc1-c1ccccc1NC(=O)NCC(Cl)Cl ZINC000880665488 DD On-Demand Reactive CCR3 30 42 COCc1cc(NC(=O)N[C@@H]2C[C@H]3C[C@H]2[C@@H]2C[C@H]32)ccc1OC ZINC000880665489 DG On-Demand Anodyne QRFPR 43 34 COCc1cc(NC(=O)N2CCN(CCCOC(C)(C)C)CC2)ccc1OC ZINC000880665490 GG On-Demand Anodyne HTR1A 22 46 COCc1cc(NC(=O)N2CCN(CCCOC(C)(C)C)CC2)ccc1OC ZINC000880665490 GG On-Demand Anodyne HTR1D 16 46 COCc1cc(NC(=O)N2CCN(CCCOC(C)(C)C)CC2)ccc1OC ZINC000880665490 GG On-Demand Anodyne HTR1B 17 46 COCc1cc(NC(=O)N2CCN(CCCOC(C)(C)C)CC2)ccc1OC ZINC000880665490 GG On-Demand Anodyne PDGFRB 55 43 COCc1cc(NC(=O)N[C@@H]2C[C@H]3C[C@H]2[C@H]2C[C@@H]23)ccc1OC ZINC000880665491 DG On-Demand Anodyne QRFPR 43 34 COCc1cc(NC(=O)N[C@@H]2C[C@H]3C[C@H]2[C@H]2C[C@H]23)ccc1OC ZINC000880665492 DG On-Demand Anodyne QRFPR 43 34 CCOc1ccc(NNC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880665493 EG On-Demand Reactive TSHR 61 37 CCOc1ccc(NNC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880665493 EG On-Demand Reactive PDGFRA 43 35 CCOc1ccc(NNC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880665493 EG On-Demand Reactive QRFPR 41 34 CCOc1ccc(NNC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880665493 EG On-Demand Reactive ENPP1 56 32 COCc1cc(NC(=O)N(C)CCN(C)C(=O)OC)ccc1OC ZINC000880665494 EE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N(C)CCN(C)C(=O)OC)ccc1OC ZINC000880665494 EE On-Demand Anodyne ENPP1 55 30 C#CCCCNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665500 CD On-Demand Mild CCR3 26 40 Cn1nnnc1-c1ccccc1NC(=O)NC1(C)CC(F)(F)C1 ZINC000880665502 DE On-Demand Anodyne CCR3 37 43 COCc1cc(NC(=O)N2CC=C[C@@H]2CO)ccc1OC ZINC000880665504 CD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC=C[C@@H]2CO)ccc1OC ZINC000880665504 CD On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CC=C[C@H]2CO)ccc1OC ZINC000880665506 CD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC=C[C@H]2CO)ccc1OC ZINC000880665506 CD On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NC2(c3ncccn3)CCC2)ccc1OC ZINC000880665513 EF On-Demand Anodyne TSHR 53 33 COCc1cc(NC(=O)NC2(c3ncccn3)CCC2)ccc1OC ZINC000880665513 EF On-Demand Anodyne PDGFRA 41 33 COCc1cc(NC(=O)NC2(c3ncccn3)CCC2)ccc1OC ZINC000880665513 EF On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)NC2(c3ncccn3)CCC2)ccc1OC ZINC000880665513 EF On-Demand Anodyne ENPP1 53 36 Cn1nnnc1-c1ccccc1NC(=O)NCC1Cc2ccccc2C1 ZINC000880665515 EE On-Demand Anodyne CCR3 47 46 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCOC2)ccc1OC ZINC000880665518 ED On-Demand Reactive QRFPR 45 37 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCOC2)ccc1OC ZINC000880665519 ED On-Demand Reactive QRFPR 45 37 COCc1cc(NC(=O)N[C@H](C2CCC2)[C@H]2CCOC2)ccc1OC ZINC000880665520 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H](C2CCC2)[C@@H]2CCOC2)ccc1OC ZINC000880665521 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H](C2CCC2)[C@H]2CCOC2)ccc1OC ZINC000880665522 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@H](C2CCC2)[C@@H]2CCOC2)ccc1OC ZINC000880665523 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NNc2nccnc2C2CCC2)ccc1OC ZINC000880665524 FG On-Demand Reactive TSHR 40 30 COCc1cc(NC(=O)NNc2nccnc2C2CCC2)ccc1OC ZINC000880665524 FG On-Demand Reactive QRFPR 43 36 C#CC1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665525 DF On-Demand Mild TSHR 67 34 C#CC1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665525 DF On-Demand Mild HTR1D 17 45 C#CC1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665525 DF On-Demand Mild HTR1B 20 45 C#CC1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665525 DF On-Demand Mild PDGFRB 42 36 C#CC1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880665525 DF On-Demand Mild QRFPR 44 36 COCc1cc(NC(=O)NCC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880665526 EH On-Demand Anodyne TSHR 65 31 COCc1cc(NC(=O)NCC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880665526 EH On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NCC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880665526 EH On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N(C)C[C@@]2(O)CCc3ccccc32)ccc1OC ZINC000880665533 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N(C)C[C@]2(O)CCc3ccccc32)ccc1OC ZINC000880665534 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NC[C@]23OCCC[C@H]2C3(F)F)ccc1OC ZINC000880665535 FF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCc3c([nH]c4ccc(OC)cc34)C2)ccc1OC ZINC000880665536 GH On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N2CCc3c([nH]c4ccc(OC)cc34)C2)ccc1OC ZINC000880665536 GH On-Demand Anodyne HTR1D 16 52 COCc1cc(NC(=O)N2CCc3c([nH]c4ccc(OC)cc34)C2)ccc1OC ZINC000880665536 GH On-Demand Anodyne HTR1B 18 52 C#CC[C@@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665538 DE On-Demand Mild CCR3 59 49 C#CC[C@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665541 DE On-Demand Mild CCR3 59 49 Cn1nnnc1-c1ccccc1NC(=O)NC1CCC(OC(C)(C)C)CC1 ZINC000880665543 FG On-Demand Anodyne CCR3 30 47 COCc1cc(NC(=O)NCCC2SCCS2)ccc1OC ZINC000880665544 EG On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCCC2SCCS2)ccc1OC ZINC000880665544 EG On-Demand Anodyne QRFPR 45 39 CCN(CCNC(=O)Nc1ccccc1-c1nnnn1C)C(C)C ZINC000880665545 ED On-Demand Anodyne CCR3 53 40 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880665547 ED On-Demand Anodyne CCR3 26 41 COCc1cc(NC(=O)N2Cc3ccccc3[C@@H](C)C2)ccc1OC ZINC000880665551 EH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2Cc3ccccc3[C@@H](C)C2)ccc1OC ZINC000880665551 EH On-Demand Anodyne HTR1B 15 42 COCc1cc(NC(=O)N2Cc3ccccc3[C@@H](C)C2)ccc1OC ZINC000880665551 EH On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@H]2C)ccc1OC ZINC000880665553 ED On-Demand Reactive TSHR 40 29 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@H]2C)ccc1OC ZINC000880665553 ED On-Demand Reactive QRFPR 47 38 COCc1cc(NC(=O)N2Cc3ccccc3[C@H](C)C2)ccc1OC ZINC000880665554 EH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2Cc3ccccc3[C@H](C)C2)ccc1OC ZINC000880665554 EH On-Demand Anodyne HTR1B 15 42 COCc1cc(NC(=O)N2Cc3ccccc3[C@H](C)C2)ccc1OC ZINC000880665554 EH On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCO[C@H]2C)ccc1OC ZINC000880665555 ED On-Demand Reactive TSHR 40 29 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCO[C@H]2C)ccc1OC ZINC000880665555 ED On-Demand Reactive QRFPR 47 38 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@@H]2C)ccc1OC ZINC000880665557 ED On-Demand Reactive TSHR 40 29 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@@H]2C)ccc1OC ZINC000880665557 ED On-Demand Reactive QRFPR 47 38 COCc1cc(NC(=O)N[C@@]2(c3ccccc3)C[C@@H](O)C2)ccc1OC ZINC000880665558 FG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)N[C@@]2(c3ccccc3)C[C@@H](O)C2)ccc1OC ZINC000880665558 FG On-Demand Anodyne QRFPR 43 39 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCO[C@@H]2C)ccc1OC ZINC000880665559 ED On-Demand Reactive TSHR 40 29 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCO[C@@H]2C)ccc1OC ZINC000880665559 ED On-Demand Reactive QRFPR 47 38 COCc1cc(NC(=O)NCC(C)(C)C(C)(F)F)ccc1OC ZINC000880665560 EH On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCCCCCNC(=O)CC2)ccc1OC ZINC000880665562 FF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCCCCCNC(=O)CC2)ccc1OC ZINC000880665562 FF On-Demand Anodyne ENPP1 41 33 Cn1nnnc1-c1ccccc1NC(=O)N1CCN(c2ccnc(F)c2)CC1 ZINC000880665563 GD On-Demand Anodyne CCR3 40 42 COCc1cc(NC(=O)NCc2ccc(N(C)C(C)=O)cc2)ccc1OC ZINC000880665564 FG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCc2ccc(N(C)C(C)=O)cc2)ccc1OC ZINC000880665564 FG On-Demand Anodyne ROCK2 19 42 COCc1cc(NC(=O)N(C)[C@@H]2CC(C)(C)OC2=O)ccc1OC ZINC000880665566 EE On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N(C)[C@H]2CC(C)(C)OC2=O)ccc1OC ZINC000880665567 EE On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NN(C)C(=O)OC)ccc1OC ZINC000880665568 CD On-Demand Reactive TSHR 40 31 COCc1cc(NC(=O)NN(C)C(=O)OC)ccc1OC ZINC000880665568 CD On-Demand Reactive QRFPR 41 34 COCc1cc(NC(=O)NN(C)C(=O)OC)ccc1OC ZINC000880665568 CD On-Demand Reactive ENPP1 55 31 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H]2C[C@@H]2Cc2ccccc2)n1 ZINC000880665569 EE On-Demand Anodyne CAPN2 41 36 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H]2C[C@H]2Cc2ccccc2)n1 ZINC000880665570 EE On-Demand Anodyne CAPN2 41 36 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H]2C[C@@H]2Cc2ccccc2)n1 ZINC000880665571 EE On-Demand Anodyne CAPN2 41 36 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H]2C[C@H]2Cc2ccccc2)n1 ZINC000880665573 EE On-Demand Anodyne CAPN2 41 36 Cn1nnnc1-c1ccccc1NC(=O)NOC1CCCC1 ZINC000880665574 DD On-Demand Anodyne CCR3 58 50 COCc1cc(NC(=O)NN=c2cc[nH]c(C)c2)ccc1OC ZINC000880665577 DE On-Demand Reactive ENPP1 62 33 COCc1cc(NC(=O)N2C[C@@H]3CC[C@H]2c2ccccc23)ccc1OC ZINC000880665582 FI On-Demand Anodyne TSHR 69 33 COCc1cc(NC(=O)N2C[C@@H]3CC[C@H]2c2ccccc23)ccc1OC ZINC000880665582 FI On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)N2CC(CC3CCOCC3)C2)ccc1OC ZINC000880665583 EG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC(CC3CCOCC3)C2)ccc1OC ZINC000880665583 EG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NC[C@@]23COCCN2C(=O)OC3)ccc1OC ZINC000880665588 FD On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NC[C@]23COCCN2C(=O)OC3)ccc1OC ZINC000880665590 FD On-Demand Anodyne TSHR 53 30 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CCC12CCOCC2 ZINC000880665591 FE On-Demand Anodyne CCR3 30 42 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CCC12CCOCC2 ZINC000880665593 FE On-Demand Anodyne CCR3 30 42 COCc1cc(NC(=O)NCc2cnc(Br)cn2)ccc1OC ZINC000880665595 GF On-Demand Anodyne TSHR 55 31 COCc1cc(NC(=O)NCc2cnc(Br)cn2)ccc1OC ZINC000880665595 GF On-Demand Anodyne ENPP1 53 36 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne TSHR 73 37 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne PDGFRB 42 40 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne GRM4 15 43 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne ROCK2 23 44 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne FLT4 21 40 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne PDGFRA 53 38 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne QPCT 15 42 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne PRMT3 61 35 COCc1cc(NC(=O)NCc2ncccn2)ccc1OC ZINC000880665599 DD On-Demand Anodyne ENPP1 73 39 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccccc1-c1nnnn1C ZINC000880665601 GD On-Demand Anodyne CCR3 23 42 COCc1cc(NC(=O)N[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665605 GG On-Demand Clean TSHR 57 34 COCc1cc(NC(=O)N[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665605 GG On-Demand Clean CCR3 21 43 COCc1cc(NC(=O)N[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665605 GG On-Demand Clean EPHX2 46 40 COCc1cc(NC(=O)N[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665605 GG On-Demand Clean MCHR1 24 45 COCc1cc(NC(=O)N[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665605 GG On-Demand Clean QRFPR 40 33 COCc1cc(NC(=O)N[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665607 GG On-Demand Clean TSHR 57 34 COCc1cc(NC(=O)N[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665607 GG On-Demand Clean CCR3 21 43 COCc1cc(NC(=O)N[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665607 GG On-Demand Clean EPHX2 46 40 COCc1cc(NC(=O)N[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665607 GG On-Demand Clean MCHR1 24 45 COCc1cc(NC(=O)N[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880665607 GG On-Demand Clean QRFPR 40 33 COCc1cc(NC(=O)NN2CCc3ccccc3C2=O)ccc1OC ZINC000880665609 FF On-Demand Anodyne TSHR 72 36 CCN1CC[C@@H]1CNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665611 DD On-Demand Anodyne CCR3 58 47 COCc1cc(NC(=O)NCc2cc(F)cnc2Cl)ccc1OC ZINC000880665612 FG On-Demand Anodyne TSHR 57 35 COCc1cc(NC(=O)NCc2cc(F)cnc2Cl)ccc1OC ZINC000880665612 FG On-Demand Anodyne ENPP1 53 36 COCc1cc(NC(=O)NN=c2cc[nH]cc2C)ccc1OC ZINC000880665614 DE On-Demand Reactive TSHR 47 31 COCc1cc(NC(=O)NN=c2cc[nH]cc2C)ccc1OC ZINC000880665614 DE On-Demand Reactive ENPP1 70 36 CN1CCN(C2CCN(C(=O)Nc3ccccc3-c3nnnn3C)CC2)CC1 ZINC000880665615 GD On-Demand Anodyne CCR3 18 44 CN1CCN(C2CCN(C(=O)Nc3ccccc3-c3nnnn3C)CC2)CC1 ZINC000880665615 GD On-Demand Anodyne L3MBTL3 46 38 COCc1cc(NC(=O)N2CCC(C(C)(C)O)CC2)ccc1OC ZINC000880665616 EF On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N2CCC(C(C)(C)O)CC2)ccc1OC ZINC000880665616 EF On-Demand Anodyne HTR1D 15 46 COCc1cc(NC(=O)N2CCC(C(C)(C)O)CC2)ccc1OC ZINC000880665616 EF On-Demand Anodyne HTR1B 18 43 COCc1cc(NC(=O)N2CCC(C(C)(C)O)CC2)ccc1OC ZINC000880665616 EF On-Demand Anodyne PDGFRB 41 39 COCc1cc(NC(=O)N2CCC(C(C)(C)O)CC2)ccc1OC ZINC000880665616 EF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCCC[C@H]2COC(=O)NC2CC2)ccc1OC ZINC000880665617 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NCC2(OC(C)C)CCC2)ccc1OC ZINC000880665628 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NCC2(OC(C)C)CCC2)ccc1OC ZINC000880665628 EG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(CCO)C3)ccc1OC ZINC000880665629 EF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(CCO)C3)ccc1OC ZINC000880665629 EF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@](OC)(C(F)(F)F)C2)ccc1OC ZINC000880665630 FG On-Demand Anodyne EPHX2 34 44 COCc1cc(NC(=O)N2CC[C@](OC)(C(F)(F)F)C2)ccc1OC ZINC000880665631 FG On-Demand Anodyne EPHX2 34 44 Cn1nnnc1-c1ccccc1NC(=O)NCCOC1CCC1 ZINC000880665632 DD On-Demand Anodyne CCR3 48 45 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne HTR1D 21 46 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne HTR1B 23 46 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne PDGFRB 45 37 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne EPHX2 36 42 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne RBP4 27 42 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne QRFPR 47 38 COCc1cc(NC(=O)N2CCC(F)CC2)ccc1OC ZINC000880665634 CF On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)NCCC(C)(C)COC)ccc1OC ZINC000880665635 DG On-Demand Anodyne TSHR 48 31 Cc1cccc2c1CCN(C(=O)Nc1ccccc1-c1nnnn1C)C2 ZINC000880665732 EF On-Demand Anodyne P2RY14 47 37 COCc1cc(NC(=O)N2CCCC[C@@H]2COC(=O)NC2CC2)ccc1OC ZINC000880665736 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@H]2CCCC23OCCO3)ccc1OC ZINC000880665737 EE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N[C@H]2CCCC23OCCO3)ccc1OC ZINC000880665737 EE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@@H]2CCCC23OCCO3)ccc1OC ZINC000880665738 EE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N[C@@H]2CCCC23OCCO3)ccc1OC ZINC000880665738 EE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NCCS(=O)(=O)C2CC2)ccc1OC ZINC000880665739 ED On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)NCCS(=O)(=O)C2CC2)ccc1OC ZINC000880665739 ED On-Demand Anodyne QRFPR 45 36 COCc1cc(NC(=O)NCC[C@@H]2CCCS2(=O)=O)ccc1OC ZINC000880665744 FD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NCC[C@H]2CCCS2(=O)=O)ccc1OC ZINC000880665746 FD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NCc2cnnn2C)ccc1OC ZINC000880665755 DD On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCc2cnnn2C)ccc1OC ZINC000880665755 DD On-Demand Anodyne HTR2A 36 42 COCc1cc(NC(=O)NCc2cnnn2C)ccc1OC ZINC000880665755 DD On-Demand Anodyne ENPP1 71 35 COCc1cc(NC(=O)Nc2cc3n(n2)CCN(C)C3)ccc1OC ZINC000880665756 EE On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N2C[C@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665757 DF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2C[C@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665757 DF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2C[C@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665757 DF On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N2C[C@@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665759 DF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2C[C@@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665759 DF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2C[C@@H]3[C@H](C2)C3(F)F)ccc1OC ZINC000880665759 DF On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N2C[C@@H]3[C@@H](C2)C3(F)F)ccc1OC ZINC000880665761 DF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2C[C@@H]3[C@@H](C2)C3(F)F)ccc1OC ZINC000880665761 DF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2C[C@@H]3[C@@H](C2)C3(F)F)ccc1OC ZINC000880665761 DF On-Demand Anodyne ENPP1 51 32 Cn1nnnc1-c1ccccc1NC(=O)NOC1CCC1 ZINC000880665762 CD On-Demand Anodyne CCR3 58 48 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne TSHR 41 33 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne HTR1B 17 41 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne PDGFRB 49 38 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne P2RY14 50 39 COCc1cc(NC(=O)N2CCc3ncncc3C2)ccc1OC ZINC000880665764 EE On-Demand Anodyne ENPP1 49 37 COCc1cc(NC(=O)NC[C@@H]2CCO[C@H]2c2cn[nH]c2)ccc1OC ZINC000880665770 FE On-Demand Anodyne TSHR 51 33 COCc1cc(NC(=O)NC[C@@H]2CCO[C@H]2c2cn[nH]c2)ccc1OC ZINC000880665770 FE On-Demand Anodyne ROCK2 30 47 COCc1cc(NC(=O)NC[C@@H]2CCO[C@H]2c2cn[nH]c2)ccc1OC ZINC000880665770 FE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC[C@@H]2CCO[C@H]2c2cn[nH]c2)ccc1OC ZINC000880665770 FE On-Demand Anodyne ENPP1 62 34 COCc1cc(NC(=O)NC[C@H]2CN(C3CC3)C(=O)O2)ccc1OC ZINC000880665776 ED On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)NC[C@H]2CN(C3CC3)C(=O)O2)ccc1OC ZINC000880665776 ED On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC[C@@H]2CN(C3CC3)C(=O)O2)ccc1OC ZINC000880665779 ED On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)NC[C@@H]2CN(C3CC3)C(=O)O2)ccc1OC ZINC000880665779 ED On-Demand Anodyne QRFPR 44 36 C#CC[C@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665781 CD On-Demand Mild QRFPR 41 33 C#CC[C@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665781 CD On-Demand Mild ENPP1 55 31 C#CC[C@@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665783 CD On-Demand Mild QRFPR 41 33 C#CC[C@@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665783 CD On-Demand Mild ENPP1 55 31 C#C[C@@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665785 DD On-Demand Mild CCR3 52 45 C#C[C@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665786 DD On-Demand Mild CCR3 52 45 COCc1cc(NC(=O)NC[C@@H](CO)Cc2ccoc2)ccc1OC ZINC000880665788 EE On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NC[C@@H](CO)Cc2ccoc2)ccc1OC ZINC000880665788 EE On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)NC[C@H](CO)Cc2ccoc2)ccc1OC ZINC000880665790 EE On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NC[C@H](CO)Cc2ccoc2)ccc1OC ZINC000880665790 EE On-Demand Anodyne ENPP1 62 33 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665792 FE On-Demand Anodyne CCR3 48 45 COCc1cc(NC(=O)NNC(=O)[C@@H]2CC[C@H](C)O2)ccc1OC ZINC000880665793 ED On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NNC(=O)[C@@H]2CC[C@H](C)O2)ccc1OC ZINC000880665793 ED On-Demand Reactive ENPP1 44 30 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880665794 FE On-Demand Anodyne CCR3 48 45 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880665798 FF On-Demand Anodyne TSHR 60 33 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880665798 FF On-Demand Anodyne QRFPR 40 33 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880665798 FF On-Demand Anodyne ENPP1 63 33 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880665805 EE On-Demand Anodyne CCR3 36 43 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880665806 EE On-Demand Anodyne CCR3 36 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2C=C[C@H]1C2 ZINC000880665807 CD On-Demand Anodyne CCR3 18 41 COCc1cc(NC(=O)N2CC3(CNC(=O)O3)C2)ccc1OC ZINC000880665808 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC3(CNC(=O)O3)C2)ccc1OC ZINC000880665808 DD On-Demand Anodyne ENPP1 58 36 C[C@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@@H](C(F)(F)F)O1 ZINC000880665809 GE On-Demand Anodyne CCR3 21 41 C[C@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@@H](C(F)(F)F)O1 ZINC000880665809 GE On-Demand Anodyne RBP4 47 34 C[C@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@H](C(F)(F)F)O1 ZINC000880665810 GE On-Demand Anodyne CCR3 21 41 C[C@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@H](C(F)(F)F)O1 ZINC000880665810 GE On-Demand Anodyne RBP4 47 34 C[C@@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@@H](C(F)(F)F)O1 ZINC000880665811 GE On-Demand Anodyne CCR3 21 41 C[C@@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@@H](C(F)(F)F)O1 ZINC000880665811 GE On-Demand Anodyne RBP4 47 34 C[C@@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@H](C(F)(F)F)O1 ZINC000880665813 GE On-Demand Anodyne CCR3 21 41 C[C@@H]1CN(C(=O)Nc2ccccc2-c2nnnn2C)CC[C@H](C(F)(F)F)O1 ZINC000880665813 GE On-Demand Anodyne RBP4 47 34 COCc1cc(NC(=O)NC[C@@H]2CCC3(CCC3)O2)ccc1OC ZINC000880665819 EG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)NC[C@H]2CCC3(CCC3)O2)ccc1OC ZINC000880665821 EG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)N2C[C@@H](CN(C)C)[C@H](CN(C)C)C2)ccc1OC ZINC000880665822 GE On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N2C[C@@H](CN(C)C)[C@H](CN(C)C)C2)ccc1OC ZINC000880665822 GE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2C[C@@H](CN(C)C)[C@H](CN(C)C)C2)ccc1OC ZINC000880665822 GE On-Demand Anodyne ENPP1 63 34 COCc1cc(NC(=O)N2CCCN(C(=O)CC(C)C)CC2)ccc1OC ZINC000880665823 GF On-Demand Anodyne PDGFRB 45 39 COCc1cc(NC(=O)N2CCCN(C(=O)CC(C)C)CC2)ccc1OC ZINC000880665823 GF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCCN(C(=O)CC(C)C)CC2)ccc1OC ZINC000880665823 GF On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N(C)c2ccc(C)cc2)ccc1OC ZINC000880665824 DH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N(C)c2ccc(C)cc2)ccc1OC ZINC000880665824 DH On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne ADRB2 25 43 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne ADRB1 41 32 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne SOAT1 24 42 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne ENPP1 54 31 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne KCNK3 50 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2OC)ccc1OC ZINC000880665838 FF On-Demand Anodyne KCNK9 43 40 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne EPHX2 38 42 COCc1cc(NC(=O)N2CCC(NC(=O)OC)CC2)ccc1OC ZINC000880665840 FE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC(CF)CF)ccc1OC ZINC000880665842 CE On-Demand Anodyne TSHR 52 32 COCc1cc(NC(=O)NC(CF)CF)ccc1OC ZINC000880665842 CE On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)NC(CF)CF)ccc1OC ZINC000880665842 CE On-Demand Anodyne ENPP1 57 32 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne MME 43 37 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne TIMP3 53 32 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne CAPNS1 59 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne HLA-DRB1 53 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne CAPN1 68 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne CAPN2 92 38 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne ACE2 51 37 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665851 ED On-Demand Anodyne FPR1 44 34 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne MME 43 37 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne TIMP3 53 32 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne CAPNS1 59 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne HLA-DRB1 53 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne CAPN1 68 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne CAPN2 92 38 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne ACE2 51 37 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665853 ED On-Demand Anodyne FPR1 44 34 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne MME 43 37 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne TIMP3 53 32 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne CAPNS1 59 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne HLA-DRB1 53 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne CAPN1 68 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne CAPN2 92 38 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne ACE2 51 37 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](F)Cc2ccccc2)n1 ZINC000880665855 ED On-Demand Anodyne FPR1 44 34 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne MME 43 37 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne TIMP3 53 32 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne CAPNS1 59 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne HLA-DRB1 53 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne CAPN1 68 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne CAPN2 92 38 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne ACE2 51 37 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](F)Cc2ccccc2)n1 ZINC000880665856 ED On-Demand Anodyne FPR1 44 34 C#CCN(C(=O)Nc1ccccc1-c1nnnn1C)C1CC1 ZINC000880665857 CD On-Demand Mild CCR3 24 43 C#CCN(C(=O)Nc1ccccc1-c1nnnn1C)C1CCCC1 ZINC000880665859 DE On-Demand Mild CCR3 29 45 COCc1cc(NC(=O)N[C@](C)(CC(=O)OC)C2CC2)ccc1OC ZINC000880665862 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)N[C@](C)(CC(=O)OC)C2CC2)ccc1OC ZINC000880665862 FF On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N[C@@](C)(CC(=O)OC)C2CC2)ccc1OC ZINC000880665864 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)N[C@@](C)(CC(=O)OC)C2CC2)ccc1OC ZINC000880665864 FF On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccc1OC ZINC000880665865 EF On-Demand Anodyne PDE4A 15 41 COCc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccc1OC ZINC000880665865 EF On-Demand Anodyne QRFPR 48 39 COCc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccc1OC ZINC000880665865 EF On-Demand Anodyne PRMT3 35 45 COCc1cc(NC(=O)NCC[C@H](O)C2CCCC2)ccc1OC ZINC000880665865 EF On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccc1OC ZINC000880665866 EF On-Demand Anodyne PDE4A 15 41 COCc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccc1OC ZINC000880665866 EF On-Demand Anodyne QRFPR 48 39 COCc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccc1OC ZINC000880665866 EF On-Demand Anodyne PRMT3 35 45 COCc1cc(NC(=O)NCC[C@@H](O)C2CCCC2)ccc1OC ZINC000880665866 EF On-Demand Anodyne ENPP1 55 31 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H](C1CCC1)[C@H]1CCOC1 ZINC000880665868 FE On-Demand Anodyne CCR3 44 33 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H](C1CCC1)[C@@H]1CCOC1 ZINC000880665871 FE On-Demand Anodyne CCR3 44 33 Cn1nnnc1-c1ccccc1NC(=O)N[C@H](C1CCC1)[C@@H]1CCOC1 ZINC000880665873 FE On-Demand Anodyne CCR3 44 33 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne HTR2A 46 43 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne HTR2C 17 43 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne PDGFRA 44 35 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)Nc2cnn(C)c2C2CC2)ccc1OC ZINC000880665874 EG On-Demand Anodyne ENPP1 52 33 Cn1nnnc1-c1ccccc1NC(=O)N[C@H](C1CCC1)[C@H]1CCOC1 ZINC000880665875 FE On-Demand Anodyne CCR3 44 33 COCc1cc(NC(=O)N2CCN(C)C(C)(C)CC2)ccc1OC ZINC000880665878 EF On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N2CCN(C)C(C)(C)CC2)ccc1OC ZINC000880665878 EF On-Demand Anodyne HTR1D 15 46 COCc1cc(NC(=O)N2CCN(C)C(C)(C)CC2)ccc1OC ZINC000880665878 EF On-Demand Anodyne HTR1B 18 46 COCc1cc(NC(=O)N2CCN(C)C(C)(C)CC2)ccc1OC ZINC000880665878 EF On-Demand Anodyne PDGFRB 49 39 COCc1cc(NC(=O)NC2CCC(OC(C)(C)C)CC2)ccc1OC ZINC000880665880 FI On-Demand Anodyne EPHX2 52 40 COCc1cc(NC(=O)NC2CCC(OC(C)(C)C)CC2)ccc1OC ZINC000880665880 FI On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne HTR1D 18 50 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne HTR1B 21 50 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC3(CCN(C)CC3)CC2)ccc1OC ZINC000880665882 FG On-Demand Anodyne ENPP1 63 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C\c2csc(C(F)(F)F)c2)n1 ZINC000880665884 GF On-Demand Anodyne UL26 58 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C\c2csc(C(F)(F)F)c2)n1 ZINC000880665884 GF On-Demand Anodyne SCAF_EBVB9 49 33 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C\c2csc(C(F)(F)F)c2)n1 ZINC000880665885 GF On-Demand Anodyne UL26 58 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C\c2csc(C(F)(F)F)c2)n1 ZINC000880665885 GF On-Demand Anodyne SCAF_EBVB9 49 33 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C/c2csc(C(F)(F)F)c2)n1 ZINC000880665886 GF On-Demand Anodyne UL26 58 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C/c2csc(C(F)(F)F)c2)n1 ZINC000880665886 GF On-Demand Anodyne SCAF_EBVB9 49 33 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C/c2csc(C(F)(F)F)c2)n1 ZINC000880665888 GF On-Demand Anodyne UL26 58 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C/c2csc(C(F)(F)F)c2)n1 ZINC000880665888 GF On-Demand Anodyne SCAF_EBVB9 49 33 COCc1cc(NC(=O)NC[C@@H]2CCC3(CCOCC3)CO2)ccc1OC ZINC000880665889 GF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@H]2CCC3(CCOCC3)CO2)ccc1OC ZINC000880665891 GF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NCC2C[C@@H]3CC[C@H](C2)S3(=O)=O)ccc1OC ZINC000880665898 GE On-Demand Anodyne QRFPR 48 39 COCc1cc(NC(=O)N[C@@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665903 GF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665903 GF On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N[C@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665904 GF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H]2C[C@H]3CC[C@H]2N(C(=O)OC)C3)ccc1OC ZINC000880665904 GF On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N[C@H]2[C@@H]3CN(C(=O)OC(C)(C)C)C[C@@H]32)ccc1OC ZINC000880665907 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@H]2[C@@H]3CN(C(=O)OC(C)(C)C)C[C@@H]32)ccc1OC ZINC000880665907 GF On-Demand Anodyne ENPP1 55 30 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880665908 EF On-Demand Anodyne QRFPR 41 34 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(CCCO)CC1 ZINC000880665910 ED On-Demand Anodyne CCR3 47 43 COCc1cc(NC(=O)N2CCCNC(=O)C2)ccc1OC ZINC000880665913 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCCNC(=O)C2)ccc1OC ZINC000880665913 DD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCCNC(=O)C2)ccc1OC ZINC000880665913 DD On-Demand Anodyne ENPP1 62 34 CN(C(=O)Nc1ccccc1-c1nnnn1C)[C@@H]1CCN(CC(F)(F)F)C1=O ZINC000880665914 GD On-Demand Anodyne CCR3 33 44 CN(C(=O)Nc1ccccc1-c1nnnn1C)[C@H]1CCN(CC(F)(F)F)C1=O ZINC000880665916 GD On-Demand Anodyne CCR3 33 44 COCc1cc(NC(=O)N2CC[C@H](NC(=O)OC(C)(C)C)[C@@H]2C)ccc1OC ZINC000880665917 GG On-Demand Anodyne QRFPR 43 36 CCC1(CC)CCCN1C(=O)Nc1ccccc1-c1nnnn1C ZINC000880665918 EG On-Demand Anodyne CCR3 20 41 COCc1cc(NC(=O)N2C[C@@H](COC)[C@H](c3cnn(C)c3)C2)ccc1OC ZINC000880665919 GE On-Demand Anodyne ENPP1 50 33 Cn1nnnc1-c1ccccc1NC(=O)NOC1CCCCC1 ZINC000880665920 DE On-Demand Anodyne CCR3 56 49 Cn1nnnc1-c1ccccc1NC(=O)N1CC(CC2CCOCC2)C1 ZINC000880665923 FE On-Demand Anodyne CCR3 36 43 COCc1cc(NC(=O)N[C@H]2CC(=O)N(CC3CC3)C2)ccc1OC ZINC000880665926 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@H]2CC(=O)N(CC3CC3)C2)ccc1OC ZINC000880665926 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H]2CC(=O)N(CC3CC3)C2)ccc1OC ZINC000880665927 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@@H]2CC(=O)N(CC3CC3)C2)ccc1OC ZINC000880665927 ED On-Demand Anodyne QRFPR 40 33 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1C[C@H]1C1CCOCC1 ZINC000880665928 FE On-Demand Anodyne CCR3 25 43 COCc1cc(NC(=O)N2CCO[C@H](C(F)(F)F)CC2)ccc1OC ZINC000880665930 FG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CCO[C@H](C(F)(F)F)CC2)ccc1OC ZINC000880665930 FG On-Demand Anodyne EPHX2 37 40 COCc1cc(NC(=O)N2CCO[C@H](C(F)(F)F)CC2)ccc1OC ZINC000880665930 FG On-Demand Anodyne RBP4 27 41 COCc1cc(NC(=O)N2CCO[C@H](C(F)(F)F)CC2)ccc1OC ZINC000880665930 FG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCO[C@@H](C(F)(F)F)CC2)ccc1OC ZINC000880665931 FG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CCO[C@@H](C(F)(F)F)CC2)ccc1OC ZINC000880665931 FG On-Demand Anodyne EPHX2 37 40 COCc1cc(NC(=O)N2CCO[C@@H](C(F)(F)F)CC2)ccc1OC ZINC000880665931 FG On-Demand Anodyne RBP4 27 41 COCc1cc(NC(=O)N2CCO[C@@H](C(F)(F)F)CC2)ccc1OC ZINC000880665931 FG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC[C@@H](c3nccs3)C2)ccc1OC ZINC000880665933 EG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@@H](c3nccs3)C2)ccc1OC ZINC000880665933 EG On-Demand Anodyne HTR1B 15 41 COCc1cc(NC(=O)N2CC[C@@H](c3nccs3)C2)ccc1OC ZINC000880665933 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)N2CC[C@@H](c3nccs3)C2)ccc1OC ZINC000880665933 EG On-Demand Anodyne ENPP1 46 33 C[C@H](Cc1ccco1)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665937 EE On-Demand Anodyne CCR3 41 38 C[C@@H](Cc1ccco1)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880665938 EE On-Demand Anodyne CCR3 41 38 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2ccc3c(C#N)c[nH]c3c2)C1 ZINC000880665957 EE On-Demand Mild EZH2 50 40 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2ccc3c(C#N)c[nH]c3c2)C1 ZINC000880665958 EE On-Demand Mild EZH2 50 40 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2ccc3c(C#N)c[nH]c3c2)C1 ZINC000880665959 EE On-Demand Mild EZH2 50 40 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2ccc3c(C#N)c[nH]c3c2)C1 ZINC000880665960 EE On-Demand Mild EZH2 50 40 O=C(c1cnc2cc[nH]c2c1)N1CCCC2(CCCC2)CC1 ZINC000880665965 CH On-Demand Anodyne ACACA 33 58 COCc1cc(NC(=O)N2CC[C@H](c3nccs3)C2)ccc1OC ZINC000880665972 EG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@H](c3nccs3)C2)ccc1OC ZINC000880665972 EG On-Demand Anodyne HTR1B 15 41 COCc1cc(NC(=O)N2CC[C@H](c3nccs3)C2)ccc1OC ZINC000880665972 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)N2CC[C@H](c3nccs3)C2)ccc1OC ZINC000880665972 EG On-Demand Anodyne ENPP1 46 33 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Cc2ccc3cccnc3c2)C1 ZINC000880665973 EF On-Demand Anodyne CDK5 17 43 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Cc2ccc3cccnc3c2)C1 ZINC000880665975 EF On-Demand Anodyne CDK5 17 43 COc1ccc(N2CC[C@H](NC(=O)Nc3ccccc3-c3nnnn3C)C2)cc1 ZINC000880665976 GE On-Demand Clean CCR3 42 45 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Cc2ccc3cccnc3c2)C1 ZINC000880665977 EF On-Demand Anodyne CDK5 17 43 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Cc2ccc3cccnc3c2)C1 ZINC000880665979 EF On-Demand Anodyne CDK5 17 43 COCc1cc(NC(=O)N[C@@H]2COC3(CCC3)C2)ccc1OC ZINC000880665980 DF On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)N[C@H]2COC3(CCC3)C2)ccc1OC ZINC000880665982 DF On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccc1OC ZINC000880665992 EG On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccc1OC ZINC000880665992 EG On-Demand Anodyne EPHX2 23 45 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H]1CCC1(C)C ZINC000880665994 DE On-Demand Anodyne CCR3 26 47 Cn1nnnc1-c1ccccc1NC(=O)N[C@H]1CCC1(C)C ZINC000880665996 DE On-Demand Anodyne CCR3 26 47 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CCC(C)(C)CO1 ZINC000880666002 EE On-Demand Anodyne CCR3 41 42 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CCC(C)(C)CO1 ZINC000880666004 EE On-Demand Anodyne CCR3 41 42 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CCC=CO1 ZINC000880666008 DD On-Demand Anodyne CCR3 37 42 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CCC=CO1 ZINC000880666010 DD On-Demand Anodyne CCR3 37 42 C#CC1(NC(=O)Nc2ccc(OC)c(COC)c2)CCCC1 ZINC000880666012 DF On-Demand Mild QRFPR 42 35 COCc1cc(NC(=O)N[C@@H]2C[C@H]2C2CCOCC2)ccc1OC ZINC000880666014 EF On-Demand Anodyne QRFPR 42 35 Cn1nnnc1-c1ccccc1NC(=O)NN1CCCC1 ZINC000880666016 CD On-Demand Anodyne CCR3 39 47 COc1ccc(N2CCN(C(=O)Nc3ccccc3-c3nnnn3C)CC2)cc1 ZINC000880666017 GE On-Demand Clean CCR3 17 40 COc1ccc(N2CCN(C(=O)Nc3ccccc3-c3nnnn3C)CC2)cc1 ZINC000880666017 GE On-Demand Clean ABCG2 29 40 COCc1cc(NC(=O)NC2(C)CC(F)(F)C2)ccc1OC ZINC000880666018 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCCC[C@H](C3CCOCC3)C2)ccc1OC ZINC000880666019 GH On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CCCC[C@@H](C3CCOCC3)C2)ccc1OC ZINC000880666021 GH On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NNC(=O)C2CCOCC2)ccc1OC ZINC000880666023 ED On-Demand Reactive TSHR 46 31 COCc1cc(NC(=O)NNC(=O)C2CCOCC2)ccc1OC ZINC000880666023 ED On-Demand Reactive QRFPR 45 37 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880666029 GE On-Demand Anodyne CCR3 61 47 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880666035 GE On-Demand Anodyne CCR3 61 47 COCc1cc(NC(=O)N(C)CCNC(=O)OC(C)(C)C)ccc1OC ZINC000880666038 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@@H](C(=O)OC)C3)ccc1OC ZINC000880666040 EE On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@@H](C(=O)OC)C3)ccc1OC ZINC000880666040 EE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@@H](C(=O)OC)C3)ccc1OC ZINC000880666040 EE On-Demand Anodyne ENPP1 61 32 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](C)Cc2ccc(F)cc2)n1 ZINC000880666041 EE On-Demand Anodyne MME 20 40 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@H](C)Cc2ccc(F)cc2)n1 ZINC000880666041 EE On-Demand Anodyne ACE2 53 40 COc1cc(C)c(C)cc1NC(=O)c1cc(C)cnc1Cl ZINC000880666042 DH On-Demand Anodyne GRM4 19 41 COc1cc(C)c(C)cc1NC(=O)c1cc(C)cnc1Cl ZINC000880666042 DH On-Demand Anodyne KCNMA1 35 43 COc1cc(C)c(C)cc1NC(=O)c1cc(C)cnc1Cl ZINC000880666042 DH On-Demand Anodyne G2YM83_BOTF4 52 34 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@H](C(=O)OC)C3)ccc1OC ZINC000880666043 EE On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@H](C(=O)OC)C3)ccc1OC ZINC000880666043 EE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2[C@H](C(=O)OC)C3)ccc1OC ZINC000880666043 EE On-Demand Anodyne ENPP1 61 32 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](C)Cc2ccc(F)cc2)n1 ZINC000880666044 EE On-Demand Anodyne MME 20 40 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@H](C)Cc2ccc(F)cc2)n1 ZINC000880666044 EE On-Demand Anodyne ACE2 53 40 Cn1nnnc1-c1ccccc1NC(=O)NN1CCCCC1 ZINC000880666045 DD On-Demand Anodyne CCR3 36 46 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](C)Cc2ccc(F)cc2)n1 ZINC000880666046 EE On-Demand Anodyne MME 20 40 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)[C@@H](C)Cc2ccc(F)cc2)n1 ZINC000880666046 EE On-Demand Anodyne ACE2 53 40 COCc1cc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)ccc1OC ZINC000880666047 GF On-Demand Clean TSHR 66 32 COCc1cc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)ccc1OC ZINC000880666047 GF On-Demand Clean HTR1D 21 51 COCc1cc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)ccc1OC ZINC000880666047 GF On-Demand Clean HTR1B 26 48 COCc1cc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)ccc1OC ZINC000880666047 GF On-Demand Clean ROCK2 15 41 COCc1cc(NC(=O)NCc2ccc(N3CCN(C)CC3)cc2)ccc1OC ZINC000880666047 GF On-Demand Clean FLT3 21 43 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](C)Cc2ccc(F)cc2)n1 ZINC000880666048 EE On-Demand Anodyne MME 20 40 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)[C@@H](C)Cc2ccc(F)cc2)n1 ZINC000880666048 EE On-Demand Anodyne ACE2 53 40 Cn1nnnc1-c1ccccc1NC(=O)NCC(C)(C)CC(F)F ZINC000880666050 EF On-Demand Anodyne CCR3 34 41 COCc1cc(NC(=O)NC2CC3(CSC3)C2)ccc1OC ZINC000880666052 DF On-Demand Anodyne EPHX2 41 36 COCc1cc(NC(=O)NC2CC3(CSC3)C2)ccc1OC ZINC000880666052 DF On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)NC2CC3(CSC3)C2)ccc1OC ZINC000880666052 DF On-Demand Anodyne ENPP1 45 30 CCn1ncc(CNC(=O)Nc2ccc(OC)c(COC)c2)n1 ZINC000880666054 DD On-Demand Anodyne TSHR 55 33 CCn1ncc(CNC(=O)Nc2ccc(OC)c(COC)c2)n1 ZINC000880666054 DD On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)N2CCO[C@H](c3ccccc3OC)C2)ccc1OC ZINC000880666057 GG On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCO[C@H](c3ccccc3OC)C2)ccc1OC ZINC000880666057 GG On-Demand Anodyne QRFPR 41 38 COCc1cc(NC(=O)N2CCO[C@@H](c3ccccc3OC)C2)ccc1OC ZINC000880666062 GG On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCO[C@@H](c3ccccc3OC)C2)ccc1OC ZINC000880666062 GG On-Demand Anodyne QRFPR 41 38 C#CC1(F)CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666067 CE On-Demand Mild TSHR 52 30 C#CC1(F)CN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666067 CE On-Demand Mild ENPP1 41 33 COCc1cc(NC(=O)NCC[C@H]2CCCC2(F)F)ccc1OC ZINC000880666070 EH On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCN(C)[C@@H]2C)ccc1OC ZINC000880666072 FD On-Demand Reactive TSHR 42 32 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCN(C)[C@@H]2C)ccc1OC ZINC000880666072 FD On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NCC[C@@H]2CCCC2(F)F)ccc1OC ZINC000880666074 EH On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NCc2ncc(Cl)s2)ccc1OC ZINC000880666076 EG On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NCc2ncc(Cl)s2)ccc1OC ZINC000880666076 EG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCc2ncc(Cl)s2)ccc1OC ZINC000880666076 EG On-Demand Anodyne PRMT3 44 32 COCc1cc(NC(=O)NCc2ncc(Cl)s2)ccc1OC ZINC000880666076 EG On-Demand Anodyne ENPP1 47 36 COCc1cc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666080 GH On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666080 GH On-Demand Anodyne EPHX2 37 46 COCc1cc(NC(=O)N2CC[C@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666080 GH On-Demand Anodyne TRPM8 29 51 COCc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666082 GH On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666082 GH On-Demand Anodyne EPHX2 37 46 COCc1cc(NC(=O)N2CC[C@@]3(CCc4ccccc4O3)C2)ccc1OC ZINC000880666082 GH On-Demand Anodyne TRPM8 29 51 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](NC2CCOCC2)C1 ZINC000880666086 GD On-Demand Anodyne CCR3 51 45 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](NC2CCOCC2)C1 ZINC000880666090 GD On-Demand Anodyne CCR3 51 45 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(COC)c2)CCC1(F)F ZINC000880666096 GF On-Demand Anodyne ENPP1 45 30 CCN1CC[C@@H]1CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666097 DE On-Demand Anodyne DRD2 38 46 CCN1CC[C@@H]1CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666097 DE On-Demand Anodyne TSHR 61 33 CCN1CC[C@@H]1CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666097 DE On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N[C@H](C)c2nccnc2C)ccc1OC ZINC000880666102 EF On-Demand Anodyne TSHR 55 35 COCc1cc(NC(=O)N[C@H](C)c2nccnc2C)ccc1OC ZINC000880666102 EF On-Demand Anodyne ENPP1 48 34 COCc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)ccc1OC ZINC000880666103 FD On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)ccc1OC ZINC000880666103 FD On-Demand Anodyne CCR3 25 45 COCc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)ccc1OC ZINC000880666103 FD On-Demand Anodyne EPHX2 44 38 COCc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)ccc1OC ZINC000880666103 FD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H](C)c2nccnc2C)ccc1OC ZINC000880666107 EF On-Demand Anodyne TSHR 55 35 COCc1cc(NC(=O)N[C@@H](C)c2nccnc2C)ccc1OC ZINC000880666107 EF On-Demand Anodyne ENPP1 48 34 COCc1cc(NC(=O)NC[C@H]2CC(C(F)(F)F)=NO2)ccc1OC ZINC000880666115 FF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@@H]2CC(C(F)(F)F)=NO2)ccc1OC ZINC000880666118 FF On-Demand Anodyne QRFPR 40 33 C=C(C)C[C@@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666123 DE On-Demand Mild ENPP1 68 32 C=C(C)C[C@H](CO)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666126 DE On-Demand Mild ENPP1 68 32 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne HTR1D 17 44 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne HTR1B 20 44 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne PDGFRB 43 36 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne QRFPR 46 37 COCc1cc(NC(=O)N2CCC(C(C)=O)CC2)ccc1OC ZINC000880666127 DF On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N[C@@H]2COc3ccccc3[C@H]2O)ccc1OC ZINC000880666128 FE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N[C@@H]2COc3ccccc3[C@H]2O)ccc1OC ZINC000880666128 FE On-Demand Anodyne QRFPR 40 36 Cn1nnnc1-c1ccccc1NC(=O)NC1CC2(CSC2)C1 ZINC000880666130 ED On-Demand Anodyne CCR3 15 44 COCc1cc(NC(=O)N[C@H]2COc3ccccc3[C@H]2O)ccc1OC ZINC000880666131 FE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N[C@H]2COc3ccccc3[C@H]2O)ccc1OC ZINC000880666131 FE On-Demand Anodyne QRFPR 40 36 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@@H]1CCSC1 ZINC000880666133 EE On-Demand Anodyne CCR3 42 44 COCc1cc(NC(=O)N[C@@H]2COc3ccccc3[C@@H]2O)ccc1OC ZINC000880666134 FE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N[C@@H]2COc3ccccc3[C@@H]2O)ccc1OC ZINC000880666134 FE On-Demand Anodyne QRFPR 40 36 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@H]1CCSC1 ZINC000880666136 EE On-Demand Anodyne CCR3 42 44 COCc1cc(NC(=O)N[C@H]2COc3ccccc3[C@@H]2O)ccc1OC ZINC000880666137 FE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N[C@H]2COc3ccccc3[C@@H]2O)ccc1OC ZINC000880666137 FE On-Demand Anodyne QRFPR 40 36 COCc1cc(NC(=O)NC[C@@H](Oc2ccccc2)C(=O)OC)ccc1OC ZINC000880666139 GF On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne CACNA1H 44 38 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne HTR1B 15 44 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne PDGFRB 46 41 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne EPHX2 30 40 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC(F)(F)CC2)ccc1OC ZINC000880666140 DG On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NC[C@@H]2CC3(CCOCC3)CO2)ccc1OC ZINC000880666143 FF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@H]2CC3(CCOCC3)CO2)ccc1OC ZINC000880666145 FF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880666146 DF On-Demand Anodyne HTR2A 40 39 COCc1cc(NC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880666146 DF On-Demand Anodyne QPCT 15 41 COCc1cc(NC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880666146 DF On-Demand Anodyne ENPP1 57 31 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCS2)ccc1OC ZINC000880666148 ED On-Demand Reactive TSHR 41 31 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCS2)ccc1OC ZINC000880666148 ED On-Demand Reactive QRFPR 49 40 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@@H](C(F)F)C1 ZINC000880666149 ED On-Demand Anodyne CCR3 41 42 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCS2)ccc1OC ZINC000880666150 ED On-Demand Reactive TSHR 41 31 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCS2)ccc1OC ZINC000880666150 ED On-Demand Reactive QRFPR 49 40 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@H](C(F)F)C1 ZINC000880666151 ED On-Demand Anodyne CCR3 41 42 COCc1cc(NC(=O)NCC[S@](C)=O)ccc1OC ZINC000880666152 DD On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NCC[S@](C)=O)ccc1OC ZINC000880666152 DD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NCC[S@](C)=O)ccc1OC ZINC000880666152 DD On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NCc2ccc(OC)c(C#N)c2)ccc1OC ZINC000880666153 FG On-Demand Mild TSHR 60 32 COCc1cc(NC(=O)NCc2ccc(OC)c(C#N)c2)ccc1OC ZINC000880666153 FG On-Demand Mild ROCK2 21 45 COCc1cc(NC(=O)NCC[S@@](C)=O)ccc1OC ZINC000880666154 DD On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NCC[S@@](C)=O)ccc1OC ZINC000880666154 DD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NCC[S@@](C)=O)ccc1OC ZINC000880666154 DD On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N[C@@H]2C(=O)OCC2(C)C)ccc1OC ZINC000880666155 DD On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)N[C@@H]2C(=O)OCC2(C)C)ccc1OC ZINC000880666155 DD On-Demand Anodyne QRFPR 43 35 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880666156 FG On-Demand Anodyne RBP4 55 34 COCc1cc(NC(=O)N[C@H]2C(=O)OCC2(C)C)ccc1OC ZINC000880666157 DD On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)N[C@H]2C(=O)OCC2(C)C)ccc1OC ZINC000880666157 DD On-Demand Anodyne QRFPR 43 35 C#CC[C@H](CCOC)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666158 ED On-Demand Mild CCR3 44 40 C#CC[C@@H](CCOC)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666160 ED On-Demand Mild CCR3 44 40 COCc1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666163 DE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666163 DE On-Demand Anodyne HTR1D 16 44 COCc1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666163 DE On-Demand Anodyne HTR1B 18 41 COCc1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666163 DE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666163 DE On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666165 DE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666165 DE On-Demand Anodyne HTR1D 16 44 COCc1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666165 DE On-Demand Anodyne HTR1B 18 41 COCc1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666165 DE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666165 DE On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)Nc2ccc(O)c(C(C)C)c2)ccc1OC ZINC000880666171 EI On-Demand Anodyne THRA 68 37 COCc1cc(NC(=O)Nc2ccc(O)c(C(C)C)c2)ccc1OC ZINC000880666171 EI On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)Nc2ccc(O)c(C(C)C)c2)ccc1OC ZINC000880666171 EI On-Demand Anodyne HTR2A 24 41 COCc1cc(NC(=O)Nc2ccc(O)c(C(C)C)c2)ccc1OC ZINC000880666171 EI On-Demand Anodyne THRB 71 41 COCc1cc(NC(=O)Nc2ccc(O)c(C(C)C)c2)ccc1OC ZINC000880666171 EI On-Demand Anodyne ENPP1 50 30 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666175 FG On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666175 FG On-Demand Anodyne HTR2A 31 43 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666175 FG On-Demand Anodyne ADRB3 23 41 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666175 FG On-Demand Anodyne QRFPR 41 42 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666175 FG On-Demand Anodyne ENPP1 66 35 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@H]1CCCS1 ZINC000880666176 EE On-Demand Anodyne CCR3 46 44 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666177 FG On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666177 FG On-Demand Anodyne HTR2A 31 43 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666177 FG On-Demand Anodyne ADRB3 23 41 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666177 FG On-Demand Anodyne QRFPR 41 42 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)cc2)ccc1OC ZINC000880666177 FG On-Demand Anodyne ENPP1 66 35 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@@H]1CCCS1 ZINC000880666178 EE On-Demand Anodyne CCR3 46 44 COCc1cc(NC(=O)NC[C@@H]2CC(=O)c3ccccc3O2)ccc1OC ZINC000880666179 FF On-Demand Anodyne TSHR 75 38 COCc1cc(NC(=O)NC[C@@H]2CC(=O)c3ccccc3O2)ccc1OC ZINC000880666179 FF On-Demand Anodyne QRFPR 40 36 COCc1cc(NC(=O)NC[C@H]2CC(=O)c3ccccc3O2)ccc1OC ZINC000880666181 FF On-Demand Anodyne TSHR 75 38 COCc1cc(NC(=O)NC[C@H]2CC(=O)c3ccccc3O2)ccc1OC ZINC000880666181 FF On-Demand Anodyne QRFPR 40 36 C[C@@H]1CC[C@H](NC(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666182 DE On-Demand Anodyne CCR3 27 47 C[C@H]1CC[C@H](NC(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666184 DE On-Demand Anodyne CCR3 27 47 C[C@H]1CC[C@@H](NC(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666186 DE On-Demand Anodyne CCR3 27 47 COCc1cc(NC(=O)N2CCN([S@](C)(=N)=O)CC2)ccc1OC ZINC000880666188 FD On-Demand Anodyne PDGFRB 46 38 COCc1cc(NC(=O)N2CCN([S@](C)(=N)=O)CC2)ccc1OC ZINC000880666188 FD On-Demand Anodyne F13A1 45 39 COCc1cc(NC(=O)N2CCN([S@](C)(=N)=O)CC2)ccc1OC ZINC000880666188 FD On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCN([S@](C)(=N)=O)CC2)ccc1OC ZINC000880666188 FD On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N2CCN([S@@](C)(=N)=O)CC2)ccc1OC ZINC000880666190 FD On-Demand Anodyne PDGFRB 46 38 COCc1cc(NC(=O)N2CCN([S@@](C)(=N)=O)CC2)ccc1OC ZINC000880666190 FD On-Demand Anodyne F13A1 45 39 COCc1cc(NC(=O)N2CCN([S@@](C)(=N)=O)CC2)ccc1OC ZINC000880666190 FD On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCN([S@@](C)(=N)=O)CC2)ccc1OC ZINC000880666190 FD On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N2C[C@H]3C(=O)OC[C@H]3C2)ccc1OC ZINC000880666191 DD On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NC[C@@H]2CCC(C)(C)CO2)ccc1OC ZINC000880666192 EG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC3=C(CCC(=O)N3)C2)ccc1OC ZINC000880666193 EE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H]2CCC(C)(C)CO2)ccc1OC ZINC000880666194 EG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2Cc3cccnc3N3C[C@H](O)C[C@H]3C2)ccc1OC ZINC000880666195 GE On-Demand Anodyne TSHR 53 31 C#C[C@@H](NC(=O)Nc1ccccc1-c1nnnn1C)C(C)C ZINC000880666197 CD On-Demand Mild CCR3 40 40 C#C[C@H](NC(=O)Nc1ccccc1-c1nnnn1C)C(C)C ZINC000880666199 CD On-Demand Mild CCR3 40 40 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](CF)C1 ZINC000880666205 DD On-Demand Anodyne CCR3 62 48 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](CF)C1 ZINC000880666208 DD On-Demand Anodyne CCR3 62 48 COCc1cc(NC(=O)N2CCOC[C@H]2c2nc(C)no2)ccc1OC ZINC000880666213 FE On-Demand Anodyne TSHR 42 33 COCc1cc(NC(=O)N2CCOC[C@H]2c2nc(C)no2)ccc1OC ZINC000880666213 FE On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)N2CCOC[C@@H]2c2nc(C)no2)ccc1OC ZINC000880666214 FE On-Demand Anodyne TSHR 42 33 COCc1cc(NC(=O)N2CCOC[C@@H]2c2nc(C)no2)ccc1OC ZINC000880666214 FE On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)NC[C@@H]2CCC23CCOCC3)ccc1OC ZINC000880666216 EG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC[C@H]2CCC23CCOCC3)ccc1OC ZINC000880666217 EG On-Demand Anodyne QRFPR 44 36 C#CC[C@@H](CCOC)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666218 DE On-Demand Mild QRFPR 41 34 C#CC[C@H](CCOC)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666219 DE On-Demand Mild QRFPR 41 34 COCc1cc(NC(=O)N[C@@H]2CCCC[C@@H]2F)ccc1OC ZINC000880666220 DG On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N[C@@H]2CCCC[C@@H]2F)ccc1OC ZINC000880666220 DG On-Demand Anodyne PDE4A 22 40 COCc1cc(NC(=O)N[C@@H]2CCCC[C@@H]2F)ccc1OC ZINC000880666220 DG On-Demand Anodyne QRFPR 50 41 COCc1cc(NC(=O)N[C@@H]2CCCC[C@@H]2F)ccc1OC ZINC000880666220 DG On-Demand Anodyne ENPP1 55 32 CCn1ncn(NC(=O)Nc2ccc(OC)c(COC)c2)c1=O ZINC000880666222 DC On-Demand Anodyne TSHR 42 33 CCn1ncn(NC(=O)Nc2ccc(OC)c(COC)c2)c1=O ZINC000880666222 DC On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)NOCC2CC2)ccc1OC ZINC000880666231 CE On-Demand Anodyne TSHR 59 32 COCc1cc(NC(=O)NOCC2CC2)ccc1OC ZINC000880666231 CE On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)NOCC2CC2)ccc1OC ZINC000880666231 CE On-Demand Anodyne ENPP1 60 31 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)CCc2ccc(Cl)c(Cl)c2)n1 ZINC000880666232 GG On-Demand Anodyne TPSAB1 42 37 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)CCc2ccc(Cl)c(Cl)c2)n1 ZINC000880666233 GG On-Demand Anodyne TPSAB1 42 37 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](CF)C1 ZINC000880666237 DE On-Demand Anodyne CCR3 67 53 COCc1cc(NC(=O)N2CCCC[C@H]2CN2CCCC2=O)ccc1OC ZINC000880666239 GF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2CCCC[C@H]2CN2CCCC2=O)ccc1OC ZINC000880666239 GF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCCC[C@@H]2CN2CCCC2=O)ccc1OC ZINC000880666240 GF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2CCCC[C@@H]2CN2CCCC2=O)ccc1OC ZINC000880666240 GF On-Demand Anodyne QRFPR 44 36 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](CF)C1 ZINC000880666241 DE On-Demand Anodyne CCR3 67 53 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1C[C@H](O)c1cccs1 ZINC000880666245 GG On-Demand Anodyne CCR3 40 31 COCc1cc(NC(=O)N2CCc3cc(Cl)nnc3C2)ccc1OC ZINC000880666247 FF On-Demand Anodyne HTR1B 15 40 COCc1cc(NC(=O)N2CCc3cc(Cl)nnc3C2)ccc1OC ZINC000880666247 FF On-Demand Anodyne ENPP1 67 33 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1C[C@H](O)c1cccs1 ZINC000880666250 GG On-Demand Anodyne CCR3 40 31 C#C[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666253 DF On-Demand Mild TSHR 56 33 C#C[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666253 DF On-Demand Mild HTR1D 15 42 C#C[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666253 DF On-Demand Mild HTR1B 18 41 C#C[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666253 DF On-Demand Mild QRFPR 45 37 C#C[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666254 DF On-Demand Mild TSHR 56 33 C#C[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666254 DF On-Demand Mild HTR1D 15 42 C#C[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666254 DF On-Demand Mild HTR1B 18 41 C#C[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666254 DF On-Demand Mild QRFPR 45 37 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1C[C@@H](O)c1cccs1 ZINC000880666255 GG On-Demand Anodyne CCR3 40 31 COCc1cc(NC(=O)NN2CCC[C@H]2COC)ccc1OC ZINC000880666256 DD On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)NN2CCC[C@H]2COC)ccc1OC ZINC000880666256 DD On-Demand Anodyne QRFPR 47 38 COCc1cc(NC(=O)NN2CCC[C@H]2COC)ccc1OC ZINC000880666256 DD On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)NN2CCC[C@@H]2COC)ccc1OC ZINC000880666257 DD On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)NN2CCC[C@@H]2COC)ccc1OC ZINC000880666257 DD On-Demand Anodyne QRFPR 47 38 COCc1cc(NC(=O)NN2CCC[C@@H]2COC)ccc1OC ZINC000880666257 DD On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)NCCN(C)OC)ccc1OC ZINC000880666258 CD On-Demand Anodyne TSHR 64 30 COCc1cc(NC(=O)NCCN(C)OC)ccc1OC ZINC000880666258 CD On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NCCN(C)OC)ccc1OC ZINC000880666258 CD On-Demand Anodyne ENPP1 45 30 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1C[C@@H](O)c1cccs1 ZINC000880666259 GG On-Demand Anodyne CCR3 40 31 COCc1cc(NC(=O)N(C)C[C@@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880666260 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N(C)C[C@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880666261 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NOC(C)(C)CO)ccc1OC ZINC000880666262 CD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NOC(C)(C)CO)ccc1OC ZINC000880666262 CD On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)NCC2SCCS2)ccc1OC ZINC000880666263 EF On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NCC2SCCS2)ccc1OC ZINC000880666263 EF On-Demand Anodyne QRFPR 49 42 COCc1cc(NC(=O)NCC2SCCS2)ccc1OC ZINC000880666263 EF On-Demand Anodyne PRMT3 44 32 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne HTR2A 39 42 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne ROCK2 15 44 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne QPCT 21 46 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne PRMT3 44 33 COCc1cc(NC(=O)NCc2cnn(C)n2)ccc1OC ZINC000880666266 DD On-Demand Anodyne ENPP1 65 35 COCc1cc(NC(=O)N2CCN(c3ccncc3)[C@@H](C)C2)ccc1OC ZINC000880666267 FF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCN(c3ccncc3)[C@@H](C)C2)ccc1OC ZINC000880666267 FF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)N2CCN(c3ccncc3)[C@H](C)C2)ccc1OC ZINC000880666272 FF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCN(c3ccncc3)[C@H](C)C2)ccc1OC ZINC000880666272 FF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)NN2CCc3ccccc3C2)ccc1OC ZINC000880666275 EF On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)NN2CCc3ccccc3C2)ccc1OC ZINC000880666275 EF On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)NN2CCc3ccccc3C2)ccc1OC ZINC000880666275 EF On-Demand Anodyne NOD1 16 40 COCc1cc(NC(=O)NN2CCc3ccccc3C2)ccc1OC ZINC000880666275 EF On-Demand Anodyne NOD2 43 40 COCc1cc(NC(=O)NCCCc2nnc(S)n2C)ccc1OC ZINC000880666277 FE On-Demand Anodyne QPCT 26 48 COCc1cc(NC(=O)NCCCc2nnc(S)n2C)ccc1OC ZINC000880666277 FE On-Demand Anodyne PRMT3 43 31 COCc1cc(NC(=O)NCCCc2nnc(S)n2C)ccc1OC ZINC000880666277 FE On-Demand Anodyne ENPP1 56 31 COCc1cc(NC(=O)N[C@H](C)C2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666281 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)C2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666281 GG On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)N2CCOC[C@H]2c2ccc(OC)cc2)ccc1OC ZINC000880666284 GG On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)N2CCOC[C@H]2c2ccc(OC)cc2)ccc1OC ZINC000880666284 GG On-Demand Anodyne ENPP1 60 32 COCc1cc(NC(=O)N[C@@H](C)C2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666285 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H](C)C2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666285 GG On-Demand Anodyne ENPP1 55 30 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666288 DG On-Demand Mild TSHR 41 31 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666288 DG On-Demand Mild HTR1D 16 44 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666288 DG On-Demand Mild HTR1B 19 42 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666288 DG On-Demand Mild PDGFRB 42 37 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666288 DG On-Demand Mild QRFPR 46 38 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666289 DG On-Demand Mild TSHR 41 31 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666289 DG On-Demand Mild HTR1D 16 44 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666289 DG On-Demand Mild HTR1B 19 42 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666289 DG On-Demand Mild PDGFRB 42 37 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880666289 DG On-Demand Mild QRFPR 46 38 COCc1cc(NC(=O)NCCc2nnc(C)s2)ccc1OC ZINC000880666290 EE On-Demand Anodyne PRMT3 62 34 COCc1cc(NC(=O)NCCc2nnc(C)s2)ccc1OC ZINC000880666290 EE On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N2CCOC[C@@H]2c2ccc(OC)cc2)ccc1OC ZINC000880666291 GG On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)N2CCOC[C@@H]2c2ccc(OC)cc2)ccc1OC ZINC000880666291 GG On-Demand Anodyne ENPP1 60 32 COCc1cc(NC(=O)N(CCO)Cc2ccc(OC)cc2)ccc1OC ZINC000880666293 FF On-Demand Anodyne TSHR 55 35 COCc1cc(NC(=O)N(CCO)Cc2ccc(OC)cc2)ccc1OC ZINC000880666293 FF On-Demand Anodyne BMP1 31 42 COCc1cc(NC(=O)N(CCO)Cc2ccc(OC)cc2)ccc1OC ZINC000880666293 FF On-Demand Anodyne ROCK2 16 46 COCc1cc(NC(=O)NC[C@@H]2[C@H](C(=O)OC)C2(F)F)ccc1OC ZINC000880666295 FE On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)NC[C@@H]2[C@H](C(=O)OC)C2(F)F)ccc1OC ZINC000880666295 FE On-Demand Anodyne QRFPR 41 34 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](C(C)(C)O)C1 ZINC000880666296 ED On-Demand Anodyne CCR3 46 44 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H](C(C)(C)O)C1 ZINC000880666296 ED On-Demand Anodyne RBP4 46 34 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](C(C)(C)O)C1 ZINC000880666299 ED On-Demand Anodyne CCR3 46 44 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H](C(C)(C)O)C1 ZINC000880666299 ED On-Demand Anodyne RBP4 46 34 COCc1cc(NC(=O)NOCCCC(=O)OC)ccc1OC ZINC000880666301 ED On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NOCCCC(=O)OC)ccc1OC ZINC000880666301 ED On-Demand Anodyne ENPP1 49 31 COCc1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1OC ZINC000880666302 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1OC ZINC000880666302 DE On-Demand Anodyne HTR1D 16 47 COCc1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1OC ZINC000880666302 DE On-Demand Anodyne HTR1B 19 44 COCc1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1OC ZINC000880666302 DE On-Demand Anodyne PDGFRB 48 38 COCc1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1OC ZINC000880666302 DE On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2[C@H]3CC[C@H]2CC(c2noc(C)n2)C3)ccc1OC ZINC000880666303 GG On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1OC ZINC000880666304 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1OC ZINC000880666304 DE On-Demand Anodyne HTR1D 16 47 COCc1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1OC ZINC000880666304 DE On-Demand Anodyne HTR1B 19 44 COCc1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1OC ZINC000880666304 DE On-Demand Anodyne PDGFRB 48 38 COCc1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1OC ZINC000880666304 DE On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2Cc3ccc(Br)cc3C2)ccc1OC ZINC000880666305 GI On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2Cc3ccc(Br)cc3C2)ccc1OC ZINC000880666305 GI On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2Cc3ccc(Br)cc3C2)ccc1OC ZINC000880666305 GI On-Demand Anodyne ENPP1 42 35 COCc1cc(NC(=O)N2CCc3cc(C(=O)OC)ccc3C2)ccc1OC ZINC000880666308 GG On-Demand Anodyne ABCG2 29 41 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@]1(C)C[C@H]1Br ZINC000880666312 FE On-Demand Reactive CCR3 54 46 Cn1nnnc1-c1ccccc1NC(=O)NC[C@]1(C)C[C@@H]1Br ZINC000880666313 FE On-Demand Reactive CCR3 54 46 Cn1nnnc1-c1ccccc1NC(=O)NC[C@]1(C)C[C@H]1Br ZINC000880666314 FE On-Demand Reactive CCR3 54 46 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@]1(C)C[C@@H]1Br ZINC000880666315 FE On-Demand Reactive CCR3 54 46 Cn1nnnc1-c1ccccc1NC(=O)NCCOC(F)(F)C(F)(F)F ZINC000880666316 GE On-Demand Anodyne CCR3 23 41 COCc1cc(NC(=O)NCc2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880666317 GF On-Demand Anodyne TSHR 70 34 COCc1cc(NC(=O)NCc2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880666317 GF On-Demand Anodyne ROCK2 17 41 COCc1cc(NC(=O)NCc2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880666317 GF On-Demand Anodyne ENPP1 50 31 COCc1cc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)ccc1OC ZINC000880666318 FD On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)ccc1OC ZINC000880666318 FD On-Demand Anodyne HTR1B 15 42 COCc1cc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)ccc1OC ZINC000880666318 FD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)ccc1OC ZINC000880666318 FD On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)ccc1OC ZINC000880666319 FD On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)ccc1OC ZINC000880666319 FD On-Demand Anodyne HTR1B 15 42 COCc1cc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)ccc1OC ZINC000880666319 FD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)ccc1OC ZINC000880666319 FD On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NCc2cnc(Cl)s2)ccc1OC ZINC000880666325 EG On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NCc2cnc(Cl)s2)ccc1OC ZINC000880666325 EG On-Demand Anodyne ROCK2 15 43 COCc1cc(NC(=O)NCc2cnc(Cl)s2)ccc1OC ZINC000880666325 EG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCc2cnc(Cl)s2)ccc1OC ZINC000880666325 EG On-Demand Anodyne ENPP1 48 36 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666328 GH On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666328 GH On-Demand Anodyne HTR2A 17 44 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666328 GH On-Demand Anodyne RAF1 23 40 COCc1cc(NC(=O)N(Cc2ccccc2OC)OC)ccc1OC ZINC000880666330 FG On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)N(Cc2ccccc2OC)OC)ccc1OC ZINC000880666330 FG On-Demand Anodyne TSPO 46 40 COCc1cc(NC(=O)N(Cc2ccccc2OC)OC)ccc1OC ZINC000880666330 FG On-Demand Anodyne QRFPR 41 36 C#C[C@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666331 DD On-Demand Mild TSHR 47 31 C#C[C@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666331 DD On-Demand Mild QRFPR 41 34 C#C[C@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666331 DD On-Demand Mild ENPP1 40 32 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666332 GH On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666332 GH On-Demand Anodyne HTR2A 17 44 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C(F)(F)F)c2)ccc1OC ZINC000880666332 GH On-Demand Anodyne RAF1 23 40 C#C[C@@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666333 DD On-Demand Mild TSHR 47 31 C#C[C@@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666333 DD On-Demand Mild QRFPR 41 34 C#C[C@@H]1COCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666333 DD On-Demand Mild ENPP1 40 32 COCc1cc(NC(=O)NCc2ccnc(F)c2)ccc1OC ZINC000880666334 DF On-Demand Anodyne TSHR 58 35 COCc1cc(NC(=O)NCc2ccnc(F)c2)ccc1OC ZINC000880666334 DF On-Demand Anodyne ROCK2 28 47 COCc1cc(NC(=O)NCc2ccnc(F)c2)ccc1OC ZINC000880666334 DF On-Demand Anodyne PDGFRA 43 37 COCc1cc(NC(=O)NCc2ccnc(F)c2)ccc1OC ZINC000880666334 DF On-Demand Anodyne ENPP1 52 34 COCc1cc(NC(=O)NCc2ccnc(F)c2)ccc1OC ZINC000880666334 DF On-Demand Anodyne DRTS_TRYCR 45 32 COCc1cc(NC(=O)NC[C@@H]2C[C@H]3CCC[C@H]3O2)ccc1OC ZINC000880666339 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NC[C@@H]2C[C@@H]3CCC[C@@H]3O2)ccc1OC ZINC000880666341 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@H]3C2)ccc1OC ZINC000880666345 EG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@H]3C2)ccc1OC ZINC000880666345 EG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@H]3C2)ccc1OC ZINC000880666345 EG On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@H]3C2)ccc1OC ZINC000880666345 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)NC[C@@H]2C[C@H]3CCC[C@@H]3O2)ccc1OC ZINC000880666346 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666347 EG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666347 EG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666347 EG On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CC[C@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666347 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666348 EG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666348 EG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666348 EG On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@@H]3C2)ccc1OC ZINC000880666348 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)NC[C@@H]2C[C@@H]3CCC[C@H]3O2)ccc1OC ZINC000880666349 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@H]3C2)ccc1OC ZINC000880666350 EG On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@H]3C2)ccc1OC ZINC000880666350 EG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@H]3C2)ccc1OC ZINC000880666350 EG On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CC[C@@H]3CSC[C@H]3C2)ccc1OC ZINC000880666350 EG On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)N2C[C@H](N(C)C)[C@H](n3ccnn3)C2)ccc1OC ZINC000880666353 FD On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)N2C[C@@H]3C[C@H]2CN3C(=O)OC(C)(C)C)ccc1OC ZINC000880666354 GG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2C[C@@H]3C[C@H]2CN3C(=O)OC(C)(C)C)ccc1OC ZINC000880666354 GG On-Demand Anodyne ENPP1 45 33 COCc1cc(NC(=O)N2CC[C@@](O)(C(F)F)C2)ccc1OC ZINC000880666355 EE On-Demand Anodyne EPHX2 31 41 COC[C@@H]1CCCN1NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666357 ED On-Demand Anodyne CCR3 56 48 COCc1cc(NC(=O)N2CC[C@](O)(C(F)F)C2)ccc1OC ZINC000880666358 EE On-Demand Anodyne EPHX2 31 41 COCc1cc(NC(=O)NN2CCCC2)ccc1OC ZINC000880666359 CD On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NN2CCCC2)ccc1OC ZINC000880666359 CD On-Demand Anodyne QRFPR 45 38 COCc1cc(NC(=O)NN2CCCC2)ccc1OC ZINC000880666359 CD On-Demand Anodyne ENPP1 63 32 Cn1nnnc1-c1ccccc1NC(=O)NCC(F)(F)Br ZINC000880666360 FD On-Demand Anodyne CCR3 34 44 COCc1cc(NC(=O)NCc2cnc(Cl)cn2)ccc1OC ZINC000880666361 EF On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NCc2cnc(Cl)cn2)ccc1OC ZINC000880666361 EF On-Demand Anodyne ROCK2 16 43 COCc1cc(NC(=O)NCc2cnc(Cl)cn2)ccc1OC ZINC000880666361 EF On-Demand Anodyne ENPP1 48 36 COCc1cc(NC(=O)NCc2ccc(N3CCCNC3=O)cc2)ccc1OC ZINC000880666362 GG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCc2ccc(N3CCCNC3=O)cc2)ccc1OC ZINC000880666362 GG On-Demand Anodyne ROCK2 15 40 COCc1cc(NC(=O)NCc2ccc(N3CCCNC3=O)cc2)ccc1OC ZINC000880666362 GG On-Demand Anodyne ENPP1 44 30 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880666363 GF On-Demand Anodyne CCR3 38 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880666368 GF On-Demand Anodyne CCR3 38 42 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne HTR1D 25 52 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne HTR1B 27 52 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne PDGFRB 41 36 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)ccc1OC ZINC000880666369 GE On-Demand Anodyne L3MBTL3 57 38 COCc1cc(NC(=O)N2CCC[C@@]3(C2)CC3(F)F)ccc1OC ZINC000880666370 EG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@]3(C2)CC3(F)F)ccc1OC ZINC000880666371 EG On-Demand Anodyne QRFPR 42 35 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@H]1[C@H](O)c1ccccc1 ZINC000880666372 GF On-Demand Anodyne CCR3 38 42 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880666376 GF On-Demand Anodyne CCR3 38 42 COCc1cc(NC(=O)NCCCc2cnn(C)n2)ccc1OC ZINC000880666378 ED On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)NCCCc2cnn(C)n2)ccc1OC ZINC000880666378 ED On-Demand Anodyne QPCT 44 52 COCc1cc(NC(=O)NCCCc2cnn(C)n2)ccc1OC ZINC000880666378 ED On-Demand Anodyne ENPP1 52 33 COCc1cc(NC(=O)N[C@@H]2CC[C@H]2O)ccc1OC ZINC000880666379 CD On-Demand Anodyne TSHR 59 32 COCc1cc(NC(=O)N[C@@H]2CC[C@H]2O)ccc1OC ZINC000880666379 CD On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)N[C@@H]2CC[C@H]2O)ccc1OC ZINC000880666379 CD On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne HTR1D 17 47 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne HTR1B 20 47 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne PDGFRB 49 39 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne EPHX2 15 45 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne RBP4 16 40 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCCCCCCC2)ccc1OC ZINC000880666380 DI On-Demand Anodyne ENPP1 69 35 COCc1cc(NC(=O)NCc2ncc(Br)s2)ccc1OC ZINC000880666381 GG On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NCc2ncc(Br)s2)ccc1OC ZINC000880666381 GG On-Demand Anodyne QRFPR 41 39 COCc1cc(NC(=O)NCc2ncc(Br)s2)ccc1OC ZINC000880666381 GG On-Demand Anodyne PRMT3 44 32 COCc1cc(NC(=O)NCc2ncc(Br)s2)ccc1OC ZINC000880666381 GG On-Demand Anodyne ENPP1 47 35 COCc1cc(NC(=O)N[C@@H]2C[C@H](COC)C2)ccc1OC ZINC000880666385 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N[C@@H]2C[C@H](COC)C2)ccc1OC ZINC000880666385 DE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@@H]2C[C@H](COC)C2)ccc1OC ZINC000880666385 DE On-Demand Anodyne ENPP1 44 30 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880666389 GF On-Demand Anodyne EPHX2 15 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880666389 GF On-Demand Anodyne TRPM8 28 45 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880666390 GF On-Demand Anodyne EPHX2 15 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880666390 GF On-Demand Anodyne TRPM8 28 45 COCc1cc(NC(=O)NC[C@@H]2C[C@@H](OC)C2)ccc1OC ZINC000880666391 DE On-Demand Anodyne TSHR 49 31 COCc1cc(NC(=O)NC[C@@H]2C[C@@H](OC)C2)ccc1OC ZINC000880666391 DE On-Demand Anodyne QRFPR 47 38 COCc1cc(NC(=O)NC[C@H](OC)C(=O)OC)ccc1OC ZINC000880666392 ED On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NC[C@H](OC)C(=O)OC)ccc1OC ZINC000880666392 ED On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N2CC(O)(C(=O)OC)C2)ccc1OC ZINC000880666394 DC On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CC(O)(C(=O)OC)C2)ccc1OC ZINC000880666394 DC On-Demand Anodyne PDGFRB 40 36 COCc1cc(NC(=O)N2CC(O)(C(=O)OC)C2)ccc1OC ZINC000880666394 DC On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC(O)(C(=O)OC)C2)ccc1OC ZINC000880666394 DC On-Demand Anodyne ENPP1 63 35 COCc1cc(NC(=O)N[C@H]2CC23CCC3)ccc1OC ZINC000880666395 CF On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)N[C@@H]2CC23CCC3)ccc1OC ZINC000880666396 CF On-Demand Anodyne QRFPR 47 39 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880666399 GF On-Demand Anodyne CCR3 60 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1C[C@H](O)c1ccccc1 ZINC000880666400 GF On-Demand Anodyne CCR3 60 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880666401 GF On-Demand Anodyne CCR3 60 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880666402 GF On-Demand Anodyne CCR3 60 43 COCc1cc(NC(=O)N2C[C@H]3C=C[C@H]2C3)ccc1OC ZINC000880666403 CF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2C[C@H]3C=C[C@H]2C3)ccc1OC ZINC000880666403 CF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@H]3C=C[C@H]2C3)ccc1OC ZINC000880666403 CF On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N2CCC(NC3CCOCC3)CC2)ccc1OC ZINC000880666404 GF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC(NC3CCOCC3)CC2)ccc1OC ZINC000880666404 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC3(CC2)COCCO3)ccc1OC ZINC000880666407 FE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)N2CCC3(CC2)COCCO3)ccc1OC ZINC000880666407 FE On-Demand Anodyne EPHX2 21 45 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666408 ED On-Demand Anodyne CCR3 55 46 CC(=O)[C@H]1CCCN(C(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666409 ED On-Demand Anodyne CCR3 55 46 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](N2CCCCC2=O)C1 ZINC000880666410 GD On-Demand Anodyne CCR3 50 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](N2CCCCC2=O)C1 ZINC000880666411 GD On-Demand Anodyne CCR3 50 44 Cn1nnnc1-c1ccccc1NC(=O)NOCC1CCC1 ZINC000880666412 DD On-Demand Anodyne CCR3 65 50 Cn1nnnc1-c1ccccc1NC(=O)N1Cc2cccnc2N2CCC[C@H]2C1 ZINC000880666413 GE On-Demand Anodyne CCR3 19 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C)(N2CCCCC2)CC1 ZINC000880666414 GF On-Demand Anodyne CCR5 17 40 CN1Cc2ccccc2[C@@H]1CNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666415 FE On-Demand Anodyne CCR3 23 41 CN1Cc2ccccc2[C@H]1CNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666416 FE On-Demand Anodyne CCR3 23 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@H]1CN1CCCC1=O ZINC000880666417 GD On-Demand Anodyne CCR3 39 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@@H]1CN1CCCC1=O ZINC000880666418 GD On-Demand Anodyne CCR3 39 43 C#CCCCCNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666419 CD On-Demand Mild CCR3 23 40 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@@H]1CCCOC1 ZINC000880666422 EG On-Demand Anodyne QRFPR 42 36 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@H]1CCCOC1 ZINC000880666423 EG On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)N(CC(C)C)CC2CCN(C)CC2)ccc1OC ZINC000880666424 GH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@H]3C2)ccc1OC ZINC000880666425 GH On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@H]3C2)ccc1OC ZINC000880666425 GH On-Demand Anodyne HTR1D 15 45 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@H]3C2)ccc1OC ZINC000880666425 GH On-Demand Anodyne HTR1B 17 45 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@H]3C2)ccc1OC ZINC000880666425 GH On-Demand Anodyne QRFPR 44 39 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@@H]3C2)ccc1OC ZINC000880666426 GH On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@@H]3C2)ccc1OC ZINC000880666426 GH On-Demand Anodyne HTR1D 15 45 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@@H]3C2)ccc1OC ZINC000880666426 GH On-Demand Anodyne HTR1B 17 45 COCc1cc(NC(=O)N2Cc3ccccc3N3CCC[C@@H]3C2)ccc1OC ZINC000880666426 GH On-Demand Anodyne QRFPR 44 39 COCc1cc(NC(=O)N2CC[C@@H](C(F)(F)F)O[C@H](C)C2)ccc1OC ZINC000880666427 GG On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2CC[C@@H](C(F)(F)F)O[C@H](C)C2)ccc1OC ZINC000880666427 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@H](C(F)(F)F)O[C@H](C)C2)ccc1OC ZINC000880666428 GG On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2CC[C@H](C(F)(F)F)O[C@H](C)C2)ccc1OC ZINC000880666428 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@H](C(F)(F)F)O[C@@H](C)C2)ccc1OC ZINC000880666429 GG On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2CC[C@@H](C(F)(F)F)O[C@@H](C)C2)ccc1OC ZINC000880666429 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@H](C(F)(F)F)O[C@@H](C)C2)ccc1OC ZINC000880666430 GG On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2CC[C@H](C(F)(F)F)O[C@@H](C)C2)ccc1OC ZINC000880666430 GG On-Demand Anodyne QRFPR 40 33 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@]1(C)C[C@@]1(F)Cl ZINC000880666434 FF On-Demand Anodyne CCR3 24 41 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@@]1(C)C[C@@]1(F)Cl ZINC000880666435 FF On-Demand Anodyne CCR3 24 41 CCC(C)(C)[C@@H](C)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880666456 DG On-Demand Anodyne KCNQ2 63 37 O=C1CC[C@H](c2ccc(C(=O)N3CCCC4(CCCC4)CC3)cc2)N1 ZINC000880666457 EH On-Demand Anodyne L3MBTL3 60 46 O=C1CC[C@@H](c2ccc(C(=O)N3CCCC4(CCCC4)CC3)cc2)N1 ZINC000880666458 EH On-Demand Anodyne L3MBTL3 60 46 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](C2OCCO2)C1 ZINC000880666459 FD On-Demand Anodyne CCR3 46 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](C2OCCO2)C1 ZINC000880666459 FD On-Demand Anodyne RBP4 44 32 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](C2OCCO2)C1 ZINC000880666460 FD On-Demand Anodyne CCR3 46 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](C2OCCO2)C1 ZINC000880666460 FD On-Demand Anodyne RBP4 44 32 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Cc2csc(COc3ccccc3)n2)C1 ZINC000880666461 GG On-Demand Anodyne ALOX5 23 42 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Cc2csc(COc3ccccc3)n2)C1 ZINC000880666462 GG On-Demand Anodyne ALOX5 23 42 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Cc2csc(COc3ccccc3)n2)C1 ZINC000880666463 GG On-Demand Anodyne ALOX5 23 42 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Cc2csc(COc3ccccc3)n2)C1 ZINC000880666464 GG On-Demand Anodyne ALOX5 23 42 Cn1nnnc1-c1ccccc1NC(=O)NCCSC(F)(F)F ZINC000880666496 EE On-Demand Anodyne CCR3 24 41 CCC(C)(C)[C@@H](C)NC(=O)c1cccn2nccc12 ZINC000880666515 CF On-Demand Anodyne JAK3 16 44 CCC(C)(C)[C@@H](C)NC(=O)c1cccn2nccc12 ZINC000880666515 CF On-Demand Anodyne TYK2 17 44 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)c2cc(F)c3ncccc3c2)C1 ZINC000880666531 EF On-Demand Anodyne MAPK13 65 34 C[S@](=O)[C@H]1CCC[C@H](NC(=O)c2cc(F)c3ncccc3c2)C1 ZINC000880666532 EF On-Demand Anodyne MAPK13 65 34 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)c2cc(F)c3ncccc3c2)C1 ZINC000880666533 EF On-Demand Anodyne MAPK13 65 34 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)c2cc(F)c3ncccc3c2)C1 ZINC000880666534 EF On-Demand Anodyne MAPK13 65 34 COCc1cc(NC(=O)NNc2cc(Cl)nc(C)n2)ccc1OC ZINC000880666536 FF On-Demand Reactive TSHR 58 38 COCc1cc(NC(=O)NNc2cc(Cl)nc(C)n2)ccc1OC ZINC000880666536 FF On-Demand Reactive HTR2A 31 40 COCc1cc(NC(=O)NNc2cc(Cl)nc(C)n2)ccc1OC ZINC000880666536 FF On-Demand Reactive ENPP1 71 37 COCc1cc(NC(=O)NOC2CCC2)ccc1OC ZINC000880666543 CE On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NOC2CCC2)ccc1OC ZINC000880666543 CE On-Demand Anodyne PDE4A 29 43 COCc1cc(NC(=O)NOC2CCC2)ccc1OC ZINC000880666543 CE On-Demand Anodyne QRFPR 51 42 COCc1cc(NC(=O)NOC2CCC2)ccc1OC ZINC000880666543 CE On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)NN2CCS(=O)(=O)CC2)ccc1OC ZINC000880666549 EC On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NN2CCS(=O)(=O)CC2)ccc1OC ZINC000880666549 EC On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NCC[C@@H]2CCSC2)ccc1OC ZINC000880666556 DG On-Demand Anodyne TSHR 51 34 COCc1cc(NC(=O)NCC[C@@H]2CCSC2)ccc1OC ZINC000880666556 DG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NCC[C@@H]2CCSC2)ccc1OC ZINC000880666556 DG On-Demand Anodyne PRMT3 25 42 COCc1cc(NC(=O)NCC[C@H]2CCSC2)ccc1OC ZINC000880666557 DG On-Demand Anodyne TSHR 51 34 COCc1cc(NC(=O)NCC[C@H]2CCSC2)ccc1OC ZINC000880666557 DG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NCC[C@H]2CCSC2)ccc1OC ZINC000880666557 DG On-Demand Anodyne PRMT3 25 42 COCc1cc(NC(=O)N2C[C@H]3C(=O)N(C)C(=O)[C@H]3C2)ccc1OC ZINC000880666558 EC On-Demand Anodyne TSHR 65 35 COCc1cc(NC(=O)N2C[C@H]3C(=O)N(C)C(=O)[C@H]3C2)ccc1OC ZINC000880666558 EC On-Demand Anodyne HTR1B 16 41 COCc1cc(NC(=O)N2C[C@H]3C(=O)N(C)C(=O)[C@H]3C2)ccc1OC ZINC000880666558 EC On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)N2C[C@H]3C(=O)N(C)C(=O)[C@H]3C2)ccc1OC ZINC000880666558 EC On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)NNc2cccc(C)n2)ccc1OC ZINC000880666563 DF On-Demand Reactive TSHR 44 35 COCc1cc(NC(=O)NNc2cccc(C)n2)ccc1OC ZINC000880666563 DF On-Demand Reactive GRM5 18 40 COCc1cc(NC(=O)NNc2cccc(C)n2)ccc1OC ZINC000880666563 DF On-Demand Reactive ENPP1 64 33 COCc1cc(NC(=O)N[C@H]2C[C@@H](O)c3ccccc32)ccc1OC ZINC000880666564 EG On-Demand Anodyne TSHR 61 32 COCc1cc(NC(=O)N[C@H]2C[C@@H](O)c3ccccc32)ccc1OC ZINC000880666564 EG On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)N[C@@H]2C[C@@H](O)c3ccccc32)ccc1OC ZINC000880666565 EG On-Demand Anodyne TSHR 61 32 COCc1cc(NC(=O)N[C@@H]2C[C@@H](O)c3ccccc32)ccc1OC ZINC000880666565 EG On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)N[C@H]2C[C@H](O)c3ccccc32)ccc1OC ZINC000880666566 EG On-Demand Anodyne TSHR 61 32 COCc1cc(NC(=O)N[C@H]2C[C@H](O)c3ccccc32)ccc1OC ZINC000880666566 EG On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)N[C@@H]2C[C@H](O)c3ccccc32)ccc1OC ZINC000880666567 EG On-Demand Anodyne TSHR 61 32 COCc1cc(NC(=O)N[C@@H]2C[C@H](O)c3ccccc32)ccc1OC ZINC000880666567 EG On-Demand Anodyne QRFPR 43 38 COCc1cc(NC(=O)N[C@@H]2COC(=O)C2)ccc1OC ZINC000880666570 CD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2COC(=O)C2)ccc1OC ZINC000880666570 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCCc2nnc(S)n2C)ccc1OC ZINC000880666575 FD On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)NCCc2nnc(S)n2C)ccc1OC ZINC000880666575 FD On-Demand Anodyne QPCT 17 45 COCc1cc(NC(=O)NCCc2nnc(S)n2C)ccc1OC ZINC000880666575 FD On-Demand Anodyne PRMT3 51 32 COCc1cc(NC(=O)NCCc2nnc(S)n2C)ccc1OC ZINC000880666575 FD On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)N2CCn3ncc(Br)c3C2)ccc1OC ZINC000880666576 GF On-Demand Anodyne PDGFRB 41 38 COCc1cc(NC(=O)N2CCn3ncc(Br)c3C2)ccc1OC ZINC000880666576 GF On-Demand Anodyne ENPP1 46 33 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@]1(C)C[C@]1(F)Cl ZINC000880666588 FF On-Demand Anodyne CCR3 24 41 Cn1nnnc1-c1ccccc1NC(=O)NCC[C@@]1(C)C[C@]1(F)Cl ZINC000880666590 FF On-Demand Anodyne CCR3 24 41 COCc1cc(NC(=O)NCc2nonc2C)ccc1OC ZINC000880666594 DD On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCc2nonc2C)ccc1OC ZINC000880666594 DD On-Demand Anodyne ENPP1 54 31 COCc1cc(NC(=O)N2CCC[C@@H](NC3CCOCC3)C2)ccc1OC ZINC000880666596 GF On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)N2CCC[C@@H](NC3CCOCC3)C2)ccc1OC ZINC000880666596 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@H](NC3CCOCC3)C2)ccc1OC ZINC000880666598 GF On-Demand Anodyne TSHR 48 32 COCc1cc(NC(=O)N2CCC[C@H](NC3CCOCC3)C2)ccc1OC ZINC000880666598 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NCc2ccc(C3(C)OCCO3)cc2)ccc1OC ZINC000880666602 GG On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NCc2ccc(C3(C)OCCO3)cc2)ccc1OC ZINC000880666602 GG On-Demand Anodyne ROCK2 16 41 COCc1cc(NC(=O)NCc2cc(Br)no2)ccc1OC ZINC000880666603 FF On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)NCc2cc(Br)no2)ccc1OC ZINC000880666603 FF On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666604 GG On-Demand Anodyne EPHX2 32 44 COCc1cc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666604 GG On-Demand Anodyne TRPM8 28 42 CSC(C)(C)CNC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666605 DE On-Demand Anodyne CCR3 28 43 COCc1cc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666606 GG On-Demand Anodyne EPHX2 32 44 COCc1cc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666606 GG On-Demand Anodyne TRPM8 28 42 COCc1cc(NC(=O)N[C@@H]2CCC[C@]23CCCO3)ccc1OC ZINC000880666607 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666608 GG On-Demand Anodyne EPHX2 32 44 COCc1cc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666608 GG On-Demand Anodyne TRPM8 28 42 COCc1cc(NC(=O)N[C@H]2CCC[C@@]23CCCO3)ccc1OC ZINC000880666609 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666610 GG On-Demand Anodyne EPHX2 32 44 COCc1cc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)ccc1OC ZINC000880666610 GG On-Demand Anodyne TRPM8 28 42 COCc1cc(NC(=O)N[C@@H]2CCC[C@@]23CCCO3)ccc1OC ZINC000880666611 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NCCC(C)(C)OC)ccc1OC ZINC000880666612 DF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@H](C)[C@@H](C)O)ccc1OC ZINC000880666613 CD On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)N[C@H](C)[C@@H](C)O)ccc1OC ZINC000880666613 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H](C)[C@@H](C)O)ccc1OC ZINC000880666613 CD On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N[C@H]2CCC[C@]23CCCO3)ccc1OC ZINC000880666614 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@@H](C)[C@H](C)O)ccc1OC ZINC000880666615 CD On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)N[C@@H](C)[C@H](C)O)ccc1OC ZINC000880666615 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@@H](C)[C@H](C)O)ccc1OC ZINC000880666615 CD On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N[C@@H](C)[C@@H](C)O)ccc1OC ZINC000880666616 CD On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)N[C@@H](C)[C@@H](C)O)ccc1OC ZINC000880666616 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@@H](C)[C@@H](C)O)ccc1OC ZINC000880666616 CD On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N[C@H](C)[C@H](C)O)ccc1OC ZINC000880666618 CD On-Demand Anodyne TSHR 40 31 COCc1cc(NC(=O)N[C@H](C)[C@H](C)O)ccc1OC ZINC000880666618 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H](C)[C@H](C)O)ccc1OC ZINC000880666618 CD On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)ccc1OC ZINC000880666619 GG On-Demand Mild HTR1B 16 52 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)ccc1OC ZINC000880666619 GG On-Demand Mild PDGFRB 59 54 COCc1cc(NC(=O)N2CCN(c3ccc(C#N)cc3)CC2)ccc1OC ZINC000880666619 GG On-Demand Mild TNIK 32 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880666620 GF On-Demand Anodyne CCR3 28 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880666622 GF On-Demand Anodyne CCR3 28 44 COCc1cc(NC(=O)NNc2ccnc(C(F)(F)F)c2)ccc1OC ZINC000880666626 FG On-Demand Reactive TSHR 47 33 COCc1cc(NC(=O)NNc2ccnc(C(F)(F)F)c2)ccc1OC ZINC000880666626 FG On-Demand Reactive PDGFRA 44 36 COCc1cc(NC(=O)NNc2ccnc(C(F)(F)F)c2)ccc1OC ZINC000880666626 FG On-Demand Reactive ENPP1 47 34 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CCC2(CCC2)O1 ZINC000880666627 EE On-Demand Anodyne CCR3 32 43 COCc1cc(NC(=O)N2CCc3c(CC(N)=O)cccc3C2)ccc1OC ZINC000880666628 GE On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N2CCc3c(CC(N)=O)cccc3C2)ccc1OC ZINC000880666628 GE On-Demand Anodyne P2RY14 46 33 COCc1cc(NC(=O)N2CCc3c(CC(N)=O)cccc3C2)ccc1OC ZINC000880666628 GE On-Demand Anodyne ENPP1 44 33 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CCC2(CCC2)O1 ZINC000880666629 EE On-Demand Anodyne CCR3 32 43 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H]1c1ccc(F)c(F)c1 ZINC000880666631 GH On-Demand Anodyne CCR3 58 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]1c1ccc(F)c(F)c1 ZINC000880666633 GH On-Demand Anodyne CCR3 58 44 COCc1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1OC ZINC000880666634 FF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1OC ZINC000880666634 FF On-Demand Anodyne PDGFRB 45 41 COCc1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1OC ZINC000880666634 FF On-Demand Anodyne EPHX2 28 41 COCc1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1OC ZINC000880666634 FF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NNC(=O)[C@@H]2C[C@H]3CC[C@H]2O3)ccc1OC ZINC000880666636 ED On-Demand Reactive QRFPR 42 34 COCc1cc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666637 EF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666637 EF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666637 EF On-Demand Anodyne PDE4A 16 46 COCc1cc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666637 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)ccc1OC ZINC000880666637 EF On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)NNC(=O)[C@H]2C[C@H]3CC[C@H]2O3)ccc1OC ZINC000880666638 ED On-Demand Reactive QRFPR 42 34 COCc1cc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666639 EF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666639 EF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666639 EF On-Demand Anodyne PDE4A 16 46 COCc1cc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666639 EF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)ccc1OC ZINC000880666639 EF On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N2CCO[C@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666644 GG On-Demand Anodyne TSHR 59 34 COCc1cc(NC(=O)N2CCO[C@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666644 GG On-Demand Anodyne EDNRA 27 40 COCc1cc(NC(=O)N2CCO[C@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666644 GG On-Demand Anodyne ENPP1 44 31 COCc1cc(NC(=O)N2CCO[C@@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666646 GG On-Demand Anodyne TSHR 59 34 COCc1cc(NC(=O)N2CCO[C@@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666646 GG On-Demand Anodyne EDNRA 27 40 COCc1cc(NC(=O)N2CCO[C@@H](c3ccc(OC)cc3)C2)ccc1OC ZINC000880666646 GG On-Demand Anodyne ENPP1 44 31 COCc1cc(NC(=O)N[C@](C)(CO)Cc2ccc(OC)cc2)ccc1OC ZINC000880666647 GF On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NO[C@@H](CO)C(C)C)ccc1OC ZINC000880666648 DD On-Demand Anodyne ENPP1 67 33 COCc1cc(NC(=O)N[C@@](C)(CO)Cc2ccc(OC)cc2)ccc1OC ZINC000880666649 GF On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NO[C@H](CO)C(C)C)ccc1OC ZINC000880666650 DD On-Demand Anodyne ENPP1 67 33 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne HTR1B 18 43 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne PDGFRB 40 35 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC(c3nnc(S)n3C)CC2)ccc1OC ZINC000880666652 GF On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N2CC[C@](C(=O)OC)(c3ccccc3)C2)ccc1OC ZINC000880666655 GG On-Demand Anodyne TSHR 66 36 COCc1cc(NC(=O)N2CC[C@](C(=O)OC)(c3ccccc3)C2)ccc1OC ZINC000880666655 GG On-Demand Anodyne EPHX2 32 45 COCc1cc(NC(=O)N2CC[C@@](C(=O)OC)(c3ccccc3)C2)ccc1OC ZINC000880666657 GG On-Demand Anodyne TSHR 66 36 COCc1cc(NC(=O)N2CC[C@@](C(=O)OC)(c3ccccc3)C2)ccc1OC ZINC000880666657 GG On-Demand Anodyne EPHX2 32 45 COCc1cc(NC(=O)NCCS(=O)(=O)C(F)(F)F)ccc1OC ZINC000880666659 FD On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NNc2cc(C(F)(F)F)ccn2)ccc1OC ZINC000880666661 FG On-Demand Reactive HTR2A 22 41 COCc1cc(NC(=O)NNc2cc(C(F)(F)F)ccn2)ccc1OC ZINC000880666661 FG On-Demand Reactive RAF1 32 42 COCc1cc(NC(=O)NNc2cc(C(F)(F)F)ccn2)ccc1OC ZINC000880666661 FG On-Demand Reactive PDGFRA 41 34 COCc1cc(NC(=O)NNc2cc(C(F)(F)F)ccn2)ccc1OC ZINC000880666661 FG On-Demand Reactive TEK 48 38 COCc1cc(NC(=O)NNc2cc(C(F)(F)F)ccn2)ccc1OC ZINC000880666661 FG On-Demand Reactive ENPP1 46 33 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne TSHR 58 35 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne HTR1D 20 48 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne HTR1B 21 48 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne CCR3 32 46 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne MLNR 24 41 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne EPHX2 47 38 COCc1cc(NC(=O)N2CC[C@H](Oc3ccc(F)cc3)C2)ccc1OC ZINC000880666662 FH On-Demand Anodyne QRFPR 41 34 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)C1CC1 ZINC000880666663 CE On-Demand Mild TSHR 60 32 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)C1CC1 ZINC000880666663 CE On-Demand Mild QRFPR 47 39 COCc1cc(NC(=O)NN(C)c2ccccn2)ccc1OC ZINC000880666664 DE On-Demand Reactive TSHR 56 35 COCc1cc(NC(=O)NN(C)c2ccccn2)ccc1OC ZINC000880666664 DE On-Demand Reactive GRM4 26 44 COCc1cc(NC(=O)NN(C)c2ccccn2)ccc1OC ZINC000880666664 DE On-Demand Reactive ENPP1 47 36 Cn1nnnc1-c1ccccc1NC(=O)NC[C@]12OCCC[C@H]1C2(F)F ZINC000880666665 FD On-Demand Anodyne CCR3 49 44 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCCO2)ccc1OC ZINC000880666666 ED On-Demand Reactive QRFPR 50 42 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCCO2)ccc1OC ZINC000880666668 ED On-Demand Reactive QRFPR 50 42 CCc1nc(CNC(=O)Nc2ccc(OC)c(COC)c2)co1 ZINC000880666670 DF On-Demand Anodyne TSHR 47 31 CCc1nc(CNC(=O)Nc2ccc(OC)c(COC)c2)co1 ZINC000880666670 DF On-Demand Anodyne ENPP1 65 30 COCc1cc(NC(=O)NC[C@@H](F)C(=O)OC)ccc1OC ZINC000880666672 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@@H](F)C(=O)OC)ccc1OC ZINC000880666672 DD On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)NC[C@H](F)C(=O)OC)ccc1OC ZINC000880666673 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H](F)C(=O)OC)ccc1OC ZINC000880666673 DD On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)NCc2cncn2C)ccc1OC ZINC000880666674 DD On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NCc2cncn2C)ccc1OC ZINC000880666674 DD On-Demand Anodyne QPCT 30 45 COCc1cc(NC(=O)NCc2cncn2C)ccc1OC ZINC000880666674 DD On-Demand Anodyne ENPP1 63 35 C#C[C@@H](CC)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666675 CD On-Demand Mild CCR3 47 40 C#C[C@H](CC)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666676 CD On-Demand Mild CCR3 47 40 COCc1cc(NC(=O)NCC2(C)CC(F)(F)C2)ccc1OC ZINC000880666677 EG On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NCC2(C)CC(F)(F)C2)ccc1OC ZINC000880666677 EG On-Demand Anodyne QRFPR 40 33 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880666679 DD On-Demand Anodyne CCR3 28 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880666679 DD On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880666680 DD On-Demand Anodyne CCR3 28 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880666680 DD On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880666681 DD On-Demand Anodyne CCR3 28 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880666681 DD On-Demand Anodyne RBP4 46 33 COCc1cc(NC(=O)N2CCn3c(nnc3-c3cn(C)cn3)C2)ccc1OC ZINC000880666682 GD On-Demand Anodyne PDGFRB 42 36 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H](c1ccccc1)C1CCOCC1 ZINC000880666683 GG On-Demand Anodyne CCR3 41 41 Cn1nnnc1-c1ccccc1NC(=O)N[C@H](c1ccccc1)C1CCOCC1 ZINC000880666684 GG On-Demand Anodyne CCR3 41 41 Cn1nnnc1-c1ccccc1NC(=O)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880666685 GD On-Demand Anodyne CCR3 48 50 Cn1nnnc1-c1ccccc1NC(=O)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880666686 GD On-Demand Anodyne CCR3 48 50 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccccc2-c2nnnn2C)CC1 ZINC000880666687 DE On-Demand Mild CCR3 21 46 COCc1cc(NC(=O)N2CCO[C@@H](C(F)F)C2)ccc1OC ZINC000880666688 EE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCO[C@@H](C(F)F)C2)ccc1OC ZINC000880666688 EE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCO[C@H](C(F)F)C2)ccc1OC ZINC000880666689 EE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCO[C@H](C(F)F)C2)ccc1OC ZINC000880666689 EE On-Demand Anodyne QRFPR 40 33 CCn1ncc(NC(=O)Nc2ccc(OC)c(COC)c2)c1C ZINC000880666690 DG On-Demand Anodyne HTR2A 39 40 CCn1ncc(NC(=O)Nc2ccc(OC)c(COC)c2)c1C ZINC000880666690 DG On-Demand Anodyne ENPP1 68 35 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666691 FD On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666691 FD On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666691 FD On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666691 FD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666692 FD On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666692 FD On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666692 FD On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666692 FD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666693 FD On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666693 FD On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666693 FD On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@@H]3C2)ccc1OC ZINC000880666693 FD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666694 FD On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666694 FD On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666694 FD On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@@H]3CS(=O)(=O)C[C@H]3C2)ccc1OC ZINC000880666694 FD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCC(C)(N3CCC3)CC2)ccc1OC ZINC000880666695 EF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC(C)(N3CCC3)CC2)ccc1OC ZINC000880666695 EF On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC(C)(N3CCC3)CC2)ccc1OC ZINC000880666695 EF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC2CCC3(CC2)COC3)ccc1OC ZINC000880666696 EF On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)NC2CCC3(CC2)COC3)ccc1OC ZINC000880666696 EF On-Demand Anodyne EPHX2 42 37 COCc1cc(NC(=O)NC2CCC3(CC2)COC3)ccc1OC ZINC000880666696 EF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC2CCC3(CC2)COC3)ccc1OC ZINC000880666696 EF On-Demand Anodyne ENPP1 44 30 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H]1C[C@@H]2CCCC[C@@H]21 ZINC000880666697 EF On-Demand Anodyne CCR3 27 53 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne TSHR 61 32 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne HTR1D 15 45 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne HTR1B 18 45 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne IL2RA 48 30 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC(c3nnnn3C)CC2)ccc1OC ZINC000880666701 FD On-Demand Anodyne ENPP1 56 34 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880666702 DE On-Demand Anodyne CCR3 16 41 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880666702 DE On-Demand Anodyne RBP4 48 35 COCc1cc(NC(=O)NCC2CC(NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666703 GG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NCC2CC(NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880666703 GG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N(C)[C@@H]2CCOC[C@H]2OC)ccc1OC ZINC000880666704 EE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)[C@H]2CCOC[C@H]2OC)ccc1OC ZINC000880666705 EE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)[C@H]2CCOC[C@@H]2OC)ccc1OC ZINC000880666706 EE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)[C@@H]2CCOC[C@@H]2OC)ccc1OC ZINC000880666707 EE On-Demand Anodyne QRFPR 41 34 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880666708 GE On-Demand Anodyne CCR3 23 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880666708 GE On-Demand Anodyne RBP4 48 39 COCc1cc(NC(=O)NCCc2ccns2)ccc1OC ZINC000880666709 DF On-Demand Anodyne PRMT3 63 35 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@H](OC2CCC2)CC1 ZINC000880666710 FF On-Demand Anodyne CCR3 42 44 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880666711 FF On-Demand Anodyne CCR3 42 44 Cn1nnnc1-c1ccccc1NC(=O)NC(CF)CF ZINC000880666712 CD On-Demand Anodyne CCR3 64 45 C#C[C@@H](CCC)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666716 CD On-Demand Mild CCR3 50 41 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne HTR1D 15 44 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne EPHX2 19 40 COCc1cc(NC(=O)N2CC[C@H](CF)C2)ccc1OC ZINC000880666720 CF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne HTR1D 15 44 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne EPHX2 19 40 COCc1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1OC ZINC000880666721 CF On-Demand Anodyne QRFPR 44 36 C#C[C@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@H]1CCCO1 ZINC000880666722 ED On-Demand Mild CCR3 43 33 C#C[C@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@@H]1CCCO1 ZINC000880666723 ED On-Demand Mild CCR3 43 33 C#C[C@@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@@H]1CCCO1 ZINC000880666724 ED On-Demand Mild CCR3 43 33 C#C[C@@H](NC(=O)Nc1ccccc1-c1nnnn1C)[C@H]1CCCO1 ZINC000880666725 ED On-Demand Mild CCR3 43 33 COCc1cc(NC(=O)N2CCc3ccsc3[C@H]2C)ccc1OC ZINC000880666727 EI On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)N2CCc3ccsc3[C@@H]2C)ccc1OC ZINC000880666728 EI On-Demand Anodyne QRFPR 43 37 CCONC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666730 CC On-Demand Anodyne CCR3 26 43 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2C[C@@]2(CO)C1 ZINC000880666734 DC On-Demand Anodyne CCR3 48 41 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2C[C@@]2(CO)C1 ZINC000880666735 DC On-Demand Anodyne CCR3 48 41 COCc1cc(NC(=O)N2CC(c3nc(C)no3)C2)ccc1OC ZINC000880666736 EE On-Demand Anodyne TSHR 48 34 COCc1cc(NC(=O)N2CC(c3nc(C)no3)C2)ccc1OC ZINC000880666736 EE On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N2CC(c3nc(C)no3)C2)ccc1OC ZINC000880666736 EE On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)N2CC(c3nc(C)no3)C2)ccc1OC ZINC000880666736 EE On-Demand Anodyne SMO 16 40 COCc1cc(NC(=O)NCCC2(C)OCCO2)ccc1OC ZINC000880666742 DE On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne PDE4A 27 42 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne EPHX2 17 42 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne PDGFRA 28 40 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne QRFPR 53 44 COCc1cc(NC(=O)NOC2CCCCC2)ccc1OC ZINC000880666745 DG On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne HTR1D 21 46 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne HTR1B 22 46 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne PDGFRB 43 36 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne ROCK2 27 43 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)ccc1OC ZINC000880666748 EF On-Demand Anodyne ENPP1 72 36 COCc1cc(NC(=O)NC[C@H](O)c2cc(F)cc(Cl)c2)ccc1OC ZINC000880666749 GG On-Demand Anodyne TSHR 48 34 COCc1cc(NC(=O)NC[C@@H](O)c2cc(F)cc(Cl)c2)ccc1OC ZINC000880666750 GG On-Demand Anodyne TSHR 48 34 COCc1cc(NC(=O)NNc2ccc(OC)cn2)ccc1OC ZINC000880666751 EE On-Demand Reactive TSHR 58 36 COCc1cc(NC(=O)NNc2ccc(OC)cn2)ccc1OC ZINC000880666751 EE On-Demand Reactive HTR2A 26 40 COCc1cc(NC(=O)NNc2ccc(OC)cn2)ccc1OC ZINC000880666751 EE On-Demand Reactive PDGFRA 52 38 COCc1cc(NC(=O)NNc2ccc(OC)cn2)ccc1OC ZINC000880666751 EE On-Demand Reactive LUCI_LUCLA 17 43 COCc1cc(NC(=O)NNc2ccc(OC)cn2)ccc1OC ZINC000880666751 EE On-Demand Reactive ENPP1 64 34 COCc1cc(NC(=O)NCc2ccc(OC(F)F)cn2)ccc1OC ZINC000880666752 FG On-Demand Anodyne TSHR 57 34 COCc1cc(NC(=O)N[C@H]2CCCCC23OCCO3)ccc1OC ZINC000880666754 FF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N[C@@H]2CCCCC23OCCO3)ccc1OC ZINC000880666755 FF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)NNC(=O)[C@H]2CCOC2)ccc1OC ZINC000880666758 DD On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCOC2)ccc1OC ZINC000880666759 DD On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NNC(=O)CC2CCCC2)ccc1OC ZINC000880666760 EF On-Demand Reactive TSHR 41 30 COCc1cc(NC(=O)NNC(=O)CC2CCCC2)ccc1OC ZINC000880666760 EF On-Demand Reactive CYSLTR1 22 41 COCc1cc(NC(=O)NNC(=O)CC2CCCC2)ccc1OC ZINC000880666760 EF On-Demand Reactive QRFPR 54 44 COCc1cc(NC(=O)NNC(=O)CC2CCCC2)ccc1OC ZINC000880666760 EF On-Demand Reactive ENPP1 57 33 COCc1cc(NC(=O)NNC(=O)CC2CC2)ccc1OC ZINC000880666761 DD On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NNC(=O)CC2CC2)ccc1OC ZINC000880666761 DD On-Demand Reactive QRFPR 50 41 COCc1cc(NC(=O)NNC(=O)CC2CC2)ccc1OC ZINC000880666761 DD On-Demand Reactive ENPP1 58 34 C#CC(C)(C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666763 CE On-Demand Mild TSHR 41 33 C#CC(C)(C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666763 CE On-Demand Mild QRFPR 41 34 C#CC(C)(C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666763 CE On-Demand Mild ENPP1 60 31 COCc1cc(NC(=O)NCCCCCCO)ccc1OC ZINC000880666764 DF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCCCCCCO)ccc1OC ZINC000880666764 DF On-Demand Anodyne QPCT 17 48 COCc1cc(NC(=O)NCCCCCCO)ccc1OC ZINC000880666764 DF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCCCCCO)ccc1OC ZINC000880666764 DF On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean TSHR 76 39 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean CA1 30 42 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean MTNR1A 45 36 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean MTNR1B 41 42 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean ROCK2 15 53 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean CA12 16 42 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean PDGFRA 43 35 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean CA9 16 42 COCc1cc(NC(=O)NCc2ccc(OC)cc2O)ccc1OC ZINC000880666768 EF On-Demand Clean ENPP1 54 29 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666769 EG On-Demand Anodyne TSHR 66 34 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666769 EG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666769 EG On-Demand Anodyne ENPP1 66 34 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666770 EG On-Demand Anodyne TSHR 66 34 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666770 EG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C)cc2)ccc1OC ZINC000880666770 EG On-Demand Anodyne ENPP1 66 34 C#CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666778 EH On-Demand Mild TSHR 59 33 C#CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666778 EH On-Demand Mild SOAT1 19 44 C#CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666778 EH On-Demand Mild QRFPR 40 37 C#CC[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666779 EH On-Demand Mild TSHR 59 33 C#CC[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666779 EH On-Demand Mild SOAT1 19 44 C#CC[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880666779 EH On-Demand Mild QRFPR 40 37 COCc1cc(NC(=O)NC[C@H](O)c2ccc(Cl)c(F)c2)ccc1OC ZINC000880666780 GG On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(Cl)c(F)c2)ccc1OC ZINC000880666781 GG On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)NCc2ccn(C)n2)ccc1OC ZINC000880666785 DD On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NCc2ccn(C)n2)ccc1OC ZINC000880666785 DD On-Demand Anodyne QPCT 20 46 COCc1cc(NC(=O)NCc2ccn(C)n2)ccc1OC ZINC000880666785 DD On-Demand Anodyne PRMT3 44 33 COCc1cc(NC(=O)NCc2ccn(C)n2)ccc1OC ZINC000880666785 DD On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)NNC(=O)CCc2ccccc2)ccc1OC ZINC000880666786 FF On-Demand Reactive TSHR 74 38 COCc1cc(NC(=O)NNC(=O)CCc2ccccc2)ccc1OC ZINC000880666786 FF On-Demand Reactive FFAR1 24 40 COCc1cc(NC(=O)NNC(=O)CCc2ccccc2)ccc1OC ZINC000880666786 FF On-Demand Reactive QRFPR 40 37 COCc1cc(NC(=O)NNC(=O)CCc2ccccc2)ccc1OC ZINC000880666786 FF On-Demand Reactive ENPP1 67 32 C#CCCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666789 CE On-Demand Mild TSHR 46 30 C#CCCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666789 CE On-Demand Mild QPCT 15 46 C#CCCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666789 CE On-Demand Mild QRFPR 42 34 COCc1cc(NC(=O)N2CCC3(CC2)CNC(=O)O3)ccc1OC ZINC000880666791 ED On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CCC3(CC2)CNC(=O)O3)ccc1OC ZINC000880666791 ED On-Demand Anodyne EPHX2 18 40 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne CCR1 37 40 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne CPT1A 54 36 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne CPT2 43 32 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne CPT1B 40 33 COCc1cc(NC(=O)N2CC[C@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666794 FI On-Demand Anodyne QRFPR 44 43 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne CCR1 37 40 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne CPT1A 54 36 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne CPT2 43 32 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne CPT1B 40 33 COCc1cc(NC(=O)N2CC[C@@H]2c2ccc(Cl)cc2)ccc1OC ZINC000880666795 FI On-Demand Anodyne QRFPR 44 43 COCc1cc(NC(=O)N2CCCC[C@H]2COC(=O)N(C)C)ccc1OC ZINC000880666796 GF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCCC[C@@H]2COC(=O)N(C)C)ccc1OC ZINC000880666797 GF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC=C(Br)C2)ccc1OC ZINC000880666800 FG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCC=C(Br)C2)ccc1OC ZINC000880666800 FG On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)N2Cc3cccc(Cl)c3C2)ccc1OC ZINC000880666802 EI On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)N2Cc3cccc(Cl)c3C2)ccc1OC ZINC000880666802 EI On-Demand Anodyne CPT1A 43 33 COCc1cc(NC(=O)N2Cc3cccc(Cl)c3C2)ccc1OC ZINC000880666802 EI On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)NOC2CCCC2)ccc1OC ZINC000880666803 CF On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NOC2CCCC2)ccc1OC ZINC000880666803 CF On-Demand Anodyne PDE4A 29 43 COCc1cc(NC(=O)NOC2CCCC2)ccc1OC ZINC000880666803 CF On-Demand Anodyne QRFPR 54 44 COCc1cc(NC(=O)NOC2CCCC2)ccc1OC ZINC000880666803 CF On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)NC[C@@H](O)c2cc(C)cc(C)c2)ccc1OC ZINC000880666805 FG On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)NC[C@@H](O)c2cc(C)cc(C)c2)ccc1OC ZINC000880666805 FG On-Demand Anodyne ENPP1 66 34 COCc1cc(NC(=O)NC[C@H](O)c2cc(C)cc(C)c2)ccc1OC ZINC000880666806 FG On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)NC[C@H](O)c2cc(C)cc(C)c2)ccc1OC ZINC000880666806 FG On-Demand Anodyne ENPP1 66 34 COCc1cc(NC(=O)N(C)[C@H](C)C(N)=O)ccc1OC ZINC000880666812 CD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N(C)[C@H](C)C(N)=O)ccc1OC ZINC000880666812 CD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N(C)[C@H](C)C(N)=O)ccc1OC ZINC000880666812 CD On-Demand Anodyne ENPP1 68 33 COCc1cc(NC(=O)N(C)[C@@H](C)C(N)=O)ccc1OC ZINC000880666813 CD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N(C)[C@@H](C)C(N)=O)ccc1OC ZINC000880666813 CD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N(C)[C@@H](C)C(N)=O)ccc1OC ZINC000880666813 CD On-Demand Anodyne ENPP1 68 33 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne CNR2 19 44 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne PDE4A 18 43 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne RAF1 33 41 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne FLT1 16 40 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne ROCK2 16 50 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne QPCT 20 48 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne PRMT3 60 33 COCc1cc(NC(=O)NCCc2ccncc2)ccc1OC ZINC000880666814 DF On-Demand Anodyne ENPP1 58 35 COCc1cc(NC(=O)N2CCC[C@H]2c2c(C)nn(C)c2Cl)ccc1OC ZINC000880666817 GH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCC[C@H]2c2c(C)nn(C)c2Cl)ccc1OC ZINC000880666817 GH On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)N2CCC[C@@H]2c2c(C)nn(C)c2Cl)ccc1OC ZINC000880666818 GH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CCC[C@@H]2c2c(C)nn(C)c2Cl)ccc1OC ZINC000880666818 GH On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)NCCCc2c(C)noc2C)ccc1OC ZINC000880666819 EG On-Demand Anodyne TSHR 54 32 CC[C@H](Nc1cccnc1Cl)C(=O)N[C@@H]1CCC[C@@H]([S@@](C)=O)C1 ZINC000880666824 FF On-Demand Anodyne G2YM83_BOTF4 58 34 CC[C@H](Nc1cccnc1Cl)C(=O)N[C@@H]1CCC[C@@H]([S@](C)=O)C1 ZINC000880666825 FF On-Demand Anodyne G2YM83_BOTF4 58 34 CC[C@H](Nc1cccnc1Cl)C(=O)N[C@@H]1CCC[C@H]([S@@](C)=O)C1 ZINC000880666826 FF On-Demand Anodyne G2YM83_BOTF4 58 34 CC[C@H](Nc1cccnc1Cl)C(=O)N[C@@H]1CCC[C@H]([S@](C)=O)C1 ZINC000880666827 FF On-Demand Anodyne G2YM83_BOTF4 58 34 COCc1cc(NC(=O)N2CCC[C@H](c3ccnn3C)C2)ccc1OC ZINC000880666845 FF On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC[C@H](c3ccnn3C)C2)ccc1OC ZINC000880666845 FF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@H](c3ccnn3C)C2)ccc1OC ZINC000880666845 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@H](c3ccnn3C)C2)ccc1OC ZINC000880666845 FF On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N2CCC[C@@H](c3ccnn3C)C2)ccc1OC ZINC000880666846 FF On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC[C@@H](c3ccnn3C)C2)ccc1OC ZINC000880666846 FF On-Demand Anodyne HTR1D 15 41 COCc1cc(NC(=O)N2CCC[C@@H](c3ccnn3C)C2)ccc1OC ZINC000880666846 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@@H](c3ccnn3C)C2)ccc1OC ZINC000880666846 FF On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N2CCC[C@H]2c2cc(C)on2)ccc1OC ZINC000880666849 EH On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CCC[C@H]2c2cc(C)on2)ccc1OC ZINC000880666849 EH On-Demand Anodyne CPT1A 40 39 COCc1cc(NC(=O)N2CCC[C@H]2c2cc(C)on2)ccc1OC ZINC000880666849 EH On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@@H]2c2cc(C)on2)ccc1OC ZINC000880666850 EH On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CCC[C@@H]2c2cc(C)on2)ccc1OC ZINC000880666850 EH On-Demand Anodyne CPT1A 40 39 COCc1cc(NC(=O)N2CCC[C@@H]2c2cc(C)on2)ccc1OC ZINC000880666850 EH On-Demand Anodyne QRFPR 41 34 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@H]2C[C@]2(CO)C1 ZINC000880666851 DC On-Demand Anodyne CCR3 48 41 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne HTR2A 22 43 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne PPIA 30 40 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne RAF1 24 45 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne KDR 24 42 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne ENPP1 40 33 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne IMDH_CRYPV 58 40 COCc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)ccc1OC ZINC000880666858 EH On-Demand Anodyne KCNK3 50 38 COCc1cc(NC(=O)NCCCSc2nccs2)ccc1OC ZINC000880666861 FH On-Demand Clean ENPP1 64 35 Cn1nnnc1-c1ccccc1NC(=O)N1C[C@@H]2C[C@]2(CO)C1 ZINC000880666862 DC On-Demand Anodyne CCR3 48 41 COCC1CC(NC(=O)Nc2ccccc2-c2nnnn2C)C1 ZINC000880666867 DD On-Demand Anodyne CCR3 39 48 Cc1cncc([C@@H]2CCCN2C(=O)Nc2ccccc2-c2nnnn2C)c1 ZINC000880666869 FF On-Demand Anodyne CCR3 54 43 Cn1nnnc1-c1ccccc1NC(=O)NC1CCN(C(C)(C)C)CC1 ZINC000880666870 FE On-Demand Anodyne CCR3 43 48 Cc1cncc([C@H]2CCCN2C(=O)Nc2ccccc2-c2nnnn2C)c1 ZINC000880666871 FF On-Demand Anodyne CCR3 54 43 COCc1cc(NC(=O)N2CC(CNC(=O)C(F)(F)F)C2)ccc1OC ZINC000880666874 GD On-Demand Anodyne QRFPR 40 32 Cn1nnnc1-c1ccccc1NC(=O)N[C@H]1C=CCC1 ZINC000880666880 CD On-Demand Anodyne CCR3 44 47 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CC1(Cl)Cl ZINC000880666881 EE On-Demand Anodyne CCR3 33 44 Cn1nnnc1-c1ccccc1NC(=O)N[C@@H]1C=CCC1 ZINC000880666882 CD On-Demand Anodyne CCR3 44 47 COCc1cc(NC(=O)NC[C@H]2C[C@H](O)C2)ccc1OC ZINC000880666883 CD On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@H]2C[C@H](O)C2)ccc1OC ZINC000880666883 CD On-Demand Anodyne QRFPR 46 38 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CC(C)(C)CO1 ZINC000880666884 ED On-Demand Anodyne CCR3 31 41 COCc1cc(NC(=O)Nc2n[nH]c(C3CC3)c2C)ccc1OC ZINC000880666885 EG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)Nc2n[nH]c(C3CC3)c2C)ccc1OC ZINC000880666885 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)Nc2n[nH]c(C3CC3)c2C)ccc1OC ZINC000880666885 EG On-Demand Anodyne ENPP1 62 33 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CC1(Cl)Cl ZINC000880666886 EE On-Demand Anodyne CCR3 33 44 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CC(C)(C)CO1 ZINC000880666887 ED On-Demand Anodyne CCR3 31 41 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@@H]1CCN(C)C1 ZINC000880666889 EG On-Demand Anodyne CCR5 15 41 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@@H]1CCN(C)C1 ZINC000880666889 EG On-Demand Anodyne PDE4D 26 40 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@@H]1CCN(C)C1 ZINC000880666889 EG On-Demand Anodyne UTS2R 22 41 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@@H]1CCN(C)C1 ZINC000880666889 EG On-Demand Anodyne CACNA1I 56 38 Cn1nnnc1-c1ccccc1NC(=O)N1CCC[C@@H]2[C@H](O)C(C)(C)[C@@H]21 ZINC000880666890 FD On-Demand Anodyne CCR3 32 42 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@H]1CCN(C)C1 ZINC000880666891 EG On-Demand Anodyne CCR5 15 41 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@H]1CCN(C)C1 ZINC000880666891 EG On-Demand Anodyne PDE4D 26 40 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@H]1CCN(C)C1 ZINC000880666891 EG On-Demand Anodyne UTS2R 22 41 CCN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@H]1CCN(C)C1 ZINC000880666891 EG On-Demand Anodyne CACNA1I 56 38 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880666893 FE On-Demand Anodyne CCR3 21 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880666893 FE On-Demand Anodyne RBP4 50 39 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880666895 FE On-Demand Anodyne CCR3 21 41 Cn1nnnc1-c1ccccc1NC(=O)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880666895 FE On-Demand Anodyne RBP4 50 39 COCc1cc(NC(=O)NNC(=O)C2CCC2)ccc1OC ZINC000880666896 DD On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NNC(=O)C2CCC2)ccc1OC ZINC000880666896 DD On-Demand Reactive QRFPR 50 41 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne HTR1B 17 43 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne PDGFRB 40 36 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC(C(=O)NOC)CC2)ccc1OC ZINC000880666898 FD On-Demand Anodyne ENPP1 40 31 Cn1nnnc1-c1ccccc1NC(=O)N1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880666900 GF On-Demand Anodyne CCR3 39 43 Cn1nnnc1-c1ccccc1NC(=O)N1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880666901 GF On-Demand Anodyne CCR3 39 43 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880666904 EE On-Demand Mild TSHR 40 31 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880666904 EE On-Demand Mild PDGFRB 44 38 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880666904 EE On-Demand Mild QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)c2ccc(C(F)(F)F)nc2)ccc1OC ZINC000880666906 GI On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N[C@@H](C)c2ccc(C(F)(F)F)nc2)ccc1OC ZINC000880666908 GI On-Demand Anodyne ENPP1 51 32 CCC1(CC)CCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666909 DI On-Demand Anodyne QRFPR 42 35 CCC1(CC)CCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880666909 DI On-Demand Anodyne ENPP1 46 32 COCc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666914 GG On-Demand Anodyne ADRB1 33 41 COCc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666914 GG On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666914 GG On-Demand Anodyne MAOB 16 43 COCc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666914 GG On-Demand Anodyne ADRB3 27 43 COCc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666914 GG On-Demand Anodyne ROCK2 15 40 COCc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666916 GG On-Demand Anodyne ADRB1 33 41 COCc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666916 GG On-Demand Anodyne TSHR 64 35 COCc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666916 GG On-Demand Anodyne MAOB 16 43 COCc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666916 GG On-Demand Anodyne ADRB3 27 43 COCc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)ccc1OC ZINC000880666916 GG On-Demand Anodyne ROCK2 15 40 Cn1nnnc1-c1ccccc1NC(=O)N1CCC(F)(F)CC1 ZINC000880666918 DE On-Demand Anodyne CCR3 21 41 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@H](O)c1ccccc1 ZINC000880666922 FG On-Demand Anodyne TSHR 60 33 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@H](O)c1ccccc1 ZINC000880666922 FG On-Demand Anodyne ENPP1 45 31 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@@H](O)c1ccccc1 ZINC000880666924 FG On-Demand Anodyne TSHR 60 33 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@@H](O)c1ccccc1 ZINC000880666924 FG On-Demand Anodyne ENPP1 45 31 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880666927 EE On-Demand Anodyne CCR3 45 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880666927 EE On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H]2CSC[C@H]2C1 ZINC000880666935 EE On-Demand Anodyne CCR3 45 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H]2CSC[C@H]2C1 ZINC000880666935 EE On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880666937 EE On-Demand Anodyne CCR3 45 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880666937 EE On-Demand Anodyne RBP4 46 33 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880666939 EE On-Demand Anodyne CCR3 45 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880666939 EE On-Demand Anodyne RBP4 46 33 CSCC[C@H](C)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666945 DE On-Demand Anodyne CCR3 55 42 CSCC[C@@H](C)NC(=O)Nc1ccccc1-c1nnnn1C ZINC000880666947 DE On-Demand Anodyne CCR3 55 42 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@H]1Cc1ccccc1 ZINC000880666949 EF On-Demand Anodyne CCR3 63 48 Cn1nnnc1-c1ccccc1NC(=O)N1CC[C@@H]1Cc1ccccc1 ZINC000880666951 EF On-Demand Anodyne CCR3 63 48 COCc1cc(NC(=O)N2CCN(C)c3ncccc3C2)ccc1OC ZINC000880666953 FF On-Demand Anodyne HTR1B 17 44 COCc1cc(NC(=O)N2CCN(C)c3ncccc3C2)ccc1OC ZINC000880666953 FF On-Demand Anodyne PDGFRB 61 41 COCc1cc(NC(=O)N2CCN(C)c3ncccc3C2)ccc1OC ZINC000880666953 FF On-Demand Anodyne RBP4 16 41 COCc1cc(NC(=O)N2CCN(C)c3ncccc3C2)ccc1OC ZINC000880666953 FF On-Demand Anodyne ENPP1 48 41 Cn1nnnc1-c1ccccc1NC(=O)NCC(C)(C)C(C)(F)F ZINC000880666956 EF On-Demand Anodyne CCR3 33 43 COCc1cc(NC(=O)N(Cc2ccccc2)[C@@H](C)CO)ccc1OC ZINC000880666962 FG On-Demand Anodyne TSHR 70 36 COCc1cc(NC(=O)N(Cc2ccccc2)[C@@H](C)CO)ccc1OC ZINC000880666962 FG On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N(Cc2ccccc2)[C@H](C)CO)ccc1OC ZINC000880666964 FG On-Demand Anodyne TSHR 70 36 COCc1cc(NC(=O)N(Cc2ccccc2)[C@H](C)CO)ccc1OC ZINC000880666964 FG On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N[C@@H]2C[C@@H]3CCCC[C@@H]32)ccc1OC ZINC000880666966 DH On-Demand Anodyne QRFPR 48 40 Cn1nnnc1-c1ccccc1NC(=O)NCC1SCCS1 ZINC000880666968 ED On-Demand Anodyne CCR3 32 44 COCc1cc(NC(=O)N[C@@H]2CC=C(C(=O)OC)C2)ccc1OC ZINC000880666987 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@H]2CC=C(C(=O)OC)C2)ccc1OC ZINC000880666988 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2Cc3cccnc3N3CCC[C@H]3C2)ccc1OC ZINC000880666997 GG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2Cc3cccnc3N3CCC[C@H]3C2)ccc1OC ZINC000880666997 GG On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2Cc3cccnc3N3CCC[C@H]3C2)ccc1OC ZINC000880666997 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC(OC[C@H]3CCCO3)CC2)ccc1OC ZINC000880667002 GG On-Demand Anodyne HTR1B 15 40 COCc1cc(NC(=O)N2CCC(OC[C@H]3CCCO3)CC2)ccc1OC ZINC000880667002 GG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC(OC[C@@H]3CCCO3)CC2)ccc1OC ZINC000880667003 GG On-Demand Anodyne HTR1B 15 40 COCc1cc(NC(=O)N2CCC(OC[C@@H]3CCCO3)CC2)ccc1OC ZINC000880667003 GG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)ccc1OC ZINC000880667004 GG On-Demand Mild HTR1D 20 54 COCc1cc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)ccc1OC ZINC000880667004 GG On-Demand Mild HTR1B 22 54 COCc1cc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)ccc1OC ZINC000880667004 GG On-Demand Mild P2RY12 15 45 COCc1cc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)ccc1OC ZINC000880667004 GG On-Demand Mild PDGFRB 52 43 COCc1cc(NC(=O)N2CCN(c3ccc(F)cc3C#N)CC2)ccc1OC ZINC000880667004 GG On-Demand Mild NPY2R 48 39 CCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667005 CE On-Demand Anodyne TSHR 55 34 CCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667005 CE On-Demand Anodyne QRFPR 41 34 CCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667005 CE On-Demand Anodyne ENPP1 68 33 COCc1cc(NC(=O)NC[C@@H]2C[C@H]2C2CCOCC2)ccc1OC ZINC000880667006 EG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@H](C)[C@@](C)(O)c2ccccc2)ccc1OC ZINC000880667007 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N[C@@H](C)[C@@](C)(O)c2ccccc2)ccc1OC ZINC000880667008 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N[C@H](C)[C@](C)(O)c2ccccc2)ccc1OC ZINC000880667009 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N[C@@H](C)[C@](C)(O)c2ccccc2)ccc1OC ZINC000880667010 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N(C)CCc2cccc(C#N)c2)ccc1OC ZINC000880667011 FG On-Demand Mild TSHR 43 33 COCc1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1OC ZINC000880667014 DC On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1OC ZINC000880667014 DC On-Demand Anodyne HTR1D 17 43 COCc1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1OC ZINC000880667014 DC On-Demand Anodyne HTR1B 20 43 COCc1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1OC ZINC000880667014 DC On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1OC ZINC000880667014 DC On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667019 GG On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667019 GG On-Demand Anodyne KCNA3 41 36 COCc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667019 GG On-Demand Anodyne EPHX2 28 57 COCc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667019 GG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667020 GG On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667020 GG On-Demand Anodyne KCNA3 41 36 COCc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667020 GG On-Demand Anodyne EPHX2 28 57 COCc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)ccc1OC ZINC000880667020 GG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)NCCc2nnc(S)n2C(C)C)ccc1OC ZINC000880667021 GF On-Demand Anodyne PRMT3 43 30 COCc1cc(NC(=O)NCCc2nnc(S)n2C(C)C)ccc1OC ZINC000880667021 GF On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)NOCCC2CC2)ccc1OC ZINC000880667024 CF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NOCCC2CC2)ccc1OC ZINC000880667024 CF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)NOCCC2CC2)ccc1OC ZINC000880667024 CF On-Demand Anodyne ENPP1 44 31 COCc1cc(NC(=O)Nc2cc(Br)nn2C)ccc1OC ZINC000880667025 FF On-Demand Anodyne HTR2A 44 45 COCc1cc(NC(=O)Nc2cc(Br)nn2C)ccc1OC ZINC000880667025 FF On-Demand Anodyne HTR2C 17 45 COCc1cc(NC(=O)Nc2cc(Br)nn2C)ccc1OC ZINC000880667025 FF On-Demand Anodyne ENPP1 73 37 CC[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)C(OC)OC ZINC000880667026 EE On-Demand Anodyne ENPP1 49 31 COCc1cc(NC(=O)N2C[C@@H](NC(=O)OC(C)(C)C)C[C@@H]2C)ccc1OC ZINC000880667028 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@@H](NC(=O)OC(C)(C)C)C[C@H]2C)ccc1OC ZINC000880667029 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@H](NC(=O)OC(C)(C)C)C[C@H]2C)ccc1OC ZINC000880667030 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@H](NC(=O)OC(C)(C)C)C[C@@H]2C)ccc1OC ZINC000880667031 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667032 FE On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CC[C@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667032 FE On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)N2CC[C@@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667033 FE On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CC[C@@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667033 FE On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)NCCOC(=O)C2CC2)ccc1OC ZINC000880667038 DD On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)NCCOC(=O)C2CC2)ccc1OC ZINC000880667038 DD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC(C#N)CC2)ccc1OC ZINC000880667039 DF On-Demand Mild TSHR 53 31 COCc1cc(NC(=O)N2CCC(C#N)CC2)ccc1OC ZINC000880667039 DF On-Demand Mild HTR1D 15 46 COCc1cc(NC(=O)N2CCC(C#N)CC2)ccc1OC ZINC000880667039 DF On-Demand Mild HTR1B 18 43 COCc1cc(NC(=O)N2CCC(C#N)CC2)ccc1OC ZINC000880667039 DF On-Demand Mild PDGFRB 43 39 COCc1cc(NC(=O)N2CCC(C#N)CC2)ccc1OC ZINC000880667039 DF On-Demand Mild QRFPR 44 36 C#CC[C@@H](COC)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667040 DE On-Demand Mild QRFPR 40 33 C#CC[C@H](COC)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667041 DE On-Demand Mild QRFPR 40 33 COCc1cc(NC(=O)N2CCC[C@@H]3[C@H](O)C(C)(C)[C@@H]32)ccc1OC ZINC000880667046 EF On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC[C@@H]3[C@H](O)C(C)(C)[C@@H]32)ccc1OC ZINC000880667046 EF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NCCNC(=O)OC)ccc1OC ZINC000880667047 DD On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NCCNC(=O)OC)ccc1OC ZINC000880667047 DD On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)NCCNC(=O)OC)ccc1OC ZINC000880667047 DD On-Demand Anodyne ENPP1 56 31 COCc1cc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)ccc1OC ZINC000880667048 FF On-Demand Anodyne HTR1B 16 51 COCc1cc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)ccc1OC ZINC000880667048 FF On-Demand Anodyne PDGFRB 64 43 COCc1cc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)ccc1OC ZINC000880667048 FF On-Demand Anodyne MET 44 39 COCc1cc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)ccc1OC ZINC000880667048 FF On-Demand Anodyne PDGFRA 21 42 COCc1cc(NC(=O)N2CCN(c3ccnc(F)c3)CC2)ccc1OC ZINC000880667048 FF On-Demand Anodyne ENPP1 47 36 COCc1cc(NC(=O)NC(C)(C)[C@@H]2CCCCO2)ccc1OC ZINC000880667049 EG On-Demand Anodyne QRFPR 48 41 COCc1cc(NC(=O)NC(C)(C)[C@H]2CCCCO2)ccc1OC ZINC000880667050 EG On-Demand Anodyne QRFPR 48 41 COCc1cc(NC(=O)N[C@H]2CCOC2=O)ccc1OC ZINC000880667051 CD On-Demand Anodyne TSHR 65 31 COCc1cc(NC(=O)N[C@H]2CCOC2=O)ccc1OC ZINC000880667051 CD On-Demand Anodyne LUXR 78 42 COCc1cc(NC(=O)N[C@H]2CCOC2=O)ccc1OC ZINC000880667051 CD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@H]2CCOC2=O)ccc1OC ZINC000880667051 CD On-Demand Anodyne TRAR 92 42 COCc1cc(NC(=O)N[C@H]2CCOC2=O)ccc1OC ZINC000880667051 CD On-Demand Anodyne LASR 64 41 COCc1cc(NC(=O)NCCc2cn(C)c3ncccc23)ccc1OC ZINC000880667053 FG On-Demand Anodyne TSHR 57 36 COCc1cc(NC(=O)NCCc2cn(C)c3ncccc23)ccc1OC ZINC000880667053 FG On-Demand Anodyne QPCT 16 44 COCc1cc(NC(=O)NCCc2cn(C)c3ncccc23)ccc1OC ZINC000880667053 FG On-Demand Anodyne ENPP1 41 36 COCc1cc(NC(=O)N2CC[C@@]3(CC(C(=O)OC)=NO3)C2)ccc1OC ZINC000880667060 GD On-Demand Anodyne EPHX2 29 44 COCc1cc(NC(=O)N2CC[C@]3(CC(C(=O)OC)=NO3)C2)ccc1OC ZINC000880667061 GD On-Demand Anodyne EPHX2 29 44 COCc1cc(NC(=O)NC2CC(COC)C2)ccc1OC ZINC000880667062 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NC2CC(COC)C2)ccc1OC ZINC000880667062 DE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC2CC(COC)C2)ccc1OC ZINC000880667062 DE On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)ccc1OC ZINC000880667063 GF On-Demand Anodyne TSHR 75 37 COCc1cc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)ccc1OC ZINC000880667063 GF On-Demand Anodyne ROCK2 18 41 COCc1cc(NC(=O)NCc2ccc(CN3CCNC3=O)cc2)ccc1OC ZINC000880667063 GF On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667070 FH On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)N2CCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667070 FH On-Demand Anodyne TACR1 19 45 COCc1cc(NC(=O)N2CCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667070 FH On-Demand Anodyne PDE4A 19 40 COCc1cc(NC(=O)N2CCC[C@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667070 FH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667071 FH On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)N2CCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667071 FH On-Demand Anodyne TACR1 19 45 COCc1cc(NC(=O)N2CCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667071 FH On-Demand Anodyne PDE4A 19 40 COCc1cc(NC(=O)N2CCC[C@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667071 FH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667072 FH On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)N2CCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667072 FH On-Demand Anodyne TACR1 19 45 COCc1cc(NC(=O)N2CCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667072 FH On-Demand Anodyne PDE4A 19 40 COCc1cc(NC(=O)N2CCC[C@@H]2[C@@H](O)c2ccccc2)ccc1OC ZINC000880667072 FH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667073 FH On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)N2CCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667073 FH On-Demand Anodyne TACR1 19 45 COCc1cc(NC(=O)N2CCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667073 FH On-Demand Anodyne PDE4A 19 40 COCc1cc(NC(=O)N2CCC[C@@H]2[C@H](O)c2ccccc2)ccc1OC ZINC000880667073 FH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CC[C@](C)(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667074 GG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N2CC[C@@](C)(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667075 GG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N[C@@H]2C=CCC2)ccc1OC ZINC000880667076 CF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@@H]2C=CCC2)ccc1OC ZINC000880667076 CF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N[C@H]2C=CCC2)ccc1OC ZINC000880667077 CF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@H]2C=CCC2)ccc1OC ZINC000880667077 CF On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N[C@@H]2CC=CC[C@H]2C(F)(F)F)ccc1OC ZINC000880667078 FH On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCO[C@](C)(C(F)(F)F)C2)ccc1OC ZINC000880667079 FG On-Demand Anodyne EPHX2 34 48 COCc1cc(NC(=O)N2CCO[C@@](C)(C(F)(F)F)C2)ccc1OC ZINC000880667080 FG On-Demand Anodyne EPHX2 34 48 COCc1cc(NC(=O)NCCC2CCN(C(C)C)CC2)ccc1OC ZINC000880667083 FG On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)NCCC2CCN(C(C)C)CC2)ccc1OC ZINC000880667083 FG On-Demand Anodyne CCR3 43 39 COCc1cc(NC(=O)NCCC2CCN(C(C)C)CC2)ccc1OC ZINC000880667083 FG On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)NCCC2CCN(C(C)C)CC2)ccc1OC ZINC000880667083 FG On-Demand Anodyne PRMT3 24 41 COCc1cc(NC(=O)NNCC(F)(F)C(F)(F)F)ccc1OC ZINC000880667084 FF On-Demand Reactive ENPP1 44 30 COCc1cc(NC(=O)NCc2nn(C)cc2C(F)F)ccc1OC ZINC000880667085 FF On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)NCc2nn(C)cc2C(F)F)ccc1OC ZINC000880667085 FF On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NO[C@H]2CCCCO2)ccc1OC ZINC000880667087 DE On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NO[C@H]2CCCCO2)ccc1OC ZINC000880667087 DE On-Demand Anodyne QRFPR 50 42 COCc1cc(NC(=O)NO[C@@H]2CCCCO2)ccc1OC ZINC000880667088 DE On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NO[C@@H]2CCCCO2)ccc1OC ZINC000880667088 DE On-Demand Anodyne QRFPR 50 42 COCc1cc(NC(=O)N[C@@H](C)[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667090 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@@H](C)[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667090 GF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)N[C@H](C)[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667091 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@H](C)[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667091 GF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)N[C@@H](C)[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667092 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@@H](C)[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667092 GF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)N[C@H](C)[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667093 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@H](C)[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880667093 GF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)NC[C@@H]2CCC=CO2)ccc1OC ZINC000880667096 DF On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)NC[C@@H]2CCC=CO2)ccc1OC ZINC000880667096 DF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NC[C@H]2CCC=CO2)ccc1OC ZINC000880667097 DF On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)NC[C@H]2CCC=CO2)ccc1OC ZINC000880667097 DF On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NCC2(C)OCCCO2)ccc1OC ZINC000880667100 DE On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NCC2(C)OCCCO2)ccc1OC ZINC000880667100 DE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667101 EE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667101 EE On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N[C@@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667101 EE On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)N[C@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667102 EE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667102 EE On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N[C@H](CC(=O)OC)C2CC2)ccc1OC ZINC000880667102 EE On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)NC[C@H]2COC3(CCCCC3)O2)ccc1OC ZINC000880667103 FG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NC[C@@H]2COC3(CCCCC3)O2)ccc1OC ZINC000880667104 FG On-Demand Anodyne QRFPR 42 35 CC[C@@H](C)C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667106 DE On-Demand Reactive QRFPR 41 35 CC[C@@H](C)C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667106 DE On-Demand Reactive ENPP1 55 31 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccc3c(c2)OCO3)ccc1OC ZINC000880667107 GF On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NCC2(O)CCC3(CC2)OCCO3)ccc1OC ZINC000880667124 GE On-Demand Anodyne TSHR 51 29 O=C(CCCn1cccn1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667127 ED On-Demand Anodyne SUCNR1 57 39 COCc1cc(NC(=O)NC[C@@]2(O)CCc3ccccc32)ccc1OC ZINC000880667132 FF On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NC[C@]2(O)CCc3ccccc32)ccc1OC ZINC000880667133 FF On-Demand Anodyne TSHR 67 32 O=C(CCn1ccnc1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667135 ED On-Demand Anodyne TBXAS1 46 42 COCc1cc(NC(=O)N2CCCC23CCC3)ccc1OC ZINC000880667139 DG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCCC23CCC3)ccc1OC ZINC000880667139 DG On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCCC23CCC3)ccc1OC ZINC000880667139 DG On-Demand Anodyne ENPP1 57 33 C#CCCCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667151 CF On-Demand Mild QRFPR 41 33 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive TSHR 58 36 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive KIT 21 41 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive KDR 27 43 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive PDGFRA 36 43 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive ENPP1 47 34 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive KCNK3 48 38 COCc1cc(NC(=O)NNC(=O)COc2cccc(C)c2)ccc1OC ZINC000880667152 FE On-Demand Reactive KCNK9 48 36 COCc1cc(NC(=O)NC2CCC(C)(O)CC2)ccc1OC ZINC000880667153 DF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NC2CCC(C)(O)CC2)ccc1OC ZINC000880667153 DF On-Demand Anodyne EPHX2 49 43 COCc1cc(NC(=O)NC2CCC(C)(O)CC2)ccc1OC ZINC000880667153 DF On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2cnn(C)c2)ccc1OC ZINC000880667154 GF On-Demand Anodyne ACKR3 62 33 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2cnn(C)c2)ccc1OC ZINC000880667155 GF On-Demand Anodyne ACKR3 62 33 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2cnn(C)c2)ccc1OC ZINC000880667156 GF On-Demand Anodyne ACKR3 62 33 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2cnn(C)c2)ccc1OC ZINC000880667157 GF On-Demand Anodyne ACKR3 62 33 COCc1cc(NC(=O)N2C[C@@H]3C[C@]3(CO)C2)ccc1OC ZINC000880667158 DD On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)N2C[C@@H]3C[C@]3(CO)C2)ccc1OC ZINC000880667158 DD On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2C[C@@H]3C[C@@]3(CO)C2)ccc1OC ZINC000880667159 DD On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)N2C[C@@H]3C[C@@]3(CO)C2)ccc1OC ZINC000880667159 DD On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2C[C@H]3C[C@]3(CO)C2)ccc1OC ZINC000880667160 DD On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)N2C[C@H]3C[C@]3(CO)C2)ccc1OC ZINC000880667160 DD On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2C[C@H]3C[C@@]3(CO)C2)ccc1OC ZINC000880667161 DD On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)N2C[C@H]3C[C@@]3(CO)C2)ccc1OC ZINC000880667161 DD On-Demand Anodyne QRFPR 40 34 O=C(Cc1cccs1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667162 EE On-Demand Anodyne CA5B 31 43 O=C(Cc1cccs1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667162 EE On-Demand Anodyne CA5A 31 43 COCc1cc(NC(=O)NC[C@@H]2CSCCS2)ccc1OC ZINC000880667163 EF On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)NC[C@@H]2CSCCS2)ccc1OC ZINC000880667163 EF On-Demand Anodyne QRFPR 45 39 COCc1cc(NC(=O)NC[C@H]2CSCCS2)ccc1OC ZINC000880667164 EF On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)NC[C@H]2CSCCS2)ccc1OC ZINC000880667164 EF On-Demand Anodyne QRFPR 45 39 COCc1cc(NC(=O)NC[C@@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667165 FF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NC[C@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667166 FF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC(=O)N(C)C[C@H]2C)ccc1OC ZINC000880667167 DD On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CC(=O)N(C)C[C@H]2C)ccc1OC ZINC000880667167 DD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC(=O)N(C)C[C@@H]2C)ccc1OC ZINC000880667168 DD On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CC(=O)N(C)C[C@@H]2C)ccc1OC ZINC000880667168 DD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NNc2nccnc2C(C)C)ccc1OC ZINC000880667169 EF On-Demand Reactive TSHR 47 31 COCc1cc(NC(=O)NNc2nccnc2C(C)C)ccc1OC ZINC000880667169 EF On-Demand Reactive ENPP1 47 34 CCCCSCC(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667173 EF On-Demand Anodyne EST1_PIG 44 37 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880667174 FD On-Demand Mild TSHR 41 30 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880667174 FD On-Demand Mild HTR1D 15 43 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880667174 FD On-Demand Mild HTR1B 17 43 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880667174 FD On-Demand Mild EPHX2 19 41 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880667174 FD On-Demand Mild QRFPR 45 38 COCc1cc(NC(=O)N2CCC[C@H](c3nccn3C)C2)ccc1OC ZINC000880667180 FF On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCC[C@H](c3nccn3C)C2)ccc1OC ZINC000880667180 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@@H](c3nccn3C)C2)ccc1OC ZINC000880667181 FF On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCC[C@@H](c3nccn3C)C2)ccc1OC ZINC000880667181 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NNC(=O)C23CC4CC(CC(C4)C2)C3)ccc1OC ZINC000880667182 GG On-Demand Reactive EPHX2 48 44 COCc1cc(NC(=O)NNC(=O)C23CC4CC(CC(C4)C2)C3)ccc1OC ZINC000880667182 GG On-Demand Reactive QRFPR 47 39 C#C[C@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667184 CD On-Demand Mild TSHR 40 30 C#C[C@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667184 CD On-Demand Mild QRFPR 41 35 C#C[C@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667184 CD On-Demand Mild ENPP1 45 30 C#C[C@@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667185 CD On-Demand Mild TSHR 40 30 C#C[C@@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667185 CD On-Demand Mild QRFPR 41 35 C#C[C@@H](C)NC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667185 CD On-Demand Mild ENPP1 45 30 COCc1cc(NC(=O)N2CCc3c(F)cccc3C2)ccc1OC ZINC000880667186 EH On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)N2CCc3c(F)cccc3C2)ccc1OC ZINC000880667186 EH On-Demand Anodyne P2RY14 46 34 COc1cc(C)c(C)cc1NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880667208 EF On-Demand Anodyne CNR2 15 41 COc1cc(C)c(C)cc1NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880667208 EF On-Demand Anodyne CSF1R 24 41 COCc1cc(NC(=O)N[C@H](C)[C@@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667264 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)[C@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667266 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H](C)[C@@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667268 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H](C)[C@H](C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880667270 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@H](CN3CCOC3=O)C2)ccc1OC ZINC000880667272 FE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2CC[C@H](CN3CCOC3=O)C2)ccc1OC ZINC000880667274 FE On-Demand Anodyne TSHR 40 30 CCON(C)C(=O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667276 ED On-Demand Anodyne TSHR 46 30 CCON(C)C(=O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667276 ED On-Demand Anodyne ENPP1 61 31 COCc1cc(NC(=O)N2CCOc3ccc(OC)cc3C2)ccc1OC ZINC000880667278 FG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCO2)ccc1OC ZINC000880667280 DD On-Demand Reactive TSHR 40 30 COCc1cc(NC(=O)NNC(=O)[C@H]2CCCO2)ccc1OC ZINC000880667280 DD On-Demand Reactive QRFPR 49 40 COCc1cc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)ccc1OC ZINC000880667282 GG On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)ccc1OC ZINC000880667282 GG On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)NC[C@@H]2CCN(C)[C@H]2c2cccnc2)ccc1OC ZINC000880667282 GG On-Demand Anodyne NAMPT 40 37 COCc1cc(NC(=O)NC[C@]2(C)CC2(Cl)Cl)ccc1OC ZINC000880667284 EH On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@]2(C)CC2(Cl)Cl)ccc1OC ZINC000880667284 EH On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)NC[C@@]2(C)CC2(Cl)Cl)ccc1OC ZINC000880667286 EH On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@@]2(C)CC2(Cl)Cl)ccc1OC ZINC000880667286 EH On-Demand Anodyne QRFPR 42 36 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CN2CCC[C@@H]2CO1 ZINC000880667289 FC On-Demand Anodyne CCR3 58 47 COCc1cc(NC(=O)N[C@@H]2C[C@@H](C)OC2=O)ccc1OC ZINC000880667291 DD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2C[C@@H](C)OC2=O)ccc1OC ZINC000880667291 DD On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)N[C@H]2C[C@H](C)OC2=O)ccc1OC ZINC000880667292 DD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@H]2C[C@H](C)OC2=O)ccc1OC ZINC000880667292 DD On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)N[C@@H]2C[C@H](C)OC2=O)ccc1OC ZINC000880667293 DD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2C[C@H](C)OC2=O)ccc1OC ZINC000880667293 DD On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)N[C@H]2C[C@@H](C)OC2=O)ccc1OC ZINC000880667294 DD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@H]2C[C@@H](C)OC2=O)ccc1OC ZINC000880667294 DD On-Demand Anodyne QRFPR 42 36 COCc1cc(NC(=O)NCc2cc(C)ccc2O)ccc1OC ZINC000880667295 EG On-Demand Clean TSHR 61 34 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CN2CCC[C@@H]2CO1 ZINC000880667296 FC On-Demand Anodyne CCR3 58 47 COCc1cc(NC(=O)NNC(=O)[C@@H]2CCCO[C@H]2C(C)(C)C)ccc1OC ZINC000880667297 GF On-Demand Reactive QRFPR 45 38 Cn1nnnc1-c1ccccc1NC(=O)NC[C@@H]1CN2CCC[C@H]2CO1 ZINC000880667298 FC On-Demand Anodyne CCR3 58 47 COCc1cc(NC(=O)N2CCC(C(=O)N(C)OC)CC2)ccc1OC ZINC000880667299 FE On-Demand Anodyne TSHR 59 32 COCc1cc(NC(=O)N2CCC(C(=O)N(C)OC)CC2)ccc1OC ZINC000880667299 FE On-Demand Anodyne HTR1D 15 42 COCc1cc(NC(=O)N2CCC(C(=O)N(C)OC)CC2)ccc1OC ZINC000880667299 FE On-Demand Anodyne HTR1B 18 42 COCc1cc(NC(=O)N2CCC(C(=O)N(C)OC)CC2)ccc1OC ZINC000880667299 FE On-Demand Anodyne QRFPR 43 35 Cn1nnnc1-c1ccccc1NC(=O)NC[C@H]1CN2CCC[C@H]2CO1 ZINC000880667300 FC On-Demand Anodyne CCR3 58 47 COCc1cc(NC(=O)N[C@@H]2CCn3ccnc32)ccc1OC ZINC000880667310 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N[C@@H]2CCn3ccnc32)ccc1OC ZINC000880667310 DE On-Demand Anodyne HTR2A 40 39 COCc1cc(NC(=O)N[C@@H]2CCn3ccnc32)ccc1OC ZINC000880667310 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@@H]2CCn3ccnc32)ccc1OC ZINC000880667310 DE On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N[C@H]2CCn3ccnc32)ccc1OC ZINC000880667311 DE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N[C@H]2CCn3ccnc32)ccc1OC ZINC000880667311 DE On-Demand Anodyne HTR2A 40 39 COCc1cc(NC(=O)N[C@H]2CCn3ccnc32)ccc1OC ZINC000880667311 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H]2CCn3ccnc32)ccc1OC ZINC000880667311 DE On-Demand Anodyne ENPP1 62 33 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)[C@@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880667314 FG On-Demand Anodyne C3AR1 46 44 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)[C@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880667316 FG On-Demand Anodyne C3AR1 46 44 COCc1cc(NC(=O)N2C[C@H]3CC=CC[C@H]3C2)ccc1OC ZINC000880667319 DG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2C[C@H]3CC=CC[C@H]3C2)ccc1OC ZINC000880667319 DG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2C[C@H]3CC=CC[C@H]3C2)ccc1OC ZINC000880667319 DG On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)ccc1OC ZINC000880667320 GG On-Demand Clean TSHR 65 34 COCc1cc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)ccc1OC ZINC000880667320 GG On-Demand Clean HTR1D 15 42 COCc1cc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)ccc1OC ZINC000880667320 GG On-Demand Clean HTR1B 17 42 COCc1cc(NC(=O)NCc2ccc(N3CCC(O)CC3)cc2)ccc1OC ZINC000880667320 GG On-Demand Clean QRFPR 41 34 CNC(=O)OC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667321 FF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC[C@H](O)c2cc(F)c(F)c(F)c2)ccc1OC ZINC000880667323 GG On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)NC[C@H](O)c2cc(F)c(F)c(F)c2)ccc1OC ZINC000880667323 GG On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)NC[C@@H](O)c2cc(F)c(F)c(F)c2)ccc1OC ZINC000880667324 GG On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)NC[C@@H](O)c2cc(F)c(F)c(F)c2)ccc1OC ZINC000880667324 GG On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)NN2CCCCC2)ccc1OC ZINC000880667327 CE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NN2CCCCC2)ccc1OC ZINC000880667327 CE On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NN2CCCCC2)ccc1OC ZINC000880667327 CE On-Demand Anodyne ENPP1 62 32 C=CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667330 CE On-Demand Mild TSHR 40 31 C=CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667330 CE On-Demand Mild QRFPR 41 34 C=CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667330 CE On-Demand Mild ENPP1 67 32 COCc1cc(NC(=O)NOC/C=C\Cl)ccc1OC ZINC000880667335 DF On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NOC/C=C/Cl)ccc1OC ZINC000880667336 DF On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NOC(C)C)ccc1OC ZINC000880667337 CE On-Demand Anodyne TSHR 48 34 COCc1cc(NC(=O)NOC(C)C)ccc1OC ZINC000880667337 CE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NOC(C)C)ccc1OC ZINC000880667337 CE On-Demand Anodyne ENPP1 73 35 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667338 GF On-Demand Anodyne TSHR 47 31 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667338 GF On-Demand Anodyne QRFPR 40 33 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667338 GF On-Demand Anodyne ACKR3 55 31 COCc1cc(NC(=O)N[C@@H]2CC(C)(C)CC[C@H]2O)ccc1OC ZINC000880667339 EF On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N[C@@H]2CC(C)(C)CC[C@H]2O)ccc1OC ZINC000880667339 EF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@H](C)[C@H](O)c2ccccc2)ccc1OC ZINC000880667340 EG On-Demand Anodyne TSHR 67 34 COCc1cc(NC(=O)N[C@H](C)[C@H](O)c2ccccc2)ccc1OC ZINC000880667340 EG On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N[C@H](C)[C@@H](O)c2ccccc2)ccc1OC ZINC000880667341 EG On-Demand Anodyne TSHR 67 34 COCc1cc(NC(=O)N[C@H](C)[C@@H](O)c2ccccc2)ccc1OC ZINC000880667341 EG On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N[C@@H](C)[C@@H](O)c2ccccc2)ccc1OC ZINC000880667342 EG On-Demand Anodyne TSHR 67 34 COCc1cc(NC(=O)N[C@@H](C)[C@@H](O)c2ccccc2)ccc1OC ZINC000880667342 EG On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccccc2)ccc1OC ZINC000880667343 EG On-Demand Anodyne TSHR 67 34 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccccc2)ccc1OC ZINC000880667343 EG On-Demand Anodyne ENPP1 45 32 COCc1cc(NC(=O)N[C@@H](C)C(OC)OC)ccc1OC ZINC000880667348 DD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N[C@@H](C)C(OC)OC)ccc1OC ZINC000880667348 DD On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)N[C@H](C)C(OC)OC)ccc1OC ZINC000880667349 DD On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N[C@H](C)C(OC)OC)ccc1OC ZINC000880667349 DD On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)NC[C@H]2CC(C)=NO2)ccc1OC ZINC000880667350 DE On-Demand Anodyne TSHR 58 31 COCc1cc(NC(=O)NC[C@H]2CC(C)=NO2)ccc1OC ZINC000880667350 DE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@@H]2CC(C)=NO2)ccc1OC ZINC000880667351 DE On-Demand Anodyne TSHR 58 31 COCc1cc(NC(=O)NC[C@@H]2CC(C)=NO2)ccc1OC ZINC000880667351 DE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@@H]2c3ccccc3CN2C)ccc1OC ZINC000880667360 FG On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)NC[C@@H]2c3ccccc3CN2C)ccc1OC ZINC000880667360 FG On-Demand Anodyne QRFPR 42 37 COCc1cc(NC(=O)NC[C@H]2c3ccccc3CN2C)ccc1OC ZINC000880667361 FG On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)NC[C@H]2c3ccccc3CN2C)ccc1OC ZINC000880667361 FG On-Demand Anodyne QRFPR 42 37 COCc1cc(NC(=O)NC(c2ccnn2C)c2ccnn2C)ccc1OC ZINC000880667362 GE On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)NC(c2ccnn2C)c2ccnn2C)ccc1OC ZINC000880667362 GE On-Demand Anodyne HTR2A 43 48 COCc1cc(NC(=O)NC(c2ccnn2C)c2ccnn2C)ccc1OC ZINC000880667362 GE On-Demand Anodyne HTR2C 15 48 COCc1cc(NC(=O)NC(c2ccnn2C)c2ccnn2C)ccc1OC ZINC000880667362 GE On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N2C[C@@H](OC)CC[C@H]2C)ccc1OC ZINC000880667363 DF On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)N2C[C@@H](OC)CC[C@H]2C)ccc1OC ZINC000880667363 DF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@H](OC)CC[C@H]2C)ccc1OC ZINC000880667364 DF On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)N2C[C@H](OC)CC[C@H]2C)ccc1OC ZINC000880667364 DF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@H](OC)CC[C@@H]2C)ccc1OC ZINC000880667365 DF On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)N2C[C@H](OC)CC[C@@H]2C)ccc1OC ZINC000880667365 DF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@@H](OC)CC[C@@H]2C)ccc1OC ZINC000880667366 DF On-Demand Anodyne TSHR 72 35 COCc1cc(NC(=O)N2C[C@@H](OC)CC[C@@H]2C)ccc1OC ZINC000880667366 DF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2C[C@@H](O)CC(C)(C)C2)ccc1OC ZINC000880667367 DE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2C[C@@H](O)CC(C)(C)C2)ccc1OC ZINC000880667367 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2C[C@H](O)CC(C)(C)C2)ccc1OC ZINC000880667368 DE On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2C[C@H](O)CC(C)(C)C2)ccc1OC ZINC000880667368 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H](C)c2ccccc2O)ccc1OC ZINC000880667369 EG On-Demand Clean TSHR 64 36 COCc1cc(NC(=O)N[C@H](C)c2ccccc2O)ccc1OC ZINC000880667369 EG On-Demand Clean CA1 15 43 COCc1cc(NC(=O)N[C@H](C)c2ccccc2O)ccc1OC ZINC000880667369 EG On-Demand Clean KCNK3 37 40 COCc1cc(NC(=O)N[C@H](C)c2ccccc2O)ccc1OC ZINC000880667369 EG On-Demand Clean KCNK9 33 40 COCc1cc(NC(=O)N[C@@H](C)c2ccccc2O)ccc1OC ZINC000880667370 EG On-Demand Clean TSHR 64 36 COCc1cc(NC(=O)N[C@@H](C)c2ccccc2O)ccc1OC ZINC000880667370 EG On-Demand Clean CA1 15 43 COCc1cc(NC(=O)N[C@@H](C)c2ccccc2O)ccc1OC ZINC000880667370 EG On-Demand Clean KCNK3 37 40 COCc1cc(NC(=O)N[C@@H](C)c2ccccc2O)ccc1OC ZINC000880667370 EG On-Demand Clean KCNK9 33 40 COCc1cc(NC(=O)NCc2ocnc2C)ccc1OC ZINC000880667371 DE On-Demand Anodyne TSHR 65 35 COCc1cc(NC(=O)NCc2ocnc2C)ccc1OC ZINC000880667371 DE On-Demand Anodyne ENPP1 46 32 CCOC(=O)C1=CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880667372 EF On-Demand Anodyne QRFPR 41 34 CCOC(=O)C1=CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880667373 EF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880667384 GG On-Demand Clean TSHR 58 35 COCc1cc(NC(=O)NC[C@@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880667384 GG On-Demand Clean QRFPR 42 34 COCc1cc(NC(=O)NC[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880667385 GG On-Demand Clean TSHR 58 35 COCc1cc(NC(=O)NC[C@H]2CCN(c3ccc(OC)cc3)C2)ccc1OC ZINC000880667385 GG On-Demand Clean QRFPR 42 34 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)[C@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880667468 FG On-Demand Anodyne C3AR1 46 44 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)[C@@H](Cc2cccnc2)C2CCCC2)C1 ZINC000880667469 FG On-Demand Anodyne C3AR1 46 44 CCN(C(=O)CCCCc1ccc(OC)c(OC)c1)[C@H]1CCN(C)C1 ZINC000880667470 EF On-Demand Anodyne FKBP1A 44 41 CCN(C(=O)CCCCc1ccc(OC)c(OC)c1)[C@H]1CCN(C)C1 ZINC000880667470 EF On-Demand Anodyne CCR5 27 43 CCN(C(=O)CCCCc1ccc(OC)c(OC)c1)[C@@H]1CCN(C)C1 ZINC000880667471 EF On-Demand Anodyne FKBP1A 44 41 CCN(C(=O)CCCCc1ccc(OC)c(OC)c1)[C@@H]1CCN(C)C1 ZINC000880667471 EF On-Demand Anodyne CCR5 27 43 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880667472 GE On-Demand Anodyne KCNQ2 58 35 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880667472 GE On-Demand Anodyne CCR3 20 41 Cn1nnnc1-c1ccccc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880667472 GE On-Demand Anodyne SCN10A 15 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1cc(F)ccc1C ZINC000880667473 FF On-Demand Reactive PAPA1_CARPA 38 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1cc(F)ccc1C ZINC000880667474 FF On-Demand Reactive PAPA1_CARPA 38 44 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880667507 GG On-Demand Anodyne SLC6A5 36 40 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880667508 GG On-Demand Anodyne SLC6A5 36 40 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880667509 GG On-Demand Anodyne SLC6A5 36 40 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Cc2ccc(OCc3ccncc3)cc2)C1 ZINC000880667510 GG On-Demand Anodyne SLC6A5 36 40 COCc1cc(NC(=O)NC[C@@H]2COCO2)ccc1OC ZINC000880667528 CD On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NC[C@@H]2COCO2)ccc1OC ZINC000880667528 CD On-Demand Anodyne QRFPR 46 39 COCc1cc(NC(=O)NC[C@H]2COCO2)ccc1OC ZINC000880667529 CD On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NC[C@H]2COCO2)ccc1OC ZINC000880667529 CD On-Demand Anodyne QRFPR 46 39 CCC(C)(C)[C@@H](C)NC(=O)[C@H](CNC(=O)OC(C)(C)C)OC ZINC000880667534 DE On-Demand Anodyne PAPA1_CARPA 38 41 COCc1cc(NC(=O)Nn2cnnc2)ccc1OC ZINC000880667571 CD On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)Nn2cnnc2)ccc1OC ZINC000880667571 CD On-Demand Anodyne QPCT 15 41 COCc1cc(NC(=O)Nn2cnnc2)ccc1OC ZINC000880667571 CD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)Nn2cnnc2)ccc1OC ZINC000880667571 CD On-Demand Anodyne ENPP1 72 34 COCc1cc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)ccc1OC ZINC000880667582 FI On-Demand Anodyne TSHR 70 34 COCc1cc(NC(=O)N2C[C@@H]3[C@@H](C[C@H]3c3ccccc3)C2)ccc1OC ZINC000880667582 FI On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)NC[C@@H]2C[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667585 GG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC[C@@H]2C[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667585 GG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@@H]2C[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667586 GG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC[C@@H]2C[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667586 GG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H]3COC(=O)N[C@H]3C2)ccc1OC ZINC000880667595 ED On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CC[C@@H]3COC(=O)N[C@H]3C2)ccc1OC ZINC000880667595 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@H]3COC(=O)N[C@H]3C2)ccc1OC ZINC000880667595 ED On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild HTR1A 45 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild DRD2 39 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild TSHR 66 32 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild DRD4 28 42 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild ADRA1D 44 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild HTR1D 17 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild HTR1B 20 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild ADRA1A 35 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild ADRA1B 34 45 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild DRD3 42 38 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild NPY1R 27 44 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild EPHX2 43 39 COCc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)ccc1OC ZINC000880667596 GH On-Demand Mild QRFPR 43 39 COCc1cc(NC(=O)N2C[C@H]3[C@@H](C2)[C@@H]3C(=O)OC)ccc1OC ZINC000880667597 ED On-Demand Anodyne TSHR 69 35 COCc1cc(NC(=O)N2C[C@H]3[C@@H](C2)[C@@H]3C(=O)OC)ccc1OC ZINC000880667597 ED On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2C[C@H]3[C@@H](C2)[C@@H]3C(=O)OC)ccc1OC ZINC000880667597 ED On-Demand Anodyne ENPP1 72 35 COCc1cc(NC(=O)NOCC2CCC2)ccc1OC ZINC000880667600 CF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NOCC2CCC2)ccc1OC ZINC000880667600 CF On-Demand Anodyne PDE4A 23 41 COCc1cc(NC(=O)NOCC2CCC2)ccc1OC ZINC000880667600 CF On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)NOCC2CCC2)ccc1OC ZINC000880667600 CF On-Demand Anodyne ENPP1 49 31 COCc1cc(NC(=O)N[C@@H](C)c2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880667607 GG On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N[C@@H](C)c2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880667607 GG On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)N[C@H](C)c2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880667608 GG On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N[C@H](C)c2ccc(N3CCNC3=O)cc2)ccc1OC ZINC000880667608 GG On-Demand Anodyne ENPP1 61 32 COCc1cc(NC(=O)N2CCC[C@](C)(F)C2)ccc1OC ZINC000880667615 DG On-Demand Anodyne EPHX2 35 42 COCc1cc(NC(=O)N2CCC[C@](C)(F)C2)ccc1OC ZINC000880667615 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC[C@@](C)(F)C2)ccc1OC ZINC000880667616 DG On-Demand Anodyne EPHX2 35 42 COCc1cc(NC(=O)N2CCC[C@@](C)(F)C2)ccc1OC ZINC000880667616 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCN(C3CC3)[C@@H](C#N)C2)ccc1OC ZINC000880667617 EE On-Demand Mild TSHR 40 30 COCc1cc(NC(=O)N2CCN(C3CC3)[C@@H](C#N)C2)ccc1OC ZINC000880667617 EE On-Demand Mild QRFPR 42 36 COCc1cc(NC(=O)N2CCN(C3CC3)[C@H](C#N)C2)ccc1OC ZINC000880667618 EE On-Demand Mild TSHR 40 30 COCc1cc(NC(=O)N2CCN(C3CC3)[C@H](C#N)C2)ccc1OC ZINC000880667618 EE On-Demand Mild QRFPR 42 36 COCc1cc(NC(=O)N2CC3(CC3)C2)ccc1OC ZINC000880667625 CE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CC3(CC3)C2)ccc1OC ZINC000880667625 CE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CC3(CC3)C2)ccc1OC ZINC000880667625 CE On-Demand Anodyne ENPP1 73 38 COCc1cc(NC(=O)N2CCc3c(nnn3-c3ccccc3)C2)ccc1OC ZINC000880667626 GG On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CCc3c(nnn3-c3ccccc3)C2)ccc1OC ZINC000880667626 GG On-Demand Anodyne ENPP1 40 35 COCc1cc(NC(=O)NCC(=O)N(C)OC)ccc1OC ZINC000880667631 DC On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NCC(=O)N(C)OC)ccc1OC ZINC000880667631 DC On-Demand Anodyne ENPP1 62 31 COCc1cc(NC(=O)NCCN(C)C(=O)OC)ccc1OC ZINC000880667632 ED On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NCCN(C)C(=O)OC)ccc1OC ZINC000880667632 ED On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCC(OC(=O)N(C)C)CC2)ccc1OC ZINC000880667634 FF On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)N2CCC(OC(=O)N(C)C)CC2)ccc1OC ZINC000880667634 FF On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC(OC(=O)N(C)C)CC2)ccc1OC ZINC000880667634 FF On-Demand Anodyne HTR1B 18 43 COCc1cc(NC(=O)N2CCC(OC(=O)N(C)C)CC2)ccc1OC ZINC000880667634 FF On-Demand Anodyne PDGFRB 41 38 COCc1cc(NC(=O)N2CCC(OC(=O)N(C)C)CC2)ccc1OC ZINC000880667634 FF On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667635 GF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667635 GF On-Demand Anodyne HTR1B 17 40 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667635 GF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667635 GF On-Demand Anodyne PDE4A 15 45 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667636 GF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667636 GF On-Demand Anodyne HTR1B 17 40 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667636 GF On-Demand Anodyne PDGFRB 42 35 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)ccc1OC ZINC000880667636 GF On-Demand Anodyne PDE4A 15 45 COCc1cc(NC(=O)N2CC[C@H](N3CCOC3=O)C2)ccc1OC ZINC000880667637 ED On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CC[C@H](N3CCOC3=O)C2)ccc1OC ZINC000880667637 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@H](N3CCOC3=O)C2)ccc1OC ZINC000880667638 ED On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CC[C@@H](N3CCOC3=O)C2)ccc1OC ZINC000880667638 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCc2ccccc2CC(=O)OC)ccc1OC ZINC000880667643 FF On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)NCc2ccccc2CC(=O)OC)ccc1OC ZINC000880667643 FF On-Demand Anodyne ROCK2 17 48 COCc1cc(NC(=O)NCc2ccccc2CC(=O)OC)ccc1OC ZINC000880667643 FF On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)N[C@H](C)[C@@H](O)c2ccc(C)cc2)ccc1OC ZINC000880667645 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@@H](C)[C@@H](O)c2ccc(C)cc2)ccc1OC ZINC000880667646 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@H](C)[C@H](O)c2ccc(C)cc2)ccc1OC ZINC000880667647 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccc(C)cc2)ccc1OC ZINC000880667648 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2CCC[C@H](N3CCCCC3=O)C2)ccc1OC ZINC000880667649 GF On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)N2CCC[C@H](N3CCCCC3=O)C2)ccc1OC ZINC000880667649 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@@H](N3CCCCC3=O)C2)ccc1OC ZINC000880667650 GF On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)N2CCC[C@@H](N3CCCCC3=O)C2)ccc1OC ZINC000880667650 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC=C(Cl)C2)ccc1OC ZINC000880667651 DG On-Demand Anodyne QRFPR 45 39 COCc1cc(NC(=O)N2CCC=C(Cl)C2)ccc1OC ZINC000880667651 DG On-Demand Anodyne ENPP1 40 33 COCc1cc(NC(=O)NN(C)C2CC2)ccc1OC ZINC000880667662 CD On-Demand Reactive TSHR 59 32 COCc1cc(NC(=O)NN(C)C2CC2)ccc1OC ZINC000880667662 CD On-Demand Reactive QRFPR 47 39 COCc1cc(NC(=O)NN(C)C2CC2)ccc1OC ZINC000880667662 CD On-Demand Reactive ENPP1 45 30 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne HTR1B 18 43 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne PDGFRB 42 36 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne PDE4A 19 49 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)ccc1OC ZINC000880667663 FH On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne TSHR 66 33 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne HTR1B 18 43 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne PDGFRB 42 36 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne PDE4A 19 49 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)ccc1OC ZINC000880667664 FH On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N[C@@H]2[C@@H]3C[C@H]4[C@H](CO[C@H]42)C3)ccc1OC ZINC000880667667 EE On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)N[C@@H]2[C@@H]3C[C@@H]4[C@@H]2OC[C@@H]4C3)ccc1OC ZINC000880667668 EE On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)N[C@@H]2[C@H]3C[C@@H]4CO[C@@H]2[C@H]4C3)ccc1OC ZINC000880667669 EE On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)N[C@@H]2[C@H]3C[C@@H]4CO[C@H]2[C@H]4C3)ccc1OC ZINC000880667670 EE On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)NC[C@@]2(C)C[C@@H]2Br)ccc1OC ZINC000880667676 FG On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NC[C@@]2(C)C[C@@H]2Br)ccc1OC ZINC000880667676 FG On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NC[C@]2(C)C[C@H]2Br)ccc1OC ZINC000880667677 FG On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NC[C@]2(C)C[C@H]2Br)ccc1OC ZINC000880667677 FG On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NC[C@@]2(C)C[C@H]2Br)ccc1OC ZINC000880667678 FG On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NC[C@@]2(C)C[C@H]2Br)ccc1OC ZINC000880667678 FG On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NC[C@]2(C)C[C@@H]2Br)ccc1OC ZINC000880667679 FG On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NC[C@]2(C)C[C@@H]2Br)ccc1OC ZINC000880667679 FG On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NC2CC(C(=O)OC)C2)ccc1OC ZINC000880667682 DD On-Demand Anodyne TSHR 69 33 COCc1cc(NC(=O)NC2CC(C(=O)OC)C2)ccc1OC ZINC000880667682 DD On-Demand Anodyne EPHX2 40 36 COCc1cc(NC(=O)NC2CC(C(=O)OC)C2)ccc1OC ZINC000880667682 DD On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC2CC(C(=O)OC)C2)ccc1OC ZINC000880667682 DD On-Demand Anodyne ENPP1 54 31 COCc1cc(NC(=O)N2CCC[C@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667683 FF On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)N2CCC[C@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667683 FF On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC[C@@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667684 FF On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)N2CCC[C@@H](OC(=O)N(C)C)C2)ccc1OC ZINC000880667684 FF On-Demand Anodyne QRFPR 44 37 CCN(CCNC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667685 GG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NN2CCCNC2=O)ccc1OC ZINC000880667686 DD On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NN2CCCNC2=O)ccc1OC ZINC000880667686 DD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NN2CCCNC2=O)ccc1OC ZINC000880667686 DD On-Demand Anodyne ENPP1 58 33 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)C1CCCC1 ZINC000880667688 DG On-Demand Mild TSHR 47 31 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)C1CCCC1 ZINC000880667688 DG On-Demand Mild PDE4A 26 41 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)C1CCCC1 ZINC000880667688 DG On-Demand Mild QRFPR 51 42 COCc1cc(NC(=O)N[C@@H]2CC[C@H]3SCCS[C@@H]23)ccc1OC ZINC000880667691 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2CC[C@H]3SCCS[C@@H]23)ccc1OC ZINC000880667691 FG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@@H]2CC[C@H]3SCCS[C@H]23)ccc1OC ZINC000880667692 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2CC[C@H]3SCCS[C@H]23)ccc1OC ZINC000880667692 FG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@@H]2CC[C@@H]3SCCS[C@H]32)ccc1OC ZINC000880667693 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2CC[C@@H]3SCCS[C@H]32)ccc1OC ZINC000880667693 FG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@@H]2CC[C@@H]3SCCS[C@@H]32)ccc1OC ZINC000880667694 FG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N[C@@H]2CC[C@@H]3SCCS[C@@H]32)ccc1OC ZINC000880667694 FG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N(CCS(C)(=O)=O)C2CC2)ccc1OC ZINC000880667701 FD On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N2CC[C@H](N(C)C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667702 GG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CC[C@@H](N(C)C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667703 GG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NCCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667704 GE On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)NCCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667704 GE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667704 GE On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880667705 FG On-Demand Anodyne TSHR 70 34 COCc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880667705 FG On-Demand Anodyne PDGFRB 53 41 COCc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880667705 FG On-Demand Anodyne TACR1 17 41 COCc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880667705 FG On-Demand Anodyne EPHX2 27 42 COCc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880667705 FG On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)N2CC[C@@H]3NC(=O)OC[C@H]3C2)ccc1OC ZINC000880667706 ED On-Demand Anodyne TSHR 59 31 COCc1cc(NC(=O)N2CC[C@@H]3NC(=O)OC[C@H]3C2)ccc1OC ZINC000880667706 ED On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CC[C@@H]3NC(=O)OC[C@H]3C2)ccc1OC ZINC000880667706 ED On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)N[C@@](C)(CO)C2CC2)ccc1OC ZINC000880667713 DE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N[C@@](C)(CO)C2CC2)ccc1OC ZINC000880667713 DE On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@](C)(CO)C2CC2)ccc1OC ZINC000880667714 DE On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N[C@](C)(CO)C2CC2)ccc1OC ZINC000880667714 DE On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)NC[C@H](O)c2cc3ccccc3s2)ccc1OC ZINC000880667720 GH On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)NC[C@@H](O)c2cc3ccccc3s2)ccc1OC ZINC000880667721 GH On-Demand Anodyne TSHR 55 33 COCc1cc(NC(=O)N[C@H]2CCCc3[nH]ccc32)ccc1OC ZINC000880667722 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H]2CCCc3[nH]ccc32)ccc1OC ZINC000880667723 EG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NNC(=O)C2CC2)ccc1OC ZINC000880667724 CD On-Demand Reactive TSHR 60 32 COCc1cc(NC(=O)NNC(=O)C2CC2)ccc1OC ZINC000880667724 CD On-Demand Reactive HTR1B 16 42 COCc1cc(NC(=O)NNC(=O)C2CC2)ccc1OC ZINC000880667724 CD On-Demand Reactive QRFPR 49 40 COCc1cc(NC(=O)NNC(=O)C2CC2)ccc1OC ZINC000880667724 CD On-Demand Reactive ENPP1 55 31 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667725 GH On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667725 GH On-Demand Anodyne HTR2A 16 43 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667725 GH On-Demand Anodyne RAF1 22 40 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667725 GH On-Demand Anodyne PPARD 28 45 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667725 GH On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667726 GH On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667726 GH On-Demand Anodyne HTR2A 16 43 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667726 GH On-Demand Anodyne RAF1 22 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667726 GH On-Demand Anodyne PPARD 28 45 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C(F)(F)F)cc2)ccc1OC ZINC000880667726 GH On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880667728 FE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880667728 FE On-Demand Anodyne CCR3 17 41 COCc1cc(NC(=O)NC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880667728 FE On-Demand Anodyne EPHX2 64 52 COCc1cc(NC(=O)NC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880667728 FE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880667728 FE On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne TSHR 82 42 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne F10 19 40 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne NPY1R 32 42 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne CCKAR 42 41 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne CCKBR 48 41 COCc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667732 GG On-Demand Anodyne QRFPR 42 38 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne TSHR 82 42 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne F10 19 40 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne NPY1R 32 42 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne CCKAR 42 41 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne CCKBR 48 41 COCc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667733 GG On-Demand Anodyne QRFPR 42 38 COCc1cc(NC(=O)NCCn2c(C)nnc2S)ccc1OC ZINC000880667737 FD On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NCCn2c(C)nnc2S)ccc1OC ZINC000880667737 FD On-Demand Anodyne ENPP1 68 33 COCCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667740 CD On-Demand Anodyne TSHR 41 31 COCCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667740 CD On-Demand Anodyne QRFPR 41 34 COCCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667740 CD On-Demand Anodyne ENPP1 66 32 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne HTR1D 18 45 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne HTR1B 21 45 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne EPHX2 24 40 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CC[C@@H](OC)C2)ccc1OC ZINC000880667744 CE On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667746 GF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667746 GF On-Demand Anodyne CACNA1I 44 32 COCc1cc(NC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667746 GF On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCC([C@@H](O)c3nccn3C)CC2)ccc1OC ZINC000880667748 GF On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2CCC([C@@H](O)c3nccn3C)CC2)ccc1OC ZINC000880667748 GF On-Demand Anodyne ENPP1 51 33 COCc1cc(NC(=O)N2CCC([C@H](O)c3nccn3C)CC2)ccc1OC ZINC000880667749 GF On-Demand Anodyne PDGFRB 44 36 COCc1cc(NC(=O)N2CCC([C@H](O)c3nccn3C)CC2)ccc1OC ZINC000880667749 GF On-Demand Anodyne ENPP1 51 33 COCc1cc(NC(=O)N2CCn3c(C(C)C)nnc3[C@H]2C)ccc1OC ZINC000880667750 FG On-Demand Anodyne ENPP1 42 35 COCc1cc(NC(=O)N2CCn3c(C(C)C)nnc3[C@@H]2C)ccc1OC ZINC000880667751 FG On-Demand Anodyne ENPP1 42 35 COCc1cc(NC(=O)NCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667752 FE On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667752 FE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667752 FE On-Demand Anodyne PRMT3 45 33 COCc1cc(NC(=O)NCc2nnc(S)n2C2CC2)ccc1OC ZINC000880667752 FE On-Demand Anodyne ENPP1 60 30 COCc1cc(NC(=O)NNC(=O)CN(C)C)ccc1OC ZINC000880667755 DC On-Demand Reactive QRFPR 41 33 COCc1cc(NC(=O)NNC(=O)CN(C)C)ccc1OC ZINC000880667755 DC On-Demand Reactive ENPP1 64 34 COCc1cc(NC(=O)NNC(=O)OC(C)(C)C)ccc1OC ZINC000880667756 EE On-Demand Reactive TSHR 47 31 COCc1cc(NC(=O)NNC(=O)OC(C)(C)C)ccc1OC ZINC000880667756 EE On-Demand Reactive QRFPR 43 35 COCc1cc(NC(=O)NNC(=O)OC(C)(C)C)ccc1OC ZINC000880667756 EE On-Demand Reactive ENPP1 55 31 COCc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccc1OC ZINC000880667757 GG On-Demand Anodyne PDGFRB 74 45 COCc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccc1OC ZINC000880667757 GG On-Demand Anodyne TRPV1 15 46 COCc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccc1OC ZINC000880667757 GG On-Demand Anodyne PDGFRA 15 43 COCc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)ccc1OC ZINC000880667757 GG On-Demand Anodyne RBP4 20 54 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)c(C)c2)ccc1OC ZINC000880667758 GF On-Demand Reactive TSHR 60 35 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)c(C)c2)ccc1OC ZINC000880667758 GF On-Demand Reactive ENPP1 58 35 COCc1cc(NC(=O)NCCc2cnccn2)ccc1OC ZINC000880667759 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NCCc2cnccn2)ccc1OC ZINC000880667759 DD On-Demand Anodyne QPCT 16 45 COCc1cc(NC(=O)NCCc2cnccn2)ccc1OC ZINC000880667759 DD On-Demand Anodyne ENPP1 50 37 COCc1cc(NC(=O)N2CCC(C)=C(Br)C2)ccc1OC ZINC000880667762 FH On-Demand Anodyne P2RY14 41 31 COCc1cc(NC(=O)N2CCC(C)=C(Br)C2)ccc1OC ZINC000880667762 FH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NNC(=O)[C@H]2OCC[C@H]2c2ccccc2)ccc1OC ZINC000880667763 GF On-Demand Reactive TSHR 70 34 COCc1cc(NC(=O)NNC(=O)[C@H]2OCC[C@H]2c2ccccc2)ccc1OC ZINC000880667763 GF On-Demand Reactive QRFPR 43 39 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)[C@H]1CCS(=O)(=O)C1 ZINC000880667764 FD On-Demand Mild QRFPR 42 34 C#CCN(C(=O)Nc1ccc(OC)c(COC)c1)[C@@H]1CCS(=O)(=O)C1 ZINC000880667765 FD On-Demand Mild QRFPR 42 34 COCc1cc(NC(=O)N2CC[C@H](NC(=O)OC(C)(C)C)[C@H]2C)ccc1OC ZINC000880667766 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@H](NC(=O)OC(C)(C)C)[C@H]2C)ccc1OC ZINC000880667767 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@H](NC(=O)OC(C)(C)C)[C@@H]2C)ccc1OC ZINC000880667768 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCN(C3=NCC(C)(C)S3)CC2)ccc1OC ZINC000880667769 GF On-Demand Anodyne PDGFRB 61 41 COCc1cc(NC(=O)NC[C@](C)(O)c2ccc(F)cc2)ccc1OC ZINC000880667770 FG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)NC[C@](C)(O)c2ccc(F)cc2)ccc1OC ZINC000880667770 FG On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccc(F)cc2)ccc1OC ZINC000880667771 FG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccc(F)cc2)ccc1OC ZINC000880667771 FG On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667772 GH On-Demand Anodyne HTR2A 15 43 COCc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667772 GH On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667773 GH On-Demand Anodyne HTR2A 15 43 COCc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667773 GH On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N[C@@H](C)C[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667774 GH On-Demand Anodyne HTR2A 15 43 COCc1cc(NC(=O)N[C@@H](C)C[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667774 GH On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N[C@@H](C)C[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667775 GH On-Demand Anodyne HTR2A 15 43 COCc1cc(NC(=O)N[C@@H](C)C[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880667775 GH On-Demand Anodyne ENPP1 60 31 COCc1cc(NC(=O)N2C[C@H](C)[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667776 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667777 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@@H](NC(=O)OC(C)(C)C)[C@H](C)C2)ccc1OC ZINC000880667778 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2C[C@H](C)[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667779 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCSCc2ccnc(Cl)c2)ccc1OC ZINC000880667780 GH On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)NCCSCc2ccnc(Cl)c2)ccc1OC ZINC000880667780 GH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCSCc2ccnc(Cl)c2)ccc1OC ZINC000880667780 GH On-Demand Anodyne ENPP1 46 33 O=C(NCc1ccc(OCC(F)(F)F)nn1)c1ccc(N2CCOCC2)nc1 ZINC000880667783 GD On-Demand Anodyne HPGDS 33 51 COCc1cc(NC(=O)NNC(=O)CC(C)C)ccc1OC ZINC000880667841 DE On-Demand Reactive TSHR 40 31 COCc1cc(NC(=O)NNC(=O)CC(C)C)ccc1OC ZINC000880667841 DE On-Demand Reactive QRFPR 41 34 COCc1cc(NC(=O)NNC(=O)CC(C)C)ccc1OC ZINC000880667841 DE On-Demand Reactive ENPP1 74 36 COCc1cc(NC(=O)N[C@H]2CCC2(C)C)ccc1OC ZINC000880667842 CG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@H]2CCC2(C)C)ccc1OC ZINC000880667842 CG On-Demand Anodyne QRFPR 47 40 COCc1cc(NC(=O)N[C@@H]2CCC2(C)C)ccc1OC ZINC000880667843 CG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@@H]2CCC2(C)C)ccc1OC ZINC000880667843 CG On-Demand Anodyne QRFPR 47 40 COCc1cc(NC(=O)N[C@@H](C)C[C@@H](O)c2ccccc2)ccc1OC ZINC000880667844 FG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@@H](C)C[C@@H](O)c2ccccc2)ccc1OC ZINC000880667844 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccccc2)ccc1OC ZINC000880667845 FG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccccc2)ccc1OC ZINC000880667845 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@@H](C)C[C@H](O)c2ccccc2)ccc1OC ZINC000880667846 FG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@@H](C)C[C@H](O)c2ccccc2)ccc1OC ZINC000880667846 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccccc2)ccc1OC ZINC000880667847 FG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccccc2)ccc1OC ZINC000880667847 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NC[C@H]2COC3(CCOCC3)O2)ccc1OC ZINC000880667848 FD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@@H]2COC3(CCOCC3)O2)ccc1OC ZINC000880667849 FD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C)c2)ccc1OC ZINC000880667851 EG On-Demand Anodyne TSHR 69 35 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C)c2)ccc1OC ZINC000880667851 EG On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C)c2)ccc1OC ZINC000880667851 EG On-Demand Anodyne KCNK3 49 36 COCc1cc(NC(=O)NC[C@H](O)c2cccc(C)c2)ccc1OC ZINC000880667851 EG On-Demand Anodyne KCNK9 48 36 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C)c2)ccc1OC ZINC000880667852 EG On-Demand Anodyne TSHR 69 35 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C)c2)ccc1OC ZINC000880667852 EG On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C)c2)ccc1OC ZINC000880667852 EG On-Demand Anodyne KCNK3 49 36 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(C)c2)ccc1OC ZINC000880667852 EG On-Demand Anodyne KCNK9 48 36 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne HTR1D 15 49 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne HTR1B 17 42 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne PDGFRB 44 40 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne EPHX2 15 44 COCc1cc(NC(=O)N2CCC(CCCO)CC2)ccc1OC ZINC000880667854 EF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667855 GF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CC[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880667856 GF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCOCC[C@H]2C)ccc1OC ZINC000880667857 DE On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CCOCC[C@H]2C)ccc1OC ZINC000880667857 DE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCOCC[C@H]2C)ccc1OC ZINC000880667857 DE On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N2CCOCC[C@@H]2C)ccc1OC ZINC000880667858 DE On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CCOCC[C@@H]2C)ccc1OC ZINC000880667858 DE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCOCC[C@@H]2C)ccc1OC ZINC000880667858 DE On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)N2CC(O)(c3ccccc3)C2)ccc1OC ZINC000880667861 EF On-Demand Anodyne TSHR 69 35 COCc1cc(NC(=O)N2CC(O)(c3ccccc3)C2)ccc1OC ZINC000880667861 EF On-Demand Anodyne QRFPR 41 38 COCc1cc(NC(=O)N2CC(O)(c3ccccc3)C2)ccc1OC ZINC000880667861 EF On-Demand Anodyne ENPP1 41 33 COCc1cc(NC(=O)NCc2cc(C)cc(Cl)n2)ccc1OC ZINC000880667864 EH On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NCc2cc(C)cc(Cl)n2)ccc1OC ZINC000880667864 EH On-Demand Anodyne ENPP1 61 34 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne TSHR 49 35 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne PTAFR 24 40 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne CHRNA7 30 42 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne ROCK2 22 41 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne ENPP1 70 37 COCc1cc(NC(=O)NOCc2cccnc2)ccc1OC ZINC000880667865 DE On-Demand Anodyne NAMPT 41 41 O=C(CCCn1ccnc1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667866 ED On-Demand Anodyne TBXAS1 49 45 O=C(CCCn1ccnc1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880667866 ED On-Demand Anodyne QPCT 36 41 COCc1cc(NC(=O)NNC(=O)COCc2ccccc2)ccc1OC ZINC000880667867 FE On-Demand Reactive TSHR 74 38 COCc1cc(NC(=O)NNC(=O)COCc2ccccc2)ccc1OC ZINC000880667867 FE On-Demand Reactive QRFPR 40 37 COCc1cc(NC(=O)NNC(=O)COCc2ccccc2)ccc1OC ZINC000880667867 FE On-Demand Reactive ENPP1 67 32 COCc1cc(NC(=O)NNc2ccc(C(F)(F)F)cn2)ccc1OC ZINC000880667870 FG On-Demand Reactive HTR2A 24 43 COCc1cc(NC(=O)NNc2ccc(C(F)(F)F)cn2)ccc1OC ZINC000880667870 FG On-Demand Reactive ENPP1 46 32 COCc1cc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)ccc1OC ZINC000880667874 GG On-Demand Anodyne TSHR 57 33 COCc1cc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)ccc1OC ZINC000880667874 GG On-Demand Anodyne PDGFRB 55 38 COCc1cc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)ccc1OC ZINC000880667874 GG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H](CCO)Cc2ccccc2)ccc1OC ZINC000880667879 FF On-Demand Anodyne TSHR 70 36 COCc1cc(NC(=O)N[C@@H](CCO)Cc2ccccc2)ccc1OC ZINC000880667880 FF On-Demand Anodyne TSHR 70 36 COCc1cc(NC(=O)NNC(C)=O)ccc1OC ZINC000880667882 CD On-Demand Reactive TSHR 72 37 COCc1cc(NC(=O)NNC(C)=O)ccc1OC ZINC000880667882 CD On-Demand Reactive MTNR1B 25 42 COCc1cc(NC(=O)NNC(C)=O)ccc1OC ZINC000880667882 CD On-Demand Reactive QRFPR 47 38 COCc1cc(NC(=O)NNC(C)=O)ccc1OC ZINC000880667882 CD On-Demand Reactive ENPP1 69 34 COCc1cc(NC(=O)NNC(=O)[C@@H](C)Oc2ccccc2F)ccc1OC ZINC000880667883 GF On-Demand Reactive TSHR 55 34 COCc1cc(NC(=O)NNC(=O)[C@@H](C)Oc2ccccc2F)ccc1OC ZINC000880667883 GF On-Demand Reactive HTR2A 17 40 COCc1cc(NC(=O)NNC(=O)[C@H](C)Oc2ccccc2F)ccc1OC ZINC000880667884 GF On-Demand Reactive TSHR 55 34 COCc1cc(NC(=O)NNC(=O)[C@H](C)Oc2ccccc2F)ccc1OC ZINC000880667884 GF On-Demand Reactive HTR2A 17 40 COCc1cc(NC(=O)NCc2nnc(S)n2C(C)C)ccc1OC ZINC000880667885 FF On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NCc2nnc(S)n2C(C)C)ccc1OC ZINC000880667885 FF On-Demand Anodyne ENPP1 62 32 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne HTR1D 17 45 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne HTR1B 20 45 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne PDGFRB 43 37 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N2CCC(OC(C)=O)CC2)ccc1OC ZINC000880667887 EE On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)NCC[C@](C)(O)c2ccccc2)ccc1OC ZINC000880667889 FG On-Demand Anodyne TSHR 69 33 COCc1cc(NC(=O)NCC[C@@](C)(O)c2ccccc2)ccc1OC ZINC000880667890 FG On-Demand Anodyne TSHR 69 33 COCc1cc(NC(=O)NOCC(C)C)ccc1OC ZINC000880667892 CF On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)NOCC(C)C)ccc1OC ZINC000880667892 CF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NOCC(C)C)ccc1OC ZINC000880667892 CF On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NNC(=O)[C@@H]2Cc3ccccc3O2)ccc1OC ZINC000880667893 FD On-Demand Reactive TSHR 59 31 COCc1cc(NC(=O)NNC(=O)[C@@H]2Cc3ccccc3O2)ccc1OC ZINC000880667893 FD On-Demand Reactive QRFPR 41 35 COCc1cc(NC(=O)NNC(=O)[C@H]2Cc3ccccc3O2)ccc1OC ZINC000880667894 FD On-Demand Reactive TSHR 59 31 COCc1cc(NC(=O)NNC(=O)[C@H]2Cc3ccccc3O2)ccc1OC ZINC000880667894 FD On-Demand Reactive QRFPR 41 35 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2C)ccc1OC ZINC000880667895 FF On-Demand Reactive TSHR 64 35 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2C)ccc1OC ZINC000880667895 FF On-Demand Reactive QRFPR 41 35 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2C)ccc1OC ZINC000880667895 FF On-Demand Reactive ENPP1 62 34 COCc1cc(NC(=O)N(CC2CCOCC2)OC)ccc1OC ZINC000880667900 EF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N(CC2CCOCC2)OC)ccc1OC ZINC000880667900 EF On-Demand Anodyne QRFPR 43 36 O=C1CCCc2cc(C(=O)NCc3ccc(OCC(F)(F)F)nn3)ccc2N1 ZINC000880667902 GF On-Demand Anodyne HDAC9 18 40 COCc1cc(NC(=O)NC2CCC(O)(c3cccnc3)CC2)ccc1OC ZINC000880667903 GG On-Demand Anodyne CHRNA7 18 41 COCc1cc(NC(=O)NC2CCC(O)(c3cccnc3)CC2)ccc1OC ZINC000880667903 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NNC(=O)c2cc3c(s2)CCC3)ccc1OC ZINC000880667904 GF On-Demand Reactive QRFPR 44 38 COCc1cc(NC(=O)NOCCSC)ccc1OC ZINC000880667905 DE On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)NOCCSC)ccc1OC ZINC000880667905 DE On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)N[C@H]2CCCC3(C2)OCCO3)ccc1OC ZINC000880667911 FF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@H]2CCCC3(C2)OCCO3)ccc1OC ZINC000880667911 FF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@@H]2CCCC3(C2)OCCO3)ccc1OC ZINC000880667912 FF On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@@H]2CCCC3(C2)OCCO3)ccc1OC ZINC000880667912 FF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N(Cc2ccccc2)OC)ccc1OC ZINC000880667913 EG On-Demand Anodyne TSHR 75 38 COCc1cc(NC(=O)N(Cc2ccccc2)OC)ccc1OC ZINC000880667913 EG On-Demand Anodyne TSPO 44 36 COCc1cc(NC(=O)N(Cc2ccccc2)OC)ccc1OC ZINC000880667913 EG On-Demand Anodyne QRFPR 40 38 COCc1cc(NC(=O)N(Cc2ccccc2)OC)ccc1OC ZINC000880667913 EG On-Demand Anodyne ENPP1 44 31 CC[C@@H](C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880667915 FG On-Demand Reactive TSHR 67 33 CC[C@@H](C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880667915 FG On-Demand Reactive KCNQ2 40 41 CC[C@@H](C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880667915 FG On-Demand Reactive SOAT1 34 40 CC[C@@H](C(=O)NNC(=O)Nc1ccc(OC)c(COC)c1)c1ccccc1 ZINC000880667915 FG On-Demand Reactive ENPP1 40 31 COCc1cc(NC(=O)NNC(=O)Cc2ccsc2)ccc1OC ZINC000880667916 EE On-Demand Reactive QRFPR 43 42 COCc1cc(NC(=O)NNC(=O)Cc2ccsc2)ccc1OC ZINC000880667916 EE On-Demand Reactive ENPP1 56 32 COCc1cc(NC(=O)NNc2ncccc2C)ccc1OC ZINC000880667919 DF On-Demand Reactive TSHR 55 35 COCc1cc(NC(=O)NNc2ncccc2C)ccc1OC ZINC000880667919 DF On-Demand Reactive PPIA 39 40 COCc1cc(NC(=O)NNc2ncccc2C)ccc1OC ZINC000880667919 DF On-Demand Reactive GRM4 16 42 COCc1cc(NC(=O)NNc2ncccc2C)ccc1OC ZINC000880667919 DF On-Demand Reactive PDGFRA 41 37 COCc1cc(NC(=O)NNc2ncccc2C)ccc1OC ZINC000880667919 DF On-Demand Reactive ENPP1 54 39 COCc1cc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667924 FG On-Demand Anodyne HTR1D 15 46 COCc1cc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667924 FG On-Demand Anodyne HTR1B 15 46 COCc1cc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667924 FG On-Demand Anodyne PDGFRB 40 36 COCc1cc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667924 FG On-Demand Anodyne S1PR2 28 40 COCc1cc(NC(=O)N2CC[C@@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667924 FG On-Demand Anodyne EPHX2 29 41 COCc1cc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667925 FG On-Demand Anodyne HTR1D 15 46 COCc1cc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667925 FG On-Demand Anodyne HTR1B 15 46 COCc1cc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667925 FG On-Demand Anodyne PDGFRB 40 36 COCc1cc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667925 FG On-Demand Anodyne S1PR2 28 40 COCc1cc(NC(=O)N2CC[C@](O)(c3ccc(F)cc3)C2)ccc1OC ZINC000880667925 FG On-Demand Anodyne EPHX2 29 41 CCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667926 CD On-Demand Reactive TSHR 47 32 CCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667926 CD On-Demand Reactive QRFPR 42 35 CCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667926 CD On-Demand Reactive ENPP1 72 35 COCc1cc(NC(=O)NCC2(C)OCCO2)ccc1OC ZINC000880667929 DD On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NCC2(C)OCCO2)ccc1OC ZINC000880667929 DD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667930 GG On-Demand Anodyne TSHR 81 40 COCc1cc(NC(=O)N(C)[C@H]2CCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667930 GG On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667931 GG On-Demand Anodyne TSHR 81 40 COCc1cc(NC(=O)N(C)[C@@H]2CCN(Cc3ccccc3)C2=O)ccc1OC ZINC000880667931 GG On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)N2CCC[C@H](C3(C)OCCO3)C2)ccc1OC ZINC000880667932 FF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@H](C3(C)OCCO3)C2)ccc1OC ZINC000880667932 FF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@@H](C3(C)OCCO3)C2)ccc1OC ZINC000880667933 FF On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCC[C@@H](C3(C)OCCO3)C2)ccc1OC ZINC000880667933 FF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N(C)OCc2ccccc2)ccc1OC ZINC000880667934 EG On-Demand Anodyne TSHR 76 39 COCc1cc(NC(=O)N(C)OCc2ccccc2)ccc1OC ZINC000880667934 EG On-Demand Anodyne QRFPR 41 38 COCc1cc(NC(=O)N(C)OCc2ccccc2)ccc1OC ZINC000880667934 EG On-Demand Anodyne ENPP1 50 31 COCc1cc(NC(=O)NCCc2cnc(C)s2)ccc1OC ZINC000880667937 EF On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NCCc2cnc(C)s2)ccc1OC ZINC000880667937 EF On-Demand Anodyne PRMT3 51 32 COCc1cc(NC(=O)NCCc2cnc(C)s2)ccc1OC ZINC000880667937 EF On-Demand Anodyne ENPP1 51 32 CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667938 CD On-Demand Anodyne TSHR 54 32 CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667938 CD On-Demand Anodyne QRFPR 43 35 CCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667938 CD On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)N(C)Cc2ncc(Cl)n2C)ccc1OC ZINC000880667941 FF On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)N(C)Cc2ncc(Cl)n2C)ccc1OC ZINC000880667941 FF On-Demand Anodyne ENPP1 58 36 COCc1cc(NC(=O)NC[C@@H]2COC(C)(C)O2)ccc1OC ZINC000880667943 DE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)NC[C@@H]2COC(C)(C)O2)ccc1OC ZINC000880667943 DE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NC[C@H]2COC(C)(C)O2)ccc1OC ZINC000880667944 DE On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)NC[C@H]2COC(C)(C)O2)ccc1OC ZINC000880667944 DE On-Demand Anodyne QRFPR 42 35 C#C[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@H]1CCCO1 ZINC000880667949 DE On-Demand Mild QRFPR 45 39 C#C[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@H]1CCCO1 ZINC000880667950 DE On-Demand Mild QRFPR 45 39 C#C[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@@H]1CCCO1 ZINC000880667951 DE On-Demand Mild QRFPR 45 39 C#C[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)[C@@H]1CCCO1 ZINC000880667952 DE On-Demand Mild QRFPR 45 39 COCc1cc(NC(=O)NC23CCC(CC2)C3)ccc1OC ZINC000880667953 DG On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NC23CCC(CC2)C3)ccc1OC ZINC000880667953 DG On-Demand Anodyne EPHX2 66 47 COCc1cc(NC(=O)NC23CCC(CC2)C3)ccc1OC ZINC000880667953 DG On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)NNC(=O)[C@@H](C)Oc2ccc(F)cc2)ccc1OC ZINC000880667955 GF On-Demand Reactive TSHR 57 33 COCc1cc(NC(=O)NNC(=O)[C@@H](C)Oc2ccc(F)cc2)ccc1OC ZINC000880667955 GF On-Demand Reactive HTR2A 19 44 COCc1cc(NC(=O)NNC(=O)[C@H](C)Oc2ccc(F)cc2)ccc1OC ZINC000880667956 GF On-Demand Reactive TSHR 57 33 COCc1cc(NC(=O)NNC(=O)[C@H](C)Oc2ccc(F)cc2)ccc1OC ZINC000880667956 GF On-Demand Reactive HTR2A 19 44 COCc1cc(NC(=O)N2CC[C@@H]2Cc2ccccc2)ccc1OC ZINC000880667959 EH On-Demand Anodyne TSHR 78 39 COCc1cc(NC(=O)N2CC[C@@H]2Cc2ccccc2)ccc1OC ZINC000880667959 EH On-Demand Anodyne TACR1 21 41 COCc1cc(NC(=O)N2CC[C@@H]2Cc2ccccc2)ccc1OC ZINC000880667959 EH On-Demand Anodyne CCR3 30 41 COCc1cc(NC(=O)N2CC[C@@H]2Cc2ccccc2)ccc1OC ZINC000880667959 EH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CC[C@@H]2Cc2ccccc2)ccc1OC ZINC000880667959 EH On-Demand Anodyne ENPP1 61 33 COCc1cc(NC(=O)N2CC[C@H]2Cc2ccccc2)ccc1OC ZINC000880667960 EH On-Demand Anodyne TSHR 78 39 COCc1cc(NC(=O)N2CC[C@H]2Cc2ccccc2)ccc1OC ZINC000880667960 EH On-Demand Anodyne TACR1 21 41 COCc1cc(NC(=O)N2CC[C@H]2Cc2ccccc2)ccc1OC ZINC000880667960 EH On-Demand Anodyne CCR3 30 41 COCc1cc(NC(=O)N2CC[C@H]2Cc2ccccc2)ccc1OC ZINC000880667960 EH On-Demand Anodyne QRFPR 44 40 COCc1cc(NC(=O)N2CC[C@H]2Cc2ccccc2)ccc1OC ZINC000880667960 EH On-Demand Anodyne ENPP1 61 33 O=C(NCc1ccc(OCC(F)(F)F)nn1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880667965 GD On-Demand Anodyne INHA 20 44 O=C(NCc1ccc(OCC(F)(F)F)nn1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880667966 GD On-Demand Anodyne INHA 20 44 COCc1cc(NC(=O)NCCn2cc(Br)cn2)ccc1OC ZINC000880667969 GF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NCCn2cc(Br)cn2)ccc1OC ZINC000880667969 GF On-Demand Anodyne HTR2A 35 44 COCc1cc(NC(=O)NCCn2cc(Br)cn2)ccc1OC ZINC000880667969 GF On-Demand Anodyne ENPP1 57 36 COCc1cc(NC(=O)NCc2ccc(N3CCOC3=O)cc2)ccc1OC ZINC000880667979 GG On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NOC2CCOCC2)ccc1OC ZINC000880667980 DE On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NOC2CCOCC2)ccc1OC ZINC000880667980 DE On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)NOC2CCOCC2)ccc1OC ZINC000880667980 DE On-Demand Anodyne ENPP1 44 31 COCc1cc(NC(=O)Nc2ccccc2O[C@H](C)C#N)ccc1OC ZINC000880667983 FH On-Demand Mild TSHR 47 32 COCc1cc(NC(=O)Nc2ccccc2O[C@@H](C)C#N)ccc1OC ZINC000880667984 FH On-Demand Mild TSHR 47 32 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne TSHR 66 35 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne HTR1D 16 44 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne HTR1B 18 44 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne PDGFRB 55 40 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne PDE4A 18 42 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne GRM4 24 44 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne EPHX2 21 40 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne QRFPR 44 39 COCc1cc(NC(=O)N2CC[C@H](c3ccccn3)C2)ccc1OC ZINC000880667985 EG On-Demand Anodyne ENPP1 53 38 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne TSHR 66 35 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne HTR1D 16 44 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne HTR1B 18 44 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne PDGFRB 55 40 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne PDE4A 18 42 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne GRM4 24 44 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne EPHX2 21 40 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne QRFPR 44 39 COCc1cc(NC(=O)N2CC[C@@H](c3ccccn3)C2)ccc1OC ZINC000880667986 EG On-Demand Anodyne ENPP1 53 38 COCc1cc(NC(=O)NCCS(=O)(=O)CC2CC2)ccc1OC ZINC000880667987 FD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC/C=C\CNC(=O)OC(C)(C)C)ccc1OC ZINC000880667991 GG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NC/C=C/CNC(=O)OC(C)(C)C)ccc1OC ZINC000880667992 GG On-Demand Anodyne TSHR 68 33 COCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667995 CC On-Demand Reactive TSHR 54 32 COCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667995 CC On-Demand Reactive QRFPR 44 37 COCC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880667995 CC On-Demand Reactive ENPP1 72 35 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2cccs2)ccc1OC ZINC000880667998 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2cccs2)ccc1OC ZINC000880667998 GI On-Demand Anodyne QRFPR 44 41 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2cccs2)ccc1OC ZINC000880667999 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2cccs2)ccc1OC ZINC000880667999 GI On-Demand Anodyne QRFPR 44 41 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2cccs2)ccc1OC ZINC000880668000 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2cccs2)ccc1OC ZINC000880668000 GI On-Demand Anodyne QRFPR 44 41 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2cccs2)ccc1OC ZINC000880668001 GI On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2cccs2)ccc1OC ZINC000880668001 GI On-Demand Anodyne QRFPR 44 41 COCc1cc(NC(=O)NOC[C@@H]2CCOC2)ccc1OC ZINC000880668002 DD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NOC[C@H]2CCOC2)ccc1OC ZINC000880668003 DD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N[C@H](C)c2ccc[nH]2)ccc1OC ZINC000880668006 DG On-Demand Anodyne TSHR 57 33 COCc1cc(NC(=O)N[C@H](C)c2ccc[nH]2)ccc1OC ZINC000880668006 DG On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N[C@H](C)c2ccc[nH]2)ccc1OC ZINC000880668006 DG On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N[C@@H](C)c2ccc[nH]2)ccc1OC ZINC000880668007 DG On-Demand Anodyne TSHR 57 33 COCc1cc(NC(=O)N[C@@H](C)c2ccc[nH]2)ccc1OC ZINC000880668007 DG On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N[C@@H](C)c2ccc[nH]2)ccc1OC ZINC000880668007 DG On-Demand Anodyne ENPP1 62 33 CCc1nc2ccccc2n1CC(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668008 GF On-Demand Anodyne IMDH_CRYPV 31 41 CN1CCC(C(=O)NCc2ccc(OCC(F)(F)F)nn2)CC1 ZINC000880668009 ED On-Demand Anodyne EPHX2 19 42 COCc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)ccc1OC ZINC000880668010 FG On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)ccc1OC ZINC000880668010 FG On-Demand Anodyne PPARA 16 41 COCc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)ccc1OC ZINC000880668010 FG On-Demand Anodyne TRPV1 32 45 COCc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)ccc1OC ZINC000880668010 FG On-Demand Anodyne ROCK2 18 44 COCc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)ccc1OC ZINC000880668010 FG On-Demand Anodyne MT-ND1 24 40 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean HTR1A 15 56 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean TSHR 57 35 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean HTR1D 20 56 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean HTR1B 23 56 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean PDGFRB 66 44 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean RBP4 16 40 COCc1cc(NC(=O)N2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668014 GG On-Demand Clean ENPP1 62 33 COCc1cc(NC(=O)N2CCC(C3(C)OCCO3)CC2)ccc1OC ZINC000880668015 FF On-Demand Anodyne TSHR 60 31 COCc1cc(NC(=O)N2CCC(C3(C)OCCO3)CC2)ccc1OC ZINC000880668015 FF On-Demand Anodyne QRFPR 41 34 CCOC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668016 CD On-Demand Reactive TSHR 47 33 CCOC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668016 CD On-Demand Reactive QRFPR 42 34 CCOC(=O)NNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668016 CD On-Demand Reactive ENPP1 68 32 COCc1cc(NC(=O)NNC(=O)C(C)C)ccc1OC ZINC000880668019 CD On-Demand Reactive TSHR 47 32 COCc1cc(NC(=O)NNC(=O)C(C)C)ccc1OC ZINC000880668019 CD On-Demand Reactive HTR2A 20 40 COCc1cc(NC(=O)NNC(=O)C(C)C)ccc1OC ZINC000880668019 CD On-Demand Reactive QRFPR 46 37 COCc1cc(NC(=O)NNC(=O)C(C)C)ccc1OC ZINC000880668019 CD On-Demand Reactive ENPP1 62 33 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne HTR2A 42 50 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne HTR2C 15 50 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne NQO2 45 32 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne QPCT 18 47 COCc1cc(NC(=O)NCCc2ccnn2C)ccc1OC ZINC000880668020 DD On-Demand Anodyne ENPP1 57 32 COCc1cc(NC(=O)NNC(=O)CCCc2cccs2)ccc1OC ZINC000880668021 GG On-Demand Reactive PTPRF 20 44 COCc1cc(NC(=O)NC2COC(C)(C)OC2)ccc1OC ZINC000880668022 DE On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)NC2COC(C)(C)OC2)ccc1OC ZINC000880668022 DE On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N[C@H]2CCCc3cn(C(C)C)nc32)ccc1OC ZINC000880668023 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@@H]2CCCc3cn(C(C)C)nc32)ccc1OC ZINC000880668024 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC2CN(C(=O)OC)C2)ccc1OC ZINC000880668026 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC2CN(C(=O)OC)C2)ccc1OC ZINC000880668026 DD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC2CN(C(=O)OC)C2)ccc1OC ZINC000880668026 DD On-Demand Anodyne ENPP1 68 32 COCc1cc(NC(=O)N2CCCC[C@H]2COC(=O)NC(C)C)ccc1OC ZINC000880668027 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCCC[C@@H]2COC(=O)NC(C)C)ccc1OC ZINC000880668028 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCOC[C@H](C)C2)ccc1OC ZINC000880668029 DE On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCOC[C@H](C)C2)ccc1OC ZINC000880668029 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N2CCOC[C@@H](C)C2)ccc1OC ZINC000880668030 DE On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCOC[C@@H](C)C2)ccc1OC ZINC000880668030 DE On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)OC)ccc1OC ZINC000880668033 CD On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N(C)OC)ccc1OC ZINC000880668033 CD On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N(C)OC)ccc1OC ZINC000880668033 CD On-Demand Anodyne ENPP1 63 32 COCc1cc(NC(=O)NCCSC(C)(C)C)ccc1OC ZINC000880668034 EG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NCCSC(C)(C)C)ccc1OC ZINC000880668034 EG On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)NCCSC(C)(C)C)ccc1OC ZINC000880668034 EG On-Demand Anodyne ENPP1 56 31 CCCCCCC(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668037 DG On-Demand Anodyne SUCNR1 46 39 COCc1cc(NC(=O)N(CCO)Cc2cccnc2Cl)ccc1OC ZINC000880668038 GF On-Demand Anodyne GRM4 20 42 CCCCCCC(=O)N[C@@H](C)c1nc(C(=O)OCC)n[nH]1 ZINC000880668039 CE On-Demand Anodyne NOD1 89 40 CCCCCCC(=O)N[C@H](C)c1nc(C(=O)OCC)n[nH]1 ZINC000880668040 CE On-Demand Anodyne NOD1 89 40 COCc1cc(NC(=O)NC[C@H](O)C(F)(F)F)ccc1OC ZINC000880668043 DD On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)NC[C@H](O)C(F)(F)F)ccc1OC ZINC000880668043 DD On-Demand Anodyne PRMT3 62 36 COCc1cc(NC(=O)NOCCO)ccc1OC ZINC000880668044 CC On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NOCCO)ccc1OC ZINC000880668044 CC On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NOCCO)ccc1OC ZINC000880668044 CC On-Demand Anodyne ENPP1 67 33 COCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668045 CD On-Demand Anodyne TSHR 53 32 COCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668045 CD On-Demand Anodyne QRFPR 43 35 COCCONC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668045 CD On-Demand Anodyne ENPP1 69 34 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668047 GG On-Demand Anodyne TSHR 40 30 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668047 GG On-Demand Anodyne QRFPR 41 33 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668047 GG On-Demand Anodyne ENPP1 67 32 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668048 GG On-Demand Anodyne TSHR 40 30 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668048 GG On-Demand Anodyne QRFPR 41 33 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668048 GG On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)N2CC(O)(C(C)C)C2)ccc1OC ZINC000880668052 DE On-Demand Anodyne PDGFRB 41 38 COCc1cc(NC(=O)N2CC(O)(C(C)C)C2)ccc1OC ZINC000880668052 DE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC(O)(C(C)C)C2)ccc1OC ZINC000880668052 DE On-Demand Anodyne ENPP1 70 36 COCc1cc(NC(=O)NC2CC(OC)C2)ccc1OC ZINC000880668056 CE On-Demand Anodyne TSHR 64 34 COCc1cc(NC(=O)NC2CC(OC)C2)ccc1OC ZINC000880668056 CE On-Demand Anodyne EPHX2 41 38 COCc1cc(NC(=O)NC2CC(OC)C2)ccc1OC ZINC000880668056 CE On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NC2CC(OC)C2)ccc1OC ZINC000880668056 CE On-Demand Anodyne ENPP1 44 30 COCc1cc(NC(=O)N2CCC3(CC2)COC(=O)N3)ccc1OC ZINC000880668057 ED On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CCC3(CC2)COC(=O)N3)ccc1OC ZINC000880668057 ED On-Demand Anodyne ENPP1 56 32 COCc1cc(NC(=O)NOCCC(F)(F)F)ccc1OC ZINC000880668059 DF On-Demand Anodyne ENPP1 54 31 COCc1cc(NC(=O)NNc2nc(C)cc(C)n2)ccc1OC ZINC000880668060 EE On-Demand Reactive ENPP1 75 37 COCc1cc(NC(=O)NNC(=O)c2cccc(N(C)C)c2)ccc1OC ZINC000880668061 FE On-Demand Reactive KCNK3 54 38 COCc1cc(NC(=O)NNC(=O)c2cccc(N(C)C)c2)ccc1OC ZINC000880668061 FE On-Demand Reactive KCNK9 49 36 COc1ccc(CC(=O)NCc2ccc(OCC(F)(F)F)nn2)cc1F ZINC000880668064 FE On-Demand Anodyne TRPV1 15 45 COCc1cc(NC(=O)NC[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668065 EF On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)NC[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668065 EF On-Demand Anodyne HTR2A 19 43 COCc1cc(NC(=O)NC[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668065 EF On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668066 EF On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668066 EF On-Demand Anodyne HTR2A 19 43 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668066 EF On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)N2CCCC3(CCCC3)C2)ccc1OC ZINC000880668068 EI On-Demand Anodyne EPHX2 34 42 COCc1cc(NC(=O)N2CCCC3(CCCC3)C2)ccc1OC ZINC000880668068 EI On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCCC3(CCCC3)C2)ccc1OC ZINC000880668068 EI On-Demand Anodyne ENPP1 69 34 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccco2)ccc1OC ZINC000880668070 FH On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccco2)ccc1OC ZINC000880668070 FH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccco2)ccc1OC ZINC000880668071 FH On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccco2)ccc1OC ZINC000880668071 FH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccco2)ccc1OC ZINC000880668072 FH On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccco2)ccc1OC ZINC000880668072 FH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccco2)ccc1OC ZINC000880668073 FH On-Demand Anodyne TSHR 48 33 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccco2)ccc1OC ZINC000880668073 FH On-Demand Anodyne QRFPR 40 34 COCc1cc(NC(=O)NCCSSC)ccc1OC ZINC000880668074 DF On-Demand Reactive TSHR 55 32 COCc1cc(NC(=O)NCCSSC)ccc1OC ZINC000880668074 DF On-Demand Reactive QRFPR 42 34 COCc1cc(NC(=O)NCCSSC)ccc1OC ZINC000880668074 DF On-Demand Reactive ENPP1 62 31 COCc1cc(NC(=O)NNC(=O)C2CCCC2)ccc1OC ZINC000880668075 DE On-Demand Reactive TSHR 48 31 COCc1cc(NC(=O)NNC(=O)C2CCCC2)ccc1OC ZINC000880668075 DE On-Demand Reactive STK17B 42 39 COCc1cc(NC(=O)NNC(=O)C2CCCC2)ccc1OC ZINC000880668075 DE On-Demand Reactive QRFPR 53 43 COCc1cc(NC(=O)N2CC(OC(=O)NC(C)C)C2)ccc1OC ZINC000880668080 FE On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)N2CC(OC(=O)NC(C)C)C2)ccc1OC ZINC000880668080 FE On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCN3C(=O)OCC[C@H]3C2)ccc1OC ZINC000880668081 ED On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)N2CCN3C(=O)OCC[C@H]3C2)ccc1OC ZINC000880668081 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCN3C(=O)OCC[C@@H]3C2)ccc1OC ZINC000880668082 ED On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)N2CCN3C(=O)OCC[C@@H]3C2)ccc1OC ZINC000880668082 ED On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3C)CC2)ccc1OC ZINC000880668083 GI On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3C)CC2)ccc1OC ZINC000880668083 GI On-Demand Anodyne QRFPR 41 36 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3C)CC2)ccc1OC ZINC000880668084 GI On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3C)CC2)ccc1OC ZINC000880668084 GI On-Demand Anodyne QRFPR 41 36 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne HTR1A 32 44 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne DRD2 28 40 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne HTR1B 18 44 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne DRD3 38 40 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne PIK3CA 29 42 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne MTOR 50 39 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne STAT6 20 40 COCc1cc(NC(=O)NCc2ccccc2N2CCOCC2)ccc1OC ZINC000880668090 GF On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)N2CCO[C@H](c3cccc(C#N)c3)C2)ccc1OC ZINC000880668091 GG On-Demand Mild TSHR 53 30 COCc1cc(NC(=O)N2CCO[C@@H](c3cccc(C#N)c3)C2)ccc1OC ZINC000880668092 GG On-Demand Mild TSHR 53 30 C=CCS(=O)(=O)CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668093 ED On-Demand Mild TSHR 40 30 COCc1cc(NC(=O)NNC(=O)COc2cc(C)ccc2C)ccc1OC ZINC000880668095 GF On-Demand Reactive ENPP1 52 35 CCc1nnc(S)n1CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668096 FE On-Demand Anodyne QPCT 17 45 CCc1nnc(S)n1CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668096 FE On-Demand Anodyne ENPP1 66 31 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne ADRB1 42 33 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne TSHR 73 35 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne CTSK 16 40 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne CPT1A 42 29 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne QRFPR 41 38 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne KCNK3 44 38 COCc1cc(NC(=O)NCCNc2ccccc2)ccc1OC ZINC000880668098 EG On-Demand Anodyne KCNK9 42 38 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne HTR1D 15 43 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne HTR1B 16 43 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne PDGFRB 40 36 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne RBP4 30 42 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCC(C(=O)C(F)(F)F)CC2)ccc1OC ZINC000880668099 FG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NNC(=O)C(C)(C)C)ccc1OC ZINC000880668100 DE On-Demand Reactive TSHR 47 32 COCc1cc(NC(=O)NNC(=O)C(C)(C)C)ccc1OC ZINC000880668100 DE On-Demand Reactive QRFPR 42 34 COCc1cc(NC(=O)NNC(=O)C(C)(C)C)ccc1OC ZINC000880668100 DE On-Demand Reactive ENPP1 57 32 COCc1cc(NC(=O)N2CCN3C(=O)OC[C@H]3C2)ccc1OC ZINC000880668101 ED On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N2CCN3C(=O)OC[C@@H]3C2)ccc1OC ZINC000880668102 ED On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NOCC(F)F)ccc1OC ZINC000880668104 CE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NOCC(F)F)ccc1OC ZINC000880668104 CE On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)NOCC(F)F)ccc1OC ZINC000880668104 CE On-Demand Anodyne ENPP1 61 32 C#CCN(CC)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668105 CE On-Demand Mild QRFPR 44 36 COCc1cc(NC(=O)NOCc2ccccc2OC)ccc1OC ZINC000880668106 EG On-Demand Anodyne TSHR 63 35 COCc1cc(NC(=O)NOCc2ccccc2OC)ccc1OC ZINC000880668106 EG On-Demand Anodyne QRFPR 42 38 COCc1cc(NC(=O)NOCc2ccccc2OC)ccc1OC ZINC000880668106 EG On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NOCc2ccccc2OC)ccc1OC ZINC000880668106 EG On-Demand Anodyne KCNK3 44 40 COCc1cc(NC(=O)NOCc2ccccc2OC)ccc1OC ZINC000880668106 EG On-Demand Anodyne KCNK9 34 40 COCc1cc(NC(=O)N(C)CCN(C)C(=O)OC(C)(C)C)ccc1OC ZINC000880668111 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NNc2cccc(OC)n2)ccc1OC ZINC000880668112 EE On-Demand Reactive TSHR 42 34 COCc1cc(NC(=O)NNc2cccc(OC)n2)ccc1OC ZINC000880668112 EE On-Demand Reactive ENPP1 65 36 COCc1cc(NC(=O)NCc2ncc(C)o2)ccc1OC ZINC000880668113 DE On-Demand Anodyne TSHR 59 35 COCc1cc(NC(=O)NCc2ncc(C)o2)ccc1OC ZINC000880668113 DE On-Demand Anodyne PDGFRA 41 33 COCc1cc(NC(=O)NCc2ncc(C)o2)ccc1OC ZINC000880668113 DE On-Demand Anodyne ENPP1 53 34 C#CCN(Cc1ccccc1)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668117 EH On-Demand Mild TSHR 70 36 C#CCN(Cc1ccccc1)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668117 EH On-Demand Mild QRFPR 40 37 COCc1cc(NC(=O)NNC(=O)CC(F)(F)F)ccc1OC ZINC000880668119 ED On-Demand Reactive QRFPR 40 33 COCc1cc(NC(=O)NNC(=O)CC(F)(F)F)ccc1OC ZINC000880668119 ED On-Demand Reactive ENPP1 63 33 COCc1cc(NC(=O)N2CC[C@]3(C)[C@@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668120 FH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CC[C@]3(C)[C@@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668120 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@]3(C)[C@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668121 FH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CC[C@]3(C)[C@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668121 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@]3(C)[C@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668122 FH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CC[C@@]3(C)[C@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668122 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CC[C@@]3(C)[C@@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668123 FH On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)N2CC[C@@]3(C)[C@@H](C2)C3(Cl)Cl)ccc1OC ZINC000880668123 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCc2ccc(Cl)nc2)ccc1OC ZINC000880668125 EG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NCCc2ccc(Cl)nc2)ccc1OC ZINC000880668125 EG On-Demand Anodyne RAF1 28 43 COCc1cc(NC(=O)NCCc2ccc(Cl)nc2)ccc1OC ZINC000880668125 EG On-Demand Anodyne PRMT3 59 33 COCc1cc(NC(=O)NCCc2ccc(Cl)nc2)ccc1OC ZINC000880668125 EG On-Demand Anodyne ENPP1 46 35 C#CCN(C)C(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668126 CD On-Demand Mild QRFPR 42 35 C#CCC[C@H](O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668127 DD On-Demand Mild QRFPR 40 35 C#CCC[C@@H](O)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668128 DD On-Demand Mild QRFPR 40 35 COCc1cc(NC(=O)NCC(F)(F)Br)ccc1OC ZINC000880668129 FF On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)NCC(F)(F)Br)ccc1OC ZINC000880668129 FF On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NCC(F)(F)Br)ccc1OC ZINC000880668129 FF On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NCC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668132 FE On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)NCC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668132 FE On-Demand Anodyne EPHX2 33 40 COCc1cc(NC(=O)NCC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668132 FE On-Demand Anodyne CACNA1I 58 35 COCc1cc(NC(=O)NCC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668132 FE On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)NCC2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668132 FE On-Demand Anodyne ENPP1 56 31 COCc1cc(NC(=O)NNC(=O)COc2cc(C)cc(C)c2)ccc1OC ZINC000880668133 GF On-Demand Reactive TSHR 56 34 COCc1cc(NC(=O)NNC(=O)COc2cc(C)cc(C)c2)ccc1OC ZINC000880668133 GF On-Demand Reactive ENPP1 63 34 COCc1cc(NC(=O)N2CCC[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668134 GG On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)N2CCC[C@@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668134 GG On-Demand Anodyne QRFPR 44 36 O=C(CCc1ccc2ccccc2n1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668139 GG On-Demand Anodyne CYSLTR1 44 39 O=C(CCc1ccc2ccccc2n1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668139 GG On-Demand Anodyne SUCNR1 63 42 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668140 EE On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668140 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668140 EE On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668141 EE On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668141 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668141 EE On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668142 EE On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668142 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@H](C(=O)OC)[C@H]2C)ccc1OC ZINC000880668142 EE On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668143 EE On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668143 EE On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CC[C@@H](C(=O)OC)[C@@H]2C)ccc1OC ZINC000880668143 EE On-Demand Anodyne ENPP1 45 31 COCc1cc(NC(=O)N2CC[C@](C(=O)OC)(C(F)(F)F)C2)ccc1OC ZINC000880668144 GF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@](C(=O)OC)(C(F)(F)F)C2)ccc1OC ZINC000880668144 GF On-Demand Anodyne EPHX2 35 45 COCc1cc(NC(=O)N2CC[C@@](C(=O)OC)(C(F)(F)F)C2)ccc1OC ZINC000880668145 GF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@@](C(=O)OC)(C(F)(F)F)C2)ccc1OC ZINC000880668145 GF On-Demand Anodyne EPHX2 35 45 COCc1cc(NC(=O)NCc2cccc(F)n2)ccc1OC ZINC000880668147 DF On-Demand Anodyne TSHR 63 35 COCc1cc(NC(=O)NCc2cccc(F)n2)ccc1OC ZINC000880668147 DF On-Demand Anodyne ROCK2 24 41 COCc1cc(NC(=O)NCc2cccc(F)n2)ccc1OC ZINC000880668147 DF On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N2CC=C(c3ccccc3)C2)ccc1OC ZINC000880668152 EH On-Demand Anodyne TSHR 63 36 COCc1cc(NC(=O)N2CC=C(c3ccccc3)C2)ccc1OC ZINC000880668152 EH On-Demand Anodyne QRFPR 40 37 COCc1cc(NC(=O)N2CCC3(CC2)CC(C(=O)OC)=NO3)ccc1OC ZINC000880668153 GE On-Demand Anodyne EPHX2 18 40 COCc1cc(NC(=O)NCCC(=O)OCc2ccccc2)ccc1OC ZINC000880668156 FG On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)NCCC(=O)OCc2ccccc2)ccc1OC ZINC000880668156 FG On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)NNC(=O)c2cccn2C)ccc1OC ZINC000880668167 ED On-Demand Reactive TSHR 55 34 COCc1cc(NC(=O)NNC(=O)c2cccn2C)ccc1OC ZINC000880668167 ED On-Demand Reactive ENPP1 45 32 COCc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668170 FG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668170 FG On-Demand Anodyne KCNA3 40 36 COCc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668170 FG On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668171 FG On-Demand Anodyne TSHR 68 33 COCc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668171 FG On-Demand Anodyne KCNA3 40 36 COCc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668171 FG On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NNC(=O)C(C)(C)c2ccccc2)ccc1OC ZINC000880668172 FF On-Demand Reactive TSHR 68 34 COCc1cc(NC(=O)NNC(=O)C(C)(C)c2ccccc2)ccc1OC ZINC000880668172 FF On-Demand Reactive NPY2R 23 41 COCc1cc(NC(=O)NNC(=O)C(C)(C)c2ccccc2)ccc1OC ZINC000880668172 FF On-Demand Reactive QRFPR 40 37 COCc1cc(NC(=O)NNC(=O)CC(C)(C)C)ccc1OC ZINC000880668174 DE On-Demand Reactive QRFPR 41 33 COCc1cc(NC(=O)NNC(=O)CC(C)(C)C)ccc1OC ZINC000880668174 DE On-Demand Reactive ENPP1 64 33 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne HTR1D 18 41 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne HTR1B 22 41 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne PDGFRB 45 37 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N2CCC(c3nccc(C)n3)CC2)ccc1OC ZINC000880668177 FG On-Demand Anodyne ENPP1 73 41 COCc1cc(NC(=O)NCc2cccnc2F)ccc1OC ZINC000880668178 DF On-Demand Anodyne TSHR 59 35 COCc1cc(NC(=O)NCc2cccnc2F)ccc1OC ZINC000880668178 DF On-Demand Anodyne GRM4 15 41 COCc1cc(NC(=O)NCc2cccnc2F)ccc1OC ZINC000880668178 DF On-Demand Anodyne ROCK2 21 45 COCc1cc(NC(=O)NCc2cccnc2F)ccc1OC ZINC000880668178 DF On-Demand Anodyne PDGFRA 42 36 COCc1cc(NC(=O)NCc2cccnc2F)ccc1OC ZINC000880668178 DF On-Demand Anodyne ENPP1 53 38 COCc1cc(NC(=O)NOCC(C)(C)O)ccc1OC ZINC000880668180 CD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NOCC(C)(C)O)ccc1OC ZINC000880668180 CD On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NOCC(C)(C)O)ccc1OC ZINC000880668180 CD On-Demand Anodyne ENPP1 66 32 COCc1cc(NC(=O)NC[C@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668181 GG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NC[C@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668181 GG On-Demand Anodyne ROCK2 16 44 COCc1cc(NC(=O)NC[C@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668181 GG On-Demand Anodyne LUCI_PHOPY 54 50 COCc1cc(NC(=O)NC[C@@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668182 GG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NC[C@@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668182 GG On-Demand Anodyne ROCK2 16 44 COCc1cc(NC(=O)NC[C@@H]2CC(c3ccc(OC)cc3)=NO2)ccc1OC ZINC000880668182 GG On-Demand Anodyne LUCI_PHOPY 54 50 COCc1cc(NC(=O)NNC(=O)CCc2ccc(OC)cc2)ccc1OC ZINC000880668184 GF On-Demand Reactive TSHR 57 35 COCc1cc(NC(=O)NNC(=O)CCc2ccc(OC)cc2)ccc1OC ZINC000880668184 GF On-Demand Reactive FFAR1 15 41 COCc1cc(NC(=O)NNC(=O)CCc2ccc(OC)cc2)ccc1OC ZINC000880668184 GF On-Demand Reactive ENPP1 63 33 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)cc2)ccc1OC ZINC000880668185 FE On-Demand Reactive TSHR 62 39 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)cc2)ccc1OC ZINC000880668185 FE On-Demand Reactive KDR 22 41 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)cc2)ccc1OC ZINC000880668185 FE On-Demand Reactive PDGFRA 41 38 COCc1cc(NC(=O)NNC(=O)COc2ccc(C)cc2)ccc1OC ZINC000880668185 FE On-Demand Reactive ENPP1 63 34 COCc1cc(NC(=O)NC2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880668188 GH On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)NC2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880668188 GH On-Demand Anodyne KCNA3 44 41 COCc1cc(NC(=O)NC2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880668188 GH On-Demand Anodyne EPHX2 45 38 COCc1cc(NC(=O)NC2CCC(O)(c3ccccc3)CC2)ccc1OC ZINC000880668188 GH On-Demand Anodyne QRFPR 43 40 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@@H]2c2ccccc2)ccc1OC ZINC000880668189 GF On-Demand Reactive TSHR 70 34 COCc1cc(NC(=O)NNC(=O)[C@H]2CCO[C@@H]2c2ccccc2)ccc1OC ZINC000880668189 GF On-Demand Reactive QRFPR 46 41 COCc1cc(NC(=O)NCc2cc(Cl)ccn2)ccc1OC ZINC000880668191 EG On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NCc2cc(Cl)ccn2)ccc1OC ZINC000880668191 EG On-Demand Anodyne HTR2A 32 42 COCc1cc(NC(=O)NCc2cc(Cl)ccn2)ccc1OC ZINC000880668191 EG On-Demand Anodyne PDGFRA 41 40 COCc1cc(NC(=O)NCc2cc(Cl)ccn2)ccc1OC ZINC000880668191 EG On-Demand Anodyne ENPP1 54 36 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2OC)ccc1OC ZINC000880668192 FE On-Demand Reactive TSHR 71 34 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2OC)ccc1OC ZINC000880668192 FE On-Demand Reactive QRFPR 42 37 COCc1cc(NC(=O)NNC(=O)Cc2ccccc2OC)ccc1OC ZINC000880668192 FE On-Demand Reactive ENPP1 64 34 COCc1cc(NC(=O)N[C@H]2CC[C@H](C)C2)ccc1OC ZINC000880668193 CG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N[C@H]2CC[C@H](C)C2)ccc1OC ZINC000880668193 CG On-Demand Anodyne EPHX2 46 40 COCc1cc(NC(=O)N[C@H]2CC[C@H](C)C2)ccc1OC ZINC000880668193 CG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N[C@@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668194 CG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N[C@@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668194 CG On-Demand Anodyne EPHX2 46 40 COCc1cc(NC(=O)N[C@@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668194 CG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N[C@@H]2CC[C@H](C)C2)ccc1OC ZINC000880668195 CG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N[C@@H]2CC[C@H](C)C2)ccc1OC ZINC000880668195 CG On-Demand Anodyne EPHX2 46 40 COCc1cc(NC(=O)N[C@@H]2CC[C@H](C)C2)ccc1OC ZINC000880668195 CG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)N[C@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668196 CG On-Demand Anodyne TSHR 41 32 COCc1cc(NC(=O)N[C@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668196 CG On-Demand Anodyne EPHX2 46 40 COCc1cc(NC(=O)N[C@H]2CC[C@@H](C)C2)ccc1OC ZINC000880668196 CG On-Demand Anodyne QRFPR 45 37 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive TSHR 72 37 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive INHA 42 34 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive HDAC8 16 40 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive MTNR1B 21 40 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive HDAC2 16 41 COCc1cc(NC(=O)NNC(=O)CCCc2ccccc2)ccc1OC ZINC000880668199 FG On-Demand Reactive ENPP1 60 31 COCc1cc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668202 GG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668202 GG On-Demand Anodyne CACNA1I 66 36 COCc1cc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668202 GG On-Demand Anodyne GPR119 35 40 COCc1cc(NC(=O)NC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668202 GG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668203 GG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668203 GG On-Demand Anodyne CACNA1I 66 36 COCc1cc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668203 GG On-Demand Anodyne GPR119 35 40 COCc1cc(NC(=O)NC[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668203 GG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N2CCCC3(C2)OCCO3)ccc1OC ZINC000880668205 EE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCCC3(C2)OCCO3)ccc1OC ZINC000880668205 EE On-Demand Anodyne EPHX2 32 42 COCc1cc(NC(=O)N2CCCC3(C2)OCCO3)ccc1OC ZINC000880668205 EE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@@H](C)CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668206 GG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NC[C@@H](C)CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668206 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@H](C)CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668207 GG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NC[C@H](C)CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668207 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)C2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668208 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@H](C)C2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668208 GF On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)N[C@@H](C)C2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668209 GF On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N[C@@H](C)C2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668209 GF On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NC[C@H]2COC3(CCCC3)O2)ccc1OC ZINC000880668210 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)NC[C@H]2COC3(CCCC3)O2)ccc1OC ZINC000880668210 FF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@@H]2COC3(CCCC3)O2)ccc1OC ZINC000880668211 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)NC[C@@H]2COC3(CCCC3)O2)ccc1OC ZINC000880668211 FF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NNC(=O)CSc2ccc(C)cc2)ccc1OC ZINC000880668212 GG On-Demand Reactive QRFPR 40 33 COCc1cc(NC(=O)NNC(=O)CSc2ccc(C)cc2)ccc1OC ZINC000880668212 GG On-Demand Reactive ENPP1 79 39 COCc1cc(NC(=O)NNC(=O)CSc2ccc(C)cc2)ccc1OC ZINC000880668212 GG On-Demand Reactive FAS 42 36 C#C[C@H](NC(=O)Nc1ccc(OC)c(COC)c1)C(C)C ZINC000880668214 CF On-Demand Mild ENPP1 49 30 C#C[C@@H](NC(=O)Nc1ccc(OC)c(COC)c1)C(C)C ZINC000880668215 CF On-Demand Mild ENPP1 49 30 C#CCOCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668216 CD On-Demand Mild QRFPR 41 33 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668217 FE On-Demand Anodyne TSHR 46 31 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668217 FE On-Demand Anodyne EPHX2 48 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668217 FE On-Demand Anodyne CCR8 23 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668217 FE On-Demand Anodyne QRFPR 41 34 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668217 FE On-Demand Anodyne ENPP1 60 32 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668218 FE On-Demand Anodyne TSHR 46 31 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668218 FE On-Demand Anodyne EPHX2 48 45 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668218 FE On-Demand Anodyne CCR8 23 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668218 FE On-Demand Anodyne QRFPR 41 34 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668218 FE On-Demand Anodyne ENPP1 60 32 COCc1cc(NC(=O)NCc2ccon2)ccc1OC ZINC000880668219 CE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NCc2ccon2)ccc1OC ZINC000880668219 CE On-Demand Anodyne PRMT3 62 35 COCc1cc(NC(=O)NCc2ccon2)ccc1OC ZINC000880668219 CE On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)NNC(=O)CCOc2ccccc2)ccc1OC ZINC000880668225 FE On-Demand Reactive TSHR 64 38 COCc1cc(NC(=O)NNC(=O)CCOc2ccccc2)ccc1OC ZINC000880668225 FE On-Demand Reactive TSPO 42 33 COCc1cc(NC(=O)NNC(=O)CCOc2ccccc2)ccc1OC ZINC000880668225 FE On-Demand Reactive PLA2G4B 44 35 COCc1cc(NC(=O)NNC(=O)CCOc2ccccc2)ccc1OC ZINC000880668225 FE On-Demand Reactive FAAH 18 40 COCc1cc(NC(=O)NNC(=O)CCOc2ccccc2)ccc1OC ZINC000880668225 FE On-Demand Reactive ENPP1 53 33 COCc1cc(NC(=O)N[C@H]2CCCc3nc(C)sc32)ccc1OC ZINC000880668226 FH On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@@H]2CCCc3nc(C)sc32)ccc1OC ZINC000880668227 FH On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)NNC(=O)CCC(C)C)ccc1OC ZINC000880668228 DE On-Demand Reactive QRFPR 40 33 COCc1cc(NC(=O)NNC(=O)CCC(C)C)ccc1OC ZINC000880668228 DE On-Demand Reactive ENPP1 63 33 COCc1cc(NC(=O)NC[C@H](O)COC)ccc1OC ZINC000880668231 CC On-Demand Anodyne ADRB1 44 34 COCc1cc(NC(=O)NC[C@H](O)COC)ccc1OC ZINC000880668231 CC On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H](O)COC)ccc1OC ZINC000880668231 CC On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC[C@H](O)COC)ccc1OC ZINC000880668231 CC On-Demand Anodyne ENPP1 60 30 COCc1cc(NC(=O)NCCC#N)ccc1OC ZINC000880668232 CD On-Demand Mild ADRB1 41 31 COCc1cc(NC(=O)NCCC#N)ccc1OC ZINC000880668232 CD On-Demand Mild TSHR 53 31 COCc1cc(NC(=O)NCCC#N)ccc1OC ZINC000880668232 CD On-Demand Mild QPCT 18 47 COCc1cc(NC(=O)NCCC#N)ccc1OC ZINC000880668232 CD On-Demand Mild QRFPR 40 33 COCc1cc(NC(=O)NCCC#N)ccc1OC ZINC000880668232 CD On-Demand Mild ENPP1 45 30 COCc1cc(NC(=O)NC(C)(C)CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668237 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N(CC(C)(C)C)OC)ccc1OC ZINC000880668238 DG On-Demand Anodyne TSHR 46 31 COCc1cc(NC(=O)N(CC(C)(C)C)OC)ccc1OC ZINC000880668238 DG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N(CC(C)(C)C)OC)ccc1OC ZINC000880668238 DG On-Demand Anodyne ENPP1 50 31 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C/c2ccsc2)n1 ZINC000880668240 DD On-Demand Anodyne UL26 80 47 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C/c2ccsc2)n1 ZINC000880668240 DD On-Demand Anodyne SCAF_EBVB9 65 35 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C\c2ccsc2)n1 ZINC000880668241 DD On-Demand Anodyne UL26 80 47 CCOC(=O)c1n[nH]c([C@H](C)NC(=O)/C=C\c2ccsc2)n1 ZINC000880668241 DD On-Demand Anodyne SCAF_EBVB9 65 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C/c2ccsc2)n1 ZINC000880668242 DD On-Demand Anodyne UL26 80 47 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C/c2ccsc2)n1 ZINC000880668242 DD On-Demand Anodyne SCAF_EBVB9 65 35 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C\c2ccsc2)n1 ZINC000880668243 DD On-Demand Anodyne UL26 80 47 CCOC(=O)c1n[nH]c([C@@H](C)NC(=O)/C=C\c2ccsc2)n1 ZINC000880668243 DD On-Demand Anodyne SCAF_EBVB9 65 35 COCc1cc(NC(=O)NCC2OCCCO2)ccc1OC ZINC000880668244 DD On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NCC2OCCCO2)ccc1OC ZINC000880668244 DD On-Demand Anodyne QRFPR 50 42 COCc1cc(NC(=O)NCc2cccc(NC(=O)OC)c2)ccc1OC ZINC000880668246 FG On-Demand Anodyne TSHR 74 37 COCc1cc(NC(=O)NCc2cccc(NC(=O)OC)c2)ccc1OC ZINC000880668246 FG On-Demand Anodyne ROCK2 35 48 COCc1cc(NC(=O)NCc2ccc([C@@H](C)O)cc2)ccc1OC ZINC000880668250 EG On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NCc2ccc([C@@H](C)O)cc2)ccc1OC ZINC000880668250 EG On-Demand Anodyne ROCK2 18 44 COCc1cc(NC(=O)NCc2ccc([C@@H](C)O)cc2)ccc1OC ZINC000880668250 EG On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)NCc2ccc([C@H](C)O)cc2)ccc1OC ZINC000880668251 EG On-Demand Anodyne TSHR 67 32 COCc1cc(NC(=O)NCc2ccc([C@H](C)O)cc2)ccc1OC ZINC000880668251 EG On-Demand Anodyne ROCK2 18 44 COCc1cc(NC(=O)NCc2ccc([C@H](C)O)cc2)ccc1OC ZINC000880668251 EG On-Demand Anodyne ENPP1 55 30 COCc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ccc1OC ZINC000880668253 EG On-Demand Anodyne TSHR 48 34 COCc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ccc1OC ZINC000880668253 EG On-Demand Anodyne HTR2A 43 44 COCc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ccc1OC ZINC000880668253 EG On-Demand Anodyne HTR2C 16 44 COCc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ccc1OC ZINC000880668253 EG On-Demand Anodyne KDR 17 40 COCc1cc(NC(=O)Nc2cnn(C(C)(C)C)c2)ccc1OC ZINC000880668253 EG On-Demand Anodyne ENPP1 64 35 COCc1cc(NC(=O)N[C@@H](CCO)C2CC2)ccc1OC ZINC000880668256 DE On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N[C@H](CCO)C2CC2)ccc1OC ZINC000880668257 DE On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)N2CCC(O)(c3cccc(C)c3C)CC2)ccc1OC ZINC000880668263 GH On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N[C@@H](Cn2ccnc2)C(C)(C)C)ccc1OC ZINC000880668264 FG On-Demand Anodyne QPCT 31 51 COCc1cc(NC(=O)N[C@@H](Cn2ccnc2)C(C)(C)C)ccc1OC ZINC000880668264 FG On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)N[C@H](Cn2ccnc2)C(C)(C)C)ccc1OC ZINC000880668265 FG On-Demand Anodyne QPCT 31 51 COCc1cc(NC(=O)N[C@H](Cn2ccnc2)C(C)(C)C)ccc1OC ZINC000880668265 FG On-Demand Anodyne ENPP1 40 32 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668268 FF On-Demand Anodyne TSHR 71 36 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668268 FF On-Demand Anodyne HTR2A 15 40 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668268 FF On-Demand Anodyne ADRB3 25 41 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668268 FF On-Demand Anodyne F7 19 41 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668268 FF On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668269 FF On-Demand Anodyne TSHR 71 36 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668269 FF On-Demand Anodyne HTR2A 15 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668269 FF On-Demand Anodyne ADRB3 25 41 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668269 FF On-Demand Anodyne F7 19 41 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC)cc2)ccc1OC ZINC000880668269 FF On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)NC[C@H]2CN3CCC[C@@H]3CO2)ccc1OC ZINC000880668275 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H]2CN3CCC[C@@H]3CO2)ccc1OC ZINC000880668275 ED On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@H]2CN3CCC[C@H]3CO2)ccc1OC ZINC000880668276 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@H]2CN3CCC[C@H]3CO2)ccc1OC ZINC000880668276 ED On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@@H]2CN3CCC[C@@H]3CO2)ccc1OC ZINC000880668277 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@@H]2CN3CCC[C@@H]3CO2)ccc1OC ZINC000880668277 ED On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@@H]2CN3CCC[C@H]3CO2)ccc1OC ZINC000880668278 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NC[C@@H]2CN3CCC[C@H]3CO2)ccc1OC ZINC000880668278 ED On-Demand Anodyne QRFPR 43 36 CN1C[C@H](C(=O)NCc2ccc(OCC(F)(F)F)nn2)c2ccccc2C1=O ZINC000880668281 GD On-Demand Anodyne P2RX7 47 39 CN1C[C@@H](C(=O)NCc2ccc(OCC(F)(F)F)nn2)c2ccccc2C1=O ZINC000880668282 GD On-Demand Anodyne P2RX7 47 39 COCc1cc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668284 GG On-Demand Anodyne PDGFRB 44 39 COCc1cc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668284 GG On-Demand Anodyne F13A1 23 41 COCc1cc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668284 GG On-Demand Anodyne GPR119 32 43 COCc1cc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668284 GG On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668284 GG On-Demand Anodyne ENPP1 56 32 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccc(OC)c(COC)c2)c1 ZINC000880668288 GH On-Demand Mild TSHR 72 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2ccc(OC)c(COC)c2)c1 ZINC000880668288 GH On-Demand Mild ROCK2 38 48 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccc(OC)c(COC)c2)c1 ZINC000880668289 GH On-Demand Mild TSHR 72 36 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2ccc(OC)c(COC)c2)c1 ZINC000880668289 GH On-Demand Mild ROCK2 38 48 COCc1cc(NC(=O)NCc2c(C)cccc2F)ccc1OC ZINC000880668296 EH On-Demand Anodyne TSHR 63 40 COCc1cc(NC(=O)NCc2c(C)cccc2F)ccc1OC ZINC000880668296 EH On-Demand Anodyne ROCK2 15 42 COCc1cc(NC(=O)N(C)CCc2ccccc2F)ccc1OC ZINC000880668305 EH On-Demand Anodyne TSHR 56 35 COCc1cc(NC(=O)NCC(=O)NCc2ccccc2)ccc1OC ZINC000880668306 FE On-Demand Anodyne TSHR 80 41 COCc1cc(NC(=O)NCC(=O)NCc2ccccc2)ccc1OC ZINC000880668306 FE On-Demand Anodyne ROCK2 26 43 COCc1cc(NC(=O)NCC(=O)NCc2ccccc2)ccc1OC ZINC000880668306 FE On-Demand Anodyne F7 28 41 COCc1cc(NC(=O)NCC(=O)NCc2ccccc2)ccc1OC ZINC000880668306 FE On-Demand Anodyne PRMT3 45 36 COCc1cc(NC(=O)NCC(=O)NCc2ccccc2)ccc1OC ZINC000880668306 FE On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)N2CCC(CCN3CCOCC3)CC2)ccc1OC ZINC000880668313 GF On-Demand Anodyne HTR1D 19 48 COCc1cc(NC(=O)N2CCC(CCN3CCOCC3)CC2)ccc1OC ZINC000880668313 GF On-Demand Anodyne HTR1B 22 42 COCc1cc(NC(=O)N2CCC(CCN3CCOCC3)CC2)ccc1OC ZINC000880668313 GF On-Demand Anodyne PDGFRB 46 42 COCc1cc(NC(=O)N2CCC(CCN3CCOCC3)CC2)ccc1OC ZINC000880668313 GF On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NC2CCN(C(C)(C)C)CC2)ccc1OC ZINC000880668315 EG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC2CCN(C(C)(C)C)CC2)ccc1OC ZINC000880668315 EG On-Demand Anodyne EPHX2 51 44 COCc1cc(NC(=O)NC2CCN(C(C)(C)C)CC2)ccc1OC ZINC000880668315 EG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N(C)Cc2c(C)nn(C)c2C)ccc1OC ZINC000880668316 EF On-Demand Anodyne ENPP1 50 32 COCc1cc(NC(=O)Nc2ccc(NC(C)=O)c(C)c2)ccc1OC ZINC000880668318 FH On-Demand Anodyne TSHR 63 36 COCc1cc(NC(=O)Nc2ccc(NC(C)=O)c(C)c2)ccc1OC ZINC000880668318 FH On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)Nc2ccc(NC(C)=O)c(C)c2)ccc1OC ZINC000880668318 FH On-Demand Anodyne ENPP1 56 34 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668319 FF On-Demand Anodyne TSHR 55 33 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668319 FF On-Demand Anodyne QRFPR 42 35 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)C1 ZINC000880668319 FF On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NCc2cccn2C)ccc1OC ZINC000880668322 DF On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NCc2cccn2C)ccc1OC ZINC000880668322 DF On-Demand Anodyne ROCK2 17 42 COCc1cc(NC(=O)NCc2cccn2C)ccc1OC ZINC000880668322 DF On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne ADRB3 43 39 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne MTNR1B 40 44 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne ROCK2 27 44 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne F7 17 47 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668325 FF On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne ADRB3 43 39 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne MTNR1B 40 44 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne ROCK2 27 44 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne F7 17 47 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC)c2)ccc1OC ZINC000880668326 FF On-Demand Anodyne ENPP1 51 32 COCc1cc(NC(=O)N[C@@H](C)c2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668329 GH On-Demand Clean PIK3CA 25 40 COCc1cc(NC(=O)N[C@@H](C)c2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668329 GH On-Demand Clean MTOR 43 39 COCc1cc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668330 GH On-Demand Clean PIK3CA 25 40 COCc1cc(NC(=O)N[C@H](C)c2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668330 GH On-Demand Clean MTOR 43 39 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668333 FF On-Demand Anodyne PDGFRB 46 44 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668333 FF On-Demand Anodyne QRFPR 42 34 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668333 FF On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)C)CC2)ccc1OC ZINC000880668335 GF On-Demand Anodyne EPHX2 53 48 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)C)CC2)ccc1OC ZINC000880668335 GF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)C)CC2)ccc1OC ZINC000880668335 GF On-Demand Anodyne ENPP1 66 31 COCc1cc(NC(=O)N2CCCN(C(=O)OCC(C)C)CC2)ccc1OC ZINC000880668336 GG On-Demand Anodyne PDGFRB 43 38 COCc1cc(NC(=O)N2CCCN(C(=O)OCC(C)C)CC2)ccc1OC ZINC000880668336 GG On-Demand Anodyne ENPP1 60 32 COCc1cc(NC(=O)NCC2Cc3ccccc3C2)ccc1OC ZINC000880668339 EG On-Demand Anodyne TSHR 70 33 COCc1cc(NC(=O)NCC2Cc3ccccc3C2)ccc1OC ZINC000880668339 EG On-Demand Anodyne QRFPR 46 41 COCc1cc(NC(=O)N[C@@H](C)C(=O)OC2CCCC2)ccc1OC ZINC000880668340 FF On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N[C@@H](C)C(=O)OC2CCCC2)ccc1OC ZINC000880668340 FF On-Demand Anodyne PDE4A 24 43 COCc1cc(NC(=O)N[C@@H](C)C(=O)OC2CCCC2)ccc1OC ZINC000880668340 FF On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)N[C@@H](C)C(=O)OC2CCCC2)ccc1OC ZINC000880668340 FF On-Demand Anodyne ENPP1 59 31 C=C(Cl)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668346 CF On-Demand Mild TSHR 68 34 C=C(Cl)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668346 CF On-Demand Mild QRFPR 41 34 C=C(Cl)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668346 CF On-Demand Mild ENPP1 70 34 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC(C)C)cc2)ccc1OC ZINC000880668354 GG On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NC[C@H](O)c2ccc(OC(C)C)cc2)ccc1OC ZINC000880668354 GG On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC(C)C)cc2)ccc1OC ZINC000880668355 GG On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(OC(C)C)cc2)ccc1OC ZINC000880668355 GG On-Demand Anodyne ENPP1 67 32 C#CCSCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668356 DE On-Demand Mild QRFPR 43 34 C#CCSCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668356 DE On-Demand Mild ENPP1 44 30 COCc1cc(NC(=O)N[C@H]2COc3ccccc32)ccc1OC ZINC000880668360 EG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@H]2COc3ccccc32)ccc1OC ZINC000880668360 EG On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)N[C@@H]2COc3ccccc32)ccc1OC ZINC000880668361 EG On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N[C@@H]2COc3ccccc32)ccc1OC ZINC000880668361 EG On-Demand Anodyne QRFPR 41 37 COCc1cc(NC(=O)NC[C@](C)(O)c2ccsc2)ccc1OC ZINC000880668362 FF On-Demand Anodyne QRFPR 40 39 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccsc2)ccc1OC ZINC000880668363 FF On-Demand Anodyne QRFPR 40 39 COCc1cc(NC(=O)NCC(C)(C)SC)ccc1OC ZINC000880668364 DG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NCC(C)(C)SC)ccc1OC ZINC000880668364 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCC(C)(C)SC)ccc1OC ZINC000880668364 DG On-Demand Anodyne ENPP1 62 31 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne HTR1D 16 49 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne HTR1B 20 49 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne PDGFRB 57 41 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne RBP4 17 42 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)N2CCN(C(=O)OC)CC2)ccc1OC ZINC000880668369 ED On-Demand Anodyne ENPP1 72 36 COCc1cc(NC(=O)NCc2cccc(N3CCOC3=O)c2)ccc1OC ZINC000880668371 GG On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NCc2cccc(N3CCOC3=O)c2)ccc1OC ZINC000880668371 GG On-Demand Anodyne ROCK2 22 40 COCc1cc(NC(=O)NC[C@H](O)c2ccsc2)ccc1OC ZINC000880668375 EF On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NC[C@H](O)c2ccsc2)ccc1OC ZINC000880668375 EF On-Demand Anodyne QRFPR 41 40 COCc1cc(NC(=O)NC[C@H](O)c2ccsc2)ccc1OC ZINC000880668375 EF On-Demand Anodyne ENPP1 59 31 COCc1cc(NC(=O)NC[C@@H](O)c2ccsc2)ccc1OC ZINC000880668376 EF On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)NC[C@@H](O)c2ccsc2)ccc1OC ZINC000880668376 EF On-Demand Anodyne QRFPR 41 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccsc2)ccc1OC ZINC000880668376 EF On-Demand Anodyne ENPP1 59 31 COCc1cc(NC(=O)NC[C@](C)(O)c2cc(C)oc2C)ccc1OC ZINC000880668378 FG On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)NC[C@@](C)(O)c2cc(C)oc2C)ccc1OC ZINC000880668379 FG On-Demand Anodyne TSHR 53 32 C[C@@H](Oc1cccc(CO)c1)C(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668380 GD On-Demand Anodyne CARM1 43 35 C[C@@H](Oc1cccc(CO)c1)C(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668380 GD On-Demand Anodyne PDS 46 36 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668382 GG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668382 GG On-Demand Anodyne EPHX2 57 48 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668382 GG On-Demand Anodyne F13A1 23 43 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668382 GG On-Demand Anodyne GPR119 44 42 COCc1cc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668382 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@@H]2COCCO2)ccc1OC ZINC000880668386 DD On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NC[C@@H]2COCCO2)ccc1OC ZINC000880668386 DD On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@H]2COCCO2)ccc1OC ZINC000880668387 DD On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NC[C@H]2COCCO2)ccc1OC ZINC000880668387 DD On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668393 FG On-Demand Clean TSHR 56 35 COCc1cc(NC(=O)N[C@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668393 FG On-Demand Clean THRB 43 34 COCc1cc(NC(=O)N[C@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668393 FG On-Demand Clean CA1 17 40 COCc1cc(NC(=O)N[C@@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668394 FG On-Demand Clean TSHR 56 35 COCc1cc(NC(=O)N[C@@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668394 FG On-Demand Clean THRB 43 34 COCc1cc(NC(=O)N[C@@H](C)c2cc(OC)ccc2O)ccc1OC ZINC000880668394 FG On-Demand Clean CA1 17 40 C#CCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668395 CD On-Demand Mild TSHR 53 30 C#CCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668395 CD On-Demand Mild QRFPR 43 35 C#CCCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668395 CD On-Demand Mild ENPP1 45 30 COCc1cc(NC(=O)N[C@H]2CC[C@H](SC)C2)ccc1OC ZINC000880668399 DG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)N[C@@H]2CC[C@H](SC)C2)ccc1OC ZINC000880668400 DG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)N[C@H]2CC[C@@H](SC)C2)ccc1OC ZINC000880668401 DG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)N[C@@H]2CC[C@@H](SC)C2)ccc1OC ZINC000880668402 DG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)NCc2ccc(Cl)nc2)ccc1OC ZINC000880668404 EG On-Demand Anodyne TSHR 72 38 COCc1cc(NC(=O)NCc2ccc(Cl)nc2)ccc1OC ZINC000880668404 EG On-Demand Anodyne ROCK2 24 47 COCc1cc(NC(=O)NCc2ccc(Cl)nc2)ccc1OC ZINC000880668404 EG On-Demand Anodyne ENPP1 48 36 COCc1cc(NC(=O)NCc2ccc(Cl)nc2)ccc1OC ZINC000880668404 EG On-Demand Anodyne NAMPT 33 52 COCc1cc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668405 GG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668405 GG On-Demand Anodyne ACACB 15 40 COCc1cc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668405 GG On-Demand Anodyne CACNA1I 55 35 COCc1cc(NC(=O)N2CC[C@@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668405 GG On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668406 GG On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668406 GG On-Demand Anodyne ACACB 15 40 COCc1cc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668406 GG On-Demand Anodyne CACNA1I 55 35 COCc1cc(NC(=O)N2CC[C@H](CNC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668406 GG On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)NCc2ccc(N3CC=CC3)cc2)ccc1OC ZINC000880668410 FH On-Demand Clean TSHR 71 35 COCc1cc(NC(=O)NCc2ccc(N3CC=CC3)cc2)ccc1OC ZINC000880668410 FH On-Demand Clean ROCK2 23 42 COCc1cc(NC(=O)NC[C@H](C)N2CCCCC2)ccc1OC ZINC000880668413 EF On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NC[C@H](C)N2CCCCC2)ccc1OC ZINC000880668413 EF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@H](C)N2CCCCC2)ccc1OC ZINC000880668413 EF On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)NC[C@@H](C)N2CCCCC2)ccc1OC ZINC000880668414 EF On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NC[C@@H](C)N2CCCCC2)ccc1OC ZINC000880668414 EF On-Demand Anodyne QRFPR 43 35 COCc1cc(NC(=O)NC[C@@H](C)N2CCCCC2)ccc1OC ZINC000880668414 EF On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)NC[C@@H]2OCCc3sccc32)ccc1OC ZINC000880668418 FG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC[C@@H]2OCCc3sccc32)ccc1OC ZINC000880668418 FG On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)NC[C@H]2OCCc3sccc32)ccc1OC ZINC000880668419 FG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)NC[C@H]2OCCc3sccc32)ccc1OC ZINC000880668419 FG On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)NCC[S@@](=O)Cc2ccccc2)ccc1OC ZINC000880668421 GF On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)NCC[S@](=O)Cc2ccccc2)ccc1OC ZINC000880668422 GF On-Demand Anodyne TSHR 74 36 COCc1cc(NC(=O)NC[C@@H](O)CC(C)C)ccc1OC ZINC000880668424 DE On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@@H](O)CC(C)C)ccc1OC ZINC000880668424 DE On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NC[C@H](O)CC(C)C)ccc1OC ZINC000880668425 DE On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)NC[C@H](O)CC(C)C)ccc1OC ZINC000880668425 DE On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne ADRB2 25 43 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne ADRB1 41 32 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne SOAT1 24 42 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne QRFPR 40 35 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne ENPP1 54 31 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne KCNK3 50 40 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2OC)ccc1OC ZINC000880668426 FF On-Demand Anodyne KCNK9 43 40 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2Cl)ccc1OC ZINC000880668427 FG On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2Cl)ccc1OC ZINC000880668428 FG On-Demand Anodyne TSHR 71 35 O=C(CCc1cccnc1Cl)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668429 FF On-Demand Anodyne SUCNR1 61 39 COCc1cc(NC(=O)N2CCCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668432 GH On-Demand Clean TSHR 48 33 COCc1cc(NC(=O)N2CCCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668432 GH On-Demand Clean HTR1D 18 52 COCc1cc(NC(=O)N2CCCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668432 GH On-Demand Clean HTR1B 21 52 COCc1cc(NC(=O)N2CCCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668432 GH On-Demand Clean PDGFRB 59 42 COCc1cc(NC(=O)N2CCCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668432 GH On-Demand Clean ENPP1 40 32 O=C(NCc1ccc(OCC(F)(F)F)nn1)c1cncc(Cl)n1 ZINC000880668433 ED On-Demand Anodyne SCN10A 35 40 CN1C[C@H](C(=O)NCc2ccc(OCC(F)(F)F)nn2)CCC1=O ZINC000880668434 EC On-Demand Anodyne P2RX7 46 41 CN1C[C@@H](C(=O)NCc2ccc(OCC(F)(F)F)nn2)CCC1=O ZINC000880668435 EC On-Demand Anodyne P2RX7 46 41 O=C(CCc1ncccn1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668436 ED On-Demand Anodyne SUCNR1 56 41 COCc1cc(NC(=O)NCc2nncn2C)ccc1OC ZINC000880668437 DD On-Demand Anodyne TSHR 55 32 COCc1cc(NC(=O)NCc2nncn2C)ccc1OC ZINC000880668437 DD On-Demand Anodyne ENPP1 70 34 COCc1cc(NC(=O)N(C)Cc2nnc3ccccn23)ccc1OC ZINC000880668438 FF On-Demand Anodyne ENPP1 55 33 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne TSHR 57 34 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne HRH2 19 40 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne ROCK2 15 41 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne PDGFRA 42 36 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne QPCT 15 44 COCc1cc(NC(=O)NCCOc2cccnc2)ccc1OC ZINC000880668439 EE On-Demand Anodyne ENPP1 49 36 COCc1cc(NC(=O)N2CCC[C@@H]2c2ccc(F)c(F)c2)ccc1OC ZINC000880668440 GI On-Demand Anodyne TSHR 54 37 COCc1cc(NC(=O)N2CCC[C@@H]2c2ccc(F)c(F)c2)ccc1OC ZINC000880668440 GI On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)ccc1OC ZINC000880668441 GI On-Demand Anodyne TSHR 54 37 COCc1cc(NC(=O)N2CCC[C@H]2c2ccc(F)c(F)c2)ccc1OC ZINC000880668441 GI On-Demand Anodyne QRFPR 43 37 COCc1cc(NC(=O)NCc2nc(C3CC3)no2)ccc1OC ZINC000880668444 EE On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NCc2nc(C3CC3)no2)ccc1OC ZINC000880668444 EE On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCc2nc(C3CC3)no2)ccc1OC ZINC000880668444 EE On-Demand Anodyne ENPP1 49 29 COCc1cc(NC(=O)NC[C@H](O)c2c(F)cccc2F)ccc1OC ZINC000880668453 FF On-Demand Anodyne TSHR 62 39 COCc1cc(NC(=O)NC[C@@H](O)c2c(F)cccc2F)ccc1OC ZINC000880668454 FF On-Demand Anodyne TSHR 62 39 COCc1cc(NC(=O)NCC[C@H](O)c2ccccc2)ccc1OC ZINC000880668458 EG On-Demand Anodyne TSHR 70 33 COCc1cc(NC(=O)NCC[C@H](O)c2ccccc2)ccc1OC ZINC000880668458 EG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NCC[C@@H](O)c2ccccc2)ccc1OC ZINC000880668459 EG On-Demand Anodyne TSHR 70 33 COCc1cc(NC(=O)NCC[C@@H](O)c2ccccc2)ccc1OC ZINC000880668459 EG On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@H](C)CCSC)ccc1OC ZINC000880668462 DG On-Demand Anodyne FPR1 30 40 COCc1cc(NC(=O)N[C@H](C)CCSC)ccc1OC ZINC000880668462 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@H](C)CCSC)ccc1OC ZINC000880668462 DG On-Demand Anodyne ENPP1 62 31 COCc1cc(NC(=O)N[C@@H](C)CCSC)ccc1OC ZINC000880668463 DG On-Demand Anodyne FPR1 30 40 COCc1cc(NC(=O)N[C@@H](C)CCSC)ccc1OC ZINC000880668463 DG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N[C@@H](C)CCSC)ccc1OC ZINC000880668463 DG On-Demand Anodyne ENPP1 62 31 CCN(CCNC(=O)Nc1ccc(OC)c(COC)c1)C(C)C ZINC000880668465 DF On-Demand Anodyne TSHR 46 31 CCN(CCNC(=O)Nc1ccc(OC)c(COC)c1)C(C)C ZINC000880668465 DF On-Demand Anodyne ENPP1 40 31 O=C(NCc1ccc(OCC(F)(F)F)nn1)c1ccccc1OC1CC1 ZINC000880668469 FF On-Demand Anodyne HCN1 42 32 O=C(NCc1ccc(OCC(F)(F)F)nn1)c1ccccc1OC1CC1 ZINC000880668469 FF On-Demand Anodyne HCN4 40 32 COCc1cc(NC(=O)Nc2ccc(CNC(=O)OC)cc2)ccc1OC ZINC000880668470 FG On-Demand Anodyne TSHR 70 36 COCc1cc(NC(=O)Nc2ccc(CNC(=O)OC)cc2)ccc1OC ZINC000880668470 FG On-Demand Anodyne ROCK2 17 44 COCc1cc(NC(=O)Nc2ccc(CNC(=O)OC)cc2)ccc1OC ZINC000880668470 FG On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)Nc2ccc(CN3CCOC3=O)cc2)ccc1OC ZINC000880668471 GG On-Demand Anodyne TSHR 71 37 COCc1cc(NC(=O)Nc2ccc(CN3CCOC3=O)cc2)ccc1OC ZINC000880668471 GG On-Demand Anodyne HTR2A 36 40 COCc1cc(NC(=O)Nc2ccc(CN3CCOC3=O)cc2)ccc1OC ZINC000880668471 GG On-Demand Anodyne CPT1A 35 40 COCc1cc(NC(=O)N2CCC3(CC2)CNC(=O)C3)ccc1OC ZINC000880668472 ED On-Demand Anodyne TSHR 48 31 COCc1cc(NC(=O)N2CCC3(CC2)CNC(=O)C3)ccc1OC ZINC000880668472 ED On-Demand Anodyne ENPP1 63 35 COCc1cc(NC(=O)NCCc2ccc(NC(=O)OC)cc2)ccc1OC ZINC000880668475 GG On-Demand Anodyne TSHR 68 35 COCc1cc(NC(=O)NCCc2ccc(NC(=O)OC)cc2)ccc1OC ZINC000880668475 GG On-Demand Anodyne NQO2 41 42 COCc1cc(NC(=O)NCCc2ccc(NC(=O)OC)cc2)ccc1OC ZINC000880668475 GG On-Demand Anodyne RAF1 26 42 COCc1cc(NC(=O)NCCc2ccc(NC(=O)OC)cc2)ccc1OC ZINC000880668475 GG On-Demand Anodyne MTNR1A 17 43 COCc1cc(NC(=O)NCCc2ccc(NC(=O)OC)cc2)ccc1OC ZINC000880668475 GG On-Demand Anodyne MTNR1B 16 42 COCc1cc(NC(=O)N[C@@H](C)COc2ccccc2)ccc1OC ZINC000880668481 EG On-Demand Anodyne ADRB1 24 42 COCc1cc(NC(=O)N[C@@H](C)COc2ccccc2)ccc1OC ZINC000880668481 EG On-Demand Anodyne TSHR 70 39 COCc1cc(NC(=O)N[C@@H](C)COc2ccccc2)ccc1OC ZINC000880668481 EG On-Demand Anodyne MTNR1B 19 45 COCc1cc(NC(=O)N[C@H](C)COc2ccccc2)ccc1OC ZINC000880668482 EG On-Demand Anodyne ADRB1 24 42 COCc1cc(NC(=O)N[C@H](C)COc2ccccc2)ccc1OC ZINC000880668482 EG On-Demand Anodyne TSHR 70 39 COCc1cc(NC(=O)N[C@H](C)COc2ccccc2)ccc1OC ZINC000880668482 EG On-Demand Anodyne MTNR1B 19 45 COCc1cc(NC(=O)N2CCC[C@@H]2C(=O)N(C)C)ccc1OC ZINC000880668485 ED On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)N2CCC[C@@H]2C(=O)N(C)C)ccc1OC ZINC000880668485 ED On-Demand Anodyne AVPR1B 41 33 COCc1cc(NC(=O)N2CCC[C@@H]2C(=O)N(C)C)ccc1OC ZINC000880668485 ED On-Demand Anodyne QRFPR 44 37 COCc1cc(NC(=O)N[C@H](C)c2ccc(C)s2)ccc1OC ZINC000880668487 EI On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N[C@@H](C)c2ccc(C)s2)ccc1OC ZINC000880668488 EI On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NCc2ccc(N3CCCC3=O)cc2)ccc1OC ZINC000880668489 GG On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NCCN(C)C(=O)OC(C)(C)C)ccc1OC ZINC000880668517 FF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCc2ncc(C)c(OC)c2C)ccc1OC ZINC000880668520 FG On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NCc2ncc(C)c(OC)c2C)ccc1OC ZINC000880668520 FG On-Demand Anodyne ENPP1 47 33 COCc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668521 GF On-Demand Anodyne ADRB2 27 46 COCc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668521 GF On-Demand Anodyne ADRB1 56 46 COCc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668521 GF On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NC[C@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668521 GF On-Demand Anodyne ADRB3 31 43 COCc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668522 GF On-Demand Anodyne ADRB2 27 46 COCc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668522 GF On-Demand Anodyne ADRB1 56 46 COCc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668522 GF On-Demand Anodyne TSHR 55 34 COCc1cc(NC(=O)NC[C@@H](O)COc2cccc(F)c2)ccc1OC ZINC000880668522 GF On-Demand Anodyne ADRB3 31 43 C=C(Br)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668523 EF On-Demand Mild TSHR 54 31 C=C(Br)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668523 EF On-Demand Mild QRFPR 41 35 C=C(Br)CNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668523 EF On-Demand Mild ENPP1 64 33 COCc1cc(NC(=O)NC[C@H](O)c2cnn(C)c2)ccc1OC ZINC000880668524 ED On-Demand Anodyne TSHR 65 32 COCc1cc(NC(=O)NC[C@H](O)c2cnn(C)c2)ccc1OC ZINC000880668524 ED On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NC[C@@H](O)c2cnn(C)c2)ccc1OC ZINC000880668525 ED On-Demand Anodyne TSHR 65 32 COCc1cc(NC(=O)NC[C@@H](O)c2cnn(C)c2)ccc1OC ZINC000880668525 ED On-Demand Anodyne ENPP1 69 33 COCc1cc(NC(=O)NCCOC2CCC2)ccc1OC ZINC000880668526 DF On-Demand Anodyne ADRB1 15 45 COCc1cc(NC(=O)NCCOC2CCC2)ccc1OC ZINC000880668526 DF On-Demand Anodyne TSHR 57 33 COCc1cc(NC(=O)NCCOC2CCC2)ccc1OC ZINC000880668526 DF On-Demand Anodyne PDE4A 22 42 COCc1cc(NC(=O)NCCOC2CCC2)ccc1OC ZINC000880668526 DF On-Demand Anodyne QRFPR 47 39 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668540 GG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668540 GG On-Demand Anodyne ADRB3 43 38 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668540 GG On-Demand Anodyne F7 20 43 COCc1cc(NC(=O)NC[C@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668540 GG On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668541 GG On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668541 GG On-Demand Anodyne ADRB3 43 38 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668541 GG On-Demand Anodyne F7 20 43 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(OC(C)C)c2)ccc1OC ZINC000880668541 GG On-Demand Anodyne ENPP1 62 33 COCc1cc(NC(=O)N2CC[C@@](F)(C(=O)OC)C2)ccc1OC ZINC000880668549 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@@](F)(C(=O)OC)C2)ccc1OC ZINC000880668549 ED On-Demand Anodyne EPHX2 31 41 COCc1cc(NC(=O)N2CC[C@@](F)(C(=O)OC)C2)ccc1OC ZINC000880668549 ED On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)N2CC[C@](F)(C(=O)OC)C2)ccc1OC ZINC000880668550 ED On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CC[C@](F)(C(=O)OC)C2)ccc1OC ZINC000880668550 ED On-Demand Anodyne EPHX2 31 41 COCc1cc(NC(=O)N2CC[C@](F)(C(=O)OC)C2)ccc1OC ZINC000880668550 ED On-Demand Anodyne ENPP1 40 31 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne HTR4 50 44 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne CCR3 32 42 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne EPHX2 51 40 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne CXCR3 18 40 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne MCHR1 19 42 COCc1cc(NC(=O)NC2CCN(CCS(C)(=O)=O)CC2)ccc1OC ZINC000880668553 GD On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)N2CCC[C@H]2CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668562 GG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC[C@H]2CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668562 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N2CCC[C@@H]2CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668563 GG On-Demand Anodyne TSHR 47 31 COCc1cc(NC(=O)N2CCC[C@@H]2CNC(=O)OC(C)(C)C)ccc1OC ZINC000880668563 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N(C)[C@@H]2CCN(CC(F)(F)F)C2=O)ccc1OC ZINC000880668565 GE On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N(C)[C@H]2CCN(CC(F)(F)F)C2=O)ccc1OC ZINC000880668566 GE On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NC[C@@H](O)c2cc(OC)cc(OC)c2)ccc1OC ZINC000880668567 GF On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)NC[C@@H](O)c2cc(OC)cc(OC)c2)ccc1OC ZINC000880668567 GF On-Demand Anodyne ENPP1 66 32 COCc1cc(NC(=O)NC[C@H](O)c2cc(OC)cc(OC)c2)ccc1OC ZINC000880668568 GF On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)NC[C@H](O)c2cc(OC)cc(OC)c2)ccc1OC ZINC000880668568 GF On-Demand Anodyne ENPP1 66 32 COCc1cc(NC(=O)N2CCC[C@H]2c2cccc(N(C)C)c2)ccc1OC ZINC000880668571 GI On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC[C@H]2c2cccc(N(C)C)c2)ccc1OC ZINC000880668571 GI On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC[C@@H]2c2cccc(N(C)C)c2)ccc1OC ZINC000880668572 GI On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC[C@@H]2c2cccc(N(C)C)c2)ccc1OC ZINC000880668572 GI On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC3(C2)OCCO3)ccc1OC ZINC000880668577 DD On-Demand Anodyne TSHR 62 33 COCc1cc(NC(=O)N2CCC3(C2)OCCO3)ccc1OC ZINC000880668577 DD On-Demand Anodyne PDGFRB 38 40 COCc1cc(NC(=O)N2CCC3(C2)OCCO3)ccc1OC ZINC000880668577 DD On-Demand Anodyne EPHX2 33 45 COCc1cc(NC(=O)N2CCN(C(=O)OCC(C)C)CC2)ccc1OC ZINC000880668578 GF On-Demand Anodyne PDGFRB 46 40 COCc1cc(NC(=O)N2CCN(C(=O)OCC(C)C)CC2)ccc1OC ZINC000880668578 GF On-Demand Anodyne ENPP1 68 33 COCc1cc(NC(=O)NC[C@](C)(O)c2ccccc2)ccc1OC ZINC000880668581 EF On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccccc2)ccc1OC ZINC000880668582 EF On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCc3c(C)cccc3C2)ccc1OC ZINC000880668586 EH On-Demand Anodyne HTR1B 15 47 COCc1cc(NC(=O)N2CCc3c(C)cccc3C2)ccc1OC ZINC000880668586 EH On-Demand Anodyne P2RY14 52 38 COCc1cc(NC(=O)NCCCN2CCOC2=O)ccc1OC ZINC000880668588 ED On-Demand Anodyne TSHR 52 32 COCc1cc(NC(=O)NCCCN2CCOC2=O)ccc1OC ZINC000880668588 ED On-Demand Anodyne QPCT 28 46 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C)o2)ccc1OC ZINC000880668591 EF On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NC[C@H](O)c2ccc(C)o2)ccc1OC ZINC000880668591 EF On-Demand Anodyne ENPP1 60 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C)o2)ccc1OC ZINC000880668592 EF On-Demand Anodyne TSHR 56 33 COCc1cc(NC(=O)NC[C@@H](O)c2ccc(C)o2)ccc1OC ZINC000880668592 EF On-Demand Anodyne ENPP1 60 33 COCc1cc(NC(=O)NCCSC(F)(F)F)ccc1OC ZINC000880668598 EG On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)NCCSC(F)(F)F)ccc1OC ZINC000880668598 EG On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NCCSC(F)(F)F)ccc1OC ZINC000880668598 EG On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne ADRB2 41 40 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne ADRB1 47 46 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne HTR2A 19 41 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne ADRB3 64 46 COCc1cc(NC(=O)NC[C@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668611 FG On-Demand Anodyne ENPP1 55 34 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne ADRB2 41 40 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne ADRB1 47 46 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne HTR2A 19 41 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne ADRB3 64 46 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(Cl)c2)ccc1OC ZINC000880668612 FG On-Demand Anodyne ENPP1 55 34 COCc1cc(NC(=O)N[C@@H](CCO)c2cccs2)ccc1OC ZINC000880668615 FG On-Demand Anodyne QRFPR 35 40 COCc1cc(NC(=O)N[C@H](CCO)c2cccs2)ccc1OC ZINC000880668616 FG On-Demand Anodyne QRFPR 35 40 COCc1cc(NC(=O)N(C)CCOc2ccccc2OC)ccc1OC ZINC000880668619 FG On-Demand Anodyne TSHR 56 34 COCc1cc(NC(=O)N(C)CCOc2ccccc2OC)ccc1OC ZINC000880668619 FG On-Demand Anodyne ENPP1 57 33 COCc1cc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668627 GF On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668627 GF On-Demand Anodyne OPRK1 20 41 COCc1cc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668627 GF On-Demand Anodyne PDGFRB 51 40 COCc1cc(NC(=O)N2CCN(C[C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668627 GF On-Demand Anodyne ABCB1 23 43 COCc1cc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668628 GF On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668628 GF On-Demand Anodyne OPRK1 20 41 COCc1cc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668628 GF On-Demand Anodyne PDGFRB 51 40 COCc1cc(NC(=O)N2CCN(C[C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880668628 GF On-Demand Anodyne ABCB1 23 43 COCc1cc(NC(=O)N2CCO[C@H](c3ccc(F)c(F)c3)C2)ccc1OC ZINC000880668630 GH On-Demand Anodyne TSHR 43 34 COCc1cc(NC(=O)N2CCO[C@@H](c3ccc(F)c(F)c3)C2)ccc1OC ZINC000880668631 GH On-Demand Anodyne TSHR 43 34 COCc1cc(NC(=O)N[C@H](CO)C2CC2)ccc1OC ZINC000880668640 CD On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N[C@H](CO)C2CC2)ccc1OC ZINC000880668640 CD On-Demand Anodyne QRFPR 46 39 COCc1cc(NC(=O)N[C@H](CO)C2CC2)ccc1OC ZINC000880668640 CD On-Demand Anodyne ENPP1 68 32 COCc1cc(NC(=O)N[C@@H](CO)C2CC2)ccc1OC ZINC000880668641 CD On-Demand Anodyne TSHR 41 30 COCc1cc(NC(=O)N[C@@H](CO)C2CC2)ccc1OC ZINC000880668641 CD On-Demand Anodyne QRFPR 46 39 COCc1cc(NC(=O)N[C@@H](CO)C2CC2)ccc1OC ZINC000880668641 CD On-Demand Anodyne ENPP1 68 32 COCc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ccc1OC ZINC000880668645 GG On-Demand Anodyne TSHR 65 32 COCc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ccc1OC ZINC000880668645 GG On-Demand Anodyne ROCK2 17 41 COCc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ccc1OC ZINC000880668645 GG On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)NCc2ccc(C(=O)N3CCCC3)cc2)ccc1OC ZINC000880668645 GG On-Demand Anodyne NAMPT 21 50 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2C)ccc1OC ZINC000880668646 EG On-Demand Anodyne ADRB2 22 40 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2C)ccc1OC ZINC000880668646 EG On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2C)ccc1OC ZINC000880668647 EG On-Demand Anodyne ADRB2 22 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2C)ccc1OC ZINC000880668647 EG On-Demand Anodyne TSHR 71 35 COCc1cc(NC(=O)N(C)Cc2cnn(-c3ccccc3)n2)ccc1OC ZINC000880668656 GG On-Demand Anodyne TSHR 55 35 COCc1cc(NC(=O)N(C)Cc2nc(O)c3ccccc3n2)ccc1OC ZINC000880668662 GG On-Demand Anodyne TSHR 54 42 COCc1cc(NC(=O)N(C)Cc2nc(O)c3ccccc3n2)ccc1OC ZINC000880668662 GG On-Demand Anodyne ENPP1 45 30 COCc1cc(NC(=O)Nc2ccc(CN(C)C(=O)OC)cc2)ccc1OC ZINC000880668665 GH On-Demand Anodyne TSHR 54 33 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne TSHR 56 35 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne HTR2A 26 40 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne CA1 32 43 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne CA12 22 43 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne CA9 20 43 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne QRFPR 41 34 CCOC(=O)Nc1ccc(NC(=O)Nc2ccc(OC)c(COC)c2)cc1 ZINC000880668674 FI On-Demand Anodyne ENPP1 68 34 COCc1cc(NC(=O)NCc2cccnc2-n2ccnc2C)ccc1OC ZINC000880668682 GG On-Demand Anodyne TSHR 63 34 COCc1cc(NC(=O)NCc2cccnc2-n2ccnc2C)ccc1OC ZINC000880668682 GG On-Demand Anodyne ROCK2 15 40 COCc1cc(NC(=O)NCc2cccnc2-n2ccnc2C)ccc1OC ZINC000880668682 GG On-Demand Anodyne ENPP1 41 36 COCc1cc(NC(=O)NC[C@H]2COc3ccccc3C2)ccc1OC ZINC000880668686 FG On-Demand Anodyne TSHR 59 30 COCc1cc(NC(=O)NC[C@H]2COc3ccccc3C2)ccc1OC ZINC000880668686 FG On-Demand Anodyne ROCK2 15 43 COCc1cc(NC(=O)NC[C@H]2COc3ccccc3C2)ccc1OC ZINC000880668686 FG On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)NC[C@@H]2COc3ccccc3C2)ccc1OC ZINC000880668687 FG On-Demand Anodyne TSHR 59 30 COCc1cc(NC(=O)NC[C@@H]2COc3ccccc3C2)ccc1OC ZINC000880668687 FG On-Demand Anodyne ROCK2 15 43 COCc1cc(NC(=O)NC[C@@H]2COc3ccccc3C2)ccc1OC ZINC000880668687 FG On-Demand Anodyne QRFPR 44 38 COCc1cc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)ccc1OC ZINC000880668692 GF On-Demand Anodyne CCR3 26 41 COCc1cc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)ccc1OC ZINC000880668692 GF On-Demand Anodyne EPHX2 43 40 COCc1cc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)ccc1OC ZINC000880668692 GF On-Demand Anodyne CXCR3 19 41 COCc1cc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)ccc1OC ZINC000880668692 GF On-Demand Anodyne MCHR1 16 43 COCc1cc(NC(=O)NC2CCN(C[C@H]3CCCO3)CC2)ccc1OC ZINC000880668692 GF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)ccc1OC ZINC000880668693 GF On-Demand Anodyne CCR3 26 41 COCc1cc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)ccc1OC ZINC000880668693 GF On-Demand Anodyne EPHX2 43 40 COCc1cc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)ccc1OC ZINC000880668693 GF On-Demand Anodyne CXCR3 19 41 COCc1cc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)ccc1OC ZINC000880668693 GF On-Demand Anodyne MCHR1 16 43 COCc1cc(NC(=O)NC2CCN(C[C@@H]3CCCO3)CC2)ccc1OC ZINC000880668693 GF On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC[C@H](C)CC2(C)OCCO2)ccc1OC ZINC000880668706 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)NC[C@@H](C)CC2(C)OCCO2)ccc1OC ZINC000880668707 FF On-Demand Anodyne TSHR 40 29 COCc1cc(NC(=O)NCC(=O)OC(C)C)ccc1OC ZINC000880668708 DD On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)NCC(=O)OC(C)C)ccc1OC ZINC000880668708 DD On-Demand Anodyne ENPP1 71 35 COCc1cc(NC(=O)N2CCC3(CCCC3)C2)ccc1OC ZINC000880668712 DH On-Demand Anodyne TSHR 52 30 COCc1cc(NC(=O)N2CCC3(CCCC3)C2)ccc1OC ZINC000880668712 DH On-Demand Anodyne EPHX2 38 45 COCc1cc(NC(=O)N2CCC3(CCCC3)C2)ccc1OC ZINC000880668712 DH On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCC3(CCCC3)C2)ccc1OC ZINC000880668712 DH On-Demand Anodyne ENPP1 63 34 COCc1cc(NC(=O)NCC[S@@](=O)C(C)(C)C)ccc1OC ZINC000880668713 EF On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NCC[S@](=O)C(C)(C)C)ccc1OC ZINC000880668714 EF On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)NCCNC(=O)OC(C)(C)C)ccc1OC ZINC000880668715 FE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)NCCNC(=O)OC(C)(C)C)ccc1OC ZINC000880668715 FE On-Demand Anodyne QRFPR 42 34 COCc1cc(NC(=O)NCCc2nnc3ccccn23)ccc1OC ZINC000880668716 FE On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCCc2nnc3ccccn23)ccc1OC ZINC000880668716 FE On-Demand Anodyne QPCT 15 43 COCc1cc(NC(=O)NCCc2nnc3ccccn23)ccc1OC ZINC000880668716 FE On-Demand Anodyne PRMT3 51 34 COCc1cc(NC(=O)NCCc2nnc3ccccn23)ccc1OC ZINC000880668716 FE On-Demand Anodyne ENPP1 56 33 COCc1cc(NC(=O)NCc2nnc(S)n2C)ccc1OC ZINC000880668723 ED On-Demand Anodyne TSHR 54 32 COCc1cc(NC(=O)NCc2nnc(S)n2C)ccc1OC ZINC000880668723 ED On-Demand Anodyne PRMT3 44 32 COCc1cc(NC(=O)NCc2nnc(S)n2C)ccc1OC ZINC000880668723 ED On-Demand Anodyne ENPP1 69 32 COCc1cc(NC(=O)NCCS(C)(=O)=O)ccc1OC ZINC000880668724 DD On-Demand Anodyne TSHR 53 30 COCc1cc(NC(=O)NCCS(C)(=O)=O)ccc1OC ZINC000880668724 DD On-Demand Anodyne QRFPR 41 35 COCc1cc(NC(=O)NCCS(C)(=O)=O)ccc1OC ZINC000880668724 DD On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)NC[C@](C)(O)c2ccco2)ccc1OC ZINC000880668726 EE On-Demand Anodyne TSHR 41 34 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccco2)ccc1OC ZINC000880668727 EE On-Demand Anodyne TSHR 41 34 COCc1cc(NC(=O)NCC(=O)OC2CCCCC2)ccc1OC ZINC000880668737 FF On-Demand Anodyne TSHR 62 34 COCc1cc(NC(=O)NCC(=O)OC2CCCCC2)ccc1OC ZINC000880668737 FF On-Demand Anodyne QRFPR 49 40 COCc1cc(NC(=O)NCC(=O)OC2CCCCC2)ccc1OC ZINC000880668737 FF On-Demand Anodyne PRMT3 50 39 COCc1cc(NC(=O)NCC(=O)OC2CCCCC2)ccc1OC ZINC000880668737 FF On-Demand Anodyne ENPP1 44 30 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668740 FD On-Demand Anodyne PDGFRB 49 40 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668740 FD On-Demand Anodyne F13A1 49 39 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668740 FD On-Demand Anodyne QRFPR 43 35 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668740 FD On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)Nc2cccc(CN3CCOC3=O)c2)ccc1OC ZINC000880668744 GG On-Demand Anodyne TSHR 70 35 COCc1cc(NC(=O)NC[C@@H](OC)C(F)(F)F)ccc1OC ZINC000880668745 EF On-Demand Anodyne TSHR 53 32 COCc1cc(NC(=O)NC[C@H](OC)C(F)(F)F)ccc1OC ZINC000880668746 EF On-Demand Anodyne TSHR 53 32 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668747 GF On-Demand Anodyne TSHR 46 31 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668747 GF On-Demand Anodyne HTR1B 15 41 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880668747 GF On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NC[C@](C)(O)c2ccc(F)cc2F)ccc1OC ZINC000880668760 GG On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NC[C@@](C)(O)c2ccc(F)cc2F)ccc1OC ZINC000880668761 GG On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)N2CCC(C3OCCO3)CC2)ccc1OC ZINC000880668764 FE On-Demand Anodyne TSHR 54 31 COCc1cc(NC(=O)N2CCC(C3OCCO3)CC2)ccc1OC ZINC000880668764 FE On-Demand Anodyne HTR1D 15 45 COCc1cc(NC(=O)N2CCC(C3OCCO3)CC2)ccc1OC ZINC000880668764 FE On-Demand Anodyne HTR1B 18 45 COCc1cc(NC(=O)N2CCC(C3OCCO3)CC2)ccc1OC ZINC000880668764 FE On-Demand Anodyne PDGFRB 41 35 COCc1cc(NC(=O)N2CCC(C3OCCO3)CC2)ccc1OC ZINC000880668764 FE On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCC[C@@H](C3OCCO3)C2)ccc1OC ZINC000880668765 FE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC[C@@H](C3OCCO3)C2)ccc1OC ZINC000880668765 FE On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCC[C@H](C3OCCO3)C2)ccc1OC ZINC000880668766 FE On-Demand Anodyne TSHR 53 31 COCc1cc(NC(=O)N2CCC[C@H](C3OCCO3)C2)ccc1OC ZINC000880668766 FE On-Demand Anodyne QRFPR 46 38 O=C(CCc1cncc2ccccc12)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668774 GG On-Demand Anodyne SUCNR1 46 37 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean TSHR 66 32 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean PIK3CA 32 41 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean ROCK2 15 41 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean MTOR 64 38 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean EPHX2 24 41 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean STAT6 54 41 COCc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880668775 GF On-Demand Clean NAMPT 23 40 COCc1cc(NC(=O)N(C)Cc2ccccc2O)ccc1OC ZINC000880668777 EG On-Demand Clean TSHR 62 35 COCc1cc(NC(=O)N(C)Cc2ccccc2O)ccc1OC ZINC000880668777 EG On-Demand Clean QRFPR 40 35 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668779 GH On-Demand Anodyne TSHR 72 36 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668779 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668779 GH On-Demand Anodyne Q8WSF8_APLCA 21 40 COCc1cc(NC(=O)N2CCC[C@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668779 GH On-Demand Anodyne ACKR3 64 35 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668780 GH On-Demand Anodyne TSHR 72 36 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668780 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668780 GH On-Demand Anodyne Q8WSF8_APLCA 21 40 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@H](O)c2ccccc2)ccc1OC ZINC000880668780 GH On-Demand Anodyne ACKR3 64 35 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668781 GH On-Demand Anodyne TSHR 72 36 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668781 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668781 GH On-Demand Anodyne Q8WSF8_APLCA 21 40 COCc1cc(NC(=O)N2CCC[C@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668781 GH On-Demand Anodyne ACKR3 64 35 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668782 GH On-Demand Anodyne TSHR 72 36 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668782 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668782 GH On-Demand Anodyne Q8WSF8_APLCA 21 40 COCc1cc(NC(=O)N2CCC[C@@H]2C[C@@H](O)c2ccccc2)ccc1OC ZINC000880668782 GH On-Demand Anodyne ACKR3 64 35 COCc1cc(NC(=O)N2CCC[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668786 GG On-Demand Anodyne TSHR 49 33 COCc1cc(NC(=O)N2CCC[C@H](NC(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668786 GG On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668796 GI On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668796 GI On-Demand Anodyne PDE4A 15 40 COCc1cc(NC(=O)N[C@@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668796 GI On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668797 GI On-Demand Anodyne TSHR 67 33 COCc1cc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668797 GI On-Demand Anodyne PDE4A 15 40 COCc1cc(NC(=O)N[C@H](c2ccccc2)C2CCOCC2)ccc1OC ZINC000880668797 GI On-Demand Anodyne QRFPR 42 39 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(COC)c2)CCO1 ZINC000880668800 FD On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)NCc2nc(Cc3ccccc3)no2)ccc1OC ZINC000880668802 GG On-Demand Anodyne TSHR 73 36 COCc1cc(NC(=O)NCc2nc(Cc3ccccc3)no2)ccc1OC ZINC000880668802 GG On-Demand Anodyne ENPP1 49 30 O=C(CCCc1ccsc1)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668811 FG On-Demand Anodyne SUCNR1 53 38 COCc1cc(NC(=O)NCC(C)(C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880668816 GG On-Demand Anodyne TSHR 47 30 COCc1cc(NC(=O)NCC(C)(C)NC(=O)OC(C)(C)C)ccc1OC ZINC000880668816 GG On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)N[C@H](C)Cc2ccco2)ccc1OC ZINC000880668821 DG On-Demand Anodyne TSHR 19 40 COCc1cc(NC(=O)N[C@@H](C)Cc2ccco2)ccc1OC ZINC000880668822 DG On-Demand Anodyne TSHR 19 40 COCc1cc(NC(=O)N2CCC(NC(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668825 GG On-Demand Anodyne TSHR 41 31 COCc1cc(NC(=O)N2CCC(NC(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880668825 GG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean TSHR 66 37 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean CA1 15 42 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean MTNR1A 40 43 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean MTNR1B 39 43 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean QRFPR 40 33 COCc1cc(NC(=O)NCc2cc(OC)ccc2O)ccc1OC ZINC000880668826 EF On-Demand Clean PRMT3 50 32 COCc1cc(NC(=O)NC[C@](C)(O)c2cccs2)ccc1OC ZINC000880668828 FF On-Demand Anodyne QRFPR 42 40 COCc1cc(NC(=O)NC[C@@](C)(O)c2cccs2)ccc1OC ZINC000880668829 FF On-Demand Anodyne QRFPR 42 40 COCc1cc(NC(=O)NCc2ccc(OCC#N)cc2)ccc1OC ZINC000880668833 FG On-Demand Mild TSHR 63 37 COCc1cc(NC(=O)NCc2ccc(OCC#N)cc2)ccc1OC ZINC000880668833 FG On-Demand Mild ROCK2 19 42 C#CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668834 BD On-Demand Mild TSHR 55 32 C#CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668834 BD On-Demand Mild QRFPR 45 37 C#CCNC(=O)Nc1ccc(OC)c(COC)c1 ZINC000880668834 BD On-Demand Mild ENPP1 56 31 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2C(F)(F)F)ccc1OC ZINC000880668846 GH On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2C(F)(F)F)ccc1OC ZINC000880668846 GH On-Demand Anodyne SOAT1 20 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2C(F)(F)F)ccc1OC ZINC000880668847 GH On-Demand Anodyne TSHR 66 32 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2C(F)(F)F)ccc1OC ZINC000880668847 GH On-Demand Anodyne SOAT1 20 40 COCc1cc(NC(=O)N[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668848 FE On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668848 FE On-Demand Anodyne CCR3 21 41 COCc1cc(NC(=O)N[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668848 FE On-Demand Anodyne EPHX2 47 40 COCc1cc(NC(=O)N[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668848 FE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668848 FE On-Demand Anodyne ENPP1 67 31 COCc1cc(NC(=O)N[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668849 FE On-Demand Anodyne TSHR 61 33 COCc1cc(NC(=O)N[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668849 FE On-Demand Anodyne CCR3 21 41 COCc1cc(NC(=O)N[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668849 FE On-Demand Anodyne EPHX2 47 40 COCc1cc(NC(=O)N[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668849 FE On-Demand Anodyne QRFPR 44 36 COCc1cc(NC(=O)N[C@@H]2CCCN(C(=O)OC)C2)ccc1OC ZINC000880668849 FE On-Demand Anodyne ENPP1 67 31 CCn1c(CNC(=O)Nc2ccc(OC)c(COC)c2)nc2ccccc21 ZINC000880668850 FH On-Demand Anodyne TSHR 74 37 CCn1c(CNC(=O)Nc2ccc(OC)c(COC)c2)nc2ccccc21 ZINC000880668850 FH On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)ccc1OC ZINC000880668854 GF On-Demand Anodyne TSHR 73 36 COCc1cc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)ccc1OC ZINC000880668854 GF On-Demand Anodyne CA1 34 42 COCc1cc(NC(=O)NCCS(=O)(=O)Cc2ccccc2)ccc1OC ZINC000880668854 GF On-Demand Anodyne CCR3 15 42 COCc1cc(NC(=O)NC[C@H](O)c2cccc(F)c2)ccc1OC ZINC000880668855 EF On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)NC[C@H](O)c2cccc(F)c2)ccc1OC ZINC000880668855 EF On-Demand Anodyne HTR2A 15 41 COCc1cc(NC(=O)NC[C@H](O)c2cccc(F)c2)ccc1OC ZINC000880668855 EF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(F)c2)ccc1OC ZINC000880668856 EF On-Demand Anodyne TSHR 61 34 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(F)c2)ccc1OC ZINC000880668856 EF On-Demand Anodyne HTR2A 15 41 COCc1cc(NC(=O)NC[C@@H](O)c2cccc(F)c2)ccc1OC ZINC000880668856 EF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)N[C@H]2CCCc3nc(C)ncc32)ccc1OC ZINC000880668860 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N[C@H]2CCCc3nc(C)ncc32)ccc1OC ZINC000880668860 FG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)N[C@@H]2CCCc3nc(C)ncc32)ccc1OC ZINC000880668861 FG On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N[C@@H]2CCCc3nc(C)ncc32)ccc1OC ZINC000880668861 FG On-Demand Anodyne QRFPR 43 36 COCc1cc(NC(=O)NC2CCC3(CC2)OCCO3)ccc1OC ZINC000880668864 FF On-Demand Anodyne TSHR 60 32 COCc1cc(NC(=O)NC2CCC3(CC2)OCCO3)ccc1OC ZINC000880668864 FF On-Demand Anodyne EPHX2 44 37 COCc1cc(NC(=O)NC2CCC3(CC2)OCCO3)ccc1OC ZINC000880668864 FF On-Demand Anodyne QRFPR 43 35 O=C(CCc1cccc2ccccc12)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880668867 GH On-Demand Anodyne SUCNR1 56 38 COCc1cc(NC(=O)N(C)Cc2cccc(C(N)=O)c2)ccc1OC ZINC000880668869 FF On-Demand Anodyne TSHR 42 32 COCc1cc(NC(=O)N(C)Cc2cccc(C(N)=O)c2)ccc1OC ZINC000880668869 FF On-Demand Anodyne ROCK2 18 43 COCc1cc(NC(=O)N(C)Cc2cccc(C(N)=O)c2)ccc1OC ZINC000880668869 FF On-Demand Anodyne ENPP1 54 30 COCc1cc(NC(=O)N(C)Cc2c(C)noc2C)ccc1OC ZINC000880668873 EG On-Demand Anodyne TSHR 42 33 COCc1cc(NC(=O)NCc2cccc(OC)c2O)ccc1OC ZINC000880668876 EF On-Demand Clean TSHR 70 36 COCc1cc(NC(=O)NCc2cccc(OC)c2O)ccc1OC ZINC000880668876 EF On-Demand Clean ROCK2 22 48 COCc1cc(NC(=O)NCc2cccc(OC)c2O)ccc1OC ZINC000880668876 EF On-Demand Clean QRFPR 40 33 COCc1cc(NC(=O)NCc2cccc(OC)c2O)ccc1OC ZINC000880668876 EF On-Demand Clean ENPP1 49 31 COCc1cc(NC(=O)NC[C@H](O)c2c(F)cccc2Cl)ccc1OC ZINC000880668878 GG On-Demand Anodyne TSHR 62 38 COCc1cc(NC(=O)NC[C@@H](O)c2c(F)cccc2Cl)ccc1OC ZINC000880668879 GG On-Demand Anodyne TSHR 62 38 COCc1cc(NC(=O)N[C@@H](C)[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668881 FG On-Demand Anodyne HTR2A 16 44 COCc1cc(NC(=O)N[C@@H](C)[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668881 FG On-Demand Anodyne ENPP1 61 31 COCc1cc(NC(=O)N[C@H](C)[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668882 FG On-Demand Anodyne HTR2A 16 44 COCc1cc(NC(=O)N[C@H](C)[C@@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668882 FG On-Demand Anodyne ENPP1 61 31 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668883 FG On-Demand Anodyne HTR2A 16 44 COCc1cc(NC(=O)N[C@@H](C)[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668883 FG On-Demand Anodyne ENPP1 61 31 COCc1cc(NC(=O)N[C@H](C)[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668884 FG On-Demand Anodyne HTR2A 16 44 COCc1cc(NC(=O)N[C@H](C)[C@H](O)c2ccc(F)cc2)ccc1OC ZINC000880668884 FG On-Demand Anodyne ENPP1 61 31 COCc1cc(NC(=O)NCc2ccc(-n3ccnc3C)nc2)ccc1OC ZINC000880668885 GG On-Demand Anodyne TSHR 56 36 COCc1cc(NC(=O)NCc2ccc(-n3ccnc3C)nc2)ccc1OC ZINC000880668885 GG On-Demand Anodyne ROCK2 15 41 COCc1cc(NC(=O)NCc2ccc(-n3ccnc3C)nc2)ccc1OC ZINC000880668885 GG On-Demand Anodyne ENPP1 41 32 COCc1cc(NC(=O)NCc2ccc(-n3ccnc3C)nc2)ccc1OC ZINC000880668885 GG On-Demand Anodyne NAMPT 32 42 COCc1cc(NC(=O)NCc2c(OC)cc(OC)cc2OC)ccc1OC ZINC000880668889 GG On-Demand Anodyne TSHR 69 33 COCc1cc(NC(=O)NCc2c(OC)cc(OC)cc2OC)ccc1OC ZINC000880668889 GG On-Demand Anodyne ROCK2 15 48 COCc1cc(NC(=O)NCc2c(OC)cc(OC)cc2OC)ccc1OC ZINC000880668889 GG On-Demand Anodyne ENPP1 55 31 COCc1cc(NC(=O)N(C)[C@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668891 GG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)N(C)[C@@H]2CCN(C(=O)OC(C)(C)C)C2)ccc1OC ZINC000880668892 GG On-Demand Anodyne QRFPR 41 34 COCc1cc(NC(=O)NCCC[S@](C)=O)ccc1OC ZINC000880668897 DD On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NCCC[S@](C)=O)ccc1OC ZINC000880668897 DD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCC[S@@](C)=O)ccc1OC ZINC000880668898 DD On-Demand Anodyne TSHR 69 34 COCc1cc(NC(=O)NCCC[S@@](C)=O)ccc1OC ZINC000880668898 DD On-Demand Anodyne QRFPR 40 33 COCc1cc(NC(=O)NCCn2cncn2)ccc1OC ZINC000880668901 DD On-Demand Anodyne TSHR 52 31 COCc1cc(NC(=O)NCCn2cncn2)ccc1OC ZINC000880668901 DD On-Demand Anodyne QPCT 22 49 COCc1cc(NC(=O)NCCn2cncn2)ccc1OC ZINC000880668901 DD On-Demand Anodyne ENPP1 71 36 COCc1cc(NC(=O)NCCCNC(=O)OC(C)(C)C)ccc1OC ZINC000880668905 FF On-Demand Anodyne TSHR 47 32 COCc1cc(NC(=O)NCCCNC(=O)OC(C)(C)C)ccc1OC ZINC000880668905 FF On-Demand Anodyne QRFPR 41 33 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean TSHR 58 35 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean CCR3 18 41 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean EPHX2 53 43 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean PDGFRA 18 40 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean PDK1 44 31 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean CXCR3 15 41 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean MCHR1 26 43 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean QRFPR 41 34 COCc1cc(NC(=O)NC2CCN(c3ccc(OC)cc3)CC2)ccc1OC ZINC000880668910 GH On-Demand Clean ENPP1 44 30 C[C@@H]1CN(CCNC(=O)c2cc3ccccc3cc2F)[C@H](C)CO1 ZINC000880668943 EF On-Demand Anodyne POLR1A 58 34 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880668958 GE On-Demand Anodyne CACNA1H 50 38 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880668958 GE On-Demand Anodyne EPHX2 36 43 C=CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880668984 CE On-Demand Mild NQO2 42 44 C=CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880668984 CE On-Demand Mild MTNR1A 77 45 C=CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880668984 CE On-Demand Mild MTNR1B 65 43 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)n1 ZINC000880668985 DB On-Demand Anodyne SIGMAR1 22 44 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)n1 ZINC000880668985 DB On-Demand Anodyne MLNR 60 37 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)n1 ZINC000880668985 DB On-Demand Anodyne HSP90AA1 16 43 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)n1 ZINC000880668985 DB On-Demand Anodyne MCHR1 23 42 C=CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880668986 CE On-Demand Mild NQO2 42 44 C=CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880668986 CE On-Demand Mild MTNR1A 77 45 C=CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880668986 CE On-Demand Mild MTNR1B 65 43 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)n1 ZINC000880668987 DB On-Demand Anodyne SIGMAR1 22 44 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)n1 ZINC000880668987 DB On-Demand Anodyne MLNR 60 37 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)n1 ZINC000880668987 DB On-Demand Anodyne HSP90AA1 16 43 Cn1nnc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)n1 ZINC000880668987 DB On-Demand Anodyne MCHR1 23 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880668999 GE On-Demand Anodyne GABRA1 17 57 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880668999 GE On-Demand Anodyne CCR3 49 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880668999 GE On-Demand Anodyne MLNR 54 36 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880668999 GE On-Demand Anodyne MCHR1 18 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880669000 GE On-Demand Anodyne GABRA1 17 57 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880669000 GE On-Demand Anodyne CCR3 49 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880669000 GE On-Demand Anodyne MLNR 54 36 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880669000 GE On-Demand Anodyne MCHR1 18 41 CO[C@]1(CO)CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880669005 GD On-Demand Anodyne CELA1 18 41 CO[C@]1(CO)CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880669005 GD On-Demand Anodyne PREP 65 49 CO[C@]1(CO)CCCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880669005 GD On-Demand Anodyne SLC12A5 73 41 C[C@@H](CCNC(=O)[C@@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669028 EE On-Demand Anodyne CHRNA3 23 40 C[C@@H](CCNC(=O)[C@@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669028 EE On-Demand Anodyne CHRNA4 18 40 C[C@H](CCNC(=O)[C@@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669030 EE On-Demand Anodyne CHRNA3 23 40 C[C@H](CCNC(=O)[C@@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669030 EE On-Demand Anodyne CHRNA4 18 40 C[C@@H](CCNC(=O)[C@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669032 EE On-Demand Anodyne CHRNA3 23 40 C[C@@H](CCNC(=O)[C@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669032 EE On-Demand Anodyne CHRNA4 18 40 C[C@H](CCNC(=O)[C@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669033 EE On-Demand Anodyne CHRNA3 23 40 C[C@H](CCNC(=O)[C@H]1CN(C(=O)OC(C)(C)C)CC1(C)C)N(C)C ZINC000880669033 EE On-Demand Anodyne CHRNA4 18 40 COCC1CC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880669037 FH On-Demand Anodyne EPHX2 44 41 O=C(COC1CC1)N1CCc2ccc(Cl)c(Cl)c2C1 ZINC000880669045 DG On-Demand Anodyne PNMT 15 48 COCc1cc(NC(=O)N2CCC(C(=O)NCC(C)C)CC2)ccc1OC ZINC000880669051 GF On-Demand Anodyne TSHR 40 30 COCc1cc(NC(=O)N2CCC(C(=O)NCC(C)C)CC2)ccc1OC ZINC000880669051 GF On-Demand Anodyne EPHX2 18 41 COCc1cc(NC(=O)N2CCC(C(=O)NCC(C)C)CC2)ccc1OC ZINC000880669051 GF On-Demand Anodyne QRFPR 42 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1F ZINC000880669053 GF On-Demand Anodyne CACNA1H 54 40 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1F ZINC000880669053 GF On-Demand Anodyne NPY5R 27 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(CO)(CO)CC2)ccc1F ZINC000880669053 GF On-Demand Anodyne EPHX2 34 41 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne HTR1B 15 44 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne PDGFRB 45 38 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne PDE4A 17 45 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne NPY2R 61 34 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669063 GH On-Demand Anodyne ENPP1 67 34 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne TSHR 71 34 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne HTR1B 15 44 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne PDGFRB 45 38 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne PDE4A 17 45 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne NPY2R 61 34 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne QRFPR 42 39 COCc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)ccc1OC ZINC000880669064 GH On-Demand Anodyne ENPP1 67 34 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne TSHR 48 33 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne HTR1D 15 47 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne HTR1B 19 47 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne P2RY12 35 40 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne PDGFRB 51 46 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne TGM2 24 40 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne F13A1 42 40 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne QRFPR 41 34 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880669083 FE On-Demand Anodyne ENPP1 72 35 C[C@@H]1CN(CCNC(=O)CC[C@H]2CCc3ccccc32)[C@H](C)CO1 ZINC000880669124 EF On-Demand Anodyne NQO2 18 41 C[C@@H]1CN(CCNC(=O)CC[C@@H]2CCc3ccccc32)[C@H](C)CO1 ZINC000880669127 EF On-Demand Anodyne NQO2 18 41 O=C(c1cnc(CC2CC2)s1)N1CCC(C2CCC2)CC1 ZINC000880669132 DH On-Demand Anodyne L3MBTL3 44 40 O=C(C[C@H]1CCNC1=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880669139 EC On-Demand Anodyne SIGMAR1 18 40 O=C(C[C@@H]1CCNC1=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880669140 EC On-Demand Anodyne SIGMAR1 18 40 O=C(C[C@H]1CCNC1=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880669141 EC On-Demand Anodyne SIGMAR1 18 40 O=C(C[C@@H]1CCNC1=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880669142 EC On-Demand Anodyne SIGMAR1 18 40 O=C([C@@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669162 GF On-Demand Anodyne SSTR1 19 42 O=C([C@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669163 GF On-Demand Anodyne SSTR1 19 42 COC[C@@H]1CCCN1NC(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880669165 FG On-Demand Anodyne CCR3 32 47 COC[C@@H]1CCCN1NC(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880669165 FG On-Demand Anodyne ACKR3 62 33 C=CC(C)(C)CC(=O)N1CCc2ccc(C)cc2C1 ZINC000880669172 CG On-Demand Mild HDAC6 33 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)CC2)ccc1F ZINC000880669173 EI On-Demand Anodyne CACNA1H 50 39 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)CC2)ccc1F ZINC000880669173 EI On-Demand Anodyne NPY2R 52 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)CC2)ccc1F ZINC000880669173 EI On-Demand Anodyne EPHX2 46 40 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)CC2)ccc1F ZINC000880669173 EI On-Demand Anodyne RBP4 43 37 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@H]3C(=O)OC[C@H]3C2)ccc1F ZINC000880669182 FF On-Demand Anodyne RBP4 46 34 C=CCCNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880669191 CD On-Demand Mild PAPA1_CARPA 41 51 C=CCCNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880669191 CD On-Demand Mild CTSK 18 52 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@H](CF)C2)ccc1F ZINC000880669192 EH On-Demand Anodyne CCR3 31 41 C=CCCNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880669193 CD On-Demand Mild PAPA1_CARPA 41 51 C=CCCNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880669193 CD On-Demand Mild CTSK 18 52 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@@H](CF)C2)ccc1F ZINC000880669198 EH On-Demand Anodyne CCR3 31 41 C=CCCNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880669199 CG On-Demand Mild INHA 80 38 C=CCCNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880669199 CG On-Demand Mild MTNR1A 27 46 C=CCCNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880669199 CG On-Demand Mild MTNR1B 32 49 C[C@H](CCNC(=O)[C@@H]1OC[C@@H]2CCC[C@@H]21)N(C)C ZINC000880669205 CD On-Demand Anodyne CHRNA4 21 43 C[C@@H](CCNC(=O)[C@@H]1OC[C@@H]2CCC[C@@H]21)N(C)C ZINC000880669207 CD On-Demand Anodyne CHRNA4 21 43 COCc1cc(NC(=O)NNC(=O)OC)ccc1OC ZINC000880669252 CD On-Demand Reactive TSHR 61 33 COCc1cc(NC(=O)NNC(=O)OC)ccc1OC ZINC000880669252 CD On-Demand Reactive QRFPR 44 36 COCc1cc(NC(=O)NNC(=O)OC)ccc1OC ZINC000880669252 CD On-Demand Reactive ENPP1 69 34 CC(C)c1ccc2c(c1)CN(C(=O)c1nnn(C)n1)CC2 ZINC000880669253 CD On-Demand Anodyne QRFPR 16 41 CS(=O)(=O)C1CCC(C(=O)NCC(F)(F)c2cccc(F)c2)CC1 ZINC000880669254 FF On-Demand Anodyne CACNA1G 37 46 Cn1ncc(Br)c1CC(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880669307 GF On-Demand Anodyne P2RX7 15 44 O=C(NCC(F)(F)c1cccc(F)c1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880669312 FE On-Demand Anodyne CACNA1G 34 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc(CC2CC2)s1 ZINC000880669344 FF On-Demand Anodyne NAMPT 29 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc(CC2CC2)s1 ZINC000880669345 FF On-Demand Anodyne NAMPT 29 42 Cc1cnc(Cl)c(C(=O)N2CCC(C3CCC3)CC2)c1 ZINC000880669348 CH On-Demand Anodyne L3MBTL3 52 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669360 GD On-Demand Anodyne SIGMAR1 20 44 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669360 GD On-Demand Anodyne CCR3 15 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669360 GD On-Demand Anodyne DPOL_VZVD 25 44 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669363 GD On-Demand Anodyne SIGMAR1 20 44 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669363 GD On-Demand Anodyne CCR3 15 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880669363 GD On-Demand Anodyne DPOL_VZVD 25 44 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne HTR1A 62 41 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne DRD2 52 48 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne DRD4 27 40 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne ADRA1D 40 41 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne ADRA1A 39 43 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne ADRA1B 31 41 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne DRD3 64 41 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne HTR7 48 44 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne KCNQ2 40 34 COc1cccc(OC)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669364 FF On-Demand Anodyne P2RX7 27 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(OCCO)CCOC1)C2 ZINC000880669369 ED On-Demand Anodyne MTNR1A 26 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(OCCO)CCOC1)C2 ZINC000880669369 ED On-Demand Anodyne MTNR1B 23 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(OCCO)CCOC1)C2 ZINC000880669372 ED On-Demand Anodyne MTNR1A 26 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(OCCO)CCOC1)C2 ZINC000880669372 ED On-Demand Anodyne MTNR1B 23 42 C=CCCNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880669387 CD On-Demand Mild PLD1 46 39 C=CCCNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880669387 CD On-Demand Mild PLD2 43 34 C=CCCNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880669389 CD On-Demand Mild PLD1 46 39 C=CCCNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880669389 CD On-Demand Mild PLD2 43 34 O=C(c1ccccc1)c1cc(NC(=O)N2CCO[C@H](C(F)F)C2)ccc1F ZINC000880669410 GH On-Demand Anodyne EPHX2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(OCC(F)(F)F)nn1)C2 ZINC000880669411 GF On-Demand Anodyne NQO2 26 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCO[C@@H](C(F)F)C2)ccc1F ZINC000880669413 GH On-Demand Anodyne EPHX2 27 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccc1F ZINC000880669417 GG On-Demand Anodyne CACNA1H 70 45 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CCNC3=O)CC2)ccc1F ZINC000880669417 GG On-Demand Anodyne NPY5R 30 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN1C[C@H](C)OC[C@H]1C ZINC000880669429 FD On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN1C[C@@H](C)OC[C@H]1C ZINC000880669431 FD On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN1C[C@H](C)OC[C@@H]1C ZINC000880669434 FD On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCN1C[C@@H](C)OC[C@@H]1C ZINC000880669436 FD On-Demand Anodyne PAPA1_CARPA 35 42 CC[C@@H](C)CCNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880669452 DF On-Demand Anodyne KCNQ2 66 35 O=C(c1cnc2cc[nH]c2c1)N1CCC(C2CCC2)CC1 ZINC000880669460 CG On-Demand Anodyne L3MBTL3 87 42 O=C(c1cnc2cc[nH]c2c1)N1CCC(C2CCC2)CC1 ZINC000880669460 CG On-Demand Anodyne HPGD 40 33 Cn1ncc(C2CCC2)c1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880669461 FD On-Demand Anodyne TBK1 41 35 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880669467 FH On-Demand Anodyne SLC6A1 96 37 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880669467 FH On-Demand Anodyne NPY2R 56 39 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880669472 GF On-Demand Anodyne NQO2 25 42 COc1ccc2c(c1)CC[C@H]2C(=O)NCc1ccc(OCC(F)(F)F)nn1 ZINC000880669472 GF On-Demand Anodyne PPARD 47 39 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880669474 FH On-Demand Anodyne SLC6A1 96 37 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880669474 FH On-Demand Anodyne NPY2R 56 39 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)CC1 ZINC000880669489 GD On-Demand Anodyne OPRK1 21 42 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)CC1 ZINC000880669489 GD On-Demand Anodyne SIGMAR1 18 54 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)CC1 ZINC000880669489 GD On-Demand Anodyne CACNA1G 31 40 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)CC1 ZINC000880669492 GD On-Demand Anodyne OPRK1 21 42 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)CC1 ZINC000880669492 GD On-Demand Anodyne SIGMAR1 18 54 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)CC1 ZINC000880669492 GD On-Demand Anodyne CACNA1G 31 40 C[C@@H]1CC(CNC(=O)c2nnn(C)n2)C[C@@H](C)C1 ZINC000880669497 CD On-Demand Anodyne CACNA1I 45 33 C[C@H]1C[C@@H](C)C[C@H](CNC(=O)c2nnn(C)n2)C1 ZINC000880669499 CD On-Demand Anodyne CACNA1I 45 33 C[C@H]1CC(CNC(=O)c2nnn(C)n2)C[C@H](C)C1 ZINC000880669501 CD On-Demand Anodyne CACNA1I 45 33 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669522 CE On-Demand Anodyne NQO2 18 40 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669522 CE On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669522 CE On-Demand Anodyne MTNR1B 15 41 O=C(CC[C@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669525 CE On-Demand Anodyne NQO2 18 40 O=C(CC[C@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669525 CE On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669525 CE On-Demand Anodyne MTNR1B 15 41 O=C(CC[C@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669527 CE On-Demand Anodyne NQO2 18 40 O=C(CC[C@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669527 CE On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@H]1CCc2ccccc21)NC/C=C\CO ZINC000880669527 CE On-Demand Anodyne MTNR1B 15 41 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669529 CE On-Demand Anodyne NQO2 18 40 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669529 CE On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@@H]1CCc2ccccc21)NC/C=C/CO ZINC000880669529 CE On-Demand Anodyne MTNR1B 15 41 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C\CO)c1ccccc1C(F)(F)F ZINC000880669541 GF On-Demand Anodyne PAPA1_CARPA 34 46 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C\CO)c1ccccc1C(F)(F)F ZINC000880669541 GF On-Demand Anodyne SCN10A 15 40 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C\CO)c1ccccc1C(F)(F)F ZINC000880669541 GF On-Demand Anodyne FPR1 43 35 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C/CO)c1ccccc1C(F)(F)F ZINC000880669544 GF On-Demand Anodyne PAPA1_CARPA 34 46 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C/CO)c1ccccc1C(F)(F)F ZINC000880669544 GF On-Demand Anodyne SCN10A 15 40 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C/CO)c1ccccc1C(F)(F)F ZINC000880669544 GF On-Demand Anodyne FPR1 43 35 O=C1NCC[C@@H]1CC(=O)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669563 FE On-Demand Anodyne SSTR1 32 49 O=C1NCC[C@@H]1CC(=O)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669563 FE On-Demand Anodyne BCL2A1 54 37 O=C1NCC[C@H]1CC(=O)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669565 FE On-Demand Anodyne SSTR1 32 49 O=C1NCC[C@H]1CC(=O)N1CCN(c2ccc(Cl)c(Cl)c2)CC1 ZINC000880669565 FE On-Demand Anodyne BCL2A1 54 37 COc1cccc(OC)c1CNC(=O)c1cc(C)cnc1Cl ZINC000880669589 DF On-Demand Anodyne HCRTR2 23 42 COc1cccc(OC)c1CNC(=O)c1cc(C)cnc1Cl ZINC000880669589 DF On-Demand Anodyne KCNK3 43 36 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne DRD2 25 43 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne PLA2G1B 43 33 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne SIGMAR1 15 44 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne P2RX7 38 42 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne PLA2G2A 52 41 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne PLA2G2D 40 33 COc1cccc(OC)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880669590 GD On-Demand Anodyne TMPRSS11D 40 32 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669593 GF On-Demand Anodyne SIGMAR1 39 46 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669593 GF On-Demand Anodyne CCR3 28 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669593 GF On-Demand Anodyne MCHR1 19 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669594 GF On-Demand Anodyne SIGMAR1 39 46 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669594 GF On-Demand Anodyne CCR3 28 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880669594 GF On-Demand Anodyne MCHR1 19 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncsc1C1CC1 ZINC000880669596 FF On-Demand Anodyne MCHR1 16 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncsc1C1CC1 ZINC000880669596 FF On-Demand Anodyne VHL 50 35 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncsc1C1CC1 ZINC000880669597 FF On-Demand Anodyne MCHR1 16 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncsc1C1CC1 ZINC000880669597 FF On-Demand Anodyne VHL 50 35 COc1cccc(OC)c1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880669598 FD On-Demand Anodyne MTNR1A 40 43 COc1cccc(OC)c1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880669598 FD On-Demand Anodyne MTNR1B 34 44 C=CCCNC(=O)[C@H]1CC[C@@H](C(N)=O)N1Cc1ccccc1 ZINC000880669625 DD On-Demand Mild SIGMAR1 20 41 O=C(C[C@H]1CCNC1=O)NCCc1ccnc2ccccc12 ZINC000880669635 CD On-Demand Anodyne MTNR1A 26 42 O=C(C[C@H]1CCNC1=O)NCCc1ccnc2ccccc12 ZINC000880669635 CD On-Demand Anodyne MTNR1B 20 42 O=C(C[C@@H]1CCNC1=O)NCCc1ccnc2ccccc12 ZINC000880669638 CD On-Demand Anodyne MTNR1A 26 42 O=C(C[C@@H]1CCNC1=O)NCCc1ccnc2ccccc12 ZINC000880669638 CD On-Demand Anodyne MTNR1B 20 42 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne TSHR 54 33 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne HTR1D 17 47 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne HTR1B 20 47 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne PDGFRB 49 39 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne EPHX2 15 45 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne RBP4 16 40 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne QRFPR 46 38 COCc1cc(NC(=O)N2CCCCCCC2)ccc1OC ZINC000880669651 DH On-Demand Anodyne ENPP1 69 35 C=CCCSCCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880669668 DF On-Demand Mild MPO 42 35 COc1cccc(OC)c1CNC(=O)c1cc(C)co1 ZINC000880669682 CF On-Demand Anodyne KCNK3 43 37 Cn1nnc(C(=O)N2CCc3ccc(Cl)c(Cl)c3C2)n1 ZINC000880669694 DD On-Demand Anodyne PNMT 15 47 CO[C@@](C)(CNC(=O)COC1CC1)COCc1ccccc1 ZINC000880669700 DD On-Demand Anodyne TIMP3 68 34 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1F ZINC000880669717 FE On-Demand Anodyne CACNA1H 46 39 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)ccc1F ZINC000880669717 FE On-Demand Anodyne RBP4 52 34 CC1(C)CC[C@@H](CC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)OC1 ZINC000880669727 FE On-Demand Anodyne CCR3 23 41 CC1(C)CC[C@@H](CC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)OC1 ZINC000880669727 FE On-Demand Anodyne NOS2 41 33 CC1(C)CC[C@@H](CC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)OC1 ZINC000880669729 FE On-Demand Anodyne CCR3 23 41 CC1(C)CC[C@@H](CC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)OC1 ZINC000880669729 FE On-Demand Anodyne NOS2 41 33 Cn1ncc(C2CCC2)c1CNC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880669761 EH On-Demand Anodyne P2RX7 15 40 O=C1NCC[C@H]1CC(=O)N1CCc2ccc(Cl)c(Cl)c2C1 ZINC000880669763 EE On-Demand Anodyne PNMT 15 43 O=C1NCC[C@@H]1CC(=O)N1CCc2ccc(Cl)c(Cl)c2C1 ZINC000880669766 EE On-Demand Anodyne PNMT 15 43 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild CELA1 19 42 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild GRIN2B 17 40 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild PREP 26 42 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild LGMN 62 38 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild TGM2 43 40 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild KLK5 40 38 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild F13A1 41 40 C=CCCNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669803 DE On-Demand Mild Q9NAW4_PLAFA 39 46 COCc1cc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880669805 GG On-Demand Clean CASR 15 40 COCc1cc(NC(=O)N(C)Cc2ccc(N3CCOCC3)cc2)ccc1OC ZINC000880669805 GG On-Demand Clean EPHB4 57 34 Cn1ncc(C2CCC2)c1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880669822 ED On-Demand Anodyne TBK1 45 34 Cn1ncc(C2CCC2)c1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880669826 ED On-Demand Anodyne TBK1 45 34 O=C(NC/C=C/CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669831 ED On-Demand Anodyne CELA1 19 43 O=C(NC/C=C/CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669831 ED On-Demand Anodyne PREP 28 45 O=C(NC/C=C/CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669831 ED On-Demand Anodyne LGMN 54 38 O=C(NC/C=C/CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669831 ED On-Demand Anodyne Q9NAW4_PLAFA 41 48 O=C(NC/C=C\CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669834 ED On-Demand Anodyne CELA1 19 43 O=C(NC/C=C\CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669834 ED On-Demand Anodyne PREP 28 45 O=C(NC/C=C\CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669834 ED On-Demand Anodyne LGMN 54 38 O=C(NC/C=C\CO)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880669834 ED On-Demand Anodyne Q9NAW4_PLAFA 41 48 COCc1cc(NC(=O)N(C)Cc2ccc(Cl)nc2)ccc1OC ZINC000880669848 EH On-Demand Anodyne TSHR 47 34 COCc1cc(NC(=O)N(C)Cc2ccc(Cl)nc2)ccc1OC ZINC000880669848 EH On-Demand Anodyne ENPP1 46 35 C[C@H](CCNC(=O)c1cc2ccccc2cc1F)N(C)C ZINC000880669850 CG On-Demand Anodyne POLR1A 56 41 C[C@@H](CCNC(=O)c1cc2ccccc2cc1F)N(C)C ZINC000880669852 CG On-Demand Anodyne POLR1A 56 41 COCc1cc(NC(=O)NC[C@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669870 GF On-Demand Anodyne TSHR 58 34 COCc1cc(NC(=O)NC[C@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669870 GF On-Demand Anodyne MTNR1A 37 44 COCc1cc(NC(=O)NC[C@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669870 GF On-Demand Anodyne MTNR1B 35 41 O=C(NCc1ccc2occc2c1)c1ccc(CN2CCOCC2)o1 ZINC000880669872 EF On-Demand Anodyne NAMPT 27 43 COCc1cc(NC(=O)NC[C@@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669873 GF On-Demand Anodyne TSHR 58 34 COCc1cc(NC(=O)NC[C@@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669873 GF On-Demand Anodyne MTNR1A 37 44 COCc1cc(NC(=O)NC[C@@H](O)c2cc(OC)ccc2OC)ccc1OC ZINC000880669873 GF On-Demand Anodyne MTNR1B 35 41 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc2c(c1)OCC(C)(C)C(=O)N2 ZINC000880669898 GI On-Demand Anodyne TRPM8 17 42 O=C(CN1CCCCS1(=O)=O)NNc1ccnc(Cl)c1 ZINC000880669923 DC On-Demand Reactive TYK2 46 32 O=C([C@@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880669955 GF On-Demand Anodyne CNR1 55 34 O=C([C@@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880669955 GF On-Demand Anodyne MC4R 45 37 O=C([C@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880669957 GF On-Demand Anodyne CNR1 55 34 O=C([C@H]1CCc2nncn2CC1)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880669957 GF On-Demand Anodyne MC4R 45 37 O=C(N[C@@H]1C=CCC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880669959 CG On-Demand Anodyne PDE4D 19 44 O=C(N[C@H]1C=CCC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880669961 CG On-Demand Anodyne PDE4D 19 44 CO[C@]1(CO)CCCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880670001 DE On-Demand Anodyne EBP 25 48 CO[C@]1(CO)CCCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880670002 DE On-Demand Anodyne EBP 25 48 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1csc(-c2ncc[nH]2)n1 ZINC000880670009 GE On-Demand Anodyne NAMPT 21 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1csc(-c2ncc[nH]2)n1 ZINC000880670010 GE On-Demand Anodyne NAMPT 21 40 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C/CO)c1ccc(Br)cc1 ZINC000880670021 GF On-Demand Anodyne PAPA1_CARPA 37 47 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C/CO)c1ccc(Br)cc1 ZINC000880670021 GF On-Demand Anodyne AMP1_PLAFQ 19 44 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C\CO)c1ccc(Br)cc1 ZINC000880670024 GF On-Demand Anodyne PAPA1_CARPA 37 47 CC(C)(C)OC(=O)N[C@@H](C(=O)NC/C=C\CO)c1ccc(Br)cc1 ZINC000880670024 GF On-Demand Anodyne AMP1_PLAFQ 19 44 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)c(Cl)c3)CC2)n1 ZINC000880670041 ED On-Demand Anodyne KCNA5 16 44 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)c(Cl)c3)CC2)n1 ZINC000880670041 ED On-Demand Anodyne CCKAR 19 43 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)c(Cl)c3)CC2)n1 ZINC000880670041 ED On-Demand Anodyne CCR1 21 40 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)c(Cl)c3)CC2)n1 ZINC000880670041 ED On-Demand Anodyne BCL2A1 52 36 C=CC(C)(C)CC(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880670058 DE On-Demand Mild SIGMAR1 19 41 C=CC(C)(C)CC(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880670059 DE On-Demand Mild SIGMAR1 19 41 COc1cccc(OC)c1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880670070 FE On-Demand Anodyne HTR1A 16 40 COc1cccc(OC)c1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880670070 FE On-Demand Anodyne DRD2 26 40 COc1cccc(OC)c1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880670070 FE On-Demand Anodyne DRD4 40 31 COc1cccc(OC)c1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880670070 FE On-Demand Anodyne DRD3 33 40 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC/C=C\CO ZINC000880670073 FG On-Demand Anodyne PPARA 17 49 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC/C=C\CO ZINC000880670073 FG On-Demand Anodyne PPARD 33 44 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC/C=C/CO ZINC000880670074 FG On-Demand Anodyne PPARA 17 49 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC/C=C/CO ZINC000880670074 FG On-Demand Anodyne PPARD 33 44 Cc1cc(-c2nc(C)c(C(=O)NC/C=C\CO)s2)ccc1F ZINC000880670091 DF On-Demand Anodyne SCD1 24 40 Cc1cc(-c2nc(C)c(C(=O)NC/C=C/CO)s2)ccc1F ZINC000880670092 DF On-Demand Anodyne SCD1 24 40 O=C(COC1CC1)NCCc1ccnc2ccccc12 ZINC000880670093 CE On-Demand Anodyne MTNR1A 47 48 O=C(COC1CC1)NCCc1ccnc2ccccc12 ZINC000880670093 CE On-Demand Anodyne MTNR1B 34 48 O=C(NCCc1ccnc2ccccc12)[C@H]1CCc2nncn2CC1 ZINC000880670095 EE On-Demand Anodyne MTNR1A 19 42 O=C(NCCc1ccnc2ccccc12)[C@H]1CCc2nncn2CC1 ZINC000880670095 EE On-Demand Anodyne MTNR1B 15 42 O=C(NCCc1ccnc2ccccc12)[C@H]1CCc2nncn2CC1 ZINC000880670095 EE On-Demand Anodyne HNMT 47 35 O=C(NCCc1ccnc2ccccc12)[C@@H]1CCc2nncn2CC1 ZINC000880670097 EE On-Demand Anodyne MTNR1A 19 42 O=C(NCCc1ccnc2ccccc12)[C@@H]1CCc2nncn2CC1 ZINC000880670097 EE On-Demand Anodyne MTNR1B 15 42 O=C(NCCc1ccnc2ccccc12)[C@@H]1CCc2nncn2CC1 ZINC000880670097 EE On-Demand Anodyne HNMT 47 35 O=C(CN1CCCCS1(=O)=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880670141 GC On-Demand Anodyne SIGMAR1 17 42 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne ACE 20 40 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne CTRA_BOVIN 52 30 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne CAPNS1 45 30 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne CELA2A 40 30 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne LGMN 70 39 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne CAPN1 46 41 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne CAPN2 55 35 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne KLK5 43 40 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1cscn1 ZINC000880670142 GG On-Demand Anodyne Q9NAW4_PLAFA 40 47 O=C(CN1CCCCS1(=O)=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880670144 GC On-Demand Anodyne SIGMAR1 17 42 O=C(C[C@@H]1C[C@H]1C1CC1)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880670169 CF On-Demand Anodyne ROCK2 24 48 CS(=O)(=O)C1CCC(C(=O)Nc2ccc3c(=O)[nH]ccc3c2)CC1 ZINC000880670186 EE On-Demand Anodyne ROCK2 27 48 O=C1CC[C@@H](c2ccc(C(=O)NCC(F)(F)c3cccc(F)c3)cc2)N1 ZINC000880670198 FG On-Demand Anodyne PLD1 51 36 O=C1CC[C@@H](c2ccc(C(=O)NCC(F)(F)c3cccc(F)c3)cc2)N1 ZINC000880670198 FG On-Demand Anodyne PLD2 51 36 O=C1CC[C@H](c2ccc(C(=O)NCC(F)(F)c3cccc(F)c3)cc2)N1 ZINC000880670201 FG On-Demand Anodyne PLD1 51 36 O=C1CC[C@H](c2ccc(C(=O)NCC(F)(F)c3cccc(F)c3)cc2)N1 ZINC000880670201 FG On-Demand Anodyne PLD2 51 36 COc1cccc(C(C)(C)C(=O)NCc2ccc(OCC(F)(F)F)nn2)c1 ZINC000880670204 GG On-Demand Anodyne PDS 40 35 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne TSHR 46 30 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne HTR1B 15 48 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne PDGFRB 49 41 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne F13A1 24 42 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne GPR119 37 45 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne QRFPR 42 35 COCc1cc(NC(=O)N2CCN(C(=O)OC(C)(C)C)CC2)ccc1OC ZINC000880670221 GF On-Demand Anodyne ENPP1 63 34 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C3CCC3)cnn1C)C2 ZINC000880670225 FG On-Demand Anodyne MTNR1A 32 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C3CCC3)cnn1C)C2 ZINC000880670225 FG On-Demand Anodyne MTNR1B 32 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C3CCC3)cnn1C)C2 ZINC000880670225 FG On-Demand Anodyne TBK1 55 34 CC[C@@H](C)CCNC(=O)[C@H](CNC(=O)OC(C)(C)C)OC ZINC000880670231 DE On-Demand Anodyne CTSK 16 43 C[C@@H](CCNC(=O)CN1CCCCS1(=O)=O)N(C)C ZINC000880670239 CB On-Demand Anodyne CHRNA4 18 40 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880670256 GI On-Demand Anodyne TIMP3 70 35 COCc1cc(NC(=O)NC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880670260 EG On-Demand Anodyne TSHR 62 34 COCc1cc(NC(=O)NC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880670260 EG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)NC[C@@H]2CC2(Cl)Cl)ccc1OC ZINC000880670260 EG On-Demand Anodyne ENPP1 55 32 COCc1cc(NC(=O)NC[C@H]2CC2(Cl)Cl)ccc1OC ZINC000880670262 EG On-Demand Anodyne TSHR 62 34 COCc1cc(NC(=O)NC[C@H]2CC2(Cl)Cl)ccc1OC ZINC000880670262 EG On-Demand Anodyne QRFPR 48 40 COCc1cc(NC(=O)NC[C@H]2CC2(Cl)Cl)ccc1OC ZINC000880670262 EG On-Demand Anodyne ENPP1 55 32 Cn1ncc(C2CCC2)c1CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880670268 GD On-Demand Anodyne TMPRSS11D 56 33 C[C@H](CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)N(C)C ZINC000880670278 EC On-Demand Anodyne ACE 41 38 C[C@H](CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)N(C)C ZINC000880670278 EC On-Demand Anodyne XIAP 41 38 C[C@@H](CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)N(C)C ZINC000880670281 EC On-Demand Anodyne ACE 41 38 C[C@@H](CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)N(C)C ZINC000880670281 EC On-Demand Anodyne XIAP 41 38 O=C(CN1CCCCS1(=O)=O)NCCc1ccnc2ccccc12 ZINC000880670282 ED On-Demand Anodyne MTNR1A 15 41 O=C(CN1CCCCS1(=O)=O)NCCc1ccnc2ccccc12 ZINC000880670282 ED On-Demand Anodyne HNMT 51 40 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne ADRB2 43 37 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne ADRB1 41 42 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne TSHR 75 36 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne ADRB3 47 42 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne SOAT1 32 42 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne QRFPR 40 38 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2)ccc1OC ZINC000880670298 EF On-Demand Anodyne ENPP1 67 32 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne ADRB2 43 37 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne ADRB1 41 42 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne TSHR 75 36 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne ADRB3 47 42 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne SOAT1 32 42 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne QRFPR 40 38 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2)ccc1OC ZINC000880670299 EF On-Demand Anodyne ENPP1 67 32 C=CC[C@@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880670315 FE On-Demand Mild PREP 70 40 C=CC[C@H]1CCCN(C(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880670316 FE On-Demand Mild PREP 70 40 O=C(Nc1ccc(F)c(C(=O)c2ccccc2)c1)N[C@@H]1CC[C@H](O)CC1 ZINC000880670349 FG On-Demand Anodyne EPHX2 53 43 CONC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880670395 GF On-Demand Anodyne CACNA1H 41 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1cscn1 ZINC000880670396 EE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1cscn1 ZINC000880670396 EE On-Demand Anodyne FPR1 44 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1cscn1 ZINC000880670398 EE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1cscn1 ZINC000880670398 EE On-Demand Anodyne FPR1 44 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1cscn1 ZINC000880670401 EE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1cscn1 ZINC000880670401 EE On-Demand Anodyne FPR1 44 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1cscn1 ZINC000880670403 EE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1cscn1 ZINC000880670403 EE On-Demand Anodyne FPR1 44 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H](O)C(F)(F)C1 ZINC000880670409 GF On-Demand Anodyne RBP4 40 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H](O)C(F)(F)C1 ZINC000880670409 GF On-Demand Anodyne SFRP1 41 32 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H](O)C(F)(F)C1 ZINC000880670411 GF On-Demand Anodyne RBP4 40 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H](O)C(F)(F)C1 ZINC000880670411 GF On-Demand Anodyne SFRP1 41 32 CSc1nccnc1C(=O)Nc1nc2ccc(CN(C)C3CC3)cc2s1 ZINC000880670457 GH On-Demand Anodyne CSNK1D 42 38 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@H]3C[C@]3(CO)C2)ccc1F ZINC000880670496 FF On-Demand Anodyne EPHX2 25 40 COCc1cc(NC(=O)NC[C@@H](O)c2ccco2)ccc1OC ZINC000880670498 DE On-Demand Anodyne TSHR 61 36 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@@H]3C[C@]3(CO)C2)ccc1F ZINC000880670499 FF On-Demand Anodyne EPHX2 25 40 COCc1cc(NC(=O)NC[C@H](O)c2ccco2)ccc1OC ZINC000880670501 DE On-Demand Anodyne TSHR 61 36 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@H]3C[C@@]3(CO)C2)ccc1F ZINC000880670504 FF On-Demand Anodyne EPHX2 25 40 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@@H]3C[C@@]3(CO)C2)ccc1F ZINC000880670507 FF On-Demand Anodyne EPHX2 25 40 Cn1ncc(C2CCC2)c1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880670536 FF On-Demand Anodyne GABRA1 17 46 Cn1ncc(C2CCC2)c1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880670536 FF On-Demand Anodyne HTR1F 61 37 O=C(c1cccn2nccc12)N1CCC(C2CCC2)CC1 ZINC000880670550 CF On-Demand Anodyne L3MBTL3 70 43 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670555 FD On-Demand Anodyne DRD4 26 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670555 FD On-Demand Anodyne SIGMAR1 19 43 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670555 FD On-Demand Anodyne MCHR1 22 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670555 FD On-Demand Anodyne NAMPT 46 39 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670558 FD On-Demand Anodyne DRD4 26 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670558 FD On-Demand Anodyne SIGMAR1 19 43 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670558 FD On-Demand Anodyne MCHR1 22 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccn2nccc12 ZINC000880670558 FD On-Demand Anodyne NAMPT 46 39 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne CHRM3 17 40 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne SIGMAR1 16 41 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne CCR3 18 41 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne PLD1 43 35 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne PLD2 40 35 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne MCHR1 20 47 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670597 GE On-Demand Anodyne NAMPT 20 42 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne CHRM3 17 40 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne SIGMAR1 16 41 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne CCR3 18 41 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne PLD1 43 35 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne PLD2 40 35 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne MCHR1 20 47 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670600 GE On-Demand Anodyne NAMPT 20 42 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne CHRM3 17 40 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne SIGMAR1 16 41 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne CCR3 18 41 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne PLD1 43 35 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne PLD2 40 35 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne MCHR1 20 47 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@@H](O)C4)cc3)cc2)N1 ZINC000880670603 GE On-Demand Anodyne NAMPT 20 42 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne CHRM3 17 40 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne SIGMAR1 16 41 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne CCR3 18 41 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne PLD1 43 35 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne PLD2 40 35 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne MCHR1 20 47 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(CN4CC[C@H](O)C4)cc3)cc2)N1 ZINC000880670606 GE On-Demand Anodyne NAMPT 20 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne NQO2 23 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne PAPA1_CARPA 43 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne CCKAR 55 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne CTSK 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne CTSL 16 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne TACR3 24 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne MTNR1A 28 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne MTNR1B 16 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne CCKBR 17 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670628 GF On-Demand Anodyne FPR1 46 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne NQO2 23 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne PAPA1_CARPA 43 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne CCKAR 55 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne CTSK 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne CTSL 16 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne TACR3 24 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne MTNR1A 28 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne MTNR1B 16 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne CCKBR 17 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccnc2ccccc12 ZINC000880670633 GF On-Demand Anodyne FPR1 46 38 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne SIGMAR1 22 44 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne CCR3 28 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne AKT2 38 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne AKT1 23 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne CXCR3 23 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670656 GF On-Demand Anodyne MCHR1 19 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne SIGMAR1 22 44 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne CCR3 28 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne AKT2 38 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne AKT1 23 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne CXCR3 23 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ncccc1-c1ccccn1 ZINC000880670658 GF On-Demand Anodyne MCHR1 19 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnccc1C ZINC000880670660 FD On-Demand Anodyne PAPA1_CARPA 40 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnccc1C ZINC000880670662 FD On-Demand Anodyne PAPA1_CARPA 40 42 O=C(NCC(F)(F)c1cccc(F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880670679 FF On-Demand Anodyne CACNA1G 25 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670684 FF On-Demand Anodyne PAPA1_CARPA 43 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670684 FF On-Demand Anodyne CTSL 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670684 FF On-Demand Anodyne FPR1 45 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670685 FF On-Demand Anodyne PAPA1_CARPA 43 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670685 FF On-Demand Anodyne CTSL 15 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc2occc2c1 ZINC000880670685 FF On-Demand Anodyne FPR1 45 37 O=C(Nc1ccc2c(=O)[nH]ccc2c1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880670713 CE On-Demand Anodyne ROCK2 23 44 C[C@H](CCNC(=O)c1cccc2nsnc12)N(C)C ZINC000880670732 CD On-Demand Anodyne AOX1 17 42 C[C@@H](CCNC(=O)c1cccc2nsnc12)N(C)C ZINC000880670734 CD On-Demand Anodyne AOX1 17 42 O=C(c1ncsc1C1CC1)N1CCC(C2CCC2)CC1 ZINC000880670736 CH On-Demand Anodyne L3MBTL3 43 34 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H](O)C(F)(F)C3)cc2)N1 ZINC000880670740 DD On-Demand Anodyne L3MBTL3 44 35 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H](O)C(F)(F)C3)cc2)N1 ZINC000880670741 DD On-Demand Anodyne L3MBTL3 44 35 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@@H](O)C(F)(F)C3)cc2)N1 ZINC000880670742 DD On-Demand Anodyne L3MBTL3 44 35 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@H](O)C(F)(F)C3)cc2)N1 ZINC000880670743 DD On-Demand Anodyne L3MBTL3 44 35 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne CNR1 61 45 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne MC4R 54 39 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne HRH4 31 41 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne P2RX7 17 43 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne NPY2R 38 41 Cn1nnc(C(=O)N2CCN(c3ccc(Cl)cc3Cl)CC2)n1 ZINC000880670754 ED On-Demand Anodyne ALPL 27 45 CO[C@]1(CO)CCCN(C(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880670773 GC On-Demand Anodyne PREP 54 40 CO[C@]1(CO)CCCN(C(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880670773 GC On-Demand Anodyne SLC12A5 64 35 C[C@H](CCNC(=O)c1ccc(OC(F)F)c(Cl)c1)N(C)C ZINC000880670778 DG On-Demand Anodyne PDE4D 16 40 C[C@@H](CCNC(=O)c1ccc(OC(F)F)c(Cl)c1)N(C)C ZINC000880670781 DG On-Demand Anodyne PDE4D 16 40 CCOC(=O)N1CCC(NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880670789 FF On-Demand Anodyne TSHR 53 31 CCOC(=O)N1CCC(NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880670789 FF On-Demand Anodyne EPHX2 58 52 CCOC(=O)N1CCC(NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880670789 FF On-Demand Anodyne CCR8 22 41 CCOC(=O)N1CCC(NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880670789 FF On-Demand Anodyne QRFPR 42 35 CCOC(=O)N1CCC(NC(=O)Nc2ccc(OC)c(COC)c2)CC1 ZINC000880670789 FF On-Demand Anodyne ENPP1 66 32 CN(Cc1ccc2nc(NC(=O)c3nnn(C)n3)sc2c1)C1CC1 ZINC000880670791 ED On-Demand Anodyne CSNK1D 42 39 Cn1nnc(C(=O)N2CCC(C3CCC3)CC2)n1 ZINC000880670795 BC On-Demand Anodyne L3MBTL3 46 37 O=C1NCC[C@@H]1CC(=O)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880670799 FE On-Demand Anodyne MC4R 62 40 O=C1NCC[C@H]1CC(=O)N1CCN(c2ccc(Cl)cc2Cl)CC1 ZINC000880670802 FE On-Demand Anodyne MC4R 62 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C=CCC1 ZINC000880670831 CD On-Demand Anodyne PAPA1_CARPA 36 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C=CCC1 ZINC000880670833 CD On-Demand Anodyne PAPA1_CARPA 36 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C=CCC1 ZINC000880670835 CD On-Demand Anodyne PAPA1_CARPA 36 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C=CCC1 ZINC000880670837 CD On-Demand Anodyne PAPA1_CARPA 36 41 C=CC(C)(C)CC(=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880670839 CG On-Demand Mild ROCK2 22 50 CC[C@@H](C)CCNC(=O)c1ncsc1C1CC1 ZINC000880670882 CG On-Demand Anodyne MAP1 40 35 O=C1CC[C@H](c2ccc(C(=O)N3CCC(C4CCC4)CC3)cc2)N1 ZINC000880670926 EG On-Demand Anodyne L3MBTL3 97 49 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(C4CCC4)CC3)cc2)N1 ZINC000880670928 EG On-Demand Anodyne L3MBTL3 97 49 COc1cccc(OC)c1CNC(=O)c1cnc(C(C)C)nc1C ZINC000880670931 EF On-Demand Anodyne KCNA3 22 40 O=C(C[C@@H]1C[C@H]1C1CC1)NCCc1ccnc2ccccc12 ZINC000880670943 CG On-Demand Anodyne MTNR1A 19 43 CN(CCOc1ccccc1C(=O)NC/C=C/CO)C(=O)OC(C)(C)C ZINC000880670974 FE On-Demand Anodyne HCN1 42 31 CC(C)(C)OC(=O)N1C[C@@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)C(C)(C)C1 ZINC000880670976 GG On-Demand Anodyne ROCK2 19 41 CN(CCOc1ccccc1C(=O)NC/C=C\CO)C(=O)OC(C)(C)C ZINC000880670977 FE On-Demand Anodyne HCN1 42 31 CC(C)(C)OC(=O)N1C[C@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)C(C)(C)C1 ZINC000880670980 GG On-Demand Anodyne ROCK2 19 41 O=C(c1ncccc1-c1ccccn1)N1CCC(C2CCC2)CC1 ZINC000880670982 DH On-Demand Anodyne L3MBTL3 48 35 O=C(NOC1CCOCC1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880670984 FG On-Demand Anodyne EPHX2 25 44 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cncc2[nH]ccc12 ZINC000880670995 FE On-Demand Anodyne PRKCQ 17 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cncc2[nH]ccc12 ZINC000880670999 FE On-Demand Anodyne PRKCQ 17 40 C=CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880671004 BG On-Demand Mild NQO2 21 45 C=CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880671004 BG On-Demand Mild MTNR1A 17 41 C=CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880671004 BG On-Demand Mild MTNR1B 17 41 C=CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880671006 BG On-Demand Mild NQO2 21 45 C=CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880671006 BG On-Demand Mild MTNR1A 17 41 C=CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880671006 BG On-Demand Mild MTNR1B 17 41 CO[C@@](C)(CNC(=O)[C@H]1CCc2nncn2CC1)COCc1ccccc1 ZINC000880671017 FD On-Demand Anodyne CACNA1G 33 41 CO[C@@](C)(CNC(=O)[C@@H]1CCc2nncn2CC1)COCc1ccccc1 ZINC000880671019 FD On-Demand Anodyne CACNA1G 33 41 COCc1cc(NC(=O)NC[C@H](O)c2ccccc2F)ccc1OC ZINC000880671048 EF On-Demand Anodyne TSHR 69 38 COCc1cc(NC(=O)NC[C@@H](O)c2ccccc2F)ccc1OC ZINC000880671051 EF On-Demand Anodyne TSHR 69 38 O=C(NC[C@H]1C[C@H](O)C1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880671053 EF On-Demand Anodyne EPHX2 19 42 COc1cccc(OC)c1CNC(=O)Cc1c(Br)cnn1C ZINC000880671061 FE On-Demand Anodyne P2RX7 23 43 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne TSHR 68 34 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne PTAFR 35 46 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne CHRNA7 21 41 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne ROCK2 24 46 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne QPCT 20 45 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne ENPP1 53 36 COCc1cc(NC(=O)NCCc2cccnc2)ccc1OC ZINC000880671078 DF On-Demand Anodyne NAMPT 50 48 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671092 FE On-Demand Anodyne HSP90AA1 17 42 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671092 FE On-Demand Anodyne MCHR1 21 41 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671092 FE On-Demand Anodyne VHL 48 33 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671093 FE On-Demand Anodyne HSP90AA1 17 42 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671093 FE On-Demand Anodyne MCHR1 21 41 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671093 FE On-Demand Anodyne VHL 48 33 COc1cccc(OC)c1CNC(=O)c1ncsc1C1CC1 ZINC000880671097 DF On-Demand Anodyne MAP1 66 38 CC[C@@H](C)CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880671108 EE On-Demand Anodyne ACE 46 38 CC[C@@H](C)CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880671108 EE On-Demand Anodyne TRY1_BOVIN 41 33 CC[C@@H](C)CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880671108 EE On-Demand Anodyne CAPN2 44 33 CC[C@@H](C)CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880671108 EE On-Demand Anodyne TPP2 41 43 CC[C@@H](C)CCNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880671108 EE On-Demand Anodyne XIAP 66 38 O=C(C[C@@H]1CCNC1=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671121 CC On-Demand Anodyne ROCK2 24 49 O=C(C[C@H]1CCNC1=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671126 CC On-Demand Anodyne ROCK2 24 49 CS(=O)(=O)C1CCC(C(=O)NNc2ccnc(Cl)c2)CC1 ZINC000880671142 ED On-Demand Reactive TYK2 60 41 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@@H]3[C@H](C2)C3(F)F)ccc1F ZINC000880671144 FH On-Demand Anodyne RBP4 45 33 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)COCCO3)ccc1F ZINC000880671150 GG On-Demand Anodyne CACNA1H 46 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)COCCO3)ccc1F ZINC000880671150 GG On-Demand Anodyne EPHX2 35 47 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)COCCO3)ccc1F ZINC000880671150 GG On-Demand Anodyne TRPM8 30 41 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@H]3[C@H](C2)C3(F)F)ccc1F ZINC000880671156 FH On-Demand Anodyne RBP4 45 33 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@@H]3[C@@H](C2)C3(F)F)ccc1F ZINC000880671160 FH On-Demand Anodyne RBP4 45 33 O=C(Nc1ccc(F)c(C(=O)c2ccccc2)c1)NC1CC2(CSC2)C1 ZINC000880671171 FI On-Demand Anodyne EPHX2 36 42 O=C(c1ccccc1)c1cc(NC(=O)N2CC(CC3CCOCC3)C2)ccc1F ZINC000880671181 GI On-Demand Anodyne EPHX2 19 40 C[C@@H](CCNC(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1)N(C)C ZINC000880671197 EG On-Demand Anodyne DRD4 41 31 C[C@H](CCNC(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1)N(C)C ZINC000880671198 EG On-Demand Anodyne DRD4 41 31 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1F ZINC000880671203 FH On-Demand Anodyne CACNA1H 41 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1F ZINC000880671203 FH On-Demand Anodyne NPY2R 42 35 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1F ZINC000880671203 FH On-Demand Anodyne CCR3 23 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@H](CO)CC2)ccc1F ZINC000880671203 FH On-Demand Anodyne EPHX2 27 48 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccc1F ZINC000880671204 GJ On-Demand Anodyne CACNA1H 46 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccc1F ZINC000880671204 GJ On-Demand Anodyne EPHX2 36 47 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CCCCO3)CC2)ccc1F ZINC000880671204 GJ On-Demand Anodyne TRPM8 30 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1F ZINC000880671205 FH On-Demand Anodyne CACNA1H 41 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1F ZINC000880671205 FH On-Demand Anodyne NPY2R 42 35 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1F ZINC000880671205 FH On-Demand Anodyne CCR3 23 41 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@H](CO)CC2)ccc1F ZINC000880671205 FH On-Demand Anodyne EPHX2 27 48 O=C(NCC(F)(F)c1cccc(F)c1)[C@H]1CCc2nncn2CC1 ZINC000880671217 EE On-Demand Anodyne CACNA1G 39 46 O=C(Cc1ccccc1N1CCCC1=O)NCCc1ccnc2ccccc12 ZINC000880671260 FG On-Demand Anodyne HNMT 48 37 C[C@@H](CCNC(=O)CC[C@H]1CCc2ccccc21)N(C)C ZINC000880671270 CF On-Demand Anodyne NQO2 21 47 C[C@@H](CCNC(=O)CC[C@H]1CCc2ccccc21)N(C)C ZINC000880671270 CF On-Demand Anodyne MTNR1A 31 44 C[C@@H](CCNC(=O)CC[C@H]1CCc2ccccc21)N(C)C ZINC000880671270 CF On-Demand Anodyne MTNR1B 32 44 O=C(NCCc1ccnc2ccccc12)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880671273 FE On-Demand Anodyne MTNR1A 20 45 O=C(NCCc1ccnc2ccccc12)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880671273 FE On-Demand Anodyne MTNR1B 15 40 O=C(NCCc1ccnc2ccccc12)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880671273 FE On-Demand Anodyne HNMT 48 38 C[C@@H](CCNC(=O)CC[C@@H]1CCc2ccccc21)N(C)C ZINC000880671274 CF On-Demand Anodyne NQO2 21 47 C[C@@H](CCNC(=O)CC[C@@H]1CCc2ccccc21)N(C)C ZINC000880671274 CF On-Demand Anodyne MTNR1A 31 44 C[C@@H](CCNC(=O)CC[C@@H]1CCc2ccccc21)N(C)C ZINC000880671274 CF On-Demand Anodyne MTNR1B 32 44 O=C(c1ccc(CN2CCOCC2)o1)N1CCC(C2CCC2)CC1 ZINC000880671292 EF On-Demand Anodyne L3MBTL3 43 45 C[C@@H](CCNC(=O)COC1CC1)N(C)C ZINC000880671298 BC On-Demand Anodyne CHRNA3 25 40 C[C@@H](CCNC(=O)COC1CC1)N(C)C ZINC000880671298 BC On-Demand Anodyne CHRNA4 23 42 CC[C@@H]1CCC[C@@]1(C)C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671313 EG On-Demand Anodyne SIGMAR1 15 40 C=CC[C@H]1CCCN(C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880671315 EH On-Demand Mild PDK1 40 32 C=CC[C@@H]1CCCN(C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880671317 EH On-Demand Mild PDK1 40 32 CC[C@@H]1CCC[C@@]1(C)C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671318 EG On-Demand Anodyne SIGMAR1 15 40 C[C@H]1C[C@@H](C)C[C@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880671323 EG On-Demand Anodyne CACNA1I 50 34 C[C@H]1CC(CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C[C@H](C)C1 ZINC000880671328 EG On-Demand Anodyne CACNA1I 50 34 C[C@H]1CC(CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C[C@H](C)C1 ZINC000880671333 EG On-Demand Anodyne CACNA1I 50 34 C[C@H]1C[C@@H](C)C[C@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880671339 EG On-Demand Anodyne CACNA1I 50 34 C[C@@H]1CC(CNC(=O)c2ccc(CN3CCOCC3)o2)C[C@@H](C)C1 ZINC000880671344 EF On-Demand Anodyne CACNA1I 58 40 C[C@H]1CC(CNC(=O)c2ccc(CN3CCOCC3)o2)C[C@H](C)C1 ZINC000880671348 EF On-Demand Anodyne CACNA1I 58 40 C[C@H]1C[C@@H](C)C[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880671351 EF On-Demand Anodyne CACNA1I 58 40 COc1cccc(OC)c1CNC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880671357 EG On-Demand Anodyne KCNA3 50 39 Cc1ccncc1CCNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880671373 ED On-Demand Anodyne NAMPT 28 40 O=C(C[C@@H]1C[C@H]1C1CC1)NNc1ccnc(Cl)c1 ZINC000880671392 CF On-Demand Reactive TYK2 50 34 O=C(NC[C@H](OC1CCCC1)C(F)(F)F)c1cccn2nccc12 ZINC000880671412 EF On-Demand Anodyne JAK3 15 41 O=C(NC[C@H](OC1CCCC1)C(F)(F)F)c1cccn2nccc12 ZINC000880671412 EF On-Demand Anodyne TYK2 19 41 O=C(NC[C@@H](OC1CCCC1)C(F)(F)F)c1cccn2nccc12 ZINC000880671413 EF On-Demand Anodyne JAK3 15 41 O=C(NC[C@@H](OC1CCCC1)C(F)(F)F)c1cccn2nccc12 ZINC000880671413 EF On-Demand Anodyne TYK2 19 41 O=C(N[C@@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671431 EF On-Demand Anodyne PREP 28 41 O=C(N[C@@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671431 EF On-Demand Anodyne LGMN 62 39 O=C(N[C@@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671431 EF On-Demand Anodyne Q9NAW4_PLAFA 41 45 O=C(N[C@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671432 EF On-Demand Anodyne PREP 28 41 O=C(N[C@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671432 EF On-Demand Anodyne LGMN 62 39 O=C(N[C@H]1C=CCC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880671432 EF On-Demand Anodyne Q9NAW4_PLAFA 41 45 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)(F)CC2)ccc1F ZINC000880671433 FI On-Demand Anodyne CACNA1H 61 43 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)(F)CC2)ccc1F ZINC000880671433 FI On-Demand Anodyne NPY5R 30 42 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(F)(F)CC2)ccc1F ZINC000880671433 FI On-Demand Anodyne EPHX2 35 42 C[C@@H](CCNC(=O)Cc1ccccc1N1CCCC1=O)N(C)C ZINC000880671477 DD On-Demand Anodyne KCNQ2 58 34 O=C(c1csc(-c2ncc[nH]2)n1)N1CCC(C2CCC2)CC1 ZINC000880671481 DG On-Demand Anodyne TRPC6 43 39 O=C(COC1CC1)NNc1ccnc(Cl)c1 ZINC000880671512 BD On-Demand Reactive TYK2 52 36 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne CCKAR 23 41 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne NPY2R 41 34 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne MTOR 27 43 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne EPHX2 72 48 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne ST14 25 40 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671527 GG On-Demand Anodyne CXCR3 18 40 COc1ccccc1-c1ccc(C(=O)N[C@H](C)C2(CO)CC2)c(O)n1 ZINC000880671580 EE On-Demand Anodyne KCNA3 43 38 COc1ccccc1-c1ccc(C(=O)N[C@@H](C)C2(CO)CC2)c(O)n1 ZINC000880671583 EE On-Demand Anodyne KCNA3 43 38 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1coc(-c2ccccn2)n1 ZINC000880671606 GE On-Demand Anodyne MCHR1 16 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1coc(-c2ccccn2)n1 ZINC000880671609 GE On-Demand Anodyne MCHR1 16 40 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H](C)N(C)C)C2 ZINC000880671613 DE On-Demand Anodyne NQO2 37 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H](C)N(C)C)C2 ZINC000880671613 DE On-Demand Anodyne MTNR1A 78 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H](C)N(C)C)C2 ZINC000880671613 DE On-Demand Anodyne MTNR1B 70 43 O=C(Nc1ccc2c(=O)[nH]ccc2c1)c1ccc(CN2CCOCC2)o1 ZINC000880671645 FE On-Demand Anodyne ROCK2 15 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671648 ED On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671648 ED On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671648 ED On-Demand Anodyne FPR1 47 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671649 ED On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671649 ED On-Demand Anodyne POLG_HCV1 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671649 ED On-Demand Anodyne FPR1 47 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671650 ED On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671650 ED On-Demand Anodyne POLG_HCV1 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1(CO)CC1 ZINC000880671650 ED On-Demand Anodyne FPR1 47 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671651 ED On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671651 ED On-Demand Anodyne POLG_HCV1 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1(CO)CC1 ZINC000880671651 ED On-Demand Anodyne FPR1 47 37 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)CO1 ZINC000880671656 GF On-Demand Anodyne ROCK2 18 41 CC(C)(C)OC(=O)CC[C@@H]1C[C@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)CO1 ZINC000880671657 GF On-Demand Anodyne ROCK2 18 41 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)CO1 ZINC000880671658 GF On-Demand Anodyne ROCK2 18 41 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)Nc2ccc3c(=O)[nH]ccc3c2)CO1 ZINC000880671659 GF On-Demand Anodyne ROCK2 18 41 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](C)N(C)C)C2 ZINC000880671661 DE On-Demand Anodyne NQO2 37 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](C)N(C)C)C2 ZINC000880671661 DE On-Demand Anodyne MTNR1A 78 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](C)N(C)C)C2 ZINC000880671661 DE On-Demand Anodyne MTNR1B 70 43 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671664 DF On-Demand Anodyne ROCK2 21 43 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671666 DF On-Demand Anodyne ROCK2 21 43 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671668 DF On-Demand Anodyne ROCK2 21 43 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880671670 DF On-Demand Anodyne ROCK2 21 43 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880671671 GH On-Demand Anodyne NPY2R 45 32 O=C(NNC(=O)C1CCOCC1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880671688 GF On-Demand Reactive EPHX2 26 44 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne ACE 32 42 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CTRA_BOVIN 62 33 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne KLK3 71 32 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne TRY1_BOVIN 45 33 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CTSG 42 33 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne PREP 26 40 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CAPNS1 61 32 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CELA2A 50 33 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne LGMN 74 42 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CAPN1 63 43 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne CAPN2 70 35 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne KLK5 40 39 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne SLC12A5 66 37 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1(CO)CC1 ZINC000880671691 FE On-Demand Anodyne Q9NAW4_PLAFA 44 52 O=C(c1ccccc1)c1cc(NC(=O)N2CC3(CC3)C2)ccc1F ZINC000880671693 DH On-Demand Anodyne CACNA1H 47 39 O=C(c1ccccc1)c1cc(NC(=O)N2CC3(CC3)C2)ccc1F ZINC000880671693 DH On-Demand Anodyne NPY5R 18 40 O=C(c1ccccc1)c1cc(NC(=O)N2CC3(CC3)C2)ccc1F ZINC000880671693 DH On-Demand Anodyne EPHX2 35 47 O=C(c1cncc2[nH]ccc12)N1CCC(C2CCC2)CC1 ZINC000880671741 CG On-Demand Anodyne L3MBTL3 57 36 C[C@@H](CCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)N(C)C ZINC000880671751 DD On-Demand Anodyne MPO 59 40 CC(C)(C(=O)N1CC[C@@H](O)C(F)(F)C1)c1ccc(C(F)(F)F)cc1 ZINC000880671752 FG On-Demand Anodyne EPHX2 19 41 CC(C)(C(=O)N1CC[C@H](O)C(F)(F)C1)c1ccc(C(F)(F)F)cc1 ZINC000880671754 FG On-Demand Anodyne EPHX2 19 41 CC(C)(C(=O)N[C@@H]1C=CCC1)c1ccc(C(F)(F)F)cc1 ZINC000880671757 CH On-Demand Anodyne EPHX2 15 41 CC(C)(C(=O)N[C@H]1C=CCC1)c1ccc(C(F)(F)F)cc1 ZINC000880671759 CH On-Demand Anodyne EPHX2 15 41 O=C(NNc1ccnc(Cl)c1)c1ncsc1C1CC1 ZINC000880671764 CF On-Demand Reactive TYK2 53 35 CC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671773 FH On-Demand Anodyne CACNA1H 49 41 CC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671773 FH On-Demand Anodyne NPY2R 63 36 CC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671773 FH On-Demand Anodyne EPHX2 42 38 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671778 FD On-Demand Anodyne MLNR 54 32 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880671779 FD On-Demand Anodyne MLNR 54 32 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671780 FD On-Demand Anodyne MLNR 54 32 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880671781 FD On-Demand Anodyne MLNR 54 32 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@@H]21 ZINC000880671810 GH On-Demand Anodyne AVPR2 42 37 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@@H]21 ZINC000880671810 GH On-Demand Anodyne NPY2R 65 36 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@@H]21 ZINC000880671810 GH On-Demand Anodyne RBP4 53 34 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@H]21 ZINC000880671812 GH On-Demand Anodyne AVPR2 42 37 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@H]21 ZINC000880671812 GH On-Demand Anodyne NPY2R 65 36 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC[C@H]21 ZINC000880671812 GH On-Demand Anodyne RBP4 53 34 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC(CC#N)C3)ccn2)CC1 ZINC000880671817 GE On-Demand Mild GPR119 49 48 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000880671838 GG On-Demand Anodyne CACNA1H 50 39 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000880671838 GG On-Demand Anodyne NPY5R 26 40 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000880671838 GG On-Demand Anodyne EPHX2 40 43 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@@](O)(C(F)F)C2)ccc1F ZINC000880671845 GG On-Demand Anodyne CACNA1H 46 39 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@@](O)(C(F)F)C2)ccc1F ZINC000880671845 GG On-Demand Anodyne EPHX2 34 44 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@](O)(C(F)F)C2)ccc1F ZINC000880671846 GG On-Demand Anodyne CACNA1H 46 39 O=C(c1ccccc1)c1cc(NC(=O)N2CC[C@](O)(C(F)F)C2)ccc1F ZINC000880671846 GG On-Demand Anodyne EPHX2 34 44 O=C(COC1CC1)Nc1nc(-c2ccccc2C(F)(F)F)ns1 ZINC000880671908 EG On-Demand Anodyne MPL 50 38 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880671922 GH On-Demand Anodyne SLC6A3 36 42 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880671925 GH On-Demand Anodyne SLC6A3 36 42 C#CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880671991 GG On-Demand Mild CACNA1H 48 36 O=C(c1ccccc1)c1cc(NC(=O)N2C[C@@H](CO)[C@@H](CO)C2)ccc1F ZINC000880672000 FE On-Demand Anodyne RBP4 45 33 C[C@H](CCNC(=O)c1cccn2nccc12)N(C)C ZINC000880672012 CD On-Demand Anodyne POLR1A 49 39 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1F ZINC000880672013 GH On-Demand Anodyne CACNA1H 47 38 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(CC2)OCCCO3)ccc1F ZINC000880672013 GH On-Demand Anodyne EPHX2 38 42 C[C@@H](CCNC(=O)c1cccn2nccc12)N(C)C ZINC000880672014 CD On-Demand Anodyne POLR1A 49 39 CC(C)(C(=O)N1CC[C@@H](O)C(F)(F)C1)c1ccc(F)cc1F ZINC000880672025 DE On-Demand Anodyne PRCP 42 33 CC(C)(C(=O)N1CC[C@H](O)C(F)(F)C1)c1ccc(F)cc1F ZINC000880672026 DE On-Demand Anodyne PRCP 42 33 C[C@@H](CCNC(=O)C1CCC(S(C)(=O)=O)CC1)N(C)C ZINC000880672041 DD On-Demand Anodyne CHRNA4 20 42 O=C(COC1CC1)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880672080 DD On-Demand Anodyne OPRK1 17 40 O=C(COC1CC1)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880672080 DD On-Demand Anodyne SIGMAR1 27 44 O=C(COC1CC1)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880672080 DD On-Demand Anodyne MCHR1 29 40 O=C(COC1CC1)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880672081 DD On-Demand Anodyne OPRK1 17 40 O=C(COC1CC1)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880672081 DD On-Demand Anodyne SIGMAR1 27 44 O=C(COC1CC1)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880672081 DD On-Demand Anodyne MCHR1 29 40 CC(C)(C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672083 GG On-Demand Anodyne SIGMAR1 21 42 CC(C)(C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672083 GG On-Demand Anodyne CCR3 51 42 CC(C)(C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672083 GG On-Demand Anodyne MLNR 59 37 CC(C)(C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672083 GG On-Demand Anodyne MCHR1 32 43 CC(C)(C(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672083 GG On-Demand Anodyne CACNA1G 39 41 CC(C)(C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672084 GG On-Demand Anodyne SIGMAR1 21 42 CC(C)(C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672084 GG On-Demand Anodyne CCR3 51 42 CC(C)(C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672084 GG On-Demand Anodyne MLNR 59 37 CC(C)(C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672084 GG On-Demand Anodyne MCHR1 32 43 CC(C)(C(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1)c1ccc(F)cc1F ZINC000880672084 GG On-Demand Anodyne CACNA1G 39 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne OPRK1 19 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne AVPR1B 41 33 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne SIGMAR1 24 44 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne CCR3 35 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne MCHR1 33 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@@H](O)C3)cc1)C2 ZINC000880672091 GF On-Demand Anodyne CACNA1G 28 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne OPRK1 19 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne AVPR1B 41 33 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne SIGMAR1 24 44 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne CCR3 35 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne MCHR1 33 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(CN3CC[C@H](O)C3)cc1)C2 ZINC000880672093 GF On-Demand Anodyne CACNA1G 28 43 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC/C=C\CO)ccn2)CC1 ZINC000880672100 GD On-Demand Anodyne DRD3 15 40 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC/C=C\CO)ccn2)CC1 ZINC000880672100 GD On-Demand Anodyne GPR119 36 46 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC/C=C/CO)ccn2)CC1 ZINC000880672101 GD On-Demand Anodyne DRD3 15 40 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC/C=C/CO)ccn2)CC1 ZINC000880672101 GD On-Demand Anodyne GPR119 36 46 CC1(C)CC[C@@H](CC(=O)NCCc2ccnc3ccccc23)OC1 ZINC000880672108 EG On-Demand Anodyne MTNR1A 27 43 CC1(C)CC[C@@H](CC(=O)NCCc2ccnc3ccccc23)OC1 ZINC000880672108 EG On-Demand Anodyne MTNR1B 20 43 Cc1ccncc1CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880672110 DH On-Demand Anodyne NQO2 17 40 Cc1ccncc1CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880672111 DH On-Demand Anodyne NQO2 17 40 Cc1nc(C(C)C)ncc1C(=O)NCCc1ccnc2ccccc12 ZINC000880672119 EG On-Demand Anodyne MTNR1A 24 40 Cc1nc(C(C)C)ncc1C(=O)NCCc1ccnc2ccccc12 ZINC000880672119 EG On-Demand Anodyne MTNR1B 20 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672120 GF On-Demand Anodyne PAPA1_CARPA 49 56 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672120 GF On-Demand Anodyne CTSK 18 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672120 GF On-Demand Anodyne CTSL 32 56 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672120 GF On-Demand Anodyne CTSS 27 56 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672120 GF On-Demand Anodyne FPR1 44 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672121 GF On-Demand Anodyne PAPA1_CARPA 49 56 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672121 GF On-Demand Anodyne CTSK 18 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672121 GF On-Demand Anodyne CTSL 32 56 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672121 GF On-Demand Anodyne CTSS 27 56 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1cccc(F)c1 ZINC000880672121 GF On-Demand Anodyne FPR1 44 37 O=C(C[C@H]1CCNC1=O)NCc1ccc2occc2c1 ZINC000880672126 CD On-Demand Anodyne NOS2 63 33 O=C(C[C@@H]1CCNC1=O)NCc1ccc2occc2c1 ZINC000880672127 CD On-Demand Anodyne NOS2 63 33 CC[C@@H](C)CCNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880672156 CF On-Demand Anodyne PLD1 46 35 CC[C@@H](C)CCNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880672157 CF On-Demand Anodyne PLD1 46 35 C[C@@H](NC(=O)c1cc2cc(F)ccc2[nH]c1=O)C1(CO)CC1 ZINC000880672169 DD On-Demand Anodyne PLD1 37 40 C[C@H](NC(=O)c1cc2cc(F)ccc2[nH]c1=O)C1(CO)CC1 ZINC000880672170 DD On-Demand Anodyne PLD1 37 40 O=C1N[C@H]2CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)C[C@@H]2CO1 ZINC000880672189 GG On-Demand Anodyne RBP4 46 34 COc1ccc(N2C[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)CC2=O)cc1 ZINC000880672214 GD On-Demand Anodyne PDK1 47 36 COc1ccc(N2C[C@H](NC(=O)c3ccc(CN4CCOCC4)o3)CC2=O)cc1 ZINC000880672214 GD On-Demand Anodyne MCHR1 24 42 O=C(COC1CC1)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880672221 CD On-Demand Anodyne ROCK1 15 50 O=C(COC1CC1)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880672221 CD On-Demand Anodyne ROCK2 25 53 N#CCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880672225 EE On-Demand Mild DPP4 16 42 N#CCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880672225 EE On-Demand Mild PREP 45 47 N#CCC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880672225 EE On-Demand Mild LGMN 67 39 O=C(CN1CCCCS1(=O)=O)Nc1ccc2c(=O)[nH]ccc2c1 ZINC000880672228 EC On-Demand Anodyne ROCK2 23 46 O=C(NO[C@H]1CCCCO1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672230 FH On-Demand Anodyne EPHX2 17 40 O=C(NO[C@@H]1CCCCO1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672231 FH On-Demand Anodyne EPHX2 17 40 O=C(NCC1OCCCO1)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672232 FF On-Demand Anodyne PRMT3 46 34 O=C(Nc1ccc2c(=O)[nH]ccc2c1)[C@@H]1CCc2nncn2CC1 ZINC000880672246 DD On-Demand Anodyne ROCK2 23 48 O=C(Nc1ccc2c(=O)[nH]ccc2c1)[C@H]1CCc2nncn2CC1 ZINC000880672247 DD On-Demand Anodyne ROCK2 23 48 O=C(NNc1ccnc(Cl)c1)c1cnc(CC2CC2)s1 ZINC000880672248 DF On-Demand Reactive TYK2 45 34 COC(OC)[C@@H](C)NC(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672249 FG On-Demand Anodyne KCNK3 47 34 COC(OC)[C@H](C)NC(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672250 FG On-Demand Anodyne KCNK3 47 34 O=C1NCC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)O1 ZINC000880672253 GG On-Demand Anodyne CACNA1H 51 39 O=C1NCC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)O1 ZINC000880672253 GG On-Demand Anodyne EPHX2 33 40 O=C1NCC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)O1 ZINC000880672253 GG On-Demand Anodyne TRPM8 31 42 CN(Cc1ccc2nc(NC(=O)[C@H]3CCc4nncn4CC3)sc2c1)C1CC1 ZINC000880672260 GG On-Demand Anodyne LCK 15 40 CN(Cc1ccc2nc(NC(=O)[C@H]3CCc4nncn4CC3)sc2c1)C1CC1 ZINC000880672260 GG On-Demand Anodyne NMT1 39 40 CN(Cc1ccc2nc(NC(=O)[C@@H]3CCc4nncn4CC3)sc2c1)C1CC1 ZINC000880672261 GG On-Demand Anodyne LCK 15 40 CN(Cc1ccc2nc(NC(=O)[C@@H]3CCc4nncn4CC3)sc2c1)C1CC1 ZINC000880672261 GG On-Demand Anodyne NMT1 39 40 Cc1coc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880672268 DE On-Demand Anodyne SIGMAR1 21 49 Cc1coc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880672268 DE On-Demand Anodyne MCHR1 38 43 Cc1coc(C(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c1 ZINC000880672268 DE On-Demand Anodyne CACNA1I 29 42 Cc1coc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880672269 DE On-Demand Anodyne SIGMAR1 21 49 Cc1coc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880672269 DE On-Demand Anodyne MCHR1 38 43 Cc1coc(C(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c1 ZINC000880672269 DE On-Demand Anodyne CACNA1I 29 42 O=C(NCCc1ccnc2ccccc12)c1ccc(CN2CCOCC2)o1 ZINC000880672289 FF On-Demand Anodyne HPGDS 24 45 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2ccc3occc3c2)N1Cc1ccccc1 ZINC000880672292 GF On-Demand Anodyne F2 29 40 NC(=O)[C@@H]1CC[C@H](C(=O)NCc2ccc3occc3c2)N1Cc1ccccc1 ZINC000880672292 GF On-Demand Anodyne TMPRSS11D 64 35 C=CC(C)(C)CC(=O)NCCc1ccnc2ccccc12 ZINC000880672300 CG On-Demand Mild NQO2 27 40 C=CC(C)(C)CC(=O)NCCc1ccnc2ccccc12 ZINC000880672300 CG On-Demand Mild MTNR1A 38 47 C=CC(C)(C)CC(=O)NCCc1ccnc2ccccc12 ZINC000880672300 CG On-Demand Mild MTNR1B 28 47 O=C(NC/C=C/CO)c1ccc(OC(F)F)c(Cl)c1 ZINC000880672342 CE On-Demand Anodyne PDE4D 15 41 O=C(NC/C=C/CO)c1ccc(OC(F)F)c(Cl)c1 ZINC000880672342 CE On-Demand Anodyne ADCYAP1R1 52 30 O=C(NC/C=C\CO)c1ccc(OC(F)F)c(Cl)c1 ZINC000880672343 CE On-Demand Anodyne PDE4D 15 41 O=C(NC/C=C\CO)c1ccc(OC(F)F)c(Cl)c1 ZINC000880672343 CE On-Demand Anodyne ADCYAP1R1 52 30 COc1cccc(OC)c1CNC(=O)COC1CC1 ZINC000880672344 CD On-Demand Anodyne MTNR1A 50 36 COc1cccc(OC)c1CNC(=O)COC1CC1 ZINC000880672344 CD On-Demand Anodyne MTNR1B 46 36 COc1cccc(OC)c1CNC(=O)COC1CC1 ZINC000880672344 CD On-Demand Anodyne MBTPS1 40 33 CO[C@@](C)(CNC(=O)C[C@H]1CCNC1=O)COCc1ccccc1 ZINC000880672349 ED On-Demand Anodyne R1A_CVHSA 20 40 CO[C@@](C)(CNC(=O)C[C@@H]1CCNC1=O)COCc1ccccc1 ZINC000880672350 ED On-Demand Anodyne R1A_CVHSA 20 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne SIGMAR1 18 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne SSTR5 47 35 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne CCR3 31 44 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne MLNR 60 35 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne CXCR3 28 49 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne MCHR1 31 49 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672358 FE On-Demand Anodyne NAMPT 53 51 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne SIGMAR1 18 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne SSTR5 47 35 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne CCR3 31 44 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne MLNR 60 35 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne CXCR3 28 49 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne MCHR1 31 49 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cnc2cc[nH]c2c1 ZINC000880672359 FE On-Demand Anodyne NAMPT 53 51 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ccnc(Cl)c1)C2 ZINC000880672386 EF On-Demand Reactive MMP3 27 40 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ccnc(Cl)c1)C2 ZINC000880672386 EF On-Demand Reactive MMP8 18 40 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ccnc(Cl)c1)C2 ZINC000880672386 EF On-Demand Reactive TYK2 34 40 O=C(NNc1ccnc(Cl)c1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880672402 ED On-Demand Reactive TYK2 58 37 O=C(Nc1ccc(F)c(C(=O)c2ccccc2)c1)NN1CCCCC1 ZINC000880672407 EH On-Demand Anodyne EPHX2 23 43 N#CC1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880672412 FH On-Demand Mild CACNA1H 43 37 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1ccc2occc2c1 ZINC000880672494 CG On-Demand Anodyne NOS2 56 32 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880672503 EE On-Demand Anodyne SIGMAR1 19 41 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880672504 EE On-Demand Anodyne SIGMAR1 19 41 COc1cccc(OC)c1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880672506 FF On-Demand Anodyne HTR1A 17 43 COc1cccc(OC)c1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880672506 FF On-Demand Anodyne DRD2 19 42 COc1cccc(OC)c1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880672507 FF On-Demand Anodyne HTR1A 17 43 COc1cccc(OC)c1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880672507 FF On-Demand Anodyne DRD2 19 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672515 FE On-Demand Anodyne SIGMAR1 17 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672515 FE On-Demand Anodyne CCR3 20 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672515 FE On-Demand Anodyne MCHR1 17 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672516 FE On-Demand Anodyne SIGMAR1 17 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672516 FE On-Demand Anodyne CCR3 20 41 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)c1cccc2nsnc12 ZINC000880672516 FE On-Demand Anodyne MCHR1 17 42 O=C(c1ccccc1)c1cc(NC(=O)N2CC3(CCOC3)C2)ccc1F ZINC000880672542 FG On-Demand Anodyne CACNA1H 41 35 O=C(c1ccccc1)c1cc(NC(=O)N2CC3(CCOC3)C2)ccc1F ZINC000880672542 FG On-Demand Anodyne EPHX2 37 43 CC1(C)CC[C@@H](CC(=O)Nc2ccc3c(=O)[nH]ccc3c2)OC1 ZINC000880672550 DG On-Demand Anodyne ROCK2 23 47 CN(Cc1ccc2nc(NC(=O)COC3CC3)sc2c1)C1CC1 ZINC000880672556 EG On-Demand Anodyne LCK 21 43 CN(Cc1ccc2nc(NC(=O)COC3CC3)sc2c1)C1CC1 ZINC000880672556 EG On-Demand Anodyne CSNK1D 51 48 CN(Cc1ccc2nc(NC(=O)COC3CC3)sc2c1)C1CC1 ZINC000880672556 EG On-Demand Anodyne ITK 20 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672571 DC On-Demand Anodyne PAPA1_CARPA 42 50 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672571 DC On-Demand Anodyne CTSK 18 51 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672571 DC On-Demand Anodyne FPR1 40 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672574 DC On-Demand Anodyne PAPA1_CARPA 42 50 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672574 DC On-Demand Anodyne CTSK 18 51 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C\CO ZINC000880672574 DC On-Demand Anodyne FPR1 40 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672576 DC On-Demand Anodyne PAPA1_CARPA 42 50 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672576 DC On-Demand Anodyne CTSK 18 51 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672576 DC On-Demand Anodyne FPR1 40 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672579 DC On-Demand Anodyne PAPA1_CARPA 42 50 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672579 DC On-Demand Anodyne CTSK 18 51 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC/C=C/CO ZINC000880672579 DC On-Demand Anodyne FPR1 40 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H](O)C(F)(F)C1 ZINC000880672583 GD On-Demand Anodyne CELA1 19 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H](O)C(F)(F)C1 ZINC000880672583 GD On-Demand Anodyne GRIN2B 23 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H](O)C(F)(F)C1 ZINC000880672583 GD On-Demand Anodyne PREP 61 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H](O)C(F)(F)C1 ZINC000880672583 GD On-Demand Anodyne SLC12A5 52 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H](O)C(F)(F)C1 ZINC000880672583 GD On-Demand Anodyne Q9NAW4_PLAFA 25 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880672584 GD On-Demand Anodyne CELA1 19 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880672584 GD On-Demand Anodyne GRIN2B 23 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880672584 GD On-Demand Anodyne PREP 61 49 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880672584 GD On-Demand Anodyne SLC12A5 52 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880672584 GD On-Demand Anodyne Q9NAW4_PLAFA 25 40 CS(=O)(=O)C1CCC(C(=O)NCCc2ccnc3ccccc23)CC1 ZINC000880672593 FE On-Demand Anodyne NQO2 31 40 CS(=O)(=O)C1CCC(C(=O)NCCc2ccnc3ccccc23)CC1 ZINC000880672593 FE On-Demand Anodyne MTNR1A 53 49 CS(=O)(=O)C1CCC(C(=O)NCCc2ccnc3ccccc23)CC1 ZINC000880672593 FE On-Demand Anodyne MTNR1B 37 48 Cc1ccncc1CCNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880672595 DD On-Demand Anodyne MTNR1A 22 43 Cc1ccncc1CCNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880672595 DD On-Demand Anodyne MTNR1B 15 40 O=C(NC[C@H](O)c1cccc2ccccc12)c1ccc(CN2CCOCC2)o1 ZINC000880672603 GF On-Demand Anodyne HPGDS 23 40 O=C(NC[C@@H](O)c1cccc2ccccc12)c1ccc(CN2CCOCC2)o1 ZINC000880672604 GF On-Demand Anodyne HPGDS 23 40 CS(=O)(=O)C1CCC(C(=O)NC[C@@H](O)c2cccc3ccccc23)CC1 ZINC000880672612 GF On-Demand Anodyne KCNJ11 18 41 CS(=O)(=O)C1CCC(C(=O)NC[C@@H](O)c2cccc3ccccc23)CC1 ZINC000880672612 GF On-Demand Anodyne MTNR1A 22 43 CS(=O)(=O)C1CCC(C(=O)NC[C@H](O)c2cccc3ccccc23)CC1 ZINC000880672614 GF On-Demand Anodyne KCNJ11 18 41 CS(=O)(=O)C1CCC(C(=O)NC[C@H](O)c2cccc3ccccc23)CC1 ZINC000880672614 GF On-Demand Anodyne MTNR1A 22 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnccc1C)C2 ZINC000880672630 DF On-Demand Anodyne NQO2 42 46 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnccc1C)C2 ZINC000880672630 DF On-Demand Anodyne MTNR1A 81 48 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnccc1C)C2 ZINC000880672630 DF On-Demand Anodyne MTNR1B 65 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(CC#N)C1 ZINC000880672640 DD On-Demand Mild PAPA1_CARPA 39 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(CC#N)C1 ZINC000880672642 DD On-Demand Mild PAPA1_CARPA 39 46 CN(Cc1ccc2nc(NC(=O)C[C@H]3CCNC3=O)sc2c1)C1CC1 ZINC000880672665 FE On-Demand Anodyne CSNK1D 46 45 CN(Cc1ccc2nc(NC(=O)C[C@H]3CCNC3=O)sc2c1)C1CC1 ZINC000880672665 FE On-Demand Anodyne ITK 15 42 CN(Cc1ccc2nc(NC(=O)C[C@@H]3CCNC3=O)sc2c1)C1CC1 ZINC000880672673 FE On-Demand Anodyne CSNK1D 46 45 CN(Cc1ccc2nc(NC(=O)C[C@@H]3CCNC3=O)sc2c1)C1CC1 ZINC000880672673 FE On-Demand Anodyne ITK 15 42 O=C(NNc1ccnc(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880672696 DD On-Demand Reactive TYK2 51 35 O=C(NNc1ccnc(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880672697 DD On-Demand Reactive TYK2 51 35 C[C@@]1(C(=O)NNc2ccnc(Cl)c2)OCCc2ccccc21 ZINC000880672706 DF On-Demand Reactive G2YM83_BOTF4 45 34 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1(CO)CC1 ZINC000880672709 DD On-Demand Anodyne KCNQ2 48 34 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@]3(C2)CC3(F)F)ccc1F ZINC000880672720 GJ On-Demand Anodyne CACNA1H 45 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@]3(C2)CC3(F)F)ccc1F ZINC000880672720 GJ On-Demand Anodyne EPHX2 39 47 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@]3(C2)CC3(F)F)ccc1F ZINC000880672721 GJ On-Demand Anodyne CACNA1H 45 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@]3(C2)CC3(F)F)ccc1F ZINC000880672721 GJ On-Demand Anodyne EPHX2 39 47 C[C@@H](NC(=O)c1ncsc1C1CC1)c1cscn1 ZINC000880672731 CF On-Demand Anodyne MAP1 53 37 C[C@H](NC(=O)c1ncsc1C1CC1)c1cscn1 ZINC000880672732 CF On-Demand Anodyne MAP1 53 37 C[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1(CO)CC1 ZINC000880672742 DF On-Demand Anodyne PDE4D 18 40 C[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1(CO)CC1 ZINC000880672743 DF On-Demand Anodyne PDE4D 18 40 CCN1CC[C@H](N(CC)C(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880672776 EE On-Demand Anodyne CCR5 36 41 CCN1CC[C@@H](N(CC)C(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880672777 EE On-Demand Anodyne CCR5 36 41 C[C@H]1CCOCCN1C(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672791 FH On-Demand Anodyne EPHX2 20 42 C[C@@H]1CCOCCN1C(=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880672792 FH On-Demand Anodyne EPHX2 20 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne DRD4 27 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne ACHE 37 50 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne HTR4 60 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne SIGMAR1 28 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne SSTR5 79 38 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne CCR3 37 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne CXCR3 29 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne MCHR1 38 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc2cc[nH]c2c1 ZINC000880672801 EF On-Demand Anodyne CACNA1I 79 50 COC[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672805 FE On-Demand Anodyne DRD4 43 33 COC[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672805 FE On-Demand Anodyne CASR 39 45 COC[C@@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672805 FE On-Demand Anodyne PSMB8 40 39 COC[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672806 FE On-Demand Anodyne DRD4 43 33 COC[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672806 FE On-Demand Anodyne CASR 39 45 COC[C@H](NC(=O)c1ccc(CN2CCOCC2)o1)c1cccc(OC)c1 ZINC000880672806 FE On-Demand Anodyne PSMB8 40 39 COC[C@H](NC(=O)CN1CCCCS1(=O)=O)c1cccc(OC)c1 ZINC000880672816 FC On-Demand Anodyne DRD4 40 31 COC[C@@H](NC(=O)CN1CCCCS1(=O)=O)c1cccc(OC)c1 ZINC000880672817 FC On-Demand Anodyne DRD4 40 31 O=C(c1ccccc1)c1cc(NC(=O)N2CCCC3(C2)OCCO3)ccc1F ZINC000880672830 GG On-Demand Anodyne CACNA1H 41 36 O=C(c1ccccc1)c1cc(NC(=O)N2CCCC3(C2)OCCO3)ccc1F ZINC000880672830 GG On-Demand Anodyne EPHX2 41 46 COC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)c1cccc(OC)c1 ZINC000880672838 GF On-Demand Anodyne DRD4 42 35 COC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)c1cccc(OC)c1 ZINC000880672838 GF On-Demand Anodyne KCNQ2 50 46 COC[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)c1cccc(OC)c1 ZINC000880672839 GF On-Demand Anodyne DRD4 42 35 COC[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)c1cccc(OC)c1 ZINC000880672839 GF On-Demand Anodyne KCNQ2 50 46 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne DRD4 15 47 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne ACHE 22 43 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne HTR4 57 47 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne SIGMAR1 15 40 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne SSTR5 50 36 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880672848 FF On-Demand Anodyne CACNA1I 71 46 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne DRD4 31 45 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne ACHE 42 50 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne HTR4 63 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne SIGMAR1 33 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne SSTR5 44 34 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne CCR3 25 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne MCHR1 22 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncccc1-c1ccccn1 ZINC000880672852 GG On-Demand Anodyne CACNA1I 64 43 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne DRD2 15 48 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne DRD4 37 48 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne ACHE 42 48 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne HTR4 69 45 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne SIGMAR1 30 42 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne SSTR5 69 40 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne CCR3 30 41 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne PDK1 33 40 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne MCHR1 43 42 Cc1coc(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880672855 DF On-Demand Anodyne CACNA1I 89 56 COC[C@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672920 FE On-Demand Anodyne CCR5 17 42 COC[C@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672920 FE On-Demand Anodyne MTNR1A 48 47 COC[C@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672920 FE On-Demand Anodyne MTNR1B 42 47 COC[C@@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672921 FE On-Demand Anodyne CCR5 17 42 COC[C@@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672921 FE On-Demand Anodyne MTNR1A 48 47 COC[C@@H](NC(=O)C1CCC(S(C)(=O)=O)CC1)c1cccc(OC)c1 ZINC000880672921 FE On-Demand Anodyne MTNR1B 42 47 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@H](C3OCCO3)C2)ccc1F ZINC000880672959 GH On-Demand Anodyne RBP4 52 33 O=C(c1ccccc1)c1cc(NC(=O)N2CCC[C@@H](C3OCCO3)C2)ccc1F ZINC000880672960 GH On-Demand Anodyne RBP4 52 33 COC[C@H](NC(=O)[C@H]1CCc2nncn2CC1)c1cccc(OC)c1 ZINC000880672962 ED On-Demand Anodyne DRD4 43 33 COC[C@H](NC(=O)[C@@H]1CCc2nncn2CC1)c1cccc(OC)c1 ZINC000880672963 ED On-Demand Anodyne DRD4 43 33 COC[C@@H](NC(=O)[C@@H]1CCc2nncn2CC1)c1cccc(OC)c1 ZINC000880672964 ED On-Demand Anodyne DRD4 43 33 COC[C@@H](NC(=O)[C@H]1CCc2nncn2CC1)c1cccc(OC)c1 ZINC000880672965 ED On-Demand Anodyne DRD4 43 33 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne ACHE 22 45 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne HTR4 68 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne SIGMAR1 19 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne SSTR5 40 34 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne CCR3 18 49 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cncc2[nH]ccc12 ZINC000880672979 EF On-Demand Anodyne CACNA1I 66 43 CCO[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880672995 DE On-Demand Anodyne NQO2 27 40 CCO[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880672995 DE On-Demand Anodyne MTNR1A 41 44 CCO[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880672996 DE On-Demand Anodyne NQO2 27 40 CCO[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880672996 DE On-Demand Anodyne MTNR1A 41 44 CCO[C@@H]1C[C@@H](NC(=O)c2cc3ccccc3cc2F)C1 ZINC000880673003 CG On-Demand Anodyne HTR4 31 41 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(Cc3ccncc3)CC2)CC1 ZINC000880673017 GE On-Demand Anodyne ACHE 30 45 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(Cc3ccncc3)CC2)CC1 ZINC000880673017 GE On-Demand Anodyne HTR4 50 41 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(Cc3ccncc3)CC2)CC1 ZINC000880673017 GE On-Demand Anodyne SIGMAR1 26 45 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(Cc3ccncc3)CC2)CC1 ZINC000880673017 GE On-Demand Anodyne CCR3 16 43 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(Cc3ccncc3)CC2)CC1 ZINC000880673017 GE On-Demand Anodyne CACNA1I 66 43 O=C(CN1CCCCS1(=O)=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673018 GC On-Demand Anodyne ACHE 25 44 O=C(CN1CCCCS1(=O)=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673018 GC On-Demand Anodyne SIGMAR1 24 42 O=C(CN1CCCCS1(=O)=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673018 GC On-Demand Anodyne CACNA1I 60 39 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880673035 GG On-Demand Anodyne CACNA1H 50 38 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)C1 ZINC000880673035 GG On-Demand Anodyne EPHX2 36 43 O=C1CC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)CN1 ZINC000880673056 GG On-Demand Anodyne CACNA1H 50 39 O=C1CC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)CN1 ZINC000880673056 GG On-Demand Anodyne EPHX2 27 40 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(CCCO)CC2)ccc1F ZINC000880673057 GI On-Demand Anodyne EPHX2 34 43 O=C(c1ccccc1)c1cc(NC(=O)N2CCC(CCCO)CC2)ccc1F ZINC000880673057 GI On-Demand Anodyne ST14 40 33 O=C(c1ccccc1)c1cc(NC(=O)N2CCN3C(=O)OCC[C@H]3C2)ccc1F ZINC000880673060 GG On-Demand Anodyne SMO 22 40 O=C(c1ccccc1)c1cc(NC(=O)N2CCN3C(=O)OCC[C@@H]3C2)ccc1F ZINC000880673061 GG On-Demand Anodyne SMO 22 40 COC[C@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673075 FD On-Demand Anodyne CCR5 16 40 COC[C@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673075 FD On-Demand Anodyne MTNR1A 30 42 COC[C@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673075 FD On-Demand Anodyne MTNR1B 33 42 COC[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673076 FD On-Demand Anodyne CCR5 16 40 COC[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673076 FD On-Demand Anodyne MTNR1A 30 42 COC[C@@H](NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1cccc(OC)c1 ZINC000880673076 FD On-Demand Anodyne MTNR1B 33 42 O=C(Cc1ccccc1N1CCCC1=O)N1CC[C@H](N2CCOC2=O)C1 ZINC000880673080 FD On-Demand Anodyne OXTR 18 43 O=C(Cc1ccccc1N1CCCC1=O)N1CC[C@@H](N2CCOC2=O)C1 ZINC000880673081 FD On-Demand Anodyne OXTR 18 43 CCN1CC[C@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673106 EF On-Demand Anodyne CCR5 15 44 CCN1CC[C@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673106 EF On-Demand Anodyne S1PR1 15 63 CCN1CC[C@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673106 EF On-Demand Anodyne PDK1 47 37 CCN1CC[C@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673106 EF On-Demand Anodyne MCHR1 20 41 CCN1CC[C@@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673107 EF On-Demand Anodyne CCR5 15 44 CCN1CC[C@@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673107 EF On-Demand Anodyne S1PR1 15 63 CCN1CC[C@@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673107 EF On-Demand Anodyne PDK1 47 37 CCN1CC[C@@H](N(CC)C(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673107 EF On-Demand Anodyne MCHR1 20 41 C=CC(C)(C)CC(=O)N[C@@H](COC)c1cccc(OC)c1 ZINC000880673116 CG On-Demand Mild MTNR1A 34 42 C=CC(C)(C)CC(=O)N[C@@H](COC)c1cccc(OC)c1 ZINC000880673116 CG On-Demand Mild MTNR1B 37 42 C=CC(C)(C)CC(=O)N[C@H](COC)c1cccc(OC)c1 ZINC000880673117 CG On-Demand Mild MTNR1A 34 42 C=CC(C)(C)CC(=O)N[C@H](COC)c1cccc(OC)c1 ZINC000880673117 CG On-Demand Mild MTNR1B 37 42 COC[C@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673124 EG On-Demand Anodyne DRD4 43 33 COC[C@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673124 EG On-Demand Anodyne PTGER3 54 41 COC[C@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673124 EG On-Demand Anodyne TACR3 17 46 COC[C@@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673125 EG On-Demand Anodyne DRD4 43 33 COC[C@@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673125 EG On-Demand Anodyne PTGER3 54 41 COC[C@@H](NC(=O)c1cc(C)cnc1Cl)c1cccc(OC)c1 ZINC000880673125 EG On-Demand Anodyne TACR3 17 46 COC[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673160 FF On-Demand Anodyne DRD4 41 32 COC[C@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673160 FF On-Demand Anodyne UTS2 37 40 COC[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673161 FF On-Demand Anodyne DRD4 41 32 COC[C@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673161 FF On-Demand Anodyne UTS2 37 40 COC[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673162 FF On-Demand Anodyne DRD4 41 32 COC[C@@H](NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673162 FF On-Demand Anodyne UTS2 37 40 COC[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673163 FF On-Demand Anodyne DRD4 41 32 COC[C@@H](NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1)c1cccc(OC)c1 ZINC000880673163 FF On-Demand Anodyne UTS2 37 40 COC[C@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673166 EG On-Demand Anodyne PTGER3 49 41 COC[C@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673166 EG On-Demand Anodyne ROCK1 20 41 COC[C@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673166 EG On-Demand Anodyne MTNR1A 15 40 COC[C@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673166 EG On-Demand Anodyne MTNR1B 15 40 COC[C@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673166 EG On-Demand Anodyne GCK 17 40 COC[C@@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673167 EG On-Demand Anodyne PTGER3 49 41 COC[C@@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673167 EG On-Demand Anodyne ROCK1 20 41 COC[C@@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673167 EG On-Demand Anodyne MTNR1A 15 40 COC[C@@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673167 EG On-Demand Anodyne MTNR1B 15 40 COC[C@@H](NC(=O)c1cnc(C(C)C)nc1C)c1cccc(OC)c1 ZINC000880673167 EG On-Demand Anodyne GCK 17 40 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H](N2CCOC2=O)C1 ZINC000880673171 FF On-Demand Anodyne L3MBTL3 46 36 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@@H](N2CCOC2=O)C1 ZINC000880673172 FF On-Demand Anodyne L3MBTL3 46 36 CCN1CC[C@@H](N(CC)C(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)C1 ZINC000880673195 GH On-Demand Anodyne CCR5 17 44 CCN1CC[C@H](N(CC)C(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)C1 ZINC000880673196 GH On-Demand Anodyne CCR5 17 44 CCN1CC[C@@H](N(CC)C(=O)Cc2c(Br)cnn2C)C1 ZINC000880673210 ED On-Demand Anodyne CCR5 26 40 CCN1CC[C@H](N(CC)C(=O)Cc2c(Br)cnn2C)C1 ZINC000880673211 ED On-Demand Anodyne CCR5 26 40 O=C1NC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)CO1 ZINC000880673219 GG On-Demand Anodyne CACNA1H 53 39 O=C1NC2(CCN(C(=O)Nc3ccc(F)c(C(=O)c4ccccc4)c3)CC2)CO1 ZINC000880673219 GG On-Demand Anodyne EPHX2 22 40 CCN1CC[C@H](N(CC)C(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880673233 EE On-Demand Anodyne PLD1 40 37 CCN1CC[C@H](N(CC)C(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880673233 EE On-Demand Anodyne WNT3A 40 35 CCN1CC[C@@H](N(CC)C(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880673234 EE On-Demand Anodyne PLD1 40 37 CCN1CC[C@@H](N(CC)C(=O)c2cc3cc(F)ccc3[nH]c2=O)C1 ZINC000880673234 EE On-Demand Anodyne WNT3A 40 35 COCc1n[nH]c(CNC(=O)CC[C@H]2CCc3ccccc32)n1 ZINC000880673249 DE On-Demand Anodyne NQO2 19 41 COCc1n[nH]c(CNC(=O)CC[C@H]2CCc3ccccc32)n1 ZINC000880673249 DE On-Demand Anodyne MTNR1B 19 40 COCc1n[nH]c(CNC(=O)CC[C@@H]2CCc3ccccc32)n1 ZINC000880673250 DE On-Demand Anodyne NQO2 19 41 COCc1n[nH]c(CNC(=O)CC[C@@H]2CCc3ccccc32)n1 ZINC000880673250 DE On-Demand Anodyne MTNR1B 19 40 CCO[C@@H]1C[C@@H](NC(=O)[C@@H]2C[C@]2(C)c2ccccc2)C1 ZINC000880673308 CF On-Demand Anodyne TIMP3 65 35 CCO[C@@H]1C[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880673311 ED On-Demand Anodyne TIMP3 66 36 CCO[C@@H]1C[C@@H](NC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880673324 CF On-Demand Anodyne TIMP3 71 36 CC[C@@H](Nc1cccnc1Cl)C(=O)Nc1nccc(C)c1C1CC1 ZINC000880673335 EI On-Demand Anodyne G2YM83_BOTF4 68 36 CC[C@H](Nc1cccnc1Cl)C(=O)Nc1nccc(C)c1C1CC1 ZINC000880673336 EI On-Demand Anodyne G2YM83_BOTF4 68 36 COC[C@@H](NC(=O)c1nnn(C)n1)c1cccc(OC)c1 ZINC000880673344 CC On-Demand Anodyne DRD4 41 31 COC[C@H](NC(=O)c1nnn(C)n1)c1cccc(OC)c1 ZINC000880673345 CC On-Demand Anodyne DRD4 41 31 COC[C@H](NC(=O)c1c2c(nn1C)CCSC2)c1cccc(OC)c1 ZINC000880673354 FE On-Demand Anodyne DRD4 42 32 COC[C@@H](NC(=O)c1c2c(nn1C)CCSC2)c1cccc(OC)c1 ZINC000880673355 FE On-Demand Anodyne DRD4 42 32 COC(=O)C12CC(CN1C(=O)c1cc(-c3ccc(OC)cc3)on1)C2 ZINC000880673378 EE On-Demand Anodyne PDK1 42 31 CCO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880673379 DE On-Demand Anodyne GABRA1 19 43 CCO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880673379 DE On-Demand Anodyne MPO 54 35 CCO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880673379 DE On-Demand Anodyne GABRA2 16 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccc2nsnc12 ZINC000880673400 FF On-Demand Anodyne DRD4 22 46 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccc2nsnc12 ZINC000880673400 FF On-Demand Anodyne ACHE 31 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccc2nsnc12 ZINC000880673400 FF On-Demand Anodyne HTR4 70 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccc2nsnc12 ZINC000880673400 FF On-Demand Anodyne CCR3 22 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccc2nsnc12 ZINC000880673400 FF On-Demand Anodyne CACNA1I 64 42 CCO[C@@H]1C[C@@H](NC(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880673426 EG On-Demand Anodyne INHA 77 39 CCO[C@@H]1C[C@@H](NC(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880673426 EG On-Demand Anodyne MTNR1B 23 41 C#CCN(CC(=O)OC(C)(C)C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673443 FE On-Demand Mild MPO 43 33 O=C(NCCCN1CCOC1=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880673460 GG On-Demand Anodyne CCR3 40 41 O=C(NCCCN1CCOC1=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880673460 GG On-Demand Anodyne CHRNA7 15 41 O=C(NCCCN1CCOC1=O)Nc1ccc(F)c(C(=O)c2ccccc2)c1 ZINC000880673460 GG On-Demand Anodyne EPHX2 20 42 COC[C@H](NC(=O)c1cc(C)co1)c1cccc(OC)c1 ZINC000880673461 CF On-Demand Anodyne MTNR1A 31 40 COC[C@H](NC(=O)c1cc(C)co1)c1cccc(OC)c1 ZINC000880673461 CF On-Demand Anodyne MTNR1B 32 40 COC[C@@H](NC(=O)c1cc(C)co1)c1cccc(OC)c1 ZINC000880673462 CF On-Demand Anodyne MTNR1A 31 40 COC[C@@H](NC(=O)c1cc(C)co1)c1cccc(OC)c1 ZINC000880673462 CF On-Demand Anodyne MTNR1B 32 40 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880673467 GH On-Demand Anodyne CACNA1H 48 37 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880673467 GH On-Demand Anodyne NPY2R 48 36 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880673467 GH On-Demand Anodyne EPHX2 51 38 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(=O)c3ccccc3)c2)CC1 ZINC000880673467 GH On-Demand Anodyne SCD1 15 55 COC[C@H](NC(=O)COC1CC1)c1cccc(OC)c1 ZINC000880673479 CD On-Demand Anodyne MTNR1A 37 40 COC[C@H](NC(=O)COC1CC1)c1cccc(OC)c1 ZINC000880673479 CD On-Demand Anodyne MTNR1B 39 40 COC[C@@H](NC(=O)COC1CC1)c1cccc(OC)c1 ZINC000880673480 CD On-Demand Anodyne MTNR1A 37 40 COC[C@@H](NC(=O)COC1CC1)c1cccc(OC)c1 ZINC000880673480 CD On-Demand Anodyne MTNR1B 39 40 O=C(C[C@@H]1C[C@H]1C1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673524 EF On-Demand Anodyne ACHE 25 46 O=C(C[C@@H]1C[C@H]1C1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673524 EF On-Demand Anodyne HTR4 40 39 O=C(C[C@@H]1C[C@H]1C1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673524 EF On-Demand Anodyne SIGMAR1 28 42 O=C(C[C@@H]1C[C@H]1C1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673524 EF On-Demand Anodyne CACNA1I 62 41 COCc1n[nH]c(CNC(=O)c2sc(-c3ccc(F)c(C)c3)nc2C)n1 ZINC000880673528 GF On-Demand Anodyne SCD1 24 44 COCc1n[nH]c(CNC(=O)c2sc(-c3ccc(F)c(C)c3)nc2C)n1 ZINC000880673528 GF On-Demand Anodyne SCD 23 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne DRD4 26 48 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne ACHE 38 48 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne HTR4 71 48 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne SIGMAR1 28 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne SSTR5 52 35 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne CCR3 23 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cccn2nccc12 ZINC000880673536 EE On-Demand Anodyne CACNA1I 65 44 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne HTR1D 21 41 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne HTR1B 19 41 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne GRIN2B 17 46 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne SIGMAR1 21 48 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne CCR3 63 43 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne MCHR1 21 41 O=C(NCC1CCN(Cc2ccncc2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673594 GF On-Demand Anodyne CACNA1I 57 38 COCc1n[nH]c(CNC(=O)c2sc(-c3ccc(C)cc3F)nc2C)n1 ZINC000880673617 GF On-Demand Anodyne SCD1 25 45 COCc1n[nH]c(CNC(=O)c2sc(-c3ccc(C)cc3F)nc2C)n1 ZINC000880673617 GF On-Demand Anodyne SCD 23 45 CCO[C@@H]1C[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1 ZINC000880673627 ED On-Demand Anodyne PAPA1_CARPA 34 44 CCO[C@@H]1C[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1 ZINC000880673627 ED On-Demand Anodyne CTSK 16 48 CCO[C@@H]1C[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1 ZINC000880673628 ED On-Demand Anodyne PAPA1_CARPA 34 44 CCO[C@@H]1C[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1 ZINC000880673628 ED On-Demand Anodyne CTSK 16 48 COC[C@@H](NC(=O)c1nccnc1SC)c1cccc(OC)c1 ZINC000880673632 EE On-Demand Anodyne MTNR1A 19 40 COC[C@@H](NC(=O)c1nccnc1SC)c1cccc(OC)c1 ZINC000880673632 EE On-Demand Anodyne MTNR1B 23 40 COC[C@H](NC(=O)c1nccnc1SC)c1cccc(OC)c1 ZINC000880673633 EE On-Demand Anodyne MTNR1A 19 40 COC[C@H](NC(=O)c1nccnc1SC)c1cccc(OC)c1 ZINC000880673633 EE On-Demand Anodyne MTNR1B 23 40 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne DRD4 20 44 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne ACHE 33 52 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne HTR4 53 44 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne SIGMAR1 25 41 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne SSTR5 45 36 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne CCR3 17 40 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne PLD1 40 34 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673638 GF On-Demand Anodyne CACNA1I 70 47 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne DRD4 20 44 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne ACHE 33 52 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne HTR4 53 44 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne SIGMAR1 25 41 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne SSTR5 45 36 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne CCR3 17 40 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne PLD1 40 34 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(Cc4ccncc4)CC3)cc2)N1 ZINC000880673639 GF On-Demand Anodyne CACNA1I 70 47 CCO[C@@H]1C[C@@H](NC(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880673648 DF On-Demand Anodyne PDK1 49 38 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(C2)OCCO3)ccc1F ZINC000880673649 FG On-Demand Anodyne CACNA1H 42 38 O=C(c1ccccc1)c1cc(NC(=O)N2CCC3(C2)OCCO3)ccc1F ZINC000880673649 FG On-Demand Anodyne EPHX2 40 46 CC1(C)CC[C@@H](CC(=O)NCC2CCN(Cc3ccncc3)CC2)OC1 ZINC000880673651 FG On-Demand Anodyne ACHE 28 42 CC1(C)CC[C@@H](CC(=O)NCC2CCN(Cc3ccncc3)CC2)OC1 ZINC000880673651 FG On-Demand Anodyne CACNA1I 67 42 CCO[C@@H]1C[C@@H](NC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880673654 CD On-Demand Anodyne SSTR5 41 37 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne ACHE 37 44 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne SIGMAR1 29 48 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne SSTR5 42 37 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne CCR3 66 44 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne CACNA1G 43 41 CC(C)(C(=O)NCC1CCN(Cc2ccncc2)CC1)c1ccc(F)cc1F ZINC000880673655 GH On-Demand Anodyne CACNA1I 78 42 CCO[C@@H]1C[C@@H](NC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880673656 DD On-Demand Anodyne SSTR5 49 34 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673672 GH On-Demand Anodyne ACHE 48 52 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673672 GH On-Demand Anodyne HTR4 33 40 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673672 GH On-Demand Anodyne SIGMAR1 40 38 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673672 GH On-Demand Anodyne CACNA1I 45 38 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673673 GH On-Demand Anodyne ACHE 48 52 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673673 GH On-Demand Anodyne HTR4 33 40 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673673 GH On-Demand Anodyne SIGMAR1 40 38 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673673 GH On-Demand Anodyne CACNA1I 45 38 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cncn1C ZINC000880673690 EF On-Demand Anodyne SOAT1 23 40 C#CCC1(O)CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)CC1 ZINC000880673692 FF On-Demand Mild EPHX2 29 42 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne ADORA1 15 67 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne DHODH 20 48 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne P2RY12 153 39 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne ADORA2A 15 52 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne CCR8 27 41 CCOC(=O)N1CCC(C(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)CC1 ZINC000880673693 JJ On-Demand Anodyne RORC 22 52 O=C(Nc1cnc2c(F)cccc2c1)c1ccc(CN2CCOCC2)o1 ZINC000880673698 FG On-Demand Anodyne EPHX2 18 41 O=C(Nc1cnc2c(F)cccc2c1)c1ccc(CN2CCOCC2)o1 ZINC000880673698 FG On-Demand Anodyne STAT6 58 34 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)CC1 ZINC000880673702 EH On-Demand Anodyne EPHX2 49 39 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)CC1 ZINC000880673702 EH On-Demand Anodyne RBP4 36 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)CC1 ZINC000880673702 EH On-Demand Anodyne SCD1 15 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)CC1 ZINC000880673702 EH On-Demand Anodyne KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)CC1 ZINC000880673702 EH On-Demand Anodyne KCNK9 29 43 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1cc(F)ccn1 ZINC000880673732 CE On-Demand Anodyne TYK2 47 34 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)Nc1cc(F)ccn1 ZINC000880673733 CE On-Demand Anodyne TYK2 47 34 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1cc(F)ccn1 ZINC000880673734 CE On-Demand Anodyne TYK2 47 34 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)Nc1cc(F)ccn1 ZINC000880673735 CE On-Demand Anodyne TYK2 47 34 N#C[C@@H]1CCCC[C@H]1NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880673743 DE On-Demand Mild SSTR3 31 44 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880673744 DE On-Demand Mild SSTR3 31 44 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880673745 DE On-Demand Mild SSTR3 31 44 N#C[C@@H]1CCCC[C@H]1NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880673746 DE On-Demand Mild SSTR3 31 44 N#C[C@@H]1CCCC[C@@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673749 DF On-Demand Mild GABRA1 19 46 N#C[C@@H]1CCCC[C@@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673749 DF On-Demand Mild GABRA2 17 46 N#C[C@@H]1CCCC[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673750 DF On-Demand Mild GABRA1 19 46 N#C[C@@H]1CCCC[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673750 DF On-Demand Mild GABRA2 17 46 N#C[C@H]1CCCC[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673751 DF On-Demand Mild GABRA1 19 46 N#C[C@H]1CCCC[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673751 DF On-Demand Mild GABRA2 17 46 N#C[C@H]1CCCC[C@@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673752 DF On-Demand Mild GABRA1 19 46 N#C[C@H]1CCCC[C@@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880673752 DF On-Demand Mild GABRA2 17 46 CCn1ccc(NC(=O)c2cc(Br)ccc2C2CC2)n1 ZINC000880673770 EH On-Demand Anodyne HTR1F 66 35 CCn1ccc(NC(=O)c2cc(Br)ccc2C2CC2)n1 ZINC000880673770 EH On-Demand Anodyne SORT1 16 42 O=C(Nc1cc(F)ccn1)c1ncsc1C1CC1 ZINC000880673772 CF On-Demand Anodyne MAP1 79 42 O=C(Nc1cc(F)ccn1)c1ncsc1C1CC1 ZINC000880673772 CF On-Demand Anodyne TYK2 60 36 CC[C@@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673783 EH On-Demand Anodyne ACHE 27 43 CC[C@@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673783 EH On-Demand Anodyne SIGMAR1 25 41 CC[C@@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673783 EH On-Demand Anodyne SSTR5 46 33 CC[C@@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673783 EH On-Demand Anodyne CACNA1I 65 43 CC[C@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673784 EH On-Demand Anodyne ACHE 27 43 CC[C@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673784 EH On-Demand Anodyne SIGMAR1 25 41 CC[C@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673784 EH On-Demand Anodyne SSTR5 46 33 CC[C@H]1CCC[C@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673784 EH On-Demand Anodyne CACNA1I 65 43 CC[C@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673785 EH On-Demand Anodyne ACHE 27 43 CC[C@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673785 EH On-Demand Anodyne SIGMAR1 25 41 CC[C@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673785 EH On-Demand Anodyne SSTR5 46 33 CC[C@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673785 EH On-Demand Anodyne CACNA1I 65 43 CC[C@@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673786 EH On-Demand Anodyne ACHE 27 43 CC[C@@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673786 EH On-Demand Anodyne SIGMAR1 25 41 CC[C@@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673786 EH On-Demand Anodyne SSTR5 46 33 CC[C@@H]1CCC[C@@]1(C)C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673786 EH On-Demand Anodyne CACNA1I 65 43 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild ACHE 41 48 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild HTR4 44 41 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild GRIN2B 22 43 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild SIGMAR1 28 44 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild SSTR5 45 36 C=CC(C)(C)CC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880673799 DG On-Demand Mild CACNA1I 80 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H](C(C)(C)O)C1 ZINC000880673802 FG On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H](C(C)(C)O)C1 ZINC000880673802 FG On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](C(C)(C)O)C1 ZINC000880673803 FG On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](C(C)(C)O)C1 ZINC000880673803 FG On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)COCCO2 ZINC000880673804 GG On-Demand Anodyne EPHX2 33 51 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)COCCO2 ZINC000880673804 GG On-Demand Anodyne TRPM8 31 42 O=C(Nc1cc(F)ccn1)c1cnn(CC2CCCC2)c1 ZINC000880673810 CF On-Demand Anodyne MAPK14 18 40 O=C(Nc1cc(F)ccn1)c1cnn(CC2CCCC2)c1 ZINC000880673810 CF On-Demand Anodyne RPS6KA3 16 43 CCn1ncc(NC(=O)Nc2c(OC)cccc2OC(F)(F)F)c1C ZINC000880673813 FH On-Demand Anodyne P2RY1 37 40 COCC1CC(NC(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673815 EG On-Demand Anodyne KCNK3 30 41 COCC1CC(NC(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673815 EG On-Demand Anodyne KCNK9 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN([S@@](C)(=N)=O)CC1 ZINC000880673821 GE On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN([S@@](C)(=N)=O)CC1 ZINC000880673821 GE On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN([S@](C)(=N)=O)CC1 ZINC000880673822 GE On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN([S@](C)(=N)=O)CC1 ZINC000880673822 GE On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)NN1CCS(=O)(=O)CC1 ZINC000880673834 GD On-Demand Anodyne KCNK3 24 41 COc1cccc(OC(F)(F)F)c1NC(=O)NN1CCS(=O)(=O)CC1 ZINC000880673834 GD On-Demand Anodyne KCNK9 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880673840 GH On-Demand Anodyne EPHX2 41 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880673840 GH On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880673840 GH On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880673841 GH On-Demand Anodyne EPHX2 41 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880673841 GH On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880673841 GH On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880673842 GH On-Demand Anodyne EPHX2 41 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880673842 GH On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880673842 GH On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@H]2C1 ZINC000880673843 GH On-Demand Anodyne EPHX2 41 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@H]2C1 ZINC000880673843 GH On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2CSC[C@H]2C1 ZINC000880673843 GH On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1nn(C)cc1C(F)F ZINC000880673845 GH On-Demand Anodyne SOAT1 34 43 COC(=O)C1(O)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673846 FD On-Demand Anodyne EPHX2 28 40 COC(=O)C1(O)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673846 FD On-Demand Anodyne KCNK3 25 41 COC(=O)C1(O)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673846 FD On-Demand Anodyne KCNK9 28 41 C#CC1(F)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673868 EF On-Demand Mild EPHX2 31 41 C#CC1(F)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673868 EF On-Demand Mild KCNK3 24 40 C#CC1(F)CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880673868 EF On-Demand Mild KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)CC(C)(C)S(C)(=O)=O ZINC000880673869 GF On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)CC(C)(C)S(C)(=O)=O ZINC000880673869 GF On-Demand Anodyne KCNK9 27 40 CCn1ccc(NC(=O)CCCCc2ccc(OC)c(OC)c2)n1 ZINC000880673872 EG On-Demand Anodyne INHA 66 39 CCn1ccc(NC(=O)CCCCc2ccc(OC)c(OC)c2)n1 ZINC000880673872 EG On-Demand Anodyne HDAC7 17 40 CCn1ccc(NC(=O)CCCCc2ccc(OC)c(OC)c2)n1 ZINC000880673872 EG On-Demand Anodyne ENPP1 66 33 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880673880 EE On-Demand Anodyne ACHE 22 43 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880673880 EE On-Demand Anodyne SIGMAR1 18 40 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880673880 EE On-Demand Anodyne CACNA1I 57 39 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)C(=O)N(C)OC ZINC000880673885 FE On-Demand Anodyne KCNK3 26 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)C(=O)N(C)OC ZINC000880673885 FE On-Demand Anodyne KCNK9 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)C(=O)N(C)OC ZINC000880673886 FE On-Demand Anodyne KCNK3 26 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)C(=O)N(C)OC ZINC000880673886 FE On-Demand Anodyne KCNK9 30 41 O=C1NCC[C@@H]1CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880673899 EE On-Demand Anodyne KCNH2 44 43 O=C1NCC[C@H]1CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880673900 EE On-Demand Anodyne KCNH2 44 43 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCSC ZINC000880673901 EG On-Demand Anodyne KCNK3 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCSC ZINC000880673901 EG On-Demand Anodyne KCNK9 33 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne DRD4 15 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne ACHE 26 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne HTR4 44 46 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne SIGMAR1 22 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne SSTR5 40 33 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ncsc1C1CC1 ZINC000880673923 FG On-Demand Anodyne CACNA1I 65 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(CO)(CO)CC1 ZINC000880673928 GE On-Demand Anodyne EPHX2 38 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(CO)(CO)CC1 ZINC000880673928 GE On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(CO)(CO)CC1 ZINC000880673928 GE On-Demand Anodyne KCNK9 27 40 N#C[C@@H]1CCCC[C@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673942 EH On-Demand Mild PDE4D 16 41 N#C[C@@H]1CCCC[C@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673942 EH On-Demand Mild EZH2 47 40 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673943 EH On-Demand Mild PDE4D 16 41 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673943 EH On-Demand Mild EZH2 47 40 N#C[C@H]1CCCC[C@@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673944 EH On-Demand Mild PDE4D 16 41 N#C[C@H]1CCCC[C@@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673944 EH On-Demand Mild EZH2 47 40 N#C[C@H]1CCCC[C@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673945 EH On-Demand Mild PDE4D 16 41 N#C[C@H]1CCCC[C@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880673945 EH On-Demand Mild EZH2 47 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@@H]1c1cc(C)on1 ZINC000880673950 GI On-Demand Anodyne CPT1A 47 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@H]1c1cc(C)on1 ZINC000880673951 GI On-Demand Anodyne CPT1A 47 40 O=C(C[C@@H]1C[C@H]1C1CC1)Nc1cc(F)ccn1 ZINC000880673954 BF On-Demand Anodyne TYK2 50 32 C=CCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673963 DF On-Demand Mild KCNK3 32 44 C=CCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673963 DF On-Demand Mild KCNK9 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)NN1CCCC1 ZINC000880673965 DF On-Demand Anodyne KCNK3 26 44 COc1cccc(OC(F)(F)F)c1NC(=O)NN1CCCC1 ZINC000880673965 DF On-Demand Anodyne KCNK9 30 44 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880673970 EG On-Demand Mild PAPA1_CARPA 35 41 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880673970 EG On-Demand Mild FPR1 41 37 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880673972 EG On-Demand Mild PAPA1_CARPA 35 41 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880673972 EG On-Demand Mild FPR1 41 37 O=C(Nc1cc(F)ccn1)c1cnc(CC2CC2)s1 ZINC000880673974 CF On-Demand Anodyne TYK2 54 34 CCN(CC)C(=O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673975 FF On-Demand Anodyne KCNK3 37 41 CCN(CC)C(=O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673975 FF On-Demand Anodyne KCNK9 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CCCCO2)CC1 ZINC000880673982 GI On-Demand Anodyne EPHX2 32 51 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CCCCO2)CC1 ZINC000880673982 GI On-Demand Anodyne TRPM8 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H]1C[C@H](O)C1 ZINC000880673985 EE On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H]1C[C@H](O)C1 ZINC000880673985 EE On-Demand Anodyne KCNK9 32 41 C#CCN(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673992 DF On-Demand Mild KCNK3 36 42 C#CCN(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880673992 DF On-Demand Mild KCNK9 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1nnc(C)s1 ZINC000880674005 GG On-Demand Anodyne KCNK3 30 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1nnc(C)s1 ZINC000880674005 GG On-Demand Anodyne KCNK9 32 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)[C@@H](C)O ZINC000880674010 DE On-Demand Anodyne KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)[C@@H](C)O ZINC000880674010 DE On-Demand Anodyne KCNK9 36 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)[C@@H](C)O ZINC000880674012 DE On-Demand Anodyne KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)[C@@H](C)O ZINC000880674012 DE On-Demand Anodyne KCNK9 36 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)[C@H](C)O ZINC000880674014 DE On-Demand Anodyne KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)[C@H](C)O ZINC000880674014 DE On-Demand Anodyne KCNK9 36 44 COC(=O)C[C@@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674015 FF On-Demand Anodyne KCNK3 32 42 COC(=O)C[C@@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674015 FF On-Demand Anodyne KCNK9 35 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)[C@H](C)O ZINC000880674016 DE On-Demand Anodyne KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)[C@H](C)O ZINC000880674016 DE On-Demand Anodyne KCNK9 36 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOC[C@@H]1CCOC1 ZINC000880674024 FF On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NOC[C@@H]1CCOC1 ZINC000880674024 FF On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)NOC[C@H]1CCOC1 ZINC000880674025 FF On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NOC[C@H]1CCOC1 ZINC000880674025 FF On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cnnn1C ZINC000880674036 EE On-Demand Anodyne SOAT1 26 40 Cc1cnc(Cl)c(C(=O)N2CCC[C@@H]2c2nccc(C(F)(F)F)n2)c1 ZINC000880674041 FH On-Demand Anodyne HCRTR1 40 37 Cc1cnc(Cl)c(C(=O)N2CCC[C@H]2c2nccc(C(F)(F)F)n2)c1 ZINC000880674042 FH On-Demand Anodyne HCRTR1 40 37 O=C(c1ccc(CN2CCOCC2)o1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674043 GG On-Demand Anodyne KCNH2 44 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne PGC 42 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne PAPA1_CARPA 38 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne CCKAR 23 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne CTSK 15 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne REN 41 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674055 FF On-Demand Anodyne FPR1 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne PGC 42 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne PAPA1_CARPA 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne CCKAR 23 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne CTSK 15 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne REN 41 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1Cc2ccccc2[C@@H]1C ZINC000880674056 FF On-Demand Anodyne FPR1 46 36 C[C@H](Oc1ccnc(NC(=O)COC2CC2)c1)c1ccccc1 ZINC000880674060 DG On-Demand Anodyne TIMP3 43 36 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC(O)(C(C)C)C1 ZINC000880674070 EF On-Demand Anodyne KCNK3 26 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC(O)(C(C)C)C1 ZINC000880674070 EF On-Demand Anodyne KCNK9 30 41 Cn1nc2c(c1C(=O)NCC1CCN(Cc3ccncc3)CC1)CSCC2 ZINC000880674103 GE On-Demand Anodyne ACHE 23 44 Cn1nc2c(c1C(=O)NCC1CCN(Cc3ccncc3)CC1)CSCC2 ZINC000880674103 GE On-Demand Anodyne HTR4 48 42 Cn1nc2c(c1C(=O)NCC1CCN(Cc3ccncc3)CC1)CSCC2 ZINC000880674103 GE On-Demand Anodyne CACNA1I 70 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2C(=O)N(C)C(=O)[C@H]2C1 ZINC000880674105 GD On-Demand Anodyne KCNK3 26 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2C(=O)N(C)C(=O)[C@H]2C1 ZINC000880674105 GD On-Demand Anodyne KCNK9 30 42 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne DRD2 17 49 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne DRD4 33 49 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne ACHE 35 48 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne HTR4 60 45 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne SIGMAR1 26 42 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne SSTR5 62 46 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne CCR3 30 44 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne CXCR3 30 43 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne MCHR1 40 44 Cc1cnc(Cl)c(C(=O)NCC2CCN(Cc3ccncc3)CC2)c1 ZINC000880674108 FG On-Demand Anodyne CACNA1I 92 58 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880674114 FD On-Demand Anodyne EPHX2 42 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880674114 FD On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880674114 FD On-Demand Anodyne KCNK9 28 41 CCn1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)n1 ZINC000880674116 CF On-Demand Anodyne MTNR1B 32 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(COC2)C1 ZINC000880674117 DE On-Demand Anodyne EPHX2 29 40 CCn1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)n1 ZINC000880674118 CF On-Demand Anodyne MTNR1B 32 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H]2C[C@H]2C1 ZINC000880674124 CG On-Demand Anodyne RBP4 58 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H]2C[C@@H]2C1 ZINC000880674126 CG On-Demand Anodyne RBP4 58 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880674128 CG On-Demand Anodyne RBP4 58 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)(F)CC1 ZINC000880674129 FH On-Demand Anodyne EPHX2 38 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)(F)CC1 ZINC000880674129 FH On-Demand Anodyne TRPM8 30 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)(F)CC1 ZINC000880674129 FH On-Demand Anodyne KCNK3 26 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(F)(F)CC1 ZINC000880674129 FH On-Demand Anodyne KCNK9 30 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H]2C[C@H]2C1 ZINC000880674130 CG On-Demand Anodyne RBP4 58 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@@H](C(C)=O)C1 ZINC000880674131 FG On-Demand Anodyne EPHX2 31 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@H](C(C)=O)C1 ZINC000880674133 FG On-Demand Anodyne EPHX2 31 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C)(N2CCC2)CC1 ZINC000880674150 GH On-Demand Anodyne CCR5 15 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C)(N2CCC2)CC1 ZINC000880674150 GH On-Demand Anodyne EPHX2 31 43 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674162 GH On-Demand Anodyne ACHE 27 44 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674162 GH On-Demand Anodyne SIGMAR1 27 45 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674162 GH On-Demand Anodyne CCR3 74 47 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674162 GH On-Demand Anodyne CACNA1I 64 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)c1ccnn1C ZINC000880674165 FG On-Demand Anodyne KCNK3 26 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)c1ccnn1C ZINC000880674165 FG On-Demand Anodyne KCNK9 30 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)c1ccnn1C ZINC000880674168 FG On-Demand Anodyne KCNK3 26 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)c1ccnn1C ZINC000880674168 FG On-Demand Anodyne KCNK9 30 40 O=C(Nc1cc(F)ccn1)c1c(Cl)n[nH]c1C1CC1 ZINC000880674170 CF On-Demand Anodyne TYK2 75 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCOCC1 ZINC000880674178 GE On-Demand Reactive KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCOCC1 ZINC000880674178 GE On-Demand Reactive KCNK9 27 40 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674198 FE On-Demand Anodyne ACHE 19 41 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674198 FE On-Demand Anodyne CACNA1I 54 39 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674200 FE On-Demand Anodyne ACHE 19 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674200 FE On-Demand Anodyne CACNA1I 54 39 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674202 FE On-Demand Anodyne ACHE 19 41 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674202 FE On-Demand Anodyne CACNA1I 54 39 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674204 FE On-Demand Anodyne ACHE 19 41 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674204 FE On-Demand Anodyne CACNA1I 54 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880674218 EE On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(F)ccn1 ZINC000880674221 EE On-Demand Anodyne PAPA1_CARPA 38 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCO[C@H](C(F)F)C1 ZINC000880674246 FG On-Demand Anodyne EPHX2 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCO[C@@H](C(F)F)C1 ZINC000880674249 FG On-Demand Anodyne EPHX2 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880674265 EG On-Demand Anodyne EPHX2 53 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880674265 EG On-Demand Anodyne KCNK3 25 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880674265 EG On-Demand Anodyne KCNK9 29 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2nccnn2)CC1 ZINC000880674289 FD On-Demand Anodyne FAAH 25 45 COC[C@@H](O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674296 ED On-Demand Anodyne ADRB1 42 32 COC[C@@H](O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674296 ED On-Demand Anodyne SOAT1 33 42 COC[C@@H](O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674296 ED On-Demand Anodyne KCNK3 31 41 COC[C@@H](O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674296 ED On-Demand Anodyne KCNK9 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1OCCCO1 ZINC000880674321 FE On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1OCCCO1 ZINC000880674321 FE On-Demand Anodyne KCNK9 28 40 O=C(CN1CCCCS1(=O)=O)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880674322 GD On-Demand Anodyne CPT1A 63 39 O=C(CN1CCCCS1(=O)=O)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880674323 GD On-Demand Anodyne CPT1A 63 39 C=CC(C)(C)CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674339 DI On-Demand Mild CHRM1 18 41 C=CC(C)(C)CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674339 DI On-Demand Mild KCNH2 47 45 C=CC(C)(C)CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674339 DI On-Demand Mild CHRM3 19 42 C=CC(C)(C)CC(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674339 DI On-Demand Mild GLRA1 43 33 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)OCCCO2 ZINC000880674340 GG On-Demand Anodyne EPHX2 36 47 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CC2)C1 ZINC000880674343 DG On-Demand Anodyne EPHX2 34 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CC2)C1 ZINC000880674343 DG On-Demand Anodyne KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CC2)C1 ZINC000880674343 DG On-Demand Anodyne KCNK9 29 43 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1C(=O)OCC1(C)C ZINC000880674352 FF On-Demand Anodyne KCNK3 25 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1C(=O)OCC1(C)C ZINC000880674352 FF On-Demand Anodyne KCNK9 29 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1C(=O)OCC1(C)C ZINC000880674353 FF On-Demand Anodyne KCNK3 25 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1C(=O)OCC1(C)C ZINC000880674353 FF On-Demand Anodyne KCNK9 29 40 CC[C@@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C(OC)OC ZINC000880674360 FG On-Demand Anodyne KCNK3 37 41 CC[C@@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C(OC)OC ZINC000880674360 FG On-Demand Anodyne KCNK9 38 41 COC(=O)[C@H](F)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674371 FE On-Demand Anodyne SOAT1 36 42 COC(=O)[C@H](F)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674371 FE On-Demand Anodyne KCNK3 32 42 COC(=O)[C@H](F)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674371 FE On-Demand Anodyne KCNK9 34 42 CCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674386 DG On-Demand Anodyne KCNK3 38 44 CCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674386 DG On-Demand Anodyne KCNK9 39 44 O=C(CC[C@H]1CCc2ccccc21)NCCS(=O)(=O)CC(F)(F)F ZINC000880674414 FF On-Demand Anodyne NQO2 21 42 O=C(CC[C@@H]1CCc2ccccc21)NCCS(=O)(=O)CC(F)(F)F ZINC000880674415 FF On-Demand Anodyne NQO2 21 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCN(C)OC ZINC000880674417 EE On-Demand Anodyne KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCN(C)OC ZINC000880674417 EE On-Demand Anodyne KCNK9 37 42 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(F)ccn1)C2 ZINC000880674434 DF On-Demand Anodyne RAF1 16 48 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(F)ccn1)C2 ZINC000880674434 DF On-Demand Anodyne NPY5R 16 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(F)ccn1)C2 ZINC000880674434 DF On-Demand Anodyne TYK2 52 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880674445 GI On-Demand Anodyne RBP4 62 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880674451 GI On-Demand Anodyne RBP4 62 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2c(F)cccc2c1 ZINC000880674467 GG On-Demand Anodyne PAPA1_CARPA 34 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2c(F)cccc2c1 ZINC000880674471 GG On-Demand Anodyne PAPA1_CARPA 34 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880674476 FG On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880674476 FG On-Demand Anodyne KCNK9 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880674478 FG On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880674478 FG On-Demand Anodyne KCNK9 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880674481 FG On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880674481 FG On-Demand Anodyne KCNK9 28 41 O=C(c1ncccc1-c1ccccn1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674508 GI On-Demand Anodyne KCNH2 41 40 CS(=O)(=O)C1CCC(C(=O)Nc2cc(F)ccn2)CC1 ZINC000880674515 DD On-Demand Anodyne GSK3B 15 45 CS(=O)(=O)C1CCC(C(=O)Nc2cc(F)ccn2)CC1 ZINC000880674515 DD On-Demand Anodyne MAPK10 15 49 CS(=O)(=O)C1CCC(C(=O)Nc2cc(F)ccn2)CC1 ZINC000880674515 DD On-Demand Anodyne TYK2 72 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCc2nc(C3CC3)ncc2C1 ZINC000880674521 FH On-Demand Anodyne MAPK1 42 33 CC(C)(C)OC(=O)N1CC2(CC(C(=O)Nc3cc(F)ccn3)=NO2)C1 ZINC000880674524 FD On-Demand Anodyne GPR119 16 51 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCC1 ZINC000880674535 DG On-Demand Anodyne KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCC1 ZINC000880674535 DG On-Demand Anodyne KCNK9 29 43 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674570 GF On-Demand Anodyne KCNH2 43 41 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674570 GF On-Demand Anodyne GLRA1 42 33 O=C(COC1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674594 DF On-Demand Anodyne CHRM1 18 43 O=C(COC1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674594 DF On-Demand Anodyne KCNH2 50 48 O=C(COC1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674594 DF On-Demand Anodyne CHRM4 20 40 O=C(COC1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674594 DF On-Demand Anodyne CHRM5 26 40 O=C(COC1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674594 DF On-Demand Anodyne GLRA1 44 33 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880674606 FG On-Demand Anodyne SFRP1 42 34 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880674609 FG On-Demand Anodyne SFRP1 42 34 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)CNC(=O)O2 ZINC000880674615 GF On-Demand Anodyne EPHX2 31 46 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)CNC(=O)O2 ZINC000880674615 GF On-Demand Anodyne TRPM8 32 44 COC[C@@H]1CCCN1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880674622 DE On-Demand Anodyne CASP7 40 35 O=C(c1cccn2nccc12)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674625 EH On-Demand Anodyne KCNH2 42 40 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne DRD4 21 45 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne ACHE 39 48 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne HTR4 69 48 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne SIGMAR1 29 45 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne SSTR5 54 34 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne CCR3 33 45 Cn1nnc(C(=O)NCC2CCN(Cc3ccncc3)CC2)n1 ZINC000880674629 DC On-Demand Anodyne CACNA1I 83 48 O=C([C@@H]1CCc2nncn2CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674636 FF On-Demand Anodyne KCNH2 41 40 O=C([C@H]1CCc2nncn2CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674637 FF On-Demand Anodyne KCNH2 41 40 COCCn1ncc(C(=O)Nc2cc(O[C@@H](C)c3ccccc3)ccn2)c1C ZINC000880674638 GH On-Demand Anodyne GCK 38 46 COCCn1ncc(C(=O)Nc2cc(O[C@H](C)c3ccccc3)ccn2)c1C ZINC000880674640 GH On-Demand Anodyne GCK 38 46 Cc1cc(OCC(=O)Nc2nc(-c3ccccc3)c(C(=O)c3ccccc3)s2)no1 ZINC000880674643 HI On-Demand Anodyne RORC 23 52 O=C(COC1CC1)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880674648 DE On-Demand Anodyne PRCP 30 41 O=C(COC1CC1)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880674648 DE On-Demand Anodyne CPT1A 109 47 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC([C@@H](F)C(N)=O)CC1 ZINC000880674675 GF On-Demand Anodyne KCNK3 25 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC([C@@H](F)C(N)=O)CC1 ZINC000880674675 GF On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC([C@H](F)C(N)=O)CC1 ZINC000880674676 GF On-Demand Anodyne KCNK3 25 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC([C@H](F)C(N)=O)CC1 ZINC000880674676 GF On-Demand Anodyne KCNK9 28 40 O=C(COC1CC1)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880674677 DE On-Demand Anodyne PRCP 30 41 O=C(COC1CC1)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880674677 DE On-Demand Anodyne CPT1A 109 47 Cn1nnc(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)n1 ZINC000880674678 DD On-Demand Anodyne KCNH2 45 45 Cn1nnc(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)n1 ZINC000880674678 DD On-Demand Anodyne GLRA1 54 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CNC(=O)O2)C1 ZINC000880674679 FD On-Demand Anodyne EPHX2 26 44 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@@](C)=O ZINC000880674688 EE On-Demand Anodyne KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@@](C)=O ZINC000880674688 EE On-Demand Anodyne KCNK9 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@](C)=O ZINC000880674689 EE On-Demand Anodyne KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@](C)=O ZINC000880674689 EE On-Demand Anodyne KCNK9 37 42 COC(=O)N1CCC(NC(=O)Nc2c(OC)cccc2OC(F)(F)F)CC1 ZINC000880674690 GF On-Demand Anodyne EPHX2 61 49 C=C[C@@H](C)ONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674713 DG On-Demand Mild KCNK3 27 42 C=C[C@@H](C)ONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674713 DG On-Demand Mild KCNK9 31 42 C=C[C@H](C)ONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674714 DG On-Demand Mild KCNK3 27 42 C=C[C@H](C)ONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674714 DG On-Demand Mild KCNK9 31 42 COC(=O)CCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674727 FF On-Demand Anodyne KCNK3 30 41 COC(=O)CCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674727 FF On-Demand Anodyne KCNK9 32 41 C[C@H](Oc1ccnc(NC(=O)[C@@H]2CCc3nncn3CC2)c1)c1ccccc1 ZINC000880674729 GG On-Demand Anodyne TYK2 55 38 C[C@H](Oc1ccnc(NC(=O)[C@H]2CCc3nncn3CC2)c1)c1ccccc1 ZINC000880674731 GG On-Demand Anodyne TYK2 55 38 O=C(C[C@@H]1C[C@H]1C1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674734 EI On-Demand Anodyne KCNH2 47 45 O=C(C[C@@H]1C[C@H]1C1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674734 EI On-Demand Anodyne GLRA1 44 33 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC#N ZINC000880674752 DF On-Demand Mild KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC#N ZINC000880674752 DF On-Demand Mild KCNK9 37 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCS(=O)(=O)CC(F)(F)F)C2 ZINC000880674754 GD On-Demand Anodyne NQO2 38 45 COc1ccc2c(c1)CC[C@H](C(=O)NCCS(=O)(=O)CC(F)(F)F)C2 ZINC000880674754 GD On-Demand Anodyne MTNR1A 59 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCS(=O)(=O)CC(F)(F)F)C2 ZINC000880674754 GD On-Demand Anodyne MTNR1B 50 40 O=C(c1cnc2cc[nH]c2c1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674755 EH On-Demand Anodyne KCNH2 44 42 O=C(c1cnc2cc[nH]c2c1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880674755 EH On-Demand Anodyne GLRA1 40 43 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)C(OC)OC ZINC000880674756 FF On-Demand Anodyne KCNK3 28 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)C(OC)OC ZINC000880674756 FF On-Demand Anodyne KCNK9 32 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)C(OC)OC ZINC000880674757 FF On-Demand Anodyne KCNK3 28 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)C(OC)OC ZINC000880674757 FF On-Demand Anodyne KCNK9 32 44 C#C[C@@H](C)N(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674777 DG On-Demand Mild KCNK3 27 42 C#C[C@@H](C)N(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674777 DG On-Demand Mild KCNK9 31 42 C#C[C@H](C)N(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674778 DG On-Demand Mild KCNK3 27 42 C#C[C@H](C)N(C)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880674778 DG On-Demand Mild KCNK9 31 42 O=C(Nc1cc(F)ccn1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880674785 CD On-Demand Anodyne MAPK10 15 46 O=C(Nc1cc(F)ccn1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880674785 CD On-Demand Anodyne TYK2 70 42 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@@H]1C[C@@H](OC)C1 ZINC000880674788 EG On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@@H]1C[C@@H](OC)C1 ZINC000880674788 EG On-Demand Anodyne KCNK9 32 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne DRD4 25 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne ACHE 36 52 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne HTR4 59 42 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne TBXA2R 17 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne SSTR5 46 34 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne CCR3 20 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne MCHR1 16 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1coc(-c2ccccn2)n1 ZINC000880674791 GF On-Demand Anodyne CACNA1I 58 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc(CC2CC2)s1 ZINC000880674792 FG On-Demand Anodyne ACHE 23 46 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc(CC2CC2)s1 ZINC000880674792 FG On-Demand Anodyne HTR4 55 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc(CC2CC2)s1 ZINC000880674792 FG On-Demand Anodyne SIGMAR1 23 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc(CC2CC2)s1 ZINC000880674792 FG On-Demand Anodyne SSTR5 41 35 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cnc(CC2CC2)s1 ZINC000880674792 FG On-Demand Anodyne CACNA1I 70 46 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne DRD4 31 43 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne ACHE 49 50 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne HTR4 38 43 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne SIGMAR1 55 44 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne CCR3 44 39 O=C(NCC1CCN(Cc2ccncc2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880674802 GG On-Demand Anodyne CACNA1I 60 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880674805 FG On-Demand Anodyne SSTR1 55 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880674805 FG On-Demand Anodyne EPHX2 40 37 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880674805 FG On-Demand Anodyne KCNK3 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880674805 FG On-Demand Anodyne KCNK9 40 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880674806 FG On-Demand Anodyne SSTR1 55 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880674806 FG On-Demand Anodyne EPHX2 40 37 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880674806 FG On-Demand Anodyne KCNK3 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880674806 FG On-Demand Anodyne KCNK9 40 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880674807 FG On-Demand Anodyne SSTR1 55 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880674807 FG On-Demand Anodyne EPHX2 40 37 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880674807 FG On-Demand Anodyne KCNK3 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880674807 FG On-Demand Anodyne KCNK9 40 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880674808 FG On-Demand Anodyne SSTR1 55 38 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880674808 FG On-Demand Anodyne EPHX2 40 37 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880674808 FG On-Demand Anodyne KCNK3 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880674808 FG On-Demand Anodyne KCNK9 40 44 O=C(C[C@@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674828 EC On-Demand Anodyne ACHE 34 45 O=C(C[C@@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674828 EC On-Demand Anodyne SIGMAR1 28 44 O=C(C[C@@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674828 EC On-Demand Anodyne CACNA1I 61 41 O=C(C[C@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674830 EC On-Demand Anodyne ACHE 34 45 O=C(C[C@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674830 EC On-Demand Anodyne SIGMAR1 28 44 O=C(C[C@H]1CCNC1=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674830 EC On-Demand Anodyne CACNA1I 61 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1csc(-c2ncc[nH]2)n1 ZINC000880674834 GF On-Demand Anodyne ACHE 17 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1csc(-c2ncc[nH]2)n1 ZINC000880674834 GF On-Demand Anodyne HTR4 40 38 O=C(NCC1CCN(Cc2ccncc2)CC1)c1csc(-c2ncc[nH]2)n1 ZINC000880674834 GF On-Demand Anodyne CACNA1I 64 42 COCCn1ncc(C(=O)Nc2cc(F)ccn2)c1C ZINC000880674847 CD On-Demand Anodyne MAPK14 15 41 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne DRD4 19 41 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne ACHE 41 49 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne HTR4 51 42 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne SIGMAR1 34 46 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne SSTR5 70 37 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne CCR3 32 42 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne MCHR1 33 41 O=C(COC1CC1)NCC1CCN(Cc2ccncc2)CC1 ZINC000880674850 DD On-Demand Anodyne CACNA1I 69 44 CC(C)(C)OC(=O)NC1CC(C(=O)Nc2cc(F)ccn2)C1 ZINC000880674854 DE On-Demand Anodyne TYK2 64 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880674929 GH On-Demand Anodyne RBP4 52 34 O=C(NCc1cccnc1N1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674946 FH On-Demand Anodyne KCNQ2 55 37 O=C(NCc1cccnc1N1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674946 FH On-Demand Anodyne TRPV1 40 43 O=C(NCc1cccnc1N1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674946 FH On-Demand Anodyne SCN2A 20 48 O=C(NCc1cccnc1N1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674946 FH On-Demand Anodyne SCN10A 23 48 O=C(NCc1cccnc1N1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674946 FH On-Demand Anodyne NAMPT 24 40 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880674952 GG On-Demand Anodyne CACNA1I 49 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880674985 EF On-Demand Anodyne RBP4 55 36 COc1cccc(OC(F)(F)F)c1NC(=O)NOC(C)(C)CO ZINC000880674993 EE On-Demand Anodyne KCNK3 32 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOC(C)(C)CO ZINC000880674993 EE On-Demand Anodyne KCNK9 34 44 Cc1coc(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)c1 ZINC000880675019 DH On-Demand Anodyne KCNH2 47 44 Cc1coc(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)c1 ZINC000880675019 DH On-Demand Anodyne GLRA1 45 37 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880675022 GJ On-Demand Anodyne CPT1A 86 41 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880675023 GJ On-Demand Anodyne CPT1A 86 41 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880675024 GJ On-Demand Anodyne CPT1A 86 41 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880675025 GJ On-Demand Anodyne CPT1A 86 41 C#C[C@@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C1CCOCC1 ZINC000880675026 FG On-Demand Mild KCNK3 25 40 C#C[C@@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C1CCOCC1 ZINC000880675026 FG On-Demand Mild KCNK9 28 40 C#C[C@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C1CCOCC1 ZINC000880675027 FG On-Demand Mild KCNK3 25 40 C#C[C@H](NC(=O)Nc1c(OC)cccc1OC(F)(F)F)C1CCOCC1 ZINC000880675027 FG On-Demand Mild KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCOC1=O ZINC000880675029 EE On-Demand Anodyne LUXR 79 45 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCOC1=O ZINC000880675029 EE On-Demand Anodyne TRAR 97 52 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCOC1=O ZINC000880675029 EE On-Demand Anodyne LASR 62 41 C#CCNC(=O)C1CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)CC1 ZINC000880675031 GF On-Demand Mild EPHX2 30 40 C#CCNC(=O)C1CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)CC1 ZINC000880675031 GF On-Demand Mild CACNA1G 36 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CCOC2)C1 ZINC000880675033 EF On-Demand Anodyne EPHX2 34 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)OCCO2 ZINC000880675036 GF On-Demand Anodyne EPHX2 36 48 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)OCCO2 ZINC000880675036 GF On-Demand Anodyne TRPM8 29 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCCN(C=O)CC1 ZINC000880675048 FE On-Demand Anodyne KCNK3 26 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCCN(C=O)CC1 ZINC000880675048 FE On-Demand Anodyne KCNK9 29 42 Cc1nc(C(C)C)ncc1C(=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880675060 FI On-Demand Anodyne GLRA1 44 36 COCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675061 DE On-Demand Anodyne KCNK3 47 48 COCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675061 DE On-Demand Anodyne KCNK9 47 48 CC(C)(C)OC(=O)N1CC[C@]2(CC(C(=O)Nc3cc(F)ccn3)=NO2)C1 ZINC000880675064 FE On-Demand Anodyne GPR119 18 56 CC(C)(C)OC(=O)N1CC[C@@]2(CC(C(=O)Nc3cc(F)ccn3)=NO2)C1 ZINC000880675065 FE On-Demand Anodyne GPR119 18 56 COc1cccc(OC(F)(F)F)c1NC(=O)NC(CF)CF ZINC000880675084 EG On-Demand Anodyne KCNK3 45 45 COc1cccc(OC(F)(F)F)c1NC(=O)NC(CF)CF ZINC000880675084 EG On-Demand Anodyne KCNK9 45 45 C[C@H]1c2ccccc2C[C@H]1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880675096 EG On-Demand Anodyne HTR7 18 40 C[C@H]1c2ccccc2C[C@H]1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880675096 EG On-Demand Anodyne KCNQ2 40 35 O=C(Nc1cc(F)ccn1)[C@@H]1CCc2nncn2CC1 ZINC000880675099 CD On-Demand Anodyne MAPK10 15 44 O=C(Nc1cc(F)ccn1)[C@@H]1CCc2nncn2CC1 ZINC000880675099 CD On-Demand Anodyne TYK2 65 39 O=C(Nc1cc(F)ccn1)[C@H]1CCc2nncn2CC1 ZINC000880675101 CD On-Demand Anodyne MAPK10 15 44 O=C(Nc1cc(F)ccn1)[C@H]1CCc2nncn2CC1 ZINC000880675101 CD On-Demand Anodyne TYK2 65 39 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCOC(C)C ZINC000880675104 FG On-Demand Anodyne KCNK3 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCOC(C)C ZINC000880675104 FG On-Demand Anodyne KCNK9 41 44 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675119 CE On-Demand Mild JAK3 18 41 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675119 CE On-Demand Mild JAK1 17 41 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675119 CE On-Demand Mild TYK2 21 41 N#C[C@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675120 CE On-Demand Mild JAK3 18 41 N#C[C@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675120 CE On-Demand Mild JAK1 17 41 N#C[C@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675120 CE On-Demand Mild TYK2 21 41 N#C[C@@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675121 CE On-Demand Mild JAK3 18 41 N#C[C@@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675121 CE On-Demand Mild JAK1 17 41 N#C[C@@H]1CCCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880675121 CE On-Demand Mild TYK2 21 41 N#C[C@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675122 CE On-Demand Mild JAK3 18 41 N#C[C@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675122 CE On-Demand Mild JAK1 17 41 N#C[C@H]1CCCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880675122 CE On-Demand Mild TYK2 21 41 CCn1ccc(NC(=O)c2ncsc2C2CC2)n1 ZINC000880675134 CE On-Demand Anodyne MAP1 96 38 CCn1ccc(NC(=O)Cc2ccccc2N2CCCC2=O)n1 ZINC000880675156 DE On-Demand Anodyne KCNQ2 61 38 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne DRD2 25 63 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne DRD4 50 63 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne ACHE 51 51 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne HRH1 22 41 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne DRD3 22 46 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne HTR4 77 48 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne GRIN2B 40 38 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne SIGMAR1 47 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne SSTR5 62 36 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne CCR3 98 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne CCR2 15 44 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne MCHR1 58 45 O=C(NCC1CCN(Cc2ccncc2)CC1)c1cc2ccccc2cc1F ZINC000880675158 GI On-Demand Anodyne CACNA1I 72 46 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1C[C@@H](S(C)(=O)=O)C1 ZINC000880675167 GE On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1C[C@@H](S(C)(=O)=O)C1 ZINC000880675167 GE On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880675168 GF On-Demand Anodyne DRD4 22 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880675168 GF On-Demand Anodyne CCR3 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880675168 GF On-Demand Anodyne EPHX2 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880675168 GF On-Demand Anodyne CXCR3 16 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@H]2C[C@H]2C1 ZINC000880675195 DH On-Demand Anodyne EPHX2 24 50 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@@H]2C[C@@H]2C1 ZINC000880675196 DH On-Demand Anodyne EPHX2 24 50 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@@H]2C[C@H]2C1 ZINC000880675197 DH On-Demand Anodyne EPHX2 24 50 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@H]2C[C@@H]2C1 ZINC000880675198 DH On-Demand Anodyne EPHX2 24 50 CS(=O)(=O)C1CCC(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)CC1 ZINC000880675227 GG On-Demand Anodyne KCNH2 42 40 CS(=O)(=O)C1CCC(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)CC1 ZINC000880675227 GG On-Demand Anodyne GLRA1 44 34 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC2(CC1)CC2 ZINC000880675230 DI On-Demand Anodyne EPHX2 19 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675233 GG On-Demand Anodyne SIGMAR1 18 43 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675233 GG On-Demand Anodyne CCR3 64 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675233 GG On-Demand Anodyne MCHR1 31 43 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675236 GG On-Demand Anodyne SIGMAR1 18 43 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675236 GG On-Demand Anodyne CCR3 64 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880675236 GG On-Demand Anodyne MCHR1 31 43 COc1cccc(OC(F)(F)F)c1NC(=O)NOC(C)C ZINC000880675275 DG On-Demand Anodyne KCNK3 49 49 COc1cccc(OC(F)(F)F)c1NC(=O)NOC(C)C ZINC000880675275 DG On-Demand Anodyne KCNK9 49 49 O=C(c1ncsc1C1CC1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880675291 FI On-Demand Anodyne KCNH2 40 38 Cc1cnc(Cl)c(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)c1 ZINC000880675321 FI On-Demand Anodyne KCNH2 43 41 Cc1cnc(Cl)c(C(=O)N2[C@H]3CC[C@H]2CC(Oc2ccccc2)C3)c1 ZINC000880675321 FI On-Demand Anodyne GLRA1 43 35 COC(=O)N(C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675328 EE On-Demand Reactive KCNK3 32 44 COC(=O)N(C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675328 EE On-Demand Reactive KCNK9 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)NCC(=O)N(C)OC ZINC000880675329 FD On-Demand Anodyne KCNK3 36 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC(=O)N(C)OC ZINC000880675329 FD On-Demand Anodyne KCNK9 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)NN(C)C1CC1 ZINC000880675330 DF On-Demand Reactive KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)NN(C)C1CC1 ZINC000880675330 DF On-Demand Reactive KCNK9 29 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@@]2(C1)CC2(F)F ZINC000880675331 GI On-Demand Anodyne EPHX2 35 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC[C@]2(C1)CC2(F)F ZINC000880675332 GI On-Demand Anodyne EPHX2 35 42 C=CC(C)(C)CC(=O)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880675352 EH On-Demand Mild CPT1A 46 38 C=CC(C)(C)CC(=O)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880675353 EH On-Demand Mild CPT1A 46 38 CCn1ccc(NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)n1 ZINC000880675380 ED On-Demand Anodyne SIGMAR1 15 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H]1c1ccc(F)cc1 ZINC000880675383 FG On-Demand Anodyne CELA1 18 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H]1c1ccc(F)cc1 ZINC000880675383 FG On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H]1c1ccc(F)cc1 ZINC000880675384 FG On-Demand Anodyne CELA1 18 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H]1c1ccc(F)cc1 ZINC000880675384 FG On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H]1c1ccc(F)cc1 ZINC000880675385 FG On-Demand Anodyne CELA1 18 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H]1c1ccc(F)cc1 ZINC000880675385 FG On-Demand Anodyne PAPA1_CARPA 32 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H]1c1ccc(F)cc1 ZINC000880675386 FG On-Demand Anodyne CELA1 18 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H]1c1ccc(F)cc1 ZINC000880675386 FG On-Demand Anodyne PAPA1_CARPA 32 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)=O)CC1 ZINC000880675387 FG On-Demand Anodyne EPHX2 42 39 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)=O)CC1 ZINC000880675387 FG On-Demand Anodyne RBP4 31 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)=O)CC1 ZINC000880675387 FG On-Demand Anodyne KCNK3 24 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)=O)CC1 ZINC000880675387 FG On-Demand Anodyne KCNK9 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2CN(C(C)=O)C[C@@H]2C1 ZINC000880675394 GF On-Demand Anodyne EPHX2 23 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2CN(C(C)=O)C[C@@H]2C1 ZINC000880675394 GF On-Demand Anodyne RBP4 53 32 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2CN(C(C)=O)C[C@@H]2C1 ZINC000880675394 GF On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H]2CN(C(C)=O)C[C@@H]2C1 ZINC000880675394 GF On-Demand Anodyne KCNK9 28 41 O=C(COC1CC1)Nc1cc(F)ccn1 ZINC000880675402 BD On-Demand Anodyne MAPK10 15 44 O=C(COC1CC1)Nc1cc(F)ccn1 ZINC000880675402 BD On-Demand Anodyne TYK2 54 35 CCn1ccc(NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)n1 ZINC000880675407 ED On-Demand Anodyne PAPA1_CARPA 37 41 CCn1ccc(NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)n1 ZINC000880675407 ED On-Demand Anodyne FPR1 41 34 CCn1ccc(NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)n1 ZINC000880675408 ED On-Demand Anodyne PAPA1_CARPA 37 41 CCn1ccc(NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)n1 ZINC000880675408 ED On-Demand Anodyne FPR1 41 34 N#C[C@@H]1CCCC[C@@H]1NC(=O)c1cncc2[nH]ccc12 ZINC000880675417 CE On-Demand Mild JAK1 17 42 N#C[C@@H]1CCCC[C@H]1NC(=O)c1cncc2[nH]ccc12 ZINC000880675418 CE On-Demand Mild JAK1 17 42 N#C[C@H]1CCCC[C@@H]1NC(=O)c1cncc2[nH]ccc12 ZINC000880675419 CE On-Demand Mild JAK1 17 42 N#C[C@H]1CCCC[C@H]1NC(=O)c1cncc2[nH]ccc12 ZINC000880675420 CE On-Demand Mild JAK1 17 42 O=C(Nc1cc(F)ccn1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880675430 CD On-Demand Anodyne TYK2 56 34 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CCNC2=O)CC1 ZINC000880675458 GF On-Demand Anodyne EPHX2 27 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne ACHE 28 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne HTR4 61 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne SIGMAR1 27 43 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne CCR3 21 40 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne CACNA1I 73 47 O=C(NCC1CCN(Cc2ccncc2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880675459 GE On-Demand Anodyne NAMPT 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H](CO)[C@@H](CO)C1 ZINC000880675460 FD On-Demand Anodyne KCNK3 31 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@@H](CO)[C@@H](CO)C1 ZINC000880675460 FD On-Demand Anodyne KCNK9 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC1CC1 ZINC000880675487 DG On-Demand Anodyne KCNK3 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC1CC1 ZINC000880675487 DG On-Demand Anodyne KCNK9 33 42 COC(=O)c1ccc2c(c1)[C@H](CNC(=O)COC1CC1)CCC2 ZINC000880675492 DE On-Demand Anodyne NQO2 22 41 COC(=O)c1ccc2c(c1)[C@H](CNC(=O)COC1CC1)CCC2 ZINC000880675492 DE On-Demand Anodyne HTR6 21 45 COC(=O)c1ccc2c(c1)[C@@H](CNC(=O)COC1CC1)CCC2 ZINC000880675493 DE On-Demand Anodyne NQO2 22 41 COC(=O)c1ccc2c(c1)[C@@H](CNC(=O)COC1CC1)CCC2 ZINC000880675493 DE On-Demand Anodyne HTR6 21 45 C=C(C)CONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675494 DG On-Demand Mild KCNK3 31 43 C=C(C)CONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675494 DG On-Demand Mild KCNK9 34 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCCC12CCC2 ZINC000880675497 EI On-Demand Anodyne KCNK3 24 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCCC12CCC2 ZINC000880675497 EI On-Demand Anodyne KCNK9 28 41 O=C1NCC[C@@H]1CC(=O)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880675503 ED On-Demand Anodyne CPT1A 46 37 O=C1NCC[C@H]1CC(=O)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880675504 ED On-Demand Anodyne CPT1A 46 37 O=C1NCC[C@H]1CC(=O)N1CCC[C@@H]1c1nccc(C(F)(F)F)n1 ZINC000880675505 ED On-Demand Anodyne CPT1A 46 37 O=C1NCC[C@@H]1CC(=O)N1CCC[C@H]1c1nccc(C(F)(F)F)n1 ZINC000880675506 ED On-Demand Anodyne CPT1A 46 37 C#CC1CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)CC1 ZINC000880675509 EG On-Demand Mild RBP4 35 41 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(C)(C)O ZINC000880675540 EE On-Demand Anodyne KCNK3 32 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(C)(C)O ZINC000880675540 EE On-Demand Anodyne KCNK9 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N(CC1CCOCC1)OC ZINC000880675546 GG On-Demand Anodyne KCNK3 30 40 COc1cccc(OC(F)(F)F)c1NC(=O)N(CC1CCOCC1)OC ZINC000880675546 GG On-Demand Anodyne KCNK9 32 40 C#C[C@H](CO)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675556 DD On-Demand Mild KCNK3 30 41 C#C[C@H](CO)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675556 DD On-Demand Mild KCNK9 33 41 C#C[C@@H](CO)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675557 DD On-Demand Mild KCNK3 30 41 C#C[C@@H](CO)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675557 DD On-Demand Mild KCNK9 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880675560 GH On-Demand Anodyne RBP4 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880675560 GH On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880675560 GH On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCCO1 ZINC000880675579 FF On-Demand Anodyne SOAT1 19 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCCO1 ZINC000880675579 FF On-Demand Anodyne KCNK3 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCCO1 ZINC000880675579 FF On-Demand Anodyne KCNK9 33 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[C@H]1CCOC1=O ZINC000880675592 GG On-Demand Anodyne TRAR 42 38 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[C@@H]1CCOC1=O ZINC000880675595 GG On-Demand Anodyne TRAR 42 38 O=C(Nc1ccc2c(n1)OCCO2)c1c[nH]nc1[C@@H]1CCCO1 ZINC000880675606 DD On-Demand Anodyne HTR1F 41 32 O=C(Nc1ccc2c(n1)OCCO2)c1c[nH]nc1[C@H]1CCCO1 ZINC000880675608 DD On-Demand Anodyne HTR1F 41 32 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(=O)(=O)C(C)C ZINC000880675631 GF On-Demand Anodyne SOAT1 36 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(=O)(=O)C(C)C ZINC000880675631 GF On-Demand Anodyne KCNK3 39 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(=O)(=O)C(C)C ZINC000880675631 GF On-Demand Anodyne KCNK9 41 43 Cc1cnc(Cl)c(C(=O)N2CC[C@H]2c2ccc(F)cc2)c1 ZINC000880675635 DH On-Demand Anodyne HCRTR1 51 37 Cc1cnc(Cl)c(C(=O)N2CC[C@H]2c2ccc(F)cc2)c1 ZINC000880675635 DH On-Demand Anodyne KCNA5 21 48 O=C1CC[C@H](c2ccc(C(=O)N3[C@H]4CC[C@H]3CC(Oc3ccccc3)C4)cc2)N1 ZINC000880675637 GH On-Demand Anodyne KCNH2 44 41 Cc1cnc(Cl)c(C(=O)N2CC[C@@H]2c2ccc(F)cc2)c1 ZINC000880675638 DH On-Demand Anodyne HCRTR1 51 37 Cc1cnc(Cl)c(C(=O)N2CC[C@@H]2c2ccc(F)cc2)c1 ZINC000880675638 DH On-Demand Anodyne KCNA5 21 48 O=C(C[C@H]1CCNC1=O)Nc1cc(F)ccn1 ZINC000880675642 BC On-Demand Anodyne TYK2 43 32 O=C(C[C@@H]1CCNC1=O)Nc1cc(F)ccn1 ZINC000880675644 BC On-Demand Anodyne TYK2 43 32 O=C(Nc1cc(F)c(F)c(F)c1F)N(CCN1CCOCC1)CC1CC1 ZINC000880675656 GF On-Demand Anodyne CASR 57 41 COC(=O)[C@@]1(O)CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880675658 GD On-Demand Anodyne EPHX2 36 45 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CC2(CSC2)C1 ZINC000880675660 FH On-Demand Anodyne KCNK3 25 42 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CC2(CSC2)C1 ZINC000880675660 FH On-Demand Anodyne KCNK9 29 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2C=C[C@H]1C2 ZINC000880675668 EG On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1C[C@H]2C=C[C@H]1C2 ZINC000880675668 EG On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)Nc1ccn(CCF)n1 ZINC000880675671 FG On-Demand Anodyne KCNK3 31 41 COc1cccc(OC(F)(F)F)c1NC(=O)Nc1ccn(CCF)n1 ZINC000880675671 FG On-Demand Anodyne KCNK9 33 41 CC(C)(C)OC(=O)N[C@H]1CC[C@@H](C(=O)Nc2cc(F)ccn2)CC1 ZINC000880675684 EG On-Demand Anodyne TYK2 63 41 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)Nc2cc(F)ccn2)CO1 ZINC000880675686 EF On-Demand Anodyne TYK2 53 33 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)Nc2cc(F)ccn2)CO1 ZINC000880675687 EF On-Demand Anodyne TYK2 53 33 CC(C)(C)OC(=O)CC[C@@H]1C[C@H](C(=O)Nc2cc(F)ccn2)CO1 ZINC000880675689 EF On-Demand Anodyne TYK2 53 33 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)Nc2cc(F)ccn2)CO1 ZINC000880675691 EF On-Demand Anodyne TYK2 53 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880675720 EI On-Demand Mild RBP4 45 32 O=C1CC[C@@H](c2ccc(C(=O)N3[C@H]4CC[C@H]3CC(Oc3ccccc3)C4)cc2)N1 ZINC000880675726 GH On-Demand Anodyne KCNH2 44 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1CC[C@H]1O ZINC000880675732 DE On-Demand Anodyne KCNK3 26 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H]1CC[C@H]1O ZINC000880675732 DE On-Demand Anodyne KCNK9 30 44 C#CCCCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675735 DG On-Demand Mild KCNK3 36 41 C#CCCCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675735 DG On-Demand Mild KCNK9 36 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CN(C)C(=O)O2)C1 ZINC000880675737 GE On-Demand Anodyne EPHX2 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CN(C)C(=O)O2)C1 ZINC000880675737 GE On-Demand Anodyne KCNK3 25 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC2(CN(C)C(=O)O2)C1 ZINC000880675737 GE On-Demand Anodyne KCNK9 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)NOC/C=C\Cl ZINC000880675741 EG On-Demand Anodyne KCNK3 44 45 COc1cccc(OC(F)(F)F)c1NC(=O)NOC/C=C\Cl ZINC000880675741 EG On-Demand Anodyne KCNK9 43 45 COc1cccc(OC(F)(F)F)c1NC(=O)NOC/C=C/Cl ZINC000880675742 EG On-Demand Anodyne KCNK3 44 45 COc1cccc(OC(F)(F)F)c1NC(=O)NOC/C=C/Cl ZINC000880675742 EG On-Demand Anodyne KCNK9 43 45 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H](O)C(F)(F)F ZINC000880675747 FF On-Demand Anodyne SOAT1 34 43 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H](O)C(F)(F)F ZINC000880675747 FF On-Demand Anodyne KCNK3 32 43 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H](O)C(F)(F)F ZINC000880675747 FF On-Demand Anodyne KCNK9 34 43 CC1(C)CC[C@@H](CC(=O)N2CCC[C@@H]2c2nccc(C(F)(F)F)n2)OC1 ZINC000880675758 FH On-Demand Anodyne CPT1A 43 39 CC1(C)CC[C@@H](CC(=O)N2CCC[C@H]2c2nccc(C(F)(F)F)n2)OC1 ZINC000880675759 FH On-Demand Anodyne CPT1A 43 39 CCON(C)C(=O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675764 FE On-Demand Anodyne KCNK3 36 41 CCON(C)C(=O)CNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675764 FE On-Demand Anodyne KCNK9 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@](O)(C(F)F)C1 ZINC000880675774 FF On-Demand Anodyne EPHX2 35 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@](O)(C(F)F)C1 ZINC000880675775 FF On-Demand Anodyne EPHX2 35 45 C#CCCN(CCOC)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675778 FG On-Demand Mild KCNK3 36 40 C#CCCN(CCOC)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675778 FG On-Demand Mild KCNK9 37 40 O=C(CN1CCCCS1(=O)=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880675782 GE On-Demand Anodyne KCNH2 45 42 O=C(CN1CCCCS1(=O)=O)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880675782 GE On-Demand Anodyne CPT1A 69 35 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cnn(C)n1 ZINC000880675790 EE On-Demand Anodyne SOAT1 24 40 COCCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675793 EF On-Demand Anodyne KCNK3 44 45 COCCCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880675793 EF On-Demand Anodyne KCNK9 44 45 COc1cccc(OC(F)(F)F)c1NC(=O)NO[C@H](CO)C(C)C ZINC000880675795 FF On-Demand Anodyne KCNK3 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NO[C@H](CO)C(C)C ZINC000880675795 FF On-Demand Anodyne KCNK9 34 41 COc1cccc(OC(F)(F)F)c1NC(=O)NO[C@@H](CO)C(C)C ZINC000880675796 FF On-Demand Anodyne KCNK3 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NO[C@@H](CO)C(C)C ZINC000880675796 FF On-Demand Anodyne KCNK9 34 41 O=C1CC[C@@H]2CN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC[C@@H]2N1 ZINC000880675847 EE On-Demand Anodyne RBP4 45 32 O=C1CC[C@H]2CN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC[C@@H]2N1 ZINC000880675849 EE On-Demand Anodyne RBP4 45 32 O=C1CC[C@H]2CN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC[C@H]2N1 ZINC000880675851 EE On-Demand Anodyne RBP4 45 32 O=C1CC[C@@H]2CN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC[C@H]2N1 ZINC000880675853 EE On-Demand Anodyne RBP4 45 32 CNc1nc(C(=O)N2CCC(O)(Cc3nc(C)cs3)CC2)cs1 ZINC000880675876 FE On-Demand Anodyne TRPC6 53 41 CNc1nc(C(=O)N2CCC(O)(Cc3nc(C)cs3)CC2)cs1 ZINC000880675876 FE On-Demand Anodyne TRPC3 47 41 C[C@H](Oc1ccnc(NC(=O)[C@H]2CCC(=O)O2)c1)c1ccccc1 ZINC000880675891 EF On-Demand Anodyne TYK2 44 35 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880675893 EG On-Demand Anodyne KCNH2 40 38 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1C[C@H](O)C1 ZINC000880675903 CD On-Demand Anodyne EPHX2 18 50 CCO[C@@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880676004 DF On-Demand Anodyne EPHX2 33 43 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCOC2)CC1 ZINC000880676007 FF On-Demand Anodyne EPHX2 29 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880676008 FF On-Demand Anodyne EPHX2 29 44 CO[C@@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880676012 CF On-Demand Anodyne EPHX2 25 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(CCF)CC1 ZINC000880676025 DH On-Demand Anodyne RBP4 41 37 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880676042 DE On-Demand Anodyne EPHX2 18 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2ccco2)CC1 ZINC000880676069 EI On-Demand Anodyne RBP4 41 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880676083 GH On-Demand Anodyne EPHX2 26 57 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880676084 GH On-Demand Anodyne EPHX2 26 57 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN2C(=O)OC[C@H]2C1 ZINC000880676136 GE On-Demand Anodyne HCRTR2 15 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCN2C(=O)OC[C@@H]2C1 ZINC000880676137 GE On-Demand Anodyne HCRTR2 15 41 CCOC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676152 EE On-Demand Reactive KCNK3 43 43 CCOC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676152 EE On-Demand Reactive KCNK9 43 43 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)COC(=O)N2 ZINC000880676159 GF On-Demand Anodyne EPHX2 29 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880676160 GG On-Demand Anodyne EPHX2 49 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880676160 GG On-Demand Anodyne RBP4 31 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880676160 GG On-Demand Anodyne SCD1 15 45 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880676160 GG On-Demand Anodyne KCNK3 24 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(OC(C)=O)CC1 ZINC000880676160 GG On-Demand Anodyne KCNK9 28 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CC1 ZINC000880676163 EE On-Demand Reactive KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CC1 ZINC000880676163 EE On-Demand Reactive KCNK9 29 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(=O)(=O)C(C)(C)C ZINC000880676170 GF On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(=O)(=O)C(C)(C)C ZINC000880676170 GF On-Demand Anodyne KCNK9 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCCC1 ZINC000880676173 EH On-Demand Anodyne KCNK3 26 43 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCCC1 ZINC000880676173 EH On-Demand Anodyne KCNK9 29 43 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880676174 DH On-Demand Mild EPHX2 26 51 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCOC[C@@H](C)C1 ZINC000880676175 EG On-Demand Anodyne EPHX2 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCOC[C@H](C)C1 ZINC000880676176 EG On-Demand Anodyne EPHX2 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCO ZINC000880676202 DD On-Demand Anodyne KCNK3 38 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCO ZINC000880676202 DD On-Demand Anodyne KCNK9 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCCC2(C1)OCCO2 ZINC000880676210 GF On-Demand Anodyne EPHX2 37 47 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCOCC[C@@H]1C ZINC000880676217 EG On-Demand Anodyne EPHX2 15 46 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCOCC[C@H]1C ZINC000880676218 EG On-Demand Anodyne EPHX2 15 46 COCCN(CCF)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880676221 DD On-Demand Anodyne MPO 54 34 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H](O)c1cnn(C)c1 ZINC000880676242 FE On-Demand Anodyne SOAT1 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@@H](O)c1cnn(C)c1 ZINC000880676243 FE On-Demand Anodyne SOAT1 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cccn1C ZINC000880676268 EG On-Demand Anodyne SOAT1 27 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cccn1C ZINC000880676268 EG On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1cccn1C ZINC000880676268 EG On-Demand Anodyne KCNK9 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(C)(=O)=O ZINC000880676279 FD On-Demand Anodyne SOAT1 19 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(C)(=O)=O ZINC000880676279 FD On-Demand Anodyne KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCS(C)(=O)=O ZINC000880676279 FD On-Demand Anodyne KCNK9 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(F)F ZINC000880676286 EF On-Demand Anodyne KCNK3 33 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(F)F ZINC000880676286 EF On-Demand Anodyne KCNK9 35 44 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)OC ZINC000880676292 CF On-Demand Anodyne KCNK3 39 47 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)OC ZINC000880676292 CF On-Demand Anodyne KCNK9 40 47 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)CCS(C)(=O)=O ZINC000880676293 FE On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)CCS(C)(=O)=O ZINC000880676293 FE On-Demand Anodyne KCNK9 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC(C)C ZINC000880676302 EF On-Demand Reactive KCNK3 33 43 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC(C)C ZINC000880676302 EF On-Demand Reactive KCNK9 35 43 COC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676305 DD On-Demand Reactive KCNK3 39 47 COC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676305 DD On-Demand Reactive KCNK9 40 47 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@](C)(CO)C1CC1 ZINC000880676310 EF On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@](C)(CO)C1CC1 ZINC000880676310 EF On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@](C)(CO)C1CC1 ZINC000880676311 EF On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@](C)(CO)C1CC1 ZINC000880676311 EF On-Demand Anodyne KCNK9 27 40 CCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676315 CF On-Demand Anodyne KCNK3 46 46 CCONC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676315 CF On-Demand Anodyne KCNK9 46 46 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2ccc(C(C)(C)C)cc2)n1 ZINC000880676322 EF On-Demand Anodyne SLC12A5 54 36 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2ccc(C(C)(C)C)cc2)n1 ZINC000880676323 EF On-Demand Anodyne SLC12A5 54 36 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(C1)OCCO2 ZINC000880676346 FF On-Demand Anodyne EPHX2 39 51 COCC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676359 ED On-Demand Reactive KCNK3 38 44 COCC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676359 ED On-Demand Reactive KCNK9 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1ccncc1 ZINC000880676375 FG On-Demand Anodyne RAF1 20 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1ccncc1 ZINC000880676375 FG On-Demand Anodyne FLT1 15 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1ccncc1 ZINC000880676375 FG On-Demand Anodyne KCNK3 37 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1ccncc1 ZINC000880676375 FG On-Demand Anodyne KCNK9 38 42 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C(C)(C)C ZINC000880676395 EF On-Demand Reactive KCNK3 33 45 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C(C)(C)C ZINC000880676395 EF On-Demand Reactive KCNK9 35 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CCNC2=O)CC1 ZINC000880676415 EE On-Demand Anodyne CACNA1H 53 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2COC[C@H]2C1 ZINC000880676423 DE On-Demand Anodyne RBP4 47 34 CN1CCN(C2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)CC1 ZINC000880676424 FE On-Demand Anodyne L3MBTL3 70 42 CCC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676428 DE On-Demand Reactive KCNK3 38 44 CCC(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676428 DE On-Demand Reactive KCNK9 39 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880676431 GI On-Demand Anodyne SMO 39 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880676431 GI On-Demand Anodyne ETHR 63 49 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCO1 ZINC000880676432 FE On-Demand Anodyne SOAT1 21 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCO1 ZINC000880676432 FE On-Demand Anodyne KCNK3 32 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCC1(C)OCCO1 ZINC000880676432 FE On-Demand Anodyne KCNK9 34 43 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCOCC1 ZINC000880676441 FF On-Demand Anodyne KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)NOC1CCOCC1 ZINC000880676441 FF On-Demand Anodyne KCNK9 28 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880676446 GG On-Demand Anodyne ETHR 47 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880676447 GG On-Demand Anodyne ETHR 47 36 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)OC(C)(C)C ZINC000880676452 FG On-Demand Reactive KCNK3 26 44 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)OC(C)(C)C ZINC000880676452 FG On-Demand Reactive KCNK9 30 44 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CCC(C)(O)CC1 ZINC000880676454 FG On-Demand Anodyne EPHX2 46 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CCC(C)(O)CC1 ZINC000880676454 FG On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CCC(C)(O)CC1 ZINC000880676454 FG On-Demand Anodyne KCNK9 27 40 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)[C@H](C)C(N)=O ZINC000880676481 ED On-Demand Anodyne KCNK3 27 43 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)[C@H](C)C(N)=O ZINC000880676481 ED On-Demand Anodyne KCNK9 31 43 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)[C@@H](C)C(N)=O ZINC000880676482 ED On-Demand Anodyne KCNK3 27 43 COc1cccc(OC(F)(F)F)c1NC(=O)N(C)[C@@H](C)C(N)=O ZINC000880676482 ED On-Demand Anodyne KCNK9 31 43 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCCC1 ZINC000880676494 FF On-Demand Reactive KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCCC1 ZINC000880676494 FF On-Demand Reactive KCNK9 28 41 C[C@@H](C#N)N(C(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1)C1CC1 ZINC000880676495 GF On-Demand Mild GPR119 40 47 C[C@H](C#N)N(C(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1)C1CC1 ZINC000880676496 GF On-Demand Mild GPR119 40 47 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880676507 GG On-Demand Anodyne EPHX2 49 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880676507 GG On-Demand Anodyne RBP4 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880676507 GG On-Demand Anodyne KCNK3 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(C2OCCO2)CC1 ZINC000880676507 GG On-Demand Anodyne KCNK9 28 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@](O)(Cc2ccc(F)cc2)C1 ZINC000880676527 GH On-Demand Anodyne S1PR2 28 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@](O)(Cc2ccc(F)cc2)C1 ZINC000880676529 GH On-Demand Anodyne S1PR2 28 40 C[C@H]1c2sccc2CCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880676534 EI On-Demand Anodyne TRPM8 26 43 COc1ccc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)nc1 ZINC000880676606 GG On-Demand Anodyne PDGFRB 52 39 COc1ccc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)nc1 ZINC000880676606 GG On-Demand Anodyne RBP4 25 40 COc1ccc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)nc1 ZINC000880676606 GG On-Demand Anodyne DGAT1 29 52 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1nncn1C ZINC000880676637 EE On-Demand Anodyne SOAT1 45 41 CC[C@@H](C)C(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676638 EF On-Demand Reactive SOAT1 46 38 CC[C@@H](C)C(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676638 EF On-Demand Reactive KCNK3 38 42 CC[C@@H](C)C(=O)NNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676638 EF On-Demand Reactive KCNK9 39 42 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCC(F)(F)F ZINC000880676644 FH On-Demand Anodyne KCNK3 32 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCCC(F)(F)F ZINC000880676644 FH On-Demand Anodyne KCNK9 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)c1ccc[nH]1 ZINC000880676665 EH On-Demand Anodyne KCNK3 26 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](C)c1ccc[nH]1 ZINC000880676665 EH On-Demand Anodyne KCNK9 29 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)c1ccc[nH]1 ZINC000880676666 EH On-Demand Anodyne KCNK3 26 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](C)c1ccc[nH]1 ZINC000880676666 EH On-Demand Anodyne KCNK9 29 40 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](CO)C1CC1 ZINC000880676672 EE On-Demand Anodyne KCNK3 32 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](CO)C1CC1 ZINC000880676672 EE On-Demand Anodyne KCNK9 34 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](CO)C1CC1 ZINC000880676673 EE On-Demand Anodyne KCNK3 32 42 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](CO)C1CC1 ZINC000880676673 EE On-Demand Anodyne KCNK9 34 42 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC(c2cn[nH]c2)CC1 ZINC000880676688 GH On-Demand Anodyne RBP4 34 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1cccnc1 ZINC000880676696 FG On-Demand Anodyne PTAFR 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1cccnc1 ZINC000880676696 FG On-Demand Anodyne RAF1 17 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCc1cccnc1 ZINC000880676696 FG On-Demand Anodyne NAMPT 34 49 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@H](O)CC1 ZINC000880676714 DF On-Demand Anodyne EPHX2 41 56 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C3)c1 ZINC000880676720 GE On-Demand Anodyne P2RX7 22 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CC(OC)C1 ZINC000880676722 EF On-Demand Anodyne KCNK3 25 42 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CC(OC)C1 ZINC000880676722 EF On-Demand Anodyne KCNK9 29 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1ccn(C)n1 ZINC000880676768 EF On-Demand Anodyne SOAT1 24 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@@](=O)C(C)(C)C ZINC000880676778 GG On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@@](=O)C(C)(C)C ZINC000880676778 GG On-Demand Anodyne KCNK9 32 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@](=O)C(C)(C)C ZINC000880676779 GG On-Demand Anodyne KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCC[S@](=O)C(C)(C)C ZINC000880676779 GG On-Demand Anodyne KCNK9 32 41 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880676781 EI On-Demand Mild EPHX2 29 40 COc1cccc(OC(F)(F)F)c1NC(=O)N1CCC2(CC1)CNC(=O)C2 ZINC000880676786 GF On-Demand Anodyne EPHX2 29 41 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC1(C)OCCO1 ZINC000880676790 FF On-Demand Anodyne SOAT1 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](C(F)(F)F)C1 ZINC000880676791 EI On-Demand Mild RBP4 45 32 C#C[C@@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676797 DF On-Demand Mild KCNK3 27 43 C#C[C@@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676797 DF On-Demand Mild KCNK9 31 43 C#C[C@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676798 DF On-Demand Mild KCNK3 27 43 C#C[C@H](C)NC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676798 DF On-Demand Mild KCNK9 31 43 C#CCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676804 CE On-Demand Mild SOAT1 18 40 C#CCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676804 CE On-Demand Mild KCNK3 38 44 C#CCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676804 CE On-Demand Mild KCNK9 39 44 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](CCO)C1CC1 ZINC000880676810 EF On-Demand Anodyne KCNK3 31 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@@H](CCO)C1CC1 ZINC000880676810 EF On-Demand Anodyne KCNK9 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](CCO)C1CC1 ZINC000880676811 EF On-Demand Anodyne KCNK3 31 41 COc1cccc(OC(F)(F)F)c1NC(=O)N[C@H](CCO)C1CC1 ZINC000880676811 EF On-Demand Anodyne KCNK9 33 41 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@H](O)c1ccsc1 ZINC000880676826 GH On-Demand Anodyne SOAT1 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)NC[C@@H](O)c1ccsc1 ZINC000880676827 GH On-Demand Anodyne SOAT1 28 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCCCN1CCOC1=O ZINC000880676831 GF On-Demand Anodyne SOAT1 23 42 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC1CC1 ZINC000880676832 EF On-Demand Reactive KCNK3 30 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC1CC1 ZINC000880676832 EF On-Demand Reactive KCNK9 32 41 C#CCCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676852 DF On-Demand Mild KCNK3 37 42 C#CCCNC(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880676852 DF On-Demand Mild KCNK9 38 42 COc1cccc(OC(F)(F)F)c1NC(=O)NCc1nnc(S)n1C ZINC000880676861 GE On-Demand Anodyne SOAT1 30 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C1CC1)[C@@H](C)C#N ZINC000880676957 ED On-Demand Mild PAPA1_CARPA 34 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C1CC1)[C@H](C)C#N ZINC000880676958 ED On-Demand Mild PAPA1_CARPA 34 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C1CC1)[C@@H](C)C#N ZINC000880676959 ED On-Demand Mild PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C1CC1)[C@H](C)C#N ZINC000880676960 ED On-Demand Mild PAPA1_CARPA 34 42 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC(F)(F)F ZINC000880676975 GF On-Demand Reactive KCNK3 32 44 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CC(F)(F)F ZINC000880676975 GF On-Demand Reactive KCNK9 34 44 CCOC(=O)[C@@H]1CN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)CCO1 ZINC000880676989 GE On-Demand Anodyne EPHX2 26 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880676991 DH On-Demand Anodyne RBP4 47 34 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](OC)C1 ZINC000880677003 EF On-Demand Anodyne EPHX2 47 39 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](OC)C1 ZINC000880677003 EF On-Demand Anodyne KCNK3 24 41 COc1cccc(OC(F)(F)F)c1NC(=O)N1CC[C@@H](OC)C1 ZINC000880677003 EF On-Demand Anodyne KCNK9 28 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC2(CC1)COC2 ZINC000880677022 EG On-Demand Anodyne EPHX2 19 50 COc1cccc(OC(F)(F)F)c1NC(=O)NC1CCC2(CC1)OCCO2 ZINC000880677130 GG On-Demand Anodyne EPHX2 42 39 C#CCN(CC)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880677132 DG On-Demand Mild KCNK3 36 41 C#CCN(CC)C(=O)Nc1c(OC)cccc1OC(F)(F)F ZINC000880677132 DG On-Demand Mild KCNK9 37 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(C)=O ZINC000880677139 DD On-Demand Reactive KCNK3 39 47 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(C)=O ZINC000880677139 DD On-Demand Reactive KCNK9 40 47 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@@](C)=O ZINC000880677145 FE On-Demand Anodyne SOAT1 23 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@@](C)=O ZINC000880677145 FE On-Demand Anodyne KCNK3 38 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@@](C)=O ZINC000880677145 FE On-Demand Anodyne KCNK9 39 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@](C)=O ZINC000880677146 FE On-Demand Anodyne SOAT1 23 40 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@](C)=O ZINC000880677146 FE On-Demand Anodyne KCNK3 38 43 COc1cccc(OC(F)(F)F)c1NC(=O)NCCC[S@](C)=O ZINC000880677146 FE On-Demand Anodyne KCNK9 39 43 COC(=O)[C@@]1(F)CCN(C(=O)Nc2c(OC)cccc2OC(F)(F)F)C1 ZINC000880677167 GF On-Demand Anodyne EPHX2 35 45 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCC1 ZINC000880677172 EF On-Demand Reactive KCNK3 25 41 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C1CCC1 ZINC000880677172 EF On-Demand Reactive KCNK9 28 41 COc1ccccc1[C@@H]1CN(C(=O)Nc2cc(F)c(F)c(F)c2F)CCO1 ZINC000880677185 GH On-Demand Anodyne RBP4 51 43 COc1ccccc1[C@H]1CN(C(=O)Nc2cc(F)c(F)c(F)c2F)CCO1 ZINC000880677186 GH On-Demand Anodyne RBP4 51 43 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C(C)C ZINC000880677197 EE On-Demand Reactive SOAT1 18 40 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C(C)C ZINC000880677197 EE On-Demand Reactive KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)C(C)C ZINC000880677197 EE On-Demand Reactive KCNK9 36 44 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CN(C)C ZINC000880677204 FD On-Demand Reactive KCNK3 31 42 COc1cccc(OC(F)(F)F)c1NC(=O)NNC(=O)CN(C)C ZINC000880677204 FD On-Demand Reactive KCNK9 33 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880677205 EG On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H]2CSC[C@H]2C1 ZINC000880677206 EG On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880677207 EG On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880677208 EG On-Demand Anodyne RBP4 44 32 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(C)C ZINC000880677216 DG On-Demand Anodyne SOAT1 22 40 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(C)C ZINC000880677216 DG On-Demand Anodyne KCNK3 34 44 COc1cccc(OC(F)(F)F)c1NC(=O)NOCC(C)C ZINC000880677216 DG On-Demand Anodyne KCNK9 36 44 CN1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)Cc2cccnc21 ZINC000880677219 FG On-Demand Anodyne RBP4 16 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](c2cccnc2)C1 ZINC000880677232 EH On-Demand Anodyne RBP4 47 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](c2cccnc2)C1 ZINC000880677233 EH On-Demand Anodyne RBP4 47 36 CN1CCC[C@@H](CCNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677273 EG On-Demand Anodyne CCR3 46 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](CC(F)(F)F)C1 ZINC000880677284 FI On-Demand Mild RBP4 44 31 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](CC(F)(F)F)C1 ZINC000880677285 FI On-Demand Mild RBP4 44 31 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880677320 GH On-Demand Anodyne TRPM8 33 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880677321 GH On-Demand Anodyne TRPM8 33 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880677322 GH On-Demand Anodyne TRPM8 33 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880677323 GH On-Demand Anodyne TRPM8 33 45 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CC=CC1 ZINC000880677353 CG On-Demand Anodyne EPHX2 15 51 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCOC1 ZINC000880677382 CE On-Demand Anodyne EPHX2 15 49 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677409 EG On-Demand Anodyne CACNA1I 55 35 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677410 EG On-Demand Anodyne CACNA1I 55 35 CC[C@@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CCO1 ZINC000880677463 DG On-Demand Anodyne EPHX2 15 43 CC[C@H]1C[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CCO1 ZINC000880677464 DG On-Demand Anodyne EPHX2 15 43 CC[C@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CCO1 ZINC000880677465 DG On-Demand Anodyne EPHX2 15 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880677507 EF On-Demand Anodyne RBP4 55 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880677508 EF On-Demand Anodyne RBP4 55 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880677509 EF On-Demand Anodyne RBP4 55 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880677510 EF On-Demand Anodyne RBP4 55 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880677519 GF On-Demand Anodyne L3MBTL3 70 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880677520 GF On-Demand Anodyne L3MBTL3 70 40 O=C1C[C@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677523 GH On-Demand Anodyne NPY5R 18 40 O=C1C[C@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677523 GH On-Demand Anodyne EPHX2 27 49 O=C1C[C@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677523 GH On-Demand Anodyne TRPM8 30 44 O=C1C[C@@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677524 GH On-Demand Anodyne NPY5R 18 40 O=C1C[C@@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677524 GH On-Demand Anodyne EPHX2 27 49 O=C1C[C@@]2(CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)C2)Oc2ccccc21 ZINC000880677524 GH On-Demand Anodyne TRPM8 30 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC(OC(F)F)CC1 ZINC000880677528 FH On-Demand Anodyne EPHX2 44 49 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC1 ZINC000880677536 CF On-Demand Anodyne EPHX2 54 67 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677546 FD On-Demand Anodyne EPHX2 44 48 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677547 FD On-Demand Anodyne EPHX2 44 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CC1)OCCc1ccccc12 ZINC000880677570 GI On-Demand Anodyne NPY5R 27 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880677587 DF On-Demand Anodyne PTGES 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCC[C@H](CO)C1 ZINC000880677588 DF On-Demand Anodyne PTGES 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCC[C@@H](CO)C1 ZINC000880677589 DF On-Demand Anodyne PTGES 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCC[C@H](CO)C1 ZINC000880677590 DF On-Demand Anodyne PTGES 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880677592 GF On-Demand Bother PDGFRB 21 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880677592 GF On-Demand Bother TRPV1 15 59 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880677592 GF On-Demand Bother RBP4 15 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880677598 CG On-Demand Anodyne EPHX2 16 51 O=C(Nc1cc(F)c(F)c(F)c1F)NC1C[C@H]2C[C@@H]2C1 ZINC000880677599 CG On-Demand Anodyne EPHX2 16 51 O=C(Nc1cc(F)c(F)c(F)c1F)NC1C[C@@H]2C[C@H]2C1 ZINC000880677600 CG On-Demand Anodyne EPHX2 16 51 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2CCCC[C@H]2C1 ZINC000880677601 DH On-Demand Anodyne RBP4 47 34 O=C(Nc1cc(F)c(F)c(F)c1F)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880677682 FG On-Demand Anodyne EPHX2 51 58 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@@H](O)CC1 ZINC000880677735 DF On-Demand Anodyne EPHX2 41 56 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880677753 GG On-Demand Anodyne EPHX2 57 48 COCC1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880677773 EH On-Demand Anodyne EPHX2 43 48 NC(=O)[C@@H]1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677792 DE On-Demand Anodyne EPHX2 19 48 CCCN(CCN1CCCC1)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880677822 EH On-Demand Anodyne CASR 44 36 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCCN(CCCO)C1 ZINC000880677846 EE On-Demand Anodyne CCR3 41 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCCN(CCCO)C1 ZINC000880677846 EE On-Demand Anodyne BIRC2 32 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCCN(CCCO)C1 ZINC000880677847 EE On-Demand Anodyne CCR3 41 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCCN(CCCO)C1 ZINC000880677847 EE On-Demand Anodyne BIRC2 32 40 CCOC(=O)C1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880677882 FG On-Demand Anodyne EPHX2 48 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880677883 EG On-Demand Anodyne CPT1A 46 37 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880677884 EG On-Demand Anodyne CPT1A 46 37 CN(C)S(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880677895 GD On-Demand Anodyne EPHX2 17 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC(C2CCOCC2)C1 ZINC000880677896 EG On-Demand Anodyne RBP4 45 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CCC2)C1 ZINC000880677924 DH On-Demand Anodyne EPHX2 30 44 CN1CCC(N2CCC(NC(=O)Nc3cc(F)c(F)c(F)c3F)CC2)CC1 ZINC000880677956 GF On-Demand Anodyne SLC6A5 17 42 CN1CCC(N2CCC(NC(=O)Nc3cc(F)c(F)c(F)c3F)CC2)CC1 ZINC000880677956 GF On-Demand Anodyne EPHX2 37 46 CN(C(=O)[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1)c1ccccc1 ZINC000880677958 GH On-Demand Anodyne RBP4 52 34 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCOC2(CCCCC2)C1 ZINC000880677986 EH On-Demand Anodyne EPHX2 20 45 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCOC1=O ZINC000880678004 CD On-Demand Anodyne LUXR 79 45 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCOC1=O ZINC000880678004 CD On-Demand Anodyne TRAR 92 42 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCOC1=O ZINC000880678004 CD On-Demand Anodyne LASR 65 40 CN(C)C1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678021 EG On-Demand Anodyne EPHX2 48 51 COc1cnccc1N1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678026 GG On-Demand Anodyne HTR1B 15 47 COc1cnccc1N1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678026 GG On-Demand Anodyne PDGFRB 52 45 COc1cnccc1N1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678026 GG On-Demand Anodyne RBP4 24 48 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1C[C@H](O)C1 ZINC000880678033 CD On-Demand Anodyne EPHX2 18 50 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](C2CCC2)C1 ZINC000880678081 DH On-Demand Anodyne RBP4 52 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](C2CCC2)C1 ZINC000880678082 DH On-Demand Anodyne RBP4 52 33 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C2CCC2)CC1 ZINC000880678088 EG On-Demand Anodyne EPHX2 48 52 CCO[C@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678108 DF On-Demand Anodyne EPHX2 33 43 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cc(F)c(F)c(F)c1F)C2 ZINC000880678111 EF On-Demand Anodyne EPHX2 26 47 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cc(F)c(F)c(F)c1F)C2 ZINC000880678111 EF On-Demand Anodyne GLRA1 44 32 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678119 DF On-Demand Anodyne CHRNA10 55 38 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678119 DF On-Demand Anodyne ACKR3 53 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678120 DF On-Demand Anodyne CHRNA10 55 38 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678120 DF On-Demand Anodyne ACKR3 53 33 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880678187 GH On-Demand Mild CACNA1I 67 40 N#Cc1ccc(OC2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)cc1 ZINC000880678206 GI On-Demand Mild EPHX2 27 55 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CC(N2CCCCC2)C1 ZINC000880678233 EG On-Demand Anodyne EPHX2 15 49 N#C[C@H]1CC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678277 DG On-Demand Mild EPHX2 15 46 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678309 DE On-Demand Anodyne EPHX2 18 46 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678333 GF On-Demand Mild EPHX2 26 41 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCc2nnnn2CC1 ZINC000880678346 ED On-Demand Anodyne EPHX2 32 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCc2nnnn2CC1 ZINC000880678347 ED On-Demand Anodyne EPHX2 32 44 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678394 GG On-Demand Anodyne EPHX2 38 46 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678394 GG On-Demand Anodyne DPP7 48 37 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678394 GG On-Demand Anodyne RBP4 52 34 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678394 GG On-Demand Anodyne CACNA1G 40 37 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678395 GG On-Demand Anodyne EPHX2 38 46 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678395 GG On-Demand Anodyne DPP7 48 37 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678395 GG On-Demand Anodyne RBP4 52 34 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678395 GG On-Demand Anodyne CACNA1G 40 37 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880678396 GH On-Demand Anodyne EPHX2 27 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880678396 GH On-Demand Anodyne SCD1 16 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880678417 GH On-Demand Anodyne CACNA1H 43 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880678417 GH On-Demand Anodyne EPHX2 21 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880678417 GH On-Demand Anodyne RBP4 53 34 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCOC1 ZINC000880678428 CE On-Demand Anodyne EPHX2 15 49 CN1CC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678443 DE On-Demand Anodyne CACNA1I 64 35 CN1CC[C@@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678444 DE On-Demand Anodyne CACNA1I 64 35 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678490 GD On-Demand Anodyne HLA-DRB1 46 35 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678493 GD On-Demand Anodyne HLA-DRB1 46 35 C[C@@H]1CN(CCCNC(=O)Nc2cc(F)c(F)c(F)c2F)CCCO1 ZINC000880678505 FF On-Demand Anodyne CCR3 38 43 COc1cc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)ncn1 ZINC000880678518 GE On-Demand Anodyne PDGFRB 52 40 COc1cc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)ncn1 ZINC000880678518 GE On-Demand Anodyne RBP4 20 40 COC(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678571 EF On-Demand Anodyne EPHX2 59 49 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880678577 GG On-Demand Anodyne FAAH 17 40 O=C(NCCCNC(=O)C1CCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880678595 EF On-Demand Anodyne TBK1 68 38 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880678625 FE On-Demand Anodyne CCR3 46 37 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880678674 FH On-Demand Anodyne NPY5R 27 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880678675 FH On-Demand Anodyne NPY5R 27 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(c2cccnn2)CC1 ZINC000880678684 FF On-Demand Anodyne EPHX2 39 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@@]2(CCOC2)C1 ZINC000880678701 EE On-Demand Anodyne EPHX2 18 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@]2(CCOC2)C1 ZINC000880678702 EE On-Demand Anodyne EPHX2 18 42 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)C1CC1 ZINC000880678716 FF On-Demand Anodyne EPHX2 39 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880678732 GI On-Demand Anodyne CACNA1H 42 31 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC2(CCOCC2)C1 ZINC000880678737 EH On-Demand Anodyne EPHX2 26 41 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678766 FE On-Demand Anodyne EPHX2 46 43 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678767 FE On-Demand Anodyne EPHX2 46 43 C[C@]1(O)CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678793 DF On-Demand Anodyne EPHX2 21 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](Cc2ccncc2)C1 ZINC000880678794 FH On-Demand Anodyne GRIN2B 40 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](Cc2ccncc2)C1 ZINC000880678794 FH On-Demand Anodyne CCR3 72 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880678795 FH On-Demand Anodyne GRIN2B 40 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880678795 FH On-Demand Anodyne CCR3 72 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880678862 FG On-Demand Anodyne EPHX2 25 47 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cc(F)c(F)c(F)c1F ZINC000880678886 GF On-Demand Anodyne PIK3CB 68 38 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cc(F)c(F)c(F)c1F ZINC000880678886 GF On-Demand Anodyne STAT6 41 35 CC1CN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678911 CF On-Demand Anodyne RBP4 52 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Oc2ncccc2F)CC1 ZINC000880678926 GH On-Demand Anodyne EPHX2 20 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Oc2ncccc2F)CC1 ZINC000880678926 GH On-Demand Anodyne SCD1 17 46 O=C(NCCN1CCCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880678927 EE On-Demand Anodyne EPHX2 23 47 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678928 EF On-Demand Anodyne EPHX2 46 41 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880678929 EF On-Demand Anodyne EPHX2 46 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCOC2(CCC2)C1 ZINC000880678993 DG On-Demand Anodyne EPHX2 22 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2cccnc2)CC1 ZINC000880679018 FI On-Demand Anodyne RBP4 41 37 O=C(NCc1cccc(OC2CC2)c1F)[C@@H]1CCc2nncn2CC1 ZINC000880679044 EE On-Demand Anodyne P2RX7 46 41 O=C(NCc1cccc(OC2CC2)c1F)[C@@H]1CCc2nncn2CC1 ZINC000880679044 EE On-Demand Anodyne EPHX2 18 41 O=C(NCc1cccc(OC2CC2)c1F)[C@H]1CCc2nncn2CC1 ZINC000880679045 EE On-Demand Anodyne P2RX7 46 41 O=C(NCc1cccc(OC2CC2)c1F)[C@H]1CCc2nncn2CC1 ZINC000880679045 EE On-Demand Anodyne EPHX2 18 41 O=C(NCC1CCN(C2CC2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880679063 EG On-Demand Anodyne CACNA1I 56 33 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(c2nccs2)CC1 ZINC000880679128 FG On-Demand Anodyne EPHX2 35 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880679133 FH On-Demand Anodyne CACNA1H 43 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880679133 FH On-Demand Anodyne OPRL1 17 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880679133 FH On-Demand Anodyne CCR1 28 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880679133 FH On-Demand Anodyne RBP4 46 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(Cc2ccccn2)CC1 ZINC000880679141 FF On-Demand Anodyne FAAH 27 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](c2ccccn2)C1 ZINC000880679150 EH On-Demand Anodyne RBP4 61 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](c2ccccn2)C1 ZINC000880679151 EH On-Demand Anodyne RBP4 61 38 O=C(Nc1cc(F)c(F)c(F)c1F)NC12CCC(CC1)C2 ZINC000880679170 DH On-Demand Anodyne EPHX2 38 57 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679223 FG On-Demand Anodyne CCR3 42 38 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679224 FG On-Demand Anodyne CCR3 42 38 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679225 FG On-Demand Anodyne CCR3 42 38 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679226 FG On-Demand Anodyne CCR3 42 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](C2CC2)C1 ZINC000880679239 DH On-Demand Anodyne RBP4 53 34 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](C2CC2)C1 ZINC000880679240 DH On-Demand Anodyne RBP4 53 34 C[C@@H]1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)[C@@H]1C ZINC000880679247 DH On-Demand Anodyne TRPC6 58 43 C[C@@H]1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)[C@@H]1C ZINC000880679247 DH On-Demand Anodyne TRPC3 40 43 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679249 DH On-Demand Anodyne TRPC6 58 43 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880679249 DH On-Demand Anodyne TRPC3 40 43 CCC1(O)CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880679257 EG On-Demand Anodyne EPHX2 34 48 O=C(CC[C@@H]1CCc2ccccc21)NCCO[C@@H]1CC1(F)F ZINC000880679258 DG On-Demand Anodyne NQO2 21 43 O=C(CC[C@H]1CCc2ccccc21)NCCO[C@H]1CC1(F)F ZINC000880679259 DG On-Demand Anodyne NQO2 21 43 O=C(CC[C@H]1CCc2ccccc21)NCCO[C@@H]1CC1(F)F ZINC000880679260 DG On-Demand Anodyne NQO2 21 43 O=C(CC[C@@H]1CCc2ccccc21)NCCO[C@H]1CC1(F)F ZINC000880679261 DG On-Demand Anodyne NQO2 21 43 O=C(NCC1CCN(c2ccncc2)CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880679268 GH On-Demand Anodyne F10 15 53 CC1(C)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880679275 DH On-Demand Anodyne CACNA1H 40 36 COC[C@@H](C)n1ccc(NC(=O)Nc2cc(F)c(F)c(F)c2F)n1 ZINC000880679289 EG On-Demand Anodyne GCK 19 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC(C2CCCC2)C1 ZINC000880679297 DH On-Demand Anodyne RBP4 47 34 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880679302 GH On-Demand Anodyne EPHX2 27 49 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC2(CC2)C1 ZINC000880679315 DH On-Demand Anodyne EPHX2 29 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCSC1 ZINC000880679318 CF On-Demand Anodyne EPHX2 15 50 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCSC1 ZINC000880679319 CF On-Demand Anodyne EPHX2 15 50 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(c2ncccc2F)CC1 ZINC000880679322 GH On-Demand Anodyne TRPV1 15 47 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(c2ncccc2F)CC1 ZINC000880679322 GH On-Demand Anodyne RBP4 18 51 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCn2ccnc2C1 ZINC000880679381 EF On-Demand Anodyne EPHX2 21 45 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCn2ccnc2C1 ZINC000880679382 EF On-Demand Anodyne EPHX2 21 45 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880679383 GJ On-Demand Anodyne SLC18A3 34 43 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880679383 GJ On-Demand Anodyne WNT3A 46 34 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880679396 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880679397 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@@H]2C1 ZINC000880679398 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880679399 GG On-Demand Anodyne CHRNA4 27 49 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880679402 GG On-Demand Anodyne EPHX2 15 41 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880679402 GG On-Demand Anodyne STAT6 51 37 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](C2CC2)C1 ZINC000880679404 DH On-Demand Anodyne RBP4 51 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](C2CC2)C1 ZINC000880679405 DH On-Demand Anodyne RBP4 51 33 O=C(NCCCCCN1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880679416 EH On-Demand Anodyne CCR3 31 41 O=C(NCCCCCN1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880679416 EH On-Demand Anodyne CHRNA7 21 54 O=C(NCCCCCN1CCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880679416 EH On-Demand Anodyne HNMT 42 35 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880679436 FG On-Demand Mild EPHX2 50 47 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880679436 FG On-Demand Mild CXCR3 21 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880679436 FG On-Demand Mild HPGDS 39 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC(C(F)(F)F)C1 ZINC000880679439 DG On-Demand Mild RBP4 54 34 CS(=O)(=O)C1CCC(C(=O)NCc2cccc(OC3CC3)c2F)CC1 ZINC000880679550 FF On-Demand Anodyne P2RX7 42 41 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880679572 GG On-Demand Anodyne CCR3 45 40 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880679572 GG On-Demand Anodyne MCHR1 17 42 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880679573 GG On-Demand Anodyne CCR3 45 40 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880679573 GG On-Demand Anodyne MCHR1 17 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2ccccn2)CC1 ZINC000880679582 FI On-Demand Anodyne CACNA1H 35 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2ccccn2)CC1 ZINC000880679582 FI On-Demand Anodyne EPHX2 15 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2ccccn2)CC1 ZINC000880679582 FI On-Demand Anodyne RBP4 64 40 Cn1ncc(Br)c1CC(=O)NCc1cccc(OC2CC2)c1F ZINC000880679619 GF On-Demand Anodyne P2RX7 46 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2F)CC1 ZINC000880679635 FG On-Demand Anodyne PDGFRB 31 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2F)CC1 ZINC000880679635 FG On-Demand Anodyne TRPV1 19 51 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2F)CC1 ZINC000880679635 FG On-Demand Anodyne FAAH 22 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccc2F)CC1 ZINC000880679635 FG On-Demand Anodyne RBP4 27 48 COc1ccccc1-c1ccc(C(=O)NCCO[C@H]2CC2(F)F)c(O)n1 ZINC000880679667 FF On-Demand Anodyne KCNA3 40 36 COc1ccccc1-c1ccc(C(=O)NCCO[C@@H]2CC2(F)F)c(O)n1 ZINC000880679668 FF On-Demand Anodyne KCNA3 40 36 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccc(OC2CC2)c1F ZINC000880679704 GG On-Demand Anodyne P2RX7 46 41 O=C(Cc1ccccc1N1CCCC1=O)NCc1cccc(OC2CC2)c1F ZINC000880679704 GG On-Demand Anodyne PLD1 42 31 O=C1CC[C@@H](c2ccc(C(=O)NCc3cccc(OC4CC4)c3F)cc2)N1 ZINC000880679722 FG On-Demand Anodyne PLD1 49 36 O=C1CC[C@@H](c2ccc(C(=O)NCc3cccc(OC4CC4)c3F)cc2)N1 ZINC000880679722 FG On-Demand Anodyne PLD2 48 35 O=C1CC[C@H](c2ccc(C(=O)NCc3cccc(OC4CC4)c3F)cc2)N1 ZINC000880679723 FG On-Demand Anodyne PLD1 49 36 O=C1CC[C@H](c2ccc(C(=O)NCc3cccc(OC4CC4)c3F)cc2)N1 ZINC000880679723 FG On-Demand Anodyne PLD2 48 35 O=C(NCCO[C@@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880679726 EE On-Demand Anodyne GABRA1 16 47 O=C(NCCO[C@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880679727 EE On-Demand Anodyne GABRA1 16 47 Cn1nnc(C(=O)NCc2cccc(OC3CC3)c2F)n1 ZINC000880679737 CC On-Demand Anodyne SCD1 22 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC(F)(F)CC1 ZINC000880679740 EH On-Demand Anodyne EPHX2 34 53 O=C1CC[C@H](c2ccc(C(=O)NCCO[C@@H]3CC3(F)F)cc2)N1 ZINC000880679745 DD On-Demand Anodyne PLD2 45 33 O=C1CC[C@H](c2ccc(C(=O)NCCO[C@H]3CC3(F)F)cc2)N1 ZINC000880679746 DD On-Demand Anodyne PLD2 45 33 O=C1CC[C@@H](c2ccc(C(=O)NCCO[C@@H]3CC3(F)F)cc2)N1 ZINC000880679747 DD On-Demand Anodyne PLD2 45 33 O=C1CC[C@@H](c2ccc(C(=O)NCCO[C@H]3CC3(F)F)cc2)N1 ZINC000880679748 DD On-Demand Anodyne PLD2 45 33 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880679784 FD On-Demand Anodyne EPHX2 21 40 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880679785 FD On-Demand Anodyne EPHX2 21 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCCOCC1 ZINC000880679797 DF On-Demand Anodyne EPHX2 19 57 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCCOCC1 ZINC000880679798 DF On-Demand Anodyne EPHX2 19 57 O=C(NCCO[C@H]1CC1(F)F)c1ccc(OC(F)F)c(Cl)c1 ZINC000880679822 EG On-Demand Anodyne PDE4D 18 41 O=C(NCCO[C@@H]1CC1(F)F)c1ccc(OC(F)F)c(Cl)c1 ZINC000880679823 EG On-Demand Anodyne PDE4D 18 41 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@@H]1CC1(F)F)C2 ZINC000880679854 EE On-Demand Anodyne NQO2 33 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@@H]1CC1(F)F)C2 ZINC000880679854 EE On-Demand Anodyne MTNR1A 53 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@@H]1CC1(F)F)C2 ZINC000880679854 EE On-Demand Anodyne MTNR1B 47 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@H]1CC1(F)F)C2 ZINC000880679857 EE On-Demand Anodyne NQO2 33 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@H]1CC1(F)F)C2 ZINC000880679857 EE On-Demand Anodyne MTNR1A 53 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCO[C@H]1CC1(F)F)C2 ZINC000880679857 EE On-Demand Anodyne MTNR1B 47 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Cc2cccnc2)CC1 ZINC000880679875 FI On-Demand Anodyne GRIN2B 49 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Cc2cccnc2)CC1 ZINC000880679875 FI On-Demand Anodyne CCR3 44 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Cc2cccnc2)CC1 ZINC000880679875 FI On-Demand Anodyne CHRNA7 52 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Cc2cccnc2)CC1 ZINC000880679875 FI On-Demand Anodyne C3AR1 44 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Cc2cccnc2)CC1 ZINC000880679875 FI On-Demand Anodyne NAMPT 42 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccc(F)cn2)CC1 ZINC000880679910 FG On-Demand Anodyne DGAT1 30 49 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccc(F)cn2)CC1 ZINC000880679910 FG On-Demand Anodyne SLC27A1 42 41 COCC1(O)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880679927 EE On-Demand Anodyne S1PR2 28 41 CS(=O)(=O)Nc1ccc(/C=C\C(=O)NCc2nc3ccccc3s2)cc1 ZINC000880679977 GF On-Demand Anodyne HDAC1 19 41 CN(C)CC1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880680053 EG On-Demand Anodyne EPHX2 44 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne PAPA1_CARPA 47 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne CTSK 20 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne CTSL 21 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne TACR3 15 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne REN 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne CTSS 16 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680082 FF On-Demand Anodyne FPR1 46 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne PAPA1_CARPA 47 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne CTSK 20 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne CTSL 21 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne TACR3 15 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne REN 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne CTSS 16 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)cc(C)c1 ZINC000880680083 FF On-Demand Anodyne FPR1 46 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CC1)OCc1ccccc12 ZINC000880680099 GI On-Demand Anodyne NPY5R 32 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CC1)OCc1ccccc12 ZINC000880680099 GI On-Demand Anodyne MCHR1 16 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(N2CC=CC2)CC1 ZINC000880680146 EG On-Demand Anodyne L3MBTL3 48 38 CC(=O)OC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880680147 EF On-Demand Anodyne SCD1 15 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@@]2(CCCOC2)C1 ZINC000880680211 EF On-Demand Anodyne EPHX2 19 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCO[C@]2(CCCOC2)C1 ZINC000880680212 EF On-Demand Anodyne EPHX2 19 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880680232 EH On-Demand Anodyne CPT1A 42 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880680233 EH On-Demand Anodyne CPT1A 42 38 CN(C(=O)Nc1cc(F)c(F)c(F)c1F)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880680239 EG On-Demand Anodyne GLRA1 43 32 O=C(NC[C@@H](O)CN1CCc2ccccc2C1)Nc1cc(F)c(F)c(F)c1F ZINC000880680241 GF On-Demand Anodyne NOD2 41 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880680359 FG On-Demand Anodyne EPHX2 32 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880680360 FG On-Demand Anodyne EPHX2 32 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC2(CC1)NC(=O)NC2=O ZINC000880680372 FD On-Demand Anodyne EPHX2 15 45 Cn1ccnc(N2CCC(NC(=O)Nc3cc(F)c(F)c(F)c3F)CC2)c1=O ZINC000880680378 GE On-Demand Anodyne EPHX2 27 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880680447 GH On-Demand Anodyne ETHR 52 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880680448 GH On-Demand Anodyne ETHR 52 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(C2CCCC2)CC1 ZINC000880680471 FH On-Demand Anodyne HRH3 24 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(C2CCCC2)CC1 ZINC000880680471 FH On-Demand Anodyne L3MBTL3 63 39 CS(=O)(=O)CC1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880680552 GF On-Demand Anodyne EPHX2 32 47 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880680600 GG On-Demand Mild EPHX2 30 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC(C2CC2)C1 ZINC000880680602 CG On-Demand Anodyne RBP4 54 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880680812 GI On-Demand Anodyne EPHX2 23 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880680812 GI On-Demand Anodyne SLC12A5 40 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880680813 GI On-Demand Anodyne EPHX2 23 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880680813 GI On-Demand Anodyne SLC12A5 40 35 CCN1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880680997 DF On-Demand Anodyne CCR3 44 42 CCN1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880680997 DF On-Demand Anodyne EPHX2 32 48 CCN1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880680998 DF On-Demand Anodyne CCR3 44 42 CCN1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880680998 DF On-Demand Anodyne EPHX2 32 48 CCn1nc2c(cc1=O)CN(C(=O)Nc1cc(F)c(F)c(F)c1F)CC2 ZINC000880681003 FE On-Demand Anodyne P2RY14 44 34 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880681034 GE On-Demand Anodyne EPHX2 46 55 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880681040 FG On-Demand Anodyne EPHX2 38 48 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880681042 FG On-Demand Anodyne EPHX2 38 48 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(c2ccccn2)C1 ZINC000880681078 FG On-Demand Anodyne EPHX2 24 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(c2ccccn2)C1 ZINC000880681080 FG On-Demand Anodyne EPHX2 24 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C2CCCC2)CC1 ZINC000880681081 FH On-Demand Anodyne EPHX2 44 55 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCOC2(CCOCC2)C1 ZINC000880681097 EF On-Demand Anodyne EPHX2 19 44 N#CCCN(CCN1CCOCC1)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681113 FE On-Demand Mild CASR 60 45 COC(=O)c1cccc(NNC(=O)Cc2ccccc2N2CCCC2=O)c1C ZINC000880681165 GF On-Demand Reactive KCNQ2 54 35 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681177 GD On-Demand Anodyne ACOX1 48 32 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681177 GD On-Demand Anodyne ABCB1 22 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880681178 GI On-Demand Anodyne GRIN2B 48 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880681178 GI On-Demand Anodyne SIGMAR1 15 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880681178 GI On-Demand Anodyne CCR3 31 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880681178 GI On-Demand Anodyne RBP4 53 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880681179 GI On-Demand Anodyne GRIN2B 48 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880681179 GI On-Demand Anodyne SIGMAR1 15 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880681179 GI On-Demand Anodyne CCR3 31 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880681179 GI On-Demand Anodyne RBP4 53 35 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cc(F)c(F)c(F)c1F)C2 ZINC000880681206 EG On-Demand Anodyne HTR3A 33 41 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cc(F)c(F)c(F)c1F)C2 ZINC000880681206 EG On-Demand Anodyne EPHX2 26 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCS(=O)(=O)CC1 ZINC000880681233 ED On-Demand Anodyne EPHX2 26 53 CS(=O)(=O)C1CCC(C(=O)NNc2cc(F)cc(Cl)c2)CC1 ZINC000880681238 EF On-Demand Reactive EPHX2 17 41 CCn1cc(CNC(=O)c2sc(-c3ccc(F)c(C)c3)nc2C)nn1 ZINC000880681289 FG On-Demand Anodyne SCD1 29 46 CCn1cc(CNC(=O)c2sc(-c3ccc(F)c(C)c3)nc2C)nn1 ZINC000880681289 FG On-Demand Anodyne SCD 29 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681312 EE On-Demand Anodyne EPHX2 42 51 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681313 EE On-Demand Anodyne EPHX2 42 51 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880681321 GF On-Demand Anodyne EPHX2 47 50 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880681322 GF On-Demand Anodyne EPHX2 47 50 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880681323 GF On-Demand Anodyne EPHX2 47 50 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880681324 GF On-Demand Anodyne EPHX2 47 50 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681326 GG On-Demand Anodyne CCR3 27 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681327 GG On-Demand Anodyne CCR3 27 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCO[C@H](c2ccccc2)C1 ZINC000880681334 FI On-Demand Anodyne RBP4 53 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCO[C@@H](c2ccccc2)C1 ZINC000880681335 FI On-Demand Anodyne RBP4 53 33 CC(C)(C)OC(=O)NC1(CNC(=O)c2c[nH]cc2C2CC2)CCCC1 ZINC000880681377 EG On-Demand Anodyne HCN4 40 31 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681422 DD On-Demand Anodyne LGMN 62 35 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880681448 GG On-Demand Anodyne SLC18A3 29 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880681448 GG On-Demand Anodyne EPHX2 44 53 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880681450 GG On-Demand Anodyne SLC18A3 29 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880681450 GG On-Demand Anodyne EPHX2 44 53 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880681451 GG On-Demand Anodyne SLC18A3 29 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880681451 GG On-Demand Anodyne EPHX2 44 53 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880681453 GG On-Demand Anodyne SLC18A3 29 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880681453 GG On-Demand Anodyne EPHX2 44 53 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CCOCC2)C1 ZINC000880681491 EG On-Demand Anodyne EPHX2 30 43 NC(=O)[C@H]1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681503 EE On-Demand Anodyne EPHX2 16 52 NC(=O)[C@H]1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681504 EE On-Demand Anodyne EPHX2 16 52 NC(=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681505 EE On-Demand Anodyne EPHX2 16 52 NC(=O)[C@@H]1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681507 EE On-Demand Anodyne EPHX2 16 52 C[C@H]1C[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CCN1C ZINC000880681522 DF On-Demand Anodyne EPHX2 34 44 C[C@@H](CCN(C)C)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681543 DF On-Demand Anodyne UTS2 51 33 CC(C)(C)OC(=O)CCC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880681573 FH On-Demand Anodyne GRIN2B 45 36 CCCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681583 EH On-Demand Anodyne HTR4 44 42 CCCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681583 EH On-Demand Anodyne CCR3 40 41 CCCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681583 EH On-Demand Anodyne EPHX2 43 45 CCCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681583 EH On-Demand Anodyne CXCR3 20 40 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681588 FI On-Demand Anodyne DRD4 15 44 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681588 FI On-Demand Anodyne RBP4 73 52 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681589 FI On-Demand Anodyne DRD4 15 44 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681589 FI On-Demand Anodyne RBP4 73 52 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(Nc2cccnn2)CC1 ZINC000880681591 FG On-Demand Anodyne FAAH 24 44 CS[C@H]1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681625 DH On-Demand Anodyne EPHX2 17 46 CS[C@@H]1CC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880681627 DH On-Demand Anodyne EPHX2 17 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2ncc[nH]2)CC1 ZINC000880681633 EG On-Demand Anodyne HTR2B 18 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880681642 GF On-Demand Anodyne EPHX2 25 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880681642 GF On-Demand Anodyne CXCR3 15 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880681644 GF On-Demand Anodyne EPHX2 25 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880681644 GF On-Demand Anodyne CXCR3 15 44 COCCC(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681645 GE On-Demand Anodyne EPHX2 48 44 COCCC(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681645 GE On-Demand Anodyne CCR8 42 36 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@H](CO)CC1 ZINC000880681658 DF On-Demand Anodyne EPHX2 40 52 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880681659 DF On-Demand Anodyne EPHX2 40 52 CCC1(O)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681660 DG On-Demand Anodyne S1PR2 29 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681753 GH On-Demand Anodyne CCR3 21 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880681754 GH On-Demand Anodyne CCR3 21 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C2CC2)CC1 ZINC000880681802 DF On-Demand Anodyne L3MBTL3 40 37 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681803 GG On-Demand Anodyne CACNA1H 42 32 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880681803 GG On-Demand Anodyne RBP4 47 34 CC(C)(C)OC(=O)CCC1CCN(C(=O)c2ncccc2-c2ccccn2)CC1 ZINC000880681935 GI On-Demand Anodyne MLNR 16 40 CC(C)(C)OC(=O)CCC1CCN(C(=O)c2ncccc2-c2ccccn2)CC1 ZINC000880681935 GI On-Demand Anodyne GPR119 20 42 CC(C)(C)N1C[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1=O ZINC000880682012 EF On-Demand Anodyne EPHX2 18 41 CC(C)(C)N1C[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1=O ZINC000880682013 EF On-Demand Anodyne EPHX2 18 41 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)c1ccccc1 ZINC000880682019 GH On-Demand Anodyne DRD4 22 43 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)c1ccccc1 ZINC000880682019 GH On-Demand Anodyne MAPK13 66 31 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)c1ccccc1 ZINC000880682019 GH On-Demand Anodyne EPHX2 41 42 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)c1ccccc1 ZINC000880682019 GH On-Demand Anodyne RBP4 48 38 O=C(NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1)c1ccccc1 ZINC000880682019 GH On-Demand Anodyne MCHR1 19 47 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC2(CCCC2)C1 ZINC000880682064 DI On-Demand Anodyne EPHX2 30 44 N#Cc1cccc(OC2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)c1 ZINC000880682119 GI On-Demand Mild CCR3 24 42 N#Cc1cccc(OC2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)c1 ZINC000880682119 GI On-Demand Mild EPHX2 22 57 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2cccnn2)CC1 ZINC000880682159 FE On-Demand Anodyne FAAH 25 45 COC(=O)C1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682172 EG On-Demand Anodyne EPHX2 47 50 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880682176 FG On-Demand Anodyne EPHX2 20 44 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880682178 FG On-Demand Anodyne EPHX2 20 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](c2ccco2)C1 ZINC000880682197 EH On-Demand Anodyne RBP4 41 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](c2ccco2)C1 ZINC000880682199 EH On-Demand Anodyne RBP4 41 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC(CC(F)(F)F)C1 ZINC000880682209 EH On-Demand Mild RBP4 51 33 O=C(NC[C@@H](O)COCC1CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880682236 EE On-Demand Anodyne ADRB1 18 40 O=C(NC[C@H](O)COCC1CC1)Nc1cc(F)c(F)c(F)c1F ZINC000880682239 EE On-Demand Anodyne ADRB1 18 40 COc1ccnc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)n1 ZINC000880682258 GE On-Demand Anodyne FAAH 24 44 COc1ccnc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)n1 ZINC000880682258 GE On-Demand Anodyne RBP4 20 42 CN(CCN1CCOCC1)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682282 EE On-Demand Anodyne CASR 53 39 COc1ccnc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)c1 ZINC000880682283 GG On-Demand Anodyne PDGFRB 44 39 COc1ccnc(N2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)c1 ZINC000880682283 GG On-Demand Anodyne RBP4 22 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCOC2(CCCC2)C1 ZINC000880682330 EG On-Demand Anodyne EPHX2 21 45 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682334 GG On-Demand Anodyne F2 43 38 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682334 GG On-Demand Anodyne P2RX7 15 41 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682334 GG On-Demand Anodyne LGMN 41 33 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682334 GG On-Demand Anodyne XIAP 16 51 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682335 GG On-Demand Anodyne F2 43 38 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682335 GG On-Demand Anodyne P2RX7 15 41 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682335 GG On-Demand Anodyne LGMN 41 33 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682335 GG On-Demand Anodyne XIAP 16 51 O=C(Nc1cc(F)c(F)c(F)c1F)N(CCO)CCN1CCOCC1 ZINC000880682338 FD On-Demand Anodyne CASR 64 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682361 FF On-Demand Anodyne PAPA1_CARPA 49 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682361 FF On-Demand Anodyne CTSK 20 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682361 FF On-Demand Anodyne CTSL 32 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682361 FF On-Demand Anodyne CTSS 17 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682361 FF On-Demand Anodyne FPR1 48 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682362 FF On-Demand Anodyne PAPA1_CARPA 49 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682362 FF On-Demand Anodyne CTSK 20 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682362 FF On-Demand Anodyne CTSL 32 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682362 FF On-Demand Anodyne CTSS 17 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccc(C)c(C)c1 ZINC000880682362 FF On-Demand Anodyne FPR1 48 40 CCn1cc(CNC(=O)c2sc(-c3ccc(C)cc3F)nc2C)nn1 ZINC000880682369 FG On-Demand Anodyne SCD1 29 46 CCn1cc(CNC(=O)c2sc(-c3ccc(C)cc3F)nc2C)nn1 ZINC000880682369 FG On-Demand Anodyne SCD 28 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880682370 FG On-Demand Anodyne EPHX2 17 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880682370 FG On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880682371 FG On-Demand Anodyne EPHX2 17 48 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880682371 FG On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@]2(CCOC2)C1 ZINC000880682480 DF On-Demand Anodyne EPHX2 30 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@]2(CCOC2)C1 ZINC000880682481 DF On-Demand Anodyne EPHX2 30 40 O=C(NCc1ccccc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880682502 GG On-Demand Anodyne KCNQ2 67 37 O=C(NCc1ccccc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880682502 GG On-Demand Anodyne SCN10A 16 49 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880682530 GH On-Demand Anodyne NAMPT 16 43 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCSCC1 ZINC000880682535 DG On-Demand Anodyne EPHX2 39 56 Cc1noc(C2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)n1 ZINC000880682538 FG On-Demand Anodyne SMO 40 46 Cc1noc(C2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)n1 ZINC000880682538 FG On-Demand Anodyne ETHR 62 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN2CCCC[C@@H]2C1 ZINC000880682560 EF On-Demand Anodyne L3MBTL3 66 39 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN2CCCC[C@H]2C1 ZINC000880682561 EF On-Demand Anodyne L3MBTL3 66 39 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](N2CCCCC2)C1 ZINC000880682575 EG On-Demand Anodyne L3MBTL3 92 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](N2CCCCC2)C1 ZINC000880682576 EG On-Demand Anodyne L3MBTL3 92 46 O=C(COC1CC1)N1CCN(c2ccc(Br)cc2)CC1 ZINC000880682606 EE On-Demand Anodyne MAPK1 16 42 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880682607 EF On-Demand Anodyne CCR3 42 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880682607 EF On-Demand Anodyne EPHX2 29 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(CC2CC2)C1 ZINC000880682608 EF On-Demand Anodyne CCR3 42 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(CC2CC2)C1 ZINC000880682608 EF On-Demand Anodyne EPHX2 29 43 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CCO)CC1 ZINC000880682610 ED On-Demand Anodyne CCR3 36 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CCO)CC1 ZINC000880682610 ED On-Demand Anodyne SLC6A5 16 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CCO)CC1 ZINC000880682610 ED On-Demand Anodyne EPHX2 43 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CCO)CC1 ZINC000880682610 ED On-Demand Anodyne CXCR3 19 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880682618 FG On-Demand Mild CCR3 19 42 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880682618 FG On-Demand Mild EPHX2 36 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880682618 FG On-Demand Mild CXCR3 15 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880682619 FG On-Demand Mild CCR3 19 42 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880682619 FG On-Demand Mild EPHX2 36 43 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880682619 FG On-Demand Mild CXCR3 15 40 C=CCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682647 EG On-Demand Mild EPHX2 40 47 CN1CCC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682656 DF On-Demand Anodyne CCR3 44 41 CN1CCC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682656 DF On-Demand Anodyne CACNA1I 52 33 CN1CCC(CNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682665 DF On-Demand Anodyne CACNA1I 62 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C2CCC2)CC1 ZINC000880682680 EF On-Demand Anodyne HRH3 23 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C2CCC2)CC1 ZINC000880682680 EF On-Demand Anodyne L3MBTL3 51 38 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H](C2CCCCC2)C1 ZINC000880682698 CH On-Demand Anodyne L3MBTL3 52 36 O=C(c1cnc2cc[nH]c2c1)N1CC[C@@H](C2CCCCC2)C1 ZINC000880682699 CH On-Demand Anodyne L3MBTL3 52 36 CCCCCN(CCO)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682722 DG On-Demand Anodyne SOAT1 28 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCOCC1 ZINC000880682736 CF On-Demand Anodyne EPHX2 35 55 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682753 GH On-Demand Anodyne CACNA1I 49 33 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682754 GH On-Demand Anodyne CACNA1I 49 33 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682756 FD On-Demand Anodyne EPHX2 35 48 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682762 FG On-Demand Anodyne CELA1 40 36 N#Cc1ccc(N2CCC(NC(=O)Nc3cc(F)c(F)c(F)c3F)CC2)nc1 ZINC000880682769 GG On-Demand Mild EPHX2 21 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN2CCC[C@@H]2C1 ZINC000880682804 DF On-Demand Anodyne L3MBTL3 45 37 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN2CCC[C@H]2C1 ZINC000880682805 DF On-Demand Anodyne L3MBTL3 45 37 CCCCNC(=O)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682813 GG On-Demand Anodyne ASAH1 49 35 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC(F)F)CC1 ZINC000880682836 FG On-Demand Anodyne EPHX2 48 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC(F)F)CC1 ZINC000880682836 FG On-Demand Anodyne CXCR3 19 42 C=C(C)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682839 EG On-Demand Mild EPHX2 37 45 C=C(C)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682839 EG On-Demand Mild CXCR3 20 42 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@@H](C4CCCCC4)C3)cc2)N1 ZINC000880682844 EH On-Demand Anodyne L3MBTL3 69 43 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@H](C4CCCCC4)C3)cc2)N1 ZINC000880682845 EH On-Demand Anodyne L3MBTL3 69 43 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H](C4CCCCC4)C3)cc2)N1 ZINC000880682846 EH On-Demand Anodyne L3MBTL3 69 43 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H](C4CCCCC4)C3)cc2)N1 ZINC000880682847 EH On-Demand Anodyne L3MBTL3 69 43 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682858 GD On-Demand Anodyne SLC6A1 105 35 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682858 GD On-Demand Anodyne CCR3 39 44 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682859 GD On-Demand Anodyne SLC6A1 105 35 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682859 GD On-Demand Anodyne CCR3 39 44 NC(=O)C1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682860 EE On-Demand Anodyne EPHX2 32 52 N#CCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682867 EE On-Demand Mild EPHX2 39 46 O=C(CNC(=O)Nc1cc(F)c(F)c(F)c1F)NC1CCCC1 ZINC000880682898 EE On-Demand Anodyne EPHX2 15 54 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682942 EF On-Demand Anodyne EPHX2 36 48 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682943 EF On-Demand Anodyne EPHX2 36 48 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682961 EF On-Demand Anodyne CCR3 15 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880682964 GG On-Demand Anodyne EPHX2 30 45 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880682964 GG On-Demand Anodyne CXCR3 17 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880682965 GG On-Demand Anodyne EPHX2 30 45 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880682965 GG On-Demand Anodyne CXCR3 17 40 C[C@@H](Cn1cncn1)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880682970 DE On-Demand Anodyne HIS3 82 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne HTR1F 56 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne PIM1 47 33 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne CCR2 26 54 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne RBP4 48 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne CALCRL 43 39 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880682974 GJ On-Demand Anodyne PIM3 48 33 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880682975 GE On-Demand Anodyne HTR2A 16 41 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880682975 GE On-Demand Anodyne MAPK10 15 46 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880682975 GE On-Demand Anodyne EPHX2 27 45 N#Cc1ccccc1N1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682976 GH On-Demand Mild KCNQ2 61 35 N#Cc1ccccc1N1CCCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880682976 GH On-Demand Mild RBP4 21 42 O=C(CNC(=O)Nc1cc(F)c(F)c(F)c1F)NC1CCCCC1 ZINC000880682995 EF On-Demand Anodyne EPHX2 20 55 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682997 GH On-Demand Anodyne ACACB 15 40 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682997 GH On-Demand Anodyne CACNA1I 59 36 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682998 GH On-Demand Anodyne ACACB 15 40 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880682998 GH On-Demand Anodyne CACNA1I 59 36 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@@H](N2CCCC2)C1 ZINC000880683008 EF On-Demand Anodyne L3MBTL3 94 47 O=C(Nc1cc(F)c(F)c(F)c1F)N1CC[C@H](N2CCCC2)C1 ZINC000880683009 EF On-Demand Anodyne L3MBTL3 94 47 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683015 GF On-Demand Anodyne STAT6 45 34 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683015 GF On-Demand Anodyne DGAT1 21 41 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683015 GF On-Demand Anodyne NAMPT 26 43 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683029 GH On-Demand Anodyne MLYCD 17 40 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683029 GH On-Demand Anodyne L3MBTL3 57 36 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880683031 FG On-Demand Mild CACNA1I 62 36 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cc(F)c(F)c(F)c1F ZINC000880683032 FG On-Demand Mild CACNA1I 62 36 CC(=O)NCC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683044 EF On-Demand Anodyne CACNA1I 53 32 CC(C)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683063 EG On-Demand Anodyne EPHX2 46 46 CC(C)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683063 EG On-Demand Anodyne CXCR3 21 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C2CCCC2)CC1 ZINC000880683064 EG On-Demand Anodyne HRH3 20 45 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C2CCCC2)CC1 ZINC000880683064 EG On-Demand Anodyne L3MBTL3 51 38 CN(C)C(=O)OCCNC(=O)c1cccc(N(C)C(=O)OC(C)(C)C)c1 ZINC000880683065 FE On-Demand Anodyne DRD4 41 31 CCCCN(CC)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683092 CH On-Demand Anodyne SOAT1 19 42 CN(C)C(=O)OCCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880683094 DD On-Demand Anodyne MPO 61 35 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC2CC2)CC1 ZINC000880683110 EG On-Demand Anodyne EPHX2 49 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(CC2CC2)CC1 ZINC000880683110 EG On-Demand Anodyne CXCR3 20 52 CN(C)C(=O)OCCNC(=O)c1cc2ccccc2cc1F ZINC000880683122 DE On-Demand Anodyne POLR1A 43 36 O=C(NCCCN1CCCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683131 EG On-Demand Anodyne CCR3 36 44 O=C(NCCCN1CCCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683131 EG On-Demand Anodyne CHRNA7 22 54 O=C(NCCCN1CCCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683131 EG On-Demand Anodyne HNMT 41 34 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880683137 GI On-Demand Anodyne RBP4 48 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880683138 GI On-Demand Anodyne RBP4 48 38 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683142 GH On-Demand Anodyne ASAH1 87 39 COc1ccccc1-c1ccc(C(=O)N[C@H]2COC3(CCC3)C2)c(O)n1 ZINC000880683152 FF On-Demand Anodyne HTR3A 17 45 COc1ccccc1-c1ccc(C(=O)N[C@@H]2COC3(CCC3)C2)c(O)n1 ZINC000880683153 FF On-Demand Anodyne HTR3A 17 45 COCCOc1ncccc1CNC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683154 FF On-Demand Anodyne P2RY1 34 42 COCCOc1ncccc1CNC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683154 FF On-Demand Anodyne SCN10A 15 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](N2CCCC2)C1 ZINC000880683166 EG On-Demand Anodyne L3MBTL3 69 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](N2CCCC2)C1 ZINC000880683167 EG On-Demand Anodyne L3MBTL3 69 40 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCC[C@H](O)C1 ZINC000880683169 DF On-Demand Anodyne EPHX2 21 54 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCC[C@@H](O)C1 ZINC000880683170 DF On-Demand Anodyne EPHX2 21 54 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCC[C@@H](O)C1 ZINC000880683171 DF On-Demand Anodyne EPHX2 21 54 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCC[C@H](O)C1 ZINC000880683172 DF On-Demand Anodyne EPHX2 21 54 CS(=O)(=O)N1CCN(CCNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683173 GC On-Demand Anodyne DRD4 40 31 CS(=O)(=O)N1CCN(CCNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683173 GC On-Demand Anodyne CCR3 30 40 O=C(c1ccccc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683183 GI On-Demand Anodyne SLC18A3 37 43 O=C(c1ccccc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683183 GI On-Demand Anodyne RBP4 56 39 O=C(NCc1ccccc1CN1CCCC1=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683184 GH On-Demand Anodyne P2RX7 41 38 COc1ccc2c(c1)CC[C@H](C(=O)NCCOC(=O)N(C)C)C2 ZINC000880683185 DD On-Demand Anodyne NQO2 37 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCOC(=O)N(C)C)C2 ZINC000880683185 DD On-Demand Anodyne MTNR1A 58 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCOC(=O)N(C)C)C2 ZINC000880683185 DD On-Demand Anodyne MTNR1B 51 41 CN1CCN(c2ncccc2CNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683215 GF On-Demand Anodyne TRPV1 39 42 CN1CCN(c2ncccc2CNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683215 GF On-Demand Anodyne P2RX7 35 41 CN1CCN(c2ncccc2CNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683215 GF On-Demand Anodyne SCN10A 19 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(C(=O)c2ccco2)CC1 ZINC000880683225 FF On-Demand Anodyne RBP4 19 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880683256 GG On-Demand Anodyne EPHX2 42 45 CNC(=O)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683263 FD On-Demand Anodyne EPHX2 42 46 CNC(=O)CN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683263 FD On-Demand Anodyne CXCR3 20 41 Cc1cc([C@@H]2CCCN2C(=O)Nc2cc(F)c(F)c(F)c2F)on1 ZINC000880683268 EH On-Demand Anodyne KCNA5 18 44 COc1cc2c(cc1OC)CN(C(=O)Nc1cc(F)c(F)c(F)c1F)CC2 ZINC000880683274 GH On-Demand Anodyne ABCB1 18 44 N#Cc1ccc(CN2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)cc1 ZINC000880683300 GG On-Demand Mild MLNR 28 41 N#Cc1ccc(CN2CCN(C(=O)Nc3cc(F)c(F)c(F)c3F)CC2)cc1 ZINC000880683300 GG On-Demand Mild FAAH 21 46 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880683301 FF On-Demand Anodyne EPHX2 54 55 O=C(NC[C@H](O)CN1CCc2ccccc2C1)Nc1cc(F)c(F)c(F)c1F ZINC000880683308 GF On-Demand Anodyne NOD2 41 35 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880683310 GH On-Demand Anodyne EPHX2 58 52 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880683310 GH On-Demand Anodyne SFRP1 35 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880683310 GH On-Demand Anodyne L3MBTL3 65 36 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683318 GI On-Demand Anodyne NPY5R 19 44 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683318 GI On-Demand Anodyne EPHX2 45 44 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683318 GI On-Demand Anodyne RBP4 56 39 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(Cc2ccncc2)CC1 ZINC000880683319 FF On-Demand Anodyne FAAH 33 49 O=C1CC[C@H]2CN(C(=O)c3cncc4[nH]ccc34)CC[C@@H]2N1 ZINC000880683322 CD On-Demand Anodyne HPGDS 17 46 O=C(CCNC(=O)Nc1cc(F)c(F)c(F)c1F)NC1CCCCC1 ZINC000880683324 FG On-Demand Anodyne EPHX2 20 54 O=C1CC[C@H]2CN(C(=O)c3cncc4[nH]ccc34)CC[C@H]2N1 ZINC000880683327 CD On-Demand Anodyne HPGDS 17 46 O=C1CC[C@@H]2CN(C(=O)c3cncc4[nH]ccc34)CC[C@@H]2N1 ZINC000880683329 CD On-Demand Anodyne HPGDS 17 46 O=C1CC[C@@H]2CN(C(=O)c3cncc4[nH]ccc34)CC[C@H]2N1 ZINC000880683331 CD On-Demand Anodyne HPGDS 17 46 O=C(NCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683334 CG On-Demand Anodyne CCR3 41 41 O=C(NCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683334 CG On-Demand Anodyne EPHX2 27 51 O=C(NCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683334 CG On-Demand Anodyne CACNA1I 60 36 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCCC1 ZINC000880683336 CH On-Demand Anodyne EPHX2 59 53 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCCC1 ZINC000880683336 CH On-Demand Anodyne CXCR3 17 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](O)C1 ZINC000880683339 CF On-Demand Anodyne EPHX2 26 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](O)C1 ZINC000880683341 CF On-Demand Anodyne EPHX2 26 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(O)(CO)CC1 ZINC000880683342 GD On-Demand Anodyne PREP 67 52 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(O)(CO)CC1 ZINC000880683342 GD On-Demand Anodyne SLC12A5 68 37 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC(O)(CO)CC1 ZINC000880683342 GD On-Demand Anodyne Q9NAW4_PLAFA 26 41 C[C@@H]1CCCN(C(=O)C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)C1 ZINC000880683344 GI On-Demand Anodyne EPHX2 24 51 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683351 GH On-Demand Anodyne EPHX2 50 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCCCC1 ZINC000880683353 CI On-Demand Anodyne CACNA1H 38 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCCCC1 ZINC000880683353 CI On-Demand Anodyne EPHX2 27 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880683366 GJ On-Demand Anodyne CACNA1H 43 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880683366 GJ On-Demand Anodyne NPY2R 73 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880683369 GJ On-Demand Anodyne CACNA1H 43 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880683369 GJ On-Demand Anodyne NPY2R 73 38 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683377 FH On-Demand Anodyne NPY2R 52 38 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683377 FH On-Demand Anodyne EPHX2 25 47 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1COC3(CCC3)C1)C2 ZINC000880683383 DF On-Demand Anodyne MTNR1A 25 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1COC3(CCC3)C1)C2 ZINC000880683383 DF On-Demand Anodyne MTNR1B 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1COC3(CCC3)C1)C2 ZINC000880683385 DF On-Demand Anodyne MTNR1A 25 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1COC3(CCC3)C1)C2 ZINC000880683385 DF On-Demand Anodyne MTNR1B 22 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880683394 GG On-Demand Anodyne EPHX2 49 48 O=C(N[C@H]1COC2(CCC2)C1)c1cc(C(F)(F)F)ccn1 ZINC000880683403 DF On-Demand Anodyne CCR2 15 40 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683411 FF On-Demand Anodyne EPHX2 60 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CO)C1 ZINC000880683416 DF On-Demand Anodyne CCR3 25 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CO)C1 ZINC000880683416 DF On-Demand Anodyne EPHX2 21 58 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(OCc2ccccc2)CC1 ZINC000880683417 GI On-Demand Anodyne GRIN2B 40 46 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(OCc2ccccc2)CC1 ZINC000880683417 GI On-Demand Anodyne RBP4 56 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CO)C1 ZINC000880683418 DF On-Demand Anodyne CCR3 25 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CO)C1 ZINC000880683418 DF On-Demand Anodyne EPHX2 21 58 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683424 GG On-Demand Anodyne MTOR 54 38 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683424 GG On-Demand Anodyne PIK3CB 29 42 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683424 GG On-Demand Anodyne STAT6 59 38 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683424 GG On-Demand Anodyne DGAT1 31 46 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683424 GG On-Demand Anodyne NAMPT 53 43 O=C(CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)N1CCCC1 ZINC000880683431 GF On-Demand Anodyne MAPK1 22 42 O=C(NCCNC(=O)C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683439 DE On-Demand Anodyne CCR3 25 41 CC(C)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683442 EH On-Demand Anodyne CACNA1H 42 45 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880683447 CG On-Demand Anodyne EPHX2 28 42 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880683456 CG On-Demand Anodyne EPHX2 28 42 CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683458 DG On-Demand Anodyne NPY2R 40 36 CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683458 DG On-Demand Anodyne CCR3 59 42 CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683458 DG On-Demand Anodyne EPHX2 63 52 CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683458 DG On-Demand Anodyne CXCR3 26 49 CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683458 DG On-Demand Anodyne MCHR1 39 40 O=C(Nc1ccc(F)c(C(F)F)c1)N(C[C@@H]1CCOC1)C1CC1 ZINC000880683460 EH On-Demand Anodyne MCHR1 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)N(C[C@H]1CCOC1)C1CC1 ZINC000880683461 EH On-Demand Anodyne MCHR1 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880683476 GH On-Demand Anodyne EPHX2 56 43 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)c1ccccc1 ZINC000880683487 GI On-Demand Anodyne DRD4 22 43 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)c1ccccc1 ZINC000880683487 GI On-Demand Anodyne EPHX2 59 39 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)c1ccccc1 ZINC000880683487 GI On-Demand Anodyne MCHR1 26 47 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)c1ccccc1 ZINC000880683487 GI On-Demand Anodyne KCNK3 43 36 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)C1CC1 ZINC000880683490 FG On-Demand Anodyne EPHX2 54 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccncc2)CC1 ZINC000880683496 FH On-Demand Anodyne CACNA1H 42 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccncc2)CC1 ZINC000880683496 FH On-Demand Anodyne NPY2R 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccncc2)CC1 ZINC000880683496 FH On-Demand Anodyne PRNP 45 38 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2nc3ccccc3[nH]2)CC1 ZINC000880683518 GJ On-Demand Anodyne SMO 31 41 C[C@@H]1C[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683521 CH On-Demand Anodyne EPHX2 16 42 C[C@@H]1C[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683521 CH On-Demand Anodyne PRMT3 52 32 C[C@@H]1C[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683525 CH On-Demand Anodyne EPHX2 16 42 C[C@@H]1C[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683525 CH On-Demand Anodyne PRMT3 52 32 C[C@H]1C[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683527 CH On-Demand Anodyne EPHX2 16 42 C[C@H]1C[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683527 CH On-Demand Anodyne PRMT3 52 32 O=C(NCC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683529 CH On-Demand Anodyne CCR3 47 39 O=C(NCC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683529 CH On-Demand Anodyne EPHX2 24 55 O=C(NCC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683529 CH On-Demand Anodyne CACNA1I 49 33 O=C(NCC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683529 CH On-Demand Anodyne PRMT3 41 38 O=C(c1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683531 GJ On-Demand Anodyne CACNA1H 46 39 O=C(c1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683531 GJ On-Demand Anodyne NPY2R 44 35 O=C(c1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683531 GJ On-Demand Anodyne SLC18A3 32 41 O=C(c1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683531 GJ On-Demand Anodyne EPHX2 33 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne DRD4 26 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne KCNH2 15 41 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne SIGMAR1 26 48 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne SSTR5 52 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne CCR3 57 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne EPHX2 44 45 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne CXCR3 32 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880683546 GG On-Demand Anodyne MCHR1 55 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccc(O)cc2)CC1 ZINC000880683557 FH On-Demand Anodyne MAPK1 21 42 O=C(N[C@H]1COC2(CCC2)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880683558 EG On-Demand Anodyne EZH2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1c1ccccc1 ZINC000880683573 EK On-Demand Anodyne NPY2R 47 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1c1ccccc1 ZINC000880683580 EK On-Demand Anodyne NPY2R 47 35 CN1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683582 CE On-Demand Anodyne HRH4 22 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2cccc(O)c2)CC1 ZINC000880683593 FH On-Demand Anodyne CACNA1H 50 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2cccc(O)c2)CC1 ZINC000880683593 FH On-Demand Anodyne MAPK1 18 43 O=C(NCc1nnc2n1CCCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880683602 FG On-Demand Anodyne F2R 49 30 O=C(NCc1nnc2n1CCCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880683602 FG On-Demand Anodyne PRMT3 56 38 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne DRD4 21 58 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne SIGMAR1 18 46 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne SSTR5 45 39 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne CCR3 41 44 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne EPHX2 39 46 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne CXCR3 22 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880683612 GG On-Demand Anodyne MCHR1 32 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccn2)CC1 ZINC000880683622 FE On-Demand Anodyne FAAH 24 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ncccn2)CC1 ZINC000880683622 FE On-Demand Anodyne RBP4 25 42 CN1CCC[C@H](NC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880683626 DE On-Demand Anodyne EPHX2 30 51 O=C(NCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880683638 CE On-Demand Anodyne CCR3 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2cnccn2)CC1 ZINC000880683639 FF On-Demand Anodyne PDGFRB 38 40 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCN(C2CC2)CC1 ZINC000880683643 EF On-Demand Anodyne EPHX2 47 51 CC(C)(C)N1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683645 EH On-Demand Anodyne EPHX2 51 49 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683649 GI On-Demand Clean NPY2R 41 33 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683649 GI On-Demand Clean EPHB4 57 33 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683649 GI On-Demand Clean STAT6 63 38 CC[C@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683665 CH On-Demand Anodyne EPHX2 16 43 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683672 GG On-Demand Mild P2RY12 17 46 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683672 GG On-Demand Mild PDGFRB 52 42 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683672 GG On-Demand Mild TRPV1 19 66 CCOCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683676 CG On-Demand Anodyne HRH2 15 40 CCOCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683676 CG On-Demand Anodyne CCR3 26 42 CCOCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683676 CG On-Demand Anodyne EPHX2 17 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(Cc2cccnc2)CC1 ZINC000880683677 FF On-Demand Anodyne FAAH 36 52 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C2CC2)CC1 ZINC000880683680 EH On-Demand Anodyne EPHX2 55 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C2CC2)CC1 ZINC000880683680 EH On-Demand Anodyne CXCR3 21 44 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(N2CCCCC2)CC1 ZINC000880683681 FH On-Demand Anodyne L3MBTL3 109 50 CCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683696 DF On-Demand Anodyne CCR3 27 41 CCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683696 DF On-Demand Anodyne EPHX2 54 49 CCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683696 DF On-Demand Anodyne CXCR3 21 43 O=C(NCCCN1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683699 EE On-Demand Anodyne CCR3 30 42 O=C(NCCCN1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683699 EE On-Demand Anodyne CHRNA7 15 45 O=C(NCCCN1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683699 EE On-Demand Anodyne EPHX2 29 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(=O)N2CCCCC2)CC1 ZINC000880683702 GI On-Demand Anodyne EPHX2 38 45 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683705 EF On-Demand Anodyne PLD1 47 36 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683705 EF On-Demand Anodyne EPHX2 33 46 CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683722 CH On-Demand Anodyne CCR3 27 41 CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683722 CH On-Demand Anodyne EPHX2 16 52 CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683722 CH On-Demand Anodyne LEF 19 46 CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683722 CH On-Demand Anodyne ASAH1 56 32 C[C@H](CN1CCOCC1)NC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683731 EE On-Demand Anodyne PLD1 41 34 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne PIK3CA 36 41 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne PIK3CD 16 42 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne MTOR 70 40 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne PIK3CB 32 42 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne STAT6 53 36 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne NAMPT 43 40 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683743 GG On-Demand Anodyne SMG1 28 41 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683745 FH On-Demand Anodyne EPHX2 72 53 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683745 FH On-Demand Anodyne CXCR3 21 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880683748 FH On-Demand Anodyne EPHX2 40 43 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H]3NC(=O)CC[C@@H]3C2)N1Cc1ccccc1 ZINC000880683750 GC On-Demand Anodyne TRHR 26 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H]3NC(=O)CC[C@H]3C2)N1Cc1ccccc1 ZINC000880683752 GC On-Demand Anodyne TRHR 26 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H]3NC(=O)CC[C@H]3C2)N1Cc1ccccc1 ZINC000880683754 GC On-Demand Anodyne TRHR 26 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H]3NC(=O)CC[C@@H]3C2)N1Cc1ccccc1 ZINC000880683757 GC On-Demand Anodyne TRHR 26 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H](c2nc3ccccc3o2)C1 ZINC000880683775 GJ On-Demand Anodyne RBP4 44 32 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H](c2nc3ccccc3o2)C1 ZINC000880683777 GJ On-Demand Anodyne RBP4 44 32 CN(C)C(=O)OCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880683791 DE On-Demand Anodyne NQO2 21 45 CN(C)C(=O)OCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880683791 DE On-Demand Anodyne MTNR1A 21 40 CN(C)C(=O)OCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880683791 DE On-Demand Anodyne MTNR1B 21 40 CN(C)C(=O)OCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880683792 DE On-Demand Anodyne NQO2 21 45 CN(C)C(=O)OCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880683792 DE On-Demand Anodyne MTNR1A 21 40 CN(C)C(=O)OCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880683792 DE On-Demand Anodyne MTNR1B 21 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683801 GE On-Demand Anodyne CCR8 84 41 CCN1CC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880683818 DF On-Demand Anodyne CCR3 50 39 CCN1CC[C@H](CNC(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880683818 DF On-Demand Anodyne CACNA1I 63 35 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC(c2nnc3ccccn23)CC1 ZINC000880683825 GH On-Demand Anodyne RBP4 48 39 NC(=O)C1CCN(CCCCNC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880683828 GE On-Demand Anodyne CCR3 41 44 CN(C)C(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683836 EG On-Demand Anodyne CACNA1H 33 40 Cc1nc(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)cs1 ZINC000880683841 EH On-Demand Anodyne PRMT3 45 34 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683844 GF On-Demand Anodyne TRPV1 32 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683844 GF On-Demand Anodyne MTOR 41 38 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683844 GF On-Demand Anodyne SCN10A 23 51 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683844 GF On-Demand Anodyne STAT6 54 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccco2)CC1 ZINC000880683845 FH On-Demand Anodyne FAAH 15 45 O=C(NCCCCn1ccnc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683846 EG On-Demand Anodyne TBXAS1 45 49 O=C(NCCCCn1ccnc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683846 EG On-Demand Anodyne HMOX2 46 33 O=C(NCCCCn1ccnc1)Nc1cc(F)c(F)c(F)c1F ZINC000880683846 EG On-Demand Anodyne QPCT 38 52 CC(=O)NCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683847 DE On-Demand Anodyne CCR3 27 40 O=C(NCc1ccc(N2CCCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683855 FI On-Demand Anodyne F2R 49 31 O=C(NCc1ccc(N2CCCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683855 FI On-Demand Anodyne PRMT3 54 36 O=C(NCc1ccc(N2CCCC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683855 FI On-Demand Anodyne NAMPT 54 42 O=C(NCCCN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683857 EF On-Demand Anodyne CCR3 39 43 O=C(NCCCN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683857 EF On-Demand Anodyne EPHX2 20 42 O=C(NCCCN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880683857 EF On-Demand Anodyne TYRO3 21 41 CCOC(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683863 FH On-Demand Anodyne CCR3 20 40 CCOC(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683863 FH On-Demand Anodyne EPHX2 27 41 CCOC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683866 EH On-Demand Anodyne CACNA1H 42 38 CCOC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683866 EH On-Demand Anodyne FDFT1 15 43 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880683869 FG On-Demand Anodyne PANC 42 34 O=C(C(=O)N1CCC(O)(CO)CC1)c1c[nH]c2cc(F)ccc12 ZINC000880683870 DC On-Demand Anodyne MPO 51 34 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccc(F)c(C(F)F)c2)c1 ZINC000880683882 GH On-Demand Anodyne MTNR1A 19 43 O=C(NC[C@@H](O)C(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880683899 DF On-Demand Anodyne PRMT3 63 37 O=C(NC[C@H](O)C(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880683900 DF On-Demand Anodyne PRMT3 63 37 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683902 GJ On-Demand Anodyne CACNA1H 43 37 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683902 GJ On-Demand Anodyne TRPV1 17 40 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683902 GJ On-Demand Anodyne NPY5R 15 44 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683902 GJ On-Demand Anodyne EPHX2 54 42 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CC1 ZINC000880683903 BF On-Demand Anodyne EPHX2 54 62 O=C(NCc1ccnc(N2CCCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683906 FI On-Demand Anodyne F2R 50 32 O=C(NCc1ccnc(N2CCCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880683906 FI On-Demand Anodyne NAMPT 42 41 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1cc(F)c(F)c(F)c1F ZINC000880683910 FG On-Demand Anodyne PANC 42 34 CN(C)C(=O)OCCNC(=O)c1ccc(OC(F)F)c(Br)c1 ZINC000880683916 GE On-Demand Anodyne NCEH1 42 36 CC(C)(C)C(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683923 FG On-Demand Anodyne CACNA1H 50 40 CC(C)(C)C(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880683923 FG On-Demand Anodyne EPHX2 26 45 O=C(N[C@H]1COC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880683925 DE On-Demand Anodyne GABRA1 15 40 O=C(N[C@H]1COC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880683925 DE On-Demand Anodyne GABRA2 15 40 O=C(N[C@@H]1COC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880683927 DE On-Demand Anodyne GABRA1 15 40 O=C(N[C@@H]1COC2(CCC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880683927 DE On-Demand Anodyne GABRA2 15 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@@H]1c1cccnc1 ZINC000880683935 EI On-Demand Anodyne CHRNA7 17 48 Cc1nc(CN2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cs1 ZINC000880683936 GH On-Demand Anodyne FAAH 17 42 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCC[C@H]1c1cccnc1 ZINC000880683937 EI On-Demand Anodyne CHRNA7 17 48 O=C(NCCN1CCCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683939 DF On-Demand Anodyne DRD4 40 30 O=C(NCCN1CCCCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880683939 DF On-Demand Anodyne CHRNA7 17 47 CN(C)C(=O)OCCNC(=O)c1coc(-c2ccccn2)n1 ZINC000880683954 DD On-Demand Anodyne TBXA2R 15 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880683963 GH On-Demand Anodyne NPY2R 20 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880683963 GH On-Demand Anodyne EPHX2 20 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880683994 GH On-Demand Clean STAT6 44 34 O=C(NCC(F)(F)F)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684000 GH On-Demand Anodyne EPHX2 52 40 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne ADRA1D 19 41 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne HTR2A 22 41 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne ADRA1B 22 41 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne DRD3 15 41 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne CCR3 71 52 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne CHRNA7 22 51 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne F2R 41 32 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne EPHX2 33 43 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684004 GF On-Demand Anodyne MCHR1 39 43 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCC2(CC1)OCCO2 ZINC000880684017 EG On-Demand Anodyne EPHX2 19 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880684022 EJ On-Demand Anodyne EPHX2 30 45 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cc(F)c(F)c(F)c1F ZINC000880684023 GG On-Demand Clean STAT6 58 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](C(F)(F)F)C1 ZINC000880684026 EJ On-Demand Anodyne EPHX2 30 45 COCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880684044 EE On-Demand Anodyne HTR4 44 40 COCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880684044 EE On-Demand Anodyne CCR3 37 45 COCCN1CCC(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC1 ZINC000880684044 EE On-Demand Anodyne EPHX2 49 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880684069 GH On-Demand Anodyne NPY2R 25 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880684069 GH On-Demand Anodyne EPHX2 24 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880684069 GH On-Demand Anodyne L3MBTL3 47 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880684071 GH On-Demand Anodyne CACNA1H 55 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880684071 GH On-Demand Anodyne NPY2R 27 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880684071 GH On-Demand Anodyne EPHX2 24 47 CNC(=O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684093 CD On-Demand Anodyne F7 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880684096 GJ On-Demand Anodyne GRIN2B 49 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880684096 GJ On-Demand Anodyne TIMP3 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880684096 GJ On-Demand Anodyne EPHX2 51 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880684096 GJ On-Demand Anodyne SCD1 17 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2cccnc2)CC1 ZINC000880684097 FH On-Demand Anodyne CHRNA7 46 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2cccnc2)CC1 ZINC000880684097 FH On-Demand Anodyne FAAH 37 56 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)N1CCOCC1 ZINC000880684098 EF On-Demand Anodyne EPHX2 28 44 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880684104 DH On-Demand Anodyne RBP4 48 34 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cc(F)c(F)c(F)c2F)C1 ZINC000880684105 DH On-Demand Anodyne RBP4 48 34 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880684112 EF On-Demand Anodyne EPHX2 21 46 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880684113 EF On-Demand Anodyne EPHX2 21 46 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880684114 EF On-Demand Anodyne EPHX2 21 46 O=C(Nc1cc(F)c(F)c(F)c1F)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880684115 EF On-Demand Anodyne EPHX2 21 46 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684135 EH On-Demand Anodyne FDFT1 21 44 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684135 EH On-Demand Anodyne EPHX2 25 41 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne TRPV1 28 44 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne PIK3CA 47 43 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne PIK3CD 18 43 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne MTOR 75 43 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne EPHX2 29 41 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne PIK3CG 33 43 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne SCN10A 27 51 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne PIK3CB 29 40 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne STAT6 61 38 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684140 GG On-Demand Anodyne NAMPT 47 42 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684141 GI On-Demand Anodyne F2R 53 32 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684141 GI On-Demand Anodyne EPHX2 31 44 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684141 GI On-Demand Anodyne L3MBTL3 68 38 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684141 GI On-Demand Anodyne NAMPT 31 53 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CC1 ZINC000880684160 CF On-Demand Anodyne MCHR1 38 43 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684161 EG On-Demand Anodyne CACNA1H 42 39 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684161 EG On-Demand Anodyne P2RY12 56 45 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684161 EG On-Demand Anodyne NPY2R 43 34 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684161 EG On-Demand Anodyne TGM2 20 42 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684161 EG On-Demand Anodyne F13A1 37 42 CCCCNC(=O)Nc1cc(F)c(F)c(F)c1F ZINC000880684166 CG On-Demand Anodyne ASAH1 60 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880684168 GH On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880684168 GH On-Demand Anodyne NPY2R 56 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880684168 GH On-Demand Anodyne FAAH 17 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880684168 GH On-Demand Anodyne EPHX2 33 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880684168 GH On-Demand Anodyne L3MBTL3 43 34 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne EGFR 15 43 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne HTR2A 22 41 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne CCR3 50 48 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne CHRNA7 24 52 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne EPHX2 44 56 O=C(NCCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684170 EF On-Demand Anodyne MCHR1 25 46 O=C(Nc1cc(F)c(F)c(F)c1F)NC1CCCC1 ZINC000880684174 CG On-Demand Anodyne EPHX2 51 71 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684181 GF On-Demand Anodyne CACNA1H 40 38 CS(=O)(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684193 FD On-Demand Anodyne NPY5R 17 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(CC(F)(F)F)CC1 ZINC000880684195 FH On-Demand Anodyne EPHX2 23 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCCC2)CC1 ZINC000880684206 EH On-Demand Anodyne HRH3 22 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCCC2)CC1 ZINC000880684206 EH On-Demand Anodyne EPHX2 23 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCCC2)CC1 ZINC000880684206 EH On-Demand Anodyne L3MBTL3 63 34 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684208 DE On-Demand Anodyne EPHX2 41 39 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684208 DE On-Demand Anodyne PRMT3 47 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)C2CC2)CC1 ZINC000880684217 EF On-Demand Anodyne CACNA1H 45 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)C2CC2)CC1 ZINC000880684217 EF On-Demand Anodyne EPHX2 38 41 O=C(NCCCN1C(=O)NC2(CCCC2)C1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684218 GG On-Demand Anodyne CCR3 36 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccccn2)CC1 ZINC000880684221 FF On-Demand Anodyne DRD4 24 41 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccccn2)CC1 ZINC000880684221 FF On-Demand Anodyne PDGFRB 27 40 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccccn2)CC1 ZINC000880684221 FF On-Demand Anodyne FAAH 23 43 O=C(Nc1cc(F)c(F)c(F)c1F)N1CCN(c2ccccn2)CC1 ZINC000880684221 FF On-Demand Anodyne RBP4 32 41 O=C(CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)NC1CC1 ZINC000880684226 FE On-Demand Anodyne CCR2 21 43 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684232 CF On-Demand Anodyne CACNA1H 37 42 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684232 CF On-Demand Anodyne HTR1D 18 52 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684232 CF On-Demand Anodyne HTR1B 21 52 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684232 CF On-Demand Anodyne HRH4 23 42 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684232 CF On-Demand Anodyne EPHX2 27 47 CCOC(=O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684269 DG On-Demand Anodyne EPHX2 18 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccn2)CC1 ZINC000880684279 FF On-Demand Anodyne CACNA1H 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccn2)CC1 ZINC000880684279 FF On-Demand Anodyne PDGFRB 53 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccn2)CC1 ZINC000880684279 FF On-Demand Anodyne TRPV1 17 56 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccn2)CC1 ZINC000880684279 FF On-Demand Anodyne NPY2R 60 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccn2)CC1 ZINC000880684279 FF On-Demand Anodyne FAAH 24 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880684283 FK On-Demand Anodyne PRCP 57 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880684284 FK On-Demand Anodyne PRCP 57 42 O=C(NCCc1nnc2n1CCCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880684290 FG On-Demand Anodyne PRMT3 42 38 CC(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684296 EI On-Demand Anodyne CCR3 53 41 CC(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684296 EI On-Demand Anodyne EPHX2 61 50 CC(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684296 EI On-Demand Anodyne CXCR3 26 50 CC(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684296 EI On-Demand Anodyne MCHR1 45 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccncc2)CC1 ZINC000880684297 FH On-Demand Anodyne FAAH 33 55 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccncc2)CC1 ZINC000880684297 FH On-Demand Anodyne MCHR1 20 42 O=C(NC[C@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684309 CG On-Demand Anodyne TNK2 27 41 CN(C[C@@H]1COCCO1)C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880684312 EE On-Demand Anodyne PDE4D 16 41 CCN(Cc1cccs1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684313 EJ On-Demand Anodyne NPY2R 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1c1cccnc1 ZINC000880684314 EJ On-Demand Anodyne CHRNA7 26 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1c1cccnc1 ZINC000880684315 EJ On-Demand Anodyne CHRNA7 26 43 O=C(NCCN1CCOCC1)Nc1cc(F)c(F)c(F)c1F ZINC000880684318 DD On-Demand Anodyne EPHX2 28 50 CCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684319 FH On-Demand Anodyne EPHX2 37 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne GRIN2B 15 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne NPY2R 45 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne CCR3 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne EPHX2 74 52 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880684320 GI On-Demand Anodyne L3MBTL3 74 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880684321 GI On-Demand Anodyne NPY2R 48 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880684321 GI On-Demand Anodyne EPHX2 32 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880684321 GI On-Demand Anodyne L3MBTL3 48 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccco2)CC1 ZINC000880684323 FG On-Demand Anodyne EPHX2 18 48 O=C(NCC(=O)N1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684332 EF On-Demand Anodyne EPHX2 30 42 O=C(NCC(=O)N1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684332 EF On-Demand Anodyne PRMT3 53 56 O=C(NCC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684339 DG On-Demand Anodyne EPHX2 27 47 O=C(NCC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684339 DG On-Demand Anodyne CACNA1I 44 32 COC(=O)CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684340 EH On-Demand Anodyne CCR3 15 43 COC(=O)CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684340 EH On-Demand Anodyne EPHX2 18 45 COC(=O)CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684340 EH On-Demand Anodyne LEF 18 44 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880684347 GF On-Demand Anodyne STAT6 42 32 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880684347 GF On-Demand Anodyne DGAT1 30 47 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)CN1CCCC1 ZINC000880684362 EH On-Demand Anodyne CCR3 35 40 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)CN1CCCC1 ZINC000880684362 EH On-Demand Anodyne EPHX2 18 44 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)CN1CCCC1 ZINC000880684362 EH On-Demand Anodyne MCHR1 22 46 CS(=O)(=O)N[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684370 FE On-Demand Anodyne EPHX2 17 49 CS(=O)(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684371 FE On-Demand Anodyne EPHX2 17 49 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684378 FH On-Demand Anodyne CCR3 19 41 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684378 FH On-Demand Anodyne EPHX2 21 41 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684378 FH On-Demand Anodyne CACNA1I 59 35 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684379 FH On-Demand Anodyne CCR3 19 41 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684379 FH On-Demand Anodyne EPHX2 21 41 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684379 FH On-Demand Anodyne CACNA1I 59 35 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC(C)(C)O1 ZINC000880684380 DH On-Demand Anodyne CACNA1H 29 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC(C)(C)O1 ZINC000880684381 DH On-Demand Anodyne CACNA1H 29 41 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne DRD4 19 42 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne HTR2A 29 41 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne CCR3 69 41 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne EPHX2 69 54 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne CXCR3 24 46 COCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684389 EF On-Demand Anodyne MCHR1 52 41 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684390 EG On-Demand Anodyne MTOR 23 42 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684390 EG On-Demand Anodyne EPHX2 72 50 COC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684390 EG On-Demand Anodyne CXCR3 20 44 Cc1noc(C)c1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684410 DH On-Demand Anodyne P2RX7 18 48 Cc1noc(C)c1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684410 DH On-Demand Anodyne NPY2R 17 42 O=C(NCCS(=O)(=O)N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684421 GD On-Demand Anodyne EPHX2 28 45 O=C(NCCS(=O)(=O)N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684421 GD On-Demand Anodyne NAMPT 15 40 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684433 GI On-Demand Anodyne F2R 51 33 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684433 GI On-Demand Anodyne NAMPT 31 46 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684434 FH On-Demand Anodyne EPHX2 68 50 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684434 FH On-Demand Anodyne CXCR3 21 55 CCNC(=O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684441 CE On-Demand Anodyne F7 24 41 N#Cc1ccnc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880684450 GG On-Demand Mild PDGFRB 30 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)N2CCCC2)CC1 ZINC000880684454 FG On-Demand Anodyne EPHX2 22 44 O=C(NCc1ccccc1CN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684455 GI On-Demand Anodyne F2R 50 31 O=C(Nc1ccc(F)c(C(F)F)c1)N(Cc1ccccn1)C1CC1 ZINC000880684458 EI On-Demand Anodyne GRM4 29 42 O=C(NCCCn1cccn1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684460 DG On-Demand Anodyne QPCT 20 42 COCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684469 CF On-Demand Anodyne CCR3 20 41 COCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684469 CF On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880684470 FG On-Demand Anodyne EPHX2 69 63 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880684470 FG On-Demand Anodyne CXCR3 19 42 CN1CCN(C(C)(C)CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684471 FF On-Demand Anodyne EPHX2 22 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC1 ZINC000880684485 CF On-Demand Anodyne CACNA1H 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC1 ZINC000880684485 CF On-Demand Anodyne ITGAL 40 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC1 ZINC000880684485 CF On-Demand Anodyne EPHX2 42 51 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne HTR2A 23 42 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne CCR3 43 43 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne CHRNA7 17 47 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne EPHX2 39 64 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne PLD2 56 32 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne MCHR1 20 41 O=C(NCCN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684493 DE On-Demand Anodyne STAT6 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne CACNA1H 55 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne PDGFRB 34 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne TRPV1 15 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne NPY2R 97 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne PRNP 47 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880684495 EI On-Demand Anodyne FAAH 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCO2 ZINC000880684501 EG On-Demand Anodyne CACNA1H 45 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCO2 ZINC000880684501 EG On-Demand Anodyne EPHX2 37 42 C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684503 CI On-Demand Anodyne EPHX2 28 56 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2O)CC1 ZINC000880684505 FH On-Demand Anodyne HTR1B 17 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2O)CC1 ZINC000880684505 FH On-Demand Anodyne PDGFRB 27 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2O)CC1 ZINC000880684505 FH On-Demand Anodyne KCNQ2 45 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccc2O)CC1 ZINC000880684505 FH On-Demand Anodyne NPY2R 104 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)CC1 ZINC000880684511 CF On-Demand Anodyne CACNA1H 40 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)CC1 ZINC000880684511 CF On-Demand Anodyne EPHX2 35 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)CC1 ZINC000880684511 CF On-Demand Anodyne SCD1 16 42 O=C(NCCCOC[C@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684526 EG On-Demand Anodyne CCR3 28 41 O=C(NCCCOC[C@@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684527 EG On-Demand Anodyne CCR3 28 41 O=C1CC[C@@H]2CN(C(=O)c3cc4cccc(C(F)(F)F)c4nc3O)CC[C@H]2N1 ZINC000880684530 GF On-Demand Anodyne RBP4 60 34 O=C1CC[C@H]2CN(C(=O)c3cc4cccc(C(F)(F)F)c4nc3O)CC[C@@H]2N1 ZINC000880684531 GF On-Demand Anodyne RBP4 60 34 Cc1noc(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880684547 FH On-Demand Anodyne SCD1 15 43 Cc1noc(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880684547 FH On-Demand Anodyne SMO 42 50 Cc1noc(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880684547 FH On-Demand Anodyne ETHR 55 36 O=C(NCCN1CCCS1(=O)=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684551 FD On-Demand Anodyne CCR3 19 41 O=C(NCc1nnc2n1CCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880684552 EG On-Demand Anodyne F2R 49 30 O=C(NCc1nnc2n1CCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880684552 EG On-Demand Anodyne PRMT3 54 36 O=C(NCc1ccc(CN2CCCC2=O)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684556 GI On-Demand Anodyne F2R 54 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCOCC1 ZINC000880684568 CG On-Demand Anodyne EPHX2 36 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CC2)CC1 ZINC000880684570 EG On-Demand Anodyne CACNA1H 41 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CC2)CC1 ZINC000880684570 EG On-Demand Anodyne CCR3 35 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CC2)CC1 ZINC000880684570 EG On-Demand Anodyne CCR2 18 56 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CC2)CC1 ZINC000880684570 EG On-Demand Anodyne MCHR1 20 40 O=C(NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)C1CCCCC1 ZINC000880684593 GI On-Demand Anodyne EPHX2 58 47 O=C(NCCC(=O)N1CCCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684599 FH On-Demand Anodyne EPHX2 25 42 O=C(NCCC(=O)N1CCCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684599 FH On-Demand Anodyne PRMT3 34 46 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880684601 GI On-Demand Anodyne P2RY14 46 33 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne DRD4 15 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne SIGMAR1 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne NPY1R 31 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne CCR3 50 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne F2R 40 30 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne CCKBR 44 37 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880684606 GH On-Demand Anodyne MCHR1 21 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne DRD4 15 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne SIGMAR1 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne NPY1R 31 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne CCR3 50 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne F2R 40 30 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne CCKBR 44 37 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880684607 GH On-Demand Anodyne MCHR1 21 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCSCC1 ZINC000880684609 CG On-Demand Anodyne CACNA1H 36 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@@](O)(C2CC2)C1 ZINC000880684610 DG On-Demand Anodyne PREP 37 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@@](O)(C2CC2)C1 ZINC000880684610 DG On-Demand Anodyne EBP 19 43 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@](O)(C2CC2)C1 ZINC000880684611 DG On-Demand Anodyne PREP 37 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCC[C@](O)(C2CC2)C1 ZINC000880684611 DG On-Demand Anodyne EBP 19 43 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@](O)(C2CC2)C1 ZINC000880684612 DG On-Demand Anodyne PREP 37 40 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@](O)(C2CC2)C1 ZINC000880684612 DG On-Demand Anodyne EBP 19 43 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@@](O)(C2CC2)C1 ZINC000880684613 DG On-Demand Anodyne PREP 37 40 O=C(CC[C@H]1CCc2ccccc21)N1CCC[C@@](O)(C2CC2)C1 ZINC000880684613 DG On-Demand Anodyne EBP 19 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)CC1 ZINC000880684614 DF On-Demand Anodyne CCR3 25 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)CC1 ZINC000880684614 DF On-Demand Anodyne EPHX2 37 56 CCN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684618 DG On-Demand Anodyne CCR3 97 41 CCN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684618 DG On-Demand Anodyne EPHX2 28 41 CCN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684618 DG On-Demand Anodyne CACNA1I 76 37 O=C1CC[C@@H]2CN(C(=O)c3cc4cccc(C(F)(F)F)c4nc3O)CC[C@@H]2N1 ZINC000880684632 GF On-Demand Anodyne RBP4 60 34 O=C1CC[C@H]2CN(C(=O)c3cc4cccc(C(F)(F)F)c4nc3O)CC[C@H]2N1 ZINC000880684633 GF On-Demand Anodyne RBP4 60 34 O=C(CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)N1CCCCC1 ZINC000880684634 GF On-Demand Anodyne MAPK1 21 42 O=C(CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)N1CCCCC1 ZINC000880684634 GF On-Demand Anodyne EPHX2 19 41 O=C(NCc1nnc2n1CCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880684640 EF On-Demand Anodyne PRMT3 54 35 Cn1cnnc1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684641 CE On-Demand Anodyne PRMT3 46 34 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684642 FE On-Demand Anodyne DRD4 19 43 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684642 FE On-Demand Anodyne CCR3 46 40 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684642 FE On-Demand Anodyne EPHX2 54 44 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684642 FE On-Demand Anodyne CXCR3 25 46 O=C(NC[C@@H](O)CN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684647 EF On-Demand Anodyne CCR3 30 40 O=C(NC[C@H](O)CN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684648 EF On-Demand Anodyne CCR3 30 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1OC ZINC000880684655 FI On-Demand Anodyne MT-ND1 18 44 COc1ccc(CN(C)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1OC ZINC000880684655 FI On-Demand Anodyne ENPP1 67 32 COc1ccc(CN(C)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1OC ZINC000880684655 FI On-Demand Anodyne DRTS_TRYCR 44 31 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684663 BG On-Demand Anodyne EPHX2 62 50 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684663 BG On-Demand Anodyne CXCR3 17 42 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880684669 GI On-Demand Anodyne ABCB1 18 43 O=C(NCCCN1CCCCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684670 FH On-Demand Anodyne CCR3 41 42 O=C(NCCCN1CCCCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684670 FH On-Demand Anodyne EPHX2 15 43 O=C(NCC(=O)N1CCc2ccccc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684689 GG On-Demand Anodyne DPP8 22 43 O=C(NCC(=O)N1CCc2ccccc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684689 GG On-Demand Anodyne NOD2 40 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC1 ZINC000880684695 CG On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC1 ZINC000880684695 CG On-Demand Anodyne EPHX2 30 48 CO[C@@H](C)CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684696 CG On-Demand Anodyne LEF 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1c1ccccn1 ZINC000880684697 EJ On-Demand Anodyne CACNA1H 35 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1c1ccccn1 ZINC000880684697 EJ On-Demand Anodyne GRM4 32 41 CCN(Cc1ccncc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684699 DI On-Demand Anodyne NPY2R 40 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1c1ccccn1 ZINC000880684700 EJ On-Demand Anodyne CACNA1H 35 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1c1ccccn1 ZINC000880684700 EJ On-Demand Anodyne GRM4 32 41 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684702 DG On-Demand Anodyne TBXAS1 38 41 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684702 DG On-Demand Anodyne QPCT 28 42 O=C(NCCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684709 EH On-Demand Anodyne TBXAS1 54 52 O=C(NCCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684709 EH On-Demand Anodyne CCR3 17 41 O=C(NCCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684709 EH On-Demand Anodyne HMOX2 48 34 O=C(NCCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684709 EH On-Demand Anodyne QPCT 63 60 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684712 GI On-Demand Anodyne EPHX2 61 53 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880684713 FH On-Demand Anodyne CCR3 55 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880684713 FH On-Demand Anodyne EPHX2 68 53 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880684713 FH On-Demand Anodyne CXCR3 26 48 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880684713 FH On-Demand Anodyne MCHR1 35 40 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2ccc(OC(F)(F)F)cc2)n1 ZINC000880684715 FE On-Demand Anodyne SLC12A5 57 35 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684716 GI On-Demand Anodyne CCR3 18 41 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684716 GI On-Demand Anodyne ACACB 15 40 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684716 GI On-Demand Anodyne CACNA1I 74 40 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2ccc(OC(F)(F)F)cc2)n1 ZINC000880684717 FE On-Demand Anodyne SLC12A5 57 35 CC(C)(C(=O)N1CCC(O)(CO)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880684718 EE On-Demand Anodyne EPHX2 19 42 O=C(NCCCOCC(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880684719 EH On-Demand Anodyne CCR3 16 41 O=C(NCCCN1CCCC1=O)Nc1cc(F)c(F)c(F)c1F ZINC000880684720 EE On-Demand Anodyne TYRO3 19 41 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684724 GI On-Demand Anodyne CCR3 18 41 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684724 GI On-Demand Anodyne ACACB 15 40 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684724 GI On-Demand Anodyne CACNA1I 74 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne CACNA1H 43 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne PDGFRB 52 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne TRPV1 16 63 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne NPY2R 45 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne FAAH 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne EPHX2 15 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880684732 FH On-Demand Anodyne DGAT1 25 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCSCC1 ZINC000880684746 DH On-Demand Anodyne EPHX2 19 40 O=C(NCCCOCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684759 DH On-Demand Anodyne CCR3 40 44 O=C(CCCNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684769 EF On-Demand Anodyne CCR3 33 42 O=C(CCCNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CC1 ZINC000880684769 EF On-Demand Anodyne EPHX2 41 39 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CCCCC1 ZINC000880684771 EG On-Demand Anodyne EPHX2 43 45 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CCCCC1 ZINC000880684771 EG On-Demand Anodyne PRMT3 51 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880684783 FH On-Demand Anodyne CCR3 46 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880684783 FH On-Demand Anodyne EPHX2 59 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880684783 FH On-Demand Anodyne CXCR3 21 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880684784 FH On-Demand Anodyne CCR3 46 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880684784 FH On-Demand Anodyne EPHX2 59 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880684784 FH On-Demand Anodyne CXCR3 21 46 CCN(CC)C(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684811 FH On-Demand Anodyne NPY2R 57 38 O=C(NC[C@H]1CCCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684818 DG On-Demand Anodyne EPHX2 15 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2nccs2)CC1 ZINC000880684828 FJ On-Demand Anodyne CACNA1H 41 37 NC(=O)c1ccc(CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C2CC2)cc1 ZINC000880684836 GI On-Demand Anodyne GCGR 18 42 NC(=O)c1ccc(CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C2CC2)cc1 ZINC000880684836 GI On-Demand Anodyne GIPR 58 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880684841 GG On-Demand Anodyne CACNA1H 43 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880684841 GG On-Demand Anodyne PDGFRB 30 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880684841 GG On-Demand Anodyne GRM4 62 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880684841 GG On-Demand Anodyne EPHX2 24 46 CC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684851 DE On-Demand Anodyne CACNA1H 37 43 O=C(NCC[C@@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684864 DG On-Demand Anodyne PRMT3 40 40 O=C(NCC[C@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684865 DG On-Demand Anodyne PRMT3 40 40 O=C(NCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684866 DG On-Demand Anodyne TBXAS1 55 49 O=C(NCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684866 DG On-Demand Anodyne CCR3 23 40 O=C(NCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684866 DG On-Demand Anodyne HMOX2 48 34 O=C(NCCCn1ccnc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684866 DG On-Demand Anodyne QPCT 80 63 COc1ccc(OC)c2c1CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C[C@@H]2O ZINC000880684878 GH On-Demand Anodyne CPT1A 40 34 COc1ccc(OC)c2c1CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C[C@@H]2O ZINC000880684878 GH On-Demand Anodyne CPT1B 44 34 COc1ccc(OC)c2c1CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C[C@H]2O ZINC000880684879 GH On-Demand Anodyne CPT1A 40 34 COc1ccc(OC)c2c1CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C[C@H]2O ZINC000880684879 GH On-Demand Anodyne CPT1B 44 34 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880684881 GH On-Demand Anodyne EPHX2 57 47 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684892 EG On-Demand Anodyne CCR3 40 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684892 EG On-Demand Anodyne EPHX2 15 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684892 EG On-Demand Anodyne CACNA1I 45 34 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684893 FH On-Demand Anodyne CACNA1H 51 38 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCOCC1 ZINC000880684919 CG On-Demand Anodyne EPHX2 60 46 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCOCC1 ZINC000880684919 CG On-Demand Anodyne CXCR3 17 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne CACNA1H 42 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne CCR1 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne CCR5 19 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne RBP4 51 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne MCHR1 31 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880684934 EJ On-Demand Anodyne ADAM10 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne CACNA1H 42 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne CCR1 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne CCR5 19 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne RBP4 51 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne MCHR1 31 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880684935 EJ On-Demand Anodyne ADAM10 18 40 CCOC(=O)N1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684938 FG On-Demand Anodyne P2RY12 48 43 CCOC(=O)N1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684938 FG On-Demand Anodyne TGM2 17 40 CCOC(=O)N1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684938 FG On-Demand Anodyne F13A1 31 40 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684939 DG On-Demand Anodyne CCR3 87 44 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684939 DG On-Demand Anodyne CCR2 15 43 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684939 DG On-Demand Anodyne EPHX2 50 42 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684939 DG On-Demand Anodyne CXCR3 21 42 CCN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684940 DG On-Demand Anodyne CCR3 87 44 CCN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684940 DG On-Demand Anodyne CCR2 15 43 CCN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684940 DG On-Demand Anodyne EPHX2 50 42 CCN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880684940 DG On-Demand Anodyne CXCR3 21 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC(F)F)CC1 ZINC000880684952 EG On-Demand Anodyne CACNA1H 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC(F)F)CC1 ZINC000880684952 EG On-Demand Anodyne FAAH 16 45 CCN(CC)C(=O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880684953 DF On-Demand Anodyne NPY2R 44 33 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc(F)c(C(F)F)c2)on1 ZINC000880684958 EI On-Demand Anodyne KCNA5 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne DRD4 25 56 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne KCNH2 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne SIGMAR1 26 53 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne SSTR5 52 39 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne CCR3 69 45 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne EPHX2 51 45 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne CXCR3 44 50 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880684966 GH On-Demand Anodyne MCHR1 70 48 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684970 EG On-Demand Anodyne CACNA1H 34 40 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880684970 EG On-Demand Anodyne EPHX2 38 41 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne MC4R 23 40 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne KCNQ2 60 37 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne NPY2R 78 38 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne PIK3CA 29 41 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne PIK3CD 21 40 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne MTOR 47 41 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne EPHX2 30 43 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne SCN10A 18 49 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne PIK3CB 35 40 O=C(NCc1ccccc1N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880684974 GH On-Demand Anodyne STAT6 57 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OC2CCCC2)CC1 ZINC000880684976 FJ On-Demand Anodyne EPHX2 42 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCCC[C@@H]12 ZINC000880684981 EH On-Demand Anodyne EPHX2 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000880684982 EH On-Demand Anodyne EPHX2 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCCC[C@H]12 ZINC000880684983 EH On-Demand Anodyne EPHX2 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCCC[C@H]12 ZINC000880684984 EH On-Demand Anodyne EPHX2 29 41 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880684991 GG On-Demand Mild PDGFRB 44 45 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880684991 GG On-Demand Mild DGAT1 28 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880685001 FH On-Demand Anodyne CCR3 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880685001 FH On-Demand Anodyne EPHX2 64 47 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880685001 FH On-Demand Anodyne CXCR3 24 50 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880685001 FH On-Demand Anodyne HPGDS 41 45 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685006 GF On-Demand Anodyne CACNA1H 29 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685006 GF On-Demand Anodyne EPHX2 34 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685006 GF On-Demand Anodyne CCR8 72 37 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685006 GF On-Demand Anodyne SFRP1 60 33 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685006 GF On-Demand Anodyne WNT3 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC2(CC1)OCCO2 ZINC000880685007 EH On-Demand Anodyne EPHX2 45 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCCCC2)CC1 ZINC000880685022 FI On-Demand Anodyne HRH3 16 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCCCC2)CC1 ZINC000880685022 FI On-Demand Anodyne EPHX2 27 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCCCC2)CC1 ZINC000880685022 FI On-Demand Anodyne L3MBTL3 130 46 Cc1cc(-c2nc(C)c(C(=O)N[C@@H]3CC[C@@H](C)S(=O)(=O)C3)s2)ccc1F ZINC000880685023 GG On-Demand Anodyne MAPK13 58 31 Cc1cc(-c2nc(C)c(C(=O)N[C@H]3CC[C@H](C)S(=O)(=O)C3)s2)ccc1F ZINC000880685024 GG On-Demand Anodyne MAPK13 58 31 Cc1cc(-c2nc(C)c(C(=O)N[C@H]3CC[C@@H](C)S(=O)(=O)C3)s2)ccc1F ZINC000880685025 GG On-Demand Anodyne MAPK13 58 31 Cc1cc(-c2nc(C)c(C(=O)N[C@@H]3CC[C@H](C)S(=O)(=O)C3)s2)ccc1F ZINC000880685026 GG On-Demand Anodyne MAPK13 58 31 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685034 GG On-Demand Anodyne TRPV1 32 45 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685034 GG On-Demand Anodyne P2RX7 19 43 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685034 GG On-Demand Anodyne NPY2R 46 37 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685034 GG On-Demand Anodyne SCN10A 21 41 COCC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685046 EE On-Demand Anodyne PDGFRB 44 35 O=C(NCCOC1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685060 DH On-Demand Anodyne ADRB1 21 48 O=C(NCCOC1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685060 DH On-Demand Anodyne CCR3 24 43 O=C(NCCOC1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685060 DH On-Demand Anodyne EPHX2 22 40 CCC(=O)N1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685066 EG On-Demand Anodyne EPHX2 30 41 CC(C)(C)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685069 EI On-Demand Anodyne EPHX2 58 47 CC(C)(C)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685069 EI On-Demand Anodyne CXCR3 21 46 CN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685077 DF On-Demand Anodyne CCR3 73 40 CN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685077 DF On-Demand Anodyne EPHX2 52 45 CN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685077 DF On-Demand Anodyne CXCR3 16 40 COCC(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685080 FF On-Demand Anodyne EPHX2 46 40 COCC(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685080 FF On-Demand Anodyne MCHR1 24 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2cscn2)CC1 ZINC000880685086 FH On-Demand Anodyne FAAH 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2cscn2)CC1 ZINC000880685086 FH On-Demand Anodyne SCN5A 41 35 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685089 GI On-Demand Anodyne EPHX2 33 41 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685089 GI On-Demand Anodyne ASAH1 60 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](N2CCCC2)C1 ZINC000880685094 EH On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](N2CCCC2)C1 ZINC000880685094 EH On-Demand Anodyne L3MBTL3 82 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](N2CCCC2)C1 ZINC000880685095 EH On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](N2CCCC2)C1 ZINC000880685095 EH On-Demand Anodyne L3MBTL3 82 40 C[C@H]1CC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CS1(=O)=O ZINC000880685104 FD On-Demand Anodyne GABRA1 18 42 C[C@H]1CC[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CS1(=O)=O ZINC000880685104 FD On-Demand Anodyne GABRA2 16 42 C[C@H]1CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CS1(=O)=O ZINC000880685107 FD On-Demand Anodyne GABRA1 18 42 C[C@H]1CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CS1(=O)=O ZINC000880685107 FD On-Demand Anodyne GABRA2 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000880685110 FH On-Demand Anodyne PANC 46 35 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000880685111 FH On-Demand Anodyne PANC 46 35 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean F2R 49 31 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean MTOR 60 39 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean EPHX2 30 44 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean PIK3CB 23 40 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean STAT6 77 41 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685114 GH On-Demand Clean NAMPT 38 41 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685118 GF On-Demand Anodyne CCR3 26 43 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685118 GF On-Demand Anodyne EPHX2 18 43 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685119 GF On-Demand Anodyne CCR3 26 43 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685119 GF On-Demand Anodyne EPHX2 18 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880685143 FG On-Demand Anodyne EPHX2 40 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880685144 FG On-Demand Anodyne EPHX2 40 39 COCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685160 CG On-Demand Anodyne CCR3 18 42 COCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685160 CG On-Demand Anodyne EPHX2 15 43 COCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685160 CG On-Demand Anodyne LEF 33 45 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne HRH2 24 43 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne CCR3 62 44 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne CHRNA7 26 55 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne F2R 50 31 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne EPHX2 28 59 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne PLD2 43 33 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne MCHR1 30 48 O=C(NCCN1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685170 DG On-Demand Anodyne PRMT3 40 38 O=C(NCCN1Cc2ccccc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685171 EH On-Demand Anodyne CCR3 33 41 O=C(NCCN1Cc2ccccc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685171 EH On-Demand Anodyne EPHX2 19 45 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685177 GH On-Demand Anodyne MAPK14 22 41 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685177 GH On-Demand Anodyne CCR3 38 40 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685177 GH On-Demand Anodyne ROCK2 22 44 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685177 GH On-Demand Anodyne EPHX2 32 44 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685177 GH On-Demand Anodyne PRMT3 50 31 O=C(NCCN1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685203 EF On-Demand Anodyne HTR2A 17 40 O=C(NCCN1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685203 EF On-Demand Anodyne CCR3 42 43 O=C(NCCN1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685203 EF On-Demand Anodyne EPHX2 26 50 O=C(NCCN1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685203 EF On-Demand Anodyne PLD2 43 32 O=C(NCCN1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685203 EF On-Demand Anodyne MCHR1 17 41 CN1CCC(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685204 DG On-Demand Anodyne HTR1F 48 37 CN1CCC(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685204 DG On-Demand Anodyne CCR3 88 45 CN1CCC(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685204 DG On-Demand Anodyne EPHX2 53 45 CN1CCC(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685204 DG On-Demand Anodyne MCHR1 30 41 CN1CCC(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685204 DG On-Demand Anodyne CACNA1I 81 39 O=C(NC[C@@H](O)C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685214 CF On-Demand Anodyne PRMT3 41 50 O=C(NC[C@H](O)C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685215 CF On-Demand Anodyne PRMT3 41 50 O=C(NCCN1C(=O)CCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685216 EE On-Demand Anodyne CCR3 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(=O)N2CCOCC2)CC1 ZINC000880685223 GF On-Demand Anodyne ITGAL 40 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(=O)N2CCOCC2)CC1 ZINC000880685223 GF On-Demand Anodyne EPHX2 42 46 COC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685224 EG On-Demand Anodyne CACNA1H 37 40 COC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685224 EG On-Demand Anodyne EPHX2 36 42 COc1ccc(CN(CCO)C(=O)Nc2ccc(F)c(C(F)F)c2)c(OC)c1 ZINC000880685232 GH On-Demand Anodyne ROCK2 15 42 Cc1ncc(CN2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)s1 ZINC000880685233 GH On-Demand Anodyne FAAH 18 40 N#CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685234 CH On-Demand Mild ADRB1 41 34 N#CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685234 CH On-Demand Mild CCR3 17 41 N#CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685237 EF On-Demand Mild CCR3 42 40 N#CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685237 EF On-Demand Mild EPHX2 51 43 N#CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685237 EF On-Demand Mild CXCR3 22 47 C[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685238 EE On-Demand Anodyne CACNA1H 40 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880685241 FE On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880685241 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880685241 FE On-Demand Anodyne CTSL 22 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880685241 FE On-Demand Anodyne REN 41 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880685241 FE On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880685242 FE On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880685242 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880685242 FE On-Demand Anodyne CTSL 22 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880685242 FE On-Demand Anodyne REN 41 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880685242 FE On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880685243 FE On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880685243 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880685243 FE On-Demand Anodyne CTSL 22 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880685243 FE On-Demand Anodyne REN 41 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880685243 FE On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880685244 FE On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880685244 FE On-Demand Anodyne CTSK 24 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880685244 FE On-Demand Anodyne CTSL 22 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880685244 FE On-Demand Anodyne REN 41 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880685244 FE On-Demand Anodyne FPR1 48 38 O=C(Nc1ccc(F)c(C(F)F)c1)N(Cc1cccnc1)C1CC1 ZINC000880685262 EI On-Demand Anodyne CHRNA7 40 38 O=C(Nc1ccc(F)c(C(F)F)c1)N(Cc1cccnc1)C1CC1 ZINC000880685262 EI On-Demand Anodyne MCHR1 30 43 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880685264 FH On-Demand Anodyne CACNA1H 77 48 O=C(CN1CCCC1)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685275 GF On-Demand Anodyne MAPK1 22 43 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685276 GI On-Demand Anodyne CCR2 22 42 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685276 GI On-Demand Anodyne EPHX2 42 40 O=C(NN1CCc2ccccc2C1)c1ccc(CN2CCOCC2)o1 ZINC000880685278 ED On-Demand Anodyne NOD1 17 40 O=C(NN1CCc2ccccc2C1)c1ccc(CN2CCOCC2)o1 ZINC000880685278 ED On-Demand Anodyne NOD2 45 37 O=C(NCC1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685281 DI On-Demand Anodyne EPHX2 15 47 O=C(NCC1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685281 DI On-Demand Anodyne CACNA1I 44 34 O=C(NCC1CCSCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685281 DI On-Demand Anodyne PRMT3 47 35 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685291 FH On-Demand Anodyne EPHX2 33 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@@H](O)C1 ZINC000880685293 DG On-Demand Anodyne EPHX2 49 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@H](O)C1 ZINC000880685294 DG On-Demand Anodyne EPHX2 49 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@@H](O)C1 ZINC000880685295 DG On-Demand Anodyne EPHX2 49 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H](O)C1 ZINC000880685296 DG On-Demand Anodyne EPHX2 49 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2cccnn2)CC1 ZINC000880685299 FF On-Demand Anodyne FAAH 24 45 O=C(NCCCn1cncn1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685306 DF On-Demand Anodyne QPCT 45 42 COCCN(Cc1ccccn1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685308 FH On-Demand Anodyne GRM4 30 43 C[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C[C@@H](C)[C@@H]1O ZINC000880685326 FG On-Demand Anodyne RBP4 43 34 C[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C[C@H](C)C1O ZINC000880685327 FG On-Demand Anodyne RBP4 43 34 CCCN(CC)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685328 CI On-Demand Anodyne NPY2R 42 34 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685342 GD On-Demand Anodyne CCR3 47 44 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685342 GD On-Demand Anodyne EPHX2 31 47 CCO[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685344 DH On-Demand Anodyne EPHX2 33 44 O=C(NCc1cn2c(n1)CCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880685353 EH On-Demand Anodyne PRMT3 52 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880685356 GG On-Demand Anodyne NPY2R 32 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880685356 GG On-Demand Anodyne EPHX2 25 43 CCN(Cc1ccoc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685362 DI On-Demand Anodyne NPY2R 42 33 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CCCC1 ZINC000880685370 EF On-Demand Anodyne EPHX2 40 44 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NC1CCCC1 ZINC000880685370 EF On-Demand Anodyne PRMT3 49 38 O=C(CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)N1CCCC1 ZINC000880685371 GI On-Demand Anodyne EPHX2 35 42 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@@H](C)[C@@H]1O ZINC000880685380 GE On-Demand Anodyne CELA1 18 41 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@@H](C)[C@@H]1O ZINC000880685380 GE On-Demand Anodyne PREP 53 49 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@@H](C)[C@@H]1O ZINC000880685380 GE On-Demand Anodyne SLC12A5 46 35 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@@H](C)[C@@H]1O ZINC000880685380 GE On-Demand Anodyne Q9NAW4_PLAFA 27 43 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@H](C)C1O ZINC000880685381 GE On-Demand Anodyne CELA1 18 41 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@H](C)C1O ZINC000880685381 GE On-Demand Anodyne PREP 53 49 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@H](C)C1O ZINC000880685381 GE On-Demand Anodyne SLC12A5 46 35 C[C@H]1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C[C@H](C)C1O ZINC000880685381 GE On-Demand Anodyne Q9NAW4_PLAFA 27 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(c2nccs2)CC1 ZINC000880685386 FH On-Demand Anodyne PDGFRB 40 38 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685392 FH On-Demand Anodyne EPHX2 33 42 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685410 FG On-Demand Anodyne NPY5R 32 40 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685411 FG On-Demand Anodyne NPY5R 32 40 O=C(NCCCN1C(=O)CNC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685412 ED On-Demand Anodyne CCR3 37 42 CN1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685417 DG On-Demand Anodyne CCR3 101 44 CN1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685417 DG On-Demand Anodyne EPHX2 28 46 CN1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685417 DG On-Demand Anodyne MCHR1 24 43 CN1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685417 DG On-Demand Anodyne CACNA1I 71 35 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCOC1 ZINC000880685418 CG On-Demand Anodyne EPHX2 48 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCOC1 ZINC000880685419 CG On-Demand Anodyne EPHX2 48 42 CCOCCN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685424 EF On-Demand Anodyne HTR1B 15 40 CCOCCN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685424 EF On-Demand Anodyne PDGFRB 40 37 CCOCCN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685424 EF On-Demand Anodyne EPHX2 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000880685447 GF On-Demand Anodyne EPHX2 24 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](C(=O)N2CCOCC2)C1 ZINC000880685448 GF On-Demand Anodyne EPHX2 24 42 O=C(NCCCN1C(=O)CCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685457 EE On-Demand Anodyne CCR3 38 43 O=C(NCCCN1C(=O)CCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685457 EE On-Demand Anodyne EPHX2 15 40 COc1ccccc1-c1ccc(C(=O)NCCCOC(C)(C)C)c(O)n1 ZINC000880685468 FG On-Demand Anodyne DRD2 20 40 COc1ccccc1-c1ccc(C(=O)NCCCOC(C)(C)C)c(O)n1 ZINC000880685468 FG On-Demand Anodyne DRD3 37 40 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685484 FH On-Demand Anodyne EPHX2 28 42 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685484 FH On-Demand Anodyne HCN1 57 39 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685484 FH On-Demand Anodyne HCN4 49 31 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne DRD4 15 54 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne SIGMAR1 16 48 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne CCR3 51 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne EPHX2 50 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne CXCR3 28 47 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880685510 GH On-Demand Anodyne MCHR1 48 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC2CC2)CC1 ZINC000880685528 EH On-Demand Anodyne SIGMAR1 19 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC2CC2)CC1 ZINC000880685528 EH On-Demand Anodyne CCR3 70 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC2CC2)CC1 ZINC000880685528 EH On-Demand Anodyne EPHX2 58 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CC2CC2)CC1 ZINC000880685528 EH On-Demand Anodyne CXCR3 25 52 COCCN(Cc1ccc(C#N)cc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685533 GI On-Demand Mild MCHR1 16 45 O=C(NCCCNc1ccccn1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685540 EH On-Demand Anodyne ADRB1 41 33 O=C(NCCCNc1ccccn1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685540 EH On-Demand Anodyne DOT1L 48 31 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880685542 GH On-Demand Anodyne EPHX2 67 67 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880685542 GH On-Demand Anodyne CXCR3 21 46 O=C(NCCCN1CCCS1(=O)=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685572 FE On-Demand Anodyne CCR3 35 44 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685581 CH On-Demand Anodyne CACNA1H 34 41 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685581 CH On-Demand Anodyne EPHX2 37 48 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685582 CH On-Demand Anodyne CACNA1H 34 41 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685582 CH On-Demand Anodyne EPHX2 37 48 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@](O)(C3CC3)C2)N1Cc1ccccc1 ZINC000880685584 FD On-Demand Anodyne PREP 57 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@](O)(C3CC3)C2)N1Cc1ccccc1 ZINC000880685585 FD On-Demand Anodyne PREP 57 40 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)Cc2ccccc21 ZINC000880685606 EI On-Demand Anodyne NPY2R 47 34 O=C1CC[C@H](c2ccc(C(=O)NN3CCc4ccccc4C3)cc2)N1 ZINC000880685607 EE On-Demand Anodyne NOD2 43 37 O=C1CC[C@@H](c2ccc(C(=O)NN3CCc4ccccc4C3)cc2)N1 ZINC000880685608 EE On-Demand Anodyne NOD2 43 37 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685616 GG On-Demand Anodyne NPY2R 43 34 O=C(COC1CC1)NN1CCc2ccccc2C1 ZINC000880685651 BD On-Demand Anodyne NOD2 40 34 CCc1noc([C@@H](C)N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880685662 GH On-Demand Anodyne NPY2R 31 47 CCc1noc([C@H](C)N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880685663 GH On-Demand Anodyne NPY2R 31 47 O=C(NC[C@@H](O)COCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685670 EF On-Demand Anodyne ADRB1 42 35 O=C(NC[C@H](O)COCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685671 EF On-Demand Anodyne ADRB1 42 35 COC(=O)C1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685672 EH On-Demand Anodyne EPHX2 57 45 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880685674 GF On-Demand Anodyne PDGFRB 54 40 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880685674 GF On-Demand Anodyne FAAH 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCCC[C@@H]2C1 ZINC000880685679 EG On-Demand Anodyne L3MBTL3 76 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCCC[C@H]2C1 ZINC000880685680 EG On-Demand Anodyne L3MBTL3 76 39 Cc1nc(CN2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)oc1C ZINC000880685681 GH On-Demand Anodyne FAAH 17 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC1 ZINC000880685682 CG On-Demand Anodyne EPHX2 62 50 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC1 ZINC000880685682 CG On-Demand Anodyne CXCR3 17 41 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685684 EE On-Demand Anodyne CCR3 49 39 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685684 EE On-Demand Anodyne CACNA1I 48 31 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685685 EE On-Demand Anodyne CCR3 49 39 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685685 EE On-Demand Anodyne CACNA1I 48 31 O=C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCN1 ZINC000880685686 DE On-Demand Anodyne CACNA1H 40 36 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685700 EG On-Demand Anodyne CCR3 33 41 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685700 EG On-Demand Anodyne EPHX2 40 43 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685700 EG On-Demand Anodyne CACNA1I 65 38 COCCOc1ccc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880685705 FH On-Demand Anodyne ROCK2 16 41 COCCOc1ccc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880685705 FH On-Demand Anodyne PRMT3 46 37 CC(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685713 EF On-Demand Anodyne EPHX2 31 41 CC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685714 EF On-Demand Anodyne EPHX2 31 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OCC(F)(F)F)C1 ZINC000880685717 FI On-Demand Anodyne EPHX2 41 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OCC(F)(F)F)C1 ZINC000880685718 FI On-Demand Anodyne EPHX2 41 36 O=C(CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)NC1CCCC1 ZINC000880685747 GI On-Demand Anodyne CCR2 17 40 O=C(CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)NC1CCCC1 ZINC000880685747 GI On-Demand Anodyne EPHX2 47 40 CCOC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685756 EI On-Demand Anodyne CCR3 25 47 CCOC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685756 EI On-Demand Anodyne EPHX2 21 45 O=C(NCC1(O)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685757 DE On-Demand Anodyne EPHX2 22 40 O=C(NCC1(O)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685757 DE On-Demand Anodyne PRMT3 43 31 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685759 EH On-Demand Mild CCR3 42 40 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685759 EH On-Demand Mild EPHX2 56 44 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685759 EH On-Demand Mild CXCR3 24 46 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685772 FH On-Demand Anodyne CCR3 78 40 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685772 FH On-Demand Anodyne CACNA1I 74 36 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685774 FH On-Demand Anodyne CCR3 78 40 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685774 FH On-Demand Anodyne CACNA1I 74 36 COC(=O)N1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685776 EG On-Demand Anodyne EPHX2 52 42 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685778 EG On-Demand Anodyne EPHX2 52 42 O=C(NC[C@@]1(N2CCOCC2)CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685780 GG On-Demand Anodyne EPHX2 24 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCO)CC1 ZINC000880685781 DG On-Demand Anodyne EPHX2 39 48 O=C(NC[C@]1(N2CCOCC2)CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685782 GG On-Demand Anodyne EPHX2 24 42 N#Cc1ccc(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880685798 GH On-Demand Mild EPHX2 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880685799 GG On-Demand Anodyne NPY2R 24 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880685799 GG On-Demand Anodyne EPHX2 23 47 CO[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685821 DG On-Demand Anodyne HTR1D 16 41 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne SLC6A1 104 38 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne CCR3 79 51 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne CHRNA7 20 47 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne F2R 52 33 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne EPHX2 18 42 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685851 FE On-Demand Anodyne MCHR1 28 43 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne SLC6A1 104 38 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne CCR3 79 51 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne CHRNA7 20 47 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne F2R 52 33 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne EPHX2 18 42 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685852 FE On-Demand Anodyne MCHR1 28 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000880685863 EH On-Demand Anodyne EPHX2 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000880685863 EH On-Demand Anodyne L3MBTL3 109 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCCCC2)C1 ZINC000880685864 EH On-Demand Anodyne EPHX2 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCCCC2)C1 ZINC000880685864 EH On-Demand Anodyne L3MBTL3 109 45 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne HTR2A 36 45 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne CHRNA7 18 43 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne MTOR 48 37 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne EPHX2 33 52 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne MCHR1 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880685875 GF On-Demand Anodyne STAT6 42 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCCC2)C1 ZINC000880685891 EG On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCCC2)C1 ZINC000880685891 EG On-Demand Anodyne L3MBTL3 110 46 O=C(NC[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685893 DG On-Demand Anodyne EPHX2 15 41 O=C(NCCC(=O)N1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685894 EG On-Demand Anodyne EPHX2 25 42 O=C(NCCC(=O)N1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685894 EG On-Demand Anodyne PRMT3 34 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@H](C)C(O)[C@@H](C)C1 ZINC000880685907 ED On-Demand Anodyne CTSK 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@H](C)[C@@H](O)[C@H](C)C1 ZINC000880685908 ED On-Demand Anodyne CTSK 15 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@H](C)[C@@H](O)[C@H](C)C1 ZINC000880685909 ED On-Demand Anodyne CTSK 15 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](C)C(O)[C@H](C)C1 ZINC000880685910 ED On-Demand Anodyne CTSK 15 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCCC2)C1 ZINC000880685923 EG On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCCC2)C1 ZINC000880685923 EG On-Demand Anodyne L3MBTL3 110 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)C(=O)N2CCCC2)CC1 ZINC000880685924 GE On-Demand Anodyne EPHX2 22 44 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685926 FE On-Demand Anodyne CCR3 33 42 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685926 FE On-Demand Anodyne EPHX2 53 42 O=C(NCc1ccnc(OC2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880685931 GI On-Demand Anodyne MAPK1 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880685944 EG On-Demand Anodyne CCR3 76 47 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880685944 EG On-Demand Anodyne CCR2 23 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880685944 EG On-Demand Anodyne EPHX2 47 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880685944 EG On-Demand Anodyne CXCR3 21 45 C[C@@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685945 FF On-Demand Anodyne PDE4D 17 41 C[C@@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685945 FF On-Demand Anodyne UTS2R 21 42 C[C@@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685945 FF On-Demand Anodyne EZH2 44 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880685946 EG On-Demand Anodyne CCR3 76 47 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880685946 EG On-Demand Anodyne CCR2 23 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880685946 EG On-Demand Anodyne EPHX2 47 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880685946 EG On-Demand Anodyne CXCR3 21 45 C[C@H]1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685947 FF On-Demand Anodyne PDE4D 17 41 C[C@H]1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685947 FF On-Demand Anodyne UTS2R 21 42 C[C@H]1CC[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685947 FF On-Demand Anodyne EZH2 44 41 C[C@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685949 FF On-Demand Anodyne PDE4D 17 41 C[C@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685949 FF On-Demand Anodyne UTS2R 21 42 C[C@H]1CC[C@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)CS1(=O)=O ZINC000880685949 FF On-Demand Anodyne EZH2 44 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCSCC1 ZINC000880685951 DH On-Demand Anodyne EPHX2 56 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCSCC1 ZINC000880685951 DH On-Demand Anodyne CXCR3 15 40 COCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685953 DH On-Demand Anodyne CCR3 17 44 COCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685953 DH On-Demand Anodyne EPHX2 15 44 COCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685953 DH On-Demand Anodyne LEF 30 44 COCCn1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880685955 EG On-Demand Anodyne HTR2A 42 40 COCCn1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880685955 EG On-Demand Anodyne HTR2C 15 42 CN1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880685958 DE On-Demand Anodyne FPR2 44 37 CN1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880685960 DE On-Demand Anodyne FPR2 44 37 CN(C)CCn1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880685969 EG On-Demand Anodyne FPR2 40 34 Cc1noc(C)c1CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685975 EH On-Demand Anodyne NPY2R 16 41 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685979 DH On-Demand Anodyne CCR3 39 49 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880685979 DH On-Demand Anodyne EPHX2 24 48 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685980 GI On-Demand Anodyne NPY2R 50 37 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685980 GI On-Demand Anodyne EPHX2 65 55 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685980 GI On-Demand Anodyne CXCR3 20 44 CCOCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685986 DH On-Demand Anodyne CCR3 26 43 CCOCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685986 DH On-Demand Anodyne EPHX2 18 44 CCOCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685986 DH On-Demand Anodyne LEF 18 44 CCN(CC)C(=O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685987 GF On-Demand Anodyne NPY2R 47 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCNC2=O)CC1 ZINC000880685988 FF On-Demand Anodyne CACNA1H 41 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCNC2=O)CC1 ZINC000880685988 FF On-Demand Anodyne SCD1 17 41 O=C(NC[C@@H](O)COc1ccc2c(c1)OCO2)Nc1ccc(F)c(C(F)F)c1 ZINC000880685989 GG On-Demand Anodyne ADRB1 42 34 O=C(NC[C@@H](O)COc1ccc2c(c1)OCO2)Nc1ccc(F)c(C(F)F)c1 ZINC000880685989 GG On-Demand Anodyne ADRB3 16 40 O=C(NC[C@H](O)COc1ccc2c(c1)OCO2)Nc1ccc(F)c(C(F)F)c1 ZINC000880685991 GG On-Demand Anodyne ADRB1 42 34 O=C(NC[C@H](O)COc1ccc2c(c1)OCO2)Nc1ccc(F)c(C(F)F)c1 ZINC000880685991 GG On-Demand Anodyne ADRB3 16 40 CC(C)(C)OC(=O)NC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880685993 GI On-Demand Anodyne EPHX2 43 38 COCCOc1ncccc1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685998 FH On-Demand Anodyne P2RY1 40 37 COCCOc1ncccc1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880685998 FH On-Demand Anodyne SCN10A 15 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880686008 EH On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880686008 EH On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880686009 EH On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880686009 EH On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880686010 EH On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880686010 EH On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880686011 EH On-Demand Anodyne EPHX2 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880686011 EH On-Demand Anodyne CXCR3 19 41 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686017 FH On-Demand Anodyne GPBAR1 19 40 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686018 FH On-Demand Anodyne GPBAR1 19 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne CACNA1H 40 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne HTR1D 20 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne HTR1B 17 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne HTR1F 56 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne CCR2 35 63 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880686029 GK On-Demand Anodyne LIMK2 24 40 O=C(NCC1(O)CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686030 DG On-Demand Anodyne PRMT3 60 33 NC(=O)CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686032 CD On-Demand Anodyne PRMT3 45 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCC[C@@H]2C1 ZINC000880686035 DG On-Demand Anodyne L3MBTL3 59 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCC[C@H]2C1 ZINC000880686036 DG On-Demand Anodyne L3MBTL3 59 37 N#Cc1ccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686045 GJ On-Demand Mild CCR3 24 41 N#Cc1ccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686045 GJ On-Demand Mild S1PR2 17 42 N#Cc1ccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686045 GJ On-Demand Mild EPHX2 37 55 O=C(Cc1ccccc1N1CCCC1=O)NN1CCc2ccccc2C1 ZINC000880686051 EE On-Demand Anodyne HTR7 15 41 CN1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880686090 DF On-Demand Anodyne EPHX2 33 41 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686094 GG On-Demand Anodyne PRNP 47 35 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686094 GG On-Demand Anodyne MAPK1 17 40 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cc1 ZINC000880686094 GG On-Demand Anodyne STAT6 50 35 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1C ZINC000880686096 CH On-Demand Anodyne CACNA1H 31 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1C ZINC000880686097 CH On-Demand Anodyne CACNA1H 31 40 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1C ZINC000880686098 CH On-Demand Anodyne CACNA1H 31 40 C[C@@](CO)(NC(=O)Nc1ccc(F)c(C(F)F)c1)C1CC1 ZINC000880686099 DG On-Demand Anodyne IMDH_CRYPV 41 33 O=C(NCCCC(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880686101 DI On-Demand Anodyne CCR3 17 40 O=C(NCCCC(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880686101 DI On-Demand Anodyne EPHX2 17 40 C[C@@H](CCN(C)C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686104 DG On-Demand Anodyne UTS2 58 34 C[C@H]1[C@H](C)CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686106 CI On-Demand Anodyne TRPC6 46 34 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H]1C ZINC000880686107 CI On-Demand Anodyne TRPC6 46 34 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H]1C ZINC000880686108 CI On-Demand Anodyne TRPC6 46 34 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H]1C ZINC000880686109 CI On-Demand Anodyne TRPC6 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](C(F)(F)F)C1 ZINC000880686129 EH On-Demand Anodyne EPHX2 32 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](C(F)(F)F)C1 ZINC000880686130 EH On-Demand Anodyne EPHX2 32 41 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686136 GF On-Demand Anodyne EPHX2 33 44 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686137 GF On-Demand Anodyne EPHX2 33 44 O=C(NCC1(O)CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686142 CF On-Demand Anodyne PRMT3 60 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(C1)OCCO2 ZINC000880686147 DF On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(C1)OCCO2 ZINC000880686147 DF On-Demand Anodyne EPHX2 39 45 CN1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCC1=O ZINC000880686157 DF On-Demand Anodyne EPHX2 42 37 CN1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCC1=O ZINC000880686158 DF On-Demand Anodyne EPHX2 42 37 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686166 FF On-Demand Mild CASR 68 54 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686166 FF On-Demand Mild EPHX2 23 42 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686166 FF On-Demand Mild MCHR1 26 43 O=C(NN1CCc2ccccc2C1)c1c[nH]cc1C1CC1 ZINC000880686194 CF On-Demand Anodyne HTR1F 64 35 NC(=O)c1ccccc1N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686200 GG On-Demand Anodyne CCR3 21 40 NC(=O)c1ccccc1N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686201 GG On-Demand Anodyne CCR3 21 40 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686212 EF On-Demand Anodyne HTR2A 18 41 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686212 EF On-Demand Anodyne CASR 62 48 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686212 EF On-Demand Anodyne EPHX2 28 46 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686212 EF On-Demand Anodyne MCHR1 39 42 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686212 EF On-Demand Anodyne STAT6 40 32 O=C(NCC1(O)CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686232 DH On-Demand Anodyne PRMT3 62 35 O=C(CC1CCCC1)N1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686243 GI On-Demand Anodyne EPHX2 28 42 COCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686256 DH On-Demand Anodyne CACNA1H 40 39 COCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686256 DH On-Demand Anodyne PDGFRB 41 35 COCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686256 DH On-Demand Anodyne CCR3 32 44 COCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686256 DH On-Demand Anodyne EPHX2 36 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ncc[nH]2)CC1 ZINC000880686268 EH On-Demand Anodyne HTR2B 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ncc[nH]2)CC1 ZINC000880686268 EH On-Demand Anodyne CCR2 15 44 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686269 EF On-Demand Anodyne EPHX2 22 41 CN(C)C(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCC1 ZINC000880686281 FH On-Demand Anodyne PRMT3 43 31 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCS(=O)(=O)CC1 ZINC000880686288 EE On-Demand Anodyne EPHX2 49 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880686289 FH On-Demand Anodyne EPHX2 49 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880686289 FH On-Demand Anodyne CXCR3 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880686291 FH On-Demand Anodyne EPHX2 49 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880686291 FH On-Demand Anodyne CXCR3 20 42 C[C@H](O)CN(Cc1ccccc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686292 FI On-Demand Anodyne NPY5R 33 40 O=C(C[C@@H]1CCNC1=O)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880686305 CC On-Demand Anodyne BDKRB1 15 43 O=C(C[C@@H]1CCNC1=O)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880686306 CC On-Demand Anodyne BDKRB1 15 43 O=C(C[C@@H]1CCNC1=O)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880686307 CC On-Demand Anodyne BDKRB1 15 43 O=C(C[C@@H]1CCNC1=O)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880686308 CC On-Demand Anodyne BDKRB1 15 43 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686325 GE On-Demand Anodyne ABCB1 25 44 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CC(=O)N2CCOCC2)c1 ZINC000880686333 GE On-Demand Anodyne MTOR 55 32 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cnn(CC(=O)N2CCOCC2)c1 ZINC000880686333 GE On-Demand Anodyne EPHX2 27 46 CC(C)(C)[C@@H](O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686338 DG On-Demand Anodyne PRMT3 45 34 CC(C)(C)N1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880686339 EG On-Demand Anodyne EPHX2 44 38 CC(C)(C)N1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880686341 EG On-Demand Anodyne EPHX2 44 38 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880686358 EE On-Demand Anodyne CCR3 65 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880686358 EE On-Demand Anodyne SLC6A5 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880686358 EE On-Demand Anodyne EPHX2 60 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880686358 EE On-Demand Anodyne CXCR3 24 46 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880686358 EE On-Demand Anodyne MCHR1 49 42 Cc1nc(C(C)(C)NC(=O)Nc2ccc(F)c(C(F)F)c2)no1 ZINC000880686360 EH On-Demand Anodyne IMDH_CRYPV 52 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCC2)C1 ZINC000880686372 DJ On-Demand Anodyne CACNA1H 46 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCC2)C1 ZINC000880686372 DJ On-Demand Anodyne EPHX2 39 51 CCOC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686377 DH On-Demand Anodyne CCR3 25 46 CCOC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686377 DH On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC[C@@H]1CO ZINC000880686381 DG On-Demand Anodyne CCR3 35 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC[C@@H]1CO ZINC000880686381 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC[C@@H]1CO ZINC000880686382 DG On-Demand Anodyne CCR3 35 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC[C@@H]1CO ZINC000880686382 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC[C@H]1CO ZINC000880686383 DG On-Demand Anodyne CCR3 35 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC[C@H]1CO ZINC000880686383 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC[C@H]1CO ZINC000880686384 DG On-Demand Anodyne CCR3 35 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC[C@H]1CO ZINC000880686384 DG On-Demand Anodyne EPHX2 24 40 CC[C@@](C)(CO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686388 CG On-Demand Anodyne IMDH_CRYPV 53 33 O=C(NCCOC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686389 DG On-Demand Anodyne ADRB1 19 46 O=C(NCCOC1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686389 DG On-Demand Anodyne CCR3 21 43 CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686394 DH On-Demand Anodyne CACNA1H 76 45 CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686394 DH On-Demand Anodyne NPY5R 15 40 CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686394 DH On-Demand Anodyne S1PR2 34 49 CS[C@@H]1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686411 DI On-Demand Anodyne EPHX2 45 39 CS[C@H]1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686412 DI On-Demand Anodyne EPHX2 45 39 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686416 EF On-Demand Anodyne CACNA1H 43 38 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686416 EF On-Demand Anodyne NPY2R 41 33 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686417 EF On-Demand Anodyne CACNA1H 43 38 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686417 EF On-Demand Anodyne NPY2R 41 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(F)(F)F)(C(F)(F)F)C1 ZINC000880686418 GK On-Demand Mild CACNA1H 44 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(F)(F)F)(C(F)(F)F)C1 ZINC000880686418 GK On-Demand Mild EPHX2 40 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880686421 EG On-Demand Anodyne CACNA1H 40 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880686421 EG On-Demand Anodyne EPHX2 40 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880686422 EG On-Demand Anodyne CACNA1H 40 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880686422 EG On-Demand Anodyne EPHX2 40 45 Cn1nc2c(cc1=O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880686429 FE On-Demand Anodyne MAPK1 47 37 Cn1nc2c(cc1=O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880686429 FE On-Demand Anodyne P2RY14 45 33 Cn1ccnc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1=O ZINC000880686432 GE On-Demand Anodyne PDGFRB 52 40 CCN(Cc1ccccn1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686437 DI On-Demand Anodyne NPY2R 48 36 O=C(NCCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686438 CH On-Demand Anodyne CCR3 43 42 O=C(NCCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686438 CH On-Demand Anodyne PRMT3 42 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CC2)CC1 ZINC000880686439 DG On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CC2)CC1 ZINC000880686439 DG On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CC2)CC1 ZINC000880686439 DG On-Demand Anodyne L3MBTL3 50 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCCCC2)C1 ZINC000880686446 EI On-Demand Anodyne EPHX2 39 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCC2)CC1 ZINC000880686447 EG On-Demand Anodyne HRH3 27 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCC2)CC1 ZINC000880686447 EG On-Demand Anodyne EPHX2 22 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCC2)CC1 ZINC000880686447 EG On-Demand Anodyne L3MBTL3 65 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2cncnc2C1 ZINC000880686477 DG On-Demand Anodyne MAPK1 59 42 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686479 GH On-Demand Anodyne PDGFRB 59 43 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne ADRA1B 15 44 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne HTR4 38 41 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne CCR3 84 41 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne CHRNA7 17 41 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne EPHX2 72 55 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne CXCR3 25 46 CCCCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686480 EI On-Demand Anodyne MCHR1 57 41 COCC(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686495 CG On-Demand Anodyne IMDH_CRYPV 58 35 NC(=O)C1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686496 EF On-Demand Anodyne EPHX2 48 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880686498 FH On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880686500 FH On-Demand Anodyne EPHX2 22 42 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686502 GI On-Demand Anodyne CCR3 29 43 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686502 GI On-Demand Anodyne EPHX2 18 45 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686502 GI On-Demand Anodyne CACNA1I 66 37 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686504 GI On-Demand Anodyne CCR3 29 43 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686504 GI On-Demand Anodyne EPHX2 18 45 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686504 GI On-Demand Anodyne CACNA1I 66 37 Cc1noc(C)c1CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686515 EI On-Demand Anodyne NPY2R 16 40 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(F)c(C(F)F)c3)C2)nn1 ZINC000880686525 GH On-Demand Anodyne CCR3 59 35 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(F)c(C(F)F)c3)C2)nn1 ZINC000880686525 GH On-Demand Anodyne EPHX2 33 41 Cn1cc(CN2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cn1 ZINC000880686527 FF On-Demand Anodyne FAAH 24 46 C[C@@H](O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686531 DG On-Demand Anodyne CACNA1H 42 43 C[C@@H](O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686531 DG On-Demand Anodyne EPHX2 29 40 CC(=O)N(CC(=O)NN1CCc2ccccc2C1)c1ccccc1 ZINC000880686536 DE On-Demand Anodyne NOD2 40 34 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCSC1 ZINC000880686540 CG On-Demand Anodyne EPHX2 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCN2CCOCC2)CC1 ZINC000880686547 GH On-Demand Anodyne ITGAL 41 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCN2CCOCC2)CC1 ZINC000880686547 GH On-Demand Anodyne CCR3 38 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCN2CCOCC2)CC1 ZINC000880686547 GH On-Demand Anodyne CCR2 17 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCN2CCOCC2)CC1 ZINC000880686547 GH On-Demand Anodyne EPHX2 46 45 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686551 DF On-Demand Anodyne EPHX2 33 40 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880686551 DF On-Demand Anodyne MCHR1 29 41 O=C(NCCCN1CCCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686557 EG On-Demand Anodyne CCR3 41 42 O=C(NCCCN1CCCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686557 EG On-Demand Anodyne EPHX2 15 44 COCCN(Cc1cccnc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686577 FH On-Demand Anodyne ROCK2 32 41 C[C@@H](Cn1cncn1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686579 DF On-Demand Anodyne HIS3 83 36 O=C(NCCOCC1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686580 DG On-Demand Anodyne CCR3 32 41 CS(=O)(=O)C1CCC(C(=O)NN2CCc3ccccc3C2)CC1 ZINC000880686581 ED On-Demand Anodyne AKR1C3 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCSC1 ZINC000880686589 CG On-Demand Anodyne EPHX2 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(C2CCOCC2)C1=O ZINC000880686590 FF On-Demand Anodyne EPHX2 31 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(C2CCOCC2)C1=O ZINC000880686591 FF On-Demand Anodyne EPHX2 31 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCS(=O)(=O)C2(CCCCC2)C1 ZINC000880686597 GH On-Demand Anodyne CACNA1H 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCS(=O)(=O)C2(CCCCC2)C1 ZINC000880686597 GH On-Demand Anodyne EPHX2 29 40 CC[C@@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)C1CCOCC1 ZINC000880686599 EI On-Demand Anodyne NPY2R 19 41 O=C(NC[C@]1(O)CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686601 DF On-Demand Anodyne PRMT3 60 32 O=C(NC[C@@]1(O)CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686602 DF On-Demand Anodyne PRMT3 60 32 C#CC(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686608 CG On-Demand Mild IMDH_CRYPV 59 35 O=C(NCc1nnnn1C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686631 EE On-Demand Anodyne PRMT3 52 32 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686634 FF On-Demand Anodyne PDGFRB 40 37 O=C(NCCCOC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686636 EG On-Demand Anodyne CCR3 29 44 O=C(NCCCOC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686636 EG On-Demand Anodyne EPHX2 25 41 O=C(C[C@@H]1C=CS(=O)(=O)C1)Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2)s1 ZINC000880686645 IH On-Demand Anodyne RORC 20 52 O=C(C[C@H]1C=CS(=O)(=O)C1)Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2)s1 ZINC000880686646 IH On-Demand Anodyne RORC 20 52 O=C(NC[C@@H](CCO)c1ccccc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686647 FI On-Demand Anodyne SOAT1 21 41 O=C(NC[C@H](CCO)c1ccccc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686648 FI On-Demand Anodyne SOAT1 21 41 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880686652 FF On-Demand Anodyne MAPK1 48 38 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880686652 FF On-Demand Anodyne P2RY14 51 37 COC(=O)CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686655 FH On-Demand Anodyne CCR3 21 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CO)C1 ZINC000880686656 CF On-Demand Anodyne CCR3 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CO)C1 ZINC000880686656 CF On-Demand Anodyne EPHX2 30 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CO)C1 ZINC000880686657 CF On-Demand Anodyne CCR3 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CO)C1 ZINC000880686657 CF On-Demand Anodyne EPHX2 30 49 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686664 GH On-Demand Anodyne CACNA1H 64 40 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686664 GH On-Demand Anodyne EPHX2 26 42 Cn1cc(CN2CCCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cn1 ZINC000880686689 GG On-Demand Anodyne FAAH 20 43 Cn1cc(CN2CCCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cn1 ZINC000880686689 GG On-Demand Anodyne MCHR1 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCO)C1 ZINC000880686691 DG On-Demand Anodyne CCR3 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCO)C1 ZINC000880686691 DG On-Demand Anodyne EPHX2 17 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCO)C1 ZINC000880686693 DG On-Demand Anodyne CCR3 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCO)C1 ZINC000880686693 DG On-Demand Anodyne EPHX2 17 48 C[C@@H]([C@@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1)N1CCOCC1 ZINC000880686714 EF On-Demand Anodyne EPHX2 24 45 NC(=O)c1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686719 GF On-Demand Anodyne PDGFRB 52 42 NC(=O)c1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686719 GF On-Demand Anodyne TRPV1 19 57 NC(=O)c1cccnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686719 GF On-Demand Anodyne STAT6 58 34 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(CCn2cccn2)CC1 ZINC000880686723 GH On-Demand Anodyne CCR5 20 54 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(CCn2cccn2)CC1 ZINC000880686723 GH On-Demand Anodyne MCHR1 47 38 N#Cc1cccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686738 GJ On-Demand Mild CACNA1H 37 44 N#Cc1cccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686738 GJ On-Demand Mild HRH1 16 43 N#Cc1cccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686738 GJ On-Demand Mild CCR3 39 43 N#Cc1cccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686738 GJ On-Demand Mild EPHX2 32 57 N#Cc1cccc(OC2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1 ZINC000880686738 GJ On-Demand Mild MCHR1 39 40 Cc1coc(C(=O)NN2CCc3ccccc3C2)c1 ZINC000880686745 CE On-Demand Anodyne AKR1C3 20 40 Cc1coc(C(=O)NN2CCc3ccccc3C2)c1 ZINC000880686745 CE On-Demand Anodyne NOD2 42 36 CN(CC(=O)N1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686757 EE On-Demand Anodyne EPHX2 20 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](O)c3ccccc31)C2 ZINC000880686767 EG On-Demand Anodyne MTNR1A 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](O)c3ccccc31)C2 ZINC000880686767 EG On-Demand Anodyne MTNR1B 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](O)c3ccccc31)C2 ZINC000880686768 EG On-Demand Anodyne MTNR1A 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](O)c3ccccc31)C2 ZINC000880686768 EG On-Demand Anodyne MTNR1B 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@@H](O)c3ccccc31)C2 ZINC000880686769 EG On-Demand Anodyne MTNR1A 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@@H](O)c3ccccc31)C2 ZINC000880686769 EG On-Demand Anodyne MTNR1B 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)c3ccccc31)C2 ZINC000880686770 EG On-Demand Anodyne MTNR1A 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)c3ccccc31)C2 ZINC000880686770 EG On-Demand Anodyne MTNR1B 23 41 CSc1nccnc1C(=O)Nc1nc(CC(C)C)ns1 ZINC000880686772 DF On-Demand Anodyne MAP1 59 43 O=C(NCCCc1nnc2n1CCCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880686775 GH On-Demand Anodyne F2R 40 31 O=C(NCCCc1nnc2n1CCCCC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880686775 GH On-Demand Anodyne PRMT3 41 37 O=C(NCCCN1CCOC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686786 EF On-Demand Anodyne CCR3 39 44 O=C(NCCCN1CCOC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686786 EF On-Demand Anodyne EPHX2 21 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686787 FE On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686787 FE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686787 FE On-Demand Anodyne CTSK 20 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686787 FE On-Demand Anodyne CTSL 21 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686787 FE On-Demand Anodyne FPR1 48 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686788 FE On-Demand Anodyne PGC 50 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686788 FE On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686788 FE On-Demand Anodyne CTSK 20 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686788 FE On-Demand Anodyne CTSL 21 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCc2ccccc2C1 ZINC000880686788 FE On-Demand Anodyne FPR1 48 36 C=CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686799 EH On-Demand Mild CCR3 39 40 C=CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686799 EH On-Demand Mild EPHX2 50 42 C=CCN1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686799 EH On-Demand Mild CXCR3 22 45 O=C(NC[C@@H](O)C1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686805 EF On-Demand Anodyne PRMT3 25 47 O=C(NC[C@H](O)C1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686807 EF On-Demand Anodyne PRMT3 25 47 O=C(NCCCOC[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686816 EG On-Demand Anodyne CCR3 27 40 O=C(NCCCOC[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880686818 EG On-Demand Anodyne CCR3 27 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(F)(F)F)CC1 ZINC000880686823 EJ On-Demand Anodyne EPHX2 41 44 O=C1CC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CN1 ZINC000880686870 EF On-Demand Anodyne CACNA1H 46 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OCCO)C1 ZINC000880686877 EF On-Demand Anodyne EPHX2 19 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OCCO)C1 ZINC000880686879 EF On-Demand Anodyne EPHX2 19 44 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCCCO)C1CC1 ZINC000880686894 DH On-Demand Anodyne MCHR1 35 42 CSCC[C@@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686895 DI On-Demand Anodyne FPR1 38 41 CSCC[C@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880686896 DI On-Demand Anodyne FPR1 38 41 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)CN1CCN(C)CC1 ZINC000880686899 FF On-Demand Anodyne EPHX2 19 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCOCC2)C1 ZINC000880686905 EF On-Demand Anodyne EPHX2 29 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CCOCC2)C1 ZINC000880686905 EF On-Demand Anodyne L3MBTL3 56 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCOCC2)C1 ZINC000880686906 EF On-Demand Anodyne EPHX2 29 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CCOCC2)C1 ZINC000880686906 EF On-Demand Anodyne L3MBTL3 56 37 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880686909 FG On-Demand Anodyne EPHX2 52 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880686909 FG On-Demand Anodyne CXCR3 20 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880686910 FG On-Demand Anodyne EPHX2 52 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880686910 FG On-Demand Anodyne CXCR3 20 44 Cn1nccc1C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880686922 FH On-Demand Anodyne CACNA1H 44 37 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1N1CCOCC1 ZINC000880686928 FF On-Demand Anodyne EPHX2 16 40 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1N1CCOCC1 ZINC000880686929 FF On-Demand Anodyne EPHX2 16 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1N1CCOCC1 ZINC000880686930 FF On-Demand Anodyne EPHX2 16 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1N1CCOCC1 ZINC000880686931 FF On-Demand Anodyne EPHX2 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880686932 GG On-Demand Anodyne P2RX7 25 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@@H]1c1ncc[nH]1 ZINC000880686936 EI On-Demand Anodyne CPT1A 21 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@H]1c1ncc[nH]1 ZINC000880686937 EI On-Demand Anodyne CPT1A 21 42 O=C(NCCC(F)(F)F)Nc1ccc(F)c(C(F)F)c1 ZINC000880687017 DH On-Demand Anodyne PRMT3 45 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](N2CC=CC2)C1 ZINC000880687018 EG On-Demand Anodyne L3MBTL3 50 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](N2CC=CC2)C1 ZINC000880687019 EG On-Demand Anodyne L3MBTL3 50 36 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCS(=O)(=O)C1 ZINC000880687026 EE On-Demand Anodyne EPHX2 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCS(=O)(=O)C1 ZINC000880687027 EE On-Demand Anodyne EPHX2 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CCO)C1 ZINC000880687032 DF On-Demand Anodyne CCR3 22 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CCO)C1 ZINC000880687032 DF On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CCO)C1 ZINC000880687033 DF On-Demand Anodyne CCR3 22 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CCO)C1 ZINC000880687033 DF On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCC2CC2)CC1 ZINC000880687040 EI On-Demand Anodyne EPHX2 29 41 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880687049 EH On-Demand Anodyne HTR3A 35 44 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880687049 EH On-Demand Anodyne CCR3 26 40 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880687049 EH On-Demand Anodyne EPHX2 50 41 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880687049 EH On-Demand Anodyne CXCR3 21 43 COCCn1nc(C)c(NC(=O)Nc2ccc(F)c(C(F)F)c2)c1C ZINC000880687069 FH On-Demand Anodyne FPR2 51 39 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687071 EF On-Demand Anodyne CACNA1H 51 43 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687071 EF On-Demand Anodyne EPHX2 35 44 CNC(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687073 EG On-Demand Anodyne CCR2 15 40 CNC(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687073 EG On-Demand Anodyne EPHX2 27 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCCN2CCCC2)CC1 ZINC000880687079 GH On-Demand Anodyne EPHX2 27 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880687080 GF On-Demand Anodyne CCR3 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880687080 GF On-Demand Anodyne EPHX2 64 63 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880687080 GF On-Demand Anodyne CXCR3 18 42 COC(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCC1 ZINC000880687084 EH On-Demand Anodyne PRMT3 44 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCCC2)C1 ZINC000880687099 EH On-Demand Anodyne CCR3 49 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCCC2)C1 ZINC000880687099 EH On-Demand Anodyne CCR2 17 53 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCCC2)C1 ZINC000880687099 EH On-Demand Anodyne MCHR1 19 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880687100 EH On-Demand Anodyne CCR3 49 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880687100 EH On-Demand Anodyne CCR2 17 53 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCCC2)C1 ZINC000880687100 EH On-Demand Anodyne MCHR1 19 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687102 DF On-Demand Anodyne UL80 40 42 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687102 DF On-Demand Anodyne LGMN 63 36 CC[C@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687109 DG On-Demand Anodyne CCR3 23 40 CC[C@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687109 DG On-Demand Anodyne LEF 19 45 CC[C@@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687110 DG On-Demand Anodyne CCR3 23 40 CC[C@@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687110 DG On-Demand Anodyne LEF 19 45 COCCCOC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687113 FH On-Demand Anodyne HTR1B 15 40 CCC[C@](C)(CO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687115 DG On-Demand Anodyne IMDH_CRYPV 47 32 CN1CCC(N(C)CCN(C)C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687125 FG On-Demand Anodyne MCHR1 44 42 O=C(NCCCCN1CCC[C@@H]1CO)Nc1ccc(F)c(C(F)F)c1 ZINC000880687126 FG On-Demand Anodyne CCR3 51 46 O=C(NCCCCN1CCC[C@H]1CO)Nc1ccc(F)c(C(F)F)c1 ZINC000880687127 FG On-Demand Anodyne CCR3 51 46 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687128 FD On-Demand Anodyne EPHX2 25 41 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687129 FD On-Demand Anodyne EPHX2 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC(Cc2ccccc2)C1 ZINC000880687131 EI On-Demand Anodyne GRIN2B 45 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC(Cc2ccccc2)C1 ZINC000880687131 EI On-Demand Anodyne CCR3 67 46 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687137 EG On-Demand Anodyne EPHX2 22 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O[C@@H]2CCOC2)CC1 ZINC000880687143 FH On-Demand Anodyne EPHX2 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O[C@H]2CCOC2)CC1 ZINC000880687144 FH On-Demand Anodyne EPHX2 20 41 Cn1c(S)nnc1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687147 EF On-Demand Anodyne PRMT3 44 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@H]1CN1CCOCC1 ZINC000880687148 FG On-Demand Anodyne EPHX2 25 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@@H]1CN1CCOCC1 ZINC000880687149 FG On-Demand Anodyne EPHX2 25 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Nc2cccnn2)CC1 ZINC000880687150 FH On-Demand Anodyne FAAH 23 44 CC(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687182 CH On-Demand Anodyne IMDH_CRYPV 64 39 O=C(NCCCOCC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687191 FH On-Demand Anodyne CCR3 35 42 O=C(NCCCOCC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687191 FH On-Demand Anodyne EPHX2 21 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880687194 GI On-Demand Anodyne SMO 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880687194 GI On-Demand Anodyne ETHR 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880687195 GI On-Demand Anodyne SMO 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880687195 GI On-Demand Anodyne ETHR 41 39 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCN1C ZINC000880687203 DG On-Demand Anodyne EPHX2 51 40 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCN1C ZINC000880687203 DG On-Demand Anodyne CXCR3 19 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCOCC2)CC1 ZINC000880687211 FG On-Demand Anodyne ITGAL 40 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCOCC2)CC1 ZINC000880687211 FG On-Demand Anodyne HRH3 15 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C2CCOCC2)CC1 ZINC000880687211 FG On-Demand Anodyne EPHX2 25 47 CC[C@@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)c1nnc2n1CCCCC2 ZINC000880687213 GI On-Demand Anodyne CCR3 48 31 CC[C@@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)c1nnc2n1CCCCC2 ZINC000880687213 GI On-Demand Anodyne F2R 51 31 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)CN1CCOCC1 ZINC000880687215 EF On-Demand Anodyne EPHX2 31 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(CCOCC2)C1 ZINC000880687229 EI On-Demand Anodyne EPHX2 44 46 C[S@@](=O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687235 DF On-Demand Anodyne CCR3 31 43 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687237 CI On-Demand Anodyne CACNA1H 64 47 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687237 CI On-Demand Anodyne NPY5R 18 42 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687237 CI On-Demand Anodyne EPHX2 38 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2ccccn12 ZINC000880687248 EE On-Demand Anodyne FPR1 47 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2ccccn12 ZINC000880687249 EE On-Demand Anodyne FPR1 47 37 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687256 GH On-Demand Anodyne F2 42 40 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687256 GH On-Demand Anodyne XIAP 17 53 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687257 GH On-Demand Anodyne F2 42 40 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687257 GH On-Demand Anodyne XIAP 17 53 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCSC1 ZINC000880687266 DH On-Demand Anodyne EPHX2 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCSC1 ZINC000880687267 DH On-Demand Anodyne EPHX2 39 41 CC[C@@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)C(=O)N1CCOCC1 ZINC000880687279 FF On-Demand Anodyne EPHX2 34 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CCOCC2)CC1 ZINC000880687286 FG On-Demand Anodyne TACR2 23 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CCOCC2)CC1 ZINC000880687286 FG On-Demand Anodyne CCR3 17 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CC2CCOCC2)CC1 ZINC000880687286 FG On-Demand Anodyne CCR2 15 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)C1 ZINC000880687295 EH On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)C1 ZINC000880687295 EH On-Demand Anodyne EPHX2 46 53 O=C(NC[C@H]1CCC[C@@H]1O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687297 DG On-Demand Anodyne PRMT3 50 37 O=C(NC[C@H]1CCC[C@H]1O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687298 DG On-Demand Anodyne PRMT3 50 37 COC(=O)C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880687321 EF On-Demand Anodyne EPHX2 23 41 COC(=O)C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880687322 EF On-Demand Anodyne EPHX2 23 41 Cc1ccoc1C(=O)NCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687327 FH On-Demand Anodyne LEF 18 43 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687332 GH On-Demand Anodyne CCR3 56 38 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687332 GH On-Demand Anodyne EPHX2 61 47 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687332 GH On-Demand Anodyne CACNA1I 68 37 Cc1nsc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880687338 FG On-Demand Anodyne FAAH 17 51 CC[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880687416 CE On-Demand Anodyne NQO2 21 43 CC[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880687416 CE On-Demand Anodyne MTNR1A 24 46 CC[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880687416 CE On-Demand Anodyne MTNR1B 26 46 CC[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880687417 CE On-Demand Anodyne NQO2 21 43 CC[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880687417 CE On-Demand Anodyne MTNR1A 24 46 CC[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880687417 CE On-Demand Anodyne MTNR1B 26 46 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)CCN1CCOCC1 ZINC000880687418 FD On-Demand Anodyne CASR 71 54 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)CCN1CCOCC1 ZINC000880687418 FD On-Demand Anodyne EPHX2 26 45 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)CCN1CCOCC1 ZINC000880687418 FD On-Demand Anodyne MCHR1 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)CCN1CCOCC1 ZINC000880687418 FD On-Demand Anodyne STAT6 45 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CC=CC2)CC1 ZINC000880687438 EH On-Demand Anodyne CACNA1H 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CC=CC2)CC1 ZINC000880687438 EH On-Demand Anodyne EPHX2 15 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CC=CC2)CC1 ZINC000880687438 EH On-Demand Anodyne L3MBTL3 74 35 CC[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880687439 CD On-Demand Anodyne NQO2 33 43 CC[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880687439 CD On-Demand Anodyne MTNR1A 65 48 CC[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880687439 CD On-Demand Anodyne MTNR1B 57 48 CC[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880687440 CD On-Demand Anodyne NQO2 33 43 CC[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880687440 CD On-Demand Anodyne MTNR1A 65 48 CC[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880687440 CD On-Demand Anodyne MTNR1B 57 48 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880687442 FH On-Demand Anodyne CCR3 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880687442 FH On-Demand Anodyne EPHX2 52 50 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880687443 FH On-Demand Anodyne CCR3 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880687443 FH On-Demand Anodyne EPHX2 52 50 O=C(CN1CCCCS1(=O)=O)N[C@@H]1CCc2ccccc21 ZINC000880687447 DD On-Demand Anodyne HTR7 15 45 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)C1=O ZINC000880687454 FD On-Demand Anodyne CACNA1H 54 43 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687474 GH On-Demand Anodyne CCR3 38 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687474 GH On-Demand Anodyne EPHX2 33 44 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687475 GH On-Demand Anodyne CCR3 38 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687475 GH On-Demand Anodyne EPHX2 33 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC1 ZINC000880687478 CF On-Demand Anodyne EPHX2 54 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC1 ZINC000880687479 CF On-Demand Anodyne EPHX2 54 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](Cn2ccnn2)C1 ZINC000880687501 FG On-Demand Anodyne CCR3 15 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](Cn2ccnn2)C1 ZINC000880687502 FG On-Demand Anodyne CCR3 15 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(O)CCCC[C@H]2C1 ZINC000880687510 EH On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(O)CCCC[C@@H]2C1 ZINC000880687511 EH On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(O)CCCC[C@H]2C1 ZINC000880687512 EH On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(O)CCCC[C@@H]2C1 ZINC000880687513 EH On-Demand Anodyne CACNA1H 39 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687564 GI On-Demand Anodyne CCR3 38 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687564 GI On-Demand Anodyne EPHX2 31 45 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687565 GI On-Demand Anodyne CCR3 38 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687565 GI On-Demand Anodyne EPHX2 31 45 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687570 FH On-Demand Anodyne CCR3 61 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687570 FH On-Demand Anodyne EPHX2 38 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687571 FH On-Demand Anodyne CCR3 61 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687571 FH On-Demand Anodyne EPHX2 38 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687572 FH On-Demand Anodyne CCR3 61 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687572 FH On-Demand Anodyne EPHX2 38 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687573 FH On-Demand Anodyne CCR3 61 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687573 FH On-Demand Anodyne EPHX2 38 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(c2ccccn2)C1 ZINC000880687588 FH On-Demand Anodyne EPHX2 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(c2ccccn2)C1 ZINC000880687589 FH On-Demand Anodyne EPHX2 41 39 O=C(NCCc1cnc(C2CC2)nc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687595 FH On-Demand Anodyne PRMT3 62 37 Cc1coc(C(=O)N[C@@H]2CCc3ccccc32)c1 ZINC000880687745 BG On-Demand Anodyne BDKRB1 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]([C@@H]2CCOC2)C1 ZINC000880687746 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]([C@H]2CCOC2)C1 ZINC000880687747 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]([C@H]2CCOC2)C1 ZINC000880687748 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]([C@@H]2CCOC2)C1 ZINC000880687749 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CCO)CC1 ZINC000880687750 DD On-Demand Anodyne FAAH 15 43 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687757 GF On-Demand Anodyne CCR3 31 40 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687757 GF On-Demand Anodyne EPHX2 32 42 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687758 GF On-Demand Anodyne CCR3 31 40 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687758 GF On-Demand Anodyne EPHX2 32 42 C=CC(C)(C)CC(=O)N1CCC[C@H]1c1ccc(OC)c(F)c1 ZINC000880687762 DI On-Demand Mild ACKR3 51 31 C=CC(C)(C)CC(=O)N1CCC[C@@H]1c1ccc(OC)c(F)c1 ZINC000880687763 DI On-Demand Mild ACKR3 51 31 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCc3ccccc32)N1Cc1ccccc1 ZINC000880687771 FE On-Demand Anodyne XIAP 26 43 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCc3ccccc32)N1Cc1ccccc1 ZINC000880687771 FE On-Demand Anodyne BIRC3 31 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCc3ccccc32)N1Cc1ccccc1 ZINC000880687771 FE On-Demand Anodyne BIRC2 44 41 CC[C@@H](O)CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880687774 CE On-Demand Anodyne PDE4D 15 41 COc1ccc([C@@H]2CCCN2C(=O)COC2CC2)cc1F ZINC000880687775 CF On-Demand Anodyne CPT1A 64 39 COc1ccc([C@@H]2CCCN2C(=O)COC2CC2)cc1F ZINC000880687775 CF On-Demand Anodyne ACKR3 50 31 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687777 FE On-Demand Anodyne CCR3 71 41 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687777 FE On-Demand Anodyne CACNA1I 60 34 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687778 FE On-Demand Anodyne CCR3 71 41 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880687778 FE On-Demand Anodyne CACNA1I 60 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC2(CCC2)C1 ZINC000880687803 EH On-Demand Anodyne EPHX2 41 42 COC(=O)C1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687820 EE On-Demand Anodyne CACNA1H 72 44 COC(=O)C1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687820 EE On-Demand Anodyne S1PR2 29 42 COC(=O)C1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687820 EE On-Demand Anodyne EPHX2 29 40 C[C@H](CO)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687822 CF On-Demand Anodyne NPY5R 35 42 C[C@@H](CO)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687823 CF On-Demand Anodyne NPY5R 35 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC2(CCOCC2)C1 ZINC000880687828 FG On-Demand Anodyne EPHX2 44 43 CCc1noc(C)c1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880687836 DI On-Demand Anodyne NPY2R 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC(F)(F)CC1 ZINC000880687847 DI On-Demand Anodyne EPHX2 54 42 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC(F)(F)CC1 ZINC000880687847 DI On-Demand Anodyne CXCR3 16 41 CO[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687849 DH On-Demand Anodyne CACNA1H 40 39 CO[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687849 DH On-Demand Anodyne EPHX2 34 41 CC[C@@H](O)CNC(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880687856 DD On-Demand Anodyne KCNA3 18 41 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880687862 DG On-Demand Anodyne EPHX2 41 39 O=C(NCC[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687868 DH On-Demand Anodyne PRMT3 41 42 O=C(NCC[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687869 DH On-Demand Anodyne PRMT3 41 42 O=C(NCC[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687885 DG On-Demand Anodyne EPHX2 15 40 O=C(NCC[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687885 DG On-Demand Anodyne PRMT3 24 40 O=C(NCC[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687886 DG On-Demand Anodyne EPHX2 15 40 O=C(NCC[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687886 DG On-Demand Anodyne PRMT3 24 40 O=C(NO[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687901 DG On-Demand Anodyne EPHX2 16 41 O=C(NO[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687902 DG On-Demand Anodyne EPHX2 16 41 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(S(C)(=O)=O)CC1 ZINC000880687912 GF On-Demand Anodyne NPY5R 15 65 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(S(C)(=O)=O)CC1 ZINC000880687912 GF On-Demand Anodyne EPHX2 23 43 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(S(C)(=O)=O)CC1 ZINC000880687912 GF On-Demand Anodyne MCHR1 24 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](C2CCOCC2)C1 ZINC000880687922 EI On-Demand Anodyne EPHX2 23 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](C2CCOCC2)C1 ZINC000880687923 EI On-Demand Anodyne EPHX2 23 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC(F)(F)C1 ZINC000880687927 DI On-Demand Anodyne EPHX2 42 38 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC(F)(F)C1 ZINC000880687927 DI On-Demand Anodyne ENV 40 37 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC(F)(F)C1 ZINC000880687928 DI On-Demand Anodyne EPHX2 42 38 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC(F)(F)C1 ZINC000880687928 DI On-Demand Anodyne ENV 40 37 CC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880687931 EF On-Demand Anodyne LIMK1 17 42 CC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880687931 EF On-Demand Anodyne LIMK2 26 42 CC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H](C)C1 ZINC000880687932 EF On-Demand Anodyne LIMK1 17 42 CC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H](C)C1 ZINC000880687932 EF On-Demand Anodyne LIMK2 26 42 O=C(NCc1nncn1C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880687949 EG On-Demand Anodyne PRMT3 54 33 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687956 FF On-Demand Anodyne EPHX2 63 53 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687956 FF On-Demand Anodyne CXCR3 19 42 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880687956 FF On-Demand Anodyne CCR8 40 35 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880687964 FG On-Demand Anodyne EPHX2 52 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880687964 FG On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880687965 FG On-Demand Anodyne EPHX2 52 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880687965 FG On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880687966 FG On-Demand Anodyne EPHX2 52 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880687966 FG On-Demand Anodyne CXCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880687967 FG On-Demand Anodyne EPHX2 52 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880687967 FG On-Demand Anodyne CXCR3 19 41 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne ACE 29 41 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CELA1 19 41 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CTRA_BOVIN 47 31 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne TRY1_BOVIN 46 31 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne PREP 29 41 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CAPNS1 50 32 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CELA2A 40 31 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne LGMN 67 40 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CAPN1 56 39 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne CAPN2 102 36 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne KLK5 40 37 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne TPP2 23 44 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne SLC12A5 45 35 CC[C@@H](O)CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880687975 ED On-Demand Anodyne Q9NAW4_PLAFA 41 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCOCC2)C1 ZINC000880687976 EG On-Demand Anodyne EPHX2 41 51 O=C(COC1CC1)N[C@@H]1CCc2ccccc21 ZINC000880688002 BD On-Demand Anodyne BDKRB1 15 41 O=C(NCCc1nc[nH]n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688033 CE On-Demand Anodyne PRMT3 61 38 O=C(NCc1nc(C2CC2)cs1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688047 EI On-Demand Anodyne PRMT3 52 32 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688061 EG On-Demand Anodyne CACNA1H 36 40 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688061 EG On-Demand Anodyne HTR1D 17 40 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688061 EG On-Demand Anodyne HTR1B 17 40 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688061 EG On-Demand Anodyne EPHX2 41 41 CC(=O)OC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688061 EG On-Demand Anodyne SCD1 18 49 CC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688069 CI On-Demand Anodyne CCR3 31 45 CC[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688069 CI On-Demand Anodyne EPHX2 33 41 C#CCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688074 CH On-Demand Mild CCR3 15 40 CS(=O)(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688080 FF On-Demand Anodyne CACNA1H 35 42 CS(=O)(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688080 FF On-Demand Anodyne EPHX2 28 40 CC[C@@H](O)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880688083 CD On-Demand Anodyne GABRA1 16 53 CC[C@@H](O)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880688083 CD On-Demand Anodyne MPO 75 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne ACE 23 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne HTR7 18 51 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne KCNQ2 22 42 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne BDKRB1 31 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne XIAP 25 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCc2ccccc21 ZINC000880688107 EG On-Demand Anodyne BIRC2 41 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880688112 FH On-Demand Anodyne EPHX2 33 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880688113 FH On-Demand Anodyne EPHX2 33 41 CC[C@@H](O)CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880688123 DC On-Demand Anodyne XIAP 58 37 CN1[C@H]2CC[C@H]1CC(N1CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC1)C2 ZINC000880688137 GH On-Demand Anodyne CACNA1H 36 42 CN1[C@H]2CC[C@H]1CC(N1CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC1)C2 ZINC000880688137 GH On-Demand Anodyne GLRA1 40 32 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@@H](O)CC1 ZINC000880688138 DG On-Demand Anodyne EPHX2 56 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@@H](O)CC1 ZINC000880688138 DG On-Demand Anodyne CXCR3 15 40 C=CC(C)(C)CC(=O)N[C@@H]1CCc2ccccc21 ZINC000880688139 BG On-Demand Mild XIAP 19 41 O=C(NCc1nnc(S)n1C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688149 FG On-Demand Anodyne PRMT3 52 32 Cc1nc(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)sc1C ZINC000880688152 EI On-Demand Anodyne PRMT3 44 32 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688164 EF On-Demand Anodyne CCR3 31 41 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688164 EF On-Demand Anodyne EPHX2 56 61 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688164 EF On-Demand Anodyne CXCR3 19 42 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688165 EF On-Demand Anodyne CCR3 31 41 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688165 EF On-Demand Anodyne EPHX2 56 61 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688165 EF On-Demand Anodyne CXCR3 19 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCCC2)C1 ZINC000880688179 EH On-Demand Anodyne EPHX2 40 51 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne CTSK 19 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne CTSL 19 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne REN 53 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne GZMB 49 30 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne FPR1 47 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne XIAP 27 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688185 EF On-Demand Anodyne BIRC2 45 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne PGC 50 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne PAPA1_CARPA 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne CTSK 19 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne CTSL 19 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne REN 53 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne GZMB 49 30 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne FPR1 47 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne XIAP 27 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccccc21 ZINC000880688186 EF On-Demand Anodyne BIRC2 45 33 NC(=O)[C@@H]1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688187 EF On-Demand Anodyne EPHX2 40 40 NC(=O)[C@H]1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688188 EF On-Demand Anodyne EPHX2 40 40 NC(=O)[C@H]1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688189 EF On-Demand Anodyne EPHX2 40 40 NC(=O)[C@@H]1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688190 EF On-Demand Anodyne EPHX2 40 40 CN(CC1=CCCOC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880688207 DE On-Demand Anodyne MPO 45 36 Cc1ncc(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)s1 ZINC000880688212 EH On-Demand Anodyne PRMT3 44 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CCCCC2=O)CC1 ZINC000880688213 FH On-Demand Anodyne L3MBTL3 49 32 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880688214 GH On-Demand Anodyne SLC18A3 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880688214 GH On-Demand Anodyne EPHX2 54 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880688214 GH On-Demand Anodyne CXCR3 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880688215 GH On-Demand Anodyne SLC18A3 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880688215 GH On-Demand Anodyne EPHX2 54 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880688215 GH On-Demand Anodyne CXCR3 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880688216 GH On-Demand Anodyne SLC18A3 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880688216 GH On-Demand Anodyne EPHX2 54 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880688216 GH On-Demand Anodyne CXCR3 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880688217 GH On-Demand Anodyne SLC18A3 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880688217 GH On-Demand Anodyne EPHX2 54 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880688217 GH On-Demand Anodyne CXCR3 18 41 O=C(NCCCO[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688218 EG On-Demand Anodyne CCR3 19 42 O=C(NCCCO[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688219 EG On-Demand Anodyne CCR3 19 42 O=C(N[C@@H]1CCc2ccccc21)c1ccc(CN2CCOCC2)o1 ZINC000880688223 EF On-Demand Anodyne BDKRB1 37 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC2(CCCC2)C1 ZINC000880688228 EI On-Demand Anodyne EPHX2 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC2(CCCC2)C1 ZINC000880688229 EI On-Demand Anodyne EPHX2 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(F)F)CC1 ZINC000880688230 DI On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(F)F)CC1 ZINC000880688230 DI On-Demand Anodyne EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880688295 FH On-Demand Anodyne TRPV1 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880688295 FH On-Demand Anodyne EPHX2 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880688296 FH On-Demand Anodyne TRPV1 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880688296 FH On-Demand Anodyne EPHX2 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC2(CCOCC2)C1 ZINC000880688298 FH On-Demand Anodyne EPHX2 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC2(CCOCC2)C1 ZINC000880688299 FH On-Demand Anodyne EPHX2 26 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]1Cc1ccccc1 ZINC000880688307 EJ On-Demand Anodyne SIGMAR1 21 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]1Cc1ccccc1 ZINC000880688307 EJ On-Demand Anodyne CCR3 55 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]1Cc1ccccc1 ZINC000880688308 EJ On-Demand Anodyne SIGMAR1 21 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]1Cc1ccccc1 ZINC000880688308 EJ On-Demand Anodyne CCR3 55 41 CC[C@@H](O)CNC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880688314 CD On-Demand Anodyne HSP90AB1 15 42 CC[C@@H](O)CNC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880688314 CD On-Demand Anodyne PDK1 45 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccccn2)CC1 ZINC000880688317 EJ On-Demand Anodyne CACNA1H 47 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccccn2)CC1 ZINC000880688317 EJ On-Demand Anodyne GRM4 32 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccccn2)CC1 ZINC000880688317 EJ On-Demand Anodyne EPHX2 30 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccccn2)CC1 ZINC000880688317 EJ On-Demand Anodyne MCHR1 17 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccccn2)CC1 ZINC000880688317 EJ On-Demand Anodyne SMO 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC2(CCC2)C1 ZINC000880688327 EH On-Demand Anodyne EPHX2 27 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC2(CCC2)C1 ZINC000880688328 EH On-Demand Anodyne EPHX2 27 41 CS(=O)(=O)N[C@@H]1CCC[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688335 GF On-Demand Anodyne PRMT3 46 34 CS(=O)(=O)N[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688336 GF On-Demand Anodyne PRMT3 46 34 CS(=O)(=O)N[C@@H]1CCC[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688337 GF On-Demand Anodyne PRMT3 46 34 CS(=O)(=O)N[C@H]1CCC[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688338 GF On-Demand Anodyne PRMT3 46 34 CC[C@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688347 DI On-Demand Anodyne CACNA1H 58 43 CC[C@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688347 DI On-Demand Anodyne EPHX2 36 41 O=C(NCC1(CO)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688349 EF On-Demand Anodyne EPHX2 25 43 CC[C@@H](O)CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880688361 CD On-Demand Anodyne KCNQ2 70 36 COc1ccc([C@@H]2CCCN2C(=O)Cc2c(Br)cnn2C)cc1F ZINC000880688370 GG On-Demand Anodyne ACKR3 56 32 CN(C)CC1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688376 EI On-Demand Anodyne EPHX2 53 41 CN(C)CC1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688376 EI On-Demand Anodyne CXCR3 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(O)cc2)CC1 ZINC000880688377 GG On-Demand Anodyne NPY2R 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(O)cc2)CC1 ZINC000880688377 GG On-Demand Anodyne EPHX2 21 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(C(=O)c2ccc(O)cc2)CC1 ZINC000880688377 GG On-Demand Anodyne L3MBTL3 44 33 O=C(NCCCF)Nc1ccc(F)c(C(F)F)c1 ZINC000880688389 CG On-Demand Anodyne CCR3 20 41 O=C(NCCCF)Nc1ccc(F)c(C(F)F)c1 ZINC000880688389 CG On-Demand Anodyne LEF 17 47 CC[C@@](C)(CCO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688406 DG On-Demand Anodyne IMDH_CRYPV 47 32 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@H](CO)CC1 ZINC000880688410 DG On-Demand Anodyne EPHX2 51 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@H](CO)CC1 ZINC000880688410 DG On-Demand Anodyne CXCR3 15 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880688411 DG On-Demand Anodyne EPHX2 51 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880688411 DG On-Demand Anodyne CXCR3 15 40 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCCO)C1CC1 ZINC000880688415 DG On-Demand Anodyne MCHR1 36 42 CC[C@@H](O)CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880688421 DE On-Demand Anodyne INHA 73 39 CC[C@@H](O)CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880688421 DE On-Demand Anodyne TRPV1 16 47 CC[C@@H](O)CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880688421 DE On-Demand Anodyne MTNR1A 18 43 CC[C@@H](O)CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880688421 DE On-Demand Anodyne HCRTR2 16 40 COc1ccc([C@H](CO)N(C)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1 ZINC000880688423 FH On-Demand Anodyne NPY5R 33 40 COc1ccc([C@@H](CO)N(C)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1 ZINC000880688424 FH On-Demand Anodyne NPY5R 33 40 CN(CC1=CCCOC1)C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880688427 DE On-Demand Anodyne WNT3A 47 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(CCOC2)C1 ZINC000880688428 DG On-Demand Anodyne CACNA1H 40 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(CCOC2)C1 ZINC000880688428 DG On-Demand Anodyne EPHX2 42 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(CCOC2)C1 ZINC000880688429 DG On-Demand Anodyne CACNA1H 40 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(CCOC2)C1 ZINC000880688429 DG On-Demand Anodyne EPHX2 42 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC2)C1 ZINC000880688430 CI On-Demand Anodyne CACNA1H 44 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC2)C1 ZINC000880688430 CI On-Demand Anodyne EPHX2 39 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H]1CN1CCOCC1 ZINC000880688431 FG On-Demand Anodyne EPHX2 25 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H]1CN1CCOCC1 ZINC000880688432 FG On-Demand Anodyne EPHX2 25 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC(F)(F)C1 ZINC000880688434 DI On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC(F)(F)C1 ZINC000880688434 DI On-Demand Anodyne ENV 40 38 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC(F)(F)C1 ZINC000880688435 DI On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC(F)(F)C1 ZINC000880688435 DI On-Demand Anodyne ENV 40 38 COc1ccc([C@@H]2CCCN2C(=O)CC[C@H]2CC(C)(C)CO2)cc1F ZINC000880688443 EI On-Demand Anodyne ACKR3 50 31 COc1ccc([C@@H]2CCCN2C(=O)CC[C@@H]2CC(C)(C)CO2)cc1F ZINC000880688444 EI On-Demand Anodyne ACKR3 50 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCc1ccccc12 ZINC000880688462 GJ On-Demand Anodyne CACNA1H 46 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCc1ccccc12 ZINC000880688462 GJ On-Demand Anodyne NPY5R 33 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCc1ccccc12 ZINC000880688462 GJ On-Demand Anodyne MCHR1 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCc1ccccc12 ZINC000880688462 GJ On-Demand Anodyne TRPM8 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2ccccc2[C@@H]1CO ZINC000880688475 FH On-Demand Anodyne TRPM8 52 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2ccccc2[C@H]1CO ZINC000880688476 FH On-Demand Anodyne TRPM8 52 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880688481 FH On-Demand Anodyne EPHX2 25 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](Oc2ccccn2)C1 ZINC000880688482 FH On-Demand Anodyne EPHX2 25 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2c[nH]nc2C1 ZINC000880688484 DG On-Demand Anodyne MAPK1 49 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C2CCOCC2)CC1 ZINC000880688489 FI On-Demand Anodyne EPHX2 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC=CC1 ZINC000880688495 CH On-Demand Anodyne EPHX2 43 40 CC(C)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688496 DI On-Demand Anodyne CACNA1H 31 41 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688512 EG On-Demand Anodyne CACNA1H 50 43 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688512 EG On-Demand Anodyne EPHX2 37 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(Cc2ccccn2)C1=O ZINC000880688531 GG On-Demand Anodyne NPY1R 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(Cc2ccccn2)C1=O ZINC000880688531 GG On-Demand Anodyne EPHX2 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(Cc2ccccn2)C1=O ZINC000880688532 GG On-Demand Anodyne NPY1R 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(Cc2ccccn2)C1=O ZINC000880688532 GG On-Demand Anodyne EPHX2 16 40 N#Cc1cccc([C@@H]2CN(C(=O)Nc3ccc(F)c(C(F)F)c3)CCO2)c1 ZINC000880688536 GI On-Demand Mild CACNA1H 28 41 N#Cc1cccc([C@H]2CN(C(=O)Nc3ccc(F)c(C(F)F)c3)CCO2)c1 ZINC000880688537 GI On-Demand Mild CACNA1H 28 41 CN1CCC(C)(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688545 EH On-Demand Anodyne EPHX2 26 40 CN1CCC(C)(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688545 EH On-Demand Anodyne MCHR1 20 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCOC[C@H]2C1 ZINC000880688553 EE On-Demand Anodyne EPHX2 19 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN2CCOC[C@@H]2C1 ZINC000880688554 EE On-Demand Anodyne EPHX2 19 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(O)C[C@H]2C=C[C@H]1C2 ZINC000880688563 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(O)C[C@H]2C=C[C@H]1C2 ZINC000880688564 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(O)C[C@H]2C=C[C@H]1C2 ZINC000880688565 FD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(O)C[C@H]2C=C[C@H]1C2 ZINC000880688566 FD On-Demand Anodyne PAPA1_CARPA 35 41 CN1C(=O)NC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)C1=O ZINC000880688567 FE On-Demand Anodyne CACNA1H 70 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC2(CC2)C1 ZINC000880688570 DG On-Demand Anodyne EPHX2 42 44 Cc1nc(CN2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n[nH]1 ZINC000880688580 FF On-Demand Anodyne FAAH 17 42 COCCCN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@@H]1CCS(=O)(=O)C1 ZINC000880688587 GF On-Demand Anodyne MCHR1 25 40 COCCCN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@H]1CCS(=O)(=O)C1 ZINC000880688588 GF On-Demand Anodyne MCHR1 25 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2cccnc2)CC1 ZINC000880688598 EJ On-Demand Anodyne CACNA1H 53 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2cccnc2)CC1 ZINC000880688598 EJ On-Demand Anodyne CCR2 17 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2cccnc2)CC1 ZINC000880688598 EJ On-Demand Anodyne MCHR1 24 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OC(F)F)C1 ZINC000880688599 EH On-Demand Anodyne EPHX2 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OC(F)F)C1 ZINC000880688600 EH On-Demand Anodyne EPHX2 22 44 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1F ZINC000880688601 DH On-Demand Anodyne EPHX2 20 40 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1F ZINC000880688602 DH On-Demand Anodyne EPHX2 20 40 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1F ZINC000880688603 DH On-Demand Anodyne EPHX2 20 40 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H]1F ZINC000880688604 DH On-Demand Anodyne EPHX2 20 40 CCC1(O)CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688617 EH On-Demand Anodyne EPHX2 49 40 CCC1(O)CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688617 EH On-Demand Anodyne CXCR3 18 42 O=C(c1ccc(CN2CCOCC2)o1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880688628 GE On-Demand Anodyne CCR5 17 40 O=C(c1cnc(CC2CC2)s1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880688629 FG On-Demand Anodyne CCR5 19 40 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880688630 EE On-Demand Anodyne CCR5 17 42 COC(=O)CCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688638 EI On-Demand Anodyne CCR3 15 43 COC(=O)CCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688638 EI On-Demand Anodyne EPHX2 18 45 COC(=O)CCCCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688638 EI On-Demand Anodyne LEF 18 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880688639 GI On-Demand Anodyne EPHX2 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880688639 GI On-Demand Anodyne SCD1 18 44 O=C(c1cc(Br)ccc1C1CC1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880688644 GH On-Demand Anodyne L3MBTL3 53 37 O=C(c1cc(Br)ccc1C1CC1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880688645 GH On-Demand Anodyne L3MBTL3 53 37 Cn1ncc(NC(=O)Nc2ccc(F)c(C(F)F)c2)c1C1CC1 ZINC000880688671 DI On-Demand Anodyne HTR2A 41 40 Cn1ncc(NC(=O)Nc2ccc(F)c(C(F)F)c2)c1C1CC1 ZINC000880688671 DI On-Demand Anodyne FPR2 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880688673 FI On-Demand Anodyne EPHX2 37 42 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne HTR2A 21 45 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne CCR3 42 41 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne CHRNA7 21 45 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne F2R 40 30 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne EPHX2 37 59 O=C(NCCN1CCCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688679 EF On-Demand Anodyne MCHR1 18 41 CCOCCOC[C@H](O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688690 FE On-Demand Anodyne ADRB1 41 33 CCOCCOC[C@@H](O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688691 FE On-Demand Anodyne ADRB1 41 33 CC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688692 DG On-Demand Anodyne CACNA1H 65 45 CC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688692 DG On-Demand Anodyne NPY5R 17 40 CC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688692 DG On-Demand Anodyne S1PR2 28 41 CC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688692 DG On-Demand Anodyne EPHX2 30 40 CS(=O)(=O)[C@@H]1CCCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688698 FG On-Demand Anodyne EPHX2 19 40 COC[C@@H](C)n1ccc(NC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880688710 EH On-Demand Anodyne FPR2 42 37 C[C@@H]1CN(Cc2ccccc2)C[C@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880688712 EC On-Demand Reactive SIGMAR1 30 40 C[C@@H]1CN(Cc2ccccc2)C[C@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880688712 EC On-Demand Reactive TIMP3 42 31 O=C(NNC(=O)[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688714 DD On-Demand Reactive EPHX2 16 40 O=C(NNC(=O)[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688715 DD On-Demand Reactive EPHX2 16 40 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880688717 GF On-Demand Anodyne CCR5 18 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne PGC 48 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne CCKAR 49 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne CTSK 30 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne CTSL 26 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne TACR3 15 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne REN 62 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne CTSS 18 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688723 GF On-Demand Anodyne FPR1 51 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne PGC 48 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne CCKAR 49 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne CTSK 30 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne CTSL 26 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne TACR3 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne REN 62 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne CTSS 18 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688724 GF On-Demand Anodyne FPR1 51 39 CC[C@@H](O)CNC(=O)[C@H](CC(C)C)N(C)C(=O)OC(C)(C)C ZINC000880688729 DE On-Demand Anodyne ECE1 30 42 NS(=O)(=O)C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688736 FE On-Demand Anodyne CCR3 33 44 NS(=O)(=O)C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688737 FE On-Demand Anodyne CCR3 33 44 O=C(NC[C@@]1(O)C[C@H]2C=C[C@H]1C2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880688738 ED On-Demand Anodyne GABRA1 16 44 O=C(NC[C@]1(O)C[C@H]2C=C[C@H]1C2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880688739 ED On-Demand Anodyne GABRA1 16 44 O=C(NC[C@@H]1CC(=O)N(Cc2ccccc2)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688741 GH On-Demand Anodyne CCR3 45 37 O=C(NC[C@@H]1CC(=O)N(Cc2ccccc2)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688741 GH On-Demand Anodyne F2R 40 30 O=C(NC[C@H]1CC(=O)N(Cc2ccccc2)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688742 GH On-Demand Anodyne CCR3 45 37 O=C(NC[C@H]1CC(=O)N(Cc2ccccc2)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880688742 GH On-Demand Anodyne F2R 40 30 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)(F)C1 ZINC000880688750 CH On-Demand Anodyne CACNA1H 57 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)(F)C1 ZINC000880688750 CH On-Demand Anodyne EPHX2 37 46 O=C(COC1CC1)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688755 CD On-Demand Anodyne EPHX2 34 42 O=C(COC1CC1)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880688755 CD On-Demand Anodyne TNKS 54 39 CC[C@@H](O)CNC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880688757 GD On-Demand Anodyne GPR119 41 44 Cn1cc([C@H](CO)NC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880688790 EE On-Demand Anodyne MAPK1 36 42 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1N1CCN(C)CC1 ZINC000880688793 GG On-Demand Anodyne HTR1D 16 41 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1N1CCN(C)CC1 ZINC000880688793 GG On-Demand Anodyne HTR1B 18 41 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1N1CCN(C)CC1 ZINC000880688794 GG On-Demand Anodyne HTR1D 16 41 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1N1CCN(C)CC1 ZINC000880688794 GG On-Demand Anodyne HTR1B 18 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1N1CCN(C)CC1 ZINC000880688795 GG On-Demand Anodyne HTR1D 16 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1N1CCN(C)CC1 ZINC000880688795 GG On-Demand Anodyne HTR1B 18 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1N1CCN(C)CC1 ZINC000880688796 GG On-Demand Anodyne HTR1D 16 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1N1CCN(C)CC1 ZINC000880688796 GG On-Demand Anodyne HTR1B 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)(F)F)CC1 ZINC000880688797 FH On-Demand Anodyne CACNA1H 46 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)(F)F)CC1 ZINC000880688797 FH On-Demand Anodyne EPHX2 38 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)(F)F)CC1 ZINC000880688797 FH On-Demand Anodyne TRPM8 31 41 O=C1NC(=O)N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C[C@@H]12 ZINC000880688798 ED On-Demand Anodyne CACNA1H 40 39 O=C1NC(=O)N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C[C@H]12 ZINC000880688799 ED On-Demand Anodyne CACNA1H 40 39 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H](C)O1 ZINC000880688802 DH On-Demand Anodyne EPHX2 43 39 C[C@@H]1CC(NC(=O)Nc2ccc(F)c(C(F)F)c2)C[C@@H](C)O1 ZINC000880688804 DH On-Demand Anodyne EPHX2 43 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCO[C@]2(CCOC2)C1 ZINC000880688807 EG On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCO[C@@]2(CCOC2)C1 ZINC000880688808 EG On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCO[C@]2(CCOC2)C1 ZINC000880688809 EG On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCO[C@@]2(CCOC2)C1 ZINC000880688810 EG On-Demand Anodyne EPHX2 20 40 N#CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688811 DH On-Demand Mild EPHX2 25 42 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cc(C2CC2)[nH]n1 ZINC000880688820 DI On-Demand Anodyne CDK2 16 54 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1cc(C2CC2)[nH]n1 ZINC000880688820 DI On-Demand Anodyne PKNB 61 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@]2(CCOC2)C1 ZINC000880688826 EF On-Demand Anodyne EPHX2 38 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@]2(CCOC2)C1 ZINC000880688827 EF On-Demand Anodyne EPHX2 38 47 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688828 FF On-Demand Anodyne CCR3 18 41 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688828 FF On-Demand Anodyne EPHX2 57 43 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688829 FF On-Demand Anodyne CCR3 18 41 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688829 FF On-Demand Anodyne EPHX2 57 43 NC(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCC1 ZINC000880688841 EF On-Demand Anodyne PRMT3 63 34 NC(=O)C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688846 EF On-Demand Anodyne EPHX2 15 45 NC(=O)C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688847 EF On-Demand Anodyne EPHX2 15 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880688852 FI On-Demand Anodyne CACNA1H 60 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880688852 FI On-Demand Anodyne OPRL1 21 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880688852 FI On-Demand Anodyne CCR1 44 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880688852 FI On-Demand Anodyne EPHX2 34 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880688852 FI On-Demand Anodyne TRPM8 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(CC2)C1 ZINC000880688856 CI On-Demand Anodyne CACNA1H 36 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(CC2)C1 ZINC000880688856 CI On-Demand Anodyne EPHX2 37 49 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H](n3ccnn3)CC2)N1Cc1ccccc1 ZINC000880688865 GD On-Demand Anodyne PREP 65 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H](n3ccnn3)CC2)N1Cc1ccccc1 ZINC000880688866 GD On-Demand Anodyne PREP 65 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880688872 GI On-Demand Anodyne PDGFRB 53 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880688872 GI On-Demand Anodyne TRPV1 20 59 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880688872 GI On-Demand Anodyne RBP4 15 48 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688873 FG On-Demand Anodyne LIMK1 16 42 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688873 FG On-Demand Anodyne LIMK2 26 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OCC2CC2)C1 ZINC000880688877 EI On-Demand Anodyne EPHX2 20 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OCC2CC2)C1 ZINC000880688878 EI On-Demand Anodyne EPHX2 20 44 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880688885 FG On-Demand Anodyne L3MBTL3 70 40 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880688886 FG On-Demand Anodyne L3MBTL3 70 40 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCS1(=O)=O ZINC000880688887 FG On-Demand Anodyne CACNA1H 49 43 CSc1nnc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)s1 ZINC000880688896 EH On-Demand Anodyne PRMT3 59 33 Cn1nccc1CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688900 DF On-Demand Anodyne HTR2A 40 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccccn2)CC1 ZINC000880688905 FH On-Demand Anodyne CACNA1H 41 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccccn2)CC1 ZINC000880688905 FH On-Demand Anodyne PDGFRB 40 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2ccccn2)CC1 ZINC000880688905 FH On-Demand Anodyne FAAH 29 47 NC(=O)CN1C[C@@H](F)C[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688906 FD On-Demand Anodyne PRMT3 45 32 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880688911 GG On-Demand Anodyne SLC6A5 19 42 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880688911 GG On-Demand Anodyne EPHX2 51 43 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880688911 GG On-Demand Anodyne CXCR3 20 43 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880688911 GG On-Demand Anodyne MCHR1 16 41 O=C(NCCCO)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688913 FF On-Demand Anodyne EPHX2 21 41 CC(C)[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880688930 DH On-Demand Anodyne EPHX2 22 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@@H]2CCOC2)CC1 ZINC000880688942 EI On-Demand Anodyne EPHX2 23 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@H]2CCOC2)CC1 ZINC000880688943 EI On-Demand Anodyne EPHX2 23 41 CCc1nnc2n1C[C@@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880688962 FG On-Demand Anodyne EPHX2 33 40 CCc1nnc2n1C[C@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880688963 FG On-Demand Anodyne EPHX2 33 40 Cc1coc(C(=O)N[C@@H]2C[C@@H](Oc3ccccc3)C2)c1 ZINC000880688969 CF On-Demand Anodyne EPHX2 16 43 CCC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688986 EH On-Demand Anodyne CACNA1H 69 43 CCC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880688986 EH On-Demand Anodyne S1PR2 28 41 CO[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880688993 DH On-Demand Anodyne PRMT3 40 34 C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688997 DG On-Demand Anodyne CACNA1H 35 42 C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880688997 DG On-Demand Anodyne EPHX2 37 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(C1)OCCO2 ZINC000880689004 EG On-Demand Anodyne EPHX2 38 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2ncsc2C1 ZINC000880689026 EH On-Demand Anodyne P2RY14 47 35 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689048 DG On-Demand Anodyne CCR3 23 44 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689048 DG On-Demand Anodyne CACNA1I 42 34 O=C(NCCCNC(=O)C1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689054 EG On-Demand Anodyne CCR3 37 43 O=C(NCCCNC(=O)C1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689054 EG On-Demand Anodyne TBK1 81 41 O=C(c1cccc2nsnc12)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880689057 EE On-Demand Anodyne L3MBTL3 62 39 O=C(c1cccc2nsnc12)N1CCC[C@H](n2ccnn2)CC1 ZINC000880689058 EE On-Demand Anodyne L3MBTL3 62 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCN(C(=O)C2CC2)CC1 ZINC000880689064 FG On-Demand Anodyne EPHX2 30 43 C[C@@H](C1CC1)n1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)cn1 ZINC000880689074 EJ On-Demand Anodyne FPR2 42 36 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccncc1 ZINC000880689082 GH On-Demand Anodyne IMDH_CRYPV 48 32 COC(=O)C[C@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccncc1 ZINC000880689083 GH On-Demand Anodyne IMDH_CRYPV 48 32 O=C(CN1CCCCS1(=O)=O)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880689084 FD On-Demand Anodyne CCR5 17 41 O=C(NC[C@H]1CCn2ccnc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689090 EG On-Demand Anodyne CCR3 51 37 O=C(NC[C@@H]1CCn2ccnc2C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689091 EG On-Demand Anodyne CCR3 51 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2ncccc2F)CC1 ZINC000880689104 GI On-Demand Anodyne EPHX2 33 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2ncccc2F)CC1 ZINC000880689104 GI On-Demand Anodyne SCD1 17 49 O=C(NCCC1CC(O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689107 DG On-Demand Anodyne PRMT3 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2cn[nH]c2)CC1 ZINC000880689114 EH On-Demand Anodyne CACNA1H 43 39 O=C(NCC1CCN(C2CC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689117 EH On-Demand Anodyne CCR3 74 41 O=C(NCC1CCN(C2CC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689117 EH On-Demand Anodyne EPHX2 32 45 O=C(NCC1CCN(C2CC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689117 EH On-Demand Anodyne CACNA1I 68 37 COCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689120 EF On-Demand Anodyne CACNA1H 78 43 COCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689120 EF On-Demand Anodyne S1PR2 33 48 O=C(NC[C@@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689137 ED On-Demand Anodyne EPHX2 30 48 O=C(NC[C@@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689137 ED On-Demand Anodyne PIK3CB 27 40 O=C(NC[C@@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689137 ED On-Demand Anodyne HIPK3 17 41 O=C(NC[C@@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689137 ED On-Demand Anodyne MUSK 18 41 O=C(NC[C@@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689137 ED On-Demand Anodyne SRMS 23 41 O=C(NC[C@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689138 ED On-Demand Anodyne EPHX2 30 48 O=C(NC[C@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689138 ED On-Demand Anodyne PIK3CB 27 40 O=C(NC[C@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689138 ED On-Demand Anodyne HIPK3 17 41 O=C(NC[C@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689138 ED On-Demand Anodyne MUSK 18 41 O=C(NC[C@H](O)CN1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689138 ED On-Demand Anodyne SRMS 23 41 C[C@H](O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCCCC1 ZINC000880689140 EI On-Demand Anodyne PYGL 18 43 COC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689157 DH On-Demand Anodyne CACNA1H 74 45 COC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689157 DH On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCCO)CC1 ZINC000880689162 EF On-Demand Anodyne EPHX2 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OCCO)CC1 ZINC000880689162 EF On-Demand Anodyne SCD1 15 45 O=C(CNC(=O)Nc1ccc(F)c(C(F)F)c1)NCC1CC1 ZINC000880689174 DE On-Demand Anodyne PRMT3 47 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne CACNA1H 42 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne PDGFRB 56 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne TRPV1 23 64 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne NPY2R 46 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne FAAH 24 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne RBP4 15 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880689178 FH On-Demand Anodyne LIMK2 17 42 CN(CC1CCOCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689179 DH On-Demand Anodyne MCHR1 20 40 O=C(CCCc1cccs1)NNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689195 FI On-Demand Reactive PTPRF 20 44 O=C(NCCCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880689197 DG On-Demand Anodyne CCR3 17 44 O=C(NCCCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880689197 DG On-Demand Anodyne LEF 15 45 CC[C@@H](O)CNC(=O)c1ncsc1C1CC1 ZINC000880689203 BD On-Demand Anodyne MAP1 51 35 C[C@@H](CO)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689209 DG On-Demand Anodyne CCR3 20 40 C[C@@H](CO)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689209 DG On-Demand Anodyne LEF 18 44 C[C@H](CO)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689210 DG On-Demand Anodyne CCR3 20 40 C[C@H](CO)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689210 DG On-Demand Anodyne LEF 18 44 CN1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689215 DF On-Demand Anodyne HTR1D 16 48 CN1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689215 DF On-Demand Anodyne HTR1B 20 48 CN1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689215 DF On-Demand Anodyne HRH4 17 43 CN1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689215 DF On-Demand Anodyne EPHX2 21 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCOCC2)CC1 ZINC000880689222 FH On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCOCC2)CC1 ZINC000880689222 FH On-Demand Anodyne EPHX2 36 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCOCC2)CC1 ZINC000880689222 FH On-Demand Anodyne TRPM8 30 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@@H]2CCCO2)CC1 ZINC000880689224 EI On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC([C@H]2CCCO2)CC1 ZINC000880689225 EI On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CCOCC1 ZINC000880689227 EF On-Demand Anodyne MCHR1 34 41 Cn1cnc2c1CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880689228 DG On-Demand Anodyne MAPK1 47 37 COC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689235 EF On-Demand Anodyne CACNA1H 71 43 COC1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689235 EF On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCn2ccnc2C1 ZINC000880689263 DG On-Demand Anodyne EPHX2 42 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCn2ccnc2C1 ZINC000880689264 DG On-Demand Anodyne EPHX2 42 42 O=C(NCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880689269 CF On-Demand Anodyne CCR3 19 43 O=C(NCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880689269 CF On-Demand Anodyne LEF 19 46 O=C(c1ncsc1C1CC1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880689281 EG On-Demand Anodyne CCR5 22 42 O=C(NCC1(CO)CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689320 DG On-Demand Anodyne PRMT3 42 30 CN(C)CCCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689321 FI On-Demand Anodyne EPHX2 25 42 C=CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CC1 ZINC000880689333 CH On-Demand Mild MCHR1 31 40 O=C1NC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CO1 ZINC000880689341 EF On-Demand Anodyne CACNA1H 55 39 O=C1NC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CO1 ZINC000880689341 EF On-Demand Anodyne EPHX2 17 40 Cn1cc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)nn1 ZINC000880689343 CE On-Demand Anodyne PRMT3 61 34 C[C@@H]1CCOCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689355 DG On-Demand Anodyne EPHX2 17 42 C[C@H]1CCOCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689356 DG On-Demand Anodyne EPHX2 17 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccc(F)cn2)CC1 ZINC000880689381 FH On-Demand Anodyne PDGFRB 38 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccc(F)cn2)CC1 ZINC000880689381 FH On-Demand Anodyne DGAT1 35 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccc(F)cn2)CC1 ZINC000880689381 FH On-Demand Anodyne SLC27A1 40 39 CC[C@@H](O)CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689394 DC On-Demand Anodyne PAPA1_CARPA 42 54 CC[C@@H](O)CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689394 DC On-Demand Anodyne CTSK 17 49 CC[C@@H](O)CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689394 DC On-Demand Anodyne POLG_HCV1 22 40 CC[C@@H](O)CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689395 DC On-Demand Anodyne PAPA1_CARPA 42 54 CC[C@@H](O)CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689395 DC On-Demand Anodyne CTSK 17 49 CC[C@@H](O)CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880689395 DC On-Demand Anodyne POLG_HCV1 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC2(CCC2)C1 ZINC000880689399 DH On-Demand Anodyne EPHX2 40 51 CC[C@@H](O)CNC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880689404 DF On-Demand Anodyne LIPE 19 40 O=C(NCc1nnc2n1CCOC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880689433 EE On-Demand Anodyne EPHX2 21 41 O=C(NCc1nnc2n1CCOC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880689433 EE On-Demand Anodyne STAT6 41 35 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880689435 DE On-Demand Anodyne L3MBTL3 76 40 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880689436 DE On-Demand Anodyne L3MBTL3 76 40 O=C1NCC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)O1 ZINC000880689440 EF On-Demand Anodyne CACNA1H 48 39 O=C1NCC2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)O1 ZINC000880689440 EF On-Demand Anodyne TRPM8 31 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880689441 GJ On-Demand Anodyne CACNA1H 74 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880689441 GJ On-Demand Anodyne NPY5R 34 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880689441 GJ On-Demand Anodyne S1PR2 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880689441 GJ On-Demand Anodyne EPHX2 28 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880689441 GJ On-Demand Anodyne TRPM8 32 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H](CO)C1CCOCC1 ZINC000880689450 EF On-Demand Anodyne MAPK1 41 35 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H](CO)C1CCOCC1 ZINC000880689451 EF On-Demand Anodyne MAPK1 41 35 Cc1noc(C2(C)CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)n1 ZINC000880689452 FI On-Demand Anodyne CACNA1H 41 39 COCCn1ccc(NC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880689455 EG On-Demand Anodyne HTR2A 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CCCCC1 ZINC000880689464 EH On-Demand Anodyne PYGL 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CCCCC1 ZINC000880689464 EH On-Demand Anodyne MCHR1 38 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCOCC1 ZINC000880689485 DG On-Demand Anodyne EPHX2 51 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCOCC1 ZINC000880689486 DG On-Demand Anodyne EPHX2 51 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689487 EG On-Demand Anodyne CCR3 31 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689487 EG On-Demand Anodyne EPHX2 58 48 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689487 EG On-Demand Anodyne CXCR3 18 41 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689489 EG On-Demand Anodyne CCR3 31 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689489 EG On-Demand Anodyne EPHX2 58 48 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689489 EG On-Demand Anodyne CXCR3 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2cnccn2)CC1 ZINC000880689495 FH On-Demand Anodyne EPHX2 21 54 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Oc2cnccn2)CC1 ZINC000880689495 FH On-Demand Anodyne SCD1 17 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(CCO)C1=O ZINC000880689509 ED On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(CCO)C1=O ZINC000880689516 ED On-Demand Anodyne EPHX2 26 40 O=C(NCCCOCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880689521 DE On-Demand Anodyne CCR3 19 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880689526 FI On-Demand Anodyne CACNA1H 46 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880689526 FI On-Demand Anodyne CCR1 24 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880689526 FI On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880689526 FI On-Demand Anodyne EPHX2 32 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880689533 FI On-Demand Anodyne CACNA1H 46 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880689533 FI On-Demand Anodyne CCR1 24 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880689533 FI On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880689533 FI On-Demand Anodyne EPHX2 32 42 CN(C)C(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689537 FG On-Demand Anodyne EPHX2 23 40 CC[C@@H](O)CNC(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880689541 EE On-Demand Anodyne CTSK 17 43 CC[C@@H](O)CNC(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880689541 EE On-Demand Anodyne ECE1 26 40 CC[C@@H](O)CNC(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880689543 EE On-Demand Anodyne CTSK 17 43 CC[C@@H](O)CNC(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880689543 EE On-Demand Anodyne ECE1 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H](c1cccnc1)C1CC1 ZINC000880689552 EI On-Demand Anodyne NAMPT 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H](c1cccnc1)C1CC1 ZINC000880689554 EI On-Demand Anodyne NAMPT 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(F)(F)C1 ZINC000880689560 CH On-Demand Anodyne EPHX2 47 39 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(F)(F)C1 ZINC000880689560 CH On-Demand Anodyne ENV 43 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880689562 GH On-Demand Anodyne CACNA1H 43 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880689562 GH On-Demand Anodyne EPHX2 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880689564 GH On-Demand Anodyne CACNA1H 43 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880689564 GH On-Demand Anodyne EPHX2 30 40 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@H](n2ccnn2)CC1 ZINC000880689565 FE On-Demand Anodyne L3MBTL3 52 35 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880689566 FE On-Demand Anodyne L3MBTL3 52 35 O=C(NOC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689581 DF On-Demand Anodyne EPHX2 23 42 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689589 EH On-Demand Anodyne EPHX2 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne GRIN2B 68 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne CCR3 63 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne CHRNA7 57 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne C3AR1 45 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne FAAH 21 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne ACHP_LYMST 25 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880689609 FJ On-Demand Anodyne NAMPT 49 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880689612 GJ On-Demand Anodyne CACNA1H 52 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880689612 GJ On-Demand Anodyne EPHX2 29 41 O=C(NCC1(CO)CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689618 DG On-Demand Anodyne PRMT3 43 31 O=C(NCC(=O)N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689624 ED On-Demand Anodyne EPHX2 39 54 O=C(NCC(=O)N1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689624 ED On-Demand Anodyne PRMT3 33 45 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689625 ED On-Demand Anodyne CACNA1H 34 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cn2cncn2)CC1 ZINC000880689661 FG On-Demand Anodyne EPHX2 15 40 COC(=O)c1cn([C@@H]2CCCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)nn1 ZINC000880689673 GG On-Demand Anodyne CCR3 17 42 COC[C@@H](O)CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689675 DE On-Demand Anodyne ADRB1 43 35 COC(=O)c1cn([C@H]2CCCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)nn1 ZINC000880689676 GG On-Demand Anodyne CCR3 17 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC2(C1)OCCO2 ZINC000880689677 EH On-Demand Anodyne EPHX2 28 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC2(C1)OCCO2 ZINC000880689679 EH On-Demand Anodyne EPHX2 28 43 N#CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689687 CG On-Demand Mild ADRB1 41 35 N#CCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689687 CG On-Demand Mild CCR3 19 40 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689693 GJ On-Demand Anodyne NPY2R 52 36 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689693 GJ On-Demand Anodyne CCR2 15 41 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689693 GJ On-Demand Anodyne EPHX2 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC2(CCCC2)C1 ZINC000880689696 EI On-Demand Anodyne EPHX2 41 42 CCC1(CC)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880689700 FH On-Demand Anodyne NPY2R 41 32 CCC1(CC)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880689703 FH On-Demand Anodyne NPY2R 41 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCCCC2)C1 ZINC000880689709 DJ On-Demand Anodyne CACNA1H 35 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCCCC2)C1 ZINC000880689709 DJ On-Demand Anodyne EPHX2 27 43 Cn1nnc(C(=O)N2CC[C@H](c3ccccc3)[C@H](CO)C2)n1 ZINC000880689712 DC On-Demand Anodyne SLC6A3 15 44 C[C@@H](O)C(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689733 CG On-Demand Anodyne FPR2 44 35 C[C@@H](O)C(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689733 CG On-Demand Anodyne IMDH_CRYPV 62 37 CC(C)(CS(C)(=O)=O)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689741 EF On-Demand Anodyne IMDH_CRYPV 48 32 CO[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1C ZINC000880689742 DH On-Demand Anodyne EPHX2 17 40 CO[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1C ZINC000880689746 DH On-Demand Anodyne EPHX2 17 40 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689747 GH On-Demand Anodyne CCR3 63 39 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689747 GH On-Demand Anodyne F2R 53 33 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689747 GH On-Demand Anodyne MCHR1 31 41 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689749 GH On-Demand Anodyne CCR3 63 39 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689749 GH On-Demand Anodyne F2R 53 33 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689749 GH On-Demand Anodyne MCHR1 31 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H](O)CC(F)(F)C1 ZINC000880689752 DF On-Demand Anodyne CACNA1H 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H](O)CC(F)(F)C1 ZINC000880689754 DF On-Demand Anodyne CACNA1H 33 40 NC(=O)CCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880689755 EG On-Demand Anodyne EPHX2 28 43 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CCC1 ZINC000880689760 DG On-Demand Anodyne MCHR1 39 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(O)C[C@H]3C=C[C@H]1C3)C2 ZINC000880689763 EE On-Demand Anodyne MTNR1A 37 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(O)C[C@H]3C=C[C@H]1C3)C2 ZINC000880689763 EE On-Demand Anodyne MTNR1B 34 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880689765 GJ On-Demand Anodyne CACNA1H 54 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880689765 GJ On-Demand Anodyne S1PR2 33 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880689765 GJ On-Demand Anodyne EPHX2 26 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(O)C[C@H]3C=C[C@H]1C3)C2 ZINC000880689766 EE On-Demand Anodyne MTNR1A 37 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(O)C[C@H]3C=C[C@H]1C3)C2 ZINC000880689766 EE On-Demand Anodyne MTNR1B 34 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](Cc2ccncc2)C1 ZINC000880689768 EI On-Demand Anodyne GRIN2B 50 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](Cc2ccncc2)C1 ZINC000880689768 EI On-Demand Anodyne CCR3 93 49 CC(C)C1(O)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689769 DF On-Demand Anodyne CACNA1H 27 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880689770 EI On-Demand Anodyne GRIN2B 50 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880689770 EI On-Demand Anodyne CCR3 93 49 C[C@@H]1CN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCO1 ZINC000880689783 FG On-Demand Anodyne CCR3 62 48 C[C@@H]1CN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCO1 ZINC000880689783 FG On-Demand Anodyne CHRNA7 20 44 C[C@@H]1CN(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCO1 ZINC000880689783 FG On-Demand Anodyne EPHX2 25 41 Cc1cnc(Cl)c(C(=O)N2CC[C@H](c3ccccc3)[C@H](CO)C2)c1 ZINC000880689786 EG On-Demand Anodyne CCR5 23 44 Cc1cc(N2CCC[C@H](NC(=O)Nc3ccc(F)c(C(F)F)c3)C2)n(C)n1 ZINC000880689799 GH On-Demand Anodyne CCR3 61 33 Cc1cc(N2CCC[C@H](NC(=O)Nc3ccc(F)c(C(F)F)c3)C2)n(C)n1 ZINC000880689799 GH On-Demand Anodyne EPHX2 30 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689838 DE On-Demand Anodyne PAPA1_CARPA 42 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689838 DE On-Demand Anodyne CTSK 18 50 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689838 DE On-Demand Anodyne POLG_HCV1 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689839 DE On-Demand Anodyne PAPA1_CARPA 42 52 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689839 DE On-Demand Anodyne CTSK 18 50 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCC(C)(C)F ZINC000880689839 DE On-Demand Anodyne POLG_HCV1 22 40 C[C@@]1(C#N)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689840 DH On-Demand Mild EPHX2 30 46 CC(CO)(CO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880689842 CD On-Demand Anodyne IMDH_CRYPV 58 34 CC[C@@H](O)CNC(=O)c1ccccc1OCCN(C)C(=O)OC(C)(C)C ZINC000880689847 FE On-Demand Anodyne HCN1 54 32 CC[C@@H](O)CNC(=O)c1ccccc1OCCN(C)C(=O)OC(C)(C)C ZINC000880689847 FE On-Demand Anodyne HCN4 41 32 COc1ccccc1-c1ccc(C(=O)NC[C@]2(O)C[C@H]3C=C[C@H]2C3)c(O)n1 ZINC000880689850 FF On-Demand Anodyne KCNA3 43 37 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(O)C[C@H]3C=C[C@H]2C3)c(O)n1 ZINC000880689851 FF On-Demand Anodyne KCNA3 43 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCCO)CC1 ZINC000880689861 EH On-Demand Anodyne EPHX2 31 47 O=C(c1ccc(CN2CCOCC2)o1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880689884 FD On-Demand Anodyne L3MBTL3 25 41 O=C(c1ccc(CN2CCOCC2)o1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880689885 FD On-Demand Anodyne L3MBTL3 25 41 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1ccn(CC(=O)N2CCOCC2)n1 ZINC000880689887 GE On-Demand Anodyne EPHX2 24 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncc(F)cn2)CC1 ZINC000880689891 FG On-Demand Anodyne PDGFRB 47 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncc(F)cn2)CC1 ZINC000880689891 FG On-Demand Anodyne FAAH 21 41 O=C(NCC(F)(F)F)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689893 GG On-Demand Anodyne MAPK1 21 40 O=C(NCC(F)(F)F)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689893 GG On-Demand Anodyne EPHX2 41 40 O=C(NCC(F)(F)F)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689894 GG On-Demand Anodyne MAPK1 21 40 O=C(NCC(F)(F)F)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689894 GG On-Demand Anodyne EPHX2 41 40 Cn1ccnc(N2CCC(NC(=O)Nc3ccc(F)c(C(F)F)c3)CC2)c1=O ZINC000880689898 GF On-Demand Anodyne EPHX2 46 39 COc1cc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)ncn1 ZINC000880689906 GF On-Demand Anodyne PDGFRB 66 46 COc1cc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)ncn1 ZINC000880689906 GF On-Demand Anodyne LIMK2 19 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H](O)C[C@H]1CO ZINC000880689907 DD On-Demand Anodyne SPHK2 43 30 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H](O)C[C@H]1CO ZINC000880689908 DD On-Demand Anodyne SPHK2 43 30 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCS1 ZINC000880689921 DI On-Demand Anodyne SCD1 16 40 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCS1 ZINC000880689922 DI On-Demand Anodyne SCD1 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCOCC2)C1 ZINC000880689923 FF On-Demand Anodyne CCR3 30 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCOCC2)C1 ZINC000880689923 FF On-Demand Anodyne CCR2 15 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCOCC2)C1 ZINC000880689923 FF On-Demand Anodyne EPHX2 34 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880689924 FF On-Demand Anodyne CCR3 30 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880689924 FF On-Demand Anodyne CCR2 15 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880689924 FF On-Demand Anodyne EPHX2 34 41 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1O ZINC000880689929 DF On-Demand Anodyne EPHX2 24 40 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1O ZINC000880689930 DF On-Demand Anodyne EPHX2 24 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@H]1O ZINC000880689931 DF On-Demand Anodyne EPHX2 24 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[C@@H]1O ZINC000880689932 DF On-Demand Anodyne EPHX2 24 40 COC[C@@H]1CCCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689940 EI On-Demand Anodyne CCR3 30 46 COC[C@@H]1CCCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689940 EI On-Demand Anodyne EPHX2 23 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880689942 GJ On-Demand Anodyne CACNA1H 68 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880689942 GJ On-Demand Anodyne S1PR2 30 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880689942 GJ On-Demand Anodyne EPHX2 26 43 O=C(NCCC1CS(=O)(=O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689946 EE On-Demand Anodyne PRMT3 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880689949 FI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880689949 FI On-Demand Anodyne EPHX2 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880689950 FI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880689950 FI On-Demand Anodyne EPHX2 31 40 CCNC(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCC1 ZINC000880689952 EG On-Demand Anodyne PRMT3 51 31 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne PIK3CA 44 42 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne PIK3CD 35 44 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne MTOR 64 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne EPHX2 30 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne PIK3CB 71 44 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880689953 GG On-Demand Anodyne STAT6 58 37 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880689954 EF On-Demand Anodyne CCR5 15 40 N#C[C@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689961 DG On-Demand Mild CACNA1H 44 42 N#C[C@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689961 DG On-Demand Mild EPHX2 32 43 N#C[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689962 DG On-Demand Mild CACNA1H 44 42 N#C[C@@]1(F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689962 DG On-Demand Mild EPHX2 32 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(c2cccnn2)CC1 ZINC000880689969 FG On-Demand Anodyne EPHX2 45 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@@H]1CCO ZINC000880689982 DG On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@@H]1CCO ZINC000880689983 DG On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@H]1CCO ZINC000880689984 DG On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H]1CCO ZINC000880689985 DG On-Demand Anodyne CCR3 28 42 Cn1cnc2c(c1=O)CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880689987 FE On-Demand Anodyne MAPK1 45 35 Cn1cnc2c(c1=O)CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880689987 FE On-Demand Anodyne P2RY14 47 35 CN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689993 DF On-Demand Anodyne CCR3 91 44 CN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689993 DF On-Demand Anodyne EPHX2 38 42 CN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689993 DF On-Demand Anodyne MCHR1 20 42 CN1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689993 DF On-Demand Anodyne CACNA1I 76 36 CN1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689994 DF On-Demand Anodyne CCR3 91 44 CN1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689994 DF On-Demand Anodyne EPHX2 38 42 CN1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689994 DF On-Demand Anodyne MCHR1 20 42 CN1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880689994 DF On-Demand Anodyne CACNA1I 76 36 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690005 FF On-Demand Anodyne CCR3 69 41 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690005 FF On-Demand Anodyne EPHX2 28 41 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690005 FF On-Demand Anodyne MCHR1 21 40 O=C(NCC1(N2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690012 EF On-Demand Anodyne EPHX2 31 46 O=C(NCC1(N2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690012 EF On-Demand Anodyne HCN1 56 37 O=C(NCC1(N2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690012 EF On-Demand Anodyne HCN4 47 30 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880690019 FH On-Demand Anodyne CACNA1H 64 41 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880690020 FH On-Demand Anodyne CACNA1H 64 41 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880690021 FH On-Demand Anodyne CACNA1H 64 41 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880690022 FH On-Demand Anodyne CACNA1H 64 41 O=C(NCC1OCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690025 DF On-Demand Anodyne PRMT3 44 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCSC2(CCOCC2)C1 ZINC000880690026 FH On-Demand Anodyne EPHX2 39 40 O=C(c1cc2ccccc2cc1F)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690034 EG On-Demand Anodyne L3MBTL3 63 40 O=C(c1cc2ccccc2cc1F)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690035 EG On-Demand Anodyne L3MBTL3 63 40 C[C@@](O)(C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1)C(F)(F)F ZINC000880690037 GI On-Demand Anodyne EPHX2 32 42 O=C(c1cccn2nccc12)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690042 DD On-Demand Anodyne L3MBTL3 63 41 O=C(c1cccn2nccc12)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690043 DD On-Demand Anodyne L3MBTL3 63 41 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690046 GG On-Demand Anodyne PIK3CA 40 38 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690046 GG On-Demand Anodyne MTOR 74 39 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690046 GG On-Demand Anodyne STAT6 63 40 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690046 GG On-Demand Anodyne NAMPT 43 43 C[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880690052 EF On-Demand Anodyne LIMK1 16 40 C[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880690052 EF On-Demand Anodyne LIMK2 28 40 C[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H](C)C1 ZINC000880690053 EF On-Demand Anodyne LIMK1 16 40 C[C@H](O)CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H](C)C1 ZINC000880690053 EF On-Demand Anodyne LIMK2 28 40 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690055 FG On-Demand Anodyne CACNA1H 45 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCCCC2)C1 ZINC000880690056 FI On-Demand Anodyne CCR3 48 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CN2CCCCC2)C1 ZINC000880690056 FI On-Demand Anodyne CCR2 15 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880690057 FI On-Demand Anodyne CCR3 48 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880690057 FI On-Demand Anodyne CCR2 15 52 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCC[C@@H]1O ZINC000880690064 DG On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCC[C@H]1O ZINC000880690065 DG On-Demand Anodyne EPHX2 26 40 O=C(COC1CC1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880690072 CD On-Demand Anodyne SLC6A3 15 43 O=C(COC1CC1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880690072 CD On-Demand Anodyne CCR5 22 40 O=C(NOC1CCCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690075 DI On-Demand Anodyne EPHX2 19 40 O=C(c1c[nH]cc1C1CC1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690083 CE On-Demand Anodyne L3MBTL3 52 36 O=C(c1c[nH]cc1C1CC1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690084 CE On-Demand Anodyne L3MBTL3 52 36 O=C(NCCC[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690086 EI On-Demand Anodyne CCR3 35 40 O=C(NCCC[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690086 EI On-Demand Anodyne PRMT3 40 39 O=C(NCCC[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690087 EI On-Demand Anodyne CCR3 35 40 O=C(NCCC[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690087 EI On-Demand Anodyne PRMT3 40 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCO[C@@H](C2CC2)C1 ZINC000880690088 EH On-Demand Anodyne EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCO[C@H](C2CC2)C1 ZINC000880690089 EH On-Demand Anodyne EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCO[C@H](C2CC2)C1 ZINC000880690090 EH On-Demand Anodyne EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCO[C@@H](C2CC2)C1 ZINC000880690091 EH On-Demand Anodyne EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)F)CC1 ZINC000880690094 EG On-Demand Anodyne CACNA1H 56 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)F)CC1 ZINC000880690094 EG On-Demand Anodyne NPY5R 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)F)CC1 ZINC000880690094 EG On-Demand Anodyne S1PR2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(C(F)F)CC1 ZINC000880690094 EG On-Demand Anodyne EPHX2 31 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCC(F)(F)C1 ZINC000880690124 DG On-Demand Anodyne EPHX2 41 41 O=C(CCCCCc1ccc(O)cc1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690126 FG On-Demand Anodyne PREP 40 37 O=C(CCCCCc1ccc(O)cc1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690127 FG On-Demand Anodyne PREP 40 37 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690129 DH On-Demand Anodyne CACNA1H 38 40 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690129 DH On-Demand Anodyne EPHX2 34 47 Cc1noc(C)c1C(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690134 EI On-Demand Anodyne IMDH_CRYPV 54 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CNC(=O)C(F)(F)F)C1 ZINC000880690150 GH On-Demand Anodyne CCR3 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CNC(=O)C(F)(F)F)C1 ZINC000880690150 GH On-Demand Anodyne EPHX2 21 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CNC(=O)C(F)(F)F)C1 ZINC000880690150 GH On-Demand Anodyne CACNA1I 44 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CNC(=O)C(F)(F)F)C1 ZINC000880690151 GH On-Demand Anodyne CCR3 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CNC(=O)C(F)(F)F)C1 ZINC000880690151 GH On-Demand Anodyne EPHX2 21 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CNC(=O)C(F)(F)F)C1 ZINC000880690151 GH On-Demand Anodyne CACNA1I 44 33 CS(=O)(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690155 GF On-Demand Anodyne CACNA1H 31 40 CS(=O)(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690155 GF On-Demand Anodyne CCR3 23 41 CS(=O)(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690155 GF On-Demand Anodyne EPHX2 44 43 CS(=O)(=O)NCC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690155 GF On-Demand Anodyne CACNA1I 41 33 COCC1(NC(=O)Nc2ccc(F)c(C(F)F)c2)CCOCC1 ZINC000880690157 EG On-Demand Anodyne EPHX2 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880690164 GH On-Demand Anodyne CHRNA4 26 45 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)CN1 ZINC000880690176 EF On-Demand Anodyne CACNA1H 42 39 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)CN1 ZINC000880690176 EF On-Demand Anodyne EPHX2 31 46 O=C1C[C@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)CN1 ZINC000880690177 EF On-Demand Anodyne CACNA1H 42 39 O=C1C[C@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)CN1 ZINC000880690177 EF On-Demand Anodyne EPHX2 31 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCO2)CC1 ZINC000880690184 DH On-Demand Anodyne CACNA1H 45 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCO2)CC1 ZINC000880690184 DH On-Demand Anodyne EPHX2 37 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCO2)CC1 ZINC000880690184 DH On-Demand Anodyne TRPM8 32 44 O=C(NCCCCF)Nc1ccc(F)c(C(F)F)c1 ZINC000880690185 CH On-Demand Anodyne CCR3 20 44 O=C(NCCCCF)Nc1ccc(F)c(C(F)F)c1 ZINC000880690185 CH On-Demand Anodyne LEF 25 47 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(N2CCCCC2)C1 ZINC000880690196 EH On-Demand Anodyne EPHX2 43 44 O=C(NCc1nc(C2CC2)n[nH]1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690202 EG On-Demand Anodyne PRMT3 51 32 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880690206 DG On-Demand Anodyne CCR3 16 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880690206 DG On-Demand Anodyne EPHX2 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880690206 DG On-Demand Anodyne PTGES 17 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H](CO)C1 ZINC000880690207 DG On-Demand Anodyne CCR3 16 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H](CO)C1 ZINC000880690207 DG On-Demand Anodyne EPHX2 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H](CO)C1 ZINC000880690207 DG On-Demand Anodyne PTGES 17 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@H](CO)C1 ZINC000880690208 DG On-Demand Anodyne CCR3 16 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@H](CO)C1 ZINC000880690208 DG On-Demand Anodyne EPHX2 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCC[C@H](CO)C1 ZINC000880690208 DG On-Demand Anodyne PTGES 17 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@@H](CO)C1 ZINC000880690209 DG On-Demand Anodyne CCR3 16 44 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@@H](CO)C1 ZINC000880690209 DG On-Demand Anodyne EPHX2 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@@H](CO)C1 ZINC000880690209 DG On-Demand Anodyne PTGES 17 44 O=C(NCCCc1nccs1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690215 EH On-Demand Anodyne PRMT3 46 34 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne HRH2 25 44 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne HTR2C 16 41 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne CCR3 64 54 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne CHRNA7 29 62 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne F2R 54 33 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne HNMT 45 35 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne EPHX2 35 52 O=C(NCCCCCN1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690218 EI On-Demand Anodyne MCHR1 37 44 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880690219 FE On-Demand Anodyne EPHX2 19 40 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880690223 FE On-Demand Anodyne EPHX2 19 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC2)S(=O)(=O)CC1 ZINC000880690246 GG On-Demand Anodyne CACNA1H 42 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690247 DE On-Demand Anodyne MAPK1 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@]2(CCSC2)C1 ZINC000880690251 EJ On-Demand Anodyne EPHX2 29 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@]2(CCSC2)C1 ZINC000880690253 EJ On-Demand Anodyne EPHX2 29 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)CC1 ZINC000880690256 EI On-Demand Anodyne CACNA1H 45 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)CC1 ZINC000880690256 EI On-Demand Anodyne NPY5R 15 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)CC1 ZINC000880690256 EI On-Demand Anodyne EPHX2 42 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCOCC2)CC1 ZINC000880690256 EI On-Demand Anodyne TRPM8 29 41 Cn1ccnc1[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880690257 FH On-Demand Anodyne EPHX2 34 41 Cn1ccnc1[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880690258 FH On-Demand Anodyne EPHX2 34 41 Cn1ccnc1[C@@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880690260 FH On-Demand Anodyne EPHX2 34 41 Cn1ccnc1[C@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880690261 FH On-Demand Anodyne EPHX2 34 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(C(F)F)C1 ZINC000880690262 DF On-Demand Anodyne CACNA1H 44 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(C(F)F)C1 ZINC000880690262 DF On-Demand Anodyne EPHX2 35 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(C(F)F)C1 ZINC000880690264 DF On-Demand Anodyne CACNA1H 44 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(C(F)F)C1 ZINC000880690264 DF On-Demand Anodyne EPHX2 35 47 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(CCCO)C1 ZINC000880690279 EF On-Demand Anodyne CCR3 72 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN(CCCO)C1 ZINC000880690279 EF On-Demand Anodyne EPHX2 48 51 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(CCCO)C1 ZINC000880690281 EF On-Demand Anodyne CCR3 72 45 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN(CCCO)C1 ZINC000880690281 EF On-Demand Anodyne EPHX2 48 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCSC2(CCC2)CC1 ZINC000880690283 EJ On-Demand Anodyne CACNA1H 44 43 NC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690303 DE On-Demand Anodyne EPHX2 16 40 NC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690306 DE On-Demand Anodyne EPHX2 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880690314 GI On-Demand Anodyne CCR3 45 52 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880690314 GI On-Demand Anodyne EPHX2 73 49 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880690317 GI On-Demand Anodyne CCR3 45 52 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880690317 GI On-Demand Anodyne EPHX2 73 49 O=C(Nc1ccc(F)c(C(F)F)c1)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880690324 FH On-Demand Anodyne EPHX2 60 50 O=C(NCCCc1nc[nH]n1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690325 DF On-Demand Anodyne PRMT3 45 34 COC[C@@H](O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690347 CD On-Demand Anodyne ADRB1 44 36 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(c2nccs2)CC1 ZINC000880690349 FI On-Demand Anodyne EPHX2 48 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](O)(C(=O)N2CCCC2)C1 ZINC000880690353 GF On-Demand Anodyne EPHX2 29 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](O)(C(=O)N2CCCC2)C1 ZINC000880690355 GF On-Demand Anodyne EPHX2 29 43 N#CC1(c2ccccn2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690368 FI On-Demand Mild CACNA1H 47 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](C(=O)N2CCCC2)C1 ZINC000880690404 FG On-Demand Anodyne EPHX2 25 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](C(=O)N2CCCC2)C1 ZINC000880690406 FG On-Demand Anodyne EPHX2 25 40 CNc1nc(C(=O)N2CCC[C@H](n3ccnn3)CC2)cs1 ZINC000880690410 DD On-Demand Anodyne TRPC6 58 44 CNc1nc(C(=O)N2CCC[C@H](n3ccnn3)CC2)cs1 ZINC000880690410 DD On-Demand Anodyne TRPC3 51 44 CNc1nc(C(=O)N2CCC[C@@H](n3ccnn3)CC2)cs1 ZINC000880690413 DD On-Demand Anodyne TRPC6 58 44 CNc1nc(C(=O)N2CCC[C@@H](n3ccnn3)CC2)cs1 ZINC000880690413 DD On-Demand Anodyne TRPC3 51 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC2)CC1 ZINC000880690414 DJ On-Demand Anodyne CACNA1H 55 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC2)CC1 ZINC000880690414 DJ On-Demand Anodyne EPHX2 33 46 N#CCNC(=O)CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690465 DD On-Demand Mild F7 25 41 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690478 GH On-Demand Anodyne HTR1D 16 52 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690478 GH On-Demand Anodyne HTR1B 20 52 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690478 GH On-Demand Anodyne PDGFRB 66 50 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690478 GH On-Demand Anodyne NPY2R 68 37 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690478 GH On-Demand Anodyne RBP4 18 44 CN(C)S(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690482 GE On-Demand Anodyne EPHX2 42 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880690488 GH On-Demand Anodyne EPHX2 41 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880690488 GH On-Demand Anodyne CACNA1I 63 37 CC(C)c1nn(C)cc1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690498 EI On-Demand Anodyne FPR2 45 39 CC[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCCO1 ZINC000880690552 DH On-Demand Anodyne NPY2R 40 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](O)(c2cnn[nH]2)C1 ZINC000880690553 EE On-Demand Anodyne EPHX2 29 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](O)(c2cnn[nH]2)C1 ZINC000880690554 EE On-Demand Anodyne EPHX2 29 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](F)(CO)C1 ZINC000880690559 DF On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](F)(CO)C1 ZINC000880690559 DF On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](F)(CO)C1 ZINC000880690560 DF On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](F)(CO)C1 ZINC000880690560 DF On-Demand Anodyne EPHX2 37 43 O=C(c1c(O)cccc1O)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690580 DD On-Demand Anodyne L3MBTL3 76 42 O=C(c1c(O)cccc1O)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690581 DD On-Demand Anodyne L3MBTL3 76 42 CCOC(=O)[C@]1(COC)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690582 GH On-Demand Anodyne EPHX2 25 43 CCOC(=O)[C@@]1(COC)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690583 GH On-Demand Anodyne EPHX2 25 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@H]1CC(F)F ZINC000880690585 EH On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@@H]1CC(F)F ZINC000880690586 EH On-Demand Anodyne EPHX2 18 40 CSC1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCN(C)CC1 ZINC000880690587 FH On-Demand Anodyne MCHR1 21 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880690588 GJ On-Demand Anodyne EPHX2 32 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880690589 GJ On-Demand Anodyne EPHX2 32 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880690590 FH On-Demand Anodyne EPHX2 42 48 CS(=O)(=O)NC[C@H]1CCC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690607 GF On-Demand Anodyne CCR3 26 41 CS(=O)(=O)NC[C@H]1CCC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690608 GF On-Demand Anodyne CCR3 26 41 CS(=O)(=O)NC[C@@H]1CCC[C@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690609 GF On-Demand Anodyne CCR3 26 41 CS(=O)(=O)NC[C@@H]1CCC[C@@H]1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690610 GF On-Demand Anodyne CCR3 26 41 NC(=O)[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690615 ED On-Demand Anodyne EPHX2 28 43 NC(=O)[C@@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690616 ED On-Demand Anodyne EPHX2 28 43 CCc1nnc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)s1 ZINC000880690626 EG On-Demand Anodyne PRMT3 61 34 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880690641 GH On-Demand Anodyne GRM4 32 43 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880690641 GH On-Demand Anodyne IMDH_CRYPV 52 35 COC(=O)C[C@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880690642 GH On-Demand Anodyne GRM4 32 43 COC(=O)C[C@](C)(NC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880690642 GH On-Demand Anodyne IMDH_CRYPV 52 35 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690657 FH On-Demand Anodyne CACNA1H 40 36 Cn1nccc1[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690658 FH On-Demand Anodyne CACNA1H 40 36 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690661 EG On-Demand Anodyne CCR3 99 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690661 EG On-Demand Anodyne EPHX2 28 44 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690661 EG On-Demand Anodyne CACNA1I 66 34 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690662 EG On-Demand Anodyne CCR3 99 41 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690662 EG On-Demand Anodyne EPHX2 28 44 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690662 EG On-Demand Anodyne CACNA1I 66 34 CN(C[C@@H](O)Cc1ccccc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690664 FH On-Demand Anodyne NPY5R 34 40 CN(C[C@H](O)Cc1ccccc1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690665 FH On-Demand Anodyne NPY5R 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](n2cccn2)C1 ZINC000880690671 DG On-Demand Anodyne EPHX2 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](n2cccn2)C1 ZINC000880690672 DG On-Demand Anodyne EPHX2 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880690683 EI On-Demand Anodyne CPT1A 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880690684 EI On-Demand Anodyne CPT1A 22 44 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880690685 GF On-Demand Anodyne LIMK1 16 41 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)C1 ZINC000880690685 GF On-Demand Anodyne LIMK2 28 41 CS(=O)(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690688 EE On-Demand Anodyne PRMT3 52 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@]2(CCCOC2)C1 ZINC000880690716 EG On-Demand Anodyne EPHX2 37 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@]2(CCCOC2)C1 ZINC000880690717 EG On-Demand Anodyne EPHX2 37 46 O=C(NCCO[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690719 EG On-Demand Anodyne EPHX2 20 40 O=C(NCCO[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690720 EG On-Demand Anodyne EPHX2 20 40 CSCC[C@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)C(=O)N(C)C ZINC000880690721 FG On-Demand Anodyne FPR1 31 41 CC1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690724 CG On-Demand Anodyne CACNA1H 37 42 CC1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690724 CG On-Demand Anodyne EPHX2 27 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](C(F)(F)F)[C@H](CO)C1 ZINC000880690726 FH On-Demand Anodyne EPHX2 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880690727 FH On-Demand Anodyne EPHX2 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](C(F)(F)F)[C@H](CO)C1 ZINC000880690728 FH On-Demand Anodyne EPHX2 33 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880690729 FH On-Demand Anodyne EPHX2 33 43 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690731 GE On-Demand Anodyne HLA-DRB1 50 35 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690733 GE On-Demand Anodyne HLA-DRB1 50 35 Cn1ncc(CNC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880690736 CE On-Demand Anodyne PRMT3 45 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCOCC2)C1 ZINC000880690742 DG On-Demand Anodyne EPHX2 38 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690743 GK On-Demand Anodyne CACNA1H 40 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690743 GK On-Demand Anodyne SLC18A3 26 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690743 GK On-Demand Anodyne SCD1 17 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690743 GK On-Demand Anodyne WNT3A 47 34 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880690761 GI On-Demand Anodyne EPHX2 51 48 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880690761 GI On-Demand Anodyne DPP7 18 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](C(F)F)C1 ZINC000880690773 DG On-Demand Anodyne EPHX2 26 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](C(F)F)C1 ZINC000880690774 DG On-Demand Anodyne EPHX2 26 43 CS(=O)(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCC1 ZINC000880690777 FG On-Demand Anodyne PRMT3 45 35 C[C@@H]1CN(C2CCOCC2)CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690787 FG On-Demand Anodyne LIMK1 17 42 C[C@@H]1CN(C2CCOCC2)CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690787 FG On-Demand Anodyne LIMK2 29 42 O=C(c1ccc2nc(Cl)ccc2c1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880690791 FG On-Demand Anodyne L3MBTL3 84 45 O=C(c1ccc2nc(Cl)ccc2c1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880690792 FG On-Demand Anodyne L3MBTL3 84 45 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690806 GH On-Demand Anodyne CACNA1H 41 41 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690806 GH On-Demand Anodyne EPHX2 38 45 C[C@@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690807 CG On-Demand Anodyne CCR3 26 41 C[C@@H](O)CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690807 CG On-Demand Anodyne LEF 25 46 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCS1 ZINC000880690823 EJ On-Demand Anodyne CACNA1H 48 45 CC(C)n1ccc(NC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880690833 DI On-Demand Anodyne FPR2 57 41 N#CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880690834 CF On-Demand Mild ADRB1 42 35 O=C(NCCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880690835 CG On-Demand Anodyne CCR3 17 44 O=C(NCCCCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880690835 CG On-Demand Anodyne LEF 15 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880690839 FH On-Demand Anodyne CACNA1H 54 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880690839 FH On-Demand Anodyne EPHX2 38 55 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880690840 FH On-Demand Anodyne CACNA1H 54 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880690840 FH On-Demand Anodyne EPHX2 38 55 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCO)C1CCSCC1 ZINC000880690842 EG On-Demand Anodyne MCHR1 32 41 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCC(F)(F)CC1 ZINC000880690865 EJ On-Demand Anodyne MCHR1 27 40 N#Cc1ccncc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690866 GG On-Demand Mild NPY2R 45 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)(F)CC1 ZINC000880690869 DI On-Demand Anodyne CACNA1H 69 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)(F)CC1 ZINC000880690869 DI On-Demand Anodyne NPY5R 17 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)(F)CC1 ZINC000880690869 DI On-Demand Anodyne EPHX2 32 42 NC(=O)C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690877 DE On-Demand Anodyne CCR3 18 42 NC(=O)C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690878 DE On-Demand Anodyne CCR3 18 42 CCN1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880690894 DF On-Demand Anodyne EPHX2 33 41 CCN1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880690895 DF On-Demand Anodyne EPHX2 33 41 CS(=O)(=O)CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690901 FG On-Demand Anodyne EPHX2 32 41 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690906 EI On-Demand Anodyne CACNA1H 53 42 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690906 EI On-Demand Anodyne EPHX2 27 42 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCC1(F)F ZINC000880690909 DI On-Demand Anodyne CACNA1H 50 44 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCC1(F)F ZINC000880690910 DI On-Demand Anodyne CACNA1H 50 44 CN(C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1)S(C)(=O)=O ZINC000880690911 GF On-Demand Anodyne CCR3 16 42 CN(C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1)S(C)(=O)=O ZINC000880690912 GF On-Demand Anodyne CCR3 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@H](C2CCC2)C1 ZINC000880690920 EI On-Demand Anodyne ITGAL 41 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@H](C2CCC2)C1 ZINC000880690920 EI On-Demand Anodyne EPHX2 21 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@@H](C2CCC2)C1 ZINC000880690921 EI On-Demand Anodyne ITGAL 41 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOC[C@@H](C2CCC2)C1 ZINC000880690921 EI On-Demand Anodyne EPHX2 21 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@](CO)(Cc2ccc(F)cc2)C1 ZINC000880690925 GI On-Demand Anodyne CACNA1H 40 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@](CO)(Cc2ccc(F)cc2)C1 ZINC000880690926 GI On-Demand Anodyne CACNA1H 40 38 O=C(NCC1(c2ccccn2)CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690931 EI On-Demand Anodyne NMBR 48 44 O=C(NCC1(c2ccccn2)CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690931 EI On-Demand Anodyne SLC6A9 24 42 O=C(NCC1(c2ccccn2)CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690931 EI On-Demand Anodyne GRPR 25 44 CS(=O)(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCC1 ZINC000880690949 FF On-Demand Anodyne PRMT3 45 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(C1)Oc1ccccc1O2 ZINC000880690960 FI On-Demand Anodyne CACNA1H 43 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(C1)Oc1ccccc1O2 ZINC000880690960 FI On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(C1)Oc1ccccc1O2 ZINC000880690960 FI On-Demand Anodyne TRPM8 27 42 O=C(NCCC1(O)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690969 EF On-Demand Anodyne EPHX2 15 40 Cc1ccncc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690972 FH On-Demand Anodyne HTR1B 15 44 Cc1ccncc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690972 FH On-Demand Anodyne PDGFRB 36 40 Cc1ccncc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880690972 FH On-Demand Anodyne NPY2R 83 35 CCC1(O)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880690973 CF On-Demand Anodyne S1PR2 27 40 O=C(NCCN1CC=CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690976 DG On-Demand Anodyne CCR3 27 43 O=C(NCCN1CC=CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880690976 DG On-Demand Anodyne EPHX2 17 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880691002 FI On-Demand Anodyne CACNA1H 40 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880691002 FI On-Demand Anodyne EPHX2 34 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880691003 FI On-Demand Anodyne CACNA1H 40 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880691003 FI On-Demand Anodyne EPHX2 34 41 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880691004 EG On-Demand Anodyne EPHX2 15 41 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880691004 EG On-Demand Anodyne SCD1 16 40 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880691005 EG On-Demand Anodyne EPHX2 15 41 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880691005 EG On-Demand Anodyne SCD1 16 40 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880691006 EG On-Demand Anodyne EPHX2 15 41 C[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880691006 EG On-Demand Anodyne SCD1 16 40 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880691007 EG On-Demand Anodyne EPHX2 15 41 C[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880691007 EG On-Demand Anodyne SCD1 16 40 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)C1 ZINC000880691011 EG On-Demand Anodyne CACNA1H 40 43 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)C1 ZINC000880691011 EG On-Demand Anodyne EPHX2 37 46 O=C(c1cnc(Cl)cn1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880691019 DD On-Demand Anodyne L3MBTL3 43 40 O=C(c1cnc(Cl)cn1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880691020 DD On-Demand Anodyne L3MBTL3 43 40 CN(C(=O)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1)c1ccccc1 ZINC000880691023 GI On-Demand Anodyne NPY2R 51 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880691027 EI On-Demand Anodyne CACNA1H 40 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880691027 EI On-Demand Anodyne EPHX2 25 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880691027 EI On-Demand Anodyne MCHR1 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2ccccn2)C1 ZINC000880691027 EI On-Demand Anodyne SMO 18 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880691028 EI On-Demand Anodyne CACNA1H 40 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880691028 EI On-Demand Anodyne EPHX2 25 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880691028 EI On-Demand Anodyne MCHR1 16 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccn2)C1 ZINC000880691028 EI On-Demand Anodyne SMO 18 40 CCC[C@]1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691042 EH On-Demand Anodyne CACNA1H 40 41 CCC[C@]1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691042 EH On-Demand Anodyne EPHX2 30 40 NC(=O)C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691044 EG On-Demand Anodyne CCR3 16 41 NC(=O)C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691044 EG On-Demand Anodyne EPHX2 17 40 NC(=O)C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691045 EG On-Demand Anodyne CCR3 16 41 NC(=O)C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691045 EG On-Demand Anodyne EPHX2 17 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CC(F)(F)F)CC1 ZINC000880691050 FJ On-Demand Anodyne EPHX2 40 47 Cc1nnc(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)s1 ZINC000880691056 EG On-Demand Anodyne PRMT3 62 34 O=C(c1ccc2c(O)nc(S)nc2c1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880691058 FE On-Demand Anodyne L3MBTL3 74 41 O=C(c1ccc2c(O)nc(S)nc2c1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880691059 FE On-Demand Anodyne L3MBTL3 74 41 O=C(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880691070 EF On-Demand Bother L3MBTL3 79 50 O=C(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC[C@H](n2ccnn2)CC1 ZINC000880691071 EF On-Demand Bother L3MBTL3 79 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](n2cc(Cl)cn2)C1 ZINC000880691079 FI On-Demand Anodyne EPHX2 23 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](n2cc(Cl)cn2)C1 ZINC000880691079 FI On-Demand Anodyne MCHR1 18 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](n2cc(Cl)cn2)C1 ZINC000880691080 FI On-Demand Anodyne EPHX2 23 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](n2cc(Cl)cn2)C1 ZINC000880691080 FI On-Demand Anodyne MCHR1 18 43 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCOCC2)O1 ZINC000880691081 FH On-Demand Anodyne CACNA1H 29 40 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCOCC2)O1 ZINC000880691082 FH On-Demand Anodyne CACNA1H 29 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(CCCOC2)C1 ZINC000880691091 EH On-Demand Anodyne EPHX2 39 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(CCCOC2)C1 ZINC000880691092 EH On-Demand Anodyne EPHX2 39 46 C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691093 DH On-Demand Anodyne CACNA1H 59 45 C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691093 DH On-Demand Anodyne S1PR2 28 41 C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691093 DH On-Demand Anodyne EPHX2 31 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(c2ccccc2)CC1 ZINC000880691095 GI On-Demand Anodyne CACNA1H 58 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(c2ccccc2)CC1 ZINC000880691095 GI On-Demand Anodyne EPHX2 31 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CN2CCOCC2)C1 ZINC000880691099 FG On-Demand Anodyne CCR3 32 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CN2CCOCC2)C1 ZINC000880691099 FG On-Demand Anodyne EPHX2 34 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CN2CCOCC2)C1 ZINC000880691100 FG On-Demand Anodyne CCR3 32 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CN2CCOCC2)C1 ZINC000880691100 FG On-Demand Anodyne EPHX2 34 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](C2CC2)C1 ZINC000880691118 DI On-Demand Anodyne EPHX2 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](C2CC2)C1 ZINC000880691119 DI On-Demand Anodyne EPHX2 19 41 Cn1nc(NC(=O)Nc2ccc(F)c(C(F)F)c2)cc1C1CC1 ZINC000880691121 DI On-Demand Anodyne FPR2 41 38 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880691132 EH On-Demand Anodyne GLRA1 42 32 O=C(NCc1nnc(C2CC2)o1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691133 EG On-Demand Anodyne PRMT3 52 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880691134 GI On-Demand Anodyne CACNA1H 45 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880691134 GI On-Demand Anodyne EPHX2 37 64 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880691135 GI On-Demand Anodyne CACNA1H 45 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880691135 GI On-Demand Anodyne EPHX2 37 64 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCO)CC1 ZINC000880691148 EH On-Demand Anodyne CCR3 17 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCO)CC1 ZINC000880691148 EH On-Demand Anodyne EPHX2 29 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCO)CC1 ZINC000880691149 EH On-Demand Anodyne CCR3 17 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCO)CC1 ZINC000880691149 EH On-Demand Anodyne EPHX2 29 45 O=C1C[C@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691158 GI On-Demand Anodyne CACNA1H 45 36 O=C1C[C@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691158 GI On-Demand Anodyne EPHX2 39 47 O=C1C[C@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691158 GI On-Demand Anodyne TRPM8 31 49 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691159 GI On-Demand Anodyne CACNA1H 45 36 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691159 GI On-Demand Anodyne EPHX2 39 47 O=C1C[C@@]2(CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)Oc2ccccc21 ZINC000880691159 GI On-Demand Anodyne TRPM8 31 49 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)Cc1ccco1 ZINC000880691169 GH On-Demand Anodyne CASR 65 52 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)Cc1ccco1 ZINC000880691169 GH On-Demand Anodyne EPHX2 23 43 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)Cc1ccco1 ZINC000880691169 GH On-Demand Anodyne MCHR1 18 41 CN1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)[C@@H]1c1cccnc1 ZINC000880691174 GH On-Demand Anodyne NAMPT 59 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCCO2 ZINC000880691178 EH On-Demand Anodyne CACNA1H 40 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCCO2 ZINC000880691178 EH On-Demand Anodyne EPHX2 36 40 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691179 DG On-Demand Anodyne TRPC6 45 33 C[C@H]1[C@H](O)CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691181 DG On-Demand Anodyne TRPC6 45 33 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691182 DG On-Demand Anodyne TRPC6 45 33 C=C1c2ccccc2C(=O)N1CCC(=O)Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2)s1 ZINC000880691188 JK On-Demand Anodyne RORC 20 50 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccnc(F)c2)CC1 ZINC000880691194 FH On-Demand Anodyne CACNA1H 40 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ccnc(F)c2)CC1 ZINC000880691194 FH On-Demand Anodyne STAT6 56 32 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691198 EI On-Demand Anodyne PDGFRB 43 35 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691198 EI On-Demand Anodyne CCR3 31 46 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691198 EI On-Demand Anodyne EPHX2 28 42 C[C@@H]1CN(CC(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691202 GI On-Demand Anodyne EPHX2 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880691203 GG On-Demand Bother PDGFRB 50 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880691203 GG On-Demand Bother TRPV1 19 67 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC(O)CC2)CC1 ZINC000880691206 FI On-Demand Anodyne CACNA1H 56 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCC(O)CC2)CC1 ZINC000880691206 FI On-Demand Anodyne EPHX2 28 41 Cn1ncc2c1CCCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880691215 EG On-Demand Anodyne MAPK1 41 35 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCc2nnnn2CC1 ZINC000880691223 EE On-Demand Anodyne EPHX2 44 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCc2nnnn2CC1 ZINC000880691224 EE On-Demand Anodyne EPHX2 44 43 Cc1ncsc1CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691228 EH On-Demand Anodyne PRMT3 44 32 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880691242 CH On-Demand Anodyne EPHX2 52 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1C[C@H]2C[C@@H]2C1 ZINC000880691243 CH On-Demand Anodyne EPHX2 52 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1C[C@@H]2C[C@H]2C1 ZINC000880691244 CH On-Demand Anodyne EPHX2 52 40 CCC(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691246 DF On-Demand Anodyne EPHX2 26 40 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@]1=O ZINC000880691249 EH On-Demand Anodyne CACNA1H 52 43 CC1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC[S@@]1=O ZINC000880691250 EH On-Demand Anodyne CACNA1H 52 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2cccc(F)n2)CC1 ZINC000880691258 FH On-Demand Anodyne FAAH 20 43 O=C(NCCC1CC(F)(F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691270 DI On-Demand Anodyne PRMT3 16 40 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(CC(F)(F)F)CC1 ZINC000880691275 GI On-Demand Anodyne MCHR1 45 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880691276 GI On-Demand Anodyne CACNA1H 42 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880691277 GI On-Demand Anodyne CACNA1H 42 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880691278 GI On-Demand Anodyne CACNA1H 42 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880691279 GI On-Demand Anodyne CACNA1H 42 37 O=C(NC[C@H]1CCCCN1CCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880691284 EF On-Demand Anodyne CCR3 44 40 O=C(NC[C@H]1CCCN1CCCO)Nc1ccc(F)c(C(F)F)c1 ZINC000880691294 EF On-Demand Anodyne CCR3 50 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCn2ccnc21 ZINC000880691299 DG On-Demand Anodyne EPHX2 33 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCn2ccnc21 ZINC000880691300 DG On-Demand Anodyne EPHX2 33 42 CC(C)(C)C1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691306 DI On-Demand Anodyne CACNA1H 38 40 COCCn1nnc2c1CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880691309 FF On-Demand Anodyne MAPK1 41 38 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691311 GF On-Demand Anodyne EPHX2 30 45 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691311 GF On-Demand Anodyne HCN1 55 40 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691311 GF On-Demand Anodyne HCN4 47 30 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CCCO)C1 ZINC000880691313 DG On-Demand Anodyne CCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CCCO)C1 ZINC000880691313 DG On-Demand Anodyne EPHX2 16 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CCCO)C1 ZINC000880691314 DG On-Demand Anodyne CCR3 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CCCO)C1 ZINC000880691314 DG On-Demand Anodyne EPHX2 16 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880691316 EG On-Demand Anodyne RBP4 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880691317 EG On-Demand Anodyne RBP4 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880691318 EG On-Demand Anodyne RBP4 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880691319 EG On-Demand Anodyne RBP4 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCOCCN1 ZINC000880691323 CE On-Demand Anodyne EPHX2 16 41 CN1C(=O)CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880691326 EE On-Demand Anodyne NPY1R 27 40 CN1C(=O)CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880691327 EE On-Demand Anodyne NPY1R 27 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCC[C@H]1CO ZINC000880691342 DG On-Demand Anodyne CCR3 30 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CO)CC1 ZINC000880691349 DG On-Demand Anodyne CCR3 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CO)CC1 ZINC000880691349 DG On-Demand Anodyne EPHX2 26 52 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CO)CC1 ZINC000880691350 DG On-Demand Anodyne CCR3 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CO)CC1 ZINC000880691350 DG On-Demand Anodyne EPHX2 26 52 COC[C@]1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691365 EF On-Demand Anodyne CACNA1H 51 41 COC[C@]1(CO)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691365 EF On-Demand Anodyne EPHX2 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC(OC(F)F)CC1 ZINC000880691366 FI On-Demand Anodyne EPHX2 62 51 NC(=O)C[C@@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691386 ED On-Demand Anodyne EPHX2 26 45 NC(=O)C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691387 ED On-Demand Anodyne EPHX2 26 45 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691397 GG On-Demand Anodyne CACNA1H 50 39 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691397 GG On-Demand Anodyne EPHX2 35 45 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691398 GG On-Demand Anodyne CACNA1H 50 39 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691398 GG On-Demand Anodyne EPHX2 35 45 Cn1c(S)nnc1CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691399 EF On-Demand Anodyne PRMT3 51 31 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880691411 EH On-Demand Anodyne EPHX2 52 43 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880691411 EH On-Demand Anodyne GLRA1 43 33 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880691411 EH On-Demand Anodyne CXCR3 19 44 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691421 FE On-Demand Anodyne EPHX2 24 46 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691422 FE On-Demand Anodyne EPHX2 24 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCc1ccccc12 ZINC000880691428 GJ On-Demand Anodyne CACNA1H 42 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCc1ccccc12 ZINC000880691428 GJ On-Demand Anodyne NPY5R 30 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)OCCc1ccccc12 ZINC000880691428 GJ On-Demand Anodyne TRPM8 31 41 CN(C)CC(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691442 DG On-Demand Anodyne IMDH_CRYPV 54 33 NC(=O)C1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691482 ED On-Demand Anodyne CACNA1H 66 43 O=C(NCCS(=O)(=O)C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691483 EE On-Demand Anodyne CCR3 25 40 O=C(c1cccc([N+](=O)[O-])c1Br)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880691491 GF On-Demand Bother L3MBTL3 39 41 O=C(c1cccc([N+](=O)[O-])c1Br)N1CCC[C@H](n2ccnn2)CC1 ZINC000880691492 GF On-Demand Bother L3MBTL3 39 41 COC(OC)c1ccc(C(=O)N2CCC[C@@H](n3ccnn3)CC2)o1 ZINC000880691494 EE On-Demand Anodyne L3MBTL3 36 43 COC(OC)c1ccc(C(=O)N2CCC[C@H](n3ccnn3)CC2)o1 ZINC000880691495 EE On-Demand Anodyne L3MBTL3 36 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](F)C1 ZINC000880691499 CG On-Demand Anodyne DPP4 21 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](F)C1 ZINC000880691500 CG On-Demand Anodyne DPP4 21 45 NC(=O)[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1c1ccccc1 ZINC000880691512 GG On-Demand Anodyne SMO 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCOC2)C1 ZINC000880691513 DG On-Demand Anodyne EPHX2 35 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OC2CCC2)CC1 ZINC000880691517 EI On-Demand Anodyne EPHX2 44 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(OC2CCC2)CC1 ZINC000880691517 EI On-Demand Anodyne SCD1 15 48 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@]2(CCS(=O)(=O)C2)C1 ZINC000880691541 GG On-Demand Anodyne EPHX2 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@]2(CCS(=O)(=O)C2)C1 ZINC000880691542 GG On-Demand Anodyne EPHX2 28 42 Cc1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)nn1C(C)C ZINC000880691546 EI On-Demand Anodyne HTR2A 20 41 Cc1cc(NC(=O)Nc2ccc(F)c(C(F)F)c2)nn1C(C)C ZINC000880691546 EI On-Demand Anodyne FPR2 50 40 COCC1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691550 EI On-Demand Anodyne EPHX2 53 43 COCC1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691550 EI On-Demand Anodyne CXCR3 17 40 NC(=O)[C@@H]1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691563 DF On-Demand Anodyne EPHX2 43 41 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(CCC(F)(F)F)CC1 ZINC000880691564 GJ On-Demand Anodyne CCR5 15 52 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CCN(CCC(F)(F)F)CC1 ZINC000880691564 GJ On-Demand Anodyne MCHR1 53 41 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne PDGFRB 64 44 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne FAAH 24 41 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne GALR2 43 34 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne MCHR1 17 40 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne DGAT1 38 50 COc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)nc1 ZINC000880691569 GH On-Demand Anodyne NPBWR1 41 39 CN(C)C1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691576 EH On-Demand Anodyne EPHX2 53 43 CN(C)C1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691576 EH On-Demand Anodyne CXCR3 16 41 Cn1nccc1[C@@H](CO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691586 EE On-Demand Anodyne HTR2A 31 40 Cn1nccc1[C@H](CO)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691587 EE On-Demand Anodyne HTR2A 31 40 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1ccc(F)c(C(F)F)c1 ZINC000880691597 EF On-Demand Anodyne CCR3 38 45 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1ccc(F)c(C(F)F)c1 ZINC000880691597 EF On-Demand Anodyne MTOR 32 40 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1ccc(F)c(C(F)F)c1 ZINC000880691597 EF On-Demand Anodyne EPHX2 19 45 COCC(COC)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691601 GF On-Demand Anodyne PDGFRB 44 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CC2)C1 ZINC000880691615 CG On-Demand Anodyne CACNA1H 39 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CC2)C1 ZINC000880691615 CG On-Demand Anodyne EPHX2 30 45 O=C(c1cccnc1I)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880691638 GE On-Demand Anodyne L3MBTL3 68 42 O=C(c1cccnc1I)N1CCC[C@H](n2ccnn2)CC1 ZINC000880691640 GE On-Demand Anodyne L3MBTL3 68 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691641 GH On-Demand Anodyne CCR3 90 42 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691641 GH On-Demand Anodyne F2R 55 33 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691641 GH On-Demand Anodyne MCHR1 46 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691643 GH On-Demand Anodyne CCR3 90 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691643 GH On-Demand Anodyne F2R 55 33 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691643 GH On-Demand Anodyne MCHR1 46 42 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691649 EG On-Demand Anodyne CCR3 47 35 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691649 EG On-Demand Anodyne FPR2 44 38 CC(=O)N1CCC[C@@H]1C(=O)NN=c1cc[nH]cc1F ZINC000880691652 CC On-Demand Reactive LGMN 43 34 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691655 EH On-Demand Anodyne EPHX2 35 46 O=C(NC[C@@]1(O)C[C@H]2C=C[C@H]1C2)Nc1ccc(F)c(C(F)F)c1 ZINC000880691660 EG On-Demand Anodyne EPHX2 19 41 O=C(NC[C@]1(O)C[C@H]2C=C[C@H]1C2)Nc1ccc(F)c(C(F)F)c1 ZINC000880691662 EG On-Demand Anodyne EPHX2 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880691665 FF On-Demand Anodyne L3MBTL3 61 34 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C2CCC2)CC1 ZINC000880691666 EH On-Demand Anodyne EPHX2 56 44 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C2CCC2)CC1 ZINC000880691666 EH On-Demand Anodyne CXCR3 21 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN(C2CCC2)CC1 ZINC000880691666 EH On-Demand Anodyne MCHR1 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880691667 FF On-Demand Anodyne L3MBTL3 61 34 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691668 DF On-Demand Anodyne EPHX2 48 39 COC1CC(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691676 DH On-Demand Anodyne CCR3 32 40 CC(C)(C)N1CC[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691678 EH On-Demand Anodyne CACNA1I 55 34 CC(C)(C)N1CC[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691679 EH On-Demand Anodyne CACNA1I 55 34 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691690 FI On-Demand Anodyne CACNA1H 70 43 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691690 FI On-Demand Anodyne EPHX2 35 41 O=C(NC[C@H]1CCCC[C@@H]1O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691695 DG On-Demand Anodyne PRMT3 52 39 O=C(NCCOC(=O)C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691699 DF On-Demand Anodyne CCR3 19 41 O=C(NCCCC1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691702 EI On-Demand Anodyne CCR3 40 42 CC(C)(C)N1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691709 EI On-Demand Anodyne CCR3 70 38 CC(C)(C)N1CC[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691709 EI On-Demand Anodyne CACNA1I 73 38 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691710 EI On-Demand Anodyne CCR3 70 38 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691710 EI On-Demand Anodyne CACNA1I 73 38 O=C(NCc1nnc(C2CC2)s1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691715 EH On-Demand Anodyne PRMT3 62 34 O=C(Nc1ccc(F)c(C(F)F)c1)NN1CCCCC1 ZINC000880691717 CG On-Demand Anodyne EPHX2 17 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccncn2)CC1 ZINC000880691721 FH On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880691732 FG On-Demand Anodyne HRH3 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880691732 FG On-Demand Anodyne EPHX2 28 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880691732 FG On-Demand Anodyne L3MBTL3 82 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880691733 FG On-Demand Anodyne HRH3 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880691733 FG On-Demand Anodyne EPHX2 28 51 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880691733 FG On-Demand Anodyne L3MBTL3 82 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(CO)CC1 ZINC000880691741 DE On-Demand Anodyne CACNA1H 55 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(O)(CO)CC1 ZINC000880691741 DE On-Demand Anodyne S1PR2 31 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880691764 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880691765 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]2COC[C@H]2C1 ZINC000880691766 DG On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880691767 DG On-Demand Anodyne EPHX2 24 40 CCNC(=O)C(C)(C)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691784 DF On-Demand Anodyne IMDH_CRYPV 48 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2ccon2)CC1 ZINC000880691793 EI On-Demand Anodyne SMO 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)CC2(F)F ZINC000880691795 DI On-Demand Anodyne CACNA1H 43 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C1)CC2(F)F ZINC000880691795 DI On-Demand Anodyne EPHX2 35 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)CC2(F)F ZINC000880691796 DI On-Demand Anodyne CACNA1H 43 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C1)CC2(F)F ZINC000880691796 DI On-Demand Anodyne EPHX2 35 43 O=C(NN=c1cc[nH]cc1F)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880691812 EF On-Demand Reactive C3AR1 40 42 O=C(NN=c1cc[nH]cc1F)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880691813 EF On-Demand Reactive C3AR1 40 42 CC(C)(C[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1)C(N)=O ZINC000880691820 FH On-Demand Anodyne CCR3 41 36 CC(C)(C[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1)C(N)=O ZINC000880691821 FH On-Demand Anodyne CCR3 41 36 O=C(NCCC[C@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691825 DH On-Demand Anodyne CCR3 35 40 O=C(NCCC[C@@H]1CCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691826 DH On-Demand Anodyne CCR3 35 40 O=C(NC[C@@H](O)C1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691827 DG On-Demand Anodyne PRMT3 43 53 O=C(NC[C@H](O)C1CCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691828 DG On-Demand Anodyne PRMT3 43 53 O=C(NCc1cccc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691829 GH On-Demand Anodyne MTOR 43 38 O=C(NCc1cccc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691829 GH On-Demand Anodyne EPHX2 29 44 O=C(NCc1cccc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691829 GH On-Demand Anodyne STAT6 61 42 O=C(NCc1cccc(N2CCOCC2)c1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691829 GH On-Demand Anodyne NAMPT 34 43 CCO[C@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691858 DG On-Demand Anodyne EPHX2 55 42 C[C@@H](F)CCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691865 CH On-Demand Anodyne LEF 18 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880691876 GI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880691876 GI On-Demand Anodyne TRPM8 38 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880691877 GI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880691877 GI On-Demand Anodyne TRPM8 38 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880691879 GI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880691879 GI On-Demand Anodyne TRPM8 38 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880691881 GI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880691881 GI On-Demand Anodyne TRPM8 38 49 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691886 GG On-Demand Anodyne CACNA1H 37 41 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691886 GG On-Demand Anodyne EPHX2 36 42 CC(C)(C)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880691890 EG On-Demand Anodyne EPHX2 41 38 CC(C)(C)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1=O ZINC000880691892 EG On-Demand Anodyne EPHX2 41 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880691901 FE On-Demand Anodyne FAAH 20 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN([C@@H]2CCOC2)CC1 ZINC000880691908 EF On-Demand Anodyne EPHX2 18 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN([C@H]2CCOC2)CC1 ZINC000880691910 EF On-Demand Anodyne EPHX2 18 42 CS(=O)(=O)CC1CCC(NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880691911 GG On-Demand Anodyne EPHX2 47 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880691913 EH On-Demand Anodyne CPT1A 48 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880691914 EH On-Demand Anodyne CPT1A 48 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2cccnc2)C1 ZINC000880691917 EI On-Demand Anodyne CACNA1H 41 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2cccnc2)C1 ZINC000880691917 EI On-Demand Anodyne MCHR1 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](c2cccnc2)C1 ZINC000880691917 EI On-Demand Anodyne NAMPT 40 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2cccnc2)C1 ZINC000880691919 EI On-Demand Anodyne CACNA1H 41 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2cccnc2)C1 ZINC000880691919 EI On-Demand Anodyne MCHR1 19 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2cccnc2)C1 ZINC000880691919 EI On-Demand Anodyne NAMPT 40 36 CCC1(CC)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691920 DI On-Demand Anodyne CACNA1H 27 40 O=C(NCCCO[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691922 EH On-Demand Anodyne CCR3 32 40 O=C(NCCCO[C@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691922 EH On-Demand Anodyne EPHX2 22 41 O=C(NCCCO[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691924 EH On-Demand Anodyne CCR3 32 40 O=C(NCCCO[C@@H]1CCCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691924 EH On-Demand Anodyne EPHX2 22 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne ACHE 28 45 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne SIGMAR1 27 44 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne CCR3 99 51 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne EPHX2 24 43 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne MCHR1 43 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691945 GI On-Demand Anodyne CACNA1I 73 43 Cn1nccc1[C@@H]1OCCC[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880691964 GH On-Demand Anodyne PRMT3 44 33 O=C(NCc1ccc(N2CCCNC2=O)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880691967 GI On-Demand Anodyne F2R 48 29 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](F)C1 ZINC000880691975 CH On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](F)C1 ZINC000880691975 CH On-Demand Anodyne DPP7 16 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](F)C1 ZINC000880691976 CH On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](F)C1 ZINC000880691976 CH On-Demand Anodyne DPP7 16 42 Cn1ncc(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880691981 EF On-Demand Anodyne CCR3 22 40 Cn1ncc(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880691981 EF On-Demand Anodyne QPCT 33 40 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691982 FG On-Demand Anodyne EPHX2 15 43 COC[C@@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691987 DH On-Demand Anodyne CACNA1H 51 41 COC[C@@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691987 DH On-Demand Anodyne EPHX2 36 40 COC[C@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691988 DH On-Demand Anodyne CACNA1H 51 41 COC[C@]1(C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880691988 DH On-Demand Anodyne EPHX2 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](O)[C@@H](CO)C1 ZINC000880691992 DD On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](O)[C@@H](CO)C1 ZINC000880691993 DD On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](O)[C@H](CO)C1 ZINC000880691994 DD On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](O)[C@H](CO)C1 ZINC000880691995 DD On-Demand Anodyne EPHX2 20 40 CC[C@H](C)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692002 EH On-Demand Anodyne CACNA1H 45 40 CC[C@H](C)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692002 EH On-Demand Anodyne NPY2R 52 36 CN1CCC[C@@H](CCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692012 EH On-Demand Anodyne CCR3 93 44 CN1CCC[C@@H](CCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692012 EH On-Demand Anodyne MCHR1 17 42 CN1CCC[C@@H](CCNC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692012 EH On-Demand Anodyne PRMT3 32 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC(F)(F)C(F)(F)C1 ZINC000880692025 EH On-Demand Mild CACNA1H 32 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1C[C@H](O)C1 ZINC000880692042 CE On-Demand Anodyne EPHX2 49 39 O=C(c1c(F)ccc(O)c1O)N1CCC[C@H](n2ccnn2)CC1 ZINC000880692057 DD On-Demand Clean L3MBTL3 53 38 O=C(c1c(F)ccc(O)c1O)N1CCC[C@@H](n2ccnn2)CC1 ZINC000880692058 DD On-Demand Clean L3MBTL3 53 38 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692060 DG On-Demand Anodyne CHRNA10 55 38 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692060 DG On-Demand Anodyne MCHR1 41 37 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692060 DG On-Demand Anodyne ACKR3 63 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692061 DG On-Demand Anodyne CHRNA10 55 38 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692061 DG On-Demand Anodyne MCHR1 41 37 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692061 DG On-Demand Anodyne ACKR3 63 33 NC(=O)[C@@H]1CC[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692064 EG On-Demand Anodyne VCP 43 41 Cc1c(NC(=O)Nc2ccc(F)c(C(F)F)c2)cnn1C1CCOCC1 ZINC000880692068 FI On-Demand Anodyne MTOR 69 36 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692154 EG On-Demand Anodyne SLC6A4 29 44 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692154 EG On-Demand Anodyne SLC6A3 62 44 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692155 EG On-Demand Anodyne SLC6A4 29 44 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692155 EG On-Demand Anodyne SLC6A3 62 44 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692156 GH On-Demand Anodyne F2R 42 32 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692156 GH On-Demand Anodyne EPHX2 43 45 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692156 GH On-Demand Anodyne DPP7 44 35 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692156 GH On-Demand Anodyne CACNA1G 43 39 CCOC(=O)C1=CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692157 EH On-Demand Anodyne EPHX2 41 39 CCOC(=O)C1=CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692158 EH On-Demand Anodyne EPHX2 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1[C@H]2CC[C@H]1CC(O)(c1ccccc1)C2 ZINC000880692159 GJ On-Demand Anodyne OPRL1 19 45 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692160 GH On-Demand Anodyne F2R 42 32 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692160 GH On-Demand Anodyne EPHX2 43 45 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692160 GH On-Demand Anodyne DPP7 44 35 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692160 GH On-Demand Anodyne CACNA1G 43 39 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CF)C1 ZINC000880692181 CH On-Demand Anodyne CCR3 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](CF)C1 ZINC000880692181 CH On-Demand Anodyne EPHX2 33 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CF)C1 ZINC000880692182 CH On-Demand Anodyne CCR3 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](CF)C1 ZINC000880692182 CH On-Demand Anodyne EPHX2 33 41 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)CC1CC1 ZINC000880692185 FG On-Demand Anodyne CASR 66 49 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)CC1CC1 ZINC000880692185 FG On-Demand Anodyne EPHX2 25 43 O=C(Nc1ccc(F)c(C(F)F)c1)N(CCN1CCOCC1)CC1CC1 ZINC000880692185 FG On-Demand Anodyne MCHR1 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(CC1)CC2 ZINC000880692187 DJ On-Demand Anodyne CACNA1H 45 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC2(CC1)CC2 ZINC000880692187 DJ On-Demand Anodyne EPHX2 31 46 C[S@](=N)(=O)N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692198 FF On-Demand Anodyne NPY5R 15 40 N#Cc1cccc(C2(NC(=O)Nc3ccc(F)c(C(F)F)c3)CCOCC2)c1 ZINC000880692202 GI On-Demand Mild MCHR1 31 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC2(CC1)CC2(F)F ZINC000880692207 EJ On-Demand Anodyne EPHX2 45 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(COC2)C1 ZINC000880692209 DG On-Demand Anodyne CACNA1H 44 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(COC2)C1 ZINC000880692209 DG On-Demand Anodyne EPHX2 39 50 O=C(NCC1(O)CCC(F)(F)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692214 FH On-Demand Anodyne PRMT3 43 31 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@]2(CCSC2)C1 ZINC000880692217 EH On-Demand Anodyne EPHX2 33 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@]2(CCSC2)C1 ZINC000880692218 EH On-Demand Anodyne EPHX2 33 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880692233 EG On-Demand Anodyne RBP4 46 34 Cn1cnc(CCCNC(=O)Nc2ccc(F)c(C(F)F)c2)n1 ZINC000880692234 EF On-Demand Anodyne QPCT 35 41 O=C(NCC1CSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692235 CG On-Demand Anodyne PRMT3 46 33 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCC2)O1 ZINC000880692246 EH On-Demand Anodyne CACNA1H 29 41 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCC2)O1 ZINC000880692247 EH On-Demand Anodyne CACNA1H 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC(F)(F)CC1 ZINC000880692254 DI On-Demand Anodyne CACNA1H 57 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC(F)(F)CC1 ZINC000880692254 DI On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(Cn2cnnc2)CC1 ZINC000880692259 FG On-Demand Anodyne EPHX2 16 40 O=C(NCCN1C[C@H]2CCCCN2C1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692278 FG On-Demand Anodyne CCR3 37 41 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)cn1 ZINC000880692279 GG On-Demand Mild PDGFRB 42 38 O=C(NCCN1C[C@@H]2CCCCN2C1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692280 FG On-Demand Anodyne CCR3 37 41 CC(C)(C)N1C[C@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880692283 FH On-Demand Anodyne CACNA1I 56 35 CC(C)(C)N1C[C@@H](CNC(=O)Nc2ccc(F)c(C(F)F)c2)CC1=O ZINC000880692285 FH On-Demand Anodyne CACNA1I 56 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880692291 GH On-Demand Anodyne SMO 31 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880692291 GH On-Demand Anodyne ETHR 46 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880692293 GH On-Demand Anodyne SMO 31 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880692293 GH On-Demand Anodyne ETHR 46 34 O=C(NCc1nc(O)c2c(n1)CCOC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880692311 FF On-Demand Anodyne MTOR 17 44 O=C(NCc1nc(O)c2c(n1)CCOC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880692311 FF On-Demand Anodyne WNT3A 41 33 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880692313 GI On-Demand Anodyne P2RY14 48 35 CCC1(N2CCCC2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692315 FJ On-Demand Anodyne CACNA1H 55 42 CCC1(N2CCCC2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692315 FJ On-Demand Anodyne S1PR2 28 40 COC(=O)[C@@]12C[C@@H](NC(=O)Nc3ccc(F)c(C(F)F)c3)C[C@@H]1C2 ZINC000880692324 EG On-Demand Anodyne EPHX2 43 37 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692341 EF On-Demand Anodyne CACNA1H 46 42 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692341 EF On-Demand Anodyne EPHX2 34 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880692378 FG On-Demand Anodyne EPHX2 55 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880692378 FG On-Demand Anodyne CXCR3 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCOC2)CC1 ZINC000880692379 FG On-Demand Anodyne EPHX2 55 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCN([C@H]2CCOC2)CC1 ZINC000880692379 FG On-Demand Anodyne CXCR3 18 41 C#CC1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692396 CH On-Demand Mild CACNA1H 36 41 O=C(NN=c1cc[nH]cc1F)C1(c2ccc([N+](=O)[O-])cc2)CCC1 ZINC000880692400 EE On-Demand Reactive NMBR 41 31 C=CCOCCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692404 DG On-Demand Mild CCR3 16 41 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692407 EF On-Demand Anodyne CACNA1H 38 40 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692407 EF On-Demand Anodyne EPHX2 33 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCF)C1 ZINC000880692420 DI On-Demand Anodyne CCR3 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CCF)C1 ZINC000880692420 DI On-Demand Anodyne EPHX2 19 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCF)C1 ZINC000880692421 DI On-Demand Anodyne CCR3 22 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CCF)C1 ZINC000880692421 DI On-Demand Anodyne EPHX2 19 47 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1C(=O)N1CCOCC1 ZINC000880692447 GF On-Demand Anodyne ITGAL 41 31 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@H]1C(=O)N1CCOCC1 ZINC000880692447 GF On-Demand Anodyne EPHX2 19 42 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)CC2 ZINC000880692455 GI On-Demand Anodyne MAPK1 43 38 CC(C)(CO)[C@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)c1cccnc1 ZINC000880692464 FI On-Demand Anodyne NAMPT 22 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCNC2=O)CC1 ZINC000880692472 EF On-Demand Anodyne CACNA1H 72 44 COC[C@@H]1CCCN1NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692473 DF On-Demand Anodyne CCR3 30 44 C#CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692477 EG On-Demand Mild CACNA1H 43 41 C#CCC1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692477 EG On-Demand Mild S1PR2 29 43 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC2(CSC2)C1 ZINC000880692484 DH On-Demand Anodyne EPHX2 41 37 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC2(CSC2)C1 ZINC000880692484 DH On-Demand Anodyne ENV 41 36 NC(=O)Cc1cccc2c1CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880692493 GG On-Demand Anodyne P2RY14 47 34 CCC1(N(C)C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692500 EI On-Demand Anodyne CACNA1H 69 43 CCC1(N(C)C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692500 EI On-Demand Anodyne NPY2R 42 33 CCC1(N(C)C)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692500 EI On-Demand Anodyne S1PR2 28 41 CCC1(N2CCOCC2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692502 GH On-Demand Anodyne CACNA1H 48 41 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692513 EJ On-Demand Anodyne TRPM8 35 48 COCC1CC(NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692526 DG On-Demand Anodyne CCR3 16 40 COCC1CC(NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692526 DG On-Demand Anodyne EPHX2 47 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(c2nccnn2)CC1 ZINC000880692528 FE On-Demand Anodyne FAAH 25 47 O=C(NC[C@@]12COCCN1C(=O)OC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880692530 FE On-Demand Anodyne EPHX2 26 41 O=C(NC[C@]12COCCN1C(=O)OC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880692531 FE On-Demand Anodyne EPHX2 26 41 COC[C@@H]1CCCN1C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692534 DG On-Demand Anodyne MCHR1 25 40 CS(=O)(=O)C1(CNC(=O)Nc2ccc(F)c(C(F)F)c2)CCCCC1 ZINC000880692589 GH On-Demand Anodyne PRMT3 47 34 CN(CCN1CCCCC1)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692590 EH On-Demand Anodyne MCHR1 52 45 C[C@@H]1CN(CCNC(=O)Nc2ccc(F)c(C(F)F)c2)[C@H](C)CO1 ZINC000880692595 EF On-Demand Anodyne CCR3 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](O)(C2CC2)C1 ZINC000880692599 EH On-Demand Anodyne CACNA1H 37 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@](O)(C2CC2)C1 ZINC000880692599 EH On-Demand Anodyne EPHX2 30 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](O)(C2CC2)C1 ZINC000880692600 EH On-Demand Anodyne CACNA1H 37 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@](O)(C2CC2)C1 ZINC000880692600 EH On-Demand Anodyne EPHX2 30 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](O)C(F)(F)C1 ZINC000880692630 DF On-Demand Anodyne CACNA1H 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](O)C(F)(F)C1 ZINC000880692631 DF On-Demand Anodyne CACNA1H 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC(F)(F)C1 ZINC000880692645 DI On-Demand Anodyne CACNA1H 37 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCCC(F)(F)C1 ZINC000880692645 DI On-Demand Anodyne EPHX2 34 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCC2)[C@@H]1c1ccncc1 ZINC000880692647 FJ On-Demand Anodyne CACNA1H 49 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCC2)[C@H]1c1ccncc1 ZINC000880692650 FJ On-Demand Anodyne CACNA1H 49 43 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880692700 FH On-Demand Anodyne HTR2A 40 41 O=C(NCC1CCC(O)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692708 DG On-Demand Anodyne CACNA1I 41 33 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)Cc2cccnc21 ZINC000880692718 FH On-Demand Anodyne TRPV1 15 52 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692720 DI On-Demand Mild EPHX2 16 44 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1(C)C ZINC000880692721 DG On-Demand Anodyne CACNA1H 30 40 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1(C)C ZINC000880692721 DG On-Demand Anodyne EPHX2 28 41 CSCC[C@H](NC(=O)Nc1ccc(F)c(C(F)F)c1)C(N)=O ZINC000880692722 EE On-Demand Anodyne FPR1 39 43 C#CC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692725 DI On-Demand Mild EPHX2 16 44 CO[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692728 CG On-Demand Anodyne EPHX2 50 41 O=C(NCc1cccnc1N1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692736 FI On-Demand Anodyne TRPV1 32 45 O=C(NCc1cccnc1N1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692736 FI On-Demand Anodyne SCN2A 20 48 O=C(NCc1cccnc1N1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692736 FI On-Demand Anodyne F2R 51 32 O=C(NCc1cccnc1N1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692736 FI On-Demand Anodyne SCN10A 31 48 O=C(NCc1cccnc1N1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692736 FI On-Demand Anodyne NAMPT 46 44 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692745 FH On-Demand Anodyne CACNA1H 45 41 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692745 FH On-Demand Anodyne EPHX2 37 44 NC(=O)C1(N2CCCCC2)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880692747 GG On-Demand Anodyne CACNA1H 40 40 O=C(NCc1ccc(CN2CCNC2=O)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692756 GH On-Demand Anodyne F2R 52 31 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880692757 DI On-Demand Anodyne GRM4 31 40 C[C@@H](CNC(=O)Nc1ccc(F)c(C(F)F)c1)c1ccccn1 ZINC000880692757 DI On-Demand Anodyne SOAT1 21 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC2(CCCO2)C1 ZINC000880692761 DG On-Demand Anodyne EPHX2 31 42 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692953 FD On-Demand Anodyne CCR3 22 48 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692953 FD On-Demand Anodyne EPHX2 57 54 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692953 FD On-Demand Anodyne CXCR3 19 41 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692954 FD On-Demand Anodyne CCR3 22 48 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692954 FD On-Demand Anodyne EPHX2 57 54 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880692954 FD On-Demand Anodyne CXCR3 19 41 O=C(NCCCc1ccco1)Nc1ccc(F)c(C(F)F)c1 ZINC000880692962 DI On-Demand Anodyne CCR3 15 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@]2(CCS(=O)(=O)C2)C1 ZINC000880692967 GE On-Demand Anodyne EPHX2 32 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@]2(CCS(=O)(=O)C2)C1 ZINC000880692968 GE On-Demand Anodyne EPHX2 32 45 C=CCOCCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880692969 CG On-Demand Mild NQO2 21 46 C=CCOCCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880692971 CG On-Demand Mild NQO2 21 46 COc1ccccc1-c1ccc(C(=O)NC[C@]23OCCC[C@H]2C3(F)F)c(O)n1 ZINC000880692974 GG On-Demand Anodyne KCNA3 44 36 COc1ccccc1-c1ccc(C(=O)NC[C@]23OCCC[C@H]2C3(F)F)c(O)n1 ZINC000880692974 GG On-Demand Anodyne HCN1 57 35 COc1ccccc1-c1ccc(C(=O)NC[C@]23OCCC[C@H]2C3(F)F)c(O)n1 ZINC000880692974 GG On-Demand Anodyne HCN4 50 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@H](C)O1)C2 ZINC000880692976 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@H](C)O1)C2 ZINC000880692976 DF On-Demand Anodyne MTNR1A 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@H](C)O1)C2 ZINC000880692976 DF On-Demand Anodyne MTNR1B 35 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@H](C)O1)C2 ZINC000880692977 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@H](C)O1)C2 ZINC000880692977 DF On-Demand Anodyne MTNR1A 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@H](C)O1)C2 ZINC000880692977 DF On-Demand Anodyne MTNR1B 35 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@@H](C)O1)C2 ZINC000880692979 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@@H](C)O1)C2 ZINC000880692979 DF On-Demand Anodyne MTNR1A 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCC[C@@H](C)O1)C2 ZINC000880692979 DF On-Demand Anodyne MTNR1B 35 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@@H](C)O1)C2 ZINC000880692980 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@@H](C)O1)C2 ZINC000880692980 DF On-Demand Anodyne MTNR1A 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCC[C@@H](C)O1)C2 ZINC000880692980 DF On-Demand Anodyne MTNR1B 35 42 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880692981 FF On-Demand Anodyne P2RX7 34 49 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880692981 FF On-Demand Anodyne SSTR3 15 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1COC2(CCC2)C1 ZINC000880693002 DH On-Demand Anodyne ENV 40 35 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1COC2(CCC2)C1 ZINC000880693003 DH On-Demand Anodyne ENV 40 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne PAPA1_CARPA 46 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne CTSL 24 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne POLC 18 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne REN 30 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne CTSS 16 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne FPR1 45 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693014 GH On-Demand Anodyne DNAE 61 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne PAPA1_CARPA 46 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne CTSL 24 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne POLC 18 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne REN 30 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne CTSS 16 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne FPR1 45 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693015 GH On-Demand Anodyne DNAE 61 36 O=C(NCC1SCCS1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693024 DH On-Demand Anodyne PRMT3 45 32 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(Cl)c(Cl)c2)CC1 ZINC000880693029 FG On-Demand Anodyne P2RX7 36 51 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(Cl)c(Cl)c2)CC1 ZINC000880693029 FG On-Demand Anodyne EPHX2 18 60 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(Cl)c(Cl)c2)CC1 ZINC000880693029 FG On-Demand Anodyne DNAE 65 33 Cn1cnnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880693087 FE On-Demand Anodyne PDGFRB 40 36 Cn1cnnc1N1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880693087 FE On-Demand Anodyne NPY2R 50 33 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880693094 CE On-Demand Anodyne LUXR 78 47 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880693094 CE On-Demand Anodyne TRAR 90 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880693094 CE On-Demand Anodyne LASR 60 39 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN2CCCC[C@@H]12 ZINC000880693105 EH On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN2CCCC[C@@H]12 ZINC000880693105 EH On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN2CCCC[C@@H]12 ZINC000880693106 EH On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN2CCCC[C@@H]12 ZINC000880693106 EH On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN2CCCC[C@H]12 ZINC000880693107 EH On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCCN2CCCC[C@H]12 ZINC000880693107 EH On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN2CCCC[C@H]12 ZINC000880693108 EH On-Demand Anodyne CCR3 28 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCCN2CCCC[C@H]12 ZINC000880693108 EH On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)CC2(F)F ZINC000880693109 EI On-Demand Anodyne CACNA1H 53 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)CC2(F)F ZINC000880693109 EI On-Demand Anodyne EPHX2 29 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)CC2(F)F ZINC000880693109 EI On-Demand Anodyne TRPM8 29 40 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693113 DF On-Demand Anodyne EPHX2 48 39 C[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCCC2)O1 ZINC000880693115 EI On-Demand Anodyne CACNA1H 29 41 C[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC2(CCCC2)O1 ZINC000880693116 EI On-Demand Anodyne CACNA1H 29 41 O=C(Nc1ccc(F)c(C(F)F)c1)Nc1ccn(C2CCOCC2)n1 ZINC000880693119 FH On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OC2CCC2)C1 ZINC000880693122 EI On-Demand Anodyne EPHX2 24 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OC2CCC2)C1 ZINC000880693123 EI On-Demand Anodyne EPHX2 24 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]2C[C@H]2C1 ZINC000880693124 CH On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]2C[C@@H]2C1 ZINC000880693125 CH On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H]2C[C@H]2C1 ZINC000880693126 CH On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880693127 CH On-Demand Anodyne RBP4 47 35 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693128 GH On-Demand Anodyne CCR3 51 39 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693128 GH On-Demand Anodyne EPHX2 28 42 O=C(NC[C@H]1CCCN(C(=O)C(F)(F)F)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693128 GH On-Demand Anodyne CACNA1I 48 33 Cn1cc(CCNC(=O)CN2CCCCS2(=O)=O)c2ccccc21 ZINC000880693188 ED On-Demand Anodyne MTNR1A 16 41 O=C(CC[C@@H]1CCc2ccccc21)NCCc1ccoc1 ZINC000880693203 CG On-Demand Anodyne NQO2 17 42 O=C(CC[C@H]1CCc2ccccc21)NCCc1ccoc1 ZINC000880693204 CG On-Demand Anodyne NQO2 17 42 O=C1CC[C@@H](c2ccc(C(=O)NCCc3ccoc3)cc2)N1 ZINC000880693214 CE On-Demand Anodyne PLD1 44 34 O=C1CC[C@H](c2ccc(C(=O)NCCc3ccoc3)cc2)N1 ZINC000880693215 CE On-Demand Anodyne PLD1 44 34 Cn1cc(CCNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c2ccccc21 ZINC000880693220 FG On-Demand Anodyne PLD1 67 40 Cn1cc(CCNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c2ccccc21 ZINC000880693220 FG On-Demand Anodyne PLD2 80 40 Cn1cc(CCNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c2ccccc21 ZINC000880693221 FG On-Demand Anodyne PLD1 67 40 Cn1cc(CCNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c2ccccc21 ZINC000880693221 FG On-Demand Anodyne PLD2 80 40 Cn1ncc(C2CC2)c1CNC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880693225 EG On-Demand Anodyne P2RX7 18 42 C=CCOCCCNC(=O)c1coc(-c2ccccn2)n1 ZINC000880693232 CE On-Demand Mild TBXA2R 26 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2nccnc2C1 ZINC000880693245 DG On-Demand Anodyne MAPK1 51 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2nccnc2C1 ZINC000880693245 DG On-Demand Anodyne P2RY14 48 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880693253 DF On-Demand Anodyne CACNA1H 40 42 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@H](CO)Cc1ccccc1 ZINC000880693255 FH On-Demand Anodyne NPY5R 38 52 CN(C(=O)Nc1ccc(F)c(C(F)F)c1)[C@@H](CO)Cc1ccccc1 ZINC000880693256 FH On-Demand Anodyne NPY5R 38 52 Cn1ncc(C2CC2)c1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693261 EH On-Demand Anodyne PRMT3 44 31 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693279 GH On-Demand Anodyne CCR3 64 39 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693279 GH On-Demand Anodyne EPHX2 31 43 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693279 GH On-Demand Anodyne CACNA1I 62 35 O=C(CCc1ccc(N2CCCS2(=O)=O)cc1)NN=c1cc[nH]cc1F ZINC000880693280 GD On-Demand Reactive CDK1 16 41 N#CC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693282 DH On-Demand Mild CCR3 24 42 N#CC[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693282 DH On-Demand Mild EPHX2 15 44 N#CC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693283 DH On-Demand Mild CCR3 24 42 N#CC[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693283 DH On-Demand Mild EPHX2 15 44 C[C@@H](Cc1ccccn1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693288 DH On-Demand Anodyne GRM4 26 40 C[C@H](Cc1ccccn1)NC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693289 DH On-Demand Anodyne GRM4 26 40 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880693290 EH On-Demand Anodyne CACNA1H 47 43 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880693290 EH On-Demand Anodyne CCR2 16 41 O=C(NCc1nnc(O)n1C1CC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693295 EF On-Demand Anodyne PRMT3 53 35 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693303 DG On-Demand Anodyne EPHX2 55 42 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CO1 ZINC000880693305 CG On-Demand Anodyne EPHX2 40 37 C[C@@]1(C#N)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693317 CH On-Demand Mild CACNA1H 45 43 C[C@@]1(C#N)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693317 CH On-Demand Mild EPHX2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2cc(Cl)nnc2C1 ZINC000880693319 FH On-Demand Anodyne MAPK1 55 42 C[C@H](O)CN(C(=O)Nc1ccc(F)c(C(F)F)c1)C1CC1 ZINC000880693328 DG On-Demand Anodyne MCHR1 34 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880693331 FG On-Demand Anodyne EPHX2 31 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](Nc2ncccn2)C1 ZINC000880693332 FG On-Demand Anodyne EPHX2 31 49 CS(=O)(=O)C1CCC(C(=O)NCCc2ccoc2)CC1 ZINC000880693336 CD On-Demand Anodyne MTNR1A 20 41 O=C(NCCN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693392 DF On-Demand Anodyne CCR3 24 40 O=C(NCCN1CCCC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693392 DF On-Demand Anodyne EPHX2 18 46 Cn1ncc(C2CC2)c1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880693393 EE On-Demand Anodyne GABRA1 17 48 Cn1ncc(C2CC2)c1CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880693393 EE On-Demand Anodyne HTR1F 76 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693397 GF On-Demand Anodyne PGC 45 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693397 GF On-Demand Anodyne PAPA1_CARPA 43 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693397 GF On-Demand Anodyne REN 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693397 GF On-Demand Anodyne FPR1 46 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693399 GF On-Demand Anodyne PGC 45 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693399 GF On-Demand Anodyne PAPA1_CARPA 43 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693399 GF On-Demand Anodyne REN 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](c2ccccc2)CO1 ZINC000880693399 GF On-Demand Anodyne FPR1 46 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(C2(O)CC2)CC1 ZINC000880693411 EH On-Demand Anodyne CACNA1H 44 42 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1C[C@@H](N2CCOCC2)C12CCC2 ZINC000880693413 GH On-Demand Anodyne EPHX2 24 41 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693416 GI On-Demand Clean CCR3 58 37 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693416 GI On-Demand Clean STAT6 47 33 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCC2=O)CC1 ZINC000880693418 EI On-Demand Anodyne CACNA1H 56 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(CO)C1 ZINC000880693421 DD On-Demand Anodyne CACNA1H 47 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(CO)C1 ZINC000880693421 DD On-Demand Anodyne EPHX2 37 43 Cc1cnc(Cl)c(C(=O)NCC2(S(C)(=O)=O)CCCCC2)c1 ZINC000880693431 EF On-Demand Anodyne SLC6A9 48 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880693449 GI On-Demand Anodyne CCR5 21 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@]2(C1)CC2(F)F ZINC000880693453 EI On-Demand Anodyne EPHX2 30 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@]2(C1)CC2(F)F ZINC000880693455 EI On-Demand Anodyne EPHX2 30 43 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693457 EH On-Demand Anodyne EPHX2 43 41 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693459 EH On-Demand Anodyne EPHX2 43 41 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693461 EH On-Demand Anodyne EPHX2 43 41 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693463 EH On-Demand Anodyne EPHX2 43 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1C[C@H](O)C1 ZINC000880693482 CE On-Demand Anodyne EPHX2 49 39 C[C@H](CCO)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693488 CF On-Demand Anodyne NPY5R 34 41 C[C@@H](CCO)N(C)C(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693490 CF On-Demand Anodyne NPY5R 34 41 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCC1=O ZINC000880693491 DE On-Demand Anodyne CACNA1H 42 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(CO)C1 ZINC000880693497 CF On-Demand Anodyne EPHX2 41 39 CCN1CC[C@@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693504 EH On-Demand Anodyne NPY2R 43 34 CCN1CC[C@@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693504 EH On-Demand Anodyne CCR5 26 49 CCN1CC[C@@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693504 EH On-Demand Anodyne MCHR1 45 42 CCN1CC[C@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693505 EH On-Demand Anodyne NPY2R 43 34 CCN1CC[C@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693505 EH On-Demand Anodyne CCR5 26 49 CCN1CC[C@H](N(CC)C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693505 EH On-Demand Anodyne MCHR1 45 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880693512 FJ On-Demand Mild CACNA1H 56 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880693512 FJ On-Demand Mild NPY5R 15 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880693512 FJ On-Demand Mild EPHX2 30 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2ncncc2C1 ZINC000880693517 DG On-Demand Anodyne MAPK1 47 37 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2ncncc2C1 ZINC000880693517 DG On-Demand Anodyne P2RY14 49 38 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C3)c1 ZINC000880693518 GF On-Demand Anodyne P2RX7 23 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880693521 FH On-Demand Anodyne EPHX2 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880693522 FH On-Demand Anodyne EPHX2 36 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CF)C1 ZINC000880693530 DH On-Demand Anodyne CCR3 26 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](CF)C1 ZINC000880693530 DH On-Demand Anodyne EPHX2 22 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CF)C1 ZINC000880693531 DH On-Demand Anodyne CCR3 26 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](CF)C1 ZINC000880693531 DH On-Demand Anodyne EPHX2 22 47 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCF)CC1 ZINC000880693535 DI On-Demand Anodyne CCR3 25 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCF)CC1 ZINC000880693535 DI On-Demand Anodyne EPHX2 40 46 O=C(NCCC[C@@H]1CCOC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693545 EG On-Demand Anodyne CCR3 28 40 O=C(NCCC[C@H]1CCOC1=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693546 EG On-Demand Anodyne CCR3 28 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H]2C[C@]2(O)C1 ZINC000880693554 CE On-Demand Anodyne CACNA1H 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H]2C[C@@]2(O)C1 ZINC000880693555 CE On-Demand Anodyne CACNA1H 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@H]2C[C@]2(O)C1 ZINC000880693556 CE On-Demand Anodyne CACNA1H 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1C[C@@H]2C[C@@]2(O)C1 ZINC000880693557 CE On-Demand Anodyne CACNA1H 31 40 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693565 EJ On-Demand Anodyne CACNA1H 40 43 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880693565 EJ On-Demand Anodyne EPHX2 39 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880693566 GE On-Demand Anodyne EPHX2 24 41 CN1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCC1(C)C ZINC000880693571 EH On-Demand Anodyne CACNA1H 51 44 Cc1csc([C@H]2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)n1 ZINC000880693582 FJ On-Demand Anodyne TRPC6 42 33 Cc1csc([C@H]2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)C2)n1 ZINC000880693582 FJ On-Demand Anodyne TRPC3 40 33 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@H](O)CC1 ZINC000880693588 DG On-Demand Anodyne EPHX2 56 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CC[C@H](O)CC1 ZINC000880693588 DG On-Demand Anodyne CXCR3 15 40 O=C(NCC[C@@H]1CCCS1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693611 DI On-Demand Anodyne PRMT3 40 42 O=C(NCC[C@H]1CCCS1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693612 DI On-Demand Anodyne PRMT3 40 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2cc(C)ccc2o1 ZINC000880693630 GG On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc2cc(C)ccc2o1 ZINC000880693631 GG On-Demand Anodyne PAPA1_CARPA 38 40 C=CC(C)(C)CC(=O)NCCc1cn(C)c2ccccc12 ZINC000880693643 CG On-Demand Mild NQO2 15 45 C=CC(C)(C)CC(=O)NCCc1cn(C)c2ccccc12 ZINC000880693643 CG On-Demand Mild MTNR1A 20 45 C=CC(C)(C)CC(=O)NCCc1cn(C)c2ccccc12 ZINC000880693643 CG On-Demand Mild MTNR1B 16 45 CS(=O)(=O)C1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880693649 ED On-Demand Anodyne HCN1 74 38 CS(=O)(=O)C1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880693649 ED On-Demand Anodyne HCN4 57 36 Cn1cc(CCNC(=O)C2CCC(S(C)(=O)=O)CC2)c2ccccc21 ZINC000880693657 FE On-Demand Anodyne NQO2 29 40 Cn1cc(CCNC(=O)C2CCC(S(C)(=O)=O)CC2)c2ccccc21 ZINC000880693657 FE On-Demand Anodyne MTNR1A 42 46 Cn1cc(CCNC(=O)C2CCC(S(C)(=O)=O)CC2)c2ccccc21 ZINC000880693657 FE On-Demand Anodyne MTNR1B 29 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693663 ED On-Demand Anodyne PAPA1_CARPA 47 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693663 ED On-Demand Anodyne CTSK 21 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693663 ED On-Demand Anodyne CTSL 17 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693663 ED On-Demand Anodyne FPR1 45 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693664 ED On-Demand Anodyne PAPA1_CARPA 47 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693664 ED On-Demand Anodyne CTSK 21 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693664 ED On-Demand Anodyne CTSL 17 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1ccoc1 ZINC000880693664 ED On-Demand Anodyne FPR1 45 40 O=C(CN1CCCCS1(=O)=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693670 FE On-Demand Anodyne DNAE 81 35 O=C(CN1CCCCS1(=O)=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693670 FE On-Demand Anodyne RPA1 40 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(C2CC2)cnn1C ZINC000880693674 FD On-Demand Anodyne PAPA1_CARPA 34 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(C2CC2)cnn1C ZINC000880693675 FD On-Demand Anodyne PAPA1_CARPA 34 40 CS(=O)(=O)C1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880693677 FE On-Demand Anodyne HCN1 53 32 CS(=O)(=O)C1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880693677 FE On-Demand Anodyne HCN4 51 32 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccoc1)C2 ZINC000880693692 CF On-Demand Anodyne NQO2 42 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccoc1)C2 ZINC000880693692 CF On-Demand Anodyne MTNR1A 92 47 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1ccoc1)C2 ZINC000880693692 CF On-Demand Anodyne MTNR1B 80 42 O=C(NC[C@@H]1CCC[C@H]2C[C@@H]21)c1cccn2nccc12 ZINC000880693705 CF On-Demand Anodyne JAK3 17 41 O=C(NC[C@@H]1CCC[C@H]2C[C@@H]21)c1cccn2nccc12 ZINC000880693705 CF On-Demand Anodyne TYK2 20 41 O=C(NC[C@@H]1CCC[C@H]2C[C@H]21)c1cccn2nccc12 ZINC000880693706 CF On-Demand Anodyne JAK3 17 41 O=C(NC[C@@H]1CCC[C@H]2C[C@H]21)c1cccn2nccc12 ZINC000880693706 CF On-Demand Anodyne TYK2 20 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880693770 EG On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880693770 EG On-Demand Anodyne EPHX2 34 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CC1)COCCO2 ZINC000880693770 EG On-Demand Anodyne TRPM8 30 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@H](OC2CCC2)CC1 ZINC000880693771 FJ On-Demand Anodyne EPHX2 38 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880693772 FJ On-Demand Anodyne EPHX2 38 40 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693793 GG On-Demand Anodyne CCR3 27 47 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693793 GG On-Demand Anodyne EPHX2 16 46 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693794 GG On-Demand Anodyne CCR3 27 47 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693794 GG On-Demand Anodyne EPHX2 16 46 CCn1ncc(NC(=O)Nc2ccc(F)c(C(F)F)c2)c1C ZINC000880693795 DH On-Demand Anodyne FPR2 33 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1COCC[C@H]1O ZINC000880693806 DE On-Demand Anodyne EPHX2 24 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(CO)(CO)C1 ZINC000880693838 DE On-Demand Anodyne EPHX2 41 39 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CC(CO)(CO)C1 ZINC000880693838 DE On-Demand Anodyne ENV 42 40 Cn1cc(CCNC(=O)[C@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693844 EE On-Demand Anodyne HTR4 15 41 Cn1cc(CCNC(=O)[C@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693844 EE On-Demand Anodyne MTNR1A 22 42 Cn1cc(CCNC(=O)[C@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693844 EE On-Demand Anodyne MTNR1B 19 44 O=C(NC[C@H]1CCN1C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693845 EH On-Demand Anodyne CCR3 34 41 O=C(NC[C@H]1CCN1C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693845 EH On-Demand Anodyne EPHX2 15 40 Cn1cc(CCNC(=O)[C@@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693846 EE On-Demand Anodyne HTR4 15 41 Cn1cc(CCNC(=O)[C@@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693846 EE On-Demand Anodyne MTNR1A 22 42 Cn1cc(CCNC(=O)[C@@H]2CCc3nncn3CC2)c2ccccc21 ZINC000880693846 EE On-Demand Anodyne MTNR1B 19 44 O=C(NC[C@@H]1CCN1C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693847 EH On-Demand Anodyne CCR3 34 41 O=C(NC[C@@H]1CCN1C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693847 EH On-Demand Anodyne EPHX2 15 40 COCc1csc(CNC(=O)CC[C@@H]2CCc3ccccc32)c1 ZINC000880693848 EI On-Demand Anodyne NQO2 20 43 COCc1csc(CNC(=O)CC[C@H]2CCc3ccccc32)c1 ZINC000880693849 EI On-Demand Anodyne NQO2 20 43 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CCc2cnccn2)CC1 ZINC000880693852 GF On-Demand Anodyne CACNA1H 40 34 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCN(CCc2cnccn2)CC1 ZINC000880693852 GF On-Demand Anodyne FAAH 19 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]13OCCC[C@H]1C3(F)F)C2 ZINC000880693853 FF On-Demand Anodyne MTNR1A 32 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]13OCCC[C@H]1C3(F)F)C2 ZINC000880693853 FF On-Demand Anodyne MTNR1B 29 43 CONC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880693854 EF On-Demand Anodyne EPHX2 33 40 O=C(C[C@H]1CCNC1=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693859 DE On-Demand Anodyne DNAE 47 33 O=C(C[C@@H]1CCNC1=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880693860 DE On-Demand Anodyne DNAE 47 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]12OCCC[C@H]1C2(F)F ZINC000880693862 GD On-Demand Anodyne PAPA1_CARPA 31 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]12OCCC[C@H]1C2(F)F ZINC000880693863 GD On-Demand Anodyne PAPA1_CARPA 31 40 Cn1cc(CCNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)c2ccccc21 ZINC000880693865 FE On-Demand Anodyne MTNR1A 25 43 Cn1cc(CCNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)c2ccccc21 ZINC000880693865 FE On-Demand Anodyne MTNR1B 19 43 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H](c1ccccn1)C1CCC1 ZINC000880693888 EJ On-Demand Anodyne GRM4 40 41 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H](c1ccccn1)C1CCC1 ZINC000880693891 EJ On-Demand Anodyne GRM4 40 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C3CC3)cnn1C)C2 ZINC000880693892 EF On-Demand Anodyne MTNR1A 32 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C3CC3)cnn1C)C2 ZINC000880693892 EF On-Demand Anodyne MTNR1B 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)NC1CCC2(CC1)COC2 ZINC000880693900 EH On-Demand Anodyne EPHX2 46 40 Cn1ccnc1[C@@H]1OCCC[C@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880693939 GH On-Demand Anodyne PRMT3 46 34 O=C(NC[C@@H](O)[C@@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693940 DE On-Demand Anodyne PRMT3 31 40 O=C(NC[C@H](O)[C@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693941 DE On-Demand Anodyne PRMT3 31 40 O=C(NC[C@H](O)[C@@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693942 DE On-Demand Anodyne PRMT3 31 40 O=C(NC[C@@H](O)[C@H]1CCCO1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693943 DE On-Demand Anodyne PRMT3 31 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCCO2)CC1 ZINC000880693944 EI On-Demand Anodyne CACNA1H 39 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCCO2)CC1 ZINC000880693944 EI On-Demand Anodyne EPHX2 33 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC2(CCCCO2)CC1 ZINC000880693944 EI On-Demand Anodyne TRPM8 30 41 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(NC2CCOCC2)CC1 ZINC000880693952 FH On-Demand Anodyne EPHX2 33 41 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693954 DD On-Demand Anodyne CCR3 66 50 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693954 DD On-Demand Anodyne EPHX2 23 45 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693954 DD On-Demand Anodyne MCHR1 30 43 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693956 DD On-Demand Anodyne CCR3 66 50 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693956 DD On-Demand Anodyne EPHX2 23 45 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(F)c(C(F)F)c1 ZINC000880693956 DD On-Demand Anodyne MCHR1 30 43 Cn1ncc(C2CC2)c1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880693964 FG On-Demand Anodyne PDE4D 17 44 Cn1ncc(C2CC2)c1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880693964 FG On-Demand Anodyne CACNA1I 42 38 O=C(COC1CC1)NCC1(Cc2ccc(Br)cc2)CC1 ZINC000880693967 EG On-Demand Anodyne TIMP3 47 32 C=CCOCCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880693969 DF On-Demand Mild NQO2 35 44 C=CCOCCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880693969 DF On-Demand Mild MTNR1A 60 42 C=CCOCCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880693969 DF On-Demand Mild MTNR1B 54 40 C=CCOCCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880693970 DF On-Demand Mild NQO2 35 44 C=CCOCCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880693970 DF On-Demand Mild MTNR1A 60 42 C=CCOCCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880693970 DF On-Demand Mild MTNR1B 54 40 Cn1ncc(C2CC2)c1CNC(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880694001 GH On-Demand Anodyne P2RX7 34 44 Cn1ncc(C2CC2)c1CNC(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880694001 GH On-Demand Anodyne RBP4 41 32 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@@H](C(F)F)CC1 ZINC000880694012 EH On-Demand Anodyne EPHX2 32 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCO[C@H](C(F)F)CC1 ZINC000880694013 EH On-Demand Anodyne EPHX2 32 42 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694016 EH On-Demand Anodyne P2RX7 15 47 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694016 EH On-Demand Anodyne DNAE 50 30 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694018 EH On-Demand Anodyne P2RX7 15 47 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694018 EH On-Demand Anodyne DNAE 50 30 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694020 EH On-Demand Anodyne P2RX7 15 47 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694020 EH On-Demand Anodyne DNAE 50 30 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694022 EH On-Demand Anodyne P2RX7 15 47 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000880694022 EH On-Demand Anodyne DNAE 50 30 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne CACNA1H 34 40 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne HTR1D 18 44 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne HTR1B 19 44 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne EPHX2 25 43 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne SCD1 18 40 CN1CCN(C2CCN(C(=O)Nc3ccc(F)c(C(F)F)c3)CC2)CC1 ZINC000880694027 FG On-Demand Anodyne L3MBTL3 73 42 Cn1cc(CCNC(=O)Cc2ccccc2N2CCCC2=O)c2ccccc21 ZINC000880694031 GG On-Demand Anodyne MTNR1A 15 40 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694033 DH On-Demand Anodyne CACNA1H 30 40 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694033 DH On-Demand Anodyne EPHX2 22 42 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694035 DH On-Demand Anodyne CACNA1H 30 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694035 DH On-Demand Anodyne EPHX2 22 42 O=C(NCc1ccc(Cl)c(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880694038 EF On-Demand Anodyne P2RX7 24 48 O=C(NCc1ccc(Cl)c(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880694038 EF On-Demand Anodyne CCR3 17 41 O=C(NCc1ccc(Cl)c(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880694038 EF On-Demand Anodyne EPHX2 18 54 O=C(NCc1ccc(Cl)c(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880694038 EF On-Demand Anodyne DNAE 79 34 O=C(NCc1ccc(Cl)c(Cl)c1)[C@@H]1CCc2nncn2CC1 ZINC000880694038 EF On-Demand Anodyne RPA1 63 36 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(CO)CC1 ZINC000880694039 EE On-Demand Anodyne CACNA1H 63 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(CO)CC1 ZINC000880694039 EE On-Demand Anodyne S1PR2 27 40 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CO)(CO)CC1 ZINC000880694039 EE On-Demand Anodyne EPHX2 30 40 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880694040 EF On-Demand Anodyne P2RX7 24 48 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880694040 EF On-Demand Anodyne CCR3 17 41 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880694040 EF On-Demand Anodyne EPHX2 18 54 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880694040 EF On-Demand Anodyne DNAE 79 34 O=C(NCc1ccc(Cl)c(Cl)c1)[C@H]1CCc2nncn2CC1 ZINC000880694040 EF On-Demand Anodyne RPA1 63 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne NQO2 21 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne CCKAR 54 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne CTSL 15 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne CCKBR 17 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694050 GF On-Demand Anodyne FPR1 45 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne NQO2 21 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne CCKAR 54 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne CTSL 15 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne CCKBR 17 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cn(C)c2ccccc12 ZINC000880694052 GF On-Demand Anodyne FPR1 45 42 O=C(NCCO)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880694053 FE On-Demand Anodyne EPHX2 27 42 C=CCOCCCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880694056 DE On-Demand Mild MPO 52 37 CS[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694059 DH On-Demand Anodyne EPHX2 42 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880694060 GJ On-Demand Anodyne SMO 39 49 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880694060 GJ On-Demand Anodyne ETHR 62 45 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)CC1 ZINC000880694066 CH On-Demand Anodyne CACNA1H 40 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)CC1 ZINC000880694066 CH On-Demand Anodyne EPHX2 44 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(F)CC1 ZINC000880694066 CH On-Demand Anodyne SCD1 16 43 O=C(NCC[C@@H]1CCCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694074 DH On-Demand Anodyne PRMT3 25 43 O=C(NCC[C@H]1CCCOC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694075 DH On-Demand Anodyne PRMT3 25 43 C[C@@]1(CO)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@]1(C)CO ZINC000880694078 EF On-Demand Anodyne CACNA1H 27 40 C[C@@]1(CO)CN(C(=O)Nc2ccc(F)c(C(F)F)c2)C[C@]1(C)CO ZINC000880694078 EF On-Demand Anodyne EPHX2 24 40 CCN1CC[C@@H]1CNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880694091 DF On-Demand Anodyne CCR3 50 38 O=C(NCC[C@@H]1CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694093 DI On-Demand Anodyne PRMT3 40 42 O=C(NCC[C@H]1CCSC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694095 DI On-Demand Anodyne PRMT3 40 42 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694107 GG On-Demand Anodyne CACNA1H 35 41 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694107 GG On-Demand Anodyne EPHX2 36 44 N#CCc1cccc2c1CCN(C(=O)Nc1ccc(F)c(C(F)F)c1)C2 ZINC000880694124 FI On-Demand Mild P2RY14 46 35 COc1ccccc1[C@@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880694133 GI On-Demand Anodyne RBP4 28 40 COc1ccccc1[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 ZINC000880694134 GI On-Demand Anodyne RBP4 28 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC[C@H]1O ZINC000880694135 DE On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1CCOC[C@@H]1O ZINC000880694136 DE On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC[C@@H]1O ZINC000880694137 DE On-Demand Anodyne EPHX2 20 40 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@H]1CCOC[C@H]1O ZINC000880694138 DE On-Demand Anodyne EPHX2 20 40 COc1ccc(CN(CCO)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1 ZINC000880694144 FH On-Demand Anodyne BMP1 35 42 COc1ccc(CN(CCO)C(=O)Nc2ccc(F)c(C(F)F)c2)cc1 ZINC000880694144 FH On-Demand Anodyne ROCK2 16 46 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCO)(CCO)CC1 ZINC000880694148 FG On-Demand Anodyne CACNA1H 50 42 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCC(CCO)(CCO)CC1 ZINC000880694148 FG On-Demand Anodyne EPHX2 27 42 CS(=O)(=O)C1(CNC(=O)c2ncccc2-c2ccccn2)CCCCC1 ZINC000880694149 FF On-Demand Anodyne HCN1 51 32 CS(=O)(=O)C1(CNC(=O)c2ncccc2-c2ccccn2)CCCCC1 ZINC000880694149 FF On-Demand Anodyne HCN4 48 32 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880694164 DI On-Demand Mild EPHX2 46 43 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694174 ED On-Demand Anodyne CACNA1H 50 43 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)C1 ZINC000880694174 ED On-Demand Anodyne EPHX2 35 44 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2nc(C3CC3)ncc2C1 ZINC000880694175 FI On-Demand Anodyne MAPK1 53 38 O=C(Nc1ccc(F)c(C(F)F)c1)N1CCc2nc(C3CC3)ncc2C1 ZINC000880694175 FI On-Demand Anodyne P2RY14 43 33 O=C(NC[C@@]12COCCN1C(=O)COC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880694177 FD On-Demand Anodyne EPHX2 21 40 O=C(NC[C@]12COCCN1C(=O)COC2)Nc1ccc(F)c(C(F)F)c1 ZINC000880694178 FD On-Demand Anodyne EPHX2 21 40 O=C(NCC[C@H](O)C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694183 EH On-Demand Anodyne CCR3 29 41 O=C(NCC[C@H](O)C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694183 EH On-Demand Anodyne PRMT3 35 44 O=C(NCC[C@@H](O)C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694184 EH On-Demand Anodyne CCR3 29 41 O=C(NCC[C@@H](O)C1CCCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694184 EH On-Demand Anodyne PRMT3 35 44 Cn1nnnc1C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880694186 FF On-Demand Anodyne CCR3 42 30 O=C(NNC(=O)C1CCOCC1)Nc1ccc(F)c(C(F)F)c1 ZINC000880694191 EE On-Demand Reactive EPHX2 24 42 CC(C)[C@H]1CN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCN1C ZINC000880694202 EH On-Demand Anodyne CACNA1H 28 40 NC(=O)[C@@H]1CCCN1CCCNC(=O)Nc1ccc(F)c(C(F)F)c1 ZINC000880694203 FE On-Demand Anodyne CCR3 51 46 O=C(Nc1ccc(F)c(C(F)F)c1)N[C@@H]1C[C@H](CO)C1 ZINC000880694204 CF On-Demand Anodyne EPHX2 41 39 CC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880694226 DH On-Demand Anodyne CACNA1H 37 44 CC(=O)C1CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CC1 ZINC000880694226 DH On-Demand Anodyne EPHX2 38 41 O=C(COC1CC1)NCc1ccc(Cl)c(Cl)c1 ZINC000880694237 CF On-Demand Anodyne P2RX7 23 49 O=C(COC1CC1)NCc1ccc(Cl)c(Cl)c1 ZINC000880694237 CF On-Demand Anodyne CCR3 30 41 O=C(COC1CC1)NCc1ccc(Cl)c(Cl)c1 ZINC000880694237 CF On-Demand Anodyne PDE6A 44 35 O=C(COC1CC1)NCc1ccc(Cl)c(Cl)c1 ZINC000880694237 CF On-Demand Anodyne SSTR3 15 44 O=C(COC1CC1)NCc1ccc(Cl)c(Cl)c1 ZINC000880694237 CF On-Demand Anodyne DNAE 80 33 Cn1nc2c(c1C(=O)NCc1ccc(Cl)c(Cl)c1)CSCC2 ZINC000880694242 FG On-Demand Anodyne DNAE 67 32 Cn1nc2c(c1C(=O)NCc1ccc(Cl)c(Cl)c1)CSCC2 ZINC000880694242 FG On-Demand Anodyne RPA1 43 35 C=CCOCCCNC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880694324 DF On-Demand Mild HDAC10 18 49 C=CCOCCCNC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880694324 DF On-Demand Mild PDK1 45 33 Cn1cc(CCNC(=O)COC2CC2)c2ccccc21 ZINC000880694398 CE On-Demand Anodyne HTR4 26 42 Cn1cc(CCNC(=O)COC2CC2)c2ccccc21 ZINC000880694398 CE On-Demand Anodyne NQO2 21 48 Cn1cc(CCNC(=O)COC2CC2)c2ccccc21 ZINC000880694398 CE On-Demand Anodyne MTNR1A 52 48 Cn1cc(CCNC(=O)COC2CC2)c2ccccc21 ZINC000880694398 CE On-Demand Anodyne MTNR1B 38 48 Cn1ncc(C2CC2)c1CNC(=O)c1cncc2[nH]ccc12 ZINC000880694431 CE On-Demand Anodyne HTR1F 42 32 C=CCOCCCNC(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880694443 EF On-Demand Mild KCNA3 40 36 Cn1cc(CCNC(=O)c2ccc(CN3CCOCC3)o2)c2ccccc21 ZINC000880694457 FF On-Demand Anodyne CNR2 16 41 Cn1cc(CCNC(=O)c2ccc(CN3CCOCC3)o2)c2ccccc21 ZINC000880694457 FF On-Demand Anodyne PTGDS 43 38 Cn1cc(CCNC(=O)c2ccc(CN3CCOCC3)o2)c2ccccc21 ZINC000880694457 FF On-Demand Anodyne DPOL_VZVD 25 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@H]2C[C@@H]21 ZINC000880694482 EE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@@H]2C[C@@H]12 ZINC000880694483 EE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@@H]2C[C@H]12 ZINC000880694484 EE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@H]2C[C@H]21 ZINC000880694485 EE On-Demand Anodyne PAPA1_CARPA 35 43 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880694597 FD On-Demand Anodyne CCR3 15 45 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880694598 FD On-Demand Anodyne CCR3 15 45 COc1ccccc1-c1ccc(C(=O)NCC[C@]2(C)CC2(F)F)c(O)n1 ZINC000880694710 FH On-Demand Anodyne DRD2 21 41 COc1ccccc1-c1ccc(C(=O)NCC[C@]2(C)CC2(F)F)c(O)n1 ZINC000880694710 FH On-Demand Anodyne DRD3 39 41 COc1ccccc1-c1ccc(C(=O)NCC[C@@]2(C)CC2(F)F)c(O)n1 ZINC000880694714 FH On-Demand Anodyne DRD2 21 41 COc1ccccc1-c1ccc(C(=O)NCC[C@@]2(C)CC2(F)F)c(O)n1 ZINC000880694714 FH On-Demand Anodyne DRD3 39 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@H](C)O1 ZINC000880694721 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCC[C@@H](C)O1 ZINC000880694722 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCC[C@H](C)O1 ZINC000880694723 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCC[C@@H](C)O1 ZINC000880694724 ED On-Demand Anodyne PAPA1_CARPA 35 43 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694771 FF On-Demand Anodyne SLC6A4 16 41 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694771 FF On-Demand Anodyne SLC6A3 33 42 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694772 FF On-Demand Anodyne SLC6A4 16 41 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694772 FF On-Demand Anodyne SLC6A3 33 42 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3CCN(C4CCCCC4)C3)cc2)N1 ZINC000880694794 FF On-Demand Anodyne SLC6A5 26 43 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCN(C4CCCCC4)C3)cc2)N1 ZINC000880694795 FF On-Demand Anodyne SLC6A5 26 43 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCN(C4CCCCC4)C3)cc2)N1 ZINC000880694796 FF On-Demand Anodyne SLC6A5 26 43 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3CCN(C4CCCCC4)C3)cc2)N1 ZINC000880694797 FF On-Demand Anodyne SLC6A5 26 43 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694817 GH On-Demand Anodyne DRD4 18 49 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694817 GH On-Demand Anodyne DRD3 19 54 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694817 GH On-Demand Anodyne HTR3A 29 45 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694818 GH On-Demand Anodyne DRD4 18 49 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694818 GH On-Demand Anodyne DRD3 19 54 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C3CCCCC3)C2)c(O)n1 ZINC000880694818 GH On-Demand Anodyne HTR3A 29 45 COC[C@@H]1CCCN1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694831 EE On-Demand Anodyne CASP7 43 38 O=C(NCc1cccnc1N1CCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694833 GG On-Demand Anodyne SCN2A 17 41 O=C(NCc1cccnc1N1CCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880694833 GG On-Demand Anodyne SCN10A 19 41 CC(C)(C)OC(=O)N1CCO[C@H](c2ccc(NC(=O)COC3CC3)cc2)C1 ZINC000880694884 GG On-Demand Anodyne GPR119 28 42 CC(C)(C)OC(=O)N1CCO[C@@H](c2ccc(NC(=O)COC3CC3)cc2)C1 ZINC000880694885 GG On-Demand Anodyne GPR119 28 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H](CCF)C3)cc2)N1 ZINC000880694915 DF On-Demand Anodyne L3MBTL3 40 36 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@H](CCF)C3)cc2)N1 ZINC000880694917 DF On-Demand Anodyne L3MBTL3 40 36 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@H](CCF)C3)cc2)N1 ZINC000880694919 DF On-Demand Anodyne L3MBTL3 40 36 O=C(NCCCC1CCC1)c1cccn2nccc12 ZINC000880694920 CF On-Demand Anodyne BMP1 43 33 O=C(NCCCC1CCC1)c1cccn2nccc12 ZINC000880694920 CF On-Demand Anodyne JAK3 17 41 O=C(NCCCC1CCC1)c1cccn2nccc12 ZINC000880694920 CF On-Demand Anodyne TYK2 20 41 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H](CCF)C3)cc2)N1 ZINC000880694921 DF On-Demand Anodyne L3MBTL3 40 36 Cc1coc(C(=O)N[C@@H]2CCN(C3CCCCC3)C2)c1 ZINC000880694950 CF On-Demand Anodyne SLC6A5 17 40 Cc1coc(C(=O)N[C@H]2CCN(C3CCCCC3)C2)c1 ZINC000880694951 CF On-Demand Anodyne SLC6A5 17 40 O=C(NCCCC1CCC1)[C@@H]1CCc2nncn2CC1 ZINC000880694972 CD On-Demand Anodyne TBK1 59 33 O=C(NCCCC1CCC1)[C@H]1CCc2nncn2CC1 ZINC000880694973 CD On-Demand Anodyne TBK1 59 33 C[C@]1(CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1(F)F ZINC000880694978 EH On-Demand Anodyne PDE4D 15 41 C[C@@]1(CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1(F)F ZINC000880694979 EH On-Demand Anodyne PDE4D 15 41 O=C(/C=C/c1cccnc1)Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2)s1 ZINC000880695060 HK On-Demand Anodyne RORC 15 46 O=C(/C=C\c1cccnc1)Nc1nc(-c2ccccc2)c(C(=O)c2ccccc2)s1 ZINC000880695065 HK On-Demand Anodyne RORC 15 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1nccc(OC)c1F ZINC000880695083 FD On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1nccc(OC)c1F ZINC000880695087 FD On-Demand Anodyne PAPA1_CARPA 39 42 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1cccn2nccc12 ZINC000880695137 DE On-Demand Anodyne JAK3 15 41 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1cccn2nccc12 ZINC000880695137 DE On-Demand Anodyne TYK2 17 41 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1cccn2nccc12 ZINC000880695138 DE On-Demand Anodyne JAK3 15 41 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1cccn2nccc12 ZINC000880695138 DE On-Demand Anodyne TYK2 17 41 O=C(NCCCC1CCC1)c1coc(-c2ccccn2)n1 ZINC000880695156 CG On-Demand Anodyne TBXA2R 39 53 O=C(NCCCC1CCC1)c1coc(-c2ccccn2)n1 ZINC000880695156 CG On-Demand Anodyne BMP1 33 42 COc1ccccc1-c1ccc(C(=O)NCCCC2CCC2)c(O)n1 ZINC000880695183 EH On-Demand Anodyne DRD2 34 42 COc1ccccc1-c1ccc(C(=O)NCCCC2CCC2)c(O)n1 ZINC000880695183 EH On-Demand Anodyne DRD3 51 42 COc1ccccc1-c1ccc(C(=O)NCCCC2CCC2)c(O)n1 ZINC000880695183 EH On-Demand Anodyne KCNA3 41 35 COc1ccccc1-c1ccc(C(=O)NCCCC2CCC2)c(O)n1 ZINC000880695183 EH On-Demand Anodyne TYRO3 16 43 CN1CCN(C2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)CC1 ZINC000880695209 GE On-Demand Anodyne L3MBTL3 50 39 CS(=O)(=O)C1CCC(C(=O)N[C@H]2CCN(C3CCCCC3)C2)CC1 ZINC000880695210 FE On-Demand Anodyne EPHX2 19 49 CS(=O)(=O)C1CCC(C(=O)N[C@@H]2CCN(C3CCCCC3)C2)CC1 ZINC000880695211 FE On-Demand Anodyne EPHX2 19 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)CC1(F)F ZINC000880695217 EE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)CC1(F)F ZINC000880695218 EE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)CC1(F)F ZINC000880695219 EE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)CC1(F)F ZINC000880695220 EE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@]1(C)CC1(F)F ZINC000880695276 FE On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@]1(C)CC1(F)F ZINC000880695278 FE On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@]1(C)CC1(F)F ZINC000880695280 FE On-Demand Anodyne PAPA1_CARPA 40 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@]1(C)CC1(F)F ZINC000880695282 FE On-Demand Anodyne PAPA1_CARPA 40 46 O=C(NCCCC1CCC1)c1ccc(CN2CCOCC2)o1 ZINC000880695297 DE On-Demand Anodyne ACHE 15 40 C[C@]1(CNC(=O)c2cccn3nccc23)CC1(F)F ZINC000880695378 CE On-Demand Anodyne HCN1 69 32 C[C@]1(CNC(=O)c2cccn3nccc23)CC1(F)F ZINC000880695378 CE On-Demand Anodyne HCN4 47 30 C[C@@]1(CNC(=O)c2cccn3nccc23)CC1(F)F ZINC000880695379 CE On-Demand Anodyne HCN1 69 32 C[C@@]1(CNC(=O)c2cccn3nccc23)CC1(F)F ZINC000880695379 CE On-Demand Anodyne HCN4 47 30 C[C@]1(CNC(=O)c2ncsc2C2CC2)CC1(F)F ZINC000880695390 CF On-Demand Anodyne MAP1 41 34 C[C@@]1(CNC(=O)c2ncsc2C2CC2)CC1(F)F ZINC000880695391 CF On-Demand Anodyne MAP1 41 34 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@H](CCF)C1 ZINC000880695459 FI On-Demand Anodyne RBP4 41 34 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC[C@@H](CCF)C1 ZINC000880695460 FI On-Demand Anodyne RBP4 41 34 CCN1CC[C@H](N(CC)C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880695517 EF On-Demand Anodyne WNT3A 42 36 CCN1CC[C@@H](N(CC)C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880695518 EF On-Demand Anodyne WNT3A 42 36 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1cnc2cc[nH]c2c1 ZINC000880695617 DF On-Demand Anodyne JAK1 43 38 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1cnc2cc[nH]c2c1 ZINC000880695617 DF On-Demand Anodyne SLC6A5 18 41 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1cnc2cc[nH]c2c1 ZINC000880695619 DF On-Demand Anodyne JAK1 43 38 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1cnc2cc[nH]c2c1 ZINC000880695619 DF On-Demand Anodyne SLC6A5 18 41 C[C@H]1CCC[C@@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)O1 ZINC000880695667 DF On-Demand Anodyne GABRA1 16 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(C)CC1(F)F)C2 ZINC000880695762 DF On-Demand Anodyne NQO2 32 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(C)CC1(F)F)C2 ZINC000880695762 DF On-Demand Anodyne MTNR1A 50 49 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@]1(C)CC1(F)F)C2 ZINC000880695762 DF On-Demand Anodyne MTNR1B 43 49 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(C)CC1(F)F)C2 ZINC000880695767 DF On-Demand Anodyne NQO2 32 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(C)CC1(F)F)C2 ZINC000880695767 DF On-Demand Anodyne MTNR1A 50 49 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@]1(C)CC1(F)F)C2 ZINC000880695767 DF On-Demand Anodyne MTNR1B 43 49 O=C(NCCCC1CCC1)c1ncccc1-c1ccccn1 ZINC000880695769 CG On-Demand Anodyne BMP1 15 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCCCC2CCC2)N1Cc1ccccc1 ZINC000880695770 EE On-Demand Anodyne FKBP1A 18 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCCCC2CCC2)N1Cc1ccccc1 ZINC000880695770 EE On-Demand Anodyne ACHE 28 41 CCC1(CC)CCCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880695796 EH On-Demand Anodyne L3MBTL3 43 35 CCC1(CC)CCCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880695797 EH On-Demand Anodyne L3MBTL3 43 35 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCCCC3)C2)N1Cc1ccccc1 ZINC000880695858 GE On-Demand Anodyne SIGMAR1 23 46 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCCCC3)C2)N1Cc1ccccc1 ZINC000880695858 GE On-Demand Anodyne SLC6A5 16 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCCCC3)C2)N1Cc1ccccc1 ZINC000880695859 GE On-Demand Anodyne SIGMAR1 23 46 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCCCC3)C2)N1Cc1ccccc1 ZINC000880695859 GE On-Demand Anodyne SLC6A5 16 41 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)CC2(F)F)c(O)n1 ZINC000880695903 EG On-Demand Anodyne KCNA3 45 40 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)CC2(F)F)c(O)n1 ZINC000880695903 EG On-Demand Anodyne HCN1 62 37 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)CC2(F)F)c(O)n1 ZINC000880695904 EG On-Demand Anodyne KCNA3 45 40 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)CC2(F)F)c(O)n1 ZINC000880695904 EG On-Demand Anodyne HCN1 62 37 O=C(NNC(=O)C1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695905 ED On-Demand Reactive WNT3A 44 30 O=C(NCCN1CC[C@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695990 ED On-Demand Anodyne CCR3 46 43 O=C(NCCN1CC[C@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695990 ED On-Demand Anodyne PLD2 50 33 O=C(NCCN1CC[C@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695990 ED On-Demand Anodyne WNT3A 47 32 O=C(NCCN1CC[C@@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695991 ED On-Demand Anodyne CCR3 46 43 O=C(NCCN1CC[C@@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695991 ED On-Demand Anodyne PLD2 50 33 O=C(NCCN1CC[C@@H](O)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880695991 ED On-Demand Anodyne WNT3A 47 32 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880696046 GG On-Demand Anodyne EPHX2 49 41 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1ccc(CN2CCOCC2)o1 ZINC000880696130 FE On-Demand Anodyne SIGMAR1 16 43 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1ccc(CN2CCOCC2)o1 ZINC000880696130 FE On-Demand Anodyne SLC6A5 21 41 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1ccc(CN2CCOCC2)o1 ZINC000880696131 FE On-Demand Anodyne SIGMAR1 16 43 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1ccc(CN2CCOCC2)o1 ZINC000880696131 FE On-Demand Anodyne SLC6A5 21 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCN(C2CCCCC2)C1 ZINC000880696174 FF On-Demand Anodyne OPRL1 17 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCN(C2CCCCC2)C1 ZINC000880696174 FF On-Demand Anodyne SIGMAR1 23 43 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1CCN(C2CCCCC2)C1 ZINC000880696175 FF On-Demand Anodyne OPRL1 17 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1CCN(C2CCCCC2)C1 ZINC000880696175 FF On-Demand Anodyne SIGMAR1 23 43 O=C(N[C@H]1CCN(C2CCCCC2)C1)c1ncccc1-c1ccccn1 ZINC000880696267 FG On-Demand Anodyne SLC6A5 16 40 O=C(N[C@@H]1CCN(C2CCCCC2)C1)c1ncccc1-c1ccccn1 ZINC000880696268 FG On-Demand Anodyne SLC6A5 16 40 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880696325 FF On-Demand Anodyne HCRTR1 22 40 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)CC1(F)F)C2 ZINC000880696375 DG On-Demand Anodyne NQO2 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)CC1(F)F)C2 ZINC000880696375 DG On-Demand Anodyne MTNR1A 57 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@]1(C)CC1(F)F)C2 ZINC000880696375 DG On-Demand Anodyne MTNR1B 47 43 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)CC1(F)F)C2 ZINC000880696376 DG On-Demand Anodyne NQO2 38 42 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)CC1(F)F)C2 ZINC000880696376 DG On-Demand Anodyne MTNR1A 57 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@]1(C)CC1(F)F)C2 ZINC000880696376 DG On-Demand Anodyne MTNR1B 47 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nccc(OC)c1F)C2 ZINC000880696409 EF On-Demand Anodyne NQO2 29 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nccc(OC)c1F)C2 ZINC000880696409 EF On-Demand Anodyne RAF1 16 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nccc(OC)c1F)C2 ZINC000880696409 EF On-Demand Anodyne MTNR1A 31 41 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1ccnn1-c1ccc(F)cc1 ZINC000880696456 FD On-Demand Anodyne WNT3A 45 31 CC(C)(C[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1)C(N)=O ZINC000880696539 GG On-Demand Anodyne CCR3 66 35 CC(C)(C[C@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1)C(N)=O ZINC000880696542 GG On-Demand Anodyne CCR3 66 35 COC(=O)N1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880696686 FE On-Demand Anodyne EPHX2 45 39 O=C(C[C@@H]1C[C@H]1C1CC1)Nc1ccc2c(c1)CCOC2 ZINC000880696775 CG On-Demand Anodyne PTPRF 42 33 CN1CCO[C@@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)[C@@H]1c1cnn(C)c1 ZINC000880696776 GD On-Demand Anodyne PLD2 41 36 O=C(Nc1ccc2c(c1)CCOC2)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880696782 EH On-Demand Anodyne PTPRF 42 32 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccnn1-c1ccc(F)cc1)C2 ZINC000880696916 EF On-Demand Anodyne HTR3A 29 41 COc1cccc([C@]2(C)CCN(C(=O)C3CCC(S(C)(=O)=O)CC3)C2)c1 ZINC000880696947 GF On-Demand Anodyne MTNR1B 15 43 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)CCCNC(=O)C(C)(C)C)C2 ZINC000880697134 GD On-Demand Reactive NQO2 32 46 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)CCCNC(=O)C(C)(C)C)C2 ZINC000880697134 GD On-Demand Reactive MTNR1A 44 38 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)CCCNC(=O)C(C)(C)C)C2 ZINC000880697134 GD On-Demand Reactive MTNR1B 40 39 CN1CCO[C@H]2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@H]21 ZINC000880697297 FD On-Demand Anodyne HTR1F 41 33 CN1CCO[C@H]2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@@H]21 ZINC000880697298 FD On-Demand Anodyne HTR1F 41 33 CN1CCO[C@@H]2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@H]21 ZINC000880697299 FD On-Demand Anodyne HTR1F 41 33 CC(CO)(CO)CNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697323 DD On-Demand Anodyne NR3C1 16 41 CN1CCO[C@@H]2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@@H]21 ZINC000880697403 FD On-Demand Anodyne HTR1F 41 33 COc1cccc([C@]2(C)CCN(C(=O)c3nnn(C)n3)C2)c1 ZINC000880697414 DD On-Demand Anodyne TACR2 16 41 CC(C)(C)C(=O)NCCCC(=O)NNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880697543 FF On-Demand Reactive NQO2 21 44 CC(C)(C)C(=O)NCCCC(=O)NNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880697544 FF On-Demand Reactive NQO2 21 44 CN1CCC[C@@H](CCNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880697565 EF On-Demand Anodyne CCR3 98 43 O=C(C(=O)N1CCC[C@H](CCF)C1)c1c[nH]c2cc(F)ccc12 ZINC000880697628 DG On-Demand Anodyne GRIN2B 15 56 O=C(C(=O)N1CCC[C@H](CCF)C1)c1c[nH]c2cc(F)ccc12 ZINC000880697628 DG On-Demand Anodyne MPO 51 35 O=C(C(=O)N1CCC[C@@H](CCF)C1)c1c[nH]c2cc(F)ccc12 ZINC000880697629 DG On-Demand Anodyne GRIN2B 15 56 O=C(C(=O)N1CCC[C@@H](CCF)C1)c1c[nH]c2cc(F)ccc12 ZINC000880697629 DG On-Demand Anodyne MPO 51 35 O=C(NC[C@H]1CCCN1CCCO)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697712 FD On-Demand Anodyne CCR3 35 40 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697759 EF On-Demand Anodyne CHRNA10 40 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697759 EF On-Demand Anodyne ACKR3 64 36 CN(C[C@H]1CCCN1C)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697760 EF On-Demand Anodyne CHRNA10 40 33 CN(C[C@H]1CCCN1C)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697760 EF On-Demand Anodyne ACKR3 64 36 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H](CCF)C2)N1Cc1ccccc1 ZINC000880697765 FE On-Demand Anodyne PREP 83 41 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H](CCF)C2)N1Cc1ccccc1 ZINC000880697766 FE On-Demand Anodyne PREP 83 41 CC(=O)N1CCC[C@@H]1C(=O)NNC(=O)c1cccc(Cl)n1 ZINC000880697817 DC On-Demand Reactive ELANE 77 37 CC(=O)N1CCC[C@@H]1C(=O)NNC(=O)c1cccc(Cl)n1 ZINC000880697817 DC On-Demand Reactive PREP 44 34 CC(=O)N1CCC[C@@H]1C(=O)NNC(=O)c1cccc(Cl)n1 ZINC000880697817 DC On-Demand Reactive LGMN 65 33 CC(=O)N1CCC[C@@H]1C(=O)NNC(=O)c1cccc(Cl)n1 ZINC000880697817 DC On-Demand Reactive XIAP 46 38 CC(=O)N1CCC[C@@H]1C(=O)NNC(=O)c1cccc(Cl)n1 ZINC000880697817 DC On-Demand Reactive BRCA1 51 32 C#C[C@@H]1COCCN1C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697881 DD On-Demand Mild WNT3A 43 30 C#C[C@H]1COCCN1C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880697882 DD On-Demand Mild WNT3A 43 30 Cc1cc(N2CCC[C@H](NC(=O)Nc3ccnn3-c3ccc(F)cc3)C2)n(C)n1 ZINC000880697958 GF On-Demand Anodyne CCR3 46 33 O=C(NCCN1CC=CCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698014 EE On-Demand Anodyne PLD2 51 35 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698095 FE On-Demand Anodyne CCR3 111 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698096 FE On-Demand Anodyne CCR3 111 41 COc1cccc([C@]2(C)CCN(C(=O)c3cnc4cc[nH]c4c3)C2)c1 ZINC000880698249 EG On-Demand Anodyne TACR2 15 40 COc1cccc([C@]2(C)CCN(C(=O)c3cnc4cc[nH]c4c3)C2)c1 ZINC000880698249 EG On-Demand Anodyne ACACA 21 45 COc1cccc([C@]2(C)CCN(C(=O)c3cc(C)cnc3Cl)C2)c1 ZINC000880698309 EH On-Demand Anodyne DRD4 41 32 COc1cccc([C@]2(C)CCN(C(=O)c3cc(C)cnc3Cl)C2)c1 ZINC000880698309 EH On-Demand Anodyne TACR2 19 42 COc1ccccc1[C@@H](NC(=O)c1ccc(NC(=O)c2ccccc2)cc1)c1nccn1C ZINC000880698415 II On-Demand Anodyne CPT1A 46 33 COc1ccccc1[C@@H](NC(=O)c1ccc(NC(=O)c2ccccc2)cc1)c1nccn1C ZINC000880698415 II On-Demand Anodyne PRNP 78 39 COc1ccccc1[C@@H](NC(=O)c1ccc(NC(=O)c2ccccc2)cc1)c1nccn1C ZINC000880698415 II On-Demand Anodyne SYK 15 40 COc1ccccc1[C@@H](NC(=O)c1ccc(NC(=O)c2ccccc2)cc1)c1nccn1C ZINC000880698415 II On-Demand Anodyne KCNK3 71 42 COc1ccccc1[C@@H](NC(=O)c1ccc(NC(=O)c2ccccc2)cc1)c1nccn1C ZINC000880698415 II On-Demand Anodyne KCNK9 51 39 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880698467 FD On-Demand Anodyne CELA1 18 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880698467 FD On-Demand Anodyne PREP 46 47 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880698467 FD On-Demand Anodyne SLC12A5 66 36 C=CC(C)(C)CC(=O)Nc1ccc2c(c1)CCOC2 ZINC000880698518 CG On-Demand Mild PTPRF 44 33 O=C(/C=C\c1cccnc1)Nc1ncc(Cc2cccc(Cl)c2Cl)s1 ZINC000880698520 GK On-Demand Anodyne SCD 18 45 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698523 GF On-Demand Anodyne PIK3CA 15 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698523 GF On-Demand Anodyne MTOR 20 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698523 GF On-Demand Anodyne STAT6 49 35 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc3c(c1)CCOC3)C2 ZINC000880698559 EH On-Demand Anodyne MTNR1A 24 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc3c(c1)CCOC3)C2 ZINC000880698559 EH On-Demand Anodyne MTNR1B 25 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc3c(c1)CCOC3)C2 ZINC000880698559 EH On-Demand Anodyne ROCK2 24 45 CN1CC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698572 DE On-Demand Anodyne CCR3 57 40 CN1CC[C@@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698573 DE On-Demand Anodyne CCR3 57 40 O=C(COC1CC1)Nc1ncc(Cc2c(F)cccc2F)s1 ZINC000880698578 DG On-Demand Anodyne CDK5 53 40 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698625 FE On-Demand Anodyne CCR3 64 46 O=C(NCC1(N2CCOCC2)CC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698635 FD On-Demand Anodyne HCN1 52 36 O=C(NCC1(N2CCOCC2)CC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698635 FD On-Demand Anodyne HCN4 47 30 C[C@@](O)(CNC(=O)Nc1ccnn1-c1ccc(F)cc1)C(F)(F)F ZINC000880698640 EE On-Demand Anodyne NR3C1 22 40 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccnn2-c2ccc(F)cc2)no1 ZINC000880698643 FH On-Demand Anodyne KCNA5 16 44 CN1CCO[C@@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)[C@@H]1c1cnn(C)c1 ZINC000880698655 GD On-Demand Anodyne PANC 49 33 CN1CCO[C@@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)[C@@H]1c1cnn(C)c1 ZINC000880698656 GD On-Demand Anodyne PANC 49 33 O=C(NC1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1)C1CC1 ZINC000880698664 FF On-Demand Anodyne EPHX2 29 41 O=C(COC1CC1)Nc1ccc2c(c1)CCOC2 ZINC000880698687 BD On-Demand Anodyne PTPRF 43 34 O=C(NCCCNC(=O)C1CCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880698714 FE On-Demand Anodyne TBK1 77 37 O=C(C[C@H]1CCNC1=O)Nc1ncc(Cc2c(F)cccc2F)s1 ZINC000880698716 FE On-Demand Anodyne CDK5 52 38 O=C(C[C@@H]1CCNC1=O)Nc1ncc(Cc2c(F)cccc2F)s1 ZINC000880698717 FE On-Demand Anodyne CDK5 52 38 CN(Cc1cn(C)nn1)C(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880698726 GD On-Demand Anodyne PREP 25 44 CN1CCO[C@@H](CN(CC2CC2)C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698809 GF On-Demand Anodyne WNT3A 49 38 CN1CCO[C@H](CN(CC2CC2)C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698810 GF On-Demand Anodyne WNT3A 49 38 NC(=O)C[C@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698947 EE On-Demand Anodyne CCR3 46 35 NC(=O)C[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880698948 EE On-Demand Anodyne CCR3 46 35 C=CC(C)(C)CC(=O)N1CCc2cc(OC)ccc2C1 ZINC000880698963 CG On-Demand Mild DRD5 16 43 O=C(/C=C\c1cccnc1)Nc1cc(Cl)ccc1OCC(F)(F)F ZINC000880698974 FI On-Demand Anodyne RBP4 15 41 C[C@@H]1CN(CCCNC(=O)Nc2ccnn2-c2ccc(F)cc2)CCCO1 ZINC000880698985 GF On-Demand Anodyne CCR3 48 46 COc1cc(N2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)ncn1 ZINC000880699184 GE On-Demand Anodyne PDGFRB 48 38 O=C(NCCN1CCCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699240 ED On-Demand Anodyne CCR3 24 41 O=C(NCCN1CCCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699240 ED On-Demand Anodyne EPHX2 18 51 O=C(NCCN1CCCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699240 ED On-Demand Anodyne PLD2 58 35 CC1(C)CC[C@@H](CC(=O)Nc2ccc3c(c2)CCOC3)OC1 ZINC000880699275 DG On-Demand Anodyne PTPRF 47 37 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccnn1-c1ccc(F)cc1)C2 ZINC000880699309 FG On-Demand Anodyne HTR3A 34 46 CCC1(O)CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880699426 EF On-Demand Anodyne S1PR2 31 44 O=C(NCCCCN1CCC[C@H]1CO)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699495 GE On-Demand Anodyne CCR3 38 44 O=C(NCCCCN1CCC[C@@H]1CO)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699496 GE On-Demand Anodyne CCR3 38 44 COC(=O)c1occc1CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880699575 EG On-Demand Anodyne NQO2 22 43 COC(=O)c1occc1CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880699576 EG On-Demand Anodyne NQO2 22 43 Cn1cc([C@@H]2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C2)cn1 ZINC000880699583 FF On-Demand Anodyne PRCP 29 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cccc3c1CCN(C)C3=O)C2 ZINC000880699585 FG On-Demand Anodyne DRD4 40 32 CCOC[C@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880699604 EG On-Demand Anodyne CCR3 46 34 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699634 GE On-Demand Anodyne PIK3CA 15 41 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699634 GE On-Demand Anodyne MTOR 24 41 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699634 GE On-Demand Anodyne EPHX2 25 49 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699634 GE On-Demand Anodyne PIK3CG 15 41 CCN(CC(C)(C)O)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699653 DF On-Demand Anodyne NR3C1 21 43 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccnn1-c1ccc(F)cc1)CC2 ZINC000880699699 FF On-Demand Anodyne CACNA1H 43 40 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccnn3-c3ccc(F)cc3)C2)nn1 ZINC000880699712 GF On-Demand Anodyne CCR3 41 36 C[C@H](O)CN1CCC(CN(C)C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880699721 GF On-Demand Anodyne WNT3A 46 34 CCC(CC)(CO)CNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699740 EF On-Demand Anodyne NR3C1 16 42 CCN1CC[C@H](N(C)C(=O)Nc2ccnn2-c2ccc(F)cc2)[C@H](C)C1 ZINC000880699759 FG On-Demand Anodyne WNT3A 40 33 CCN1CC[C@@H](N(C)C(=O)Nc2ccnn2-c2ccc(F)cc2)[C@H](C)C1 ZINC000880699760 FG On-Demand Anodyne WNT3A 40 33 CCN1CC[C@@H](N(C)C(=O)Nc2ccnn2-c2ccc(F)cc2)[C@@H](C)C1 ZINC000880699761 FG On-Demand Anodyne WNT3A 40 33 CCN1CC[C@H](N(C)C(=O)Nc2ccnn2-c2ccc(F)cc2)[C@@H](C)C1 ZINC000880699762 FG On-Demand Anodyne WNT3A 40 33 COC[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880699820 EF On-Demand Anodyne CCR3 56 35 CN(C[C@@H]1CCOC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699923 DF On-Demand Anodyne WNT3A 46 33 CN(CCN1CCOCC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699936 ED On-Demand Anodyne CASR 52 38 CN(CCN1CCOCC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880699936 ED On-Demand Anodyne EPHX2 16 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCc3ccc(O)cc31)C2 ZINC000880699945 EG On-Demand Anodyne NQO2 24 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCc3ccc(O)cc31)C2 ZINC000880699945 EG On-Demand Anodyne MTNR1A 24 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCc3ccc(O)cc31)C2 ZINC000880699945 EG On-Demand Anodyne MTNR1B 22 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCc3ccc(O)cc31)C2 ZINC000880699946 EG On-Demand Anodyne NQO2 24 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCc3ccc(O)cc31)C2 ZINC000880699946 EG On-Demand Anodyne MTNR1A 24 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCc3ccc(O)cc31)C2 ZINC000880699946 EG On-Demand Anodyne MTNR1B 22 40 COC(=O)C1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880699971 FF On-Demand Anodyne EPHX2 32 41 CCN1CCC[C@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880700066 EF On-Demand Anodyne CCR3 97 42 CCN1CCC[C@@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880700068 EF On-Demand Anodyne CCR3 97 42 CN(CC1CCOCC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700078 EF On-Demand Anodyne WNT3A 53 36 COCCC(=O)N1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880700108 GE On-Demand Anodyne EPHX2 39 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1[C@@H](C)O ZINC000880700109 ED On-Demand Anodyne CELA1 40 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1[C@@H](C)O ZINC000880700110 ED On-Demand Anodyne CELA1 40 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1[C@H](C)O ZINC000880700113 ED On-Demand Anodyne CELA1 40 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1[C@H](C)O ZINC000880700114 ED On-Demand Anodyne CELA1 40 41 COC(=O)c1occc1CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880700118 EE On-Demand Anodyne MTNR1A 38 40 COC(=O)c1occc1CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880700120 EE On-Demand Anodyne MTNR1A 38 40 Cc1ccc(CC2CN(C(=O)COC3CC3)C2)cc1 ZINC000880700164 CE On-Demand Anodyne GRIN2B 16 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700168 GG On-Demand Anodyne CCR3 62 44 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700172 GG On-Demand Anodyne CCR3 62 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCC[C@@H]1Cc1cnn(C)c1)C2 ZINC000880700198 FG On-Demand Anodyne MTNR1A 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCC[C@@H]1Cc1cnn(C)c1)C2 ZINC000880700198 FG On-Demand Anodyne MTNR1B 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC[C@H]1Cc1cnn(C)c1)C2 ZINC000880700200 FG On-Demand Anodyne MTNR1A 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC[C@H]1Cc1cnn(C)c1)C2 ZINC000880700200 FG On-Demand Anodyne MTNR1B 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC[C@@H]1Cc1cnn(C)c1)C2 ZINC000880700202 FG On-Demand Anodyne MTNR1A 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCC[C@@H]1Cc1cnn(C)c1)C2 ZINC000880700202 FG On-Demand Anodyne MTNR1B 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCC[C@H]1Cc1cnn(C)c1)C2 ZINC000880700203 FG On-Demand Anodyne MTNR1A 21 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCC[C@H]1Cc1cnn(C)c1)C2 ZINC000880700203 FG On-Demand Anodyne MTNR1B 21 40 Cn1cc(CN2CCCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)cn1 ZINC000880700211 GE On-Demand Anodyne IKBKB 40 39 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880700229 GD On-Demand Anodyne ABCB1 19 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880700350 EE On-Demand Anodyne EPHX2 35 45 CCC(=O)N1CC[C@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880700351 EE On-Demand Anodyne EPHX2 35 45 C[C@H](C[C@@H]1CCOC1)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700422 EF On-Demand Anodyne CCR3 46 39 C[C@@H](C[C@H]1CCOC1)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700423 EF On-Demand Anodyne CCR3 46 39 C[C@@H](C[C@@H]1CCOC1)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700424 EF On-Demand Anodyne CCR3 46 39 O=C1NC(=O)N2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@H]12 ZINC000880700494 FC On-Demand Anodyne SMO 18 51 O=C1NC(=O)N2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)C[C@@H]12 ZINC000880700495 FC On-Demand Anodyne SMO 18 51 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700512 FF On-Demand Anodyne CCR3 70 43 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700513 FF On-Demand Anodyne CCR3 70 43 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700514 FF On-Demand Anodyne CCR3 70 43 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700516 FF On-Demand Anodyne CCR3 70 43 CC[C@@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700518 CG On-Demand Anodyne NQO2 27 43 CC[C@@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700518 CG On-Demand Anodyne MTNR1A 50 41 CC[C@@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700518 CG On-Demand Anodyne MTNR1B 45 40 CC[C@@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700520 CG On-Demand Anodyne NQO2 27 43 CC[C@@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700520 CG On-Demand Anodyne MTNR1A 50 41 CC[C@@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700520 CG On-Demand Anodyne MTNR1B 45 40 CC[C@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700522 CG On-Demand Anodyne NQO2 27 43 CC[C@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700522 CG On-Demand Anodyne MTNR1A 50 41 CC[C@H](NC(=O)[C@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700522 CG On-Demand Anodyne MTNR1B 45 40 CC[C@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700524 CG On-Demand Anodyne NQO2 27 43 CC[C@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700524 CG On-Demand Anodyne MTNR1A 50 41 CC[C@H](NC(=O)[C@@H]1CCc2cc(OC)ccc2C1)C1CC1 ZINC000880700524 CG On-Demand Anodyne MTNR1B 45 40 CNC(=O)CN1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880700552 FC On-Demand Anodyne SLC27A1 46 40 C[C@H](CC[S@](C)=O)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700566 EE On-Demand Anodyne CCR3 43 37 C[C@@H](CC[S@@](C)=O)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700568 EE On-Demand Anodyne CCR3 43 37 C[C@H](CC[S@@](C)=O)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700569 EE On-Demand Anodyne CCR3 43 37 C[C@@H](CC[S@](C)=O)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700570 EE On-Demand Anodyne CCR3 43 37 CCN(CC)C(=O)CCCNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700584 FF On-Demand Anodyne NR3C1 17 40 CC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CC1 ZINC000880700624 DF On-Demand Anodyne KCNQ2 69 35 CC[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CC1 ZINC000880700626 DF On-Demand Anodyne KCNQ2 69 35 O=C(NCCN1CCSCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700662 EE On-Demand Anodyne PLD2 62 35 CS(=O)(=O)N1CCC[C@@H]1CNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700666 GD On-Demand Anodyne CCR3 40 36 Cn1nccc1C1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880700927 FG On-Demand Anodyne PRCP 36 40 Cc1cc(-c2nc(C)c(C(=O)N3CCC[C@@H]3[C@@H](C)O)s2)ccc1F ZINC000880700961 EH On-Demand Anodyne TRPC6 40 35 Cc1cc(-c2nc(C)c(C(=O)N3CCC[C@@H]3[C@H](C)O)s2)ccc1F ZINC000880700962 EH On-Demand Anodyne TRPC6 40 35 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700984 GE On-Demand Mild CASR 57 42 C[C@@H](O)CC(C)(C)CNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880700985 EF On-Demand Anodyne NR3C1 15 41 COCC1(O)CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880700993 EE On-Demand Anodyne S1PR2 30 43 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701073 DE On-Demand Anodyne PAPA1_CARPA 35 46 CC[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701073 DE On-Demand Anodyne CTSK 15 47 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701074 DE On-Demand Anodyne PAPA1_CARPA 35 46 CC[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701074 DE On-Demand Anodyne CTSK 15 47 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701075 DE On-Demand Anodyne PAPA1_CARPA 35 46 CC[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701075 DE On-Demand Anodyne CTSK 15 47 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701076 DE On-Demand Anodyne PAPA1_CARPA 35 46 CC[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CC1 ZINC000880701076 DE On-Demand Anodyne CTSK 15 47 COCCn1nc(C)c(NC(=O)Nc2ccnn2-c2ccc(F)cc2)c1C ZINC000880701083 FG On-Demand Anodyne P2RX7 15 44 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880701124 GD On-Demand Anodyne CCR3 46 39 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880701125 GD On-Demand Anodyne CCR3 46 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccc(C)cc2)C1 ZINC000880701177 GF On-Demand Anodyne FPR1 48 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccc(C)cc2)C1 ZINC000880701178 GF On-Demand Anodyne FPR1 48 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1nc2ccccc2n1C(C)C ZINC000880701235 GG On-Demand Anodyne FPR1 48 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1nc2ccccc2n1C(C)C ZINC000880701236 GG On-Demand Anodyne FPR1 48 39 O=C(CC[C@@H]1CCc2ccccc21)NCC(O)(C1CC1)C1CC1 ZINC000880701287 DG On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@@H]1CCc2ccccc21)NCC(O)(C1CC1)C1CC1 ZINC000880701287 DG On-Demand Anodyne MTNR1B 17 41 O=C(CC[C@H]1CCc2ccccc21)NCC(O)(C1CC1)C1CC1 ZINC000880701289 DG On-Demand Anodyne MTNR1A 15 41 O=C(CC[C@H]1CCc2ccccc21)NCC(O)(C1CC1)C1CC1 ZINC000880701289 DG On-Demand Anodyne MTNR1B 17 41 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)Nc2ccc3c(c2)CCOC3)CO1 ZINC000880701309 GG On-Demand Anodyne PTPRF 41 32 CN1C[C@@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)CC1=O ZINC000880701312 FE On-Demand Anodyne DRD4 40 30 CN1C[C@@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)CC1=O ZINC000880701312 FE On-Demand Anodyne CACNA1I 64 44 CC(C)(C)OC(=O)CC[C@@H]1C[C@H](C(=O)Nc2ccc3c(c2)CCOC3)CO1 ZINC000880701313 GG On-Demand Anodyne PTPRF 41 32 CN1C[C@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)CC1=O ZINC000880701314 FE On-Demand Anodyne DRD4 40 30 CN1C[C@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)CC1=O ZINC000880701314 FE On-Demand Anodyne CACNA1I 64 44 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)Nc2ccc3c(c2)CCOC3)CO1 ZINC000880701316 GG On-Demand Anodyne PTPRF 41 32 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)Nc2ccc3c(c2)CCOC3)CO1 ZINC000880701318 GG On-Demand Anodyne PTPRF 41 32 CN1C[C@@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CC1=O ZINC000880701344 DD On-Demand Anodyne GABRA1 16 45 O=C(NCC(O)(C1CC1)C1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880701372 EG On-Demand Anodyne PDE4D 21 50 O=C(NCC(O)(C1CC1)C1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880701372 EG On-Demand Anodyne CACNA1I 47 37 COc1ccccc1-c1ccc(C(=O)NC[C@@H](CO)CC2CC2)c(O)n1 ZINC000880701373 FF On-Demand Anodyne KCNA3 40 38 COc1ccccc1-c1ccc(C(=O)NC[C@H](CO)CC2CC2)c(O)n1 ZINC000880701374 FF On-Demand Anodyne KCNA3 40 38 O=C(NCC(O)(C1CC1)C1CC1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880701375 GG On-Demand Anodyne KCNJ11 49 31 Cc1ccc(CC2CN(C(=O)c3nnn(C)n3)C2)cc1 ZINC000880701425 CC On-Demand Anodyne GRIN2B 16 40 C[C@H](NC(=O)Nc1ccnn1-c1ccc(F)cc1)[C@H]1CN(C)CCO1 ZINC000880701520 ED On-Demand Anodyne CCR3 47 36 C[C@H](NC(=O)Nc1ccnn1-c1ccc(F)cc1)[C@@H]1CN(C)CCO1 ZINC000880701522 ED On-Demand Anodyne CCR3 47 36 CC[C@@H](NC(=O)CCCCc1ccc(OC)c(OC)c1)C1CC1 ZINC000880701543 DH On-Demand Anodyne INHA 51 37 CC[C@@H](NC(=O)CCCCc1ccc(OC)c(OC)c1)C1CC1 ZINC000880701543 DH On-Demand Anodyne MTNR1B 24 44 CC[C@@H](NC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880701600 CF On-Demand Anodyne GABRA1 18 44 CC[C@@H](NC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880701600 CF On-Demand Anodyne MPO 60 36 CC[C@@H](NC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880701600 CF On-Demand Anodyne GABRA2 16 44 Cc1noc(C)c1CCCNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701617 FG On-Demand Anodyne P2RX7 15 43 Cc1ccc(CC2CN(C(=O)c3cnc4cc[nH]c4c3)C2)cc1 ZINC000880701646 DG On-Demand Anodyne GRIN2B 36 42 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCC3(CN(C(=O)OC(C)(C)C)C3)O2)c1 ZINC000880701664 GF On-Demand Anodyne CACNA1I 41 32 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCC3(CN(C(=O)OC(C)(C)C)C3)O2)c1 ZINC000880701666 GF On-Demand Anodyne CACNA1I 41 32 CC[C@@](C)(O)CNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701696 DE On-Demand Anodyne NR3C1 21 40 Cc1noc(C2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)n1 ZINC000880701701 FG On-Demand Anodyne SMO 42 41 Cc1noc(C2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)n1 ZINC000880701701 FG On-Demand Anodyne ETHR 56 35 COCCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880701718 FE On-Demand Anodyne SSTR5 40 39 COCCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880701718 FE On-Demand Anodyne CCR3 60 41 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701738 GF On-Demand Anodyne STAT6 50 35 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701738 GF On-Demand Anodyne DGAT1 18 43 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701738 GF On-Demand Anodyne NAMPT 26 41 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701738 GF On-Demand Anodyne SLC27A1 51 35 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701791 FG On-Demand Anodyne PANC 51 37 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701792 FG On-Demand Anodyne PANC 51 37 O=C(NCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701795 ED On-Demand Anodyne EPHX2 22 54 O=C(NCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701795 ED On-Demand Anodyne PLD2 64 37 O=C(NCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701795 ED On-Demand Anodyne WNT3A 44 30 CN1CCN(C(=O)c2cc3ccccc3cc2F)CCC1=O ZINC000880701814 DE On-Demand Anodyne HRH4 20 40 CN1CCN(C(=O)c2cc3ccccc3cc2F)CCC1=O ZINC000880701814 DE On-Demand Anodyne PARP1 43 37 O=C(NCC(O)(C1CC1)C1CC1)c1cccn2nccc12 ZINC000880701820 CD On-Demand Anodyne JAK3 18 42 O=C(NCC(O)(C1CC1)C1CC1)c1cccn2nccc12 ZINC000880701820 CD On-Demand Anodyne TYK2 21 42 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](C)CN1CCC(C)CC1 ZINC000880701822 DF On-Demand Anodyne PLD1 50 38 Cc1nc(C(C)C)ncc1C(=O)N[C@H](C)CN1CCC(C)CC1 ZINC000880701824 DF On-Demand Anodyne PLD1 50 38 COc1ccccc1-c1ccc(C(=O)NCC(O)(C2CC2)C2CC2)c(O)n1 ZINC000880701851 FF On-Demand Anodyne KCNA3 42 34 CS(=O)(=O)NC[C@@H]1CCCCN1C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701854 GD On-Demand Anodyne WNT3A 40 33 CS(=O)(=O)NC[C@H]1CCCCN1C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701855 GD On-Demand Anodyne WNT3A 40 33 C[C@@H]1[C@@H](c2cccc(Cl)c2)OCCN1C(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880701863 GG On-Demand Anodyne MDM2 72 35 CN(CC1CC1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880701865 CF On-Demand Anodyne WNT3A 40 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccc(O)cc21 ZINC000880701876 FE On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCc2ccc(O)cc21 ZINC000880701877 FE On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCc2ccc(O)cc21 ZINC000880701878 FE On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCc2ccc(O)cc21 ZINC000880701879 FE On-Demand Anodyne PAPA1_CARPA 35 40 Cn1cc(CN2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)cn1 ZINC000880701897 GE On-Demand Anodyne PLA2G7 46 35 Cn1cc(CN2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)cn1 ZINC000880701897 GE On-Demand Anodyne IKBKB 43 40 COc1ccnc(N2CCN(C(=O)Nc3ccnn3-c3ccc(F)cc3)CC2)n1 ZINC000880701903 GE On-Demand Anodyne FAAH 22 41 O=C(CNC(=O)Nc1ccnn1-c1ccc(F)cc1)NC1CCCCC1 ZINC000880701905 FF On-Demand Anodyne EPHX2 17 41 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccnn2-c2ccc(F)cc2)on1 ZINC000880701926 FH On-Demand Anodyne KCNA5 21 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880701937 FE On-Demand Anodyne CCR3 68 36 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880701947 FF On-Demand Anodyne GPBAR1 21 45 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880701948 FF On-Demand Anodyne GPBAR1 21 45 CN1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CCC1=O ZINC000880702003 DC On-Demand Anodyne L3MBTL3 53 39 CN1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CCC1=O ZINC000880702004 DC On-Demand Anodyne L3MBTL3 53 39 CN1C[C@@H](CNC(=O)c2ccc(OC(F)F)c(Br)c2)CC1=O ZINC000880702009 GE On-Demand Anodyne CACNA1I 64 36 CN1C[C@H](CNC(=O)c2ccc(OC(F)F)c(Br)c2)CC1=O ZINC000880702010 GE On-Demand Anodyne CACNA1I 64 36 O=C(NCC(O)(C1CC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702022 EE On-Demand Anodyne GABRA1 19 50 O=C(NCC(O)(C1CC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702022 EE On-Demand Anodyne MPO 59 34 O=C(NCC(O)(C1CC1)C1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702022 EE On-Demand Anodyne GABRA2 16 50 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702109 GG On-Demand Anodyne CCR3 45 40 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702110 GG On-Demand Anodyne CCR3 45 40 CC1(C)CC[C@@H](CC(=O)N[C@@H]2CCc3ccc(O)cc32)OC1 ZINC000880702142 DG On-Demand Anodyne STS 40 32 CC1(C)CC[C@@H](CC(=O)N[C@H]2CCc3ccc(O)cc32)OC1 ZINC000880702143 DG On-Demand Anodyne STS 40 32 O=C(NCC(=O)N1CCCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702187 EE On-Demand Anodyne PRMT3 18 44 CSc1nccnc1C(=O)N[C@H](C)CN1CCC(C)CC1 ZINC000880702196 DE On-Demand Anodyne P2RX3 28 40 CSc1nccnc1C(=O)N[C@H](C)CN1CCC(C)CC1 ZINC000880702196 DE On-Demand Anodyne PLD1 49 37 CSc1nccnc1C(=O)N[C@@H](C)CN1CCC(C)CC1 ZINC000880702197 DE On-Demand Anodyne P2RX3 28 40 CSc1nccnc1C(=O)N[C@@H](C)CN1CCC(C)CC1 ZINC000880702197 DE On-Demand Anodyne PLD1 49 37 CCCCNC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702203 CF On-Demand Anodyne ASAH1 53 32 O=C(NCCCN1CCCC1=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702204 EE On-Demand Anodyne CCR3 31 40 CC[C@H](C)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702251 CF On-Demand Anodyne CCR3 42 37 O=C(NCc1ccc(N2CCCC2)nc1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702263 GG On-Demand Anodyne SLC27A1 55 37 CN1C[C@H](CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1=O ZINC000880702269 GD On-Demand Anodyne Q9NAW4_PLAFA 28 42 CN1C[C@@H](CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CC1=O ZINC000880702272 GD On-Demand Anodyne Q9NAW4_PLAFA 28 42 CN1CCN(C(=O)c2cc3cc(F)ccc3[nH]c2=O)CCC1=O ZINC000880702286 DC On-Demand Anodyne HRH4 27 55 O=C(NCCN1CCCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702296 EF On-Demand Anodyne CCR3 38 41 O=C(NCCN1CCCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702296 EF On-Demand Anodyne CHRNA7 17 52 O=C(NCCN1CCCCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702296 EF On-Demand Anodyne PLD2 62 36 CN1CCC[C@H](NC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702321 DE On-Demand Anodyne CCR3 92 37 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1 ZINC000880702339 IH On-Demand Bother WDR5 33 41 Cn1nnc(C(=O)N2CCc3sccc3[C@@H]2c2ccc(Cl)cc2)n1 ZINC000880702345 FF On-Demand Anodyne TRPM8 17 55 Cn1nnc(C(=O)N2CCc3sccc3[C@H]2c2ccc(Cl)cc2)n1 ZINC000880702346 FF On-Demand Anodyne TRPM8 17 55 CN1CCC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702349 EE On-Demand Anodyne CCR3 114 44 O=C(CNC(=O)Nc1ccnn1-c1ccc(F)cc1)NC1CCCC1 ZINC000880702367 EE On-Demand Anodyne EPHX2 15 40 O=C(NC(CCC(F)(F)F)CCC(F)(F)F)c1cccn2nccc12 ZINC000880702405 FI On-Demand Anodyne JAK3 16 40 O=C(NC(CCC(F)(F)F)CCC(F)(F)F)c1cccn2nccc12 ZINC000880702405 FI On-Demand Anodyne TYK2 20 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H]([C@@H]3CCCCO3)C2)N1Cc1ccccc1 ZINC000880702419 GE On-Demand Anodyne PREP 56 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H]([C@@H]3CCCCO3)C2)N1Cc1ccccc1 ZINC000880702420 GE On-Demand Anodyne PREP 56 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@@H]([C@H]3CCCCO3)C2)N1Cc1ccccc1 ZINC000880702421 GE On-Demand Anodyne PREP 56 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC[C@H]([C@H]3CCCCO3)C2)N1Cc1ccccc1 ZINC000880702422 GE On-Demand Anodyne PREP 56 40 COc1ccccc1[C@@H]1C[C@H]1NC(=O)CN1CCCCS1(=O)=O ZINC000880702429 ED On-Demand Anodyne HTR1A 16 40 Cc1cncc(CCNC(=O)CC[C@@H]2CCc3ccccc32)n1 ZINC000880702442 DF On-Demand Anodyne NQO2 18 40 Cc1cncc(CCNC(=O)CC[C@@H]2CCc3ccccc32)n1 ZINC000880702442 DF On-Demand Anodyne MTNR1A 17 40 Cc1cncc(CCNC(=O)CC[C@@H]2CCc3ccccc32)n1 ZINC000880702442 DF On-Demand Anodyne MTNR1B 18 40 Cc1cncc(CCNC(=O)CC[C@H]2CCc3ccccc32)n1 ZINC000880702443 DF On-Demand Anodyne NQO2 18 40 Cc1cncc(CCNC(=O)CC[C@H]2CCc3ccccc32)n1 ZINC000880702443 DF On-Demand Anodyne MTNR1A 17 40 Cc1cncc(CCNC(=O)CC[C@H]2CCc3ccccc32)n1 ZINC000880702443 DF On-Demand Anodyne MTNR1B 18 40 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC([C@H]2CCCCO2)CC1 ZINC000880702467 FG On-Demand Anodyne L3MBTL3 47 33 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880702468 FG On-Demand Anodyne L3MBTL3 47 33 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne TIMP3 42 34 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne SYK 16 41 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne MTNR1A 31 53 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne MTNR1B 37 53 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne ROCK2 40 39 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne GALR2 24 43 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne EPHX2 15 43 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne AKR1C3 18 42 COc1cccc(Nc2ccc(NC(=O)COC3CC3)nc2)c1 ZINC000880702480 DF On-Demand Anodyne KCNK3 40 35 O=C(c1cccn2nccc12)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880702484 DF On-Demand Anodyne L3MBTL3 53 37 O=C(c1cccn2nccc12)N1CCC([C@H]2CCCCO2)CC1 ZINC000880702485 DF On-Demand Anodyne L3MBTL3 53 37 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702519 GD On-Demand Anodyne CCR8 56 38 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nc(C(N)=O)cs1)C2 ZINC000880702527 ED On-Demand Anodyne IKBKE 18 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1nc(C(N)=O)cs1)C2 ZINC000880702527 ED On-Demand Anodyne TBK1 17 41 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702538 GF On-Demand Anodyne MTOR 24 40 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702538 GF On-Demand Anodyne STAT6 45 35 Nc1ccc(C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)cc1[N+](=O)[O-] ZINC000880702543 HH On-Demand Bother WDR5 20 40 O=C(N[C@H]1C[C@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702546 DD On-Demand Anodyne GABRA1 16 40 O=C(N[C@H]1C[C@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702546 DD On-Demand Anodyne GABRA2 15 40 O=C(N[C@@H]1C[C@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702547 DD On-Demand Anodyne GABRA1 16 40 O=C(N[C@@H]1C[C@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702547 DD On-Demand Anodyne GABRA2 15 40 O=C(N[C@H]1C[C@@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702549 DD On-Demand Anodyne GABRA1 16 40 O=C(N[C@H]1C[C@@H](O)C12CCC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880702549 DD On-Demand Anodyne GABRA2 15 40 CN1C[C@@H](CNC(=O)c2cc3ccccc3cc2F)CC1=O ZINC000880702553 DE On-Demand Anodyne POLR1A 48 30 CN1C[C@H](CNC(=O)c2cc3ccccc3cc2F)CC1=O ZINC000880702555 DE On-Demand Anodyne POLR1A 48 30 C[C@@H]1[C@@H](c2cccc(Cl)c2)OCCN1C(=O)C[C@@H]1CCNC1=O ZINC000880702562 EE On-Demand Anodyne MDM2 41 33 C[C@@H]1[C@@H](c2cccc(Cl)c2)OCCN1C(=O)C[C@H]1CCNC1=O ZINC000880702565 EE On-Demand Anodyne MDM2 41 33 CN(C[C@@H]1CCCCO1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702581 EG On-Demand Anodyne WNT3A 40 32 CN(C[C@H]1CCCCO1)C(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702583 EG On-Demand Anodyne WNT3A 40 32 CCN(CC)C(=O)C1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702585 GG On-Demand Anodyne WNT3A 42 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2c(C)cccn12 ZINC000880702605 FF On-Demand Anodyne FPR1 44 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnc2c(C)cccn12 ZINC000880702608 FF On-Demand Anodyne FPR1 44 35 N#CCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702627 EE On-Demand Mild WNT3A 44 30 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](CO)CC1CC1)C2 ZINC000880702653 DE On-Demand Anodyne MTNR1A 36 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](CO)CC1CC1)C2 ZINC000880702653 DE On-Demand Anodyne MTNR1B 31 45 CN1CCC(CNC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702654 EE On-Demand Anodyne HTR1F 47 36 CN1CCC(CNC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702654 EE On-Demand Anodyne CCR3 52 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](CO)CC1CC1)C2 ZINC000880702658 DE On-Demand Anodyne MTNR1A 36 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](CO)CC1CC1)C2 ZINC000880702658 DE On-Demand Anodyne MTNR1B 31 45 Cc1cnc(Cl)c(C(=O)NC[C@H]2CC(=O)N(C)C2)c1 ZINC000880702659 CD On-Demand Anodyne CACNA1I 59 35 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC(=O)N(C)C2)c1 ZINC000880702660 CD On-Demand Anodyne CACNA1I 59 35 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702662 GF On-Demand Anodyne HCN1 58 38 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702662 GF On-Demand Anodyne HCN4 48 31 O=C(NC1(CN2CCN(c3ccccc3)CC2)CC1)[C@@H]1CCc2nncn2CC1 ZINC000880702677 GD On-Demand Anodyne DRD3 15 41 O=C(NC1(CN2CCN(c3ccccc3)CC2)CC1)[C@H]1CCc2nncn2CC1 ZINC000880702678 GD On-Demand Anodyne DRD3 15 41 CN1C[C@@H](CNC(=O)Cc2ccccc2N2CCCC2=O)CC1=O ZINC000880702680 EC On-Demand Anodyne KCNQ2 40 35 C[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)CC[C@@H](C)O1 ZINC000880702716 FH On-Demand Anodyne RBP4 57 37 O=C1CC[C@H](c2ccc(C(=O)N3CCC([C@@H]4CCCCO4)CC3)cc2)N1 ZINC000880702718 FG On-Demand Anodyne L3MBTL3 72 43 O=C1CC[C@@H](c2ccc(C(=O)N3CCC([C@@H]4CCCCO4)CC3)cc2)N1 ZINC000880702719 FG On-Demand Anodyne L3MBTL3 72 43 O=C1CC[C@@H](c2ccc(C(=O)N3CCC([C@H]4CCCCO4)CC3)cc2)N1 ZINC000880702720 FG On-Demand Anodyne L3MBTL3 72 43 O=C1CC[C@H](c2ccc(C(=O)N3CCC([C@H]4CCCCO4)CC3)cc2)N1 ZINC000880702721 FG On-Demand Anodyne L3MBTL3 72 43 O=C(c1cc2ccccc2cc1F)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880702746 EI On-Demand Anodyne L3MBTL3 61 38 O=C(c1cc2ccccc2cc1F)N1CCC([C@H]2CCCCO2)CC1 ZINC000880702747 EI On-Demand Anodyne L3MBTL3 61 38 COc1ccccc1[C@@H]1C[C@H]1NC(=O)C[C@H]1CCNC1=O ZINC000880702754 CD On-Demand Anodyne MBTPS1 44 32 COc1ccccc1[C@@H]1C[C@H]1NC(=O)C[C@@H]1CCNC1=O ZINC000880702755 CD On-Demand Anodyne MBTPS1 44 32 N#CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880702774 CF On-Demand Mild HCN1 63 37 N#CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880702774 CF On-Demand Mild HCN4 55 35 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC([C@@H]3CCCCO3)CC2)N1Cc1ccccc1 ZINC000880702779 GE On-Demand Anodyne PREP 48 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCC([C@H]3CCCCO3)CC2)N1Cc1ccccc1 ZINC000880702780 GE On-Demand Anodyne PREP 48 40 COc1ccccc1[C@@H]1C[C@H]1NC(=O)COC1CC1 ZINC000880702788 CD On-Demand Anodyne MBTPS1 50 32 CCN1CC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702820 EE On-Demand Anodyne CCR3 84 40 CCN1CC[C@H](CNC(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702820 EE On-Demand Anodyne WNT3A 40 33 O=C1NCC[C@@H]1CC(=O)N1CCc2sccc2[C@@H]1c1ccc(Cl)cc1 ZINC000880702822 FG On-Demand Anodyne TRPM8 15 52 O=C1NCC[C@@H]1CC(=O)N1CCc2sccc2[C@H]1c1ccc(Cl)cc1 ZINC000880702823 FG On-Demand Anodyne TRPM8 15 52 O=C1NCC[C@H]1CC(=O)N1CCc2sccc2[C@H]1c1ccc(Cl)cc1 ZINC000880702824 FG On-Demand Anodyne TRPM8 15 52 O=C1NCC[C@H]1CC(=O)N1CCc2sccc2[C@@H]1c1ccc(Cl)cc1 ZINC000880702825 FG On-Demand Anodyne TRPM8 15 52 CN1C[C@@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880702867 EE On-Demand Anodyne PDE4D 20 43 CN1C[C@@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880702867 EE On-Demand Anodyne CACNA1I 71 44 CN1C[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880702869 EE On-Demand Anodyne PDE4D 20 43 CN1C[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880702869 EE On-Demand Anodyne CACNA1I 71 44 CN1C[C@@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)CC1=O ZINC000880702870 FC On-Demand Anodyne F2 24 42 CN1C[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)CC1=O ZINC000880702871 FC On-Demand Anodyne F2 24 42 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702879 GD On-Demand Anodyne CCR3 41 34 O=C(CN1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1)NC1CC1 ZINC000880702880 GD On-Demand Anodyne WNT3A 44 32 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)C1 ZINC000880702882 GD On-Demand Anodyne CCR3 41 34 CCNC(=O)CN1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880702884 FD On-Demand Anodyne SLC27A1 39 40 COc1ccccc1-c1ccc(C(=O)N[C@@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702886 GG On-Demand Anodyne HTR1A 21 42 COc1ccccc1-c1ccc(C(=O)N[C@@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702886 GG On-Demand Anodyne DRD2 24 42 COc1ccccc1-c1ccc(C(=O)N[C@@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702886 GG On-Demand Anodyne PLD1 42 36 COc1ccccc1-c1ccc(C(=O)N[C@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702890 GG On-Demand Anodyne HTR1A 21 42 COc1ccccc1-c1ccc(C(=O)N[C@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702890 GG On-Demand Anodyne DRD2 24 42 COc1ccccc1-c1ccc(C(=O)N[C@H](C)CN2CCC(C)CC2)c(O)n1 ZINC000880702890 GG On-Demand Anodyne PLD1 42 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(=O)N(C)CC1 ZINC000880702893 EC On-Demand Anodyne P2RY12 62 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(=O)N(C)CC1 ZINC000880702895 EC On-Demand Anodyne P2RY12 62 36 CN1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CCC1=O ZINC000880702899 GD On-Demand Anodyne CELA1 18 40 CN1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CCC1=O ZINC000880702899 GD On-Demand Anodyne GRIN2B 18 41 CN1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CCC1=O ZINC000880702899 GD On-Demand Anodyne PREP 57 50 CN1CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)CCC1=O ZINC000880702899 GD On-Demand Anodyne SLC12A5 45 33 CN1C[C@H](CNC(=O)c2cc(Br)ccc2C2CC2)CC1=O ZINC000880702925 FF On-Demand Anodyne CACNA1I 56 36 CN1C[C@@H](CNC(=O)c2cc(Br)ccc2C2CC2)CC1=O ZINC000880702926 FF On-Demand Anodyne CACNA1I 56 36 Cc1cc(-c2nc(C)c(C(=O)NC[C@H]3CC(=O)N(C)C3)s2)ccc1F ZINC000880702940 FF On-Demand Anodyne SCD1 26 41 Cc1cc(-c2nc(C)c(C(=O)NC[C@@H]3CC(=O)N(C)C3)s2)ccc1F ZINC000880702941 FF On-Demand Anodyne SCD1 26 41 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3ccc(C)cc3C)c2)CC1 ZINC000880702962 GI On-Demand Anodyne EPHX2 35 43 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3ccc(C)cc3C)c2)CC1 ZINC000880702962 GI On-Demand Anodyne LIMK2 27 42 O=C(NCCCN1CCCCC1=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880702964 FF On-Demand Anodyne CCR3 35 41 COc1ccccc1[C@@H]1C[C@H]1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880703022 GE On-Demand Anodyne DRD2 26 42 COc1ccccc1[C@@H]1C[C@H]1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880703022 GE On-Demand Anodyne DRD3 15 40 N#CC1(CNC(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)CCCCC1 ZINC000880703089 FE On-Demand Mild NPFFR1 43 37 O=C(COC1CC1)N1CCc2sccc2[C@H]1c1ccc(Cl)cc1 ZINC000880703151 EI On-Demand Anodyne TRPM8 15 57 O=C(COC1CC1)N1CCc2sccc2[C@@H]1c1ccc(Cl)cc1 ZINC000880703152 EI On-Demand Anodyne TRPM8 15 57 O=C(NCCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703171 ED On-Demand Anodyne HTR2A 18 40 O=C(NCCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703171 ED On-Demand Anodyne CCR3 36 45 O=C(NCCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703171 ED On-Demand Anodyne CHRNA7 15 48 O=C(NCCCN1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703171 ED On-Demand Anodyne EPHX2 22 48 O=C(C[C@@H]1CCNC1=O)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703194 FC On-Demand Anodyne HTR1A 20 40 O=C(C[C@@H]1CCNC1=O)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703194 FC On-Demand Anodyne HTR7 28 40 O=C(C[C@H]1CCNC1=O)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703195 FC On-Demand Anodyne HTR1A 20 40 O=C(C[C@H]1CCNC1=O)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703195 FC On-Demand Anodyne HTR7 28 40 CCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703202 EF On-Demand Anodyne SSTR5 41 38 CCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703202 EF On-Demand Anodyne CCR3 46 38 CCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703202 EF On-Demand Anodyne MCHR1 17 42 CCN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703202 EF On-Demand Anodyne WNT3A 47 35 C[C@H](CN1CCOCC1)NC(=O)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703204 ED On-Demand Anodyne P2RX3 24 41 O=C(COC1CC1)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703207 ED On-Demand Anodyne HTR1A 29 46 O=C(COC1CC1)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703207 ED On-Demand Anodyne DRD2 18 46 O=C(COC1CC1)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703207 ED On-Demand Anodyne HTR2A 17 42 O=C(COC1CC1)NC1(CN2CCN(c3ccccc3)CC2)CC1 ZINC000880703207 ED On-Demand Anodyne DRD3 20 46 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1cc(=O)c2ccccc2o1 ZINC000880703230 HI On-Demand Anodyne GPR35 43 33 COC(=O)C[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880703234 EE On-Demand Anodyne GABRA1 18 44 COC(=O)C[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880703234 EE On-Demand Anodyne MPO 50 35 COC(=O)C[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CC1 ZINC000880703234 EE On-Demand Anodyne GABRA2 15 44 O=C(NC[C@@H](CO)CC1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880703249 EG On-Demand Anodyne PDE4D 22 48 O=C(NC[C@@H](CO)CC1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880703249 EG On-Demand Anodyne CACNA1I 46 37 O=C(NC[C@H](CO)CC1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880703250 EG On-Demand Anodyne PDE4D 22 48 O=C(NC[C@H](CO)CC1CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880703250 EG On-Demand Anodyne CACNA1I 46 37 O=C(NCc1cccnc1N1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703252 GF On-Demand Anodyne SCN10A 20 45 O=C(NCc1cccnc1N1CCOCC1)Nc1ccnn1-c1ccc(F)cc1 ZINC000880703252 GF On-Demand Anodyne STAT6 55 35 CCOC(=O)N1CCN(C(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703259 FE On-Demand Anodyne P2RY12 45 35 COC(=O)N(C)CCNC(=O)c1cc2ccccc2cc1F ZINC000880703275 DE On-Demand Anodyne POLR1A 46 40 O=C(c1cccc2nsnc12)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880703297 EG On-Demand Anodyne L3MBTL3 59 36 O=C(c1cccc2nsnc12)N1CCC([C@H]2CCCCO2)CC1 ZINC000880703298 EG On-Demand Anodyne L3MBTL3 59 36 COC[C@@H](CO)NC(=O)Nc1cccc(Oc2ccc(C)cc2C)c1 ZINC000880703326 EG On-Demand Anodyne KCNK3 55 36 COC[C@@H](CO)NC(=O)Nc1cccc(Oc2ccc(C)cc2C)c1 ZINC000880703326 EG On-Demand Anodyne KCNK9 58 36 CCOC(=O)N1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703371 GF On-Demand Anodyne GRIN2B 18 42 CCOC(=O)N1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703371 GF On-Demand Anodyne EPHX2 47 42 CN1C[C@@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703375 DC On-Demand Anodyne PYGL 21 42 CN1C[C@@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703375 DC On-Demand Anodyne PLD1 43 38 CN1C[C@@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703375 DC On-Demand Anodyne PYGM 19 42 CN1C[C@@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703375 DC On-Demand Anodyne PLD2 44 37 CN1C[C@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703376 DC On-Demand Anodyne PYGL 21 42 CN1C[C@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703376 DC On-Demand Anodyne PLD1 43 38 CN1C[C@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703376 DC On-Demand Anodyne PYGM 19 42 CN1C[C@H](CNC(=O)c2cc3cc(F)ccc3[nH]c2=O)CC1=O ZINC000880703376 DC On-Demand Anodyne PLD2 44 37 CN1CCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)CCC1=O ZINC000880703381 FE On-Demand Anodyne P2RX7 45 40 O=C(NC[C@H](CO)CC1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880703395 DE On-Demand Anodyne GABRA1 18 47 O=C(NC[C@H](CO)CC1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880703395 DE On-Demand Anodyne GABRA2 16 47 O=C(NC[C@@H](CO)CC1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880703396 DE On-Demand Anodyne GABRA1 18 47 O=C(NC[C@@H](CO)CC1CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880703396 DE On-Demand Anodyne GABRA2 16 47 CNC(=O)CN1CCC(NC(=O)Nc2ccnn2-c2ccc(F)cc2)CC1 ZINC000880703450 FD On-Demand Anodyne WNT3A 47 33 CN1C[C@@H](CNC(=O)CC[C@@H]2CCc3ccccc32)CC1=O ZINC000880703458 DE On-Demand Anodyne MTNR1A 21 44 CN1C[C@@H](CNC(=O)CC[C@@H]2CCc3ccccc32)CC1=O ZINC000880703458 DE On-Demand Anodyne MTNR1B 23 44 CN1C[C@@H](CNC(=O)CC[C@H]2CCc3ccccc32)CC1=O ZINC000880703459 DE On-Demand Anodyne MTNR1A 21 44 CN1C[C@@H](CNC(=O)CC[C@H]2CCc3ccccc32)CC1=O ZINC000880703459 DE On-Demand Anodyne MTNR1B 23 44 O=C(NCC(O)(C1CC1)C1CC1)c1cc2ccccc2cc1F ZINC000880703463 DG On-Demand Anodyne KCNJ11 65 34 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@@H]([C@@H]2CCCCO2)C1 ZINC000880703492 FG On-Demand Anodyne WNT3A 47 33 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@@H]([C@H]2CCCCO2)C1 ZINC000880703493 FG On-Demand Anodyne WNT3A 47 33 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@H]([C@H]2CCCCO2)C1 ZINC000880703494 FG On-Demand Anodyne WNT3A 47 33 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC[C@H]([C@@H]2CCCCO2)C1 ZINC000880703495 FG On-Demand Anodyne WNT3A 47 33 C[C@H]1CN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC[C@@H](C)O1 ZINC000880703510 DE On-Demand Anodyne L3MBTL3 47 37 C[C@H]1CN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC[C@@H](C)O1 ZINC000880703511 DE On-Demand Anodyne L3MBTL3 47 37 N#CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880703516 DF On-Demand Mild HCN1 51 31 N#CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880703516 DF On-Demand Mild HCN4 48 31 Cc1coc(C(=O)N[C@H](C)CN2CCC(C)CC2)c1 ZINC000880703572 CE On-Demand Anodyne P2RX3 29 40 Cc1coc(C(=O)N[C@H](C)CN2CCC(C)CC2)c1 ZINC000880703572 CE On-Demand Anodyne PLD1 52 39 Cc1coc(C(=O)N[C@@H](C)CN2CCC(C)CC2)c1 ZINC000880703573 CE On-Demand Anodyne P2RX3 29 40 Cc1coc(C(=O)N[C@@H](C)CN2CCC(C)CC2)c1 ZINC000880703573 CE On-Demand Anodyne PLD1 52 39 Cc1coc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)c1 ZINC000880703582 EF On-Demand Anodyne HTR1A 30 41 Cc1coc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)c1 ZINC000880703582 EF On-Demand Anodyne DRD2 18 41 Cc1coc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)c1 ZINC000880703582 EF On-Demand Anodyne HTR2A 23 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C)C1)C2 ZINC000880703602 DD On-Demand Anodyne MTNR1A 40 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C)C1)C2 ZINC000880703602 DD On-Demand Anodyne MTNR1B 37 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C)C1)C2 ZINC000880703605 DD On-Demand Anodyne MTNR1A 40 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C)C1)C2 ZINC000880703605 DD On-Demand Anodyne MTNR1B 37 41 Cn1nnc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)n1 ZINC000880703651 EC On-Demand Anodyne HTR1A 40 42 Cn1nnc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)n1 ZINC000880703651 EC On-Demand Anodyne DRD2 21 41 Cn1nnc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)n1 ZINC000880703651 EC On-Demand Anodyne DRD3 29 40 Cn1nnc(C(=O)NC2(CN3CCN(c4ccccc4)CC3)CC2)n1 ZINC000880703651 EC On-Demand Anodyne HTR7 45 37 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cncc(C)n1)C2 ZINC000880703662 EE On-Demand Anodyne NQO2 41 45 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cncc(C)n1)C2 ZINC000880703662 EE On-Demand Anodyne MTNR1A 66 45 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cncc(C)n1)C2 ZINC000880703662 EE On-Demand Anodyne MTNR1B 54 41 O=C(c1cnc2cc[nH]c2c1)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880703686 DF On-Demand Anodyne L3MBTL3 58 36 O=C(c1cnc2cc[nH]c2c1)N1CCC([C@H]2CCCCO2)CC1 ZINC000880703687 DF On-Demand Anodyne L3MBTL3 58 36 COc1ccccc1[C@@H]1C[C@H]1NC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880703693 EH On-Demand Anodyne KCNA3 40 34 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880703694 GG On-Demand Bother L3MBTL3 19 44 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CCC([C@H]2CCCCO2)CC1 ZINC000880703695 GG On-Demand Bother L3MBTL3 19 44 COC(=O)N(C)CCNC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880703709 EF On-Demand Anodyne LIPE 18 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1OC ZINC000880703714 GF On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1OC ZINC000880703715 GF On-Demand Anodyne FPR1 45 36 COC[C@]1(CO)CCN(C(=O)Nc2cccc(Oc3ccc(C)cc3C)c2)C1 ZINC000880703750 GH On-Demand Anodyne S1PR2 25 40 COC(=O)N(C)CCNC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880703776 DD On-Demand Anodyne RAF1 24 41 Cc1cncc(CCNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)n1 ZINC000880703792 GE On-Demand Anodyne Q9NAW4_PLAFA 27 42 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)nc2)c1 ZINC000880703818 GG On-Demand Anodyne DRD4 40 31 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)nc2)c1 ZINC000880703818 GG On-Demand Anodyne MTNR1B 22 56 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)nc2)c1 ZINC000880703819 GG On-Demand Anodyne DRD4 40 31 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)nc2)c1 ZINC000880703819 GG On-Demand Anodyne MTNR1B 22 56 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703863 GG On-Demand Anodyne PAPA1_CARPA 37 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703863 GG On-Demand Anodyne CCKAR 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703863 GG On-Demand Anodyne FPR1 46 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703864 GG On-Demand Anodyne PAPA1_CARPA 37 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703864 GG On-Demand Anodyne CCKAR 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccccc1Cl ZINC000880703864 GG On-Demand Anodyne FPR1 46 38 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880703881 FG On-Demand Anodyne HTR1A 42 39 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880703881 FG On-Demand Anodyne ADRA1A 25 41 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880703881 FG On-Demand Anodyne MBTPS1 40 32 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@@H](O)C13CCC3)C2 ZINC000880703902 DE On-Demand Anodyne MTNR1A 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@@H](O)C13CCC3)C2 ZINC000880703902 DE On-Demand Anodyne MTNR1B 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](O)C13CCC3)C2 ZINC000880703903 DE On-Demand Anodyne MTNR1A 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H](O)C13CCC3)C2 ZINC000880703903 DE On-Demand Anodyne MTNR1B 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](O)C13CCC3)C2 ZINC000880703904 DE On-Demand Anodyne MTNR1A 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](O)C13CCC3)C2 ZINC000880703904 DE On-Demand Anodyne MTNR1B 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)C13CCC3)C2 ZINC000880703905 DE On-Demand Anodyne MTNR1A 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)C13CCC3)C2 ZINC000880703905 DE On-Demand Anodyne MTNR1B 24 41 COC(=O)N(C)CCNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880703919 EE On-Demand Anodyne PDE4D 15 41 COC(=O)N(C)CCNC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880703943 ED On-Demand Anodyne PDK1 43 33 O=C(c1ccc(CN2CCOCC2)o1)N1CCC([C@H]2CCCCO2)CC1 ZINC000880704046 FF On-Demand Anodyne L3MBTL3 25 40 O=C(c1ccc(CN2CCOCC2)o1)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880704047 FF On-Demand Anodyne L3MBTL3 25 40 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)nc2)c1 ZINC000880704062 EE On-Demand Anodyne CHRNA7 18 40 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)nc2)c1 ZINC000880704062 EE On-Demand Anodyne MTNR1A 17 48 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)nc2)c1 ZINC000880704062 EE On-Demand Anodyne MTNR1B 23 48 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)nc2)c1 ZINC000880704063 EE On-Demand Anodyne CHRNA7 18 40 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)nc2)c1 ZINC000880704063 EE On-Demand Anodyne MTNR1A 17 48 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)nc2)c1 ZINC000880704063 EE On-Demand Anodyne MTNR1B 23 48 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCCC2)c(O)n1 ZINC000880704072 FH On-Demand Mild KCNA3 45 40 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCCC2)c(O)n1 ZINC000880704072 FH On-Demand Mild HCN1 74 42 COc1ccccc1-c1ccc(C(=O)NCC2(C#N)CCCCC2)c(O)n1 ZINC000880704072 FH On-Demand Mild HCN4 57 42 COC(=O)N(C)CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880704101 DD On-Demand Anodyne NQO2 42 44 COC(=O)N(C)CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880704101 DD On-Demand Anodyne MTNR1A 63 46 COC(=O)N(C)CCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880704101 DD On-Demand Anodyne MTNR1B 54 41 COC(=O)N(C)CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880704102 DD On-Demand Anodyne NQO2 42 44 COC(=O)N(C)CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880704102 DD On-Demand Anodyne MTNR1A 63 46 COC(=O)N(C)CCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880704102 DD On-Demand Anodyne MTNR1B 54 41 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1nc(Cl)ccc1Cl ZINC000880704148 HJ On-Demand Anodyne CNR1 55 33 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)NC[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880704236 GE On-Demand Anodyne SMO 29 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)NC[C@H]3C2)n(-c2ccccc2)n1 ZINC000880704237 GE On-Demand Anodyne SMO 29 43 C[C@@H]1C[C@H]1c1cc(NC(=O)NCCn2ccnc2)n(-c2ccccc2)n1 ZINC000880704280 FG On-Demand Anodyne TNF 30 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NCCn2ccnc2)n(-c2ccccc2)n1 ZINC000880704280 FG On-Demand Anodyne MAPK14 26 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NCCn2ccnc2)n(-c2ccccc2)n1 ZINC000880704280 FG On-Demand Anodyne QPCT 25 41 O=C(COc1ccc(-c2ccccc2)cc1)Nc1cc(-c2nnc3n2CCCCC3)ccc1F ZINC000880704294 JK On-Demand Anodyne CPT1A 83 44 N#CC1(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CCCCC1 ZINC000880704344 EG On-Demand Mild GABRA1 16 47 C[C@@H]1C[C@H]1c1cc(NC(=O)Nc2cnn(CCO)c2)n(-c2ccccc2)n1 ZINC000880704350 FF On-Demand Anodyne MAPK10 15 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc([C@@H]2C[C@H]2C)nn1-c1ccccc1 ZINC000880704362 FF On-Demand Anodyne P2RY12 17 41 CC(=O)NCCCNC(=O)Nc1cc([C@@H]2C[C@H]2C)nn1-c1ccccc1 ZINC000880704464 FF On-Demand Anodyne MAPK14 15 41 C[C@@H](Cn1cncn1)NC(=O)Nc1cc([C@@H]2C[C@H]2C)nn1-c1ccccc1 ZINC000880704497 FF On-Demand Anodyne HIS3 67 37 C[C@@H]1C[C@H]1c1cc(NC(=O)NCc2cccnc2)n(-c2ccccc2)n1 ZINC000880704506 EH On-Demand Anodyne CYP2C9 16 45 C[C@@H]1C[C@H]1c1cc(NC(=O)NCc2cccnc2)n(-c2ccccc2)n1 ZINC000880704506 EH On-Demand Anodyne NAMPT 85 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CCC2(CC1)CC2(F)F ZINC000880704514 GG On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CCC2(CC1)CC2(F)F ZINC000880704515 GG On-Demand Anodyne PAPA1_CARPA 33 40 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PLG 20 44 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne ACE 47 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne TYR 37 43 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne OPRM1 56 44 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne OPRD1 55 44 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PPIA 35 40 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CELA1 18 42 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MME 111 45 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne ANPEP 78 38 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne TACR1 20 60 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTRA_BOVIN 40 32 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne FCER2 107 43 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne GRB2 21 40 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CASP3 21 52 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne BMP1 25 47 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne TACR2 17 42 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne KLK3 90 42 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTSB 117 59 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PAPA1_CARPA 111 57 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CYSP_TRYCR 84 56 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CCKAR 33 43 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTSK 52 57 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTSL 92 57 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PGA 34 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne TIMP3 95 43 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CAPNS1 90 48 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP2 31 47 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP3 52 51 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP8 35 44 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne GRIA1 48 37 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne HLA-DRB1 83 40 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CELA2A 41 32 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne HDAC1 15 52 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne HDAC2 17 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne REN 45 46 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne REN1 22 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP11 75 37 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTSS 42 57 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CAPN1 128 54 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP9 37 48 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CASP1 29 44 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CTRC 45 45 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CAPN2 163 59 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne ACE2 74 39 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PLAU 42 45 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CASP6 20 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne CASP9 42 41 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne LAP3 44 34 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne TPSAB1 45 37 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP7 25 40 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne MMP1 51 48 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne FPR1 81 48 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne NPR 83 42 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne PSMB5 51 45 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne BLA1_STEMA 51 35 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne KDM1A 20 60 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne GPR142 79 42 CNC(=O)Nc1cccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1 ZINC000880704517 IH On-Demand Anodyne KCNK3 50 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC[C@H]2C(=O)NC2CC2)n(-c2ccccc2)n1 ZINC000880704529 GG On-Demand Anodyne P2RY12 19 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)n(-c2ccccc2)n1 ZINC000880704530 GG On-Demand Anodyne P2RY12 19 43 CCNC(=O)CNC(=O)Nc1cc([C@@H]2C[C@H]2C)nn1-c1ccccc1 ZINC000880704573 EE On-Demand Anodyne MAPK14 15 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NCCCO)n(-c2ccccc2)n1 ZINC000880704601 DE On-Demand Anodyne MAPK14 15 40 O=C(NC1CCC2(CC1)CC2(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880704681 FH On-Demand Anodyne GABRA1 17 43 O=C(NC1CCC2(CC1)CC2(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880704681 FH On-Demand Anodyne GABRA2 16 43 Cc1cc([C@@H]2CCCN2C(=O)Nc2cc([C@@H]3C[C@H]3C)nn2-c2ccccc2)on1 ZINC000880704710 GJ On-Demand Anodyne CPT1A 43 37 C[C@@H]1C[C@H]1c1cc(NC(=O)NC2CCN(C)CC2)n(-c2ccccc2)n1 ZINC000880704712 FG On-Demand Anodyne EPHX2 26 40 NC(=O)[C@@H]1CC[C@H](C(=O)NC2CCC3(CC2)CC3(F)F)N1Cc1ccccc1 ZINC000880704771 GF On-Demand Anodyne SIGMAR1 17 43 Cc1cc([C@@H]2CCCN2C(=O)Nc2cc([C@@H]3C[C@H]3C)nn2-c2ccccc2)no1 ZINC000880704804 GJ On-Demand Anodyne CPT1A 59 40 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3ccc(C)cc3C)c2)CC1 ZINC000880704815 GJ On-Demand Anodyne LIMK2 27 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC(O)CC2)n(-c2ccccc2)n1 ZINC000880704836 EF On-Demand Anodyne EPHX2 15 43 C[C@@H]1C[C@H]1c1cc(NC(=O)Nc2cnn(C)c2)n(-c2ccccc2)n1 ZINC000880704947 EG On-Demand Anodyne MAPK10 15 44 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc([C@@H]3C[C@H]3C)nn2-c2ccccc2)C1 ZINC000880705025 GG On-Demand Anodyne EPHX2 26 46 CCC(=O)N1CC[C@H](NC(=O)Nc2cc([C@@H]3C[C@H]3C)nn2-c2ccccc2)C1 ZINC000880705026 GG On-Demand Anodyne EPHX2 26 46 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)CC[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880705027 GF On-Demand Anodyne SMO 30 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)CC[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705028 GF On-Demand Anodyne SMO 30 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2C[C@H]3C[C@H](O)CC[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705177 GH On-Demand Anodyne RBP4 45 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2C[C@@H]3CC[C@H](O)C[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705178 GH On-Demand Anodyne RBP4 45 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2C[C@H]3C[C@@H](O)CC[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705179 GH On-Demand Anodyne RBP4 45 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2C[C@@H]3CC[C@@H](O)C[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705180 GH On-Demand Anodyne RBP4 45 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC(O)(C(F)F)CC2)n(-c2ccccc2)n1 ZINC000880705235 GH On-Demand Anodyne CACNA1H 42 33 C[C@@H]1C[C@H]1c1cc(NC(=O)NC[C@H](O)CN2CCOCC2)n(-c2ccccc2)n1 ZINC000880705289 GD On-Demand Anodyne TNF 32 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NC[C@H](O)CN2CCOCC2)n(-c2ccccc2)n1 ZINC000880705289 GD On-Demand Anodyne MAPK14 17 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NC[C@@H](O)CN2CCOCC2)n(-c2ccccc2)n1 ZINC000880705290 GD On-Demand Anodyne TNF 32 41 C[C@@H]1C[C@H]1c1cc(NC(=O)NC[C@@H](O)CN2CCOCC2)n(-c2ccccc2)n1 ZINC000880705290 GD On-Demand Anodyne MAPK14 17 41 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)OC[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705298 GF On-Demand Anodyne SMO 28 42 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)OC[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880705299 GF On-Demand Anodyne SMO 28 42 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H](N3CCCC3=O)C2)n(-c2ccccc2)n1 ZINC000880705301 GG On-Demand Anodyne SMO 28 41 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@@H](N3CCCC3=O)C2)n(-c2ccccc2)n1 ZINC000880705302 GG On-Demand Anodyne SMO 28 41 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCOC3(CCOCC3)C2)n(-c2ccccc2)n1 ZINC000880705303 GG On-Demand Anodyne EPHX2 17 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCO[C@@]3(CCOC3)C2)n(-c2ccccc2)n1 ZINC000880705345 GG On-Demand Anodyne EPHX2 16 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCO[C@]3(CCOC3)C2)n(-c2ccccc2)n1 ZINC000880705346 GG On-Demand Anodyne EPHX2 16 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC(F)(F)CC2)n(-c2ccccc2)n1 ZINC000880705355 FI On-Demand Anodyne CACNA1H 45 34 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC(C(F)(F)F)C2)n(-c2ccccc2)n1 ZINC000880705375 FI On-Demand Anodyne RBP4 54 33 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@@H](F)C2)n(-c2ccccc2)n1 ZINC000880705542 EH On-Demand Anodyne RBP4 43 30 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H](F)C2)n(-c2ccccc2)n1 ZINC000880705546 EH On-Demand Anodyne RBP4 43 30 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@@H](N3CCOC3=O)C2)n(-c2ccccc2)n1 ZINC000880705618 GG On-Demand Anodyne SMO 24 41 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H](N3CCOC3=O)C2)n(-c2ccccc2)n1 ZINC000880705619 GG On-Demand Anodyne SMO 24 41 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC3(CCNC3=O)CC2)n(-c2ccccc2)n1 ZINC000880705641 GG On-Demand Anodyne CACNA1H 42 37 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1cc(Cl)nc(Cl)c1 ZINC000880705680 HJ On-Demand Anodyne CNR1 52 32 CCN1CC[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880705681 EG On-Demand Bother CCR3 20 41 CCN1CC[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880705681 EG On-Demand Bother CACNA1I 63 37 C[C@@H]1C[C@H]1c1cc(NC(=O)NCC(=O)N2CCOCC2)n(-c2ccccc2)n1 ZINC000880705703 GD On-Demand Anodyne TNF 31 40 C[C@@H]1C[C@H]1c1cc(NC(=O)NCC(=O)N2CCOCC2)n(-c2ccccc2)n1 ZINC000880705703 GD On-Demand Anodyne MAPK14 17 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)NC(=O)[C@H]3C2)n(-c2ccccc2)n1 ZINC000880705787 GD On-Demand Anodyne SMO 32 45 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCN3C(=O)NC(=O)[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880705788 GD On-Demand Anodyne SMO 32 45 COC1CC(CCNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880705909 EH On-Demand Bother TBXA2R 21 41 COC[C@]1(C)CCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880705953 EH On-Demand Bother CACNA1D 51 32 COC[C@@]1(C)CCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880705954 EH On-Demand Bother CACNA1D 51 32 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCCC[C@H]2c2nc[nH]n2)n(-c2ccccc2)n1 ZINC000880706062 GH On-Demand Anodyne CPT1A 107 42 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCCC[C@@H]2c2nc[nH]n2)n(-c2ccccc2)n1 ZINC000880706063 GH On-Demand Anodyne CPT1A 107 42 C[C@@H]1C[C@H]1c1cc(NC(=O)NCc2ccc(N)nc2)n(-c2ccccc2)n1 ZINC000880706107 FG On-Demand Anodyne NAMPT 22 46 C[C@@H]1C[C@H]1c1cc(NC(=O)Nc2ccn(CCO)n2)n(-c2ccccc2)n1 ZINC000880706140 FF On-Demand Anodyne TNF 40 38 CCN1CCC(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880706252 EG On-Demand Bother EPHX2 32 40 CCN1CCC(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880706252 EG On-Demand Bother CXCR3 19 40 CN1CCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880706255 DF On-Demand Bother WDR5 40 44 COCC[C@@H](C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706312 DG On-Demand Bother KCNMA1 20 42 COCC[C@H](C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706313 DG On-Demand Bother KCNMA1 20 42 COCCCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706317 EH On-Demand Bother TBXA2R 20 43 COCCCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706317 EH On-Demand Bother CACNA1D 51 33 COCCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706448 DG On-Demand Bother TBXA2R 20 41 COCCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706448 DG On-Demand Bother CACNA1D 53 33 CN1CCC[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706566 EG On-Demand Bother NMBR 40 30 CN1CCC[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706566 EG On-Demand Bother CACNA1I 49 33 CN1CCC[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706566 EG On-Demand Bother WDR5 34 40 CN(CCN1CCOCC1)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706570 FF On-Demand Bother CASR 46 37 CCOCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706624 DG On-Demand Bother TBXA2R 22 43 C[C@@H]1C[C@H]1c1cc(NC(=O)N[C@H]2CCOC2=O)n(-c2ccccc2)n1 ZINC000880706644 EE On-Demand Anodyne LUXR 68 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N[C@H]2CCOC2=O)n(-c2ccccc2)n1 ZINC000880706644 EE On-Demand Anodyne TRAR 81 42 C[C@@H]1C[C@H]1c1cc(NC(=O)N[C@H]2CCOC2=O)n(-c2ccccc2)n1 ZINC000880706644 EE On-Demand Anodyne LASR 58 42 Cc1cccc(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)n1 ZINC000880706645 EH On-Demand Bother CACNA1C 51 35 Cc1cccc(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)n1 ZINC000880706645 EH On-Demand Bother CACNA1D 78 35 CN1CCC(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880706673 EG On-Demand Bother CACNA1I 61 39 CN1CCC(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880706673 EG On-Demand Bother WDR5 36 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CCC(F)CC2)n(-c2ccccc2)n1 ZINC000880706721 EH On-Demand Anodyne EPHX2 15 41 CN1CCC[C@H](NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706754 EG On-Demand Bother BIRC2 16 43 COCCN(CCOC)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706777 FG On-Demand Bother CACNA1D 41 34 COCCN(CCOC)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706777 FG On-Demand Bother KCNMA1 19 40 CN1CCN(C)[C@@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706801 FE On-Demand Bother WDR5 36 40 CN1CCN(C)[C@H](CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880706802 FE On-Demand Bother WDR5 36 40 CCOCCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706825 EH On-Demand Bother TBXA2R 22 44 CCN(Cc1ccncc1)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706832 FI On-Demand Bother MMP8 23 41 CCN(Cc1ccncc1)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706832 FI On-Demand Bother MMP1 17 41 CNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706848 CF On-Demand Bother TBXA2R 24 40 CNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706848 CF On-Demand Bother KCNMA1 18 40 COCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706856 DG On-Demand Bother TBXA2R 21 40 COCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706856 DG On-Demand Bother CACNA1D 56 36 COCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880706856 DG On-Demand Bother KCNMA1 19 40 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H]3C[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880706960 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@@H]3C[C@@H]3C2)n(-c2ccccc2)n1 ZINC000880706961 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@@H]3C[C@H]3C2)n(-c2ccccc2)n1 ZINC000880706962 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H]3C[C@H]3C2)n(-c2ccccc2)n1 ZINC000880706963 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H]3CC[C@@H](C2)[S@]3=O)n(-c2ccccc2)n1 ZINC000880707020 GH On-Demand Anodyne SMO 29 42 C[C@@H]1C[C@H]1c1cc(NC(=O)N2CC[C@H]3CC[C@@H](C2)[S@@]3=O)n(-c2ccccc2)n1 ZINC000880707021 GH On-Demand Anodyne SMO 29 42 C[C@@H]1C[C@H]1c1cc(NC(=O)NCCN2CCCC2=O)n(-c2ccccc2)n1 ZINC000880707036 FF On-Demand Anodyne MAPK14 15 48 COC[C@H](C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880707040 DG On-Demand Bother CACNA1D 40 35 COC[C@@H](C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880707041 DG On-Demand Bother CACNA1D 40 35 COCC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCC1 ZINC000880707269 EH On-Demand Bother CACNA1C 45 34 COCC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCC1 ZINC000880707269 EH On-Demand Bother CACNA1D 70 34 COCC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCC1 ZINC000880707269 EH On-Demand Bother NMBR 52 31 CSC1(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCN(C)CC1 ZINC000880707328 GH On-Demand Bother NMBR 46 30 CSC1(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880707353 EH On-Demand Bother NMBR 61 33 CO[C@@](C)(CNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C)C1CC1 ZINC000880707425 EH On-Demand Bother NMBR 42 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCO[C@H]1c1nccn1C)C2 ZINC000880707464 FE On-Demand Anodyne MTNR1A 25 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCO[C@H]1c1nccn1C)C2 ZINC000880707464 FE On-Demand Anodyne MTNR1B 23 42 CCC1(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)COC1 ZINC000880707616 EG On-Demand Bother NMBR 64 34 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880707759 GE On-Demand Anodyne F10 23 47 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880707759 GE On-Demand Anodyne PRNP 57 48 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(S(=O)(=O)C(F)F)cc1 ZINC000880707759 GE On-Demand Anodyne STAT6 53 32 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880707794 JK On-Demand Anodyne F10 18 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880707794 JK On-Demand Anodyne PRNP 46 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880707794 JK On-Demand Anodyne STAT6 58 36 N#Cc1cc(NC(=O)NCC[C@@H](O)COCc2ccccc2)c(F)cc1F ZINC000880707972 GF On-Demand Mild ADRB1 51 45 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cc(C#N)c(F)cc1F)CC2 ZINC000880708021 GI On-Demand Mild SLC18A2 44 32 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cc(C#N)c(F)cc1F)CC2 ZINC000880708022 GI On-Demand Mild SLC18A2 44 32 N#Cc1cc(NC(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880708042 GH On-Demand Mild EPHX2 20 42 N#Cc1cc(NC(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880708043 GH On-Demand Mild EPHX2 20 42 CN(C)CC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCC1 ZINC000880708167 EG On-Demand Bother NMBR 41 30 CC1CN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880708191 CG On-Demand Bother RBP4 51 33 N#Cc1cc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)c(F)cc1F ZINC000880708295 GD On-Demand Mild EPHX2 18 48 N#Cc1cc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)c(F)cc1F ZINC000880708297 GD On-Demand Mild EPHX2 18 48 CSC1(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CCOCC1 ZINC000880708347 GH On-Demand Bother NMBR 47 31 COCC(C)(C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880708388 DG On-Demand Bother CACNA1D 44 36 O=C(CN1C(=O)N[C@@]2(CCc3ccccc32)C1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880708482 HD On-Demand Anodyne STAT6 65 36 O=C(CN1C(=O)N[C@]2(CCc3ccccc32)C1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880708483 HD On-Demand Anodyne STAT6 65 36 CC(C)(C)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880708635 CH On-Demand Bother TBXA2R 24 46 COCC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880708648 DG On-Demand Bother CACNA1C 53 37 COCC1(NC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880708648 DG On-Demand Bother CACNA1D 83 37 C[C@H]1c2sccc2CCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880708680 EI On-Demand Mild TRPM8 16 40 Cn1nccc1[C@@H]1OCCC[C@H]1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880708681 GH On-Demand Anodyne PDE4D 21 40 Cn1nccc1[C@@H]1OCCC[C@H]1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880708681 GH On-Demand Anodyne CACNA1I 57 38 CN(C)[C@@H]1CCCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880708737 FH On-Demand Bother SFRP1 67 34 CN(C)[C@@H]1CCCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880708737 FH On-Demand Bother WNT3 57 34 CCONC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880708771 CF On-Demand Bother CACNA1D 52 34 CCONC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880708771 CF On-Demand Bother KCNMA1 24 40 N#Cc1cc(NC(=O)N2CCC[C@@](O)(c3ccccc3)C2)c(F)cc1F ZINC000880708781 FG On-Demand Mild EPHX2 16 43 N#Cc1cc(NC(=O)N2CCC[C@](O)(c3ccccc3)C2)c(F)cc1F ZINC000880708783 FG On-Demand Mild EPHX2 16 43 N#Cc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c(F)cc1F ZINC000880708816 GG On-Demand Mild KCNQ2 42 33 N#Cc1cc(NC(=O)NC2CCN(c3ccccc3C#N)CC2)c(F)cc1F ZINC000880708816 GG On-Demand Mild EPHX2 33 40 N#Cc1cc(NC(=O)NCC[C@H](O)C(F)F)c(F)cc1F ZINC000880708904 DD On-Demand Mild ADRB1 40 34 N#Cc1cc(NC(=O)NCC[C@@H](O)C(F)F)c(F)cc1F ZINC000880708905 DD On-Demand Mild ADRB1 40 34 CCn1nccc1[C@@H]1OCC[C@H]1NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880708941 GF On-Demand Anodyne PDK1 43 34 CN(C)C[C@@H]1CCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880708966 EG On-Demand Bother NR1D1 16 42 CN1CCCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)CC1 ZINC000880708980 EG On-Demand Bother WDR5 38 41 CC(C)(C)OC(=O)CN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880709092 GF On-Demand Mild CXCR3 18 41 COc1ccccc1[C@H]1CN(C(=O)Nc2cc(C#N)c(F)cc2F)CCO1 ZINC000880709100 FG On-Demand Mild RBP4 40 40 COc1ccccc1[C@@H]1CN(C(=O)Nc2cc(C#N)c(F)cc2F)CCO1 ZINC000880709101 FG On-Demand Mild RBP4 40 40 N#Cc1cc(NC(=O)N2CCC(c3nc(C4CCC4)no3)CC2)c(F)cc1F ZINC000880709123 GH On-Demand Mild SMO 38 49 N#Cc1cc(NC(=O)N2CCC(c3nc(C4CCC4)no3)CC2)c(F)cc1F ZINC000880709123 GH On-Demand Mild ETHR 63 49 N#Cc1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)c(F)cc1F ZINC000880709148 CE On-Demand Mild EPHX2 16 44 CN1CCN(C2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)CC1 ZINC000880709171 FE On-Demand Mild L3MBTL3 64 40 COC[C@@H]1CCCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880709256 EH On-Demand Bother CACNA1D 48 36 C[C@@H](CNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C)CN1CCN(C)CC1 ZINC000880709263 GF On-Demand Bother WDR5 35 40 C#CCCCNC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880709298 DG On-Demand Mild TBXA2R 23 41 N#Cc1cc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)c(F)cc1F ZINC000880709310 FG On-Demand Mild EPHX2 19 53 N#Cc1cc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)c(F)cc1F ZINC000880709313 FG On-Demand Mild EPHX2 19 53 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)C2)cc1F ZINC000880709326 GI On-Demand Mild RBP4 33 42 COC[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880709330 CE On-Demand Mild LGMN 42 33 Cc1cncc(CNC(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)c1 ZINC000880709507 EH On-Demand Bother NAMPT 17 48 N#Cc1cc(NC(=O)NCCN2CC[C@H](O)C2)c(F)cc1F ZINC000880709688 DD On-Demand Mild CCR3 29 42 N#Cc1cc(NC(=O)NCCN2CC[C@@H](O)C2)c(F)cc1F ZINC000880709690 DD On-Demand Mild CCR3 29 42 CC[C@@H](O)CNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880709810 CD On-Demand Mild ADRB1 41 35 N#Cc1cc(NC(=O)NC[C@H]2CCCN(CC3CC3)C2)c(F)cc1F ZINC000880709900 EG On-Demand Mild CCR3 65 39 N#Cc1cc(NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(F)cc1F ZINC000880709901 EG On-Demand Mild CCR3 65 39 N#Cc1cc(NC(=O)NCC2CCN(CC3CC3)CC2)c(F)cc1F ZINC000880709927 EG On-Demand Mild CCR3 47 40 N#Cc1cc(NC(=O)NCC2CCN(CC3CC3)CC2)c(F)cc1F ZINC000880709927 EG On-Demand Mild CACNA1I 64 37 N#Cc1cc(NC(=O)NCCCC2CC2)c(F)cc1F ZINC000880709946 CG On-Demand Mild CCR3 27 41 N#Cc1cc(NC(=O)N2CCN(c3nccnn3)CC2)c(F)cc1F ZINC000880709968 ED On-Demand Mild FAAH 23 42 COC[C@@H]1CCCCN(C(=O)Nc2cc([N+](=O)[O-])ccc2C(C)(C)C)C1 ZINC000880709969 FI On-Demand Bother CACNA1D 44 36 Cn1ncc(C2CC2)c1CNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880709973 EF On-Demand Mild CSNK2A1 34 40 C[C@H](O)CN(C)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880710020 DF On-Demand Bother COLA 41 36 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880710055 GG On-Demand Bother WDR5 36 41 N#Cc1cc(NC(=O)NCc2cccnc2N2CCCC2)c(F)cc1F ZINC000880710060 FG On-Demand Mild TRPV1 34 40 N#Cc1cc(NC(=O)NCc2cccnc2N2CCCC2)c(F)cc1F ZINC000880710060 FG On-Demand Mild SCN2A 19 47 N#Cc1cc(NC(=O)NCc2cccnc2N2CCCC2)c(F)cc1F ZINC000880710060 FG On-Demand Mild SCN10A 22 47 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c(F)cc1F ZINC000880710101 GF On-Demand Mild CCR3 57 38 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c(F)cc1F ZINC000880710101 GF On-Demand Mild CXCR3 15 40 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@H](O)C3)cc2)c(F)cc1F ZINC000880710101 GF On-Demand Mild MCHR1 27 41 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c(F)cc1F ZINC000880710102 GF On-Demand Mild CCR3 57 38 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c(F)cc1F ZINC000880710102 GF On-Demand Mild CXCR3 15 40 N#Cc1cc(NC(=O)NCc2ccc(CN3CC[C@@H](O)C3)cc2)c(F)cc1F ZINC000880710102 GF On-Demand Mild MCHR1 27 41 CCn1nccc1[C@@H]1OCC[C@H]1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880710112 GG On-Demand Anodyne PDE4D 24 41 N#Cc1cc(NC(=O)N2C[C@H]3CC[C@@H](O)C[C@H]3C2)c(F)cc1F ZINC000880710158 DE On-Demand Mild RBP4 40 33 N#Cc1cc(NC(=O)N2C[C@@H]3CC[C@H](O)C[C@H]3C2)c(F)cc1F ZINC000880710159 DE On-Demand Mild RBP4 40 33 N#Cc1cc(NC(=O)N2C[C@H]3C[C@H](O)CC[C@H]3C2)c(F)cc1F ZINC000880710160 DE On-Demand Mild RBP4 40 33 N#Cc1cc(NC(=O)N2C[C@H]3C[C@@H](O)CC[C@H]3C2)c(F)cc1F ZINC000880710161 DE On-Demand Mild RBP4 40 33 N#Cc1cc(NC(=O)N2C[C@@H]3CC[C@@H](O)C[C@H]3C2)c(F)cc1F ZINC000880710162 DE On-Demand Mild RBP4 40 33 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880710163 EG On-Demand Mild CACNA1I 53 34 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880710164 EG On-Demand Mild CACNA1I 53 34 N#Cc1cc(NC(=O)N2CCC(OCc3ccc(F)cc3)CC2)c(F)cc1F ZINC000880710175 GI On-Demand Mild LIPG 20 41 N#Cc1cc(NC(=O)NCC2CCN(C3CCOCC3)CC2)c(F)cc1F ZINC000880710214 GF On-Demand Mild CACNA1I 41 32 N#Cc1cc(NC(=O)N(CCN2CCOCC2)CC2CC2)c(F)cc1F ZINC000880710233 FE On-Demand Mild CASR 57 45 N#Cc1cc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880710398 GG On-Demand Mild ACHE 25 43 N#Cc1cc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880710398 GG On-Demand Mild SIGMAR1 24 44 N#Cc1cc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880710398 GG On-Demand Mild CCR3 70 44 N#Cc1cc(NC(=O)NCC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880710398 GG On-Demand Mild CACNA1I 62 41 COC[C@@H](CCNC(=O)Nc1cc(C#N)c(F)cc1F)OC ZINC000880710475 DE On-Demand Mild ADRB1 41 33 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@H](O)c4ccccc4O3)C2)c(F)cc1F ZINC000880710489 GG On-Demand Mild TRPM8 28 42 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@H](O)c4ccccc4O3)C2)c(F)cc1F ZINC000880710491 GG On-Demand Mild TRPM8 28 42 N#Cc1cc(NC(=O)N2CC[C@]3(C[C@@H](O)c4ccccc4O3)C2)c(F)cc1F ZINC000880710492 GG On-Demand Mild TRPM8 28 42 CN(CC1(O)CCCC1)C(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C ZINC000880710494 EH On-Demand Bother NMBR 41 31 N#Cc1cc(NC(=O)N2CC[C@@]3(C[C@@H](O)c4ccccc4O3)C2)c(F)cc1F ZINC000880710526 GG On-Demand Mild TRPM8 28 42 N#Cc1cc(NC(=O)N2CC[C@H](C(=O)NCc3ccccc3)C2)c(F)cc1F ZINC000880710531 GG On-Demand Mild EPHX2 20 42 N#Cc1cc(NC(=O)N2CC[C@@H](C(=O)NCc3ccccc3)C2)c(F)cc1F ZINC000880710532 GG On-Demand Mild EPHX2 20 42 CO[C@@H](C)CNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880710548 CD On-Demand Mild ADRB1 40 39 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild DRD4 24 44 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild HRH2 18 40 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild CHRM3 26 44 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild SIGMAR1 26 47 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild SSTR5 41 35 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild CCR3 67 51 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild MLNR 19 42 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild CXCR3 25 42 N#Cc1cccc(CN2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880710600 GG On-Demand Mild MCHR1 69 50 N#Cc1cc(NC(=O)N2CCC(c3ccon3)CC2)c(F)cc1F ZINC000880710615 EG On-Demand Mild SMO 19 45 N#Cc1cc(NC(=O)N2CCC[C@H](N3CCOCC3)CC2)c(F)cc1F ZINC000880710656 FF On-Demand Mild L3MBTL3 65 39 N#Cc1cc(NC(=O)N2CCC[C@@H](N3CCOCC3)CC2)c(F)cc1F ZINC000880710657 FF On-Demand Mild L3MBTL3 65 39 N#Cc1cc(NC(=O)N2CC[C@@H]3C[C@@H]3C2)c(F)cc1F ZINC000880710677 CF On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N2CC[C@@H]3C[C@H]3C2)c(F)cc1F ZINC000880710679 CF On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N2CC[C@H]3C[C@@H]3C2)c(F)cc1F ZINC000880710681 CF On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N2CC[C@H]3C[C@H]3C2)c(F)cc1F ZINC000880710684 CF On-Demand Mild RBP4 47 35 N#Cc1cc(NC(=O)N[C@H]2CCOC2=O)c(F)cc1F ZINC000880710739 CD On-Demand Mild LUXR 74 42 N#Cc1cc(NC(=O)N[C@H]2CCOC2=O)c(F)cc1F ZINC000880710739 CD On-Demand Mild TRAR 86 39 N#Cc1cc(NC(=O)N[C@H]2CCOC2=O)c(F)cc1F ZINC000880710739 CD On-Demand Mild LASR 61 38 N#Cc1cc(NC(=O)N2CCC(Oc3cccc(F)c3)CC2)c(F)cc1F ZINC000880710835 GI On-Demand Mild EPHX2 21 46 COC[C@H](NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C)C1CC1 ZINC000880710896 EG On-Demand Bother CACNA1D 43 35 COC[C@@H](NC(=O)Nc1cc([N+](=O)[O-])ccc1C(C)(C)C)C1CC1 ZINC000880710897 EG On-Demand Bother CACNA1D 43 35 CCn1nccc1[C@@H]1OCC[C@H]1NC(=O)c1cccc2nsnc12 ZINC000880710918 EE On-Demand Anodyne HTR3A 23 42 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880710941 FF On-Demand Mild EPHX2 44 40 CN(C)CCn1cc(NC(=O)Nc2cc(C#N)c(F)cc2F)cn1 ZINC000880710950 EE On-Demand Mild CSNK2A1 30 40 N#Cc1cc(NC(=O)N2C[C@H]3CCCC[C@H]3C2)c(F)cc1F ZINC000880711016 DG On-Demand Mild RBP4 44 32 CN1CCC[C@@H](CCNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880711047 DF On-Demand Mild CCR3 43 42 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711116 DE On-Demand Mild LGMN 56 33 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711117 DE On-Demand Mild LGMN 56 33 N#Cc1cc(NC(=O)NC2CCN(C3CCC3)CC2)c(F)cc1F ZINC000880711144 EF On-Demand Mild EPHX2 29 42 N#Cc1cc(NC(=O)NCCCCCN2CCCC2)c(F)cc1F ZINC000880711155 EG On-Demand Mild CCR3 35 45 N#Cc1cc(NC(=O)NCCCCCN2CCCC2)c(F)cc1F ZINC000880711155 EG On-Demand Mild CHRNA7 18 49 N#Cc1cc(NC(=O)N2CCC[C@](CO)(Cc3ccccc3)C2)c(F)cc1F ZINC000880711284 GH On-Demand Mild EPHX2 15 42 N#Cc1cc(NC(=O)N2CCC[C@](CO)(Cc3ccccc3)C2)c(F)cc1F ZINC000880711284 GH On-Demand Mild SLC12A5 46 34 N#Cc1cc(NC(=O)N2CCC[C@@](CO)(Cc3ccccc3)C2)c(F)cc1F ZINC000880711285 GH On-Demand Mild EPHX2 15 42 N#Cc1cc(NC(=O)N2CCC[C@@](CO)(Cc3ccccc3)C2)c(F)cc1F ZINC000880711285 GH On-Demand Mild SLC12A5 46 34 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711343 DE On-Demand Mild CHRNA10 54 37 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711343 DE On-Demand Mild ACKR3 52 32 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711344 DE On-Demand Mild CHRNA10 54 37 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880711344 DE On-Demand Mild ACKR3 52 32 CC(=O)N[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880711413 DD On-Demand Mild CSNK2A1 41 38 CC(=O)N[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880711414 DD On-Demand Mild CSNK2A1 41 38 N#Cc1cc(NC(=O)N2CC(C(F)(F)F)C2)c(F)cc1F ZINC000880711447 DF On-Demand Mild RBP4 50 32 N#Cc1cc(NC(=O)N2C[C@@H]3C[C@H](C2)c2cccc(=O)n2C3)c(F)cc1F ZINC000880711520 FF On-Demand Mild CHRNA4 25 46 CN(C)C1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880711535 DF On-Demand Mild EPHX2 18 41 N#Cc1cc(NC(=O)NC2CCC2)c(F)cc1F ZINC000880711587 CF On-Demand Mild EPHX2 24 52 N#Cc1cc(NC(=O)N[C@@H]2CCCN(CCCO)C2)c(F)cc1F ZINC000880711594 ED On-Demand Mild CCR3 32 41 N#Cc1cc(NC(=O)N[C@H]2CCCN(CCCO)C2)c(F)cc1F ZINC000880711595 ED On-Demand Mild CCR3 32 41 N#Cc1cc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3[nH]2)c(F)cc1F ZINC000880711655 GI On-Demand Mild PRCP 45 38 N#Cc1cc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3[nH]2)c(F)cc1F ZINC000880711655 GI On-Demand Mild CPT1A 31 40 N#Cc1cc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3[nH]2)c(F)cc1F ZINC000880711656 GI On-Demand Mild PRCP 45 38 N#Cc1cc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3[nH]2)c(F)cc1F ZINC000880711656 GI On-Demand Mild CPT1A 31 40 N#Cc1cc(NC(=O)N[C@@H]2CC[C@@H](O)CC2)c(F)cc1F ZINC000880711659 CE On-Demand Mild EPHX2 16 44 N#Cc1cc(NC(=O)N2CCC(CO)(c3ccccc3)CC2)c(F)cc1F ZINC000880711776 FG On-Demand Mild RBP4 44 32 CC(C)(C)OC(=O)N1C[C@@H]2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)[C@@H]2C1 ZINC000880711779 GG On-Demand Mild GPR119 26 49 N#Cc1cc(NC(=O)N2CC[C@](O)(Cc3ccc(F)cc3)C2)c(F)cc1F ZINC000880711871 GG On-Demand Mild S1PR2 27 41 N#Cc1cc(NC(=O)N2CC[C@@](O)(Cc3ccc(F)cc3)C2)c(F)cc1F ZINC000880711872 GG On-Demand Mild S1PR2 27 41 N#Cc1cc(NC(=O)N2CC[C@](CO)(c3ccccc3)C2)c(F)cc1F ZINC000880711887 FG On-Demand Mild EPHX2 20 46 N#Cc1cc(NC(=O)N2CC[C@@](CO)(c3ccccc3)C2)c(F)cc1F ZINC000880711888 FG On-Demand Mild EPHX2 20 46 N#Cc1cc(NC(=O)N(CCN2CCOCC2)Cc2ccco2)c(F)cc1F ZINC000880711911 GF On-Demand Mild CASR 59 45 N#Cc1cc(NC(=O)NC[C@@H](O)CN2CCc3ccccc3C2)c(F)cc1F ZINC000880711932 GE On-Demand Mild ADRB1 40 33 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880712001 EH On-Demand Mild PTAFR 37 49 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)nc1 ZINC000880712044 FF On-Demand Mild P2RY12 17 41 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)nc1 ZINC000880712044 FF On-Demand Mild PDGFRB 51 38 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)nc1 ZINC000880712044 FF On-Demand Mild DGAT1 25 49 N#Cc1cc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880712049 GG On-Demand Mild EPHX2 18 46 N#Cc1cc(NC(=O)N2CC[C@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880712049 GG On-Demand Mild TRPM8 20 41 N#Cc1cc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880712050 GG On-Demand Mild EPHX2 18 46 N#Cc1cc(NC(=O)N2CC[C@@]3(CC(=O)c4ccccc4O3)C2)c(F)cc1F ZINC000880712050 GG On-Demand Mild TRPM8 20 41 N#Cc1cc(NC(=O)NC23C[C@H]4C[C@@H](CC(O)(C4)C2)C3)c(F)cc1F ZINC000880712083 EG On-Demand Mild EPHX2 36 45 N#Cc1cc(NC(=O)N2CC(C3CC3)C2)c(F)cc1F ZINC000880712085 CF On-Demand Mild RBP4 44 32 COC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880712142 EE On-Demand Mild EPHX2 46 40 CCCN(CCN1CCCC1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880712177 EG On-Demand Mild CASR 44 38 N#Cc1cc(NC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(F)cc1F ZINC000880712291 GI On-Demand Mild SLC18A3 26 41 N#Cc1cc(NC(=O)N2CCC(C(=O)c3ccc(F)cc3)CC2)c(F)cc1F ZINC000880712291 GI On-Demand Mild WNT3A 47 33 Cc1c(NC(=O)Nc2cc(C#N)c(F)cc2F)cnn1C1CCCC1 ZINC000880712296 EI On-Demand Mild CSNK2A1 41 38 N#Cc1cc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c(F)cc1F ZINC000880712300 FF On-Demand Mild CXCR3 17 44 N#Cc1cc(NC(=O)NC2CCN(CC(F)(F)F)CC2)c(F)cc1F ZINC000880712300 FF On-Demand Mild HPGDS 38 41 N#Cc1cc(NC(=O)NCC[C@H](O)C(F)(F)F)c(F)cc1F ZINC000880712368 DE On-Demand Mild ADRB1 41 34 N#Cc1cc(NC(=O)NCC[C@@H](O)C(F)(F)F)c(F)cc1F ZINC000880712369 DE On-Demand Mild ADRB1 41 34 CNC(=O)OC[C@@H]1CCCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880712462 FF On-Demand Mild LGMN 49 33 COc1cccc([C@H]2C[C@@H](O)CN2C(=O)Nc2cc(C#N)c(F)cc2F)c1 ZINC000880712469 FG On-Demand Mild TAAR1 18 43 COc1cccc([C@H]2C[C@H](O)CN2C(=O)Nc2cc(C#N)c(F)cc2F)c1 ZINC000880712470 FG On-Demand Mild TAAR1 18 43 C[C@@H]1CN(CCCNC(=O)Nc2cc(C#N)c(F)cc2F)CCCO1 ZINC000880712513 FE On-Demand Mild CCR3 35 46 COc1cnccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880712535 FF On-Demand Mild PDGFRB 46 42 COc1cnccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880712535 FF On-Demand Mild RBP4 19 44 N#Cc1cc(NC(=O)N2CCCC[C@H]2c2cc[nH]n2)c(F)cc1F ZINC000880712546 EG On-Demand Mild CPT1A 28 40 N#Cc1cc(NC(=O)N2CCCC[C@@H]2c2cc[nH]n2)c(F)cc1F ZINC000880712547 EG On-Demand Mild CPT1A 28 40 COC[C@@H](O)CNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880712559 CC On-Demand Mild ADRB1 48 39 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c(F)cc1F ZINC000880712591 GI On-Demand Mild CACNA1H 42 35 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3Cl)CC2)c(F)cc1F ZINC000880712591 GI On-Demand Mild NPY5R 21 40 N#Cc1cc(NC(=O)N2CCC[C@@H](c3ncc(C(F)(F)F)[nH]3)C2)c(F)cc1F ZINC000880712651 GH On-Demand Mild RBP4 47 34 N#Cc1cc(NC(=O)N2CCC[C@H](c3ncc(C(F)(F)F)[nH]3)C2)c(F)cc1F ZINC000880712652 GH On-Demand Mild RBP4 47 34 N#Cc1cc(NC(=O)NCC2CCN(C3CC3)CC2)c(F)cc1F ZINC000880712660 EF On-Demand Mild CACNA1I 44 32 COc1ccc([C@@H](CN(C)C)NC(=O)Nc2cc(C#N)c(F)cc2F)cc1 ZINC000880712682 FG On-Demand Mild UTS2 43 39 COc1ccc([C@H](CN(C)C)NC(=O)Nc2cc(C#N)c(F)cc2F)cc1 ZINC000880712683 FG On-Demand Mild UTS2 43 39 Cc1ccncc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880712690 FF On-Demand Mild NPY2R 40 37 N#Cc1cc(NC(=O)NCC2(c3ccccn3)CCC2)c(F)cc1F ZINC000880712708 EG On-Demand Mild NMBR 44 42 N#Cc1cc(NC(=O)NCC2(c3ccccn3)CCC2)c(F)cc1F ZINC000880712708 EG On-Demand Mild GRPR 23 42 N#Cc1cc(NC(=O)Nc2cc(C3CCCC3)[nH]n2)c(F)cc1F ZINC000880712727 EH On-Demand Mild PKNB 40 36 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3F)C[C@@H]2C1 ZINC000880712740 GG On-Demand Mild GPR119 26 55 N#Cc1cc(NC(=O)N2CCC(Oc3ncccc3F)CC2)c(F)cc1F ZINC000880712751 GG On-Demand Mild GPR119 21 42 N#Cc1cc(NC(=O)N2CCC(CNC(=O)C(F)(F)F)CC2)c(F)cc1F ZINC000880712766 GF On-Demand Mild CACNA1I 41 33 N#Cc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880712787 GH On-Demand Mild PRSS2 54 30 N#Cc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880712787 GH On-Demand Mild EPHX2 24 54 N#Cc1cc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)c(F)cc1F ZINC000880712905 GH On-Demand Mild CACNA1H 44 40 N#Cc1cc(NC(=O)N2CCC(NC(=O)C3CC3)CC2)c(F)cc1F ZINC000880712921 EE On-Demand Mild EPHX2 27 42 N#Cc1cc(NC(=O)N2CC[C@H](Cc3ccncc3)C2)c(F)cc1F ZINC000880712953 EG On-Demand Mild CCR3 63 41 N#Cc1cc(NC(=O)N2CC[C@@H](Cc3ccncc3)C2)c(F)cc1F ZINC000880712954 EG On-Demand Mild CCR3 63 41 N#Cc1cc(NC(=O)NCCN2CCCOCC2)c(F)cc1F ZINC000880712969 DD On-Demand Mild EPHX2 18 44 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@H](O)C2)c(F)cc1F ZINC000880713039 GF On-Demand Mild OPRK1 16 40 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@H](O)C2)c(F)cc1F ZINC000880713039 GF On-Demand Mild CCR3 40 40 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@H](O)C2)c(F)cc1F ZINC000880713039 GF On-Demand Mild MCHR1 17 41 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@@H](O)C2)c(F)cc1F ZINC000880713040 GF On-Demand Mild OPRK1 16 40 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@@H](O)C2)c(F)cc1F ZINC000880713040 GF On-Demand Mild CCR3 40 40 N#Cc1cc(NC(=O)NCc2ccccc2CN2CC[C@@H](O)C2)c(F)cc1F ZINC000880713040 GF On-Demand Mild MCHR1 17 41 N#Cc1cc(NC(=O)N2CC[C@H](CN3CCCCC3)C2)c(F)cc1F ZINC000880713139 EG On-Demand Mild CCR3 15 40 N#Cc1cc(NC(=O)N2CC[C@@H](CN3CCCCC3)C2)c(F)cc1F ZINC000880713140 EG On-Demand Mild CCR3 15 40 N#Cc1cc(NC(=O)N2CCC(O)(Cc3ccc(F)cc3)CC2)c(F)cc1F ZINC000880713172 GH On-Demand Mild S1PR2 29 43 N#Cc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)c(F)cc1F ZINC000880713192 GG On-Demand Mild P2RY12 15 41 N#Cc1cc(NC(=O)N2CCCN(c3ncccc3F)CC2)c(F)cc1F ZINC000880713192 GG On-Demand Mild RBP4 15 48 N#Cc1cc(NC(=O)NCC2CCN(CC(F)(F)F)CC2)c(F)cc1F ZINC000880713193 GG On-Demand Mild CACNA1I 65 39 N#Cc1cc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c(F)cc1F ZINC000880713254 FH On-Demand Mild GRIN2B 21 43 N#Cc1cc(NC(=O)N2CC[C@@H](COc3ccccc3)C2)c(F)cc1F ZINC000880713254 FH On-Demand Mild CCR3 34 41 N#Cc1cc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c(F)cc1F ZINC000880713255 FH On-Demand Mild GRIN2B 21 43 N#Cc1cc(NC(=O)N2CC[C@H](COc3ccccc3)C2)c(F)cc1F ZINC000880713255 FH On-Demand Mild CCR3 34 41 N#Cc1cc(NC(=O)NC23CCC(CC2)C3)c(F)cc1F ZINC000880713281 CG On-Demand Mild EPHX2 25 43 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c(F)cc1F ZINC000880713348 FG On-Demand Mild CACNA1H 40 34 N#Cc1cc(NC(=O)N2CCC(O)(c3ccccc3)CC2)c(F)cc1F ZINC000880713348 FG On-Demand Mild CCR1 34 42 N#Cc1cc(NC(=O)NCCOCC(F)F)c(F)cc1F ZINC000880713507 DE On-Demand Mild ADRB1 43 35 CN1CCC(N2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)CC1 ZINC000880713577 GF On-Demand Mild SLC6A5 17 41 COc1cc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)ncn1 ZINC000880713578 FD On-Demand Mild PDGFRB 42 42 COc1cc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)ncn1 ZINC000880713578 FD On-Demand Mild RBP4 15 41 N#Cc1cc(NC(=O)N2CCC(Oc3ccc(F)nc3)CC2)c(F)cc1F ZINC000880713586 GG On-Demand Mild EPHX2 15 41 CC(C)n1ncc2c1C[C@H](NC(=O)Nc1cc(C#N)c(F)cc1F)CC2 ZINC000880713637 FG On-Demand Mild CSNK2A1 40 35 CC(C)n1ncc2c1C[C@@H](NC(=O)Nc1cc(C#N)c(F)cc1F)CC2 ZINC000880713638 FG On-Demand Mild CSNK2A1 40 35 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713647 GG On-Demand Mild CACNA1I 66 37 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713647 GG On-Demand Mild GPR119 40 49 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713648 GG On-Demand Mild CACNA1I 66 37 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713648 GG On-Demand Mild GPR119 40 49 N#Cc1cc(NC(=O)NCc2cccc(N3CCOCC3)n2)c(F)cc1F ZINC000880713722 FE On-Demand Mild PIK3CB 44 36 CN1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713733 CD On-Demand Mild CACNA1I 59 34 CN1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713734 CD On-Demand Mild CACNA1I 59 34 N#Cc1cc(NC(=O)N2CCCC[C@H]2c2nc3ccccc3o2)c(F)cc1F ZINC000880713758 GJ On-Demand Mild CPT1A 48 39 N#Cc1cc(NC(=O)N2CCCC[C@@H]2c2nc3ccccc3o2)c(F)cc1F ZINC000880713759 GJ On-Demand Mild CPT1A 48 39 N#Cc1cc(NC(=O)NCCCNC(=O)C2CCC2)c(F)cc1F ZINC000880713776 EE On-Demand Mild TBK1 48 35 N#Cc1cc(NC(=O)N2CCC(OCc3ccccc3F)CC2)c(F)cc1F ZINC000880713820 GI On-Demand Mild EPHX2 18 42 CO[C@@H](CCNC(=O)Nc1cc(C#N)c(F)cc1F)C(F)(F)F ZINC000880713837 EF On-Demand Mild ADRB1 40 33 CC(C)(C)OC(=O)N1CC(CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713925 FF On-Demand Mild CACNA1I 41 33 CC(C)(C)OC(=O)N1CC(CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880713925 FF On-Demand Mild GPR119 24 49 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713927 GG On-Demand Mild ACE 25 42 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713927 GG On-Demand Mild F10 18 40 N#Cc1cc(NC(=O)N[C@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713927 GG On-Demand Mild MME 17 42 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713928 GG On-Demand Mild ACE 25 42 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713928 GG On-Demand Mild F10 18 40 N#Cc1cc(NC(=O)N[C@@H]2CCCN(Cc3ccccc3)C2=O)c(F)cc1F ZINC000880713928 GG On-Demand Mild MME 17 42 N#Cc1ccccc1NC1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC1 ZINC000880713960 GG On-Demand Mild L3MBTL3 42 33 N#Cc1ccccc1NC1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC1 ZINC000880713961 GG On-Demand Mild L3MBTL3 42 33 N#Cc1cc(NC(=O)N2CCC[C@H]2C(=O)NCc2ccco2)c(F)cc1F ZINC000880713969 FF On-Demand Mild LGMN 72 36 N#Cc1cc(NC(=O)N2CCC[C@@H]2C(=O)NCc2ccco2)c(F)cc1F ZINC000880713970 FF On-Demand Mild LGMN 72 36 COCCC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880713980 FD On-Demand Mild EPHX2 36 42 N#Cc1cc(NC(=O)N2CCN(C3CCCCC3)CC2)c(F)cc1F ZINC000880713994 EG On-Demand Mild L3MBTL3 46 34 N#Cc1cc(NC(=O)N[C@@H](c2ccccc2)[C@@H]2CCOC2)c(F)cc1F ZINC000880714024 FH On-Demand Mild NPY2R 15 40 N#Cc1cc(NC(=O)N[C@H](c2ccccc2)[C@@H]2CCOC2)c(F)cc1F ZINC000880714025 FH On-Demand Mild NPY2R 15 40 N#Cc1cc(NC(=O)N[C@H](c2ccccc2)[C@H]2CCOC2)c(F)cc1F ZINC000880714026 FH On-Demand Mild NPY2R 15 40 N#Cc1cc(NC(=O)N[C@@H](c2ccccc2)[C@H]2CCOC2)c(F)cc1F ZINC000880714027 FH On-Demand Mild NPY2R 15 40 CC[C@@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714043 CE On-Demand Mild ADRB1 43 36 CC[C@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714044 CE On-Demand Mild ADRB1 43 36 C[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)[C@@H]1C ZINC000880714050 CG On-Demand Mild TRPC6 54 40 C[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)[C@@H]1C ZINC000880714050 CG On-Demand Mild TRPC3 37 40 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714053 CG On-Demand Mild TRPC6 54 40 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714053 CG On-Demand Mild TRPC3 37 40 N#Cc1cc(NC(=O)N[C@@H]2CCN(C(=O)C3CCCC3)C2)c(F)cc1F ZINC000880714079 FF On-Demand Mild EPHX2 26 40 N#Cc1cc(NC(=O)N[C@H]2CCN(C(=O)C3CCCC3)C2)c(F)cc1F ZINC000880714080 FF On-Demand Mild EPHX2 26 40 COc1cccc([C@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3F)CCO2)c1 ZINC000880714097 FG On-Demand Mild TAAR1 17 42 N#Cc1cc(NC(=O)NCC2CCN(C(=O)C(F)(F)F)CC2)c(F)cc1F ZINC000880714144 GF On-Demand Mild CACNA1I 49 35 N#Cc1cc(NC(=O)N[C@H]2CCN(C(=O)CCc3ccccc3)C2)c(F)cc1F ZINC000880714159 GG On-Demand Mild C3AR1 42 42 N#Cc1cc(NC(=O)N[C@@H]2CCN(C(=O)CCc3ccccc3)C2)c(F)cc1F ZINC000880714160 GG On-Demand Mild C3AR1 42 42 CC[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714161 FH On-Demand Mild PTGES 21 41 CC[C@@H](O)CN(Cc1ccccc1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714162 FH On-Demand Mild PTGES 21 41 CN(c1ccccc1)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714163 FH On-Demand Mild RBP4 56 38 N#Cc1cc(NC(=O)N2CCC3(CC2)OCc2ccccc23)c(F)cc1F ZINC000880714165 FH On-Demand Mild NPY5R 22 40 N#Cc1ccccc1NC1CCN(C(=O)CCc2cn[nH]c2)CC1 ZINC000880714174 DE On-Demand Mild C3AR1 41 39 N#Cc1ccccc1NC1CCN(C(=O)c2cccn3nccc23)CC1 ZINC000880714201 EF On-Demand Mild CSNK2A1 51 31 N#Cc1cc(NC(=O)N2CCCO[C@@H](c3ccccc3)C2)c(F)cc1F ZINC000880714254 FH On-Demand Mild RBP4 44 31 N#Cc1cc(NC(=O)N2CCCO[C@H](c3ccccc3)C2)c(F)cc1F ZINC000880714255 FH On-Demand Mild RBP4 44 31 N#Cc1ccccc1NC1CCN(C(=O)c2cncc3[nH]ccc23)CC1 ZINC000880714259 EG On-Demand Mild PRKCD 72 38 N#Cc1ccccc1NC1CCN(C(=O)c2cncc3[nH]ccc23)CC1 ZINC000880714259 EG On-Demand Mild PRKCQ 93 38 N#Cc1ccccc1NC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880714289 EG On-Demand Mild CSNK2A1 49 33 N#Cc1ccccc1NC1CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880714289 EG On-Demand Mild MLNR 16 49 Cc1cnc(Cl)c(C(=O)N2CCC(Nc3ccccc3C#N)CC2)c1 ZINC000880714306 FH On-Demand Mild CSNK2A1 51 35 Cc1cnc(Cl)c(C(=O)N2CCC(Nc3ccccc3C#N)CC2)c1 ZINC000880714306 FH On-Demand Mild FASN 41 35 N#Cc1cc(NC(=O)N2CCC[C@H]2C(=O)NC2CC2)c(F)cc1F ZINC000880714352 EE On-Demand Mild LGMN 69 36 N#Cc1cc(NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)c(F)cc1F ZINC000880714353 EE On-Demand Mild LGMN 69 36 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880714375 FG On-Demand Mild CSNK2A1 55 33 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880714376 FG On-Demand Mild CSNK2A1 55 33 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880714377 FG On-Demand Mild CSNK2A1 55 33 N#Cc1cc(NC(=O)N2CCC(Cc3cccnc3)CC2)c(F)cc1F ZINC000880714389 FH On-Demand Mild GRIN2B 43 39 N#Cc1cc(NC(=O)N2CCC(Cc3cccnc3)CC2)c(F)cc1F ZINC000880714389 FH On-Demand Mild CCR3 46 39 N#Cc1cc(NC(=O)N2CCC(Cc3cccnc3)CC2)c(F)cc1F ZINC000880714389 FH On-Demand Mild CHRNA7 49 40 N#Cc1cc(NC(=O)N2CCC(Cc3cccnc3)CC2)c(F)cc1F ZINC000880714389 FH On-Demand Mild C3AR1 43 43 C=CC(C)(C)CC(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880714519 DH On-Demand Mild CCR8 57 36 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880714554 FF On-Demand Mild GPR119 15 45 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714572 DD On-Demand Mild LGMN 75 39 N#Cc1cc(NC(=O)N(CCO)CCN2CCOCC2)c(F)cc1F ZINC000880714578 FC On-Demand Mild CASR 63 49 N#Cc1cc(NC(=O)NCc2ccccc2N2CCOCC2)c(F)cc1F ZINC000880714592 FF On-Demand Mild KCNQ2 43 34 N#Cc1cc(NC(=O)NCc2ccccc2N2CCOCC2)c(F)cc1F ZINC000880714592 FF On-Demand Mild SCN10A 15 48 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880714609 DD On-Demand Mild EPHX2 33 47 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880714610 DD On-Demand Mild EPHX2 33 47 COC[C@@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714612 CD On-Demand Mild ADRB1 46 38 N#Cc1cc(NC(=O)NC2CCN([C@H]3CCC[C@H]3O)CC2)c(F)cc1F ZINC000880714652 FE On-Demand Mild EPHX2 25 40 N#Cc1cc(NC(=O)NC2CCN([C@@H]3CCC[C@H]3O)CC2)c(F)cc1F ZINC000880714653 FE On-Demand Mild EPHX2 25 40 N#Cc1cc(NC(=O)NC2CCN([C@H]3CCC[C@@H]3O)CC2)c(F)cc1F ZINC000880714654 FE On-Demand Mild EPHX2 25 40 N#Cc1cc(NC(=O)NC2CCN([C@@H]3CCC[C@@H]3O)CC2)c(F)cc1F ZINC000880714655 FE On-Demand Mild EPHX2 25 40 N#Cc1cc(NC(=O)NC2CCN([C@@H]3CCCC[C@@H]3O)CC2)c(F)cc1F ZINC000880714658 GF On-Demand Mild EPHX2 27 41 N#Cc1cc(NC(=O)NC2CCN([C@@H]3CCCC[C@H]3O)CC2)c(F)cc1F ZINC000880714659 GF On-Demand Mild EPHX2 27 41 N#Cc1cc(NC(=O)NC2CCN([C@H]3CCCC[C@@H]3O)CC2)c(F)cc1F ZINC000880714660 GF On-Demand Mild EPHX2 27 41 N#Cc1cc(NC(=O)NC2CCN([C@H]3CCCC[C@H]3O)CC2)c(F)cc1F ZINC000880714661 GF On-Demand Mild EPHX2 27 41 Cn1nnc(C(=O)N2CCC(Nc3ccccc3C#N)CC2)n1 ZINC000880714686 DC On-Demand Mild MLNR 16 49 N#Cc1ccccc1NC1CCN(C(=O)c2ccc(CN3CCOCC3)o2)CC1 ZINC000880714700 GF On-Demand Mild MLNR 26 51 Cc1nc(C(C)C)ncc1C(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880714732 FG On-Demand Mild CSNK2A1 57 36 COCC1(O)CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714748 ED On-Demand Mild S1PR2 27 41 N#Cc1cc(NC(=O)N2CCC(c3ccccn3)CC2)c(F)cc1F ZINC000880714761 EH On-Demand Mild RBP4 50 37 N#Cc1cc(NC(=O)N2CCC(c3ccccn3)CC2)c(F)cc1F ZINC000880714761 EH On-Demand Mild SMO 20 44 N#Cc1ccccc1NC1CCN(C(=O)COC2CC2)CC1 ZINC000880714807 CE On-Demand Mild CCR8 41 33 CS(=O)(=O)C1CCC(C(=O)N2CCC(Nc3ccccc3C#N)CC2)CC1 ZINC000880714810 GF On-Demand Mild CSNK2A1 41 32 CS(=O)(=O)C1CCC(C(=O)N2CCC(Nc3ccccc3C#N)CC2)CC1 ZINC000880714810 GF On-Demand Mild CCR8 50 39 CS(=O)(=O)C1CCC(C(=O)N2CCC(Nc3ccccc3C#N)CC2)CC1 ZINC000880714810 GF On-Demand Mild SFRP1 55 31 CS(=O)(=O)C1CCC(C(=O)N2CCC(Nc3ccccc3C#N)CC2)CC1 ZINC000880714810 GF On-Demand Mild WNT3 49 30 CN1CCC(CNC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714825 DE On-Demand Mild CACNA1I 60 37 CN(C[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1)C(=O)OC(C)(C)C ZINC000880714841 GH On-Demand Mild GPR119 17 43 N#Cc1cc(NC(=O)N2CC[C@@H](N3CCCC3)C2)c(F)cc1F ZINC000880714842 DF On-Demand Mild L3MBTL3 89 44 N#Cc1cc(NC(=O)N2CC[C@H](N3CCCC3)C2)c(F)cc1F ZINC000880714843 DF On-Demand Mild L3MBTL3 89 44 N#Cc1cc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c(F)cc1F ZINC000880714855 GG On-Demand Mild KCNQ2 64 36 N#Cc1cc(NC(=O)N2CCCN(c3ccccc3C#N)CC2)c(F)cc1F ZINC000880714855 GG On-Demand Mild RBP4 19 42 N#Cc1cc(NC(=O)N2CCC(NC(=O)C3CCCCC3)CC2)c(F)cc1F ZINC000880714856 GH On-Demand Mild EPHX2 25 45 CN(CCN1CCOCC1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714873 DD On-Demand Mild CASR 53 42 COc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)n1 ZINC000880714885 FD On-Demand Mild FAAH 22 41 N#CCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714898 DD On-Demand Mild CXCR3 18 41 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild DRD4 21 44 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild SIGMAR1 23 44 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild SSTR5 50 39 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild CCR3 51 41 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild CXCR3 29 45 N#Cc1cc(NC(=O)NC2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880714909 FG On-Demand Mild MCHR1 48 43 CCCCN(CCOC)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714931 DG On-Demand Mild SOAT1 22 40 N#Cc1cc(NC(=O)NCC(=O)N2CCCCC2)c(F)cc1F ZINC000880714934 DD On-Demand Mild PRMT3 17 42 N#Cc1cc(NC(=O)N2CCC[C@@H](N3CCCC3)C2)c(F)cc1F ZINC000880714938 EF On-Demand Mild L3MBTL3 65 39 N#Cc1cc(NC(=O)N2CCC[C@H](N3CCCC3)C2)c(F)cc1F ZINC000880714939 EF On-Demand Mild L3MBTL3 65 39 N#Cc1cc(NC(=O)N2CCC(Oc3ccc(F)cc3F)CC2)c(F)cc1F ZINC000880714957 GI On-Demand Mild SCD1 28 47 CC(C)CN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714960 EG On-Demand Mild CXCR3 20 41 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714966 GH On-Demand Mild CACNA1I 54 34 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880714966 GH On-Demand Mild GPR119 23 45 COCCCCN(Cc1ccccc1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880714974 FI On-Demand Mild SOAT1 25 44 COc1ccc(N2CCCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880714981 GH On-Demand Mild RBP4 17 40 N#Cc1cc(NC(=O)N2CCC(OCc3ccccc3)CC2)c(F)cc1F ZINC000880714986 FI On-Demand Mild GRIN2B 24 43 N#Cc1cc(NC(=O)N2CCC(OCc3ccccc3)CC2)c(F)cc1F ZINC000880714986 FI On-Demand Mild EPHX2 18 41 N#Cc1cc(NC(=O)N2CCC(OCc3ccccc3)CC2)c(F)cc1F ZINC000880714986 FI On-Demand Mild RBP4 44 38 N#Cc1cc(NC(=O)NC[C@@H](O)COCC2CC2)c(F)cc1F ZINC000880714988 ED On-Demand Mild ADRB1 44 36 N#Cc1cc(NC(=O)NC[C@H](O)COCC2CC2)c(F)cc1F ZINC000880714989 ED On-Demand Mild ADRB1 44 36 CN1CCC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715025 DE On-Demand Mild CCR3 43 40 CN1CCC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715025 DE On-Demand Mild CACNA1I 44 32 COC(=O)C1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715031 EF On-Demand Mild EPHX2 23 40 N#Cc1cc(NC(=O)NCCOC2CCCCC2)c(F)cc1F ZINC000880715044 DG On-Demand Mild ADRB1 15 42 N#Cc1cc(NC(=O)NCCCN2CCOC2=O)c(F)cc1F ZINC000880715045 DD On-Demand Mild CCR3 20 40 Cc1noc(C2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)n1 ZINC000880715053 EF On-Demand Mild SMO 40 50 Cc1noc(C2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)n1 ZINC000880715053 EF On-Demand Mild ETHR 57 37 N#Cc1cc(NC(=O)NCc2cccc(CN3CCOCC3)c2)c(F)cc1F ZINC000880715064 GF On-Demand Mild CHRM3 18 43 N#Cc1cc(NC(=O)N2CCC(N3CCCCC3)CC2)c(F)cc1F ZINC000880715065 EG On-Demand Mild L3MBTL3 94 44 N#Cc1cc(NC(=O)Nc2cnn(C[C@H]3CCCO3)c2)c(F)cc1F ZINC000880715075 EF On-Demand Mild PANC 42 34 N#Cc1cc(NC(=O)Nc2cnn(C[C@@H]3CCCO3)c2)c(F)cc1F ZINC000880715076 EF On-Demand Mild PANC 42 34 N#Cc1cc(NC(=O)N2CCCC[C@H](N3CCCC3)C2)c(F)cc1F ZINC000880715077 EG On-Demand Mild L3MBTL3 68 39 N#Cc1cc(NC(=O)N2CCCC[C@@H](N3CCCC3)C2)c(F)cc1F ZINC000880715078 EG On-Demand Mild L3MBTL3 68 39 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715083 EI On-Demand Mild TRPM8 19 50 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715084 EI On-Demand Mild TRPM8 19 50 COc1ccc(N2CCC(NC(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880715094 GH On-Demand Mild EPHX2 44 37 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c(F)cc1F ZINC000880715096 FF On-Demand Mild CSF1R 17 42 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)cc2)c(F)cc1F ZINC000880715096 FF On-Demand Mild STAT6 45 33 COCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715101 EE On-Demand Mild CCR3 37 42 COCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715101 EE On-Demand Mild CXCR3 19 40 C=C(C)CN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715102 EF On-Demand Mild CXCR3 18 41 N#Cc1cc(NC(=O)NC2CCN(CCO)CC2)c(F)cc1F ZINC000880715119 DD On-Demand Mild SLC6A5 16 40 N#Cc1cc(NC(=O)NC2CCN(CCO)CC2)c(F)cc1F ZINC000880715119 DD On-Demand Mild CXCR3 18 41 N#Cc1cc(NC(=O)N2CC[C@@H](N3CCCCC3)C2)c(F)cc1F ZINC000880715120 EF On-Demand Mild L3MBTL3 88 43 N#Cc1cc(NC(=O)N2CC[C@H](N3CCCCC3)C2)c(F)cc1F ZINC000880715121 EF On-Demand Mild L3MBTL3 88 43 CCN1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715142 DE On-Demand Mild CCR3 50 39 CCN1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715142 DE On-Demand Mild CACNA1I 62 35 N#Cc1cc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)c(F)cc1F ZINC000880715147 DE On-Demand Mild CCR3 41 40 N#Cc1cc(NC(=O)N[C@H]2CCN(CC3CC3)C2)c(F)cc1F ZINC000880715148 DE On-Demand Mild CCR3 41 40 N#Cc1cc(NC(=O)NC2CCN(CC3CC3)CC2)c(F)cc1F ZINC000880715157 EF On-Demand Mild CXCR3 20 48 N#Cc1cc(NC(=O)NC2CCN(C(=O)CC(F)(F)F)CC2)c(F)cc1F ZINC000880715165 GF On-Demand Mild EPHX2 41 55 N#Cc1ccccc1NC1CCN(C(=O)c2ccc(Cl)c([N+](=O)[O-])c2)CC1 ZINC000880715173 GH On-Demand Mild L3MBTL3 43 44 N#Cc1cccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880715174 GH On-Demand Mild CCR3 24 41 N#Cc1cccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)c1 ZINC000880715174 GH On-Demand Mild EPHX2 20 56 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715178 GG On-Demand Mild EPHX2 37 45 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715207 GG On-Demand Mild ASAH1 59 36 COc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880715213 GH On-Demand Mild PRSS2 77 33 COc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880715213 GH On-Demand Mild EPHX2 25 47 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild DRD4 15 54 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild SIGMAR1 16 43 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild SSTR5 43 35 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild CCR3 38 41 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild EPHX2 25 42 N#Cc1cc(NC(=O)NC2CCN(Cc3ccccn3)CC2)c(F)cc1F ZINC000880715220 FG On-Demand Mild CXCR3 22 41 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715223 GG On-Demand Mild BMP1 41 38 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715226 GG On-Demand Mild HTR1A 50 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715226 GG On-Demand Mild DRD2 41 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715226 GG On-Demand Mild ADRA1D 40 36 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715226 GG On-Demand Mild DRD3 48 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715226 GG On-Demand Mild CCR3 45 36 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715227 GG On-Demand Mild HTR1A 50 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715227 GG On-Demand Mild DRD2 41 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715227 GG On-Demand Mild ADRA1D 40 36 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715227 GG On-Demand Mild DRD3 48 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715227 GG On-Demand Mild CCR3 45 36 N#Cc1cc(NC(=O)N2CCC(c3ccccc3)CC2)c(F)cc1F ZINC000880715231 EI On-Demand Mild CCR1 29 41 N#Cc1cc(NC(=O)N2CCC(c3ccccc3)CC2)c(F)cc1F ZINC000880715231 EI On-Demand Mild SLC18A3 42 38 N#Cc1cc(NC(=O)N2CCC(c3ccccc3)CC2)c(F)cc1F ZINC000880715231 EI On-Demand Mild RBP4 54 42 N#Cc1cc(NC(=O)N2CCC(c3ccccc3)CC2)c(F)cc1F ZINC000880715231 EI On-Demand Mild SMO 31 42 N#Cc1cc(NC(=O)NC2CCSCC2)c(F)cc1F ZINC000880715241 CF On-Demand Mild EPHX2 15 44 N#Cc1cc(NC(=O)NCCN2CCSCC2)c(F)cc1F ZINC000880715255 EE On-Demand Mild CCR3 18 40 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715258 GG On-Demand Mild EPHX2 48 36 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715258 GG On-Demand Mild GPR119 43 54 N#Cc1cc(NC(=O)N2CCC(C(N)=O)(c3ccccc3)CC2)c(F)cc1F ZINC000880715288 GF On-Demand Mild RBP4 43 31 N#Cc1cc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c(F)cc1F ZINC000880715305 GG On-Demand Mild FAAH 24 44 N#Cc1cc(NC(=O)N2CCN(Cc3ccc(Cl)nc3)CC2)c(F)cc1F ZINC000880715305 GG On-Demand Mild NACHRBETA2 40 35 N#Cc1cc(NC(=O)NCCN2CCCCC2)c(F)cc1F ZINC000880715325 DE On-Demand Mild CCR3 24 41 N#Cc1cc(NC(=O)NCCN2CCCCC2)c(F)cc1F ZINC000880715325 DE On-Demand Mild CHRNA7 15 43 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild HTR1A 64 42 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild DRD2 55 52 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild DRD4 35 42 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild ADRA1D 66 52 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild HTR2A 15 40 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild ADRA1A 57 52 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild ADRA1B 52 52 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild DRD3 59 40 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild HTR7 43 38 COc1ccccc1N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715328 GH On-Demand Mild NPY2R 40 34 CC[C@H](O)CCCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715360 CF On-Demand Mild ADRB1 42 35 CC[C@@H](O)CCCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715361 CF On-Demand Mild ADRB1 42 35 N#Cc1cc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c(F)cc1F ZINC000880715368 GF On-Demand Mild NPFFR2 40 40 N#Cc1cc(NC(=O)NC[C@@]2(O)CCN(Cc3ccccc3)C2)c(F)cc1F ZINC000880715368 GF On-Demand Mild NPFFR1 50 40 N#Cc1cc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c(F)cc1F ZINC000880715369 GF On-Demand Mild NPFFR2 40 40 N#Cc1cc(NC(=O)NC[C@]2(O)CCN(Cc3ccccc3)C2)c(F)cc1F ZINC000880715369 GF On-Demand Mild NPFFR1 50 40 N#Cc1cc(NC(=O)N2CCN(C3CCC3)CC2)c(F)cc1F ZINC000880715391 DF On-Demand Mild HRH3 21 41 N#Cc1cc(NC(=O)N2CCN(C3CCC3)CC2)c(F)cc1F ZINC000880715391 DF On-Demand Mild L3MBTL3 48 33 N#Cc1cc(NC(=O)NCCCCn2ccnc2)c(F)cc1F ZINC000880715430 DF On-Demand Mild TBXAS1 34 47 N#Cc1cc(NC(=O)NCCCCn2ccnc2)c(F)cc1F ZINC000880715430 DF On-Demand Mild QPCT 33 48 N#Cc1cc(NC(=O)NC[C@H]2CCN(CC(F)(F)F)C2)c(F)cc1F ZINC000880715459 FF On-Demand Mild CACNA1I 60 36 N#Cc1cc(NC(=O)NC[C@@H]2CCN(CC(F)(F)F)C2)c(F)cc1F ZINC000880715460 FF On-Demand Mild CACNA1I 60 36 N#Cc1cc(NC(=O)NC2CCN(CC(F)F)CC2)c(F)cc1F ZINC000880715468 EF On-Demand Mild CXCR3 18 41 N#Cc1cc(NC(=O)N2CCCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715476 GG On-Demand Mild NPY2R 24 41 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild ACE 36 45 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild MME 49 45 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild MC4R 95 41 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild TRY2_BOVIN 73 38 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild PAPA1_CARPA 41 42 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild CTSL 39 42 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild F2R 44 33 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild CYP51A1 23 40 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild MC3R 40 35 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild MC5R 53 37 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild CCKBR 20 40 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild CTSS 29 42 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild ACE2 51 34 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild ST14 62 35 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild CTRB_BOVIN 45 32 N#Cc1cc(NC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715514 GG On-Demand Mild BLA1_STEMA 50 32 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild ACE 36 45 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild MME 49 45 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild MC4R 95 41 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild TRY2_BOVIN 73 38 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild PAPA1_CARPA 41 42 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild CTSL 39 42 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild F2R 44 33 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild CYP51A1 23 40 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild MC3R 40 35 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild MC5R 53 37 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild CCKBR 20 40 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild CTSS 29 42 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild ACE2 51 34 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild ST14 62 35 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild CTRB_BOVIN 45 32 N#Cc1cc(NC(=O)N[C@H](Cc2ccccc2)C(=O)N2CCCC2)c(F)cc1F ZINC000880715516 GG On-Demand Mild BLA1_STEMA 50 32 N#Cc1ccc(CN2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880715560 GG On-Demand Mild MLNR 31 40 N#Cc1ccc(CN2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)cc1 ZINC000880715560 GG On-Demand Mild FAAH 19 46 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880715566 GH On-Demand Mild GPR119 42 54 N#Cc1cc(NC(=O)N2CC[C@H](COCc3ccccc3)C2)c(F)cc1F ZINC000880715589 FH On-Demand Mild RBP4 41 33 N#Cc1cc(NC(=O)N2CC[C@@H](COCc3ccccc3)C2)c(F)cc1F ZINC000880715590 FH On-Demand Mild RBP4 41 33 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715593 GG On-Demand Mild F13A1 16 43 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715593 GG On-Demand Mild GPR119 31 57 N#Cc1cc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715603 GG On-Demand Mild EPHX2 45 48 N#Cc1cc(NC(=O)NC2CCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715603 GG On-Demand Mild L3MBTL3 43 34 CC(=O)NCC1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715621 EE On-Demand Mild CACNA1I 45 32 N#Cc1cc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c(F)cc1F ZINC000880715635 GH On-Demand Mild CCR3 32 44 N#Cc1cc(NC(=O)N2CCC(NC(=O)Nc3ccccc3)CC2)c(F)cc1F ZINC000880715635 GH On-Demand Mild EPHX2 54 44 N#Cc1cc(NC(=O)N2CCN(c3cccnn3)CC2)c(F)cc1F ZINC000880715660 ED On-Demand Mild FAAH 23 42 N#Cc1cc(NC(=O)NC2CCN(c3ccccc3)CC2)c(F)cc1F ZINC000880715672 FH On-Demand Mild EPHX2 35 47 CCCCNC(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715687 FF On-Demand Mild ASAH1 48 34 CCOC(=O)N1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715691 FF On-Demand Mild P2RY12 28 41 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715716 GG On-Demand Mild CACNA1I 58 35 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715716 GG On-Demand Mild GPR119 19 43 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715717 GG On-Demand Mild CACNA1I 58 35 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715717 GG On-Demand Mild GPR119 19 43 N#Cc1cc(NC(=O)N2CCC(C(=O)NC3CCCCC3)CC2)c(F)cc1F ZINC000880715722 GH On-Demand Mild EPHX2 26 50 N#Cc1cc(NC(=O)N2CCN3CCCC[C@@H]3C2)c(F)cc1F ZINC000880715732 DF On-Demand Mild L3MBTL3 65 38 N#Cc1cc(NC(=O)N2CCN3CCCC[C@H]3C2)c(F)cc1F ZINC000880715733 DF On-Demand Mild L3MBTL3 65 38 N#Cc1cc(NC(=O)NCCCN2CCCCC2=O)c(F)cc1F ZINC000880715736 EE On-Demand Mild CCR3 29 42 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715739 FI On-Demand Mild ACKR3 50 31 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715740 FI On-Demand Mild ACKR3 50 31 N#Cc1cc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c(F)cc1F ZINC000880715743 GI On-Demand Mild HTR1F 43 35 N#Cc1cc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c(F)cc1F ZINC000880715743 GI On-Demand Mild PIM1 40 31 N#Cc1cc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c(F)cc1F ZINC000880715743 GI On-Demand Mild CCR2 20 50 N#Cc1cc(NC(=O)N2CCC(c3c[nH]c4ncccc34)CC2)c(F)cc1F ZINC000880715743 GI On-Demand Mild CALCRL 40 38 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715773 FH On-Demand Mild RBP4 60 48 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715774 FH On-Demand Mild RBP4 60 48 CCCCCN(CCO)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880715779 DF On-Demand Mild SOAT1 27 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1OC ZINC000880715792 GJ On-Demand Anodyne NR3C1 18 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1OC ZINC000880715792 GJ On-Demand Anodyne NR3C2 26 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1OC ZINC000880715792 GJ On-Demand Anodyne MT-ND1 25 52 N#Cc1cc(NC(=O)NC2CC2)c(F)cc1F ZINC000880715808 BE On-Demand Mild EPHX2 32 48 N#Cc1cc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c(F)cc1F ZINC000880715822 GH On-Demand Mild NPY2R 15 40 N#Cc1cc(NC(=O)N2CCC(C(=O)Nc3ccccc3)CC2)c(F)cc1F ZINC000880715822 GH On-Demand Mild EPHX2 21 40 N#Cc1ccccc1NC1CCN(C(=O)c2cnc(Cl)cn2)CC1 ZINC000880715837 EF On-Demand Mild CSNK2A1 44 33 N#Cc1cc(NC(=O)NCCCN2CCOCC2)c(F)cc1F ZINC000880715872 DD On-Demand Mild CCR3 33 46 N#Cc1cc(NC(=O)NCCCN2CCOCC2)c(F)cc1F ZINC000880715872 DD On-Demand Mild EPHX2 24 43 CCCN(CCC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880715883 DJ On-Demand Anodyne SOAT1 27 47 Cc1nc(NC2CC2)sc1C(=O)N1CCC(Nc2ccccc2C#N)CC1 ZINC000880715884 GH On-Demand Mild CSNK2A1 46 34 CCOC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715913 EE On-Demand Mild P2RY12 40 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)O1 ZINC000880715914 DH On-Demand Anodyne RBP4 57 43 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)O1 ZINC000880715915 DH On-Demand Anodyne RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)O1 ZINC000880715916 DH On-Demand Anodyne RBP4 57 43 N#Cc1cc(NC(=O)N2CC[C@H](CN3CCCC3)C2)c(F)cc1F ZINC000880715922 EF On-Demand Mild CCR3 17 41 N#Cc1cc(NC(=O)N2CC[C@@H](CN3CCCC3)C2)c(F)cc1F ZINC000880715924 EF On-Demand Mild CCR3 17 41 N#Cc1cc(NC(=O)NC2CCN(C3CCCC3)CC2)c(F)cc1F ZINC000880715925 EG On-Demand Mild EPHX2 28 43 N#Cc1cc(NC(=O)NC2CCN(C(=O)C3CC3)CC2)c(F)cc1F ZINC000880715932 EE On-Demand Mild EPHX2 42 50 CCOC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715934 FF On-Demand Mild P2RY12 17 40 CCOC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715934 FF On-Demand Mild EPHX2 46 40 CCOC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880715936 FH On-Demand Anodyne RBP4 42 37 CCOC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880715936 FH On-Demand Anodyne CCR8 19 41 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715950 GG On-Demand Mild CACNA1I 41 32 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2F)C1 ZINC000880715951 GG On-Demand Mild CACNA1I 41 32 CC(=O)N(Cc1ccc(NC(=O)Nc2cc(C#N)c(F)cc2F)cc1)C1CC1 ZINC000880715952 GH On-Demand Mild CSNK2A1 44 33 CNc1nc(C(=O)N2CCC(Nc3ccccc3C#N)CC2)cs1 ZINC000880715959 EF On-Demand Mild CCR8 57 34 CNc1nc(C(=O)N2CCC(Nc3ccccc3C#N)CC2)cs1 ZINC000880715959 EF On-Demand Mild TRPC6 66 45 CNc1nc(C(=O)N2CCC(Nc3ccccc3C#N)CC2)cs1 ZINC000880715959 EF On-Demand Mild TRPC3 59 45 N#Cc1cc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c(F)cc1F ZINC000880715972 GE On-Demand Mild CSNK2A1 16 41 N#Cc1cc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c(F)cc1F ZINC000880715972 GE On-Demand Mild MAP2K1 21 43 N#Cc1cc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)c(F)cc1F ZINC000880715972 GE On-Demand Mild EPHX2 22 44 N#Cc1cc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715980 GH On-Demand Mild GRIN2B 44 37 N#Cc1cc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715980 GH On-Demand Mild CCR3 45 39 N#Cc1cc(NC(=O)NCC2CCN(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880715980 GH On-Demand Mild EPHX2 15 51 CCCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715981 EG On-Demand Mild HTR4 33 40 CCCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715981 EG On-Demand Mild CCR3 39 40 CCCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715981 EG On-Demand Mild EPHX2 29 40 CCCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880715981 EG On-Demand Mild CXCR3 18 41 CNc1ncc(C(=O)N2CCC(Nc3ccccc3C#N)CC2)s1 ZINC000880715995 EF On-Demand Mild CSNK2A1 42 33 N#Cc1cc(NC(=O)N2CCC(Nc3cccnn3)CC2)c(F)cc1F ZINC000880716019 FF On-Demand Mild FAAH 22 41 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild PGR 17 42 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild DRD2 18 42 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild DRD4 48 40 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild ACHE 42 43 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild SIGMAR1 48 49 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild CCR3 51 48 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild CCR5 21 46 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild MCHR1 51 42 CN(C(=O)Nc1cc(C#N)c(F)cc1F)C1CCN(Cc2ccccc2)CC1 ZINC000880716027 GH On-Demand Mild CACNA1G 33 41 N#Cc1cc(NC(=O)NCCCCN2CCC[C@@H]2CO)c(F)cc1F ZINC000880716031 FE On-Demand Mild CCR3 36 41 N#Cc1cc(NC(=O)NCCCCN2CCC[C@H]2CO)c(F)cc1F ZINC000880716032 FE On-Demand Mild CCR3 36 41 CCCCN(CCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716069 DH On-Demand Anodyne SOAT1 30 41 N#Cc1cc(NC(=O)NC2CCC(C(F)(F)F)CC2)c(F)cc1F ZINC000880716070 EI On-Demand Mild EPHX2 30 42 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880716071 FH On-Demand Anodyne SLC6A1 41 37 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880716071 FH On-Demand Anodyne FDFT1 17 40 N#Cc1cc(NC(=O)N2CCN(Cc3cccnc3)CC2)c(F)cc1F ZINC000880716084 FF On-Demand Mild PTAFR 17 45 N#Cc1cc(NC(=O)N2CCN(Cc3cccnc3)CC2)c(F)cc1F ZINC000880716084 FF On-Demand Mild FAAH 34 49 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716085 FH On-Demand Anodyne NR3C1 16 40 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716085 FH On-Demand Anodyne SOAT1 27 40 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716085 FH On-Demand Anodyne KCNK3 41 35 N#Cc1cc(NC(=O)NCCCN2CCCCCC2=O)c(F)cc1F ZINC000880716096 FF On-Demand Mild CCR3 28 41 N#Cc1cc(NC(=O)NC2CCCC2)c(F)cc1F ZINC000880716111 CF On-Demand Mild EPHX2 22 53 CCN(Cc1ccncc1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716112 EI On-Demand Anodyne SOAT1 17 46 N#Cc1cc(NC(=O)NCCN2CCOCC2)c(F)cc1F ZINC000880716120 DD On-Demand Mild CCR3 17 40 N#Cc1cc(NC(=O)NCCN2CCOCC2)c(F)cc1F ZINC000880716120 DD On-Demand Mild EPHX2 22 47 N#Cc1cc(NC(=O)N2CCC[C@@H](c3nc4ccccc4o3)C2)c(F)cc1F ZINC000880716121 GI On-Demand Mild SMO 19 41 N#Cc1cc(NC(=O)N2CCC[C@H](c3nc4ccccc4o3)C2)c(F)cc1F ZINC000880716122 GI On-Demand Mild SMO 19 41 CN(Cc1cnn(C)c1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716123 EG On-Demand Anodyne PLA2G7 49 38 CN(C)C(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716161 FG On-Demand Anodyne RBP4 42 39 COCC(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716170 FF On-Demand Anodyne RBP4 46 40 COCC(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716170 FF On-Demand Anodyne SFRP1 54 33 COCC(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716170 FF On-Demand Anodyne WNT3 43 32 N#CCCN(CCN1CCOCC1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716237 FD On-Demand Mild CASR 62 48 COc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716254 EH On-Demand Anodyne PPIA 15 41 COc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716254 EH On-Demand Anodyne TRPV1 52 38 COc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716254 EH On-Demand Anodyne P2RX7 30 43 COc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716254 EH On-Demand Anodyne P2RY1 55 48 N#Cc1cc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880716259 FH On-Demand Mild SLC18A3 30 41 N#Cc1cc(NC(=O)N2CCC(C(=O)c3ccccc3)CC2)c(F)cc1F ZINC000880716259 FH On-Demand Mild RBP4 40 38 CCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716288 GI On-Demand Anodyne RBP4 40 38 CCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716288 GI On-Demand Anodyne CACNA1G 38 41 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716290 EF On-Demand Anodyne CTSS 17 40 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716290 EF On-Demand Anodyne EPHX2 15 40 CN(Cc1ccsc1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716296 EJ On-Demand Anodyne HSD17B2 21 43 N#Cc1cc(NC(=O)N2CCC([C@@H](O)c3ccccc3)CC2)c(F)cc1F ZINC000880716304 FH On-Demand Mild NPY2R 44 35 N#Cc1cc(NC(=O)N2CCC([C@H](O)c3ccccc3)CC2)c(F)cc1F ZINC000880716306 FH On-Demand Mild NPY2R 44 35 CCCCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716313 CF On-Demand Mild ASAH1 59 34 CC(C)(C)C(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716321 FH On-Demand Anodyne RBP4 47 40 COc1cc2c(cc1OC)CN(C(=O)Nc1cc(C#N)c(F)cc1F)CC2 ZINC000880716327 FG On-Demand Mild ABCB1 15 40 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716331 FE On-Demand Anodyne DRD4 15 49 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716331 FE On-Demand Anodyne CCR3 52 41 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716331 FE On-Demand Anodyne EPHX2 47 40 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716331 FE On-Demand Anodyne CXCR3 22 42 CNC(=O)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716331 FE On-Demand Anodyne MCHR1 19 42 CCOC(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716340 FG On-Demand Anodyne P2RY12 54 38 CN(C)C(=O)c1cccc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716342 GH On-Demand Anodyne ROCK2 21 40 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild HTR1A 86 54 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild DRD2 65 45 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild DRD1 20 45 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild DRD4 38 43 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild ADRA1D 76 42 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild HTR1D 18 54 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild HTR1B 20 54 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild HTR2A 20 45 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild ADRA1A 69 42 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild ADRA1B 61 42 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild DRD3 69 43 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild PDGFRB 45 42 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild HTR7 53 47 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild NPY2R 54 39 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild SSTR1 34 42 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild RBP4 30 54 COc1ccccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716344 FG On-Demand Mild WDR5 31 41 CCCCCNC(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716350 CG On-Demand Mild ASAH1 82 36 CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716354 DF On-Demand Anodyne HRH4 18 41 CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716354 DF On-Demand Anodyne RBP4 54 41 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne DRD4 54 41 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne KCNJ11 15 44 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne CTSL 28 42 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne CCR3 19 41 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne RAF1 26 42 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne CTSS 21 48 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne TAAR1 39 45 COc1cccc(C(=O)NCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880716357 GG On-Demand Anodyne KCNK3 39 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716358 GF On-Demand Anodyne EPHX2 22 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716358 GF On-Demand Anodyne RBP4 42 37 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716358 GF On-Demand Anodyne CCR8 96 43 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716358 GF On-Demand Anodyne SFRP1 124 38 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716358 GF On-Demand Anodyne WNT3 86 38 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)c1 ZINC000880716389 JK On-Demand Anodyne NR1H4 15 44 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)c1 ZINC000880716389 JK On-Demand Anodyne KCNK3 62 40 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)c1 ZINC000880716389 JK On-Demand Anodyne KCNK9 45 39 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716413 GH On-Demand Mild PGR 17 45 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716413 GH On-Demand Mild GCGR 18 42 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716413 GH On-Demand Mild MCHR1 28 41 CCC1(O)CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716460 DF On-Demand Mild S1PR2 28 42 C[C@@H]1[C@@H](C(=O)N2CCC(Nc3ccccc3C#N)CC2)CCN1C ZINC000880716465 EE On-Demand Mild CSNK2A1 43 32 C[C@@H]1[C@@H](C(=O)N2CCC(Nc3ccccc3C#N)CC2)CCN1C ZINC000880716465 EE On-Demand Mild CCR8 41 32 C[C@H]1[C@H](C(=O)N2CCC(Nc3ccccc3C#N)CC2)CCN1C ZINC000880716466 EE On-Demand Mild CSNK2A1 43 32 C[C@H]1[C@H](C(=O)N2CCC(Nc3ccccc3C#N)CC2)CCN1C ZINC000880716466 EE On-Demand Mild CCR8 41 32 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716483 GI On-Demand Anodyne EPHX2 58 45 CCCCN(CC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716495 DJ On-Demand Anodyne SOAT1 30 40 N#Cc1cc(NC(=O)NCCN2CCCCCC2)c(F)cc1F ZINC000880716496 DF On-Demand Mild CCR3 24 41 N#Cc1cc(NC(=O)NCCN2CCCCCC2)c(F)cc1F ZINC000880716496 DF On-Demand Mild CHRNA7 15 43 CC(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716498 EF On-Demand Anodyne RBP4 55 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716499 FF On-Demand Mild F13A1 16 42 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716499 FF On-Demand Mild GPR119 36 60 COCCOc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716506 GH On-Demand Anodyne TRPV1 41 38 COCCOc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716506 GH On-Demand Anodyne P2RX7 27 40 COCCOc1ncccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716506 GH On-Demand Anodyne P2RY1 47 46 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)CC2 ZINC000880716514 GJ On-Demand Anodyne ABCB1 20 42 N#Cc1cc(NC(=O)NCc2ccc(N3CCOCC3)nc2)c(F)cc1F ZINC000880716516 FE On-Demand Mild NAMPT 16 42 COCCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716520 CG On-Demand Anodyne CCR3 18 40 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716529 GG On-Demand Mild CSF1R 19 42 CNC(=O)CN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716535 FD On-Demand Mild CXCR3 19 41 CCCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716543 CH On-Demand Anodyne ASAH1 55 32 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716547 FH On-Demand Anodyne TRPV1 20 42 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716548 FH On-Demand Anodyne TRPV1 20 42 CCCN(CC1CC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716566 DJ On-Demand Anodyne SOAT1 17 44 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild PGR 15 40 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild DRD4 35 41 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild ACHE 42 45 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild SIGMAR1 40 42 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild CCR3 70 40 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cc(C#N)c(F)cc1F ZINC000880716571 GH On-Demand Mild MLNR 52 38 CCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2F)CC1 ZINC000880716576 DE On-Demand Mild CXCR3 20 43 N#Cc1cc(NC(=O)N2CCC[C@H]2[C@H](C#N)c2ccccc2)c(F)cc1F ZINC000880716607 FI On-Demand Mild LGMN 41 34 N#Cc1cc(NC(=O)N2CCC[C@@H]2[C@H](C#N)c2ccccc2)c(F)cc1F ZINC000880716608 FI On-Demand Mild LGMN 41 34 N#Cc1cc(NC(=O)N2CCC[C@@H]2[C@@H](C#N)c2ccccc2)c(F)cc1F ZINC000880716609 FI On-Demand Mild LGMN 41 34 N#Cc1cc(NC(=O)N2CCC[C@H]2[C@@H](C#N)c2ccccc2)c(F)cc1F ZINC000880716610 FI On-Demand Mild LGMN 41 34 N#Cc1cc(NC(=O)NCCOC2CCC2)c(F)cc1F ZINC000880716650 CF On-Demand Mild ADRB1 15 42 N#Cc1cc(NC(=O)N2CCC[C@@H](CNC(=O)c3ccccc3)C2)c(F)cc1F ZINC000880716666 GH On-Demand Mild CACNA1I 51 32 N#Cc1cc(NC(=O)N2CCC[C@H](CNC(=O)c3ccccc3)C2)c(F)cc1F ZINC000880716707 GH On-Demand Mild CACNA1I 51 32 C[C@@H]1CN(CCCNC(=O)Nc2cc(C#N)c(F)cc2F)C[C@@H](C)O1 ZINC000880716714 FE On-Demand Mild CCR3 31 42 N#Cc1cc(NC(=O)N2CCCN(C3CCCC3)CC2)c(F)cc1F ZINC000880716720 EG On-Demand Mild HRH3 24 40 N#Cc1cc(NC(=O)N2CCCN(C3CCCC3)CC2)c(F)cc1F ZINC000880716720 EG On-Demand Mild L3MBTL3 63 36 N#Cc1cc(NC(=O)NCCCN2CCCCC2)c(F)cc1F ZINC000880716731 DF On-Demand Mild CCR3 39 47 N#Cc1cc(NC(=O)NCCCN2CCCCC2)c(F)cc1F ZINC000880716731 DF On-Demand Mild CHRNA7 21 49 N#Cc1cc(NC(=O)NC2CCN(C3CC3)CC2)c(F)cc1F ZINC000880716733 DF On-Demand Mild EPHX2 28 41 Cn1cccc1C(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716734 GG On-Demand Anodyne RBP4 42 38 N#Cc1cc(NC(=O)N2CCC(c3nc4ccccc4[nH]3)CC2)c(F)cc1F ZINC000880716740 GI On-Demand Mild FASN 17 42 N#Cc1cc(NC(=O)N2CCC(c3nc4ccccc4[nH]3)CC2)c(F)cc1F ZINC000880716740 GI On-Demand Mild SMO 31 44 N#Cc1cc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c(F)cc1F ZINC000880716755 EI On-Demand Mild PREP 54 36 N#Cc1cc(NC(=O)N2CCC[C@H]2Cc2ccccc2)c(F)cc1F ZINC000880716755 EI On-Demand Mild LGMN 55 37 CCOc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)n1 ZINC000880716757 GE On-Demand Mild P2RY12 24 42 CCOc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3F)CC2)n1 ZINC000880716757 GE On-Demand Mild FAAH 22 40 N#Cc1cc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c(F)cc1F ZINC000880716759 EI On-Demand Mild PREP 54 36 N#Cc1cc(NC(=O)N2CCC[C@@H]2Cc2ccccc2)c(F)cc1F ZINC000880716759 EI On-Demand Mild LGMN 55 37 N#Cc1cc(NC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c(F)cc1F ZINC000880716764 GG On-Demand Mild EPHX2 28 43 N#Cc1cc(NC(=O)N2CCN(C3CCCC3)CC2)c(F)cc1F ZINC000880716768 EF On-Demand Mild L3MBTL3 49 33 CC(C)(C)CC(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716777 GI On-Demand Anodyne RBP4 47 40 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716795 FH On-Demand Anodyne EPHX2 59 44 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716795 FH On-Demand Anodyne CXCR3 15 43 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716795 FH On-Demand Anodyne CCR8 64 41 CCOC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716795 FH On-Demand Anodyne GPR119 19 40 Cn1cnnc1C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716796 FG On-Demand Anodyne RBP4 54 38 N#Cc1cc(NC(=O)NC2CCN(C(=O)c3ccoc3)CC2)c(F)cc1F ZINC000880716800 FF On-Demand Mild EPHX2 34 40 CCCN(CCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716839 DG On-Demand Anodyne SOAT1 23 44 N#Cc1cc(NC(=O)N2CCC[C@@H](c3noc(C4CC4)n3)C2)c(F)cc1F ZINC000880716866 FH On-Demand Mild SMO 25 43 N#Cc1cc(NC(=O)N2CCC[C@@H](c3noc(C4CC4)n3)C2)c(F)cc1F ZINC000880716866 FH On-Demand Mild ETHR 52 43 N#Cc1cc(NC(=O)N2CCC[C@H](c3noc(C4CC4)n3)C2)c(F)cc1F ZINC000880716867 FH On-Demand Mild SMO 25 43 N#Cc1cc(NC(=O)N2CCC[C@H](c3noc(C4CC4)n3)C2)c(F)cc1F ZINC000880716867 FH On-Demand Mild ETHR 52 43 N#Cc1ccccc1NC1CCN(C(=O)c2cncc(Cl)n2)CC1 ZINC000880716896 EF On-Demand Mild CSNK2A1 50 35 N#Cc1cc(NC(=O)NC[C@H](O)CN2CCc3ccccc3C2)c(F)cc1F ZINC000880716948 GE On-Demand Mild ADRB1 40 33 C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880716957 DI On-Demand Anodyne RBP4 58 42 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880716961 DH On-Demand Anodyne RBP4 57 41 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880716966 DG On-Demand Anodyne RBP4 55 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880716967 DG On-Demand Anodyne RBP4 55 41 CN(C)S(=O)(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880716972 GD On-Demand Anodyne RBP4 49 41 N#Cc1cc(NC(=O)N2CCN(c3ncccn3)CC2)c(F)cc1F ZINC000880716973 ED On-Demand Mild FAAH 22 41 COCCCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716976 DG On-Demand Anodyne CCR3 18 42 N#Cc1cc(NC(=O)NCCCN2CCCC2=O)c(F)cc1F ZINC000880716977 DD On-Demand Mild CCR3 24 42 N#Cc1cc(NC(=O)NCCCN2CCCC2=O)c(F)cc1F ZINC000880716977 DD On-Demand Mild TYRO3 18 40 N#Cc1cc(NC(=O)N2CCN(Cc3ccncc3)CC2)c(F)cc1F ZINC000880716985 FF On-Demand Mild FAAH 26 46 Cn1nccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880716990 DF On-Demand Anodyne P2RX7 19 50 N#Cc1cc(NC(=O)NC2CCCCC2)c(F)cc1F ZINC000880717004 CG On-Demand Mild EPHX2 26 56 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717006 GI On-Demand Anodyne RBP4 40 37 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717006 GI On-Demand Anodyne CACNA1G 38 40 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717006 GI On-Demand Anodyne ASAH1 68 34 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717008 DI On-Demand Anodyne RBP4 70 48 C[C@H]1C[C@@H](C)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717009 DI On-Demand Anodyne RBP4 70 48 CC(C)CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717022 EH On-Demand Anodyne RBP4 43 39 CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717061 EH On-Demand Anodyne SIGMAR1 15 40 CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717061 EH On-Demand Anodyne CCR3 66 46 CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717061 EH On-Demand Anodyne EPHX2 56 42 CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717061 EH On-Demand Anodyne CXCR3 23 44 CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717061 EH On-Demand Anodyne MCHR1 22 42 N#Cc1cc(NC(=O)NCc2cccnc2N2CCOCC2)c(F)cc1F ZINC000880717062 FE On-Demand Mild MTOR 50 38 N#Cc1cc(NC(=O)NCc2cccnc2N2CCOCC2)c(F)cc1F ZINC000880717062 FE On-Demand Mild SCN10A 21 50 COCCN(CCOC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717073 EG On-Demand Anodyne SOAT1 23 41 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)c1 ZINC000880717084 GH On-Demand Anodyne RBP4 29 43 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cccc2nsnc12 ZINC000880717107 DE On-Demand Anodyne FKBP1A 77 39 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cccc2nsnc12 ZINC000880717107 DE On-Demand Anodyne PREP 44 38 CC[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717108 DI On-Demand Anodyne DPP4 16 40 CC[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717108 DI On-Demand Anodyne ACKR3 59 34 CC[C@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717109 DI On-Demand Anodyne DPP4 16 40 CC[C@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717109 DI On-Demand Anodyne ACKR3 59 34 CC(C)c1nnc2n1CCN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C2 ZINC000880717110 FH On-Demand Anodyne P2RX7 24 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne F2 21 42 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne PLG 19 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne FKBP1A 41 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne CELA1 47 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne TRHR 48 34 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717119 FD On-Demand Anodyne HLA-DRB3 45 32 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne F2 21 42 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne PLG 19 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne FKBP1A 41 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne CELA1 47 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne TRHR 48 34 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880717120 FD On-Demand Anodyne HLA-DRB3 45 32 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717148 FI On-Demand Mild CCR3 55 41 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717148 FI On-Demand Mild EPHX2 43 42 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717148 FI On-Demand Mild CXCR3 22 43 C=C(C)CN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717148 FI On-Demand Mild MCHR1 15 40 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717152 FG On-Demand Anodyne RBP4 59 41 CCN1CC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717153 EG On-Demand Anodyne CCR3 92 44 CCN1CC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717153 EG On-Demand Anodyne CACNA1I 74 39 CN1CCC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717159 EG On-Demand Anodyne CCR3 105 41 CN1CCC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717159 EG On-Demand Anodyne CACNA1I 63 40 CN1CCC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717159 EG On-Demand Anodyne ACKR3 45 32 CN1CCC(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717172 EG On-Demand Anodyne P2RX7 16 40 CN1CCC(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717172 EG On-Demand Anodyne CCR3 69 45 CN1CCC(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717172 EG On-Demand Anodyne CACNA1I 76 42 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717174 FH On-Demand Anodyne CELA1 41 38 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717177 GI On-Demand Anodyne RBP4 53 39 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717178 GI On-Demand Anodyne RBP4 53 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCCO1 ZINC000880717179 DH On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCCO1 ZINC000880717180 DH On-Demand Anodyne RBP4 53 40 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)n1 ZINC000880717189 GG On-Demand Anodyne FAAH 23 45 COc1ccnc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)n1 ZINC000880717189 GG On-Demand Anodyne RBP4 30 43 Nc1nc(O)cc([C@H]2CCN(C(=O)CC[C@H]3CCc4ccccc43)C2)n1 ZINC000880717200 FF On-Demand Anodyne ETHR 41 34 Nc1nc(O)cc([C@H]2CCN(C(=O)CC[C@@H]3CCc4ccccc43)C2)n1 ZINC000880717201 FF On-Demand Anodyne ETHR 41 34 Nc1nc(O)cc([C@@H]2CCN(C(=O)CC[C@H]3CCc4ccccc43)C2)n1 ZINC000880717202 FF On-Demand Anodyne ETHR 41 34 Nc1nc(O)cc([C@@H]2CCN(C(=O)CC[C@@H]3CCc4ccccc43)C2)n1 ZINC000880717203 FF On-Demand Anodyne ETHR 41 34 C[C@@H](O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717205 EH On-Demand Anodyne RBP4 53 41 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717206 DG On-Demand Anodyne RBP4 61 44 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717206 DG On-Demand Anodyne MCHR1 24 45 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717206 DG On-Demand Anodyne SFRP1 60 35 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717206 DG On-Demand Anodyne WNT3 43 35 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717216 CH On-Demand Anodyne RBP4 60 44 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717217 CH On-Demand Anodyne RBP4 60 44 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cccn2nccc12 ZINC000880717222 DD On-Demand Anodyne FKBP1A 73 39 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cccn2nccc12 ZINC000880717222 DD On-Demand Anodyne PREP 53 36 CCOC(=O)[C@@H]1CCCCN1C(=O)Cc1c(Br)cnn1C ZINC000880717227 FD On-Demand Anodyne FKBP1A 50 38 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CNC(=O)OC(C)(C)C)OC ZINC000880717234 FD On-Demand Anodyne F2 19 42 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H](CNC(=O)OC(C)(C)C)OC ZINC000880717234 FD On-Demand Anodyne FKBP1A 54 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne FKBP1A 110 45 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne CPT1A 32 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne CPT2 40 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne PREP 43 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne MTNR1B 22 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne MMP3 30 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne MMP8 17 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880717237 EF On-Demand Anodyne FAAH 15 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne FKBP1A 110 45 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne CPT1A 32 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne CPT2 40 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne PREP 43 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne MTNR1B 22 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne MMP3 30 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne MMP8 17 41 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880717240 EF On-Demand Anodyne FAAH 15 40 CCc1nnc2n1CCN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C2 ZINC000880717245 FG On-Demand Anodyne P2RX7 25 49 CCCCN(CCOC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717258 EI On-Demand Anodyne SOAT1 29 48 CCOC(=O)[C@@H]1CCCCN1C(=O)CCCn1ccc(C(=O)OC)n1 ZINC000880717261 FD On-Demand Anodyne FKBP1A 66 39 COC(=O)C1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717276 FH On-Demand Anodyne EPHX2 50 41 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717279 GI On-Demand Anodyne RBP4 40 38 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717279 GI On-Demand Anodyne CACNA1I 46 35 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717280 GI On-Demand Anodyne RBP4 40 38 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717280 GI On-Demand Anodyne CACNA1I 46 35 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717285 FG On-Demand Anodyne EPHX2 20 40 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717285 FG On-Demand Anodyne RBP4 43 38 CC(=O)NCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717285 FG On-Demand Anodyne CACNA1I 60 37 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717288 GG On-Demand Anodyne ROCK2 22 44 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717288 GG On-Demand Anodyne PDS 53 37 C=CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717298 EH On-Demand Mild CCR3 56 42 C=CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717298 EH On-Demand Mild EPHX2 48 38 C=CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717298 EH On-Demand Mild CXCR3 22 43 C=CCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717298 EH On-Demand Mild MCHR1 19 42 Cc1noc(C)c1CCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717310 EH On-Demand Anodyne P2RX7 23 52 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1 ZINC000880717316 DH On-Demand Anodyne RBP4 55 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1 ZINC000880717317 DH On-Demand Anodyne RBP4 55 41 Cc1noc(C2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)n1 ZINC000880717325 FI On-Demand Anodyne RBP4 48 37 Cc1noc(C2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)n1 ZINC000880717325 FI On-Demand Anodyne SMO 39 49 Cc1noc(C2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)n1 ZINC000880717325 FI On-Demand Anodyne ETHR 67 44 CN1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717327 DG On-Demand Anodyne CCR3 81 40 CN1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717327 DG On-Demand Anodyne EPHX2 41 42 CO[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717344 DH On-Demand Anodyne RBP4 53 40 COC(=O)[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880717346 EE On-Demand Anodyne RBP4 46 39 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880717347 EE On-Demand Anodyne RBP4 46 39 C[C@@H](Cn1cncn1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717355 EF On-Demand Anodyne HIS3 78 38 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880717362 EE On-Demand Anodyne FKBP1A 65 39 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880717362 EE On-Demand Anodyne TRHR 47 32 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880717362 EE On-Demand Anodyne PREP 33 42 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880717363 EE On-Demand Anodyne FKBP1A 65 39 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880717363 EE On-Demand Anodyne TRHR 47 32 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880717363 EE On-Demand Anodyne PREP 33 42 CCOC(=O)[C@@H]1CCCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880717371 EE On-Demand Anodyne FKBP1A 71 41 CCOC(=O)[C@@H]1CCCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880717371 EE On-Demand Anodyne CPT1A 88 42 CC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717432 DJ On-Demand Anodyne CACNA1H 57 39 CC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717432 DJ On-Demand Anodyne RBP4 49 40 CC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717432 DJ On-Demand Anodyne TRPM8 25 42 CCOC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CCNC1=O ZINC000880717437 CC On-Demand Anodyne FKBP1A 58 41 CCOC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CCNC1=O ZINC000880717438 CC On-Demand Anodyne FKBP1A 58 41 CCCCCN(CCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717440 EH On-Demand Anodyne SOAT1 36 44 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cc(C)cnc1Cl ZINC000880717442 DF On-Demand Anodyne FKBP1A 57 36 Cc1noc(C)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717447 EH On-Demand Anodyne P2RX7 33 57 COC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717484 FG On-Demand Anodyne CCR3 30 42 COC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717484 FG On-Demand Anodyne EPHX2 59 43 COC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717484 FG On-Demand Anodyne CXCR3 15 41 COC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717484 FG On-Demand Anodyne SFRP1 42 34 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc(F)cc2C(C)(F)F)on1 ZINC000880717504 FJ On-Demand Anodyne KCNA5 18 45 COCCCCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717510 DH On-Demand Anodyne CCR3 16 41 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880717514 DF On-Demand Anodyne FKBP1A 72 38 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880717514 DF On-Demand Anodyne PREP 48 36 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880717514 DF On-Demand Anodyne PTR1 47 33 CCOC(=O)[C@@H]1CCCCN1C(=O)COC1CC1 ZINC000880717516 CD On-Demand Anodyne FKBP1A 51 42 CCOC(=O)[C@@H]1CCCCN1C(=O)COC1CC1 ZINC000880717516 CD On-Demand Anodyne CPT2 41 38 CCOC(=O)[C@@H]1CCCCN1C(=O)COC1CC1 ZINC000880717516 CD On-Demand Anodyne PREP 30 41 C=CC(C)(C)CC(=O)N1CCCC[C@@H]1C(=O)OCC ZINC000880717521 CF On-Demand Mild FKBP1A 53 44 C=CC(C)(C)CC(=O)N1CCCC[C@@H]1C(=O)OCC ZINC000880717521 CF On-Demand Mild PREP 26 40 C=CC(C)(C)CC(=O)N1CCCC[C@@H]1C(=O)OCC ZINC000880717521 CF On-Demand Mild LGMN 40 35 C=CC(C)(C)CC(=O)N1CCCC[C@H]1C(=O)OCC ZINC000880717522 CF On-Demand Mild FKBP1A 53 44 C=CC(C)(C)CC(=O)N1CCCC[C@H]1C(=O)OCC ZINC000880717522 CF On-Demand Mild PREP 26 40 C=CC(C)(C)CC(=O)N1CCCC[C@H]1C(=O)OCC ZINC000880717522 CF On-Demand Mild LGMN 40 35 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880717527 GH On-Demand Anodyne FKBP1A 68 38 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880717527 GH On-Demand Anodyne WNT3 42 32 CCOC(=O)N1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717537 FH On-Demand Anodyne P2RY12 46 37 C=CC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717541 DI On-Demand Mild RBP4 49 40 CCOCCN(CC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717544 DH On-Demand Anodyne SOAT1 19 41 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717557 EF On-Demand Anodyne RBP4 55 41 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717557 EF On-Demand Anodyne SFRP1 44 37 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717558 EF On-Demand Anodyne RBP4 55 41 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717558 EF On-Demand Anodyne SFRP1 44 37 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717572 EH On-Demand Anodyne CCR3 104 44 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717572 EH On-Demand Anodyne EPHX2 37 40 CCN1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717572 EH On-Demand Anodyne BIRC2 29 42 CCN1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717573 EH On-Demand Anodyne CCR3 104 44 CCN1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717573 EH On-Demand Anodyne EPHX2 37 40 CCN1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717573 EH On-Demand Anodyne BIRC2 29 42 CCOC(=O)[C@@H]1CCCCN1C(=O)CC(C)(C)CC(F)(F)F ZINC000880717579 DG On-Demand Anodyne FKBP1A 47 42 CCOC(=O)[C@@H]1CCCCN1C(=O)CC(C)(C)CC(F)(F)F ZINC000880717579 DG On-Demand Anodyne PREP 18 43 CNS(=O)(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717588 GE On-Demand Anodyne RBP4 44 41 CC(C)(C)CN(CCCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717602 EI On-Demand Anodyne SOAT1 22 48 CCN(CC)C(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717608 GI On-Demand Anodyne RBP4 40 37 CCOC(=O)[C@@H]1CCCCN1C(=O)CC(C)(C)CC(F)F ZINC000880717610 DG On-Demand Anodyne FKBP1A 47 42 CCOC(=O)[C@@H]1CCCCN1C(=O)CC(C)(C)CC(F)F ZINC000880717610 DG On-Demand Anodyne PREP 21 51 CC(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717622 EG On-Demand Anodyne RBP4 53 39 CC(=O)N[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717623 EG On-Demand Anodyne RBP4 53 39 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717627 EE On-Demand Anodyne CCR3 40 38 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717627 EE On-Demand Anodyne CACNA1I 41 33 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717628 EE On-Demand Anodyne CCR3 40 38 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717628 EE On-Demand Anodyne CACNA1I 41 33 CCOC(=O)[C@@H]1CCCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880717675 FE On-Demand Anodyne FKBP1A 92 46 CCOC(=O)[C@@H]1CCCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880717675 FE On-Demand Anodyne CPT2 41 36 CCOC(=O)[C@@H]1CCCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880717675 FE On-Demand Anodyne PREP 53 40 CCn1cc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)cn1 ZINC000880717677 DH On-Demand Anodyne PANC 43 37 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717679 GI On-Demand Anodyne HRH2 26 42 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717679 GI On-Demand Anodyne MTNR1A 26 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717679 GI On-Demand Anodyne MTNR1B 25 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880717679 GI On-Demand Anodyne EPHX2 22 44 CC(C)(C(=O)N1CC[C@H](c2cc(O)nc(N)n2)C1)c1ccc(F)cc1F ZINC000880717687 FE On-Demand Anodyne PRCP 49 37 CC(C)(C(=O)N1CC[C@@H](c2cc(O)nc(N)n2)C1)c1ccc(F)cc1F ZINC000880717688 FE On-Demand Anodyne PRCP 49 37 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717689 FH On-Demand Anodyne RBP4 47 39 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717690 FH On-Demand Anodyne RBP4 47 39 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717697 GI On-Demand Anodyne RBP4 46 38 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717697 GI On-Demand Anodyne SFRP1 51 35 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717697 GI On-Demand Anodyne WNT3 41 32 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880717708 DE On-Demand Anodyne FKBP1A 79 40 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880717708 DE On-Demand Anodyne CPT1A 56 36 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880717708 DE On-Demand Anodyne CPT2 43 36 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880717708 DE On-Demand Anodyne PREP 54 44 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1O ZINC000880717715 FI On-Demand Anodyne NR3C1 18 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1O ZINC000880717715 FI On-Demand Anodyne NR3C2 25 40 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1O ZINC000880717715 FI On-Demand Anodyne MT-ND1 18 44 COc1ccc(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1O ZINC000880717715 FI On-Demand Anodyne HSD17B2 20 42 CC(C)(C)CN(CCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717729 EH On-Demand Anodyne SOAT1 17 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717737 FG On-Demand Anodyne CCR3 50 39 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717737 FG On-Demand Anodyne RBP4 40 38 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717737 FG On-Demand Anodyne CACNA1I 45 35 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717738 EF On-Demand Anodyne CASR 52 40 CN(CCN1CCOCC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717738 EF On-Demand Anodyne EPHX2 21 42 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc(CN2CCOCC2)o1 ZINC000880717739 FD On-Demand Anodyne FKBP1A 63 38 CCCO[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717741 FJ On-Demand Anodyne RBP4 40 37 CCCO[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717742 FJ On-Demand Anodyne RBP4 40 37 Cn1cc(CN2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)cn1 ZINC000880717743 GG On-Demand Anodyne FAAH 17 40 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717756 GI On-Demand Anodyne EPHX2 54 50 CCOC(=O)[C@@H]1CCCCN1C(=O)c1nnn(C)n1 ZINC000880717768 CB On-Demand Anodyne FKBP1A 50 38 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cncc2[nH]ccc12 ZINC000880717770 DE On-Demand Anodyne FKBP1A 68 40 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1c2c[nH]nc2CC[C@H]1C ZINC000880717821 DE On-Demand Anodyne FKBP1A 51 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1c2c[nH]nc2CC[C@@H]1C ZINC000880717822 DE On-Demand Anodyne FKBP1A 51 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1c2c[nH]nc2CC[C@@H]1C ZINC000880717823 DE On-Demand Anodyne FKBP1A 51 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1c2c[nH]nc2CC[C@H]1C ZINC000880717824 DE On-Demand Anodyne FKBP1A 51 36 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880717828 GG On-Demand Anodyne FKBP1A 104 40 CCOC(=O)[C@@H]1CCCCN1C(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880717828 GG On-Demand Anodyne HCRTR1 17 41 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880717837 EE On-Demand Anodyne FKBP1A 52 36 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880717837 EE On-Demand Anodyne WNT3A 40 34 CCCN(CC)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717859 CI On-Demand Anodyne SOAT1 23 46 CCOC(=O)[C@@H]1CCCCN1C(=O)c1nccnc1SC ZINC000880717868 DD On-Demand Anodyne FKBP1A 55 37 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717873 GE On-Demand Anodyne RBP4 55 42 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@@H]1CCc2nncn2CC1 ZINC000880717875 DD On-Demand Anodyne FKBP1A 50 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1CCc2nncn2CC1 ZINC000880717877 DD On-Demand Anodyne FKBP1A 50 36 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717879 FG On-Demand Anodyne CCR3 37 42 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717879 FG On-Demand Anodyne EPHX2 45 40 COC(=O)N1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717880 FG On-Demand Anodyne CCR3 37 42 COC(=O)N1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717880 FG On-Demand Anodyne EPHX2 45 40 CCOC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880717881 CE On-Demand Anodyne FKBP1A 43 39 CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880717891 EE On-Demand Anodyne FKBP1A 78 46 CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880717891 EE On-Demand Anodyne MPO 58 35 C[C@H](O)c1ccc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)cc1 ZINC000880717905 FI On-Demand Anodyne TRPV1 85 42 CCOC(=O)[C@@H]1CCCCN1C(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880717916 ED On-Demand Anodyne FKBP1A 50 39 CCO[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717919 EH On-Demand Anodyne RBP4 48 40 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717924 GI On-Demand Anodyne RBP4 42 38 COCCn1cc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)cn1 ZINC000880717933 EG On-Demand Anodyne HTR2A 20 41 COCCn1cc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)cn1 ZINC000880717933 EG On-Demand Anodyne PANC 52 38 CN(C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1)S(C)(=O)=O ZINC000880717934 GF On-Demand Anodyne RBP4 60 42 CN(C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1)S(C)(=O)=O ZINC000880717934 GF On-Demand Anodyne SFRP1 81 35 CN(C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1)S(C)(=O)=O ZINC000880717934 GF On-Demand Anodyne WNT3 58 35 COCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717940 EH On-Demand Anodyne RBP4 49 40 COCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717940 EH On-Demand Anodyne CACNA1I 44 33 COCCN(Cc1cccnc1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717946 FI On-Demand Anodyne SOAT1 20 42 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cnc(C(C)C)nc1C ZINC000880717947 DE On-Demand Anodyne FKBP1A 51 39 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne DRD2 19 44 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne DRD4 16 41 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne ADRA1B 15 42 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne CCR3 75 49 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne EPHX2 50 38 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne CXCR3 22 42 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne MCHR1 27 41 COCCN1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717955 FG On-Demand Anodyne CACNA1I 51 36 CCOC(=O)[C@@H]1CCCCN1C(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880717956 ED On-Demand Anodyne FKBP1A 46 40 COCCN(Cc1ccccn1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717959 FI On-Demand Anodyne SOAT1 21 40 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717961 FF On-Demand Mild EPHX2 22 40 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717961 FF On-Demand Mild RBP4 49 39 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880717961 FF On-Demand Mild CACNA1G 37 40 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717980 EH On-Demand Anodyne CCR3 51 44 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880717980 EH On-Demand Anodyne RBP4 47 39 Cc1nonc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880717986 DF On-Demand Anodyne P2RX7 24 41 C[C@H]1C[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1C ZINC000880718027 EH On-Demand Anodyne EPHX2 40 37 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880718060 GJ On-Demand Anodyne P2RY1 45 40 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880718060 GJ On-Demand Anodyne RIPK1 45 32 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880718060 GJ On-Demand Anodyne KCNK3 59 38 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880718060 GJ On-Demand Anodyne KCNK9 57 38 CCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718085 EH On-Demand Anodyne CACNA1H 51 36 CCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718085 EH On-Demand Anodyne S1PR2 31 45 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1 ZINC000880718104 EI On-Demand Anodyne RBP4 53 39 Cn1ccnc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)c1=O ZINC000880718105 GE On-Demand Anodyne RBP4 25 43 COc1ccccc1[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718111 GJ On-Demand Anodyne RBP4 96 54 COc1ccccc1[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718111 GJ On-Demand Anodyne ACKR3 66 34 COc1ccccc1[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718112 GJ On-Demand Anodyne RBP4 96 54 COc1ccccc1[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718112 GJ On-Demand Anodyne ACKR3 66 34 C[S@@](=O)CCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718132 DF On-Demand Anodyne CCR3 23 42 COC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718167 EG On-Demand Anodyne RBP4 50 42 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718172 EG On-Demand Anodyne RBP4 53 39 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718172 EG On-Demand Anodyne SFRP1 43 34 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718172 EG On-Demand Anodyne WNT3 52 31 CO/C(=C/c1ccccc1)C(=O)NC(C)(C)C(=O)NCC(C)(C)C ZINC000880718178 EF On-Demand Anodyne TLR4 25 42 CO/C(=C\c1ccccc1)C(=O)NC(C)(C)C(=O)NCC(C)(C)C ZINC000880718179 EF On-Demand Anodyne TLR4 25 42 CCOC[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718197 EI On-Demand Anodyne CCR3 35 42 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1(=O)=O ZINC000880718235 FF On-Demand Anodyne RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1(=O)=O ZINC000880718236 FF On-Demand Anodyne RBP4 57 43 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718289 FI On-Demand Anodyne TRPV1 19 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)S1 ZINC000880718300 EI On-Demand Anodyne RBP4 57 43 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)S1 ZINC000880718301 EI On-Demand Anodyne RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)S1 ZINC000880718302 EI On-Demand Anodyne RBP4 57 43 Cn1cc([C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)cn1 ZINC000880718345 FH On-Demand Anodyne RBP4 55 40 CNC(=O)CC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718347 FG On-Demand Anodyne RBP4 41 38 C[C@H]1c2ccccc2CN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718357 EK On-Demand Anodyne RBP4 51 40 C[C@H]1c2ccccc2CN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718357 EK On-Demand Anodyne TRPM8 32 45 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718360 GF On-Demand Anodyne CCR3 21 40 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718360 GF On-Demand Anodyne EPHX2 15 42 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718361 GF On-Demand Anodyne CCR3 21 40 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718361 GF On-Demand Anodyne EPHX2 15 42 CC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718393 DI On-Demand Anodyne CACNA1H 40 39 CC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718393 DI On-Demand Anodyne RBP4 47 39 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(F)cc1C(C)(F)F)C2 ZINC000880718399 FI On-Demand Anodyne HTR3A 33 42 CCOC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718424 EH On-Demand Anodyne CCR3 29 41 CCOC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718424 EH On-Demand Anodyne RBP4 43 38 CCOC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718424 EH On-Demand Anodyne CACNA1I 45 32 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(F)cc1C(C)(F)F)CC2 ZINC000880718429 FH On-Demand Anodyne CACNA1H 49 40 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(F)cc1C(C)(F)F)CC2 ZINC000880718429 FH On-Demand Anodyne RBP4 45 37 C[C@H](O)CN1CCC(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718497 GG On-Demand Anodyne CACNA1I 54 37 CNC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718503 EF On-Demand Anodyne RBP4 54 41 COCCCOC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718530 FH On-Demand Anodyne SCD1 21 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880718533 DI On-Demand Anodyne RBP4 63 45 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C ZINC000880718534 DI On-Demand Anodyne RBP4 63 45 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880718535 DI On-Demand Anodyne RBP4 63 45 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880718568 FI On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880718569 FI On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880718570 FI On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880718571 FI On-Demand Anodyne RBP4 53 40 CCCN(C)C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718648 FI On-Demand Anodyne RBP4 46 39 CCCN(C)C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718649 FI On-Demand Anodyne RBP4 46 39 C[C@H](CS(C)(=O)=O)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718650 EE On-Demand Anodyne TRPV1 40 34 CC(C)(C)CNC(=O)C(C)(C)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880718652 FF On-Demand Anodyne GABRA1 15 47 CC(C)(C)CNC(=O)C(C)(C)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880718652 FF On-Demand Anodyne MPO 64 37 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718654 EH On-Demand Anodyne ACKR3 59 34 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718655 EH On-Demand Anodyne ACKR3 59 34 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718667 FH On-Demand Anodyne CCR3 75 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718668 FH On-Demand Anodyne CCR3 75 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718669 FH On-Demand Anodyne CCR3 75 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718670 FH On-Demand Anodyne CCR3 75 40 Cn1cc([C@@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CCO2)cn1 ZINC000880718671 FG On-Demand Anodyne RBP4 45 36 CN(CCOCC1CC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718673 EH On-Demand Anodyne RBP4 15 42 C[C@H](CS(C)(=O)=O)N(C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CC1 ZINC000880718686 GG On-Demand Anodyne TRPV1 71 33 Cc1noc(C)c1CCCNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718690 FI On-Demand Anodyne P2RX7 17 52 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718712 EF On-Demand Anodyne LGMN 46 35 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718712 EF On-Demand Anodyne WNT3 43 34 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718794 GF On-Demand Anodyne HLA-DRB1 51 32 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880718796 GF On-Demand Anodyne HLA-DRB1 51 32 CC1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718806 CG On-Demand Anodyne RBP4 70 48 CC(=O)N(C[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CC1 ZINC000880718820 GH On-Demand Anodyne ACKR3 67 35 CC(=O)N(C[C@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CC1 ZINC000880718821 GH On-Demand Anodyne ACKR3 67 35 CN1C[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1=O ZINC000880718893 EF On-Demand Anodyne P2RX7 22 42 CN1C[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1=O ZINC000880718894 EF On-Demand Anodyne P2RX7 22 42 COCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718905 EF On-Demand Anodyne CACNA1H 55 35 COCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718905 EF On-Demand Anodyne S1PR2 30 43 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C2CC2)O1 ZINC000880718914 EH On-Demand Anodyne RBP4 55 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C2CC2)O1 ZINC000880718919 EH On-Demand Anodyne RBP4 55 41 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C2CC2)O1 ZINC000880718922 EH On-Demand Anodyne RBP4 55 41 Cn1nccc1C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718923 FI On-Demand Anodyne RBP4 60 38 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C2CC2)O1 ZINC000880718925 EH On-Demand Anodyne RBP4 55 41 COC(=O)CCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880718951 FI On-Demand Anodyne RBP4 44 40 CC(C)[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718987 DI On-Demand Anodyne RBP4 61 43 CN1C(=O)NC2(CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)C1=O ZINC000880718988 GE On-Demand Anodyne CACNA1H 54 40 CC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718999 DI On-Demand Anodyne CCR3 42 40 CC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718999 DI On-Demand Anodyne RBP4 55 41 CC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880718999 DI On-Demand Anodyne CACNA1I 48 32 O=C(Nc1ccccc1C(=O)Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccccc1 ZINC000880719008 JK On-Demand Anodyne DHODH 15 41 O=C(Nc1ccccc1C(=O)Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccccc1 ZINC000880719008 JK On-Demand Anodyne F10 22 43 O=C(Nc1ccccc1C(=O)Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccccc1 ZINC000880719008 JK On-Demand Anodyne PRNP 44 36 O=C(Nc1ccccc1C(=O)Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccccc1 ZINC000880719008 JK On-Demand Anodyne NR1H4 21 49 Cc1c(NC(=O)Nc2ccc(F)cc2C(C)(F)F)cnn1C ZINC000880719026 DH On-Demand Anodyne HTR2A 15 42 CCC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719028 EH On-Demand Anodyne CACNA1H 44 35 CCC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719028 EH On-Demand Anodyne RBP4 46 38 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1CC(C)(C)O ZINC000880719048 FG On-Demand Anodyne RBP4 47 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1CC(C)(C)O ZINC000880719049 FG On-Demand Anodyne RBP4 47 39 CN1CCO[C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C[C@H]21 ZINC000880719051 FF On-Demand Anodyne RBP4 41 38 CN1CCO[C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C[C@@H]21 ZINC000880719052 FF On-Demand Anodyne RBP4 41 38 CN1CCO[C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C[C@H]21 ZINC000880719053 FF On-Demand Anodyne RBP4 41 38 CN1CCO[C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C[C@@H]21 ZINC000880719054 FF On-Demand Anodyne RBP4 41 38 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1(=O)=O ZINC000880719055 FF On-Demand Anodyne RBP4 41 38 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1(=O)=O ZINC000880719056 FF On-Demand Anodyne RBP4 41 38 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719061 EH On-Demand Anodyne RBP4 58 40 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719061 EH On-Demand Anodyne SFRP1 86 35 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719061 EH On-Demand Anodyne WNT3 71 35 COCCO[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719070 FH On-Demand Anodyne ACKR3 45 32 COCCO[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719071 FH On-Demand Anodyne ACKR3 45 32 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1=O ZINC000880719152 DG On-Demand Anodyne RBP4 55 41 COC(=O)[C@H]1C[C@@H](C)CCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880719248 DF On-Demand Anodyne PTR1 44 32 COC(=O)[C@@H]1C[C@@H](C)CCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880719250 DF On-Demand Anodyne PTR1 44 32 COC(=O)[C@@H]1C[C@H](C)CCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880719252 DF On-Demand Anodyne PTR1 44 32 COC(=O)[C@H]1C[C@H](C)CCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880719254 DF On-Demand Anodyne PTR1 44 32 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719261 GH On-Demand Anodyne RBP4 54 41 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719308 EG On-Demand Anodyne RBP4 54 40 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719308 EG On-Demand Anodyne CACNA1I 52 33 CNC(=O)[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880719311 ED On-Demand Anodyne RBP4 46 39 CNC(=O)[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880719312 ED On-Demand Anodyne RBP4 46 39 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880719317 GH On-Demand Anodyne RBP4 52 39 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880719318 GH On-Demand Anodyne RBP4 52 39 Cn1cc([C@@H]2CCCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)cn1 ZINC000880719330 FI On-Demand Anodyne RBP4 49 39 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880719387 EG On-Demand Anodyne ACKR3 68 36 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880719388 EG On-Demand Anodyne ACKR3 68 36 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1=O ZINC000880719464 DG On-Demand Anodyne RBP4 55 41 CO[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1OC ZINC000880719465 EF On-Demand Anodyne RBP4 58 44 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719467 FG On-Demand Anodyne CCR3 35 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719467 FG On-Demand Anodyne EPHX2 49 41 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719467 FG On-Demand Anodyne CCR8 72 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719467 FG On-Demand Anodyne SFRP1 44 33 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719468 FG On-Demand Anodyne CCR3 35 42 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719468 FG On-Demand Anodyne EPHX2 49 41 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719468 FG On-Demand Anodyne CCR8 72 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719468 FG On-Demand Anodyne SFRP1 44 33 C[C@@H]1CN(CCCNC(=O)Nc2ccc(F)cc2C(C)(F)F)CCCO1 ZINC000880719500 FH On-Demand Anodyne CCR3 49 45 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1F ZINC000880719563 DI On-Demand Anodyne RBP4 56 41 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1F ZINC000880719564 DI On-Demand Anodyne RBP4 56 41 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1F ZINC000880719566 DI On-Demand Anodyne RBP4 56 41 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1F ZINC000880719567 DI On-Demand Anodyne RBP4 56 41 CS[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N(C)C ZINC000880719569 FG On-Demand Anodyne RBP4 52 39 CS[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N(C)C ZINC000880719570 FG On-Demand Anodyne RBP4 52 39 CS[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N(C)C ZINC000880719572 FG On-Demand Anodyne RBP4 52 39 CS[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N(C)C ZINC000880719573 FG On-Demand Anodyne RBP4 52 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C(N)=O ZINC000880719618 EF On-Demand Anodyne RBP4 53 41 COCC(=O)NC1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719630 ED On-Demand Anodyne RBP4 54 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719689 FG On-Demand Anodyne CCR3 107 39 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719689 FG On-Demand Anodyne CACNA1I 56 38 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719692 FG On-Demand Anodyne CCR3 107 39 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880719692 FG On-Demand Anodyne CACNA1I 56 38 CC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719737 EH On-Demand Anodyne CACNA1H 43 36 CC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719737 EH On-Demand Anodyne RBP4 48 39 COC(=O)[C@H]1C[C@@H](C)CCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880719747 ED On-Demand Anodyne TRPC6 40 37 COC(=O)[C@@H]1C[C@H](C)CCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880719748 ED On-Demand Anodyne TRPC6 40 37 COC(=O)[C@H]1C[C@H](C)CCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880719749 ED On-Demand Anodyne TRPC6 40 37 COC(=O)[C@@H]1C[C@@H](C)CCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880719750 ED On-Demand Anodyne TRPC6 40 37 COC(=O)c1cn([C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)nn1 ZINC000880719751 GF On-Demand Anodyne RBP4 37 40 COC(=O)c1cn([C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)nn1 ZINC000880719752 GF On-Demand Anodyne RBP4 37 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1c1ccccc1 ZINC000880719791 EK On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1c1ccccc1 ZINC000880719793 EK On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@H]1c1ccccc1 ZINC000880719795 EK On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@H]1c1ccccc1 ZINC000880719797 EK On-Demand Anodyne RBP4 53 40 CC(=O)Nc1ccn([C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)n1 ZINC000880719798 GH On-Demand Anodyne RBP4 45 37 CC(=O)Nc1ccn([C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)n1 ZINC000880719799 GH On-Demand Anodyne RBP4 45 37 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1CCO ZINC000880719824 EE On-Demand Anodyne RBP4 53 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1CCO ZINC000880719825 EE On-Demand Anodyne RBP4 53 39 COC[C@@H](C)n1ccc(NC(=O)Nc2ccc(F)cc2C(C)(F)F)n1 ZINC000880719925 FH On-Demand Anodyne GCK 18 40 COC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719964 EF On-Demand Anodyne CACNA1H 41 35 COC1(CO)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880719964 EF On-Demand Anodyne RBP4 53 39 C[C@@H]1CSCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720024 EI On-Demand Anodyne RBP4 55 41 COC(=O)[C@H]1C[C@H](OC)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720049 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@@H]1C[C@@H](OC)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720051 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@@H]1C[C@H](OC)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720052 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@H]1C[C@@H](OC)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720054 DD On-Demand Anodyne PREP 22 44 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1O ZINC000880720055 DF On-Demand Anodyne RBP4 57 43 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1O ZINC000880720057 DF On-Demand Anodyne RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1O ZINC000880720058 DF On-Demand Anodyne RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1O ZINC000880720060 DF On-Demand Anodyne RBP4 57 43 CCNc1nc(C)c(C(=O)NCc2cncc(OC)c2)s1 ZINC000880720095 DE On-Demand Anodyne CHRM4 20 42 CCNc1nc(C)c(C(=O)NCc2cncc(OC)c2)s1 ZINC000880720095 DE On-Demand Anodyne SCD1 33 46 CCNc1nc(C)c(C(=O)NCc2cncc(OC)c2)s1 ZINC000880720095 DE On-Demand Anodyne SCD 32 43 COC[C@@H]1CCCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720102 EI On-Demand Anodyne CCR3 33 41 COC[C@@H]1CCCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720102 EI On-Demand Anodyne RBP4 46 38 COC(=O)[C@@H]1C[C@@H](C)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720105 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@H]1C[C@@H](C)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720107 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@H]1C[C@H](C)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720108 DD On-Demand Anodyne PREP 22 44 COC(=O)[C@@H]1C[C@H](C)CCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880720109 DD On-Demand Anodyne PREP 22 44 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1O ZINC000880720115 DG On-Demand Anodyne RBP4 56 42 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H]1O ZINC000880720116 DG On-Demand Anodyne RBP4 56 42 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1O ZINC000880720117 DG On-Demand Anodyne RBP4 56 42 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H]1O ZINC000880720118 DG On-Demand Anodyne RBP4 56 42 COC1(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720150 EH On-Demand Anodyne CACNA1H 43 36 CCCN(CCCN(C)C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720175 EI On-Demand Anodyne SOAT1 27 47 COc1cncc(CNC(=O)CCc2cn[nH]c2)c1 ZINC000880720196 CD On-Demand Anodyne ROCK1 39 40 COc1cncc(CNC(=O)CCc2cn[nH]c2)c1 ZINC000880720196 CD On-Demand Anodyne ROCK2 47 41 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720215 GE On-Demand Anodyne RBP4 41 38 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720217 GE On-Demand Anodyne RBP4 41 38 COCCO[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720218 EG On-Demand Anodyne RBP4 44 38 COCCO[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720218 EG On-Demand Anodyne LIPG 40 41 COCCO[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720220 EG On-Demand Anodyne RBP4 44 38 COCCO[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720220 EG On-Demand Anodyne LIPG 40 41 CCn1cccc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1=O ZINC000880720228 FG On-Demand Anodyne P2RX7 55 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS(=O)(=O)C1 ZINC000880720231 FF On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS(=O)(=O)C1 ZINC000880720233 FF On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](CO)O1 ZINC000880720243 EF On-Demand Anodyne RBP4 46 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](CO)O1 ZINC000880720245 EF On-Demand Anodyne RBP4 46 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](CO)O1 ZINC000880720247 EF On-Demand Anodyne RBP4 46 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](CO)O1 ZINC000880720249 EF On-Demand Anodyne RBP4 46 39 CN1C(=O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@H]1c1ccccc1 ZINC000880720296 GH On-Demand Anodyne P2RX7 18 40 CN1C(=O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@H]1c1ccccc1 ZINC000880720296 GH On-Demand Anodyne RBP4 45 38 CN1C(=O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1c1ccccc1 ZINC000880720297 GH On-Demand Anodyne P2RX7 18 40 CN1C(=O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1c1ccccc1 ZINC000880720297 GH On-Demand Anodyne RBP4 45 38 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(F)cc1C(C)(F)F)c1ccccn1 ZINC000880720307 GH On-Demand Anodyne P2RY1 34 43 COC(=O)C[C@](C)(NC(=O)Nc1ccc(F)cc1C(C)(F)F)c1ccccn1 ZINC000880720308 GH On-Demand Anodyne P2RY1 34 43 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCCO1 ZINC000880720331 EH On-Demand Anodyne RBP4 55 41 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1 ZINC000880720342 EI On-Demand Anodyne RBP4 44 38 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCS1 ZINC000880720344 EI On-Demand Anodyne RBP4 44 38 COc1cncc(CNC(=O)c2sc(NC3CC3)nc2C)c1 ZINC000880720413 DE On-Demand Anodyne CHRM4 15 40 COc1cncc(CNC(=O)c2sc(NC3CC3)nc2C)c1 ZINC000880720413 DE On-Demand Anodyne SCD1 31 44 COc1cncc(CNC(=O)c2sc(NC3CC3)nc2C)c1 ZINC000880720413 DE On-Demand Anodyne SCD 31 43 COc1cc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)ncn1 ZINC000880720429 GG On-Demand Anodyne PDGFRB 51 40 COc1cc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)ncn1 ZINC000880720429 GG On-Demand Anodyne RBP4 31 42 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720456 FG On-Demand Anodyne CCR1 25 42 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720462 GH On-Demand Anodyne HTR1A 20 44 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720462 GH On-Demand Anodyne PDGFRB 40 42 COc1cnccc1N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720462 GH On-Demand Anodyne RBP4 33 46 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne TRPV1 15 50 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne MTNR1A 30 40 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne MTNR1B 26 40 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne GRIA1 49 35 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne FAAH 42 39 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne SLC6A5 17 43 COc1cncc(CNC(=O)CCCCCc2ccc(O)cc2)c1 ZINC000880720487 EG On-Demand Anodyne SUCNR1 26 40 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720504 FI On-Demand Anodyne RBP4 47 38 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720506 FI On-Demand Anodyne RBP4 47 38 CO[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H]1C ZINC000880720509 EH On-Demand Anodyne RBP4 54 40 CO[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1C ZINC000880720514 EH On-Demand Anodyne RBP4 54 40 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720518 FI On-Demand Anodyne RBP4 48 39 Cn1nccc1[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720519 FI On-Demand Anodyne RBP4 48 39 COC(=O)[C@H]1C[C@@H](OC)CCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880720535 GF On-Demand Anodyne FKBP1A 78 47 COC(=O)[C@H]1C[C@H](OC)CCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880720537 GF On-Demand Anodyne FKBP1A 78 47 COC(=O)[C@@H]1C[C@@H](OC)CCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880720539 GF On-Demand Anodyne FKBP1A 78 47 COC(=O)[C@@H]1C[C@H](OC)CCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880720541 GF On-Demand Anodyne FKBP1A 78 47 CN1C(=O)N[C@@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC[C@@H]21 ZINC000880720546 FF On-Demand Anodyne RBP4 47 38 CCCCN(CCCO)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720583 EH On-Demand Anodyne SOAT1 30 41 C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1C ZINC000880720603 DJ On-Demand Anodyne WNT3 41 32 C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@@H]1C ZINC000880720603 DJ On-Demand Anodyne TRPC6 52 39 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720605 DJ On-Demand Anodyne WNT3 41 32 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720605 DJ On-Demand Anodyne TRPC6 52 39 Cc1noc(C2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)n1 ZINC000880720610 EG On-Demand Anodyne RBP4 48 40 COC(=O)C1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720611 FE On-Demand Anodyne CACNA1H 43 36 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720672 FG On-Demand Anodyne CCR3 63 39 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720672 FG On-Demand Anodyne CCR2 15 40 CN(C)S(=O)(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720831 GF On-Demand Anodyne RBP4 40 38 CN(C)S(=O)(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720832 GF On-Demand Anodyne RBP4 40 38 C[C@H]1C[C@@H](C)N1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880720850 CH On-Demand Anodyne RBP4 46 41 CC(C)[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880720865 EH On-Demand Anodyne RBP4 53 39 COC(=O)[C@@H]1C[C@@H](C)CCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880720887 EF On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@H]1C[C@H](C)CCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880720889 EF On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@H]1C[C@H](C)CCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880720891 EF On-Demand Anodyne MTNR1B 18 40 COC(=O)[C@@H]1C[C@@H](C)CCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880720893 EF On-Demand Anodyne MTNR1B 18 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1C ZINC000880720940 DI On-Demand Anodyne RBP4 58 42 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1C ZINC000880720940 DI On-Demand Anodyne SFRP1 64 32 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H]1C ZINC000880720940 DI On-Demand Anodyne WNT3 47 32 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720942 DI On-Demand Anodyne RBP4 58 42 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720942 DI On-Demand Anodyne SFRP1 64 32 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720942 DI On-Demand Anodyne WNT3 47 32 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720944 DI On-Demand Anodyne RBP4 58 42 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720944 DI On-Demand Anodyne SFRP1 64 32 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880720944 DI On-Demand Anodyne WNT3 47 32 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C ZINC000880720946 DI On-Demand Anodyne RBP4 58 42 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C ZINC000880720946 DI On-Demand Anodyne SFRP1 64 32 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C ZINC000880720946 DI On-Demand Anodyne WNT3 47 32 CC(=O)OC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720965 EG On-Demand Anodyne RBP4 46 39 Cc1cncc(CNC(=O)Nc2ccc(F)cc2C(C)(F)F)c1 ZINC000880720979 DH On-Demand Anodyne NAMPT 15 48 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720989 FH On-Demand Anodyne RBP4 53 39 Cn1ccnc1[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880720991 FH On-Demand Anodyne RBP4 53 39 CN(CCO)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880720998 FF On-Demand Anodyne RBP4 60 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880721134 GE On-Demand Anodyne HSD11B1 22 47 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880721134 GE On-Demand Anodyne RBP4 52 39 CCC1(O)CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721136 EI On-Demand Anodyne EPHX2 43 39 CN(C)C(=O)CC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721150 FH On-Demand Anodyne RBP4 40 37 CC(=O)N1CCc2c(NC(=O)Nc3ccc(F)cc3C(C)(F)F)cccc21 ZINC000880721175 GI On-Demand Anodyne P2RY1 45 35 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)CC1 ZINC000880721183 GH On-Demand Anodyne SLC6A5 21 45 CN1CCC(N2CCC(NC(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)CC1 ZINC000880721183 GH On-Demand Anodyne EPHX2 45 39 COCCOC1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721202 EF On-Demand Anodyne RBP4 53 40 CO[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721217 EH On-Demand Anodyne RBP4 46 40 CN1CC[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721227 DG On-Demand Anodyne CCR3 73 44 CN1CC[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721227 DG On-Demand Anodyne CACNA1I 65 39 CN1CC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721228 DG On-Demand Anodyne CCR3 73 44 CN1CC[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721228 DG On-Demand Anodyne CACNA1I 65 39 Cc1cnc(CN(C)[C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)o1 ZINC000880721276 GH On-Demand Anodyne RBP4 46 36 Cc1cnc(CN(C)[C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)o1 ZINC000880721277 GH On-Demand Anodyne RBP4 46 36 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1O ZINC000880721327 DG On-Demand Anodyne RBP4 55 42 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1O ZINC000880721328 DG On-Demand Anodyne RBP4 55 42 CN(C)CCCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721330 FJ On-Demand Anodyne RBP4 47 38 CN(C)CCCC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721330 FJ On-Demand Anodyne ACKR3 45 32 CCN(CC(C)(C)O)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721367 DH On-Demand Anodyne SOAT1 15 41 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721368 GG On-Demand Anodyne CCR3 24 44 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721368 GG On-Demand Anodyne EPHX2 53 48 COCCC(=O)N1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880721368 GG On-Demand Anodyne CCR8 53 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721392 GI On-Demand Anodyne CCR3 49 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721393 GI On-Demand Anodyne CCR3 49 42 CCC[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880721417 EH On-Demand Anodyne RBP4 54 41 CCC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880721418 EH On-Demand Anodyne RBP4 54 41 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CCN(S(C)(=O)=O)CC1 ZINC000880721428 GF On-Demand Anodyne EPHX2 17 45 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CCN(S(C)(=O)=O)CC1 ZINC000880721428 GF On-Demand Anodyne ADAMTS4 45 38 COc1cncc(CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c1 ZINC000880721455 ED On-Demand Anodyne GRIN2B 15 43 COc1cncc(CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c1 ZINC000880721456 ED On-Demand Anodyne GRIN2B 15 43 CCc1noc(C)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721488 EI On-Demand Anodyne P2RX7 19 47 CC(C)(C[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1)C(N)=O ZINC000880721501 GI On-Demand Anodyne CCR3 52 36 CC(C)(C[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1)C(N)=O ZINC000880721501 GI On-Demand Anodyne RBP4 47 39 CC(C)(C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1)C(N)=O ZINC000880721502 GI On-Demand Anodyne CCR3 52 36 CC(C)(C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1)C(N)=O ZINC000880721502 GI On-Demand Anodyne RBP4 47 39 COC[C@@H]1CCCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721508 EH On-Demand Anodyne ACKR3 65 34 CCN1C[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1=O ZINC000880721521 EF On-Demand Anodyne P2RX7 16 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721522 FD On-Demand Anodyne PAPA1_CARPA 41 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721522 FD On-Demand Anodyne CTSL 19 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721522 FD On-Demand Anodyne FPR1 40 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721523 FD On-Demand Anodyne PAPA1_CARPA 41 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721523 FD On-Demand Anodyne CTSL 19 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cncc(OC)c1 ZINC000880721523 FD On-Demand Anodyne FPR1 40 35 COC(=O)C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880721549 FF On-Demand Anodyne RBP4 54 40 COC(=O)C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880721550 FF On-Demand Anodyne RBP4 54 40 COCCn1nc(C)c(NC(=O)Nc2ccc(F)cc2C(C)(F)F)c1C ZINC000880721556 FI On-Demand Anodyne P2RX7 25 51 COc1cccc([C@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CCO2)c1 ZINC000880721611 GJ On-Demand Anodyne RBP4 53 38 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721616 EG On-Demand Anodyne CCR3 32 41 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721616 EG On-Demand Anodyne EPHX2 46 51 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721616 EG On-Demand Anodyne CCR8 42 36 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721617 EG On-Demand Anodyne CCR3 32 41 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721617 EG On-Demand Anodyne EPHX2 46 51 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721617 EG On-Demand Anodyne CCR8 42 36 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N(C)C ZINC000880721619 EG On-Demand Anodyne RBP4 53 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N(C)C ZINC000880721620 EG On-Demand Anodyne RBP4 53 41 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N(C)C ZINC000880721621 EG On-Demand Anodyne RBP4 53 41 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N(C)C ZINC000880721622 EG On-Demand Anodyne RBP4 53 41 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne ACE 17 40 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CTRA_BOVIN 53 31 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CTSG 40 31 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CAPNS1 45 30 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CELA2A 41 31 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne LGMN 69 39 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CAPN1 43 40 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne CAPN2 52 35 C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)c1nccn1C ZINC000880721727 FE On-Demand Anodyne Q9NAW4_PLAFA 40 47 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@]1=O ZINC000880721734 EG On-Demand Anodyne RBP4 42 38 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@]1=O ZINC000880721735 EG On-Demand Anodyne RBP4 42 38 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@@]1=O ZINC000880721736 EG On-Demand Anodyne RBP4 42 38 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@@]1=O ZINC000880721737 EG On-Demand Anodyne RBP4 42 38 CC(C)[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCCO1 ZINC000880721752 EI On-Demand Anodyne RBP4 40 38 C[C@@H]1CN(CC(F)(F)F)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880721753 GI On-Demand Anodyne RBP4 52 39 COc1cncc(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721788 EF On-Demand Anodyne NQO2 28 40 COc1cncc(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721788 EF On-Demand Anodyne MTNR1A 39 41 COc1cncc(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721788 EF On-Demand Anodyne MTNR1B 35 40 COc1cncc(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721789 EF On-Demand Anodyne NQO2 28 40 COc1cncc(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721789 EF On-Demand Anodyne MTNR1A 39 41 COc1cncc(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c1 ZINC000880721789 EF On-Demand Anodyne MTNR1B 35 40 COCC[C@@H]1COCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721796 EG On-Demand Anodyne ACKR3 45 31 COCC[C@H]1COCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721797 EG On-Demand Anodyne ACKR3 45 31 Cc1ccncc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721808 DH On-Demand Anodyne P2RX7 37 41 COc1cncc(CNC(=O)Cc2ccccc2N2CCCC2=O)c1 ZINC000880721815 EE On-Demand Anodyne HTR1A 15 40 COc1cncc(CNC(=O)Cc2ccccc2N2CCCC2=O)c1 ZINC000880721815 EE On-Demand Anodyne DRD4 40 33 COc1cncc(CNC(=O)Cc2ccccc2N2CCCC2=O)c1 ZINC000880721815 EE On-Demand Anodyne HTR7 23 40 COc1cncc(CNC(=O)Cc2ccccc2N2CCCC2=O)c1 ZINC000880721815 EE On-Demand Anodyne CYP11B2 20 42 O=C(Nc1ccc(N2CCOCC2)cn1)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880721816 IG On-Demand Anodyne CFTR 78 46 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880721828 FG On-Demand Anodyne RBP4 54 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880721829 FG On-Demand Anodyne RBP4 54 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880721830 FG On-Demand Anodyne RBP4 54 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880721831 FG On-Demand Anodyne RBP4 54 40 C#CC(C)(C)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880721869 CG On-Demand Mild P2RY1 15 42 Cc1nc(CN(C)[C@@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)no1 ZINC000880721893 GG On-Demand Anodyne RBP4 45 36 Cc1nc(CN(C)[C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)no1 ZINC000880721894 GG On-Demand Anodyne RBP4 45 36 C[C@@H](CNC(=O)Nc1ccc(F)cc1C(C)(F)F)S(C)(=O)=O ZINC000880721896 EE On-Demand Anodyne TRPV1 53 35 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722101 GI On-Demand Anodyne CCR3 46 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722101 GI On-Demand Anodyne EPHX2 20 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722104 GI On-Demand Anodyne CCR3 46 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722104 GI On-Demand Anodyne EPHX2 20 41 COCCNc1ccccc1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722125 GI On-Demand Anodyne P2RX7 21 41 COc1cncc(CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)c1 ZINC000880722142 FG On-Demand Anodyne DRD4 42 32 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC(=O)N1 ZINC000880722199 DE On-Demand Anodyne RBP4 42 38 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC(=O)N1 ZINC000880722200 DE On-Demand Anodyne RBP4 42 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1nccn1C ZINC000880722218 ED On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1nccn1C ZINC000880722219 ED On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1nccn1C ZINC000880722220 ED On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1nccn1C ZINC000880722221 ED On-Demand Anodyne FPR1 45 36 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C1CCN(CC(F)(F)F)CC1 ZINC000880722232 GI On-Demand Anodyne CCR3 23 40 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)C1 ZINC000880722253 EG On-Demand Anodyne EPHX2 25 42 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne INHA 45 37 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne PTAFR 22 42 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne TRPV1 17 52 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne MTNR1A 32 42 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne MTNR1B 32 44 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne MT-ND1 23 40 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne HCRTR2 15 40 COc1cncc(CNC(=O)CCCCc2ccc(OC)c(OC)c2)c1 ZINC000880722293 FG On-Demand Anodyne SUCNR1 26 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN(C2CCC2)C1 ZINC000880722305 FI On-Demand Anodyne RBP4 53 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN(C2CCC2)C1 ZINC000880722306 FI On-Demand Anodyne RBP4 53 39 CON(C)C(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880722430 FG On-Demand Anodyne RBP4 41 39 CC1(CO)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722442 DF On-Demand Anodyne RBP4 46 38 COc1cncc(CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)c1 ZINC000880722447 FD On-Demand Anodyne F2 28 44 COc1cncc(CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)c1 ZINC000880722447 FD On-Demand Anodyne TMPRSS11D 40 32 COc1cncc(CNC(=O)C2CCC(S(C)(=O)=O)CC2)c1 ZINC000880722448 ED On-Demand Anodyne MTNR1A 18 41 CN(C)C(=O)OC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880722467 FH On-Demand Anodyne RBP4 56 39 COc1cncc(CNC(=O)CC[C@@H]2CCc3ccccc32)c1 ZINC000880722470 DG On-Demand Anodyne NQO2 26 51 COc1cncc(CNC(=O)CC[C@@H]2CCc3ccccc32)c1 ZINC000880722470 DG On-Demand Anodyne MTNR1A 34 41 COc1cncc(CNC(=O)CC[C@@H]2CCc3ccccc32)c1 ZINC000880722470 DG On-Demand Anodyne MTNR1B 40 39 COc1cncc(CNC(=O)CC[C@H]2CCc3ccccc32)c1 ZINC000880722471 DG On-Demand Anodyne NQO2 26 51 COc1cncc(CNC(=O)CC[C@H]2CCc3ccccc32)c1 ZINC000880722471 DG On-Demand Anodyne MTNR1A 34 41 COc1cncc(CNC(=O)CC[C@H]2CCc3ccccc32)c1 ZINC000880722471 DG On-Demand Anodyne MTNR1B 40 39 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)[C@H](C)C1 ZINC000880722484 GF On-Demand Anodyne HSD11B1 15 40 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)S1(=O)=O ZINC000880722486 GG On-Demand Anodyne RBP4 54 41 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880722487 GG On-Demand Anodyne RBP4 54 41 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722541 FG On-Demand Anodyne RBP4 44 42 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1(F)F ZINC000880722545 EI On-Demand Anodyne RBP4 55 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1(F)F ZINC000880722546 EI On-Demand Anodyne RBP4 55 41 COc1cncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)c1 ZINC000880722563 GE On-Demand Anodyne Q9NAW4_PLAFA 26 41 COc1cncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)c1 ZINC000880722563 GE On-Demand Anodyne VHL 40 32 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722603 FH On-Demand Anodyne RBP4 53 39 CN(C)C(=O)O[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722619 FG On-Demand Anodyne RBP4 55 40 C[C@@H](NC(=O)c1ncsc1C1CC1)c1nccn1C ZINC000880722658 CE On-Demand Anodyne MAP1 47 35 C[C@H](NC(=O)c1ncsc1C1CC1)c1nccn1C ZINC000880722659 CE On-Demand Anodyne MAP1 47 35 COc1cncc(CNC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880722670 ED On-Demand Anodyne ROCK1 22 46 COc1cncc(CNC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880722670 ED On-Demand Anodyne ROCK2 20 46 COc1cncc(CNC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880722670 ED On-Demand Anodyne DPOL_VZVD 23 40 COc1cncc(CNC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880722670 ED On-Demand Anodyne NAMPT 38 43 COc1ccc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)nc1 ZINC000880722677 GH On-Demand Anodyne PDGFRB 47 39 COc1ccc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)nc1 ZINC000880722677 GH On-Demand Anodyne RBP4 29 41 COc1ccc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)nc1 ZINC000880722677 GH On-Demand Anodyne SCD1 25 40 COc1ccc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)nc1 ZINC000880722677 GH On-Demand Anodyne DGAT1 35 49 COc1ccc(N2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)nc1 ZINC000880722677 GH On-Demand Anodyne NPBWR1 40 36 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)[C@@H](CO)c1ccccc1 ZINC000880722688 FI On-Demand Anodyne NPY5R 28 40 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)[C@H](CO)c1ccccc1 ZINC000880722689 FI On-Demand Anodyne NPY5R 28 40 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C ZINC000880722719 EG On-Demand Anodyne RBP4 53 40 C#CC1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880722748 DH On-Demand Mild RBP4 59 41 C[C@@H]1CC(=O)Nc2ccccc2N1C(=O)CN(C)C(=O)/C=C\c1cccnc1 ZINC000880722759 GE On-Demand Anodyne FABI 44 34 C[C@H]1CC(=O)Nc2ccccc2N1C(=O)CN(C)C(=O)/C=C\c1cccnc1 ZINC000880722760 GE On-Demand Anodyne FABI 44 34 COCCN(Cc1c(C)nn(C)c1C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722778 GH On-Demand Anodyne P2RX7 19 42 COc1ccc([C@@H](CO)CNC(=O)Nc2ccc(F)cc2C(C)(F)F)cc1 ZINC000880722791 GH On-Demand Anodyne TRPV1 19 42 COc1ccc([C@H](CO)CNC(=O)Nc2ccc(F)cc2C(C)(F)F)cc1 ZINC000880722792 GH On-Demand Anodyne TRPV1 19 42 C#C[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722879 DH On-Demand Mild RBP4 57 41 C#C[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880722881 DH On-Demand Mild RBP4 57 41 CCOC[C@H]1CCCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722930 EI On-Demand Anodyne ACKR3 45 32 CN1C(=O)CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1=O ZINC000880722933 EE On-Demand Anodyne P2RX7 21 42 CN1C(=O)CC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1=O ZINC000880722935 EE On-Demand Anodyne P2RX7 21 42 COc1ccc2c(c1)CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)C2 ZINC000880722949 FI On-Demand Anodyne RBP4 22 40 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880722950 EG On-Demand Anodyne CCR3 41 33 C[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)c1nccn1C ZINC000880722982 EG On-Demand Anodyne PDE4D 19 41 C[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)c1nccn1C ZINC000880722986 EG On-Demand Anodyne PDE4D 19 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880723044 FF On-Demand Anodyne RBP4 56 42 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880723045 FF On-Demand Anodyne RBP4 56 42 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)S1(=O)=O ZINC000880723046 FF On-Demand Anodyne RBP4 56 42 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)N1C ZINC000880723047 EG On-Demand Anodyne RBP4 61 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)N1CCO ZINC000880723054 FF On-Demand Anodyne RBP4 56 43 C[C@@H]1C[C@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723061 DG On-Demand Anodyne RBP4 66 45 C[C@H]1C[C@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723063 DG On-Demand Anodyne RBP4 66 45 COc1cncc(CNC(=O)C(C)(C)c2ccc(F)cc2F)c1 ZINC000880723108 DF On-Demand Anodyne GRIN2B 20 44 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723124 EI On-Demand Anodyne CCR3 30 42 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723124 EI On-Demand Anodyne RBP4 41 38 COC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723124 EI On-Demand Anodyne ACKR3 46 32 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723164 DI On-Demand Mild RBP4 61 42 C#CC[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723165 DI On-Demand Mild RBP4 61 42 CC(=O)N[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723173 EF On-Demand Anodyne RBP4 55 41 CC(=O)N[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723174 EF On-Demand Anodyne RBP4 55 41 CO[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880723200 DF On-Demand Anodyne RBP4 53 40 CN(C)C1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723208 EH On-Demand Anodyne EPHX2 50 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880723212 JD On-Demand Anodyne F10 48 33 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880723212 JD On-Demand Anodyne AKR1C3 16 45 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880723212 JD On-Demand Anodyne MERTK 33 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880723212 JD On-Demand Anodyne STAT6 52 35 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880723212 JD On-Demand Anodyne NAMPT 31 41 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880723224 JF On-Demand Anodyne F10 41 47 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880723224 JF On-Demand Anodyne CNR2 21 52 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880723224 JF On-Demand Anodyne PRNP 30 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880723224 JF On-Demand Anodyne STAT6 53 37 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1CO ZINC000880723274 EG On-Demand Anodyne RBP4 53 39 C[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1CO ZINC000880723275 EG On-Demand Anodyne RBP4 53 39 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1CO ZINC000880723276 EG On-Demand Anodyne RBP4 53 39 C[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1CO ZINC000880723277 EG On-Demand Anodyne RBP4 53 39 CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)Cc2cccnc21 ZINC000880723298 FH On-Demand Anodyne RBP4 33 42 Cn1nccc1[C@@H](O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723307 GH On-Demand Anodyne RBP4 47 38 Cn1nccc1[C@H](O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723308 GH On-Demand Anodyne RBP4 47 38 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723368 EG On-Demand Anodyne CHRNA10 57 38 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723368 EG On-Demand Anodyne ACKR3 76 40 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723370 EG On-Demand Anodyne CHRNA10 57 38 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723370 EG On-Demand Anodyne ACKR3 76 40 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723372 FH On-Demand Anodyne EPHX2 24 40 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723374 FH On-Demand Anodyne EPHX2 24 40 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723375 FH On-Demand Anodyne EPHX2 24 40 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723376 FH On-Demand Anodyne EPHX2 24 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@]1(C)CO ZINC000880723500 EG On-Demand Anodyne RBP4 46 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@]1(C)CO ZINC000880723501 EG On-Demand Anodyne RBP4 46 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@]1(C)CO ZINC000880723503 EG On-Demand Anodyne RBP4 46 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@]1(C)CO ZINC000880723504 EG On-Demand Anodyne RBP4 46 39 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)[C@H](CO)Cc1ccccc1 ZINC000880723535 FI On-Demand Anodyne NPY5R 25 42 CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)[C@@H](CO)Cc1ccccc1 ZINC000880723538 FI On-Demand Anodyne NPY5R 25 42 COc1ccccc1[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880723545 GJ On-Demand Anodyne RBP4 72 45 COc1ccccc1[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880723545 GJ On-Demand Anodyne ACKR3 44 30 COc1ccccc1[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880723546 GJ On-Demand Anodyne RBP4 72 45 COc1ccccc1[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCO1 ZINC000880723546 GJ On-Demand Anodyne ACKR3 44 30 CN1C[C@@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1=O ZINC000880723574 EF On-Demand Anodyne P2RX7 20 41 CN1C[C@H](CNC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1=O ZINC000880723576 EF On-Demand Anodyne P2RX7 20 41 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)N1CC#N ZINC000880723578 FG On-Demand Mild RBP4 57 43 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)N1CC#N ZINC000880723582 FG On-Demand Mild RBP4 57 43 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)N1CC#N ZINC000880723584 FG On-Demand Mild RBP4 57 43 CN1CCO[C@@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C[C@@H]21 ZINC000880723605 EE On-Demand Anodyne RBP4 53 40 C[C@@H](CNC(=O)Nc1ccc(F)cc1C(C)(F)F)c1ccccn1 ZINC000880723627 EI On-Demand Anodyne P2RY1 28 42 C[C@H]1C[C@H](CO)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723654 EG On-Demand Anodyne RBP4 59 44 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723672 GH On-Demand Anodyne CACNA1I 52 32 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723672 GH On-Demand Anodyne ACKR3 68 35 CN(C)C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1CN(C)C ZINC000880723675 GG On-Demand Anodyne RBP4 55 41 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC[C@@H]21 ZINC000880723689 EG On-Demand Anodyne RBP4 59 43 CN1CC[C@H]2CN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC[C@H]21 ZINC000880723690 EG On-Demand Anodyne RBP4 59 43 O=C(NOCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880723724 GD On-Demand Anodyne CELA1 19 40 O=C(NOCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880723724 GD On-Demand Anodyne PREP 28 41 O=C(NOCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880723724 GD On-Demand Anodyne LGMN 57 38 O=C(NOCCN1CCCC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880723724 GD On-Demand Anodyne Q9NAW4_PLAFA 36 41 CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCC1(C)C ZINC000880723745 EH On-Demand Anodyne RBP4 43 39 CNC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723806 EF On-Demand Anodyne EPHX2 19 42 CNC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723806 EF On-Demand Anodyne RBP4 55 43 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723818 FF On-Demand Anodyne RBP4 46 39 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723819 FF On-Demand Anodyne RBP4 46 39 CCn1c(O)nnc1C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880723841 GH On-Demand Anodyne RBP4 44 38 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@@](=O)C1 ZINC000880723845 EG On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@@](=O)C1 ZINC000880723846 EG On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@](=O)C1 ZINC000880723847 EG On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[S@](=O)C1 ZINC000880723848 EG On-Demand Anodyne RBP4 53 40 CN1CCC[C@@H](CCNC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880723867 EH On-Demand Anodyne CCR3 96 42 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)[C@@H]1O ZINC000880723875 EG On-Demand Anodyne RBP4 57 44 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)C1O ZINC000880723876 EG On-Demand Anodyne RBP4 57 44 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)C1O ZINC000880723877 EG On-Demand Anodyne RBP4 57 44 O=C(NOCCN1CCCC1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880723899 EC On-Demand Anodyne PLD2 40 37 CCc1nccn1C[C@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723905 GI On-Demand Anodyne ACKR3 44 31 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)C1(F)F ZINC000880723907 FJ On-Demand Anodyne RBP4 59 45 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)C1(F)F ZINC000880723908 FJ On-Demand Anodyne RBP4 59 45 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C)C1(F)F ZINC000880723909 FJ On-Demand Anodyne RBP4 59 45 Cn1cc(CCNC(=O)Nc2ccc(F)cc2C(C)(F)F)c2cccnc21 ZINC000880723930 GI On-Demand Anodyne P2RY1 34 40 COC[C@@H]1CCCN1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723942 EG On-Demand Anodyne CCR3 23 41 COC[C@@H]1CCCN1NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880723942 EG On-Demand Anodyne ACKR3 65 34 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H](C)O1 ZINC000880723980 EH On-Demand Anodyne RBP4 57 43 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H]1C ZINC000880723991 FH On-Demand Anodyne RBP4 47 39 Cc1nnc([C@@H]2CCCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)o1 ZINC000880724097 FI On-Demand Anodyne RBP4 47 38 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880724111 JF On-Demand Anodyne F10 41 46 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880724111 JF On-Demand Anodyne LCK 15 40 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880724111 JF On-Demand Anodyne MAPK14 16 40 CCN(CC)S(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880724111 JF On-Demand Anodyne STAT6 52 34 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C(=O)N1CCOCC1 ZINC000880724142 GF On-Demand Anodyne RBP4 55 40 COC(=O)[C@H]1C[C@@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724160 FE On-Demand Anodyne RBP4 48 41 COC(=O)[C@@H]1C[C@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724161 FE On-Demand Anodyne RBP4 48 41 COC(=O)[C@@H]1C[C@@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724162 FE On-Demand Anodyne RBP4 48 41 COC(=O)[C@H]1C[C@H](O)CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724163 FE On-Demand Anodyne RBP4 48 41 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724183 EH On-Demand Anodyne RBP4 48 39 CC(C)[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1C ZINC000880724222 EH On-Demand Anodyne RBP4 59 41 Cn1ncc(Br)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724227 GH On-Demand Anodyne HTR2A 20 42 Cn1ncc(Br)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724227 GH On-Demand Anodyne P2RX7 15 42 C=CC[C@@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724263 DI On-Demand Mild RBP4 53 39 C=CC[C@H]1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724264 DI On-Demand Mild RBP4 53 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C(N)=O)O1 ZINC000880724266 EE On-Demand Anodyne RBP4 53 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C(N)=O)O1 ZINC000880724267 EE On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H](C(N)=O)O1 ZINC000880724268 EE On-Demand Anodyne RBP4 53 40 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C(N)=O)O1 ZINC000880724269 EE On-Demand Anodyne RBP4 53 40 CCC1(N(C)C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724273 FI On-Demand Anodyne RBP4 54 40 CCC1(N(C)C)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724273 FI On-Demand Anodyne TRPM8 17 40 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@H]1C1CC1 ZINC000880724345 FH On-Demand Anodyne RBP4 54 40 CCO[C@H]1C[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724355 DH On-Demand Anodyne EPHX2 40 37 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724356 DH On-Demand Anodyne EPHX2 40 37 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C[C@@H](C)C1=O ZINC000880724362 EH On-Demand Anodyne RBP4 57 43 COCC1CCC(NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724396 EI On-Demand Anodyne EPHX2 49 39 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724397 GJ On-Demand Anodyne CACNA1H 51 36 COC[C@@H]1CCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724437 DH On-Demand Anodyne ACKR3 69 36 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)CC2 ZINC000880724450 GI On-Demand Anodyne RBP4 40 38 C[C@H](Cc1ccccn1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724457 EI On-Demand Anodyne P2RY1 23 41 C[C@@H](Cc1ccccn1)NC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724460 EI On-Demand Anodyne P2RY1 23 41 CCn1nc(C)c(CN(C)C(=O)Nc2ccc(F)cc2C(C)(F)F)c1C ZINC000880724479 FI On-Demand Anodyne P2RX7 21 47 CN1CCN(C2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)CC1 ZINC000880724488 GG On-Demand Anodyne RBP4 42 39 CN1CCN(C2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)CC2)CC1 ZINC000880724488 GG On-Demand Anodyne L3MBTL3 67 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880724645 GE On-Demand Anodyne HSD11B1 22 47 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880724645 GE On-Demand Anodyne RBP4 52 39 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724668 FG On-Demand Anodyne ACKR3 46 33 COc1ccc2c(c1)CC[C@H](C(=O)NOCCN1CCCC1=O)C2 ZINC000880724695 ED On-Demand Anodyne NQO2 21 41 COc1ccc2c(c1)CC[C@H](C(=O)NOCCN1CCCC1=O)C2 ZINC000880724695 ED On-Demand Anodyne MTNR1A 25 44 Cn1ncc(C2CC2)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724698 FH On-Demand Anodyne P2RX7 20 40 O=C(Cc1ccc2cccnc2c1)NC1CSC1 ZINC000880724734 CE On-Demand Anodyne CDK5 18 45 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880724743 GI On-Demand Anodyne P2RX7 21 43 C=CCCONC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880724768 GE On-Demand Mild GPR119 33 42 Cn1nnnc1C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724774 FF On-Demand Anodyne CCR3 42 31 Cn1nnnc1C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724774 FF On-Demand Anodyne RBP4 53 38 O=C(NC1CSC1)c1cccn2nccc12 ZINC000880724775 BD On-Demand Anodyne JAK3 18 43 O=C(NC1CSC1)c1cccn2nccc12 ZINC000880724775 BD On-Demand Anodyne TYK2 21 43 O=C(NC1CSC1)c1cccn2nccc12 ZINC000880724775 BD On-Demand Anodyne EPHB3 34 42 C=CCCONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880724792 CE On-Demand Mild NQO2 24 40 C=CCCONC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880724792 CE On-Demand Mild MTNR1A 35 42 C=CCCONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880724793 CE On-Demand Mild NQO2 24 40 C=CCCONC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880724793 CE On-Demand Mild MTNR1A 35 42 C=CCCONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880724799 EE On-Demand Mild PREP 24 42 C=CCCONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880724799 EE On-Demand Mild LGMN 59 37 C=CCCONC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880724799 EE On-Demand Mild Q9NAW4_PLAFA 38 45 C#CCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724825 EG On-Demand Mild S1PR2 28 40 C#CCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724825 EG On-Demand Mild RBP4 45 37 C[C@@H](CCc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880724833 CF On-Demand Anodyne LEF 48 36 C[C@@H](CCc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880724833 CF On-Demand Anodyne BIRC2 21 41 C[C@H](CCc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880724834 CF On-Demand Anodyne LEF 48 36 C[C@H](CCc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880724834 CF On-Demand Anodyne BIRC2 21 41 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC3CSC3)ccn2)CC1 ZINC000880724840 GD On-Demand Anodyne GPR119 43 47 CC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724847 EH On-Demand Anodyne RBP4 57 40 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724855 FH On-Demand Anodyne RBP4 44 42 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1ccc(F)cc1C(C)(F)F)CC2 ZINC000880724885 GI On-Demand Anodyne TRPM8 23 40 COc1cc(I)ccc1C(=O)NC1CSC1 ZINC000880724886 EE On-Demand Anodyne DRD2 21 40 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne PIK3CA 41 39 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne CPT1A 82 45 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne PRNP 50 43 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne JAK2 15 42 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne MTOR 48 39 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne MCHR1 18 44 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne LUCI_LUCLA 34 40 O=C(COc1ccc(-c2ccccc2)cc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880724915 GH On-Demand Anodyne STAT6 67 41 O=C(NC1CSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880724929 CF On-Demand Anodyne PDE4D 18 44 O=C(NC1CSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880724929 CF On-Demand Anodyne EZH2 42 40 Cc1csc([C@H]2CCN(C(=O)Nc3ccc(F)cc3C(C)(F)F)C2)n1 ZINC000880724947 FJ On-Demand Anodyne RBP4 55 38 O=C(NC1CSC1)c1cnn(-c2cccc(F)c2)c1C(F)(F)F ZINC000880724949 EF On-Demand Anodyne MAPK14 16 44 O=C(NC1CSC1)c1cnn(-c2cccc(F)c2)c1C(F)(F)F ZINC000880724949 EF On-Demand Anodyne MST1R 40 37 COc1ccc(CN(CCO)C(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880724951 GH On-Demand Anodyne ROCK2 15 43 CONC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880724957 FF On-Demand Anodyne RBP4 44 40 O=C(NC1CSC1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880724962 CF On-Demand Anodyne CHRNA7 43 37 O=C(NC1CSC1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880724962 CF On-Demand Anodyne C3AR1 51 50 O=C(NC1CSC1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880724963 CF On-Demand Anodyne CHRNA7 43 37 O=C(NC1CSC1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880724963 CF On-Demand Anodyne C3AR1 51 50 Cn1c(S)nnc1[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724964 GH On-Demand Anodyne RBP4 46 38 Cn1c(S)nnc1[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880724965 GH On-Demand Anodyne RBP4 46 38 C[C@H](CC(=O)NC1CSC1)NC(=O)OC(C)(C)C ZINC000880724986 CD On-Demand Anodyne CTSK 15 40 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne CELA1 19 40 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne GRIN2B 18 40 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne PREP 28 47 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne LGMN 60 39 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne SLC12A5 42 34 O=C(NC1CSC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880725012 ED On-Demand Anodyne Q9NAW4_PLAFA 42 48 COC(=O)c1cc(C(=O)NC2CSC2)ccc1C ZINC000880725017 CD On-Demand Anodyne MAPK11 29 40 COC(=O)c1cc(C(=O)NC2CSC2)ccc1C ZINC000880725017 CD On-Demand Anodyne MAPK14 39 40 CN1CCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC1(C)C ZINC000880725036 EG On-Demand Anodyne RBP4 40 39 O=C(NC1CSC1)c1ccc(OCc2ccccc2)cn1 ZINC000880725049 DF On-Demand Anodyne LTA4H 19 40 O=C(NC1CSC1)c1ccc(OCc2ccccc2)cn1 ZINC000880725049 DF On-Demand Anodyne SLC6A5 36 43 O=C(NC1CSC1)c1ccc(OCc2ccccc2)cn1 ZINC000880725049 DF On-Demand Anodyne NAAA 17 43 COc1ccc(CN(CCO)C(=O)Nc2ccc(F)cc2C(C)(F)F)cc1 ZINC000880725065 GH On-Demand Anodyne SOAT1 17 48 O=C(CCc1ccc(N2CCCS2(=O)=O)cc1)NC1CSC1 ZINC000880725071 ED On-Demand Anodyne CDK1 17 40 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880725092 GJ On-Demand Anodyne RBP4 47 39 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880725093 GJ On-Demand Anodyne RBP4 47 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880725094 GJ On-Demand Anodyne RBP4 47 39 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880725095 GJ On-Demand Anodyne RBP4 47 39 O=C(NC1CSC1)c1cccn(C2CC2)c1=O ZINC000880725104 CD On-Demand Anodyne POLR1A 25 40 NC(=O)[C@@H]1CC[C@H](C(=O)NC2CSC2)N1Cc1ccccc1 ZINC000880725117 DC On-Demand Anodyne SIGMAR1 19 42 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725147 FI On-Demand Anodyne EPHX2 29 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880725198 DD On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880725198 DD On-Demand Anodyne CTSK 15 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880725199 DD On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880725199 DD On-Demand Anodyne CTSK 15 49 COc1ccccc1-c1ccc(C(=O)NC2CSC2)s1 ZINC000880725256 DG On-Demand Anodyne MAPK11 20 42 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1c1ccncc1 ZINC000880725257 GI On-Demand Anodyne RBP4 52 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1c1ccncc1 ZINC000880725258 GI On-Demand Anodyne RBP4 52 34 O=C(CCc1cccc2ccccc12)NC1CSC1 ZINC000880725261 CG On-Demand Anodyne MTNR1A 27 44 O=C(CCc1cccc2ccccc12)NC1CSC1 ZINC000880725261 CG On-Demand Anodyne TNKS 57 32 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725285 FH On-Demand Anodyne RBP4 52 33 O=C(NC1CSC1)c1ccc(OC(F)F)c(Br)c1 ZINC000880725287 EF On-Demand Anodyne EZH2 27 40 O=C(Cc1cccc2ncccc12)NC1CSC1 ZINC000880725319 CE On-Demand Anodyne TNKS 41 35 COc1ccc(Nc2ccc(C(=O)NC3CSC3)cc2)c(OC)c1 ZINC000880725325 EG On-Demand Anodyne PDGFRA 16 41 COc1ccc(Nc2ccc(C(=O)NC3CSC3)cc2)c(OC)c1 ZINC000880725325 EG On-Demand Anodyne AKR1C3 28 45 COc1ccc(Nc2ccc(C(=O)NC3CSC3)cc2)c(OC)c1 ZINC000880725325 EG On-Demand Anodyne AKR1C2 53 45 O=C(CCNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880725331 DD On-Demand Anodyne CCKAR 15 53 O=C(CCNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880725331 DD On-Demand Anodyne PYGL 79 43 O=C(CCNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880725331 DD On-Demand Anodyne PLD1 31 44 O=C(CCNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880725331 DD On-Demand Anodyne PYGM 29 43 O=C(CCNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880725331 DD On-Demand Anodyne PLD2 32 45 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725337 EE On-Demand Anodyne EPHX2 29 43 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880725338 EH On-Demand Anodyne RBP4 54 41 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(F)cc2C(C)(F)F)C1 ZINC000880725339 EH On-Demand Anodyne RBP4 54 41 Cc1csc([C@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)n1 ZINC000880725357 FJ On-Demand Anodyne RBP4 56 37 O=C(NC1CSC1)c1cn2c(n1)COCC2 ZINC000880725359 BC On-Demand Anodyne BLAT-6 17 42 CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C(=O)NC2CSC2)C1 ZINC000880725363 DD On-Demand Anodyne GPR119 20 42 CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C(=O)NC2CSC2)C1 ZINC000880725364 DD On-Demand Anodyne GPR119 20 42 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C(=O)NC2CSC2)C1 ZINC000880725365 DD On-Demand Anodyne GPR119 20 42 CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C(=O)NC2CSC2)C1 ZINC000880725366 DD On-Demand Anodyne GPR119 20 42 COCC1CC(NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725381 DG On-Demand Anodyne EPHX2 28 41 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne PGC 56 37 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne PAPA1_CARPA 55 52 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CYSP_TRYCR 46 37 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CCKAR 50 42 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CTSK 26 47 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CTSL 63 52 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CACNA1B 26 42 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne TACR3 15 41 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne REN 77 44 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CTSS 39 52 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CAPN1 19 41 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne CTSV 48 35 COc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725383 FE On-Demand Anodyne FPR1 64 43 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne PGC 56 37 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne PAPA1_CARPA 55 52 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CYSP_TRYCR 46 37 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CCKAR 50 42 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CTSK 26 47 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CTSL 63 52 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CACNA1B 26 42 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne TACR3 15 41 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne REN 77 44 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CTSS 39 52 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CAPN1 19 41 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne CTSV 48 35 COc1cccc(C[C@@H](NC(=O)OC(C)(C)C)C(=O)NC2CSC2)c1 ZINC000880725384 FE On-Demand Anodyne FPR1 64 43 CC(=O)N1CCC[C@@H]1C(=O)NC1CSC1 ZINC000880725385 BC On-Demand Anodyne CELA1 30 45 O=C(NC1CSC1)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725391 CD On-Demand Anodyne SLC18A3 18 43 O=C(NC1CSC1)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725391 CD On-Demand Anodyne EPHX2 33 67 O=C(NC1CSC1)[C@@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725391 CD On-Demand Anodyne L3MBTL3 77 40 O=C(NC1CSC1)[C@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725392 CD On-Demand Anodyne SLC18A3 18 43 O=C(NC1CSC1)[C@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725392 CD On-Demand Anodyne EPHX2 33 67 O=C(NC1CSC1)[C@H]1CCN(C(=O)c2ccccc2)C1 ZINC000880725392 CD On-Demand Anodyne L3MBTL3 77 40 CN1CC[C@H]2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC[C@@H]21 ZINC000880725400 EG On-Demand Anodyne RBP4 57 36 CN1CC[C@H]2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC[C@H]21 ZINC000880725402 EG On-Demand Anodyne RBP4 57 36 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)Cc2cccnc21 ZINC000880725422 FH On-Demand Anodyne RBP4 16 41 Cc1cc(C(=O)NC2CSC2)ccc1OC(F)(F)F ZINC000880725424 CF On-Demand Anodyne MAPK13 50 35 Cc1cc(C(=O)NC2CSC2)ccc1OC(F)(F)F ZINC000880725424 CF On-Demand Anodyne EZH2 26 41 O=C(NC1CSC1)[C@H]1COc2cc(F)ccc2C1 ZINC000880725428 CD On-Demand Anodyne ROCK2 17 42 O=C(NC1CSC1)[C@@H]1COc2cc(F)ccc2C1 ZINC000880725429 CD On-Demand Anodyne ROCK2 17 42 O=C(NC1CSC1)c1ccc(SC(F)(F)F)nc1 ZINC000880725434 CF On-Demand Anodyne HPGDS 38 41 O=C(NC1CSC1)c1cc2ccnc(Cl)c2s1 ZINC000880725443 CF On-Demand Anodyne TYK2 41 32 CCN1CC[C@@H]1CNC(=O)Nc1ccc(F)cc1C(C)(F)F ZINC000880725463 DG On-Demand Anodyne CCR3 40 37 C[C@@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1c1ccncc1 ZINC000880725468 GI On-Demand Anodyne RBP4 47 38 C[C@H]1CN(C(=O)Nc2ccc(F)cc2C(C)(F)F)CCN1c1ccncc1 ZINC000880725469 GI On-Demand Anodyne RBP4 47 38 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(F)cc2C(C)(F)F)CC1 ZINC000880725490 DI On-Demand Mild EPHX2 42 43 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(F)F ZINC000880725506 CH On-Demand Anodyne DAC 22 40 COc1ccc2c(c1)CC[C@H]2C(=O)NC1CSC1 ZINC000880725512 CD On-Demand Anodyne NQO2 24 40 COc1ccc2c(c1)CC[C@H]2C(=O)NC1CSC1 ZINC000880725512 CD On-Demand Anodyne PPARD 30 41 COc1ccc2c(c1)CC[C@H]2C(=O)NC1CSC1 ZINC000880725512 CD On-Demand Anodyne MTNR1A 24 41 COc1ccc(-c2cncc(C(=O)NC3CSC3)c2)c(C)c1 ZINC000880725529 DF On-Demand Anodyne MAPK14 20 44 COc1ccc(-c2cncc(C(=O)NC3CSC3)c2)c(C)c1 ZINC000880725529 DF On-Demand Anodyne CYP11B2 24 43 Cc1ccc2nc(C(=O)NC3CSC3)cn2c1 ZINC000880725531 BD On-Demand Anodyne MAP3K5 36 42 O=C(Cc1ccc(F)c(Cl)c1)NC1CSC1 ZINC000880725586 CE On-Demand Anodyne LUXR 40 40 O=C(NC1CSC1)c1cc(C(F)(F)F)ccc1Cl ZINC000880725593 CG On-Demand Anodyne CCR2 21 40 CCOC(=O)[C@@]1(C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880725599 FG On-Demand Anodyne EPHX2 20 41 C[C@@H](O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725608 EH On-Demand Anodyne RBP4 56 40 O=C(CCCc1ccc2c(c1)OCCCO2)NC1CSC1 ZINC000880725614 DE On-Demand Anodyne LUXR 46 47 O=C(NC1CSC1)c1cccc(Cn2cncn2)c1 ZINC000880725617 CD On-Demand Anodyne HIS3 50 35 CONC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725620 FF On-Demand Anodyne RBP4 42 42 CS(=O)(=O)N1CCC[C@H](C(=O)NC2CSC2)C1 ZINC000880725645 CB On-Demand Anodyne EPHX2 17 40 CC(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725662 EH On-Demand Anodyne RBP4 53 35 CC(=O)[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725663 EH On-Demand Anodyne RBP4 53 35 C[C@@H](CC(=O)NC1CSC1)NC(=O)OC(C)(C)C ZINC000880725665 CD On-Demand Anodyne CTSK 15 40 Cn1ncc(Br)c1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880725671 GH On-Demand Anodyne HTR2A 17 40 COC(=O)C1=NO[C@@]2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)C1 ZINC000880725682 GF On-Demand Anodyne EPHX2 31 42 COC(=O)C1=NO[C@@]2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)C1 ZINC000880725682 GF On-Demand Anodyne TRPM8 28 41 COC(=O)C1=NO[C@]2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)C1 ZINC000880725683 GF On-Demand Anodyne EPHX2 31 42 COC(=O)C1=NO[C@]2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)C1 ZINC000880725683 GF On-Demand Anodyne TRPM8 28 41 O=C(NC1CSC1)C1CCc2ccccc2CC1 ZINC000880725688 CE On-Demand Anodyne EPHX2 15 40 CC[C@@H](Nc1cccnc1Cl)C(=O)NC1CSC1 ZINC000880725709 CE On-Demand Anodyne G2YM83_BOTF4 70 38 CC[C@H](Nc1cccnc1Cl)C(=O)NC1CSC1 ZINC000880725710 CE On-Demand Anodyne G2YM83_BOTF4 70 38 O=C(NC1CSC1)c1ccc(C(=O)N2CCOCC2)cc1 ZINC000880725713 DD On-Demand Anodyne EPHX2 15 49 O=C(NC1CSC1)c1ccc(C(=O)N2CCOCC2)cc1 ZINC000880725713 DD On-Demand Anodyne L3MBTL3 59 37 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS1 ZINC000880725715 DH On-Demand Anodyne RBP4 53 34 O=C(Cc1cccc2cnccc12)NC1CSC1 ZINC000880725733 CE On-Demand Anodyne TRPV1 19 42 O=C(Cc1cccc2cnccc12)NC1CSC1 ZINC000880725733 CE On-Demand Anodyne CDK5 25 41 Cn1nnnc1C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725788 FF On-Demand Anodyne RBP4 54 40 CC(C)[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1C ZINC000880725803 EH On-Demand Anodyne RBP4 58 35 Cn1c(S)nnc1[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725806 GH On-Demand Anodyne RBP4 51 32 Cn1c(S)nnc1[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725807 GH On-Demand Anodyne RBP4 51 32 CC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725813 EH On-Demand Anodyne EPHX2 22 42 CC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725813 EH On-Demand Anodyne RBP4 57 41 O=C(NC1CSC1)[C@@H]1C[C@H]1c1ccsc1 ZINC000880725824 BE On-Demand Anodyne NPBWR1 79 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880725854 GJ On-Demand Anodyne RBP4 47 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880725855 GJ On-Demand Anodyne RBP4 47 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880725856 GJ On-Demand Anodyne RBP4 47 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880725857 GJ On-Demand Anodyne RBP4 47 35 Cc1nn(C2CCOCC2)c(C)c1C(=O)NC1CSC1 ZINC000880725867 CD On-Demand Anodyne FPR1 15 41 O=C(CCc1ccc(Cl)c(F)c1)NC1CSC1 ZINC000880725877 CF On-Demand Anodyne ENV 41 37 O=C(CCc1ccc(Cl)c(F)c1)NC1CSC1 ZINC000880725877 CF On-Demand Anodyne LUXR 35 40 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880725918 DI On-Demand Mild EPHX2 41 48 CN(C)[C@@H](C(=O)NC1CSC1)c1ccc(Cl)cc1 ZINC000880725925 CE On-Demand Anodyne UTS2 40 33 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880725928 GI On-Demand Anodyne TRPV1 16 45 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880725928 GI On-Demand Anodyne P2RX7 27 48 COc1ccccc1Cn1cnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880725955 FF On-Demand Anodyne DRD4 18 40 COc1ccccc1Cn1cnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880725955 FF On-Demand Anodyne NR1I2 42 32 COc1ccccc1Cn1cnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880725955 FF On-Demand Anodyne HPGD 23 42 C=CC[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725966 DI On-Demand Mild RBP4 46 35 C=CC[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880725967 DI On-Demand Mild RBP4 46 35 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)C[C@H]1C(F)(F)F ZINC000880725975 EF On-Demand Anodyne DRD4 24 41 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)C[C@H]1C(F)(F)F ZINC000880725975 EF On-Demand Anodyne SIGMAR1 26 43 O=C(NC1CSC1)[C@H]1Cc2ccccc2CO1 ZINC000880726018 BD On-Demand Anodyne PTPRF 43 33 O=C(NC1CSC1)[C@@H]1Cc2ccccc2CO1 ZINC000880726019 BD On-Demand Anodyne PTPRF 43 33 Cn1cc([C@@H]2CN(Cc3ccccc3)C[C@H]2C(=O)NC2CSC2)cn1 ZINC000880726024 FD On-Demand Anodyne SIGMAR1 16 42 Cn1cc([C@@H]2CN(Cc3ccccc3)C[C@H]2C(=O)NC2CSC2)cn1 ZINC000880726024 FD On-Demand Anodyne PDE1C 46 39 O=C(NC1CSC1)c1ccnc(N2CCOCC2)n1 ZINC000880726040 CC On-Demand Anodyne PIK3CA 21 40 Cn1nc(C(=O)NC2CSC2)c2ccccc21 ZINC000880726045 BD On-Demand Anodyne HTR3A 24 65 Cn1nc(C(=O)NC2CSC2)c2ccccc21 ZINC000880726045 BD On-Demand Anodyne HTR4 25 42 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccncc1 ZINC000880726054 FF On-Demand Anodyne SIGMAR1 22 42 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCC1(C)C ZINC000880726076 EH On-Demand Anodyne RBP4 45 35 COc1ccccc1[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880726078 GJ On-Demand Anodyne RBP4 56 43 COc1ccccc1[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880726079 GJ On-Demand Anodyne RBP4 56 43 O=C(COc1ccc(Br)cn1)NC1CSC1 ZINC000880726084 DD On-Demand Anodyne TRAR 32 40 C[C@@H](CNC(=O)Nc1cccc(F)c1C(C)(F)F)c1ccncc1 ZINC000880726127 EI On-Demand Anodyne TRPV1 17 49 C[C@H]1c2ccccc2CN1C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880726132 EK On-Demand Anodyne TRPM8 31 45 CC(C)(C)OC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880726146 DE On-Demand Anodyne DRD4 43 33 CC(C)(C)OC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880726146 DE On-Demand Anodyne PLA2G4B 36 41 COC[C@]1(C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880726180 EG On-Demand Anodyne EPHX2 21 40 COC[C@@]1(C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880726181 EG On-Demand Anodyne EPHX2 21 40 O=C(NC1CSC1)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880726192 FD On-Demand Anodyne EPHX2 32 49 O=C(NC1CSC1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880726193 FD On-Demand Anodyne EPHX2 32 49 Cn1nccc1[C@@H](O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726208 GH On-Demand Anodyne RBP4 45 38 Cn1nccc1[C@H](O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726209 GH On-Demand Anodyne RBP4 45 38 CCC1(N(C)C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726235 FI On-Demand Anodyne CACNA1H 40 32 CCC1(N(C)C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726235 FI On-Demand Anodyne RBP4 54 34 CCC1(N(C)C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726235 FI On-Demand Anodyne TRPM8 30 41 O=C(NC1CSC1)c1cccc(Nc2nccc(C(F)(F)F)n2)c1 ZINC000880726238 FG On-Demand Anodyne ABL1 16 41 O=C(NC1CSC1)c1cccc(Nc2nccc(C(F)(F)F)n2)c1 ZINC000880726238 FG On-Demand Anodyne SYK 20 42 O=C(NC1CSC1)c1cccc(Nc2nccc(C(F)(F)F)n2)c1 ZINC000880726238 FG On-Demand Anodyne BTK 28 41 O=C(NC1CSC1)c1cccc(Nc2nccc(C(F)(F)F)n2)c1 ZINC000880726238 FG On-Demand Anodyne TXK 47 39 O=C(NC1CSC1)c1cccc(Nc2nccc(C(F)(F)F)n2)c1 ZINC000880726238 FG On-Demand Anodyne SMG1 45 33 O=C(Cc1ccc(O)c(Cl)c1)NC1CSC1 ZINC000880726246 CD On-Demand Anodyne NCE103 20 55 O=C(Cc1ccc(O)c(Cl)c1)NC1CSC1 ZINC000880726246 CD On-Demand Anodyne P96878_MYCTU 15 52 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)C[C@H]1c1nccs1 ZINC000880726275 FF On-Demand Anodyne SIGMAR1 18 40 O=C(OCc1ccccc1)N1CC(O)(C(=O)NC2CSC2)C1 ZINC000880726295 DC On-Demand Anodyne GRIN2B 24 44 O=C(OCc1ccccc1)N1CC(O)(C(=O)NC2CSC2)C1 ZINC000880726295 DC On-Demand Anodyne PREP 25 42 O=C(OCc1ccccc1)N1CC(O)(C(=O)NC2CSC2)C1 ZINC000880726295 DC On-Demand Anodyne SLC12A5 65 38 COc1ccc(OC(C)(C)C(=O)NC2CSC2)cc1 ZINC000880726303 CE On-Demand Anodyne HSD11B1 16 53 CN1CCN(C2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)CC1 ZINC000880726305 GG On-Demand Anodyne L3MBTL3 57 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C(N)=O)O1 ZINC000880726325 EE On-Demand Anodyne RBP4 51 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C(N)=O)O1 ZINC000880726326 EE On-Demand Anodyne RBP4 51 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C(N)=O)O1 ZINC000880726327 EE On-Demand Anodyne RBP4 51 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C(N)=O)O1 ZINC000880726328 EE On-Demand Anodyne RBP4 51 33 O=C(NC1CSC1)c1ccccc1COCc1ccccc1 ZINC000880726331 DG On-Demand Anodyne SLC6A5 41 36 CS[C@@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726352 DH On-Demand Anodyne EPHX2 15 42 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(Cl)c(Cl)c1 ZINC000880726370 FF On-Demand Anodyne F10 48 51 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(Cl)c(Cl)c1 ZINC000880726370 FF On-Demand Anodyne PRNP 46 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(Cl)c(Cl)c1 ZINC000880726370 FF On-Demand Anodyne MAPK10 42 39 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(Cl)c(Cl)c1 ZINC000880726370 FF On-Demand Anodyne AKR1C3 17 50 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(Cl)c(Cl)c1 ZINC000880726370 FF On-Demand Anodyne STAT6 56 36 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne FKBP1A 16 41 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne TBXAS1 76 55 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne PTAFR 39 45 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne CHRNA7 46 37 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne C3AR1 42 43 O=C(CCCc1cccnc1)NC1CSC1 ZINC000880726373 BD On-Demand Anodyne NAMPT 28 40 O=C(NC1CSC1)c1ccn2nnnc2c1 ZINC000880726381 BB On-Demand Anodyne MAPK13 56 34 O=C(NC1CSC1)[C@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726402 EE On-Demand Anodyne GRIN2B 19 42 O=C(NC1CSC1)[C@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726402 EE On-Demand Anodyne SLC12A5 58 38 O=C(NC1CSC1)[C@@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726403 EE On-Demand Anodyne GRIN2B 19 42 O=C(NC1CSC1)[C@@H]1C[C@@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726403 EE On-Demand Anodyne SLC12A5 58 38 O=C(NC1CSC1)[C@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726404 EE On-Demand Anodyne GRIN2B 19 42 O=C(NC1CSC1)[C@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726404 EE On-Demand Anodyne SLC12A5 58 38 O=C(NC1CSC1)[C@@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726405 EE On-Demand Anodyne GRIN2B 19 42 O=C(NC1CSC1)[C@@H]1C[C@]12CCN(C(=O)OCc1ccccc1)C2 ZINC000880726405 EE On-Demand Anodyne SLC12A5 58 38 O=C(NC1CSC1)c1c(Cl)nc2cc(Cl)ccn12 ZINC000880726406 DE On-Demand Anodyne MAPK13 45 33 CN(C)C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1CN(C)C ZINC000880726408 GG On-Demand Anodyne RBP4 53 34 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS1(=O)=O ZINC000880726440 FF On-Demand Anodyne RBP4 53 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)C1(F)F ZINC000880726500 FJ On-Demand Anodyne RBP4 61 37 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)C1(F)F ZINC000880726501 FJ On-Demand Anodyne RBP4 61 37 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)C1(F)F ZINC000880726502 FJ On-Demand Anodyne RBP4 61 37 O=C(NC1CSC1)c1cccc(Cn2ccnn2)c1 ZINC000880726543 CD On-Demand Anodyne DRD4 15 42 COc1cccc(C(=O)NC2CSC2)c1C ZINC000880726544 BD On-Demand Anodyne DRD2 17 41 COc1cccc(C(=O)NC2CSC2)c1C ZINC000880726544 BD On-Demand Anodyne KCNK3 48 43 COc1cccc(C(=O)NC2CSC2)c1C ZINC000880726544 BD On-Demand Anodyne KCNK9 45 43 CC(C)(C)OC(=O)N1CCC(n2nncc2C(=O)NC2CSC2)CC1 ZINC000880726558 FD On-Demand Anodyne GPR119 41 41 O=C(NC1CSC1)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880726560 ED On-Demand Anodyne AKR1C3 50 37 O=C(NC1CSC1)c1cccc(S(=O)(=O)C(F)(F)F)c1 ZINC000880726560 ED On-Demand Anodyne SFRP1 43 38 O=C(NC1CSC1)c1coc2ccc(Cl)cc12 ZINC000880726564 CF On-Demand Anodyne INHA 41 31 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne ALOX5 17 55 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne MAOB 28 45 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne LTA4H 57 50 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne SIGMAR1 16 47 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne ADAM17 44 45 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne FAAH 17 42 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne SLC6A5 38 44 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne EPHX2 16 47 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne ACE2 15 40 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne NAAA 21 47 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne TAAR1 15 44 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne FFAR1 54 50 O=C(Cc1ccc(OCc2ccccc2)cc1)NC1CSC1 ZINC000880726569 DG On-Demand Anodyne FFAR4 48 40 O=C(NC1CSC1)c1cnn2cccc(Cl)c12 ZINC000880726574 CD On-Demand Anodyne EPHB3 43 45 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1CO ZINC000880726583 EG On-Demand Anodyne RBP4 52 36 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1CO ZINC000880726584 EG On-Demand Anodyne RBP4 52 36 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1CO ZINC000880726585 EG On-Demand Anodyne RBP4 52 36 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1CO ZINC000880726586 EG On-Demand Anodyne RBP4 52 36 O=C(NC1CSC1)c1cccc(N2CCCC2)c1 ZINC000880726614 CE On-Demand Anodyne DRD4 42 33 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726615 EG On-Demand Anodyne EPHX2 25 42 CCC(CC)C(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726654 GI On-Demand Anodyne EPHX2 15 42 COc1cccc(C(=O)NC2CSC2)c1OC(C)C ZINC000880726659 CE On-Demand Anodyne DRD2 15 44 COc1cccc(C(=O)NC2CSC2)c1OC(C)C ZINC000880726659 CE On-Demand Anodyne KDR 21 40 COc1cccc(C(=O)NC2CSC2)c1OC(C)C ZINC000880726659 CE On-Demand Anodyne KCNK3 40 40 COc1cccc(C(=O)NC2CSC2)c1OC(C)C ZINC000880726659 CE On-Demand Anodyne KCNK9 35 40 O=C(NC1CSC1)c1cccn2cc(C(F)(F)F)nc12 ZINC000880726672 DE On-Demand Anodyne POLR1A 25 40 O=C(NC1CSC1)c1ccc(C(F)(F)Br)nc1 ZINC000880726690 DE On-Demand Anodyne HPGDS 36 40 CC(C)(C)OC(=O)N1CCC(c2cc(C(=O)NC3CSC3)on2)CC1 ZINC000880726693 FF On-Demand Anodyne GPR119 42 38 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726738 FF On-Demand Anodyne EPHX2 30 42 CO[C@@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726748 DG On-Demand Anodyne EPHX2 33 42 COC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880726766 FF On-Demand Anodyne RBP4 43 32 O=C(NC1CSC1)c1ccc(CF)cc1 ZINC000880726768 BE On-Demand Anodyne SSTR3 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@H](C(=O)NC2CSC2)O1 ZINC000880726775 DD On-Demand Anodyne DRD4 26 40 C[C@@H]1CN(Cc2ccccc2)C[C@H](C(=O)NC2CSC2)O1 ZINC000880726775 DD On-Demand Anodyne SIGMAR1 29 43 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS1(=O)=O ZINC000880726859 FF On-Demand Anodyne RBP4 53 34 C#CC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726863 DH On-Demand Mild RBP4 59 42 C#C[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726867 DH On-Demand Mild RBP4 56 38 C#C[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726868 DH On-Demand Mild RBP4 56 38 COC(=O)N[C@@H](CC(C)C)C(=O)NC1CSC1 ZINC000880726877 CC On-Demand Anodyne CTSK 29 45 COC(=O)N[C@@H](CC(C)C)C(=O)NC1CSC1 ZINC000880726877 CC On-Demand Anodyne CAPNS1 53 33 COC(=O)N[C@@H](CC(C)C)C(=O)NC1CSC1 ZINC000880726877 CC On-Demand Anodyne CAPN1 69 52 COC(=O)N[C@@H](CC(C)C)C(=O)NC1CSC1 ZINC000880726877 CC On-Demand Anodyne CAPN2 82 40 COC(=O)N[C@@H](CC(C)C)C(=O)NC1CSC1 ZINC000880726877 CC On-Demand Anodyne FPR1 44 34 O=C(CCc1ccc2ccccc2c1O)NC1CSC1 ZINC000880726894 CF On-Demand Anodyne TNKS 58 33 COC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726910 EF On-Demand Anodyne CACNA1H 42 32 COC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726910 EF On-Demand Anodyne RBP4 52 34 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726952 GG On-Demand Anodyne EPHX2 25 40 CO[C@]1(CO)CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726965 EF On-Demand Anodyne EPHX2 27 40 CO[C@]1(CO)CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880726965 EF On-Demand Anodyne RBP4 44 32 CO[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880726992 EH On-Demand Anodyne RBP4 42 42 CO[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880726995 DF On-Demand Anodyne RBP4 52 34 O=C(NC1CSC1)[C@@H]1C[C@H]1c1ccc(Cl)cc1 ZINC000880727034 CF On-Demand Anodyne SLC6A3 20 43 Cc1cc(C(=O)NC2CSC2)ccc1N1CCOCC1 ZINC000880727056 CD On-Demand Anodyne MAPK11 27 46 Cc1cc(C(=O)NC2CSC2)ccc1N1CCOCC1 ZINC000880727056 CD On-Demand Anodyne MAPK14 39 46 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880727074 GI On-Demand Anodyne EPHX2 55 45 O=C(CC12C[C@H]3C[C@@H](CC(Br)(C3)C1)C2)Nc1ccc(N2CCOCC2)cn1 ZINC000880727088 IH On-Demand Anodyne STAT6 53 32 O=C(NC1CSC1)c1cc(F)c(N2CCOCC2)c(F)c1 ZINC000880727133 DD On-Demand Anodyne MAPK13 52 30 O=C(NC1CSC1)[C@@H]1C[C@H]1c1cccnc1 ZINC000880727155 BD On-Demand Anodyne NAMPT 28 52 CN(C)S(=O)(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880727166 GD On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C(=O)N1CCOCC1 ZINC000880727183 GF On-Demand Anodyne RBP4 53 33 C[C@@H](CO)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880727214 EH On-Demand Anodyne RBP4 47 38 O=C(Cc1cnn2ccccc12)NC1CSC1 ZINC000880727265 BD On-Demand Anodyne JAK3 17 41 O=C(Cc1cnn2ccccc12)NC1CSC1 ZINC000880727265 BD On-Demand Anodyne TYK2 20 41 O=C(Cc1cnn2ccccc12)NC1CSC1 ZINC000880727265 BD On-Demand Anodyne EPHB3 31 41 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@]1(C)CO ZINC000880727270 EG On-Demand Anodyne RBP4 45 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@]1(C)CO ZINC000880727271 EG On-Demand Anodyne RBP4 45 32 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@]1(C)CO ZINC000880727272 EG On-Demand Anodyne RBP4 45 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@]1(C)CO ZINC000880727273 EG On-Demand Anodyne RBP4 45 32 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880727282 GE On-Demand Anodyne RBP4 51 36 C[C@H]1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CS1(=O)=O ZINC000880727307 FG On-Demand Anodyne EPHX2 20 42 C[C@H]1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CS1(=O)=O ZINC000880727308 FG On-Demand Anodyne EPHX2 20 42 C[C@@H]1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CS1(=O)=O ZINC000880727310 FG On-Demand Anodyne EPHX2 20 42 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne PSEN2 48 31 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP13 37 48 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP2 41 47 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP3 15 47 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP8 19 47 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP14 34 47 O=C(NC1CSC1)C1(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000880727321 ED On-Demand Anodyne MMP10 71 34 O=C(NC1CSC1)c1cc2c(Br)c(F)ccc2[nH]1 ZINC000880727324 EF On-Demand Anodyne PYGL 44 35 C[C@@H](OCCc1ccccc1)C(=O)NC1CSC1 ZINC000880727330 CD On-Demand Anodyne ACE 60 38 C[C@@H](OCCc1ccccc1)C(=O)NC1CSC1 ZINC000880727330 CD On-Demand Anodyne MME 48 35 C[C@@H](OCCc1ccccc1)C(=O)NC1CSC1 ZINC000880727330 CD On-Demand Anodyne NAAA 42 39 O=C(NC1CSC1)[C@@H]1CCc2nc[nH]c2C1 ZINC000880727338 BC On-Demand Anodyne HTR3A 15 46 O=C(NC1CSC1)[C@H]1CCc2nc[nH]c2C1 ZINC000880727339 BC On-Demand Anodyne HTR3A 15 46 O=C(NC1CSC1)c1ccc(OC(F)F)c(F)c1 ZINC000880727342 CE On-Demand Anodyne EZH2 27 41 COC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C1CC1 ZINC000880727362 FH On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](CC(F)(F)F)O1 ZINC000880727408 GJ On-Demand Anodyne RBP4 43 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](CC(F)(F)F)O1 ZINC000880727410 GJ On-Demand Anodyne RBP4 43 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](CC(F)(F)F)O1 ZINC000880727412 GJ On-Demand Anodyne RBP4 43 32 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](CC(F)(F)F)O1 ZINC000880727415 GJ On-Demand Anodyne RBP4 43 32 O=C(NC1CSC1)c1ccn(CCc2ccccc2)n1 ZINC000880727436 CD On-Demand Anodyne SIGMAR1 15 42 O=C(Cc1cc2ccccc2c(O)n1)NC1CSC1 ZINC000880727438 CD On-Demand Anodyne TNKS 63 36 O=C(CN1CCCC[C@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727447 ED On-Demand Anodyne PRSS1 18 41 O=C(CN1CCCC[C@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727447 ED On-Demand Anodyne ACE 39 42 O=C(CN1CCCC[C@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727447 ED On-Demand Anodyne MME 19 42 O=C(CN1CCCC[C@@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727449 ED On-Demand Anodyne PRSS1 18 41 O=C(CN1CCCC[C@@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727449 ED On-Demand Anodyne ACE 39 42 O=C(CN1CCCC[C@@H](OCc2ccccc2)C1=O)NC1CSC1 ZINC000880727449 ED On-Demand Anodyne MME 19 42 Cc1cnc2cc(C(=O)NC3CSC3)ccn12 ZINC000880727453 BD On-Demand Anodyne MAPK13 85 39 O=C(CCC(=O)c1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880727485 CD On-Demand Bother CACNA1D 56 32 O=C(CCC(=O)c1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880727485 CD On-Demand Bother LUXR 17 42 O=C(NC1CSC1)[C@@H]1CCN(c2ccccc2)C1 ZINC000880727491 CD On-Demand Anodyne EPHX2 22 44 O=C(NC1CSC1)[C@H]1CCN(c2ccccc2)C1 ZINC000880727493 CD On-Demand Anodyne EPHX2 22 44 COc1cc(Br)c(Cl)cc1C(=O)NC1CSC1 ZINC000880727506 EF On-Demand Anodyne DRD2 28 41 COc1cc(Br)c(Cl)cc1C(=O)NC1CSC1 ZINC000880727506 EF On-Demand Anodyne DRD4 15 44 COc1cc(Br)c(Cl)cc1C(=O)NC1CSC1 ZINC000880727506 EF On-Demand Anodyne DRD3 16 44 COc1cc(Br)c(Cl)cc1C(=O)NC1CSC1 ZINC000880727506 EF On-Demand Anodyne HTR4 70 51 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727520 FH On-Demand Anodyne EPHX2 20 45 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727521 FH On-Demand Anodyne EPHX2 20 45 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727523 FH On-Demand Anodyne EPHX2 20 45 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727525 FH On-Demand Anodyne EPHX2 20 45 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne DRD2 18 54 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne DRD4 40 31 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne ACHE 24 47 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne HRH2 44 48 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne CHRM3 23 43 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne HRH3 18 43 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne SIGMAR1 31 54 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne SSTR5 46 42 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne CCR3 29 51 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne BDKRB1 47 53 O=C(NC1CSC1)c1cccc(CN2CCCCC2)c1 ZINC000880727532 CF On-Demand Anodyne MCHR1 41 51 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)C1=O ZINC000880727533 EH On-Demand Anodyne RBP4 55 35 CN(C)CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880727545 DD On-Demand Anodyne PAPA1_CARPA 34 42 CN(C)CC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880727546 DD On-Demand Anodyne PAPA1_CARPA 34 42 Cc1nnc([C@@H]2CCCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)o1 ZINC000880727571 FI On-Demand Anodyne RBP4 51 33 COC(=O)[C@@H]1C[C@@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727584 FE On-Demand Anodyne RBP4 52 34 COC(=O)[C@H]1C[C@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727585 FE On-Demand Anodyne RBP4 52 34 COC(=O)[C@H]1C[C@@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727586 FE On-Demand Anodyne RBP4 52 34 COC(=O)[C@@H]1C[C@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727587 FE On-Demand Anodyne RBP4 52 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)N1CC#N ZINC000880727617 FG On-Demand Mild RBP4 66 38 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)N1CC#N ZINC000880727618 FG On-Demand Mild RBP4 66 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)N1CC#N ZINC000880727619 FG On-Demand Mild RBP4 66 38 COC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C ZINC000880727626 EG On-Demand Anodyne RBP4 51 33 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NC2CSC2)CC1 ZINC000880727636 DE On-Demand Anodyne EPHX2 17 49 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NC2CSC2)CC1 ZINC000880727637 DE On-Demand Anodyne EPHX2 17 49 O=C(Cc1ccc2c(c1)CCCO2)NC1CSC1 ZINC000880727645 CD On-Demand Anodyne LUXR 45 36 O=C(NC1CSC1)c1cnn(C2CCCC2)c1-c1ccccc1 ZINC000880727647 EH On-Demand Anodyne HTR3A 20 41 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)[C@@H]1O ZINC000880727649 EG On-Demand Anodyne RBP4 55 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)C1O ZINC000880727650 EG On-Demand Anodyne RBP4 55 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)C1O ZINC000880727651 EG On-Demand Anodyne RBP4 55 35 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne PLG 17 42 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne ADAM17 22 40 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne SLC6A5 45 51 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne PLAU 19 41 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne ST14 16 42 O=C(NC1CSC1)c1ccc(OCc2ccncc2)cc1 ZINC000880727654 DF On-Demand Anodyne SMO 17 41 O=C(NC1CSC1)c1cc2cccnc2[nH]1 ZINC000880727656 BD On-Demand Anodyne PYGL 23 41 Cc1cc(C(=O)NC2CSC2)ccc1-n1cccn1 ZINC000880727658 CE On-Demand Anodyne MAPK14 56 39 Cc1cc(C(=O)NC2CSC2)ccc1-n1cccn1 ZINC000880727658 CE On-Demand Anodyne MAPK13 85 37 Cc1cccc(CNC(=O)c2ccc(C(=O)NC3CSC3)cc2)c1 ZINC000880727671 EF On-Demand Anodyne DRD4 18 47 Cc1cccc(CNC(=O)c2ccc(C(=O)NC3CSC3)cc2)c1 ZINC000880727671 EF On-Demand Anodyne CHRM3 15 44 Cc1cccc(CNC(=O)c2ccc(C(=O)NC3CSC3)cc2)c1 ZINC000880727671 EF On-Demand Anodyne MAPK14 18 51 O=C(Cc1cccc(C2CC2)c1)NC1CSC1 ZINC000880727676 BE On-Demand Anodyne SIGMAR1 15 42 O=C(Cc1cccc(C2CC2)c1)NC1CSC1 ZINC000880727676 BE On-Demand Anodyne LUXR 49 38 C#CCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880727681 CD On-Demand Mild PLA2G4B 40 33 COc1cccc([C@H](CO)NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880727684 FH On-Demand Anodyne KCNQ2 24 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne F2 47 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne ACE 34 43 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne TRY1_BOVIN 47 36 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne PREP 94 51 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne XIAP 40 37 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne SFRP1 41 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne WNT3 45 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1 ZINC000880727688 CD On-Demand Anodyne TMPRSS11D 57 34 CO/C(=C\c1ccccc1)C(=O)NC1CSC1 ZINC000880727698 BD On-Demand Anodyne TLR4 26 45 CO/C(=C/c1ccccc1)C(=O)NC1CSC1 ZINC000880727700 BD On-Demand Anodyne TLR4 26 45 COC(=O)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1C ZINC000880727718 FH On-Demand Anodyne RBP4 47 39 Cn1ncc(C2CCC2)c1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880727738 FI On-Demand Anodyne TRPV1 19 41 Cc1ccncc1CCNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880727739 EI On-Demand Anodyne TRPV1 19 46 CC(C)(C)CC(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880727747 GI On-Demand Anodyne RBP4 52 35 CCn1c(O)nnc1C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880727759 GH On-Demand Anodyne RBP4 47 39 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne ACE 71 42 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne PPARA 15 40 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne MME 137 40 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne ANPEP 47 35 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne CYSP_TRYCR 41 34 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne CPA1 41 36 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne TIMP3 66 38 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne CAPNS1 55 32 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne MMP3 15 40 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne CAPN1 57 38 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne CAPN2 45 32 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne ACE2 53 36 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne MMP1 17 40 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne AMP1_PLAFQ 53 36 CO[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880727782 CD On-Demand Anodyne NAAA 44 33 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne CELA1 19 43 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne PREP 31 48 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne LGMN 70 42 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne KLK5 33 43 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne SLC12A5 42 35 O=C(NC1CSC1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727791 ED On-Demand Anodyne Q9NAW4_PLAFA 36 40 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne CELA1 19 43 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne PREP 31 48 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne LGMN 70 42 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne KLK5 33 43 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne SLC12A5 42 35 O=C(NC1CSC1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880727792 ED On-Demand Anodyne Q9NAW4_PLAFA 36 40 Cn1nc(-c2ccccc2)cc1C(=O)NC1CSC1 ZINC000880727794 CD On-Demand Anodyne INHA 76 36 Cc1ccccc1[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880727797 EF On-Demand Anodyne FPR1 40 35 Cc1ccccc1[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880727798 EF On-Demand Anodyne FPR1 40 35 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne FKBP1A 20 53 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP13 46 45 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne ITGA4 36 49 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne CAPNS1 23 47 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP2 21 45 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP3 52 49 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP8 33 44 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne CAPN1 20 54 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP9 29 41 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne EPHX2 17 50 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP7 55 45 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne MMP1 51 49 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne SFRP1 115 36 O=C(NC1CSC1)[C@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880727817 ED On-Demand Anodyne WNT3 83 35 COc1ccc(OC(F)(F)F)c(C(=O)NC2CSC2)c1 ZINC000880727834 DE On-Demand Anodyne KCNK9 20 40 COc1cc(Br)c(C(=O)NC2CSC2)cc1OC ZINC000880727842 EE On-Demand Anodyne HTR4 28 41 COC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)O1 ZINC000880727849 FF On-Demand Anodyne RBP4 43 32 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne ELANE 32 42 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne KLK3 84 37 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CTSB 60 41 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne PAPA1_CARPA 61 36 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CYSP_TRYCR 56 42 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CTSK 42 45 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CTSL 45 40 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CAPNS1 65 36 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CTSS 19 45 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CAPN1 81 42 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne CAPN2 132 41 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne NPR 65 34 O=C(CC[C@H](NC(=O)OCc1ccccc1)C(F)(F)F)NC1CSC1 ZINC000880727851 GF On-Demand Anodyne PSMB5 45 39 O=C(COc1ccc(Cl)c(F)c1)NC1CSC1 ZINC000880727861 CE On-Demand Anodyne ENV 42 37 O=C(COc1ccc(Cl)c(F)c1)NC1CSC1 ZINC000880727861 CE On-Demand Anodyne TRAR 30 42 Cc1nnc(COC2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)o1 ZINC000880727863 FG On-Demand Anodyne RBP4 50 32 CN(C(=O)Nc1cccc(F)c1C(C)(F)F)[C@H](CO)Cc1ccccc1 ZINC000880727919 FI On-Demand Anodyne NPY5R 24 43 CN(C(=O)Nc1cccc(F)c1C(C)(F)F)[C@@H](CO)Cc1ccccc1 ZINC000880727920 FI On-Demand Anodyne NPY5R 24 43 Cc1cc(C(=O)NC2CSC2)nn1-c1cccc(C(F)(F)F)c1 ZINC000880727951 EG On-Demand Anodyne CCR2 40 34 C#CC[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727953 DI On-Demand Mild RBP4 57 39 C#CC[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880727954 DI On-Demand Mild RBP4 57 39 COc1cccc(Oc2ccc(C(=O)NC3CSC3)nc2)c1 ZINC000880727966 DF On-Demand Anodyne DRD4 41 31 COc1cccc(Oc2ccc(C(=O)NC3CSC3)nc2)c1 ZINC000880727966 DF On-Demand Anodyne PDE4B 45 33 COc1cccc(Oc2ccc(C(=O)NC3CSC3)nc2)c1 ZINC000880727966 DF On-Demand Anodyne MTNR1A 31 44 COc1cccc(Oc2ccc(C(=O)NC3CSC3)nc2)c1 ZINC000880727966 DF On-Demand Anodyne MTNR1B 31 44 CC(C)(C)OC(=O)N[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880727976 DE On-Demand Anodyne PAPA1_CARPA 36 40 CC(C)(C)OC(=O)N[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880727976 DE On-Demand Anodyne CTSK 15 50 CC(C)(C)OC(=O)N[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880727976 DE On-Demand Anodyne FPR1 47 37 CC(C)(C)OC(=O)N[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880727976 DE On-Demand Anodyne AMP1_PLAFQ 19 45 CC(C)(C)OC(=O)N[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880727976 DE On-Demand Anodyne Q82323_9DELA 68 31 O=C(NC1CSC1)c1ccc(I)cc1F ZINC000880727984 EE On-Demand Anodyne MAP2K1 45 32 O=C(NC1CSC1)C1CCN(c2noc3ccc(Cl)cc23)CC1 ZINC000880727987 FF On-Demand Anodyne PTGES 32 47 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880728010 JH On-Demand Anodyne F10 25 46 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880728010 JH On-Demand Anodyne CPT1A 53 41 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880728010 JH On-Demand Anodyne CPT2 35 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880728010 JH On-Demand Anodyne CPT1B 39 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880728010 JH On-Demand Anodyne STAT6 48 36 CC(C)(C)OC(=O)N1CCC(c2ncc(C(=O)NC3CSC3)o2)CC1 ZINC000880728061 FF On-Demand Anodyne GPR119 43 40 O=C(NC1CSC1)c1cc2c(Br)cncc2s1 ZINC000880728073 EF On-Demand Anodyne SELE 138 41 O=C(NC1CSC1)c1cc2c(Br)cncc2s1 ZINC000880728073 EF On-Demand Anodyne ICAM1 131 41 O=C(NC1CSC1)c1cc2c(Br)cncc2s1 ZINC000880728073 EF On-Demand Anodyne VCAM1 92 37 O=C(NC1CSC1)c1cnc(Nc2ccccc2)nc1C(F)(F)F ZINC000880728094 FG On-Demand Anodyne ATF1 43 38 O=C(NC1CSC1)c1cnc(Nc2ccccc2)nc1C(F)(F)F ZINC000880728094 FG On-Demand Anodyne NFKB1 40 38 O=C(NC1CSC1)c1cnc(Nc2ccccc2)nc1C(F)(F)F ZINC000880728094 FG On-Demand Anodyne STAT6 43 34 O=C(NC1CSC1)c1nn(-c2ccc(F)cc2F)c2c1CCC2 ZINC000880728121 EE On-Demand Anodyne CNR1 53 33 O=C(NC1CSC1)c1nn(-c2ccc(F)cc2F)c2c1CCC2 ZINC000880728121 EE On-Demand Anodyne CNR2 16 52 O=C(NC1CSC1)c1nn(-c2ccc(F)cc2F)c2c1CCC2 ZINC000880728121 EE On-Demand Anodyne MAPK14 15 42 Cn1nc(CC(=O)NC2CSC2)c2ccccc21 ZINC000880728137 CD On-Demand Anodyne HTR3A 16 43 Cn1nc(CC(=O)NC2CSC2)c2ccccc21 ZINC000880728137 CD On-Demand Anodyne IMDH_CRYPV 29 42 Cn1ncc(C2CC2)c1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880728152 FH On-Demand Anodyne TRPV1 23 42 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H](C)O1 ZINC000880728153 EH On-Demand Anodyne RBP4 55 37 O=C(NC1CSC1)[C@@H]1CCc2ccccc2C1 ZINC000880728168 BE On-Demand Anodyne PREP 21 41 O=C(NC1CSC1)[C@H]1CCc2ccccc2C1 ZINC000880728169 BE On-Demand Anodyne PREP 21 41 CCO[C@@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728176 DH On-Demand Anodyne EPHX2 37 40 CCN1CC[C@@H](N(CC)C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728218 EH On-Demand Anodyne CCR5 20 43 CCN1CC[C@H](N(CC)C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728219 EH On-Demand Anodyne CCR5 20 43 O=C(Cc1cc2cc(Cl)ccc2[nH]1)NC1CSC1 ZINC000880728231 CF On-Demand Anodyne PYGL 77 42 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880728239 DF On-Demand Anodyne TIMP3 17 40 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880728239 DF On-Demand Anodyne EPHX2 33 43 C[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880728239 DF On-Demand Anodyne ACE2 53 36 O=C(NC1CSC1)c1coc(C2CCCCC2)n1 ZINC000880728271 CF On-Demand Anodyne TBXA2R 17 41 O=C(Cc1sc(N2CCOCC2)nc1-c1ccccc1)NC1CSC1 ZINC000880728275 GE On-Demand Anodyne PIK3CA 21 40 O=C(Cc1sc(N2CCOCC2)nc1-c1ccccc1)NC1CSC1 ZINC000880728275 GE On-Demand Anodyne PIK3CD 23 40 O=C(Cc1sc(N2CCOCC2)nc1-c1ccccc1)NC1CSC1 ZINC000880728275 GE On-Demand Anodyne PIK3CB 34 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne F2 75 44 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne PLG 33 46 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne PRSS1 33 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne ACE 51 51 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne FKBP1A 63 45 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne OPRM1 30 44 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne OPRD1 16 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne CELA1 35 58 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne GRIN2B 25 43 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne ELANE 43 47 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne TACR1 15 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne CTRA_BOVIN 65 36 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne TRY1_BOVIN 94 39 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne CTSG 45 36 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne CTSL 18 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne DPP4 19 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne PREP 107 58 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne CELA2A 54 36 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne LGMN 102 58 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne ACE2 20 45 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne KLK5 30 52 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne XIAP 57 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne BRCA1 62 33 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne SLC12A5 66 39 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne Q9NAW4_PLAFA 39 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880728281 DE On-Demand Anodyne TMPRSS11D 69 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880728283 DG On-Demand Anodyne RBP4 53 35 O=C(NC1CSC1)c1ccc2nnc(S)n2c1 ZINC000880728304 CC On-Demand Anodyne MAPK13 77 35 CC(C)(C[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1)C(N)=O ZINC000880728325 GI On-Demand Anodyne RBP4 52 32 CC(C)(C[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1)C(N)=O ZINC000880728326 GI On-Demand Anodyne RBP4 52 32 O=C(NC1CSC1)c1coc2cc(F)ccc12 ZINC000880728329 CE On-Demand Anodyne INHA 47 34 COc1ccccc1-n1ncc(C(=O)NC2CSC2)c1C ZINC000880728367 DE On-Demand Anodyne DRD2 31 40 COc1ccccc1-n1ncc(C(=O)NC2CSC2)c1C ZINC000880728367 DE On-Demand Anodyne DRD4 22 40 COc1ccccc1-n1ncc(C(=O)NC2CSC2)c1C ZINC000880728367 DE On-Demand Anodyne DRD3 43 39 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc(F)c1C(C)(F)F)C2 ZINC000880728375 EH On-Demand Anodyne HTR3A 33 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc(F)c1C(C)(F)F)C2 ZINC000880728375 EH On-Demand Anodyne EPHX2 34 43 CN(C(=O)Nc1cccc(F)c1C(C)(F)F)[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880728383 GE On-Demand Anodyne EPHX2 15 41 CN(C(=O)Nc1cccc(F)c1C(C)(F)F)[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880728384 GE On-Demand Anodyne EPHX2 15 41 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728386 FG On-Demand Anodyne RBP4 52 33 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne ACE 61 38 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne GRIN2B 15 43 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne MME 70 38 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne CTSB 19 42 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne CASP1 30 49 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne CAPN2 19 42 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne NAAA 34 43 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne PSMB5 32 41 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne BIRC2 54 38 C[C@@H](NC(=O)CCc1ccccc1)C(=O)NC1CSC1 ZINC000880728387 CD On-Demand Anodyne BIRC8 44 31 O=C(CCCC(=O)c1ccc(Br)cc1)NC1CSC1 ZINC000880728388 EG On-Demand Anodyne HDAC8 30 52 O=C(CCCC(=O)c1ccc(Br)cc1)NC1CSC1 ZINC000880728388 EG On-Demand Anodyne HAO1 15 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne ELANE 39 44 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP13 29 41 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne PREP 29 45 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP3 37 41 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP8 15 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP9 25 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP7 36 40 COc1ccc(C(=O)N2CCC[C@H]2C(=O)NC2CSC2)cc1 ZINC000880728394 DD On-Demand Anodyne MMP1 33 43 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne ELANE 39 44 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP13 29 41 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne PREP 29 45 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP3 37 41 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP8 15 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP9 25 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP7 36 40 COc1ccc(C(=O)N2CCC[C@@H]2C(=O)NC2CSC2)cc1 ZINC000880728395 DD On-Demand Anodyne MMP1 33 43 C[C@@H]1[C@H](C(=O)NC2CSC2)[C@H]1c1ccccc1 ZINC000880728420 BE On-Demand Anodyne HDAC4 33 43 C[C@@H]1[C@@H](C(=O)NC2CSC2)[C@@H]1c1ccccc1 ZINC000880728421 BE On-Demand Anodyne HDAC4 33 43 C[C@@H]1[C@H](C(=O)NC2CSC2)[C@@H]1c1ccccc1 ZINC000880728422 BE On-Demand Anodyne HDAC4 33 43 C[C@H]1[C@H](c2ccccc2)[C@@H]1C(=O)NC1CSC1 ZINC000880728423 BE On-Demand Anodyne HDAC4 33 43 COCCn1cc(C(=O)NC2CSC2)c(=O)cc1C ZINC000880728433 CC On-Demand Anodyne CNR2 20 56 COc1cccc(C2=NO[C@@H](C(=O)NC3CSC3)C2)c1 ZINC000880728450 CD On-Demand Anodyne LUCI_PHOPY 34 47 COc1cccc(C2=NO[C@H](C(=O)NC3CSC3)C2)c1 ZINC000880728451 CD On-Demand Anodyne LUCI_PHOPY 34 47 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)N1C ZINC000880728452 EG On-Demand Anodyne RBP4 60 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C(N)=O ZINC000880728501 EF On-Demand Anodyne RBP4 52 33 O=C(NC1CSC1)C1CCN(CC(F)(F)F)CC1 ZINC000880728567 CD On-Demand Anodyne HPGDS 34 40 O=C(NC1CSC1)c1cccc(Cn2ccnc2)c1 ZINC000880728604 CD On-Demand Anodyne CYP19A1 21 59 O=C(NC1CSC1)c1cccc(Cn2ccnc2)c1 ZINC000880728604 CD On-Demand Anodyne CYP11B1 53 50 O=C(NC1CSC1)c1cccc(Cn2ccnc2)c1 ZINC000880728604 CD On-Demand Anodyne TBXAS1 54 50 O=C(NC1CSC1)c1cccc(Cn2ccnc2)c1 ZINC000880728604 CD On-Demand Anodyne CYP11B2 28 47 CN(C)C(=O)OC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880728605 FH On-Demand Anodyne RBP4 55 39 Cn1ncc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)n1 ZINC000880728610 DE On-Demand Anodyne TRPV1 15 41 CC1(CO)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728631 DF On-Demand Anodyne RBP4 50 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)N1CCO ZINC000880728663 FF On-Demand Anodyne RBP4 55 35 O=C(NC1CSC1)c1ccc(COC(F)(F)F)cc1 ZINC000880728713 CF On-Demand Anodyne SLC6A5 40 46 N#Cc1ccc(C[C@H](C#N)C(=O)NC2CSC2)cc1 ZINC000880728715 CD On-Demand Mild CTSC 32 40 N#Cc1ccc(C[C@@H](C#N)C(=O)NC2CSC2)cc1 ZINC000880728716 CD On-Demand Mild CTSC 32 40 Cc1ccncc1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880728725 DH On-Demand Anodyne TRPV1 25 48 C[C@@H](CF)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880728737 CG On-Demand Anodyne ANPEP 16 49 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728752 FH On-Demand Anodyne RBP4 51 34 CCN1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1=O ZINC000880728847 EF On-Demand Anodyne EPHX2 23 40 CN1C(=O)CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728876 EE On-Demand Anodyne NPY1R 15 41 CN1C(=O)CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728876 EE On-Demand Anodyne CCKAR 19 40 CN1C(=O)CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728876 EE On-Demand Anodyne CCKBR 21 40 O=C(CCSCc1ccccc1)NC1CSC1 ZINC000880728877 CF On-Demand Anodyne CACNA2D1 25 45 O=C(CCSCc1ccccc1)NC1CSC1 ZINC000880728877 CF On-Demand Anodyne TNKS 61 35 CN1C(=O)CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728878 EE On-Demand Anodyne NPY1R 15 41 CN1C(=O)CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728878 EE On-Demand Anodyne CCKAR 19 40 CN1C(=O)CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880728878 EE On-Demand Anodyne CCKBR 21 40 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880728888 FH On-Demand Anodyne EPHX2 28 43 CN1CC[C@@]2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)C1 ZINC000880728901 EG On-Demand Anodyne EPHX2 29 48 Cc1cc(O)nc2cc(C(=O)NC3CSC3)ccc12 ZINC000880728920 CE On-Demand Anodyne MAPK14 43 41 CN(CCC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880728942 DD On-Demand Anodyne GRIN2B 21 40 CN(CCC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880728942 DD On-Demand Anodyne CAPNS1 46 31 CN(CCC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880728942 DD On-Demand Anodyne CAPN2 40 32 CN(CCC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880728942 DD On-Demand Anodyne NPR 42 35 CN(CCC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880728942 DD On-Demand Anodyne F13A1 15 41 O=C(NC1CSC1)c1ccc(CN2CCOCC2)cn1 ZINC000880728963 CC On-Demand Anodyne PDE4B 39 40 C[C@H]1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CS1 ZINC000880729053 DH On-Demand Anodyne EPHX2 15 41 O=C(NC1CSC1)[C@H]1CCN(c2ccccc2Cl)C1 ZINC000880729055 CE On-Demand Anodyne EPHX2 26 46 O=C(NC1CSC1)[C@@H]1CCN(c2ccccc2Cl)C1 ZINC000880729056 CE On-Demand Anodyne EPHX2 26 46 CN1CCC[C@@H](CCNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729061 EH On-Demand Anodyne CCR3 47 41 CCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1C(=O)NC1CSC1 ZINC000880729076 GC On-Demand Anodyne PDE5A 38 44 CCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1C(=O)NC1CSC1 ZINC000880729076 GC On-Demand Anodyne HCN1 49 37 O=C(NC1CSC1)c1ccnc(NC(=O)C2CC2)c1 ZINC000880729077 CD On-Demand Anodyne TYK2 74 47 O=C(NC1CSC1)c1cccc2oc(O)nc12 ZINC000880729091 CD On-Demand Anodyne HTR3A 32 47 CN1C[C@@H]2CCCN(C(=O)Nc3cccc(F)c3C(C)(F)F)[C@@H]2C1 ZINC000880729105 EG On-Demand Anodyne RBP4 44 32 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1Cl ZINC000880729121 DE On-Demand Anodyne DRD4 21 42 Cn1c(C(=O)NC2CSC2)cc2ccccc2c1=O ZINC000880729132 CD On-Demand Anodyne POLR1A 52 38 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729140 EE On-Demand Anodyne DRD4 31 42 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729140 EE On-Demand Anodyne SIGMAR1 57 46 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729140 EE On-Demand Anodyne CCR3 18 41 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729140 EE On-Demand Anodyne CACNA1G 17 41 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729140 EE On-Demand Anodyne NPFFR1 42 37 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729142 EE On-Demand Anodyne DRD4 31 42 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729142 EE On-Demand Anodyne SIGMAR1 57 46 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729142 EE On-Demand Anodyne CCR3 18 41 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729142 EE On-Demand Anodyne CACNA1G 17 41 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCC1(F)F ZINC000880729142 EE On-Demand Anodyne NPFFR1 42 37 O=C(CCc1cnc2ccccc2c1)NC1CSC1 ZINC000880729164 CE On-Demand Anodyne TNKS 57 33 Cc1cc(OCC(=O)NC2CSC2)ccc1[N+](=O)[O-] ZINC000880729183 CD On-Demand Bother TRAR 28 41 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880729184 JI On-Demand Anodyne P2RX7 20 44 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880729185 JI On-Demand Anodyne P2RX7 20 44 O=C(NC1CSC1)[C@@H]1C[C@H]1c1ccc(OC(F)(F)F)cc1 ZINC000880729187 DF On-Demand Anodyne EPHX2 27 41 CNS(=O)(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880729188 GE On-Demand Anodyne RBP4 44 43 CC(C)[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCCO1 ZINC000880729197 EI On-Demand Anodyne RBP4 44 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN(C2CCC2)C1 ZINC000880729212 FI On-Demand Anodyne RBP4 51 34 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN(C2CCC2)C1 ZINC000880729213 FI On-Demand Anodyne RBP4 51 34 O=C(NC1CSC1)c1cc(Cc2ccccc2)[nH]n1 ZINC000880729218 CD On-Demand Anodyne HAO2 73 34 O=C(CCc1cccc(CCC(=O)NC2CSC2)c1)NC1CSC1 ZINC000880729228 FE On-Demand Anodyne LUXR 44 45 O=C(NC1CSC1)c1sc(N2CCOCC2)nc1-c1ccccc1 ZINC000880729245 FE On-Demand Anodyne PIK3CD 19 41 COc1ccc(-c2ocnc2C(=O)NC2CSC2)cc1 ZINC000880729279 CE On-Demand Anodyne PDK1 48 40 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NC2CSC2)C1 ZINC000880729448 DD On-Demand Anodyne EPHX2 17 44 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729449 EF On-Demand Anodyne RBP4 53 37 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729449 EF On-Demand Anodyne CCR8 46 32 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729450 EF On-Demand Anodyne RBP4 53 37 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729450 EF On-Demand Anodyne CCR8 46 32 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne ACE 134 45 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne MME 208 45 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne ANPEP 88 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne TACR1 15 41 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne FCER2 82 36 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne RNPEP 23 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CTSB 57 40 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne PAPA1_CARPA 47 38 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CYSP_TRYCR 66 38 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CTSL 47 40 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CPA1 63 44 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne TIMP3 76 38 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CTRB1 30 41 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CAPNS1 83 36 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne MMP8 28 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne ECE1 41 38 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne HLA-DRB1 54 33 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CTSS 20 40 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CAPN1 98 47 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne MMP9 30 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne CAPN2 81 40 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne ACE2 104 44 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne LAP3 45 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne FPR1 79 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne NPR 63 38 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne AMP1_PLAFQ 57 43 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne GAG-PRO 53 32 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne NAAA 42 33 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne BLA1_STEMA 64 35 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne BIRC2 25 41 C[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880729502 BE On-Demand Anodyne Q82323_9DELA 63 31 O=C(Cc1cccc(Cl)c1Cl)NC1CSC1 ZINC000880729572 CF On-Demand Anodyne P2RX7 30 45 CNC(=O)COc1cccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880729587 GG On-Demand Anodyne ROCK2 22 44 CNC(=O)COc1cccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880729587 GG On-Demand Anodyne PDS 53 34 Cc1nc2ccc(C(=O)NC3CSC3)cc2s1 ZINC000880729589 CE On-Demand Anodyne LCK 31 47 CC(=O)NC[C@@H]1CCn2ncc(C(=O)NC3CSC3)c2C1 ZINC000880729595 DC On-Demand Anodyne CACNA1I 43 30 O=C(COc1cccc(I)c1)NC1CSC1 ZINC000880729599 ED On-Demand Anodyne TRAR 29 41 CCC[C@]1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729602 EH On-Demand Anodyne RBP4 44 31 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880729618 DG On-Demand Anodyne RBP4 53 35 COc1cccc([C@H](C)CCCC(=O)NC2CSC2)c1 ZINC000880729630 CG On-Demand Anodyne MTNR1A 32 45 COc1cccc([C@H](C)CCCC(=O)NC2CSC2)c1 ZINC000880729630 CG On-Demand Anodyne MTNR1B 34 45 COc1cccc([C@@H](C)CCCC(=O)NC2CSC2)c1 ZINC000880729631 CG On-Demand Anodyne MTNR1A 32 45 COc1cccc([C@@H](C)CCCC(=O)NC2CSC2)c1 ZINC000880729631 CG On-Demand Anodyne MTNR1B 34 45 CN(C)S(=O)(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729649 GF On-Demand Anodyne RBP4 40 37 CN(C)S(=O)(=O)[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729650 GF On-Demand Anodyne RBP4 40 37 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729653 GH On-Demand Anodyne EPHX2 29 42 COCCOc1cc(OC)ccc1C(=O)NC1CSC1 ZINC000880729654 CD On-Demand Anodyne MTNR1A 48 37 COCCOc1cc(OC)ccc1C(=O)NC1CSC1 ZINC000880729654 CD On-Demand Anodyne LUCI_LUCLA 15 42 O=C(NC1CSC1)c1ccc(OC(F)(F)Cl)cc1 ZINC000880729656 CF On-Demand Anodyne SLC6A5 34 41 O=C(NC1CSC1)c1ccc(OC(F)(F)Cl)cc1 ZINC000880729656 CF On-Demand Anodyne EPHX2 26 40 COc1cccc(C(=O)NC2CSC2)c1[N+](=O)[O-] ZINC000880729657 CD On-Demand Bother KCNMA1 24 40 O=C(NC1CSC1)c1ccc(C(F)(F)F)cc1N1CCCC1 ZINC000880729693 EG On-Demand Anodyne MC4R 20 41 O=C(NC1CSC1)c1ccc(C(F)(F)F)cc1N1CCCC1 ZINC000880729693 EG On-Demand Anodyne LIPG 50 34 O=C(Cc1cccc(Cl)c1F)NC1CSC1 ZINC000880729710 CE On-Demand Anodyne P2RX7 28 47 O=C(NC1CSC1)c1c[nH]nc1-c1ccccn1 ZINC000880729716 CD On-Demand Anodyne TGFBR1 22 47 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[S@@](=O)C1 ZINC000880729750 EG On-Demand Anodyne RBP4 52 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[S@@](=O)C1 ZINC000880729751 EG On-Demand Anodyne RBP4 52 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[S@](=O)C1 ZINC000880729752 EG On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[S@](=O)C1 ZINC000880729753 EG On-Demand Anodyne RBP4 52 33 COCC1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880729754 EI On-Demand Anodyne EPHX2 46 44 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729755 FF On-Demand Anodyne RBP4 44 32 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729756 FF On-Demand Anodyne RBP4 44 32 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729762 EG On-Demand Anodyne EPHX2 25 42 O=C(Cc1ccc(Cl)c(F)c1)NC1CSC1 ZINC000880729778 CE On-Demand Anodyne ENV 44 40 O=C(NC1CSC1)c1ccc(NCC2CC2)nc1 ZINC000880729783 CD On-Demand Anodyne SSTR5 22 40 O=C(NC1CSC1)c1ccc(NCC2CC2)nc1 ZINC000880729783 CD On-Demand Anodyne IKBKB 20 43 O=C(NC1CSC1)c1ccc(NCC2CC2)nc1 ZINC000880729783 CD On-Demand Anodyne VCP 41 32 C[C@@H](Oc1cccc2ccccc12)C(=O)NC1CSC1 ZINC000880729799 CF On-Demand Anodyne IMDH_CRYPV 22 46 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne DRD4 35 49 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne ACHE 22 46 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne HRH3 29 46 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne SIGMAR1 30 53 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne SSTR5 49 40 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne CCR3 18 50 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne BDKRB1 28 44 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne UTS2R 20 42 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne SLC6A5 36 45 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne MCHR1 46 50 O=C(NC1CSC1)c1ccc(CN2CCCC2)cc1 ZINC000880729820 CE On-Demand Anodyne NOD2 41 34 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne GRIN2B 45 53 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne SIGMAR1 16 49 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne CTSK 16 44 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne CTSL 21 44 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne PREP 34 45 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne EPHX2 35 47 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne TGM2 44 46 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne F13A1 42 46 O=C(NC1CSC1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729843 DD On-Demand Anodyne CCR8 20 40 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne GRIN2B 45 53 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne SIGMAR1 16 49 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne CTSK 16 44 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne CTSL 21 44 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne PREP 34 45 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne EPHX2 35 47 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne TGM2 44 46 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne F13A1 42 46 O=C(NC1CSC1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880729844 DD On-Demand Anodyne CCR8 20 40 COC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880729855 EH On-Demand Anodyne CACNA1H 54 33 COC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880729855 EH On-Demand Anodyne TRPM8 29 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880729869 FF On-Demand Anodyne RBP4 56 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880729870 FF On-Demand Anodyne RBP4 56 38 COc1ccc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)nc1 ZINC000880729890 GH On-Demand Anodyne PDGFRB 41 36 COc1ccc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)nc1 ZINC000880729890 GH On-Demand Anodyne RBP4 31 41 COc1ccc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)nc1 ZINC000880729890 GH On-Demand Anodyne DGAT1 34 53 COc1ccc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)nc1 ZINC000880729890 GH On-Demand Anodyne NPBWR1 43 38 CC(C)(C)OC(=O)N1CCC([C@@H]2C[C@H]2C(=O)NC2CSC2)CC1 ZINC000880729893 EF On-Demand Anodyne GPR119 23 44 C[C@@H]1CN(CC(F)(F)F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729896 GI On-Demand Anodyne RBP4 51 32 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729902 EF On-Demand Anodyne EPHX2 21 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880729902 EF On-Demand Anodyne RBP4 54 37 COC[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880729923 EI On-Demand Anodyne RBP4 35 40 CN(C)CCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880729947 CD On-Demand Anodyne SLC6A5 30 41 Cc1ccnc2ccc(C(=O)NC3CSC3)cc12 ZINC000880729948 CE On-Demand Anodyne MAPK14 48 36 CN(C[C@H]1CCCN1C)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880729956 EG On-Demand Anodyne CHRNA10 55 39 CN(C[C@H]1CCCN1C)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880729956 EG On-Demand Anodyne ACKR3 52 32 CN(C[C@@H]1CCCN1C)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880729957 EG On-Demand Anodyne CHRNA10 55 39 CN(C[C@@H]1CCCN1C)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880729957 EG On-Demand Anodyne ACKR3 52 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)S1(=O)=O ZINC000880729971 FF On-Demand Anodyne RBP4 56 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCC1(F)F ZINC000880729986 EI On-Demand Anodyne RBP4 53 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCC1(F)F ZINC000880729987 EI On-Demand Anodyne RBP4 53 33 N#CCCCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880730001 CF On-Demand Mild CNR1 29 44 N#CCCCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880730001 CF On-Demand Mild CNR2 52 44 CCOc1nc2ccc(C(=O)NC3CSC3)cc2[nH]1 ZINC000880730025 CD On-Demand Anodyne SSTR5 45 35 O=C(NC1CSC1)[C@H]1CCC(=O)N1Cc1ccc(Br)cc1 ZINC000880730027 FE On-Demand Anodyne P2RX7 29 44 O=C(NC1CSC1)[C@@H]1CCC(=O)N1Cc1ccc(Br)cc1 ZINC000880730028 FE On-Demand Anodyne P2RX7 29 44 O=C(CCc1ccccn1)NC1CSC1 ZINC000880730029 BD On-Demand Anodyne GRIN2B 15 61 O=C(NC1CSC1)c1cc(F)c(C(F)(F)F)c(F)c1 ZINC000880730051 CF On-Demand Anodyne MAPK13 68 35 O=C(Cc1ccc(Br)c(Cl)c1)NC1CSC1 ZINC000880730054 DF On-Demand Anodyne LUXR 43 35 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730084 EG On-Demand Anodyne RBP4 61 36 Cn1cnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880730094 BD On-Demand Anodyne HPGD 45 36 O=C(NC1CSC1)[C@H]1CCN(c2ccccc2F)C1 ZINC000880730095 CD On-Demand Anodyne EPHX2 17 46 O=C(NC1CSC1)[C@@H]1CCN(c2ccccc2F)C1 ZINC000880730096 CD On-Demand Anodyne EPHX2 17 46 O=C(NC1CSC1)c1ccccc1N1CCCCC1 ZINC000880730105 CF On-Demand Anodyne KCNQ2 69 38 CN1CCO[C@@H]2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)C[C@@H]21 ZINC000880730114 EE On-Demand Anodyne RBP4 52 33 COC1(C(F)(F)F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730115 GJ On-Demand Anodyne CACNA1H 56 34 CCO[C@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730125 DH On-Demand Anodyne EPHX2 37 40 CC[C@H]1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880730127 EI On-Demand Anodyne EPHX2 23 40 CC[C@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880730128 EI On-Demand Anodyne EPHX2 23 40 CC[C@@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880730129 EI On-Demand Anodyne EPHX2 23 40 O=C(Cc1coc2ccccc12)NC1CSC1 ZINC000880730139 BE On-Demand Anodyne INHA 66 34 COc1cc(C)c(Br)cc1C(=O)NC1CSC1 ZINC000880730163 DF On-Demand Anodyne HTR4 29 44 CN(C)C1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730172 EH On-Demand Anodyne EPHX2 47 49 COC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880730173 CC On-Demand Anodyne PAPA1_CARPA 38 42 O=C(COCc1cccnc1)NC1CSC1 ZINC000880730182 BC On-Demand Anodyne CHRNA7 47 39 C[C@H]1C[C@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730190 DG On-Demand Anodyne RBP4 69 38 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730192 DG On-Demand Anodyne RBP4 69 38 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730225 FG On-Demand Anodyne RBP4 32 41 C[C@@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730239 CF On-Demand Anodyne SSTR2 46 33 C[C@@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730239 CF On-Demand Anodyne MMP2 18 41 C[C@@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730239 CF On-Demand Anodyne MMP8 27 41 C[C@@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730239 CF On-Demand Anodyne MMP9 15 41 C[C@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730240 CF On-Demand Anodyne SSTR2 46 33 C[C@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730240 CF On-Demand Anodyne MMP2 18 41 C[C@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730240 CF On-Demand Anodyne MMP8 27 41 C[C@H](CC(=O)NC1CSC1)c1c[nH]c2ccccc12 ZINC000880730240 CF On-Demand Anodyne MMP9 15 41 COCCOc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880730276 CD On-Demand Anodyne PLA2G4B 54 39 O=C(NC1CSC1)[C@H]1CCCN1c1ccccc1 ZINC000880730283 CD On-Demand Anodyne PREP 45 37 O=C(NC1CSC1)[C@@H]1CCCN1c1ccccc1 ZINC000880730284 CD On-Demand Anodyne PREP 45 37 C[S@@](=O)Cc1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880730286 GI On-Demand Anodyne TRPV1 15 42 C[S@](=O)Cc1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880730287 GI On-Demand Anodyne TRPV1 15 42 O=C(Cc1cncn1Cc1ccccc1)NC1CSC1 ZINC000880730382 CD On-Demand Anodyne CYP11B1 17 51 O=C(Cc1cncn1Cc1ccccc1)NC1CSC1 ZINC000880730382 CD On-Demand Anodyne SIGMAR1 17 45 CN1C(=O)N[C@@H]2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC[C@@H]21 ZINC000880730420 FF On-Demand Anodyne RBP4 51 35 O=C(NC1CSC1)c1ccc(O[C@@H]2CCOC2)cc1 ZINC000880730502 CD On-Demand Anodyne EPHX2 21 41 O=C(NC1CSC1)c1ccc(O[C@H]2CCOC2)cc1 ZINC000880730503 CD On-Demand Anodyne EPHX2 21 41 O=C(NC1CSC1)[C@@H]1CCCc2cccnc21 ZINC000880730515 BD On-Demand Anodyne CXCR4 48 34 O=C(NC1CSC1)[C@H]1CCCc2cccnc21 ZINC000880730516 BD On-Demand Anodyne CXCR4 48 34 O=C(CCCCN1CCOCC1)NC1CSC1 ZINC000880730517 CC On-Demand Anodyne PAOX 19 46 O=C(CCCCN1CCOCC1)NC1CSC1 ZINC000880730517 CC On-Demand Anodyne EPHX2 18 44 CN(CC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880730526 CD On-Demand Anodyne CAPNS1 51 32 CN(CC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880730526 CD On-Demand Anodyne CAPN2 54 33 CN(CC(=O)NC1CSC1)C(=O)OCc1ccccc1 ZINC000880730526 CD On-Demand Anodyne NPR 57 38 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)S1(=O)=O ZINC000880730532 GG On-Demand Anodyne RBP4 53 33 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)S1(=O)=O ZINC000880730533 GG On-Demand Anodyne RBP4 53 33 O=C(Cn1ccc2ccccc2c1=O)NC1CSC1 ZINC000880730551 CD On-Demand Anodyne PSMB1 17 50 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne DRD4 33 48 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne ACHE 20 48 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne HRH3 32 48 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne SIGMAR1 30 52 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne SSTR5 48 40 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne CCR3 17 49 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne BDKRB1 38 45 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne UTS2R 19 41 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne SLC6A5 35 44 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne MCHR1 43 49 O=C(NC1CSC1)c1ccc(CN2CCCCC2)cc1 ZINC000880730574 CF On-Demand Anodyne NOD2 41 34 CC(=O)c1cc(C(=O)NC2CSC2)ccc1C ZINC000880730586 BE On-Demand Anodyne MAPK14 42 39 CCCOc1cccnc1C(=O)NC1CSC1 ZINC000880730591 CD On-Demand Anodyne MAP1 33 43 O=C(Cc1ccc(I)cc1)NC1CSC1 ZINC000880730592 EE On-Demand Anodyne LUXR 37 50 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NC2CSC2)c1 ZINC000880730594 CE On-Demand Anodyne MTNR1A 15 56 COc1ccc(OC)c([C@H]2C[C@H]2C(=O)NC2CSC2)c1 ZINC000880730594 CE On-Demand Anodyne MTNR1B 16 56 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NC2CSC2)c1 ZINC000880730596 CE On-Demand Anodyne MTNR1A 15 56 COc1ccc(OC)c([C@H]2C[C@@H]2C(=O)NC2CSC2)c1 ZINC000880730596 CE On-Demand Anodyne MTNR1B 16 56 CCCOc1ccc(C(=O)NC2CSC2)c(OCCCOC)c1 ZINC000880730617 EF On-Demand Anodyne PLA2G4B 49 32 CCCOc1cc(OC)ccc1C(=O)NC1CSC1 ZINC000880730650 CE On-Demand Anodyne MTNR1A 51 46 CCCOc1cc(OC)ccc1C(=O)NC1CSC1 ZINC000880730650 CE On-Demand Anodyne MTNR1B 41 46 CC(C)(C(=O)NC1CSC1)c1ccc(OC(F)(F)F)cc1 ZINC000880730651 DG On-Demand Anodyne EPHX2 45 42 CO[C@@]1(C)CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730692 EI On-Demand Anodyne EPHX2 19 40 COc1cc(C)ccc1C(=O)NC1CSC1 ZINC000880730704 BD On-Demand Anodyne HTR4 26 40 CC(C)(C)OC(=O)NCCCCCC(=O)NC1CSC1 ZINC000880730706 DE On-Demand Anodyne EPHX2 15 43 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730733 FG On-Demand Anodyne CCR3 42 38 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730734 FG On-Demand Anodyne CCR3 42 38 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C2CC2)O1 ZINC000880730739 EH On-Demand Anodyne RBP4 53 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C2CC2)O1 ZINC000880730740 EH On-Demand Anodyne RBP4 53 34 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C2CC2)O1 ZINC000880730741 EH On-Demand Anodyne RBP4 53 34 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C2CC2)O1 ZINC000880730742 EH On-Demand Anodyne RBP4 53 34 O=C(CCC(=O)c1ccccn1)NC1CSC1 ZINC000880730767 CD On-Demand Anodyne GRIN2B 17 43 C[C@@H]1OCC[C@]12CN(C(=O)Nc1cccc(F)c1C(C)(F)F)CCO2 ZINC000880730776 FG On-Demand Anodyne EPHX2 20 42 COC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730790 FG On-Demand Anodyne EPHX2 58 49 COC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880730790 FG On-Demand Anodyne CCR8 42 35 O=C(NC1CSC1)c1cccnc1I ZINC000880730798 DD On-Demand Anodyne G2YM83_BOTF4 52 35 O=C(NC1CSC1)c1ccc(-c2nnc(S)o2)cc1 ZINC000880730832 CD On-Demand Anodyne CYP73A16 58 42 COc1ccc(-n2nc(C(=O)NC3CSC3)cc2C)cc1 ZINC000880730834 DE On-Demand Anodyne RPA1 18 42 O=C(NC1CSC1)c1cccc(C(=O)NC2CSC2)c1 ZINC000880730852 DD On-Demand Anodyne KCNK3 60 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS(=O)(=O)C1 ZINC000880730859 FF On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS(=O)(=O)C1 ZINC000880730860 FF On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(CCCNC(=O)Nc2cccc(F)c2C(C)(F)F)CCCO1 ZINC000880730868 FH On-Demand Anodyne CCR3 36 43 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCC1=O ZINC000880730892 DG On-Demand Anodyne RBP4 53 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCC1=O ZINC000880730894 DG On-Demand Anodyne RBP4 53 34 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)N1CCCC1 ZINC000880730901 EG On-Demand Anodyne KCNQ2 45 35 COc1ccc(O)cc1C(=O)NC1CSC1 ZINC000880730906 BD On-Demand Anodyne HTR4 25 40 C[C@H]1C[C@@H](C)N1C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880730907 CH On-Demand Anodyne RBP4 44 33 COc1ccc2cc([C@H](C)C(=O)NC3CSC3)ccc2c1 ZINC000880730928 DG On-Demand Anodyne MTNR1A 40 39 O=C(NC1CSC1)c1ccc(O)c(F)c1 ZINC000880730952 BD On-Demand Anodyne MAPK13 63 32 O=C(Cc1ccc(CC(=O)NC2CSC2)cc1)NC1CSC1 ZINC000880730970 ED On-Demand Anodyne LUXR 44 41 O=C(NC1CSC1)c1cc(F)c(O)c(Cl)c1 ZINC000880730971 CE On-Demand Anodyne MAPK13 69 33 COCC(=O)NC1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880730982 ED On-Demand Anodyne RBP4 53 34 O=C(NC1CSC1)c1cccc(NS(=O)(=O)C(F)(F)F)c1 ZINC000880730992 ED On-Demand Anodyne KCNK3 48 35 Cc1cc(C(=O)NC2CSC2)nn1-c1ccc(F)cc1 ZINC000880731027 CE On-Demand Anodyne MAPK14 19 42 O=C(NC1CSC1)c1ccc([N+](=O)[O-])cc1O ZINC000880731029 CD On-Demand Bother KCNMA1 25 43 N#Cc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880731032 CE On-Demand Mild EZH2 52 43 O=C(NC1CSC1)c1ccc(OC2CCCC2)nc1 ZINC000880731046 CE On-Demand Anodyne HPGDS 33 41 Cc1cc([C@@H]2CCCN2C(=O)Nc2cccc(F)c2C(C)(F)F)no1 ZINC000880731056 FJ On-Demand Anodyne KCNA5 15 42 Cc1noc(C2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)n1 ZINC000880731063 EG On-Demand Anodyne RBP4 52 33 Cn1nnc2cc(C(=O)NC3CSC3)cnc21 ZINC000880731071 BC On-Demand Anodyne MAPK13 57 33 O=C(CCCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731088 DG On-Demand Anodyne PTGFR 34 43 O=C(CCCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731088 DG On-Demand Anodyne CCR2 62 40 O=C(CCCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731088 DG On-Demand Anodyne LUXR 21 53 O=C(CCc1cncc2ccccc12)NC1CSC1 ZINC000880731132 CE On-Demand Anodyne TNKS 57 34 N#Cc1ccc(C(=O)NC2CSC2)cc1Cl ZINC000880731151 CE On-Demand Mild EZH2 53 45 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880731189 CD On-Demand Anodyne PAPA1_CARPA 37 43 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880731189 CD On-Demand Anodyne CTSK 18 44 O=C(NC1CSC1)c1cccn2c(O)nnc12 ZINC000880731194 CC On-Demand Anodyne POLR1A 77 46 CCCc1c(C(=O)NC2CSC2)cnn1-c1ccc(F)cc1 ZINC000880731196 DF On-Demand Anodyne MAPK14 16 41 COCCO[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731199 EG On-Demand Anodyne RBP4 47 39 COCCO[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731199 EG On-Demand Anodyne LIPG 29 40 COCCO[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731200 EG On-Demand Anodyne RBP4 47 39 COCCO[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731200 EG On-Demand Anodyne LIPG 29 40 C[C@@H]1CSCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731213 EI On-Demand Anodyne RBP4 53 35 CO[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H]1C ZINC000880731249 EH On-Demand Anodyne RBP4 52 36 CO[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H]1C ZINC000880731251 EH On-Demand Anodyne RBP4 52 36 O=C(NC1CSC1)c1ccccc1OC(F)(F)F ZINC000880731270 CE On-Demand Anodyne KCNK3 41 48 O=C(NC1CSC1)c1ccccc1OC(F)(F)F ZINC000880731270 CE On-Demand Anodyne KCNK9 44 48 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne ACE 92 43 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne GHRHR 47 37 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MME 84 40 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne ANPEP 48 35 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MTNR1B 17 41 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MMP2 37 46 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MMP3 64 45 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MMP8 19 43 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MMP9 16 40 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne ACE2 44 38 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne LAP3 49 36 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne MMP1 24 41 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne AMP1_PLAFQ 41 40 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne NAAA 44 41 C[C@@H](CCCc1ccccc1)C(=O)NC1CSC1 ZINC000880731275 CF On-Demand Anodyne BIRC2 32 40 CO[C@@]1(C)CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731276 EH On-Demand Anodyne EPHX2 30 42 CO[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1OC ZINC000880731282 EF On-Demand Anodyne RBP4 64 38 CCn1cc(C(=O)NC2CSC2)c(=O)c2cc(Cl)ccc21 ZINC000880731285 DF On-Demand Anodyne CNR1 19 44 CCn1cc(C(=O)NC2CSC2)c(=O)c2cc(Cl)ccc21 ZINC000880731285 DF On-Demand Anodyne CNR2 44 49 CCn1cc(C(=O)NC2CSC2)c(=O)c2cc(Cl)ccc21 ZINC000880731285 DF On-Demand Anodyne UL54 43 40 O=C(NC1CSC1)c1ccc2nc(C(F)(F)F)cn2c1 ZINC000880731321 DE On-Demand Anodyne MAP3K5 50 35 C=CCOc1cc(OC)ccc1C(=O)NC1CSC1 ZINC000880731323 CE On-Demand Mild LUCI_LUCLA 15 40 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NC2CSC2)C1 ZINC000880731331 CD On-Demand Anodyne EPHX2 19 50 CN(C)C(=O)Nc1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880731339 GI On-Demand Anodyne GNRHR 43 32 CN(C)C(=O)Nc1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880731339 GI On-Demand Anodyne TRPV1 15 41 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCCO1 ZINC000880731374 EH On-Demand Anodyne RBP4 54 35 O=C(CCCCC(=O)c1ccc(F)cc1)NC1CSC1 ZINC000880731377 CF On-Demand Anodyne HDAC8 28 40 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731384 FI On-Demand Anodyne RBP4 52 33 Cn1nccc1[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731385 FI On-Demand Anodyne RBP4 52 33 Cc1nc(C(=O)NC2CSC2)c(-c2ccccc2)s1 ZINC000880731390 CF On-Demand Anodyne HCRTR1 29 41 CCCc1c(C(=O)NC2CSC2)cnn1-c1cccc(F)c1 ZINC000880731401 DF On-Demand Anodyne MAPK14 19 44 CCOc1cc(Cl)ccc1C(=O)NC1CSC1 ZINC000880731402 CF On-Demand Anodyne SSTR5 41 36 CCOc1cc(Cl)ccc1C(=O)NC1CSC1 ZINC000880731402 CF On-Demand Anodyne HCN1 42 30 CSc1cc(C(=O)NC2CSC2)ccc1F ZINC000880731409 CE On-Demand Anodyne MAPK13 47 33 Cc1cc(F)ccc1-n1ccc(C(=O)NC2CSC2)n1 ZINC000880731418 CE On-Demand Anodyne MAPK13 46 31 O=C(NC1CSC1)c1ncoc1-c1cccc(C(F)(F)F)c1 ZINC000880731449 EG On-Demand Anodyne TRPV1 16 44 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne DRD4 17 43 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne PTGER1 27 45 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne SSTR5 48 40 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne HCN1 42 30 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne HCN4 40 30 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne EZH2 43 34 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne KCNK3 26 41 CCOc1ccccc1-c1cccc(C(=O)NC2CSC2)c1 ZINC000880731467 DH On-Demand Anodyne KCNK9 20 41 Cc1cc(C(=O)NC2CSC2)nn1-c1ccc(Cl)cc1 ZINC000880731502 DF On-Demand Anodyne CNR1 52 52 Cc1cc(C(=O)NC2CSC2)nn1-c1ccc(Cl)cc1 ZINC000880731502 DF On-Demand Anodyne CNR2 23 41 Cc1cc(C(=O)NC2CSC2)nn1-c1ccc(Cl)cc1 ZINC000880731502 DF On-Demand Anodyne RPA1 16 40 CN1CCO[C@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C[C@@H]21 ZINC000880731593 FF On-Demand Anodyne RBP4 47 37 CN1CCO[C@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C[C@H]21 ZINC000880731594 FF On-Demand Anodyne RBP4 47 37 CN1CCO[C@@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C[C@@H]21 ZINC000880731595 FF On-Demand Anodyne RBP4 47 37 CN1CCO[C@@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C[C@H]21 ZINC000880731596 FF On-Demand Anodyne RBP4 47 37 O=C(CCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731600 CF On-Demand Anodyne PTGFR 32 42 O=C(CCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731600 CF On-Demand Anodyne CSNK1D 20 41 O=C(CCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731600 CF On-Demand Anodyne CCR2 69 41 O=C(CCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731600 CF On-Demand Anodyne LUXR 42 60 O=C(CCc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880731600 CF On-Demand Anodyne TRAR 17 42 O=C(NC1CSC1)c1cc(F)ccc1N1CCOCC1 ZINC000880731630 CD On-Demand Anodyne PIK3CB 17 41 O=C(Cc1ccc(F)cc1Br)NC1CSC1 ZINC000880731657 DE On-Demand Anodyne P2RX7 17 46 O=C(NC1CSC1)c1ccnc(C2CC2)c1 ZINC000880731769 BD On-Demand Anodyne MAPK13 43 35 CC(C)(C)OC(=O)N1CCC[C@H](n2cc(C(=O)NC3CSC3)cn2)C1 ZINC000880731796 FE On-Demand Anodyne MTOR 18 40 CC(C)(C)OC(=O)N1CCC[C@@H](n2cc(C(=O)NC3CSC3)cn2)C1 ZINC000880731797 FE On-Demand Anodyne MTOR 18 40 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne ACE 32 43 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CTRA_BOVIN 49 32 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CASP3 26 46 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne BMP1 20 42 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne KLK3 98 43 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CTSB 81 47 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne PAPA1_CARPA 85 49 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CYSP_TRYCR 66 45 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CTSK 64 53 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CTSL 65 51 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CAPNS1 75 43 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne HLA-DRB1 41 34 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CELA2A 41 35 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne MMP11 61 34 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CTSS 42 51 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CAPN1 108 48 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CASP1 30 46 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CAPN2 160 47 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne PLAU 16 40 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne CASP9 37 41 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne TPSAB1 46 37 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne NPR 82 39 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne NAAA 64 39 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne PSMB5 55 45 COCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731821 ED On-Demand Anodyne Q9NAW4_PLAFA 39 42 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne ACE 32 43 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CTRA_BOVIN 49 32 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CASP3 26 46 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne BMP1 20 42 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne KLK3 98 43 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CTSB 81 47 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne PAPA1_CARPA 85 49 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CYSP_TRYCR 66 45 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CTSK 64 53 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CTSL 65 51 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CAPNS1 75 43 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne HLA-DRB1 41 34 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CELA2A 41 35 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne MMP11 61 34 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CTSS 42 51 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CAPN1 108 48 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CASP1 30 46 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CAPN2 160 47 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne PLAU 16 40 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne CASP9 37 41 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne TPSAB1 46 37 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne NPR 82 39 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne NAAA 64 39 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne PSMB5 55 45 COCC[C@@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880731822 ED On-Demand Anodyne Q9NAW4_PLAFA 39 42 CC[C@@H](C(=O)NC1CSC1)c1ccc(OC)cc1 ZINC000880731824 CE On-Demand Anodyne KCNQ2 29 49 CC[C@H](C(=O)NC1CSC1)c1ccc(OC)cc1 ZINC000880731825 CE On-Demand Anodyne KCNQ2 29 49 CC(C)(C)OC(=O)N1CCC(OCC(=O)NC2CSC2)CC1 ZINC000880731832 ED On-Demand Anodyne GPR119 34 40 O=C(NC1CSC1)c1ccc(C(F)(F)F)c(F)c1 ZINC000880731846 CF On-Demand Anodyne MAPK14 38 40 O=C(NC1CSC1)c1ccc(C(F)(F)F)c(F)c1 ZINC000880731846 CF On-Demand Anodyne MAPK13 72 37 CCCc1c(C(=O)NC2CSC2)cnn1-c1ccccc1 ZINC000880731847 DF On-Demand Anodyne GPR142 43 36 Cn1cnc(-c2ccc(C(=O)NC3CSC3)cc2)n1 ZINC000880731852 CD On-Demand Anodyne MAPK13 45 32 COc1cnccc1N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880731853 GH On-Demand Anodyne HTR1A 15 46 COc1cnccc1N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880731853 GH On-Demand Anodyne PDGFRB 32 42 COc1cnccc1N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880731853 GH On-Demand Anodyne RBP4 30 46 O=C(NC1CSC1)[C@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880731863 DD On-Demand Anodyne CCR2 73 38 O=C(NC1CSC1)[C@@H](O)Cc1cccc(C(F)(F)F)c1 ZINC000880731865 DD On-Demand Anodyne CCR2 73 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1CC(C)(C)O ZINC000880731875 FG On-Demand Anodyne RBP4 46 36 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1CC(C)(C)O ZINC000880731878 FG On-Demand Anodyne RBP4 46 36 COc1ccc2[nH]c(C(=O)NC3CSC3)cc2c1 ZINC000880731885 CE On-Demand Anodyne PYGL 84 40 COc1ccc2[nH]c(C(=O)NC3CSC3)cc2c1 ZINC000880731885 CE On-Demand Anodyne PYGM 34 40 COc1ccc2[nH]c(C(=O)NC3CSC3)cc2c1 ZINC000880731885 CE On-Demand Anodyne TUBB2B 53 53 CC(C)(C)OC(=O)N1CCC2(CC1)CC(C(=O)NC1CSC1)=NO2 ZINC000880731901 FD On-Demand Anodyne GPR119 15 55 Cn1c(C(=O)NC2CSC2)cc2c(=O)n3ccccc3nc21 ZINC000880731936 DD On-Demand Anodyne INHA 40 32 Cn1c(C(=O)NC2CSC2)cc2c(=O)n3ccccc3nc21 ZINC000880731936 DD On-Demand Anodyne POLR1A 83 46 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731958 FI On-Demand Anodyne RBP4 51 33 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880731959 FI On-Demand Anodyne RBP4 51 33 O=C(Cc1cccc(OCc2cccnc2)c1)NC1CSC1 ZINC000880731990 DE On-Demand Anodyne PTAFR 20 44 O=C(Cc1cccc(OCc2cccnc2)c1)NC1CSC1 ZINC000880731990 DE On-Demand Anodyne CHRNA7 43 36 O=C(NC1CSC1)[C@H](F)Cc1ccccc1 ZINC000880731996 BD On-Demand Anodyne ACE 62 44 O=C(NC1CSC1)[C@H](F)Cc1ccccc1 ZINC000880731996 BD On-Demand Anodyne MME 118 42 O=C(NC1CSC1)[C@H](F)Cc1ccccc1 ZINC000880731996 BD On-Demand Anodyne ANPEP 45 36 O=C(NC1CSC1)[C@H](F)Cc1ccccc1 ZINC000880731996 BD On-Demand Anodyne CPA1 48 38 O=C(NC1CSC1)[C@H](F)Cc1ccccc1 ZINC000880731996 BD On-Demand Anodyne AMP1_PLAFQ 45 37 O=C(NC1CSC1)[C@@H](F)Cc1ccccc1 ZINC000880731997 BD On-Demand Anodyne ACE 62 44 O=C(NC1CSC1)[C@@H](F)Cc1ccccc1 ZINC000880731997 BD On-Demand Anodyne MME 118 42 O=C(NC1CSC1)[C@@H](F)Cc1ccccc1 ZINC000880731997 BD On-Demand Anodyne ANPEP 45 36 O=C(NC1CSC1)[C@@H](F)Cc1ccccc1 ZINC000880731997 BD On-Demand Anodyne CPA1 48 38 O=C(NC1CSC1)[C@@H](F)Cc1ccccc1 ZINC000880731997 BD On-Demand Anodyne AMP1_PLAFQ 45 37 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880732016 GF On-Demand Anodyne HLA-DRB1 62 36 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880732018 GF On-Demand Anodyne HLA-DRB1 62 36 N#Cc1ccc(C(=O)NC2CSC2)cc1O ZINC000880732021 BD On-Demand Mild EZH2 42 41 CC[C@@H](C(=O)NC1CSC1)c1ccc(F)cc1 ZINC000880732028 CF On-Demand Anodyne KCNQ2 38 47 CC[C@H](C(=O)NC1CSC1)c1ccc(F)cc1 ZINC000880732030 CF On-Demand Anodyne KCNQ2 38 47 Cn1cc(-c2ccc(F)c(C(=O)NC3CSC3)c2)cn1 ZINC000880732055 CE On-Demand Anodyne MAPK13 51 30 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880732068 FF On-Demand Mild RBP4 46 39 CN1C(=O)CC[C@H]1C(=O)NC1CSC1 ZINC000880732072 BB On-Demand Anodyne P2RX7 17 46 Cc1ccc(C[C@@H](C)C(=O)NC2CSC2)cc1 ZINC000880732118 BE On-Demand Anodyne MME 76 39 Cc1ccc(C[C@@H](C)C(=O)NC2CSC2)cc1 ZINC000880732118 BE On-Demand Anodyne ACE2 54 39 Cc1cc(C(=O)NC2CSC2)cnn1 ZINC000880732130 BC On-Demand Anodyne MAPK13 42 31 O=C(CNC(=O)c1cccc(O)c1)NC1CSC1 ZINC000880732138 CC On-Demand Anodyne CCR2 69 47 CC1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732149 CG On-Demand Anodyne RBP4 69 42 COc1ccc(Cn2cc(C(=O)NC3CSC3)cn2)cc1OC ZINC000880732156 ED On-Demand Anodyne SSTR5 62 40 COc1ccc(Cn2cc(C(=O)NC3CSC3)cn2)cc1OC ZINC000880732156 ED On-Demand Anodyne MCHR1 18 48 COC[C@@H](O)CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880732163 DE On-Demand Anodyne ADRB1 25 40 COc1nn(C)cc1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880732182 EG On-Demand Anodyne P2RY1 40 36 Cn1nnc2ccc(C(=O)NC3CSC3)cc21 ZINC000880732186 BC On-Demand Anodyne MAPK14 43 37 Cn1nnc2ccc(C(=O)NC3CSC3)cc21 ZINC000880732186 BC On-Demand Anodyne MAPK13 69 37 CC[C@]1(C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880732190 EH On-Demand Anodyne EPHX2 19 42 Cc1cc(C(=O)NC2CSC2)nn1-c1cccc(Cl)c1 ZINC000880732212 DF On-Demand Anodyne CNR1 38 43 Cc1cc(C(=O)NC2CSC2)nn1-c1cccc(Cl)c1 ZINC000880732212 DF On-Demand Anodyne CNR2 19 41 Cc1cc(C(=O)NC2CSC2)nn1-c1cccc(Cl)c1 ZINC000880732212 DF On-Demand Anodyne PTGER1 25 40 O=C(NC1CSC1)c1ncccc1C(F)(F)F ZINC000880732214 CD On-Demand Anodyne TRPV1 21 40 CN(C)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880732223 EH On-Demand Anodyne RBP4 58 41 CN(C)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880732223 EH On-Demand Anodyne SFRP1 63 35 CN(C)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880732223 EH On-Demand Anodyne WNT3 56 35 Cc1cc(C(=O)NC2CSC2)nn1-c1ccccc1Cl ZINC000880732225 DF On-Demand Anodyne CNR1 54 39 O=C(CCc1cc2ccccc2nc1O)NC1CSC1 ZINC000880732236 CE On-Demand Anodyne TNKS 63 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](CO)O1 ZINC000880732239 EF On-Demand Anodyne RBP4 51 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](CO)O1 ZINC000880732240 EF On-Demand Anodyne RBP4 51 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](CO)O1 ZINC000880732241 EF On-Demand Anodyne RBP4 51 32 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](CO)O1 ZINC000880732242 EF On-Demand Anodyne RBP4 51 32 O=C(CCCNC(=O)c1cccnc1)NC1CSC1 ZINC000880732360 CC On-Demand Anodyne TBXA2R 37 41 O=C(CCCNC(=O)c1cccnc1)NC1CSC1 ZINC000880732360 CC On-Demand Anodyne TBXAS1 76 41 O=C(CCCNC(=O)c1cccnc1)NC1CSC1 ZINC000880732360 CC On-Demand Anodyne PTAFR 15 41 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880732370 GH On-Demand Anodyne RBP4 55 38 CNC(=O)COc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732377 CC On-Demand Anodyne UPP1 56 33 CNC(=O)COc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732377 CC On-Demand Anodyne PLA2G4B 18 40 CNC(=O)COc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732377 CC On-Demand Anodyne HAO2 41 37 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne HRH2 29 41 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne UPP1 44 39 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne MTNR1A 33 41 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne PLA2G4B 52 47 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne FAAH 20 44 CCCOc1cccc(CC(=O)NC2CSC2)c1 ZINC000880732379 CE On-Demand Anodyne PDS 47 34 Cc1cc(C(=O)NC2CSC2)ccc1NC(=O)c1cccs1 ZINC000880732381 EG On-Demand Anodyne MAPK11 31 44 Cc1cc(C(=O)NC2CSC2)ccc1NC(=O)c1cccs1 ZINC000880732381 EG On-Demand Anodyne MAPK14 33 42 O=C(NC1CSC1)c1ccc2nnc(O)n2c1 ZINC000880732382 CC On-Demand Anodyne MAPK13 80 34 O=C(Cc1ccc(OCCOc2ccccc2)cc1)NC1CSC1 ZINC000880732389 EF On-Demand Anodyne ADRB1 15 40 O=C(Cc1ccc(OCCOc2ccccc2)cc1)NC1CSC1 ZINC000880732389 EF On-Demand Anodyne LTA4H 76 43 O=C(Cc1ccc(OCCOc2ccccc2)cc1)NC1CSC1 ZINC000880732389 EF On-Demand Anodyne CYSLTR2 63 37 O=C(Cc1ccc(OCCOc2ccccc2)cc1)NC1CSC1 ZINC000880732389 EF On-Demand Anodyne PLA2G4B 67 39 O=C(Cc1ccc(OCCOc2ccccc2)cc1)NC1CSC1 ZINC000880732389 EF On-Demand Anodyne TRAR 41 33 CC(C)(C)OC(=O)N1CCC(CCC(=O)NC2CSC2)CC1 ZINC000880732416 EF On-Demand Anodyne GPR119 34 41 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732418 DD On-Demand Anodyne REN 24 41 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732418 DD On-Demand Anodyne POLG_HCV1 31 51 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732418 DD On-Demand Anodyne FPR1 46 38 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732419 DD On-Demand Anodyne REN 24 41 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732419 DD On-Demand Anodyne POLG_HCV1 31 51 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NC1CSC1 ZINC000880732419 DD On-Demand Anodyne FPR1 46 38 C[C@@H](Oc1cccc(CO)c1)C(=O)NC1CSC1 ZINC000880732473 CD On-Demand Anodyne FAAH 16 46 COc1cccc(C(=O)NC2CSC2)c1F ZINC000880732495 BD On-Demand Anodyne DRD2 20 44 COc1cccc(C(=O)NC2CSC2)c1F ZINC000880732495 BD On-Demand Anodyne DRD3 19 47 COc1cccc(C(=O)NC2CSC2)c1F ZINC000880732495 BD On-Demand Anodyne KCNK3 39 40 COc1cccc(C(=O)NC2CSC2)c1F ZINC000880732495 BD On-Demand Anodyne KCNK9 34 40 O=C(Nc1ccc(N2CCOCC2)cn1)C12C[C@H]3C[C@@H](CC(Br)(C3)C1)C2 ZINC000880732517 HH On-Demand Anodyne STAT6 50 31 O=C(NC1CSC1)C1=Cc2cc(F)ccc2OC1 ZINC000880732522 CD On-Demand Anodyne ALOX12 15 43 Cn1cc([C@@H]2CCCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)cn1 ZINC000880732524 FI On-Demand Anodyne RBP4 52 33 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880732537 DD On-Demand Anodyne PAPA1_CARPA 35 59 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880732537 DD On-Demand Anodyne CTSK 15 59 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880732537 DD On-Demand Anodyne FPR1 33 47 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne MAOB 16 41 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne MAPK11 26 41 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne MAPK14 36 41 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne MAPK13 69 38 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne SSTR3 22 44 O=C(NC1CSC1)c1ccc(Cl)c(F)c1 ZINC000880732542 BE On-Demand Anodyne ENV 46 43 COC(=O)C1=NOC2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)C1 ZINC000880732543 GG On-Demand Anodyne TRPM8 31 44 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880732547 GH On-Demand Anodyne CACNA1H 40 31 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880732548 GH On-Demand Anodyne CACNA1H 40 31 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880732549 GH On-Demand Anodyne CACNA1H 40 31 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880732550 GH On-Demand Anodyne CACNA1H 40 31 O=C(NC1CSC1)c1cnc2ccccn12 ZINC000880732553 BD On-Demand Anodyne EPHB3 28 53 CC1(C)C[C@@H]1C(=O)NC1CSC1 ZINC000880732555 AD On-Demand Anodyne DPEP1 89 42 CN1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1=O ZINC000880732560 DE On-Demand Anodyne TRPV1 15 42 O=C(NC1CSC1)c1cccc2nc(O)oc12 ZINC000880732623 CD On-Demand Anodyne HTR3A 26 45 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1CCO ZINC000880732632 EE On-Demand Anodyne RBP4 51 32 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1CCO ZINC000880732633 EE On-Demand Anodyne RBP4 51 32 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1c1ncc[nH]1 ZINC000880732640 FG On-Demand Anodyne RBP4 49 30 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1c1ncc[nH]1 ZINC000880732641 FG On-Demand Anodyne RBP4 49 30 O=C(NC1CSC1)c1cccc(OCC(F)(F)F)c1 ZINC000880732652 CE On-Demand Anodyne DRD4 41 31 O=C(NC1CSC1)c1cccc(OCC(F)(F)F)c1 ZINC000880732652 CE On-Demand Anodyne CCR2 42 36 CN1CC[C@@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732679 DG On-Demand Anodyne CCR3 45 41 CN1CC[C@@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732679 DG On-Demand Anodyne CACNA1I 64 37 CN1CC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732680 DG On-Demand Anodyne CCR3 45 41 CN1CC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732680 DG On-Demand Anodyne CACNA1I 64 37 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1c1nccn1C ZINC000880732681 GG On-Demand Anodyne RBP4 49 30 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1c1nccn1C ZINC000880732682 GG On-Demand Anodyne RBP4 49 30 C[C@@H](Cc1cccc(Cl)c1)C(=O)NC1CSC1 ZINC000880732689 CF On-Demand Anodyne AVPR1A 32 41 C[C@@H](Cc1cccc(Cl)c1)C(=O)NC1CSC1 ZINC000880732689 CF On-Demand Anodyne CTSL 20 45 C[C@@H](Cc1cccc(Cl)c1)C(=O)NC1CSC1 ZINC000880732689 CF On-Demand Anodyne CTSV 36 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732717 FG On-Demand Anodyne EPHX2 45 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732717 FG On-Demand Anodyne CCR8 77 43 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732718 FG On-Demand Anodyne EPHX2 45 45 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880732718 FG On-Demand Anodyne CCR8 77 43 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne ACE 71 53 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne MME 67 53 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne LTA4H 21 47 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne FCER2 44 41 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CASP3 44 35 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CASP8 50 34 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CTSB 17 43 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CYSP_TRYCR 43 38 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CTSK 21 40 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CAPN1 34 43 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne CAPN2 37 43 C[C@H](CSCc1ccccc1)C(=O)NC1CSC1 ZINC000880732719 CF On-Demand Anodyne FPR1 45 34 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne ACE 76 39 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne OPRM1 36 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne OPRD1 33 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CELA1 23 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne MME 138 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne ANPEP 55 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne TACR1 17 53 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSD 30 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne PGC 71 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CMA1 37 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTRA_BOVIN 30 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne FCER2 94 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CASP3 19 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSB 80 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne PAPA1_CARPA 100 63 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CYSP_TRYCR 80 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CCKAR 74 53 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSK 51 62 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSL 75 63 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CACNA1B 65 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne PGA 41 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne TIMP3 90 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne TACR3 23 52 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CAPNS1 70 37 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne MMP3 23 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne HLA-DRB1 63 49 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne REN 112 56 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne REN1 37 48 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CCKBR 29 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSS 35 63 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CAPN1 104 52 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne MMP9 24 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CAPN2 99 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTSE 18 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne ACE2 69 39 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne KLK5 24 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne MMP1 33 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne FPR1 99 55 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne CTRB_BOVIN 58 46 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne NAAA 40 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne BLA1_STEMA 46 34 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880732725 EE On-Demand Anodyne NPFFR1 41 32 O=C(Cc1ccc(OCc2ccccn2)cc1)NC1CSC1 ZINC000880732730 DE On-Demand Anodyne GRIN2B 16 42 O=C(Cc1ccc(OCc2ccccn2)cc1)NC1CSC1 ZINC000880732730 DE On-Demand Anodyne SMO 20 41 CCC(=O)N1CC[C@@H](C(=O)NC2CSC2)C1 ZINC000880732733 BC On-Demand Anodyne EPHX2 29 48 CCC(=O)N1CC[C@H](C(=O)NC2CSC2)C1 ZINC000880732734 BC On-Demand Anodyne EPHX2 29 48 CC(C)(C)OC(=O)N[C@@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732751 EF On-Demand Anodyne CTSK 16 49 CC(C)(C)OC(=O)N[C@@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732751 EF On-Demand Anodyne REN 41 40 CC(C)(C)OC(=O)N[C@@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732751 EF On-Demand Anodyne FPR1 48 38 CC(C)(C)OC(=O)N[C@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732752 EF On-Demand Anodyne CTSK 16 49 CC(C)(C)OC(=O)N[C@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732752 EF On-Demand Anodyne REN 41 40 CC(C)(C)OC(=O)N[C@H](CC(=O)NC1CSC1)c1ccccc1 ZINC000880732752 EF On-Demand Anodyne FPR1 48 38 CC(=O)Nc1ccn([C@@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)n1 ZINC000880732762 GH On-Demand Anodyne RBP4 49 33 CC(=O)Nc1ccn([C@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)n1 ZINC000880732763 GH On-Demand Anodyne RBP4 49 33 O=C(Cc1cccc(OC(F)(F)F)c1)NC1CSC1 ZINC000880732786 CE On-Demand Anodyne DHODH 15 40 O=C(Cc1cccc(OC(F)(F)F)c1)NC1CSC1 ZINC000880732786 CE On-Demand Anodyne CSNK1D 20 44 O=C(Cc1cccc(OC(F)(F)F)c1)NC1CSC1 ZINC000880732786 CE On-Demand Anodyne HAO2 15 48 O=C(NC1CSC1)c1ccc(OCC(F)F)nc1 ZINC000880732805 CD On-Demand Anodyne HPGDS 35 42 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H]1O ZINC000880732814 DG On-Demand Anodyne RBP4 55 38 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H]1O ZINC000880732815 DG On-Demand Anodyne RBP4 55 38 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H]1O ZINC000880732816 DG On-Demand Anodyne RBP4 55 38 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@@H]1O ZINC000880732817 DG On-Demand Anodyne RBP4 55 38 COCCOc1cc(C(=O)NC2CSC2)nc2ccccc12 ZINC000880732823 DE On-Demand Anodyne TNKS 45 32 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)Nc2ccc(N3CCOCC3)cn2)c1 ZINC000880732826 JH On-Demand Anodyne F10 47 32 O=C(Cc1cccc(OCC(F)(F)F)c1)NC1CSC1 ZINC000880732831 DE On-Demand Anodyne PDS 43 36 O=C(NC1CC1)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880732844 CD On-Demand Anodyne MAPK11 34 43 O=C(NC1CC1)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880732844 CD On-Demand Anodyne MAPK14 45 43 O=C(NC1CC1)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880732844 CD On-Demand Anodyne MAPK13 67 35 O=C(NC1CC1)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880732844 CD On-Demand Anodyne ST14 17 40 O=C(NC1CSC1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000880732845 CG On-Demand Anodyne MAPK14 39 40 O=C(NC1CSC1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000880732845 CG On-Demand Anodyne RAF1 23 44 O=C(NC1CSC1)c1ccc(Cl)c(C(F)(F)F)c1 ZINC000880732845 CG On-Demand Anodyne MAPK13 51 37 Cc1c(CC(=O)NC2CSC2)cccc1[N+](=O)[O-] ZINC000880732847 CD On-Demand Bother COLA 102 33 O=C(NC1CSC1)c1c[nH]c2cccc([N+](=O)[O-])c12 ZINC000880732859 CD On-Demand Bother GABRA1 16 40 O=C(NC1CSC1)c1c[nH]c2cccc([N+](=O)[O-])c12 ZINC000880732859 CD On-Demand Bother GABRA2 16 40 NS(=O)(=O)c1cc(Cl)c(F)c(C(=O)NC2CSC2)c1 ZINC000880732865 DC On-Demand Anodyne CA2 17 44 NS(=O)(=O)c1cc(Cl)c(F)c(C(=O)NC2CSC2)c1 ZINC000880732865 DC On-Demand Anodyne CA7 22 41 NS(=O)(=O)c1cc(Cl)c(F)c(C(=O)NC2CSC2)c1 ZINC000880732865 DC On-Demand Anodyne CA4 20 46 O=C(NC1CSC1)c1ccc(S[C@@H]2CCOC2=O)cc1 ZINC000880732871 DD On-Demand Anodyne TRAR 62 32 O=C(NC1CSC1)c1ccc(S[C@H]2CCOC2=O)cc1 ZINC000880732872 DD On-Demand Anodyne TRAR 62 32 O=C(NC1CSC1)[C@H](c1ccccc1)C1CC1 ZINC000880732882 BE On-Demand Anodyne C3AR1 38 43 O=C(NC1CSC1)[C@@H](c1ccccc1)C1CC1 ZINC000880732883 BE On-Demand Anodyne C3AR1 38 43 CCOc1ccccc1C(F)(F)C(=O)NC1CSC1 ZINC000880732884 CE On-Demand Anodyne HCN1 42 30 CCOc1ccccc1C(F)(F)C(=O)NC1CSC1 ZINC000880732884 CE On-Demand Anodyne KCNK3 19 41 CCOc1ccccc1C(F)(F)C(=O)NC1CSC1 ZINC000880732884 CE On-Demand Anodyne KCNK9 19 41 CC(=O)CCCCCCC(=O)NC1CSC1 ZINC000880732891 BE On-Demand Anodyne PAOX 43 37 O=C1CCc2cc(C(=O)NC3CSC3)c(F)cc2N1 ZINC000880732905 CD On-Demand Anodyne PKM 33 43 C[C@H](Cc1ccccc1Cl)C(=O)NC1CSC1 ZINC000880732909 CF On-Demand Anodyne ANPEP 18 43 C[C@H](Cc1ccccc1Cl)C(=O)NC1CSC1 ZINC000880732909 CF On-Demand Anodyne CXCL8 46 34 C[C@@H](Cc1ccccc1Cl)C(=O)NC1CSC1 ZINC000880732910 CF On-Demand Anodyne ANPEP 18 43 C[C@@H](Cc1ccccc1Cl)C(=O)NC1CSC1 ZINC000880732910 CF On-Demand Anodyne CXCL8 46 34 O=C(NC1CSC1)c1cn(Cc2cccc(F)c2)nn1 ZINC000880732924 CD On-Demand Anodyne CCR3 19 42 CN1CCC(N2CCC(NC(=O)Nc3cccc(F)c3C(C)(F)F)CC2)CC1 ZINC000880732927 GH On-Demand Anodyne SLC6A5 21 44 CN1CCC(N2CCC(NC(=O)Nc3cccc(F)c3C(C)(F)F)CC2)CC1 ZINC000880732927 GH On-Demand Anodyne EPHX2 39 43 COC(=O)c1cn(C2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)nn1 ZINC000880732928 GE On-Demand Anodyne RBP4 42 30 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880732942 FG On-Demand Anodyne CCR3 43 36 COc1cc2c(cc1OC)CN(CC(=O)NC1CSC1)CC2 ZINC000880732967 DD On-Demand Anodyne SLC18A2 48 34 COc1cc2c(cc1OC)CN(CC(=O)NC1CSC1)CC2 ZINC000880732967 DD On-Demand Anodyne ABCB1B 65 39 COc1cc2c(cc1OC)CN(CC(=O)NC1CSC1)CC2 ZINC000880732967 DD On-Demand Anodyne ABCB1 25 46 COc1cccc(OC)c1CC(=O)NC1CSC1 ZINC000880732977 CD On-Demand Anodyne KCNA3 28 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne F2 75 44 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne PLG 33 46 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne PRSS1 33 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne ACE 51 51 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne FKBP1A 63 45 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne OPRM1 30 44 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne OPRD1 16 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne CELA1 35 58 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne GRIN2B 25 43 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne ELANE 43 47 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne TACR1 15 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne CTRA_BOVIN 65 36 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne TRY1_BOVIN 94 39 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne CTSG 45 36 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne CTSL 18 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne DPP4 19 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne PREP 107 58 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne CELA2A 54 36 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne LGMN 102 58 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne ACE2 20 45 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne KLK5 30 52 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne XIAP 57 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne BRCA1 62 33 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne SLC12A5 66 39 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne Q9NAW4_PLAFA 39 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880732983 DE On-Demand Anodyne TMPRSS11D 69 40 Cc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880732984 CF On-Demand Anodyne MAPK14 24 40 Cc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880732984 CF On-Demand Anodyne MAPK13 49 32 Cc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880732984 CF On-Demand Anodyne SCN10A 54 49 COc1ccc(OCC(=O)NC2CSC2)cc1C ZINC000880733004 CD On-Demand Anodyne PPARD 51 39 COCCSc1ccc([N+](=O)[O-])cc1C(=O)NC1CSC1 ZINC000880733067 EE On-Demand Bother CACNA1D 45 33 COC[C@@H]1CCCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880733071 EI On-Demand Anodyne RBP4 45 33 CCOC(=O)CCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733087 GJ On-Demand Anodyne EPHX2 15 41 CCOC(=O)CCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733087 GJ On-Demand Anodyne CCR8 61 39 O=C(Cc1cccnc1)NC1CSC1 ZINC000880733088 BC On-Demand Anodyne TBXAS1 44 44 O=C(Cc1cccnc1)NC1CSC1 ZINC000880733088 BC On-Demand Anodyne CHRNA7 50 39 O=C(Cc1cccnc1)NC1CSC1 ZINC000880733088 BC On-Demand Anodyne C3AR1 39 40 O=C(Cc1cccnc1)NC1CSC1 ZINC000880733088 BC On-Demand Anodyne NAMPT 46 37 O=C(CNC(=O)c1ccccc1C(F)(F)F)NC1CSC1 ZINC000880733116 DD On-Demand Anodyne CCR2 67 40 O=C(CNC(=O)c1ccccc1C(F)(F)F)NC1CSC1 ZINC000880733116 DD On-Demand Anodyne RBP4 45 34 COc1cccc([C@@H](C)CC(=O)NC2CSC2)c1 ZINC000880733120 CE On-Demand Anodyne MTNR1A 39 41 COc1cccc([C@@H](C)CC(=O)NC2CSC2)c1 ZINC000880733120 CE On-Demand Anodyne MTNR1B 40 41 COc1cccc([C@H](C)CC(=O)NC2CSC2)c1 ZINC000880733121 CE On-Demand Anodyne MTNR1A 39 41 COc1cccc([C@H](C)CC(=O)NC2CSC2)c1 ZINC000880733121 CE On-Demand Anodyne MTNR1B 40 41 COc1cccc(C(=O)NC2CSC2)n1 ZINC000880733135 BC On-Demand Anodyne ALS 55 31 COc1cc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)ncn1 ZINC000880733155 GG On-Demand Anodyne PDGFRB 54 40 COc1cc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)ncn1 ZINC000880733155 GG On-Demand Anodyne RBP4 32 44 O=C(CCCOc1ccc2c(c1)OCO2)NC1CSC1 ZINC000880733159 CD On-Demand Anodyne EDNRB 53 41 O=C(CCCOc1ccc2c(c1)OCO2)NC1CSC1 ZINC000880733159 CD On-Demand Anodyne EDNRA 51 41 CN(C)C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880733179 EG On-Demand Anodyne RBP4 52 36 CC[C@@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733198 DG On-Demand Anodyne KCNQ2 39 54 CC[C@@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733198 DG On-Demand Anodyne CCR2 66 39 CC[C@@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733198 DG On-Demand Anodyne PDS 43 35 CC[C@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733199 DG On-Demand Anodyne KCNQ2 39 54 CC[C@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733199 DG On-Demand Anodyne CCR2 66 39 CC[C@H](C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733199 DG On-Demand Anodyne PDS 43 35 CC(C)[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880733212 EH On-Demand Anodyne RBP4 51 34 COCCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880733215 CD On-Demand Anodyne CYSLTR2 53 37 COCCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880733215 CD On-Demand Anodyne HRH3 17 44 COCCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880733215 CD On-Demand Anodyne PLA2G4B 83 40 COCCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880733215 CD On-Demand Anodyne SLC6A5 36 41 O=C(COc1ccc(O)cc1)NC1CSC1 ZINC000880733232 BD On-Demand Anodyne TRAR 35 42 O=C(NC1CSC1)C1(Cc2ccccc2)CCC1 ZINC000880733252 CF On-Demand Anodyne SLC12A5 42 33 O=C(Cc1ccc(F)cc1Cl)NC1CSC1 ZINC000880733264 CE On-Demand Anodyne P2RX7 86 46 CC(=O)[C@H](C)CCCCC(=O)NC1CSC1 ZINC000880733270 BE On-Demand Anodyne NOD1 43 34 CC(=O)[C@@H](C)CCCCC(=O)NC1CSC1 ZINC000880733271 BE On-Demand Anodyne NOD1 43 34 O=C(Cn1cc(-c2ccccc2)nn1)NC1CSC1 ZINC000880733280 CD On-Demand Anodyne FIMH 19 45 O=C(CCC(=O)N1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880733282 ED On-Demand Anodyne SSTR1 42 39 O=C(CCC(=O)N1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880733282 ED On-Demand Anodyne ADAM10 37 40 O=C(CCc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880733289 CD On-Demand Bother CACNA1C 52 36 O=C(CCc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880733289 CD On-Demand Bother CACNA1D 82 36 O=C(CCc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880733289 CD On-Demand Bother LUXR 46 61 O=C(CCc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880733289 CD On-Demand Bother TRAR 23 48 CC(C)(C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733296 DG On-Demand Anodyne NPY2R 16 42 CC(C)(C(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880733296 DG On-Demand Anodyne CCR2 42 38 CC(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880733303 BD On-Demand Anodyne KCNK3 74 37 CN1CCC(C)(CNC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733337 EH On-Demand Anodyne P2RY1 47 33 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne TACR1 15 42 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MPO 64 35 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MC5R 51 39 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MMP2 17 42 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MMP8 28 42 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne GRPR 59 35 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne GHSR 25 45 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MMP9 17 42 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne MC1R 49 39 CC(=O)N[C@@H](Cc1c[nH]c2cc(F)ccc12)C(=O)NC1CSC1 ZINC000880733339 ED On-Demand Anodyne KISS1R 40 33 CC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733346 EH On-Demand Anodyne CACNA1H 51 33 CC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733346 EH On-Demand Anodyne RBP4 46 35 CC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733346 EH On-Demand Anodyne TRPM8 28 40 COC(=O)c1ccc(C(=O)NC2CSC2)cc1F ZINC000880733359 CD On-Demand Anodyne MAPK13 62 34 O=C(NC1CSC1)c1cc(F)cc(Cl)c1 ZINC000880733364 BE On-Demand Anodyne CACNA1H 17 43 O=C(NC1CSC1)c1cc(F)cc(Cl)c1 ZINC000880733364 BE On-Demand Anodyne CACNA1I 53 33 O=C(NC1CSC1)c1cccn2c(I)cnc12 ZINC000880733367 FD On-Demand Anodyne POLR1A 60 42 O=C(NC1CSC1)c1cccc(OC(F)(F)F)c1 ZINC000880733369 CE On-Demand Anodyne DRD4 40 31 O=C(NC1CSC1)c1cccc(OC(F)(F)F)c1 ZINC000880733369 CE On-Demand Anodyne DHODH 18 43 O=C(NC1CSC1)c1cccc(OC(F)(F)F)c1 ZINC000880733369 CE On-Demand Anodyne EPHX2 21 47 O=C(NC1CSC1)c1cccc(OC(F)(F)F)c1 ZINC000880733369 CE On-Demand Anodyne TAAR1 15 41 COc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880733379 DF On-Demand Anodyne CYP11B1 16 53 COc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880733379 DF On-Demand Anodyne CYP11B2 33 53 COc1ccc(-c2cncc(C(=O)NC3CSC3)c2)cc1 ZINC000880733379 DF On-Demand Anodyne SCN10A 55 40 O=C(NC1CSC1)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880733412 DD On-Demand Anodyne PREP 18 40 O=C(NC1CSC1)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880733412 DD On-Demand Anodyne EPHX2 42 74 O=C(NC1CSC1)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880733412 DD On-Demand Anodyne SFRP1 36 40 O=C(NC1CSC1)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880733412 DD On-Demand Anodyne L3MBTL3 92 42 CC(=O)Nc1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880733414 CE On-Demand Anodyne ENV 43 39 Cc1nnc(-c2cccc(C(=O)NC3CSC3)c2)o1 ZINC000880733415 CD On-Demand Anodyne MAPK11 26 46 Cc1nnc(-c2cccc(C(=O)NC3CSC3)c2)o1 ZINC000880733415 CD On-Demand Anodyne MAPK14 25 56 Cc1nnc(-c2cccc(C(=O)NC3CSC3)c2)o1 ZINC000880733415 CD On-Demand Anodyne MAPK13 42 32 C[C@H](CC(=O)NC1CSC1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880733419 EF On-Demand Anodyne GPR119 30 47 C[C@@H](CC(=O)NC1CSC1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880733423 EF On-Demand Anodyne GPR119 30 47 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCC2)ccc1Cl ZINC000880733427 ED On-Demand Anodyne TGM2 43 36 O=C(CSc1nccc2ccccc12)NC1CSC1 ZINC000880733428 CF On-Demand Anodyne TNKS 57 35 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)NC2CCCC2)C1 ZINC000880733451 DD On-Demand Anodyne EPHX2 24 44 O=C(NC1CSC1)[C@H]1CCCN(C(=O)NC2CCCC2)C1 ZINC000880733452 DD On-Demand Anodyne EPHX2 24 44 COC(=O)C1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733466 FE On-Demand Anodyne CACNA1H 50 32 COC(=O)C1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733466 FE On-Demand Anodyne EPHX2 21 40 CO[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880733467 DH On-Demand Anodyne RBP4 52 34 O=C(CCc1ccc(Br)cc1)NC1CSC1 ZINC000880733500 DF On-Demand Anodyne LUXR 38 43 O=C(CCc1ccc(Br)cc1)NC1CSC1 ZINC000880733500 DF On-Demand Anodyne TRAR 28 54 C[C@]1(C(=O)NC2CSC2)CCc2ccccc2C1 ZINC000880733503 CE On-Demand Anodyne MME 15 42 C[C@@]1(C(=O)NC2CSC2)CCc2ccccc2C1 ZINC000880733504 CE On-Demand Anodyne MME 15 42 CC(C)(C)OC(=O)NC[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880733512 EF On-Demand Anodyne FPR1 47 36 O=C(Cc1ccc(F)cc1F)NC1CSC1 ZINC000880733526 BD On-Demand Anodyne P2RX7 28 40 O=C(Cc1cccc(I)c1)NC1CSC1 ZINC000880733532 EE On-Demand Anodyne SIGMAR1 16 55 O=C(Cc1cccc(I)c1)NC1CSC1 ZINC000880733532 EE On-Demand Anodyne LUXR 31 44 COc1cc(C)c(C(=O)NC2CSC2)cc1OC ZINC000880733533 CD On-Demand Anodyne HTR4 27 42 C[C@@H](Cc1ccc(F)c(Br)c1)C(=O)NC1CSC1 ZINC000880733567 EF On-Demand Anodyne LEF 45 33 C[C@H]1CCN(c2cc(C(=O)NC3CSC3)ccn2)C1 ZINC000880733569 CD On-Demand Anodyne MAPK13 42 34 C[C@@H]1CCN(c2cc(C(=O)NC3CSC3)ccn2)C1 ZINC000880733570 CD On-Demand Anodyne MAPK13 42 34 CC(C)(C)OC(=O)NC[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880733583 EF On-Demand Anodyne FPR1 47 36 O=C(NC1CSC1)c1ccccc1NCc1cccnc1 ZINC000880733587 CF On-Demand Anodyne KIT 19 42 O=C(NC1CSC1)c1ccccc1NCc1cccnc1 ZINC000880733587 CF On-Demand Anodyne CHRNA7 42 38 O=C(NC1CSC1)c1ccccc1NCc1cccnc1 ZINC000880733587 CF On-Demand Anodyne BRAF 17 42 O=C(NC1CSC1)c1ccccc1NCc1cccnc1 ZINC000880733587 CF On-Demand Anodyne NAMPT 46 37 O=C(NC1CSC1)c1cc(OCc2ccccc2)ccn1 ZINC000880733598 DF On-Demand Anodyne FAAH 15 41 O=C(NC1CSC1)c1cc(F)c(O)c(F)c1 ZINC000880733601 BD On-Demand Anodyne MAPK13 66 32 CC(C)(C)C(=O)Nc1ccc(F)c(C(=O)NC2CSC2)c1 ZINC000880733611 DF On-Demand Anodyne NPY2R 17 41 O=C(NC1CSC1)[C@@H]1CCN(C2CCCCC2)C1 ZINC000880733616 CD On-Demand Anodyne EPHX2 18 42 O=C(NC1CSC1)[C@H]1CCN(C2CCCCC2)C1 ZINC000880733617 CD On-Demand Anodyne EPHX2 18 42 COc1cc2c(cc1OC)CN(C(=O)CCC(=O)NC1CSC1)CC2 ZINC000880733626 FD On-Demand Anodyne ABCB1 16 48 O=C(NC1CSC1)c1ccc(OC2CCC2)cc1 ZINC000880733631 CE On-Demand Anodyne EPHX2 28 45 O=C(NC1CSC1)c1ccc(OC2CCC2)cc1 ZINC000880733631 CE On-Demand Anodyne PLAU 19 40 O=C(NC1CSC1)c1ccc(OC2CCC2)cc1 ZINC000880733631 CE On-Demand Anodyne ST14 16 40 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC[C@H]1C ZINC000880733683 DI On-Demand Anodyne RBP4 58 39 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1C ZINC000880733684 DI On-Demand Anodyne RBP4 58 39 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1C ZINC000880733685 DI On-Demand Anodyne RBP4 58 39 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C ZINC000880733686 DI On-Demand Anodyne RBP4 58 39 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCN1S(C)(=O)=O ZINC000880733706 GE On-Demand Anodyne RBP4 51 36 Cc1n[nH]c(C)c1CCC(=O)NC1CSC1 ZINC000880733709 BD On-Demand Anodyne HAO2 63 35 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1O ZINC000880733711 DG On-Demand Anodyne RBP4 53 34 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1O ZINC000880733712 DG On-Demand Anodyne RBP4 53 34 O=C(COC/C=C\c1ccccc1)NC1CSC1 ZINC000880733726 CD On-Demand Anodyne PLM1_PLAFA 22 41 O=C(COC/C=C/c1ccccc1)NC1CSC1 ZINC000880733727 CD On-Demand Anodyne PLM1_PLAFA 22 41 O=C(NC1CSC1)c1ccc(F)c(Cl)c1 ZINC000880733731 BE On-Demand Anodyne SSTR3 20 41 COC(=O)c1cn([C@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)nn1 ZINC000880733739 GF On-Demand Anodyne RBP4 33 42 COC(=O)c1cn([C@@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)nn1 ZINC000880733740 GF On-Demand Anodyne RBP4 33 42 CC(=O)N1CCc2c(NC(=O)Nc3cccc(F)c3C(C)(F)F)cccc21 ZINC000880733748 GI On-Demand Anodyne P2RY1 49 33 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733755 DJ On-Demand Anodyne CACNA1H 58 36 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733755 DJ On-Demand Anodyne EPHX2 26 40 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733755 DJ On-Demand Anodyne RBP4 48 38 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733755 DJ On-Demand Anodyne TRPM8 34 42 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880733783 DH On-Demand Anodyne RBP4 55 35 C[C@H]1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880733820 EI On-Demand Anodyne EPHX2 15 42 C[C@@H]1CC(NC(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880733822 EI On-Demand Anodyne EPHX2 15 42 CCC1(O)CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880733831 EI On-Demand Anodyne EPHX2 40 44 O=C(CSc1nnc(-c2ccncc2)n1Cc1ccco1)NC1CSC1 ZINC000880733844 GE On-Demand Anodyne HCRTR2 17 49 O=C(NC1CSC1)c1ccc(N2CCCCC2)cc1 ZINC000880733846 CF On-Demand Anodyne L3MBTL3 19 40 O=C(NC1CSC1)c1ccccc1Cn1cncn1 ZINC000880733860 CD On-Demand Anodyne HIS3 66 37 COCCOC1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880733871 EF On-Demand Anodyne RBP4 51 33 O=C(NC1CSC1)[C@@H]1CN(Cc2nc(O)c3ccccc3n2)CCO1 ZINC000880733886 FC On-Demand Anodyne TNKS 57 32 O=C(NC1CSC1)[C@H]1CN(Cc2nc(O)c3ccccc3n2)CCO1 ZINC000880733887 FC On-Demand Anodyne TNKS 57 32 O=C(Cc1ccc(F)c(F)c1)NC1CSC1 ZINC000880733915 BD On-Demand Anodyne LUXR 30 40 O=C(CSc1nnc(-c2cccnc2)n1Cc1ccco1)NC1CSC1 ZINC000880733929 GE On-Demand Anodyne HCRTR2 16 47 CNC(=O)[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880733935 ED On-Demand Anodyne RBP4 46 34 CNC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880733936 ED On-Demand Anodyne RBP4 46 34 Cc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880733950 BE On-Demand Anodyne MAPK11 33 42 Cc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880733950 BE On-Demand Anodyne MAPK14 48 42 Cc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880733950 BE On-Demand Anodyne MAPK13 51 38 O=C(CSc1nnc(-c2ccco2)n1Cc1ccco1)NC1CSC1 ZINC000880733953 GF On-Demand Anodyne HCRTR2 17 51 O=C(CNC(=O)c1cccnc1)NC1CSC1 ZINC000880733969 CC On-Demand Anodyne TBXAS1 40 38 O=C(CNC(=O)c1cccnc1)NC1CSC1 ZINC000880733969 CC On-Demand Anodyne CCR2 47 46 Cc1ncsc1-c1nc2ccccc2n1CC(=O)NC1CSC1 ZINC000880733986 EF On-Demand Anodyne IMDH_CRYPV 40 42 CC(C)(C)CNC(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880734008 DE On-Demand Anodyne MAPK11 15 46 CC(C)[C@H]1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734022 EI On-Demand Anodyne EPHX2 18 40 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734026 FH On-Demand Anodyne RBP4 56 37 Cn1ccnc1[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734027 FH On-Demand Anodyne RBP4 56 37 Cc1cncc(C(=O)NC2CSC2)c1 ZINC000880734034 BD On-Demand Anodyne SSTR5 35 48 CN(CCCC(=O)NC1CSC1)C1=NS(=O)(=O)c2ccccc21 ZINC000880734046 FD On-Demand Anodyne KCNA3 28 46 C[C@]1(C(=O)NC2CSC2)CCCN(C(=O)c2ccccc2)C1 ZINC000880734052 DE On-Demand Anodyne EPHX2 16 40 C[C@@]1(C(=O)NC2CSC2)CCCN(C(=O)c2ccccc2)C1 ZINC000880734053 DE On-Demand Anodyne EPHX2 16 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1O ZINC000880734054 DF On-Demand Anodyne RBP4 55 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1O ZINC000880734055 DF On-Demand Anodyne RBP4 55 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1O ZINC000880734056 DF On-Demand Anodyne RBP4 55 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1O ZINC000880734057 DF On-Demand Anodyne RBP4 55 35 COc1ccc(Cl)cc1NCCC(=O)NC1CSC1 ZINC000880734065 DE On-Demand Anodyne HTR4 16 40 COc1ccc(Cl)cc1NCCC(=O)NC1CSC1 ZINC000880734065 DE On-Demand Anodyne CPT1A 44 31 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne ACE 15 41 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MME 22 41 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MC5R 54 39 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MMP2 19 45 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MMP8 30 45 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne GRPR 64 36 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne ECE1 41 41 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne GHSR 25 46 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MMP9 18 45 CC(=O)N[C@@H](Cc1c[nH]c2ccc(Br)cc12)C(=O)NC1CSC1 ZINC000880734087 GE On-Demand Anodyne MC1R 53 39 CN(CC(=O)NC1CSC1)c1ccccc1[N+](=O)[O-] ZINC000880734099 CD On-Demand Bother COLA 72 33 CCC[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734111 EH On-Demand Anodyne RBP4 53 33 CCC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734112 EH On-Demand Anodyne RBP4 53 33 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne CCKAR 15 49 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne CYP51A1 21 40 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne PYGL 93 44 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne PLD1 17 41 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne PYGM 30 44 O=C(CNC(=O)c1cc2ccccc2[nH]1)NC1CSC1 ZINC000880734114 CD On-Demand Anodyne PLD2 18 42 Cc1cncc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880734117 DH On-Demand Anodyne TRPV1 24 43 Cc1cncc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880734117 DH On-Demand Anodyne NAMPT 25 50 C[C@@H](CCc1cccc(F)c1)C(=O)NC1CSC1 ZINC000880734125 CF On-Demand Anodyne BIRC2 15 44 C[C@H](CCc1cccc(F)c1)C(=O)NC1CSC1 ZINC000880734126 CF On-Demand Anodyne BIRC2 15 44 CN(CCO)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734137 FF On-Demand Anodyne RBP4 60 40 C[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)[C@@H]1C ZINC000880734138 DJ On-Demand Anodyne TRPC6 52 38 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734139 DJ On-Demand Anodyne TRPC6 52 38 O=C(CCCOc1cccnc1)NC1CSC1 ZINC000880734147 CD On-Demand Anodyne CHRNA7 18 40 CCOCCOC1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734168 EG On-Demand Anodyne RBP4 43 32 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734189 GI On-Demand Anodyne EPHX2 21 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734192 GI On-Demand Anodyne EPHX2 21 41 Cn1cc(-c2cccc(C(=O)NC3CSC3)c2)cn1 ZINC000880734197 CD On-Demand Anodyne TYRO3 26 43 CCC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734222 EH On-Demand Anodyne CACNA1H 44 32 CCC1(CO)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734222 EH On-Demand Anodyne RBP4 45 34 O=C(NC1CSC1)C1(c2ccc(F)cc2)CCC1 ZINC000880734224 CE On-Demand Anodyne AVPR1A 32 42 CN1C(=O)NC2(CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)C1=O ZINC000880734240 GE On-Demand Anodyne CACNA1H 57 37 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734254 GE On-Demand Anodyne RBP4 41 37 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734255 GE On-Demand Anodyne RBP4 41 37 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734258 CE On-Demand Anodyne SIGMAR1 20 43 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734258 CE On-Demand Anodyne HSD11B1 49 48 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734258 CE On-Demand Anodyne CCR3 62 38 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734259 CE On-Demand Anodyne SIGMAR1 20 43 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734259 CE On-Demand Anodyne HSD11B1 49 48 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccc(F)cc1 ZINC000880734259 CE On-Demand Anodyne CCR3 62 38 Cc1cc(C(=O)NC2CSC2)ccc1-n1cncn1 ZINC000880734262 CD On-Demand Anodyne MAPK14 44 37 Cc1cc(C(=O)NC2CSC2)ccc1-n1cncn1 ZINC000880734262 CD On-Demand Anodyne MAPK13 69 39 C[C@H](CCOc1ccccc1)C(=O)NC1CSC1 ZINC000880734263 CE On-Demand Anodyne LTA4H 34 40 C[C@H](CCOc1ccccc1)C(=O)NC1CSC1 ZINC000880734263 CE On-Demand Anodyne CASP3 16 45 C[C@@H](CCOc1ccccc1)C(=O)NC1CSC1 ZINC000880734264 CE On-Demand Anodyne LTA4H 34 40 C[C@@H](CCOc1ccccc1)C(=O)NC1CSC1 ZINC000880734264 CE On-Demand Anodyne CASP3 16 45 O=C(NC1CSC1)c1c[nH]nc1-c1cccc(OC(F)F)c1 ZINC000880734266 EF On-Demand Anodyne PDE4B 44 32 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne GRIN2B 32 49 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne SIGMAR1 18 42 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne CTSK 15 41 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne CTSL 22 41 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne PREP 28 42 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne TGM2 44 42 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne F13A1 47 42 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NC1CSC1 ZINC000880734281 ED On-Demand Anodyne SLC12A5 49 35 Cc1nn(C)c2sc(C(=O)N[C@H](C)C(=O)NC3CSC3)cc12 ZINC000880734285 ED On-Demand Anodyne P2RX3 15 46 Cc1nn(C)c2sc(C(=O)N[C@@H](C)C(=O)NC3CSC3)cc12 ZINC000880734286 ED On-Demand Anodyne P2RX3 15 46 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880734287 CD On-Demand Bother CACNA1C 58 39 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880734287 CD On-Demand Bother CACNA1D 91 39 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880734287 CD On-Demand Bother LUXR 28 58 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880734287 CD On-Demand Bother TRAR 15 58 COCCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880734297 CD On-Demand Anodyne DRD4 46 35 COCCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880734297 CD On-Demand Anodyne MTNR1B 23 40 COCCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880734297 CD On-Demand Anodyne PLA2G4B 48 44 COCCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880734297 CD On-Demand Anodyne EPHX2 17 40 CS[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N(C)C ZINC000880734302 FG On-Demand Anodyne RBP4 51 32 CS[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N(C)C ZINC000880734303 FG On-Demand Anodyne RBP4 51 32 CS[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N(C)C ZINC000880734304 FG On-Demand Anodyne RBP4 51 32 CS[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N(C)C ZINC000880734305 FG On-Demand Anodyne RBP4 51 32 O=C(NC1CSC1)c1ccc(OC2CCOCC2)cc1 ZINC000880734324 CE On-Demand Anodyne EPHX2 23 42 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1F ZINC000880734330 DI On-Demand Anodyne RBP4 54 38 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1F ZINC000880734331 DI On-Demand Anodyne RBP4 54 38 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1F ZINC000880734332 DI On-Demand Anodyne RBP4 54 38 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1F ZINC000880734333 DI On-Demand Anodyne RBP4 54 38 CCCCN(CCCO)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734339 EH On-Demand Anodyne SOAT1 21 41 C[C@H]1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734349 DH On-Demand Anodyne EPHX2 16 42 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccncc2)C1 ZINC000880734360 DD On-Demand Anodyne EPHX2 19 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccncc2)C1 ZINC000880734360 DD On-Demand Anodyne L3MBTL3 53 38 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccncc2)C1 ZINC000880734361 DD On-Demand Anodyne EPHX2 19 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccncc2)C1 ZINC000880734361 DD On-Demand Anodyne L3MBTL3 53 38 CN(C)CCCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734398 FJ On-Demand Anodyne RBP4 47 37 COCC1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734409 EF On-Demand Anodyne CACNA1H 59 34 COCC1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734409 EF On-Demand Anodyne TRPM8 29 40 O=C(NC1CSC1)c1ccc(N2CCCCCC2)nc1 ZINC000880734442 CE On-Demand Anodyne HDAC1 18 40 O=C(NC1CSC1)c1ccc(N2CCCCCC2)nc1 ZINC000880734442 CE On-Demand Anodyne HPGDS 37 62 O=C(NC1CSC1)c1ccc(N2CCOCC2)c(F)c1 ZINC000880734453 CD On-Demand Anodyne MAPK14 24 41 O=C(NC1CSC1)c1ccc(N2CCOCC2)c(F)c1 ZINC000880734453 CD On-Demand Anodyne SLC6A9 15 44 O=C(Cc1ccccc1C(F)(F)F)NC1CSC1 ZINC000880734454 CE On-Demand Anodyne P2RX7 41 38 O=C(Cc1ccccc1C(F)(F)F)NC1CSC1 ZINC000880734454 CE On-Demand Anodyne RBP4 41 36 Cn1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)c1=O ZINC000880734480 GE On-Demand Anodyne TRPV1 15 45 Cn1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)c1=O ZINC000880734480 GE On-Demand Anodyne RBP4 25 43 CCOc1cn(-c2ccccc2)nc1C(=O)NC1CSC1 ZINC000880734487 DE On-Demand Anodyne HCN1 48 32 CCOc1cn(-c2ccccc2)nc1C(=O)NC1CSC1 ZINC000880734487 DE On-Demand Anodyne HCN4 41 31 O=C(Cc1ccccc1Br)NC1CSC1 ZINC000880734495 CE On-Demand Anodyne CA9 20 44 O=C(NC1CSC1)c1ccc2c(c1)C(=O)NC2=O ZINC000880734497 CC On-Demand Anodyne MAPK14 31 40 O=C(CNc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880734513 CE On-Demand Anodyne CCR2 104 45 O=C(CNc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880734513 CE On-Demand Anodyne EPHX2 15 48 O=C(NC1CSC1)c1ccc(OCC(F)(F)C(F)F)nc1 ZINC000880734543 DE On-Demand Anodyne HPGDS 37 44 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734553 EG On-Demand Anodyne EPHX2 29 43 COc1ccccc1/C(C)=C/C(=O)NC1CSC1 ZINC000880734574 CE On-Demand Anodyne KCNA3 45 49 COc1ccccc1/C(C)=C\C(=O)NC1CSC1 ZINC000880734575 CE On-Demand Anodyne KCNA3 45 49 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS1 ZINC000880734587 EI On-Demand Anodyne RBP4 52 32 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880734604 CD On-Demand Anodyne PAPA1_CARPA 37 57 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880734604 CD On-Demand Anodyne CTSK 22 47 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880734604 CD On-Demand Anodyne PGA5 23 42 C[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880734623 CD On-Demand Anodyne CTSK 15 44 O=C(NC1CSC1)c1cc2cc(F)ccc2o1 ZINC000880734670 CE On-Demand Anodyne KCNH2 15 44 O=C(NC1CSC1)c1cc2cc(F)ccc2o1 ZINC000880734670 CE On-Demand Anodyne MCHR1 15 44 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880734677 DG On-Demand Anodyne ACE 17 40 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880734677 DG On-Demand Anodyne CACNA1B 17 40 C[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)NC1CSC1 ZINC000880734677 DG On-Demand Anodyne ACE2 47 43 COC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734679 EG On-Demand Anodyne RBP4 47 44 CC(C)(C)NC(=O)Nc1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880734707 EG On-Demand Anodyne ENV 40 37 CC(C)(C)NC(=O)Nc1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880734707 EG On-Demand Anodyne IMDH_CRYPV 54 45 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734728 GI On-Demand Anodyne RBP4 45 35 O=C(NC1CSC1)c1ccccc1CN1CCOCC1 ZINC000880734736 CD On-Demand Anodyne DRD4 17 47 O=C(NC1CSC1)c1ccccc1CN1CCOCC1 ZINC000880734736 CD On-Demand Anodyne CNR2 19 45 O=C(NC1CSC1)c1ccccc1CN1CCOCC1 ZINC000880734736 CD On-Demand Anodyne SIGMAR1 15 43 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne ACE 78 42 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne MME 128 41 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne ANPEP 43 39 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne CPA1 41 35 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne CAPN1 42 35 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne CAPN2 43 30 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne ACE2 51 36 CN(C)[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880734740 CD On-Demand Anodyne AMP1_PLAFQ 42 36 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880734742 GH On-Demand Anodyne RBP4 51 32 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880734746 GH On-Demand Anodyne RBP4 51 32 Cc1nsc(N2CCCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880734757 GH On-Demand Anodyne FAAH 15 53 O=C(CNC(=O)c1ccccn1)NC1CSC1 ZINC000880734761 CC On-Demand Anodyne GRM4 53 38 CCCN(C)C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734800 FI On-Demand Anodyne RBP4 50 33 CCCN(C)C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734801 FI On-Demand Anodyne RBP4 50 33 O=C(NC1CSC1)c1ccc(CNC(=O)C2CCCC2)cc1 ZINC000880734828 DE On-Demand Anodyne SSTR3 26 44 Cc1ccc(-n2nc(C(=O)NC3CSC3)c3c2CCC3)c(F)c1 ZINC000880734829 EF On-Demand Anodyne CNR1 55 39 Cc1ccc(-n2nc(C(=O)NC3CSC3)c3c2CCC3)c(F)c1 ZINC000880734829 EF On-Demand Anodyne CNR2 20 46 Cc1ccc(-n2nc(C(=O)NC3CSC3)c3c2CCC3)c(F)c1 ZINC000880734829 EF On-Demand Anodyne MAPK13 47 31 CC(C)(C)OC(=O)N1CCC(n2cccc2C(=O)NC2CSC2)CC1 ZINC000880734830 FF On-Demand Anodyne GPR119 38 40 C[C@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734840 EF On-Demand Anodyne HTR4 15 41 C[C@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734840 EF On-Demand Anodyne CNR2 25 41 C[C@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734840 EF On-Demand Anodyne HRH3 42 37 C[C@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734840 EF On-Demand Anodyne HCN1 70 36 C[C@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734840 EF On-Demand Anodyne HCN4 54 36 C[C@@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734841 EF On-Demand Anodyne HTR4 15 41 C[C@@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734841 EF On-Demand Anodyne CNR2 25 41 C[C@@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734841 EF On-Demand Anodyne HRH3 42 37 C[C@@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734841 EF On-Demand Anodyne HCN1 70 36 C[C@@H]1CCCCN1CCOc1ccccc1C(=O)NC1CSC1 ZINC000880734841 EF On-Demand Anodyne HCN4 54 36 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734849 FD On-Demand Anodyne FKBP1A 16 42 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734849 FD On-Demand Anodyne SIGMAR1 15 45 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734849 FD On-Demand Anodyne EPHX2 24 45 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734849 FD On-Demand Anodyne TMPRSS11D 40 32 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734850 FD On-Demand Anodyne FKBP1A 16 42 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734850 FD On-Demand Anodyne SIGMAR1 15 45 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734850 FD On-Demand Anodyne EPHX2 24 45 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)Cc2ccccc2)C1 ZINC000880734850 FD On-Demand Anodyne TMPRSS11D 40 32 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734868 GF On-Demand Anodyne LPL 43 32 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734868 GF On-Demand Anodyne EPHX2 20 42 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734869 GF On-Demand Anodyne LPL 43 32 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880734869 GF On-Demand Anodyne EPHX2 20 42 CN(C(=O)Nc1cccc(F)c1C(C)(F)F)C1CCN(S(C)(=O)=O)CC1 ZINC000880734883 GF On-Demand Anodyne EPHX2 18 45 COC(=O)CCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734886 FI On-Demand Anodyne RBP4 42 41 Cc1ccc(OCc2cccc(C(=O)NC3CSC3)c2)cn1 ZINC000880734947 DF On-Demand Anodyne FFAR1 54 38 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734949 EG On-Demand Anodyne EPHX2 43 55 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734949 EG On-Demand Anodyne CCR8 52 38 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734950 EG On-Demand Anodyne EPHX2 43 55 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734950 EG On-Demand Anodyne CCR8 52 38 CC(=O)OC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880734955 EG On-Demand Anodyne RBP4 40 41 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734956 EG On-Demand Anodyne EPHX2 30 43 O=C(CCCCCNC(=O)NC1CCCCC1)NC1CSC1 ZINC000880734960 EE On-Demand Anodyne EPHX2 35 61 COCCCOC1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880734963 EG On-Demand Anodyne RBP4 44 32 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734979 DD On-Demand Anodyne SLC6A1 60 36 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734979 DD On-Demand Anodyne PREP 39 45 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734979 DD On-Demand Anodyne EPHX2 24 60 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734979 DD On-Demand Anodyne L3MBTL3 72 39 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734979 DD On-Demand Anodyne MAP3K12 32 42 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734980 DD On-Demand Anodyne SLC6A1 60 36 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734980 DD On-Demand Anodyne PREP 39 45 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734980 DD On-Demand Anodyne EPHX2 24 60 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734980 DD On-Demand Anodyne L3MBTL3 72 39 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccccc2)C1 ZINC000880734980 DD On-Demand Anodyne MAP3K12 32 42 COC(=O)C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734985 FF On-Demand Anodyne RBP4 52 34 COC(=O)C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880734986 FF On-Demand Anodyne RBP4 52 34 O=C(CCc1nc2cc(C(F)(F)F)ccc2s1)NC1CSC1 ZINC000880734989 EG On-Demand Anodyne AKR1B1 16 42 O=C(NC1CSC1)[C@H]1C[C@@H]1c1ccc2ccccc2c1 ZINC000880734990 CG On-Demand Anodyne SLC6A3 21 42 O=C(NC1CSC1)[C@H]1C[C@H]1c1ccc2ccccc2c1 ZINC000880734991 CG On-Demand Anodyne SLC6A3 21 42 O=C(NC1CSC1)[C@@H]1C[C@@H]1c1ccc2ccccc2c1 ZINC000880734992 CG On-Demand Anodyne SLC6A3 21 42 O=C(NC1CSC1)[C@@H]1C[C@H]1c1ccc2ccccc2c1 ZINC000880734993 CG On-Demand Anodyne SLC6A3 21 42 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA2 163 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA6 30 41 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA1 139 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA7 100 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA13 33 43 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA5B 88 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA4 110 48 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA5A 94 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA14 98 49 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA12 112 50 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA9 119 51 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CAH_METTE 26 43 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CYNT 47 39 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne NCE103 33 46 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne CA15 17 43 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne MTCA1 51 43 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne P96878_MYCTU 62 43 NS(=O)(=O)c1ccc(CC(=O)NC2CSC2)cc1 ZINC000880734996 CC On-Demand Anodyne A6YCJ1_9METZ 31 42 O=C(CC[C@H]1NC(=O)N(c2ccc(Cl)c(Cl)c2)C1=O)NC1CSC1 ZINC000880734997 GE On-Demand Anodyne BCL2A1 52 35 O=C(CC[C@@H]1NC(=O)N(c2ccc(Cl)c(Cl)c2)C1=O)NC1CSC1 ZINC000880734998 GE On-Demand Anodyne BCL2A1 52 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1C ZINC000880735000 DI On-Demand Anodyne RBP4 65 40 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1C ZINC000880735001 DI On-Demand Anodyne RBP4 65 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1C ZINC000880735002 DI On-Demand Anodyne RBP4 65 40 O=C(CCc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880735003 DF On-Demand Anodyne EPHX2 31 42 O=C(CCc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880735003 DF On-Demand Anodyne LUXR 45 38 O=C(CCc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880735003 DF On-Demand Anodyne TRAR 26 43 Cc1cc(C(=O)NC2CSC2)cc(C)c1OC(F)F ZINC000880735004 CF On-Demand Anodyne MAPK13 54 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880735009 FG On-Demand Anodyne RBP4 53 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880735010 FG On-Demand Anodyne RBP4 53 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N1CCOCC1 ZINC000880735011 FG On-Demand Anodyne RBP4 53 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N1CCOCC1 ZINC000880735012 FG On-Demand Anodyne RBP4 53 33 O=C(NC1CSC1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880735030 DD On-Demand Anodyne LGMN 75 38 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880735031 DD On-Demand Anodyne LGMN 75 38 CCN1CCCC[C@H]1C(=O)NC1CSC1 ZINC000880735040 BD On-Demand Anodyne HSD11B1 48 39 CCN1CCCC[C@@H]1C(=O)NC1CSC1 ZINC000880735041 BD On-Demand Anodyne HSD11B1 48 39 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880735055 DD On-Demand Anodyne EPHX2 20 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880735055 DD On-Demand Anodyne L3MBTL3 63 40 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880735056 DD On-Demand Anodyne EPHX2 20 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccc(F)cc2)C1 ZINC000880735056 DD On-Demand Anodyne L3MBTL3 63 40 Nc1ncnc2c1ncn2CC(=O)NC1CSC1 ZINC000880735057 CB On-Demand Anodyne AHCY 91 49 Nc1ncnc2c1ncn2CC(=O)NC1CSC1 ZINC000880735057 CB On-Demand Anodyne ADCY5 42 43 Nc1ncnc2c1ncn2CC(=O)NC1CSC1 ZINC000880735057 CB On-Demand Anodyne OXGR1 117 42 Nc1ncnc2c1ncn2CC(=O)NC1CSC1 ZINC000880735057 CB On-Demand Anodyne DOT1L 56 37 O=C(NC1CSC1)c1cccc(OC2CCCC2)c1 ZINC000880735058 CF On-Demand Anodyne DRD4 40 30 O=C(NC1CSC1)c1cccc(OC2CCCC2)c1 ZINC000880735058 CF On-Demand Anodyne KCNH2 41 37 O=C(NC1CSC1)c1cccc(OC2CCCC2)c1 ZINC000880735058 CF On-Demand Anodyne EPHX2 24 44 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735063 EF On-Demand Anodyne LGMN 62 35 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735063 EF On-Demand Anodyne WNT3 40 32 CN(C)C(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880735066 CD On-Demand Anodyne MAPK11 23 44 CN(C)C(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880735066 CD On-Demand Anodyne MAPK14 17 44 O=C(NC1CSC1)c1cc(-n2cccn2)ccn1 ZINC000880735082 CD On-Demand Anodyne AMP1_PLAFQ 50 35 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735090 FH On-Demand Anodyne FDFT1 17 45 CN1C(=O)CC[C@H](C(=O)NC2CSC2)[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000880735093 FF On-Demand Anodyne TRPM8 45 39 CN1C(=O)CC[C@@H](C(=O)NC2CSC2)[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000880735094 FF On-Demand Anodyne TRPM8 45 39 CN1C(=O)CC[C@@H](C(=O)NC2CSC2)[C@H]1c1ccc(C(F)(F)F)cc1 ZINC000880735095 FF On-Demand Anodyne TRPM8 45 39 CN1C(=O)CC[C@H](C(=O)NC2CSC2)[C@@H]1c1ccc(C(F)(F)F)cc1 ZINC000880735096 FF On-Demand Anodyne TRPM8 45 39 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne ACE 31 46 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne AVPR1A 16 40 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne MME 42 46 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne CTSL 30 45 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne FURIN 62 47 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne FPR1 43 41 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne GAG-PRO 40 34 CSCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735102 ED On-Demand Anodyne POLG_WNV 42 34 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne ACE 31 46 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne AVPR1A 16 40 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne MME 42 46 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne CTSL 30 45 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne FURIN 62 47 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne FPR1 43 41 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne GAG-PRO 40 34 CSCC[C@@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735103 ED On-Demand Anodyne POLG_WNV 42 34 O=C(CNC(=O)c1ccc(O)cc1)NC1CSC1 ZINC000880735112 CC On-Demand Anodyne CCR2 43 41 O=C(NC1CSC1)c1csc(Nc2ccccn2)n1 ZINC000880735128 CE On-Demand Anodyne GRM4 15 44 O=C(NC1CSC1)c1csc(Nc2ccccn2)n1 ZINC000880735128 CE On-Demand Anodyne KCNN1 28 48 O=C(NC1CSC1)c1csc(Nc2ccccn2)n1 ZINC000880735128 CE On-Demand Anodyne TRPC6 48 33 O=C(NC1CSC1)c1csc(Nc2ccccn2)n1 ZINC000880735128 CE On-Demand Anodyne TRPC3 42 32 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne ACE 23 41 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne MME 37 40 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne PTAFR 27 43 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTSB 30 43 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne PAPA1_CARPA 27 46 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CYSP_TRYCR 49 41 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTSK 17 45 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTSL 39 46 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CHRNA7 38 44 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne TIMP3 44 42 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne C3AR1 40 39 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTRB1 23 40 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTSS 25 52 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne CTSV 35 42 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne MMP1 17 45 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne PSMB5 50 40 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne BLA1_STEMA 41 35 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne ACHP_LYMST 18 44 O=C(N[C@@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735152 ED On-Demand Anodyne PSMB8 21 40 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne ACE 23 41 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne MME 37 40 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne PTAFR 27 43 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTSB 30 43 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne PAPA1_CARPA 27 46 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CYSP_TRYCR 49 41 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTSK 17 45 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTSL 39 46 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CHRNA7 38 44 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne TIMP3 44 42 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne C3AR1 40 39 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTRB1 23 40 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTSS 25 52 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne CTSV 35 42 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne MMP1 17 45 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne PSMB5 50 40 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne BLA1_STEMA 41 35 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne ACHP_LYMST 18 44 O=C(N[C@H](Cc1cccnc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880735153 ED On-Demand Anodyne PSMB8 21 40 O=C(CN1CCN(c2ccccn2)CC1)NC1CSC1 ZINC000880735159 CC On-Demand Anodyne HTR1A 21 51 O=C(CN1CCN(c2ccccn2)CC1)NC1CSC1 ZINC000880735159 CC On-Demand Anodyne DRD2 20 51 O=C(CN1CCN(c2ccccn2)CC1)NC1CSC1 ZINC000880735159 CC On-Demand Anodyne DRD4 41 44 O=C(CN1CCN(c2ccccn2)CC1)NC1CSC1 ZINC000880735159 CC On-Demand Anodyne SLC27A1 67 54 C#CCN1CCC[C@H]1C(=O)NC1CSC1 ZINC000880735170 BC On-Demand Mild HSD11B1 49 38 O=C(NCCCc1ccccc1)C(=O)NC1CSC1 ZINC000880735171 CC On-Demand Anodyne SIGMAR1 22 43 O=C(NCCCc1ccccc1)C(=O)NC1CSC1 ZINC000880735171 CC On-Demand Anodyne FAAH 19 41 O=C(NCCCc1ccccc1)C(=O)NC1CSC1 ZINC000880735171 CC On-Demand Anodyne AMP1_PLAFQ 26 46 O=C(NCCCc1ccccc1)C(=O)NC1CSC1 ZINC000880735171 CC On-Demand Anodyne CRTM 35 42 Cn1nnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880735192 BC On-Demand Anodyne MAPK14 45 37 Cn1nnc2cc(C(=O)NC3CSC3)ccc21 ZINC000880735192 BC On-Demand Anodyne MAPK13 63 36 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735222 CH On-Demand Anodyne EPHX2 18 44 C[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735222 CH On-Demand Anodyne RBP4 60 40 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735223 CH On-Demand Anodyne EPHX2 18 44 C[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735223 CH On-Demand Anodyne RBP4 60 40 CS[C@H]1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735239 EI On-Demand Anodyne EPHX2 27 42 CS[C@@H]1CC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735240 EI On-Demand Anodyne EPHX2 27 42 CCC1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880735247 EH On-Demand Anodyne CACNA1H 56 33 CCC1(O)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880735247 EH On-Demand Anodyne TRPM8 29 40 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880735248 FI On-Demand Anodyne RBP4 51 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880735249 FI On-Demand Anodyne RBP4 51 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880735250 FI On-Demand Anodyne RBP4 51 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880735251 FI On-Demand Anodyne RBP4 51 33 O=C(CCCCOc1ccc(Br)cc1)NC1CSC1 ZINC000880735263 EG On-Demand Anodyne PLA2G4B 56 36 O=C(CCCCOc1ccc(Br)cc1)NC1CSC1 ZINC000880735263 EG On-Demand Anodyne LSS 28 44 O=C(CCCCOc1ccc(Br)cc1)NC1CSC1 ZINC000880735263 EG On-Demand Anodyne TRAR 38 43 CCCCCS(=O)(=O)CC(=O)NC1CSC1 ZINC000880735269 CC On-Demand Anodyne EST1_PIG 25 43 O=C(NC1CSC1)c1cnn2ccccc12 ZINC000880735288 BD On-Demand Anodyne JAK3 19 45 O=C(NC1CSC1)c1cnn2ccccc12 ZINC000880735288 BD On-Demand Anodyne JAK1 15 45 O=C(NC1CSC1)c1cnn2ccccc12 ZINC000880735288 BD On-Demand Anodyne TYK2 22 45 O=C(NC1CSC1)c1cnn2ccccc12 ZINC000880735288 BD On-Demand Anodyne EPHB3 46 57 O=C(Cc1cccc(Cl)c1)NC1CSC1 ZINC000880735296 BE On-Demand Anodyne SIGMAR1 17 60 O=C(NC1CSC1)c1cnc(-c2ccc3c(c2)OCO3)s1 ZINC000880735304 DE On-Demand Anodyne CLK4 50 33 O=C(NC1CSC1)c1coc2ccccc12 ZINC000880735308 BE On-Demand Anodyne INHA 84 40 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NC2CSC2)C1 ZINC000880735319 CD On-Demand Anodyne EPHX2 19 50 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne ACE 58 37 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne AVPR1A 21 42 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne MME 72 37 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne NPR1 49 37 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CTSB 30 41 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CTSK 36 41 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CTSL 39 44 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne NPFFR2 24 40 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne PCSK5 38 40 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne FURIN 65 40 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CTSS 18 44 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CAPN1 50 40 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne CAPN2 66 39 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne ACE2 55 36 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne BLA1_STEMA 56 41 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne POLG_WNV 57 36 CCC[C@H](NC(=O)Cc1ccccc1)C(=O)NC1CSC1 ZINC000880735321 DD On-Demand Anodyne NPFFR1 39 40 O=C(COc1ccccc1OCc1ccccc1)NC1CSC1 ZINC000880735364 EF On-Demand Anodyne PPIA 39 40 O=C(COc1ccccc1OCc1ccccc1)NC1CSC1 ZINC000880735364 EF On-Demand Anodyne PTGER1 44 38 C[C@@H](CC[S@](C)=O)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735399 EG On-Demand Anodyne ANPEP 15 46 C[C@H](CC[S@](C)=O)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735401 EG On-Demand Anodyne ANPEP 15 46 C[C@@H](CC[S@@](C)=O)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735403 EG On-Demand Anodyne ANPEP 15 46 C[C@H](CC[S@@](C)=O)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880735404 EG On-Demand Anodyne ANPEP 15 46 O=C(CCCCCc1cccs1)NC1CSC1 ZINC000880735414 CG On-Demand Anodyne PTPRF 19 42 CCN1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735421 EH On-Demand Anodyne CCR3 37 40 CCN1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735421 EH On-Demand Anodyne EPHX2 34 44 CCN1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735421 EH On-Demand Anodyne BIRC2 34 40 CCN1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735424 EH On-Demand Anodyne CCR3 37 40 CCN1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735424 EH On-Demand Anodyne EPHX2 34 44 CCN1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735424 EH On-Demand Anodyne BIRC2 34 40 CCOc1ncc(C(=O)NC2CSC2)cc1Cl ZINC000880735434 CD On-Demand Anodyne SSTR5 47 44 COc1ccc(Nc2nc(C(=O)NC3CSC3)cs2)cc1 ZINC000880735445 DF On-Demand Anodyne TRPC6 69 57 COc1ccc(Nc2nc(C(=O)NC3CSC3)cs2)cc1 ZINC000880735445 DF On-Demand Anodyne TRPC3 61 57 O=C(CNC(=O)c1c(F)cccc1Cl)NC1CSC1 ZINC000880735483 DD On-Demand Anodyne PPIA 25 43 O=C(CNC(=O)c1c(F)cccc1Cl)NC1CSC1 ZINC000880735483 DD On-Demand Anodyne CCR2 44 38 O=C(NC1CSC1)c1ccc(I)c(F)c1 ZINC000880735489 EE On-Demand Anodyne MAPK13 57 31 CCOC[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735492 EH On-Demand Anodyne RBP4 44 35 CCn1nc2c(cc1=O)CN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880735498 GG On-Demand Anodyne P2RY14 47 34 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)S1 ZINC000880735521 EI On-Demand Anodyne RBP4 55 35 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)S1 ZINC000880735522 EI On-Demand Anodyne RBP4 55 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)S1 ZINC000880735523 EI On-Demand Anodyne RBP4 55 35 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735530 DI On-Demand Anodyne CACNA1H 50 33 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735530 DI On-Demand Anodyne EPHX2 34 44 CC1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735530 DI On-Demand Anodyne RBP4 46 33 CCCN(CCC)C(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880735585 DF On-Demand Anodyne BACE1 20 44 Cn1cccc(C(=O)NC2CSC2)c1=O ZINC000880735590 BC On-Demand Anodyne CNR2 17 44 Cn1cccc(C(=O)NC2CSC2)c1=O ZINC000880735590 BC On-Demand Anodyne POLR1A 48 41 COCCc1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880735592 DE On-Demand Anodyne CYSLTR2 65 34 COCCc1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880735592 DE On-Demand Anodyne PLA2G4B 55 34 O=C(CN1C(=O)CCc2ccccc21)NC1CSC1 ZINC000880735595 CD On-Demand Anodyne ACE 19 42 CCCNC(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880735604 CD On-Demand Anodyne DRD4 44 34 COCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880735609 CD On-Demand Anodyne CYSLTR2 45 36 COCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880735609 CD On-Demand Anodyne PLA2G4B 80 39 COCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880735609 CD On-Demand Anodyne SLC6A5 37 42 COCCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880735609 CD On-Demand Anodyne AOC3 15 46 COc1ccccc1-c1nn(C)cc1C(=O)NC1CSC1 ZINC000880735644 DD On-Demand Anodyne DRD2 31 44 COc1ccccc1-c1nn(C)cc1C(=O)NC1CSC1 ZINC000880735644 DD On-Demand Anodyne DRD3 39 40 COc1ccccc1-c1nn(C)cc1C(=O)NC1CSC1 ZINC000880735644 DD On-Demand Anodyne HTR4 30 42 O=C(NC1CSC1)c1cn(-c2cccc(C(F)(F)F)c2)nn1 ZINC000880735648 EE On-Demand Anodyne ESRRA 15 43 O=C(NC1CSC1)c1cn(-c2cccc(C(F)(F)F)c2)nn1 ZINC000880735648 EE On-Demand Anodyne CCR2 45 35 CCCc1c(C(=O)NC2CSC2)nnn1-c1cccc(Cl)c1 ZINC000880735656 EF On-Demand Anodyne CNR1 27 43 CCCc1c(C(=O)NC2CSC2)nnn1-c1cccc(Cl)c1 ZINC000880735656 EF On-Demand Anodyne CNR2 17 43 CC(C)[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735662 DI On-Demand Anodyne RBP4 61 38 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HTR1A 118 55 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne DRD2 82 55 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne DRD4 52 47 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne ADRA1D 21 41 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HTR2A 66 55 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HTR2C 26 43 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne ADRA1A 30 45 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HRH1 16 45 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne ADRA1B 20 45 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne DRD3 87 49 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HTR4 16 41 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne DRD5 18 46 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne HTR7 141 55 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne SIGMAR1 33 49 O=C(CCCN1CCN(c2ccccc2)CC1)NC1CSC1 ZINC000880735690 DD On-Demand Anodyne CYP2J2 48 34 O=C(CN(Cc1cccnc1)c1ccccc1)NC1CSC1 ZINC000880735699 DE On-Demand Anodyne NAMPT 38 40 O=C(CCc1nc(-c2ccoc2)no1)NC1CSC1 ZINC000880735710 CD On-Demand Anodyne HCAR2 21 40 N#Cc1cccc(OCCCCC(=O)NC2CSC2)c1 ZINC000880735715 CE On-Demand Mild CYSLTR2 46 32 N#Cc1cccc(OCCCCC(=O)NC2CSC2)c1 ZINC000880735715 CE On-Demand Mild TNKS 28 43 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N(C)C ZINC000880735726 EG On-Demand Anodyne RBP4 52 33 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N(C)C ZINC000880735727 EG On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H]1N(C)C ZINC000880735728 EG On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H]1N(C)C ZINC000880735729 EG On-Demand Anodyne RBP4 52 33 COc1cccc([C@H]2CN(C(=O)Nc3cccc(F)c3C(C)(F)F)CCO2)c1 ZINC000880735736 GJ On-Demand Anodyne RBP4 46 39 O=C(NC1CSC1)C1CCCCCCC1 ZINC000880735768 BF On-Demand Anodyne EPHX2 18 45 C[C@@]1(C(=O)NC2CSC2)CCCN1C(=O)c1ccccc1 ZINC000880735769 DD On-Demand Anodyne SLC12A5 47 32 C[C@]1(C(=O)NC2CSC2)CCCN1C(=O)c1ccccc1 ZINC000880735770 DD On-Demand Anodyne SLC12A5 47 32 CCCCSCCC(=O)NC1CSC1 ZINC000880735774 BE On-Demand Anodyne EST1_PIG 40 35 O=C(C[C@@H]1CCc2ccccc2C1)NC1CSC1 ZINC000880735780 CE On-Demand Anodyne PREP 30 50 O=C(C[C@H]1CCc2ccccc2C1)NC1CSC1 ZINC000880735781 CE On-Demand Anodyne PREP 30 50 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735790 ED On-Demand Anodyne CPT1A 128 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735790 ED On-Demand Anodyne CPT2 51 39 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735790 ED On-Demand Anodyne EPHX2 22 44 O=C(NC1CSC1)[C@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735791 ED On-Demand Anodyne CPT1A 128 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735791 ED On-Demand Anodyne CPT2 51 39 O=C(NC1CSC1)[C@H]1CCCN(C(=O)COc2ccccc2)C1 ZINC000880735791 ED On-Demand Anodyne EPHX2 22 44 O=C(NC1CSC1)c1ccc(N2CCCS2(=O)=O)cc1Cl ZINC000880735792 ED On-Demand Anodyne CDK1 17 41 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NC1CSC1 ZINC000880735809 DG On-Demand Anodyne CACNA1B 18 43 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NC1CSC1 ZINC000880735809 DG On-Demand Anodyne CCR2 95 41 C[C@@H](Cc1cccc(C(F)(F)F)c1)C(=O)NC1CSC1 ZINC000880735809 DG On-Demand Anodyne PDS 40 38 O=C(CCCn1ccnc1)NC1CSC1 ZINC000880735847 BC On-Demand Anodyne TBXAS1 53 52 O=C(CCCn1ccnc1)NC1CSC1 ZINC000880735847 BC On-Demand Anodyne HMOX2 46 34 O=C(CCCn1ccnc1)NC1CSC1 ZINC000880735847 BC On-Demand Anodyne QPCT 40 42 CC[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735867 DI On-Demand Anodyne RBP4 54 38 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne FKBP1A 43 39 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne DRD4 18 40 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne SIGMAR1 32 53 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne HSD11B1 46 44 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne PREP 65 38 O=C(NC1CSC1)[C@@H]1CCCCN1Cc1ccccc1 ZINC000880735877 CE On-Demand Anodyne EPHX2 17 40 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne FKBP1A 43 39 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne DRD4 18 40 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne SIGMAR1 32 53 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne HSD11B1 46 44 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne PREP 65 38 O=C(NC1CSC1)[C@H]1CCCCN1Cc1ccccc1 ZINC000880735878 CE On-Demand Anodyne EPHX2 17 40 COCCC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880735879 GG On-Demand Anodyne EPHX2 50 48 COCCC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880735879 GG On-Demand Anodyne CCR8 58 40 Cc1ccc(N2CCC(C(=O)NC3CSC3)CC2)nc1 ZINC000880735888 CD On-Demand Anodyne EPHX2 28 45 CN(C)C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880735889 CD On-Demand Anodyne KCNK3 100 40 CN(C)C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880735889 CD On-Demand Anodyne KCNK9 54 40 Cc1ccccc1[C@H](C)CC(=O)NC1CSC1 ZINC000880735915 BF On-Demand Anodyne CTSA 44 33 Cc1ccccc1[C@@H](C)CC(=O)NC1CSC1 ZINC000880735916 BF On-Demand Anodyne CTSA 44 33 O=C(NC1CSC1)c1ccn(-c2cccc(C(F)(F)F)c2)n1 ZINC000880735924 EF On-Demand Anodyne CCR2 42 34 C[C@H](CC(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880735940 DG On-Demand Anodyne CCR2 91 45 C[C@@H](CC(=O)NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880735941 DG On-Demand Anodyne CCR2 91 45 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000880735953 CD On-Demand Anodyne DRD4 41 46 O=C(NC1CSC1)[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000880735953 CD On-Demand Anodyne SIGMAR1 43 45 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCO1 ZINC000880735954 CD On-Demand Anodyne DRD4 41 46 O=C(NC1CSC1)[C@H]1CN(Cc2ccccc2)CCO1 ZINC000880735954 CD On-Demand Anodyne SIGMAR1 43 45 CC[C@]1(C)CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880735957 DJ On-Demand Anodyne EPHX2 30 41 O=C(COc1cccnc1)NC1CSC1 ZINC000880736034 BC On-Demand Anodyne CHRNA7 34 40 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cccc(F)c1C(C)(F)F)C2 ZINC000880736061 FI On-Demand Anodyne HTR3A 35 44 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cccc(F)c1C(C)(F)F)C2 ZINC000880736061 FI On-Demand Anodyne EPHX2 37 45 O=C(NC1CSC1)c1nnn(-c2cccc(C(F)(F)F)c2)c1C1CC1 ZINC000880736071 FG On-Demand Anodyne CCR2 60 38 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne DRD4 34 48 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne ACHE 18 48 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne CHRM3 22 45 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne CNR2 17 41 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne SIGMAR1 25 52 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne SSTR5 46 41 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne CCR3 20 49 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne BDKRB1 17 43 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne EPHX2 18 41 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne MCHR1 34 52 O=C(NC1CSC1)c1cccc(CN2CCOCC2)c1 ZINC000880736073 CD On-Demand Anodyne HPGDS 43 36 CN1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCC1=O ZINC000880736076 EF On-Demand Anodyne EPHX2 21 41 CN1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCC1=O ZINC000880736077 EF On-Demand Anodyne EPHX2 21 41 CC(=O)CCc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880736186 CD On-Demand Anodyne PPO2 27 40 CC(=O)CCc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880736186 CD On-Demand Anodyne FFAR4 42 32 CC(=O)CCc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880736186 CD On-Demand Anodyne TRAR 41 37 Cc1cc(C(=O)NC2CSC2)c(C)n1Cc1ccccn1 ZINC000880736187 DE On-Demand Anodyne NOX4 28 40 C[C@@H](CCN(C)C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880736195 DG On-Demand Anodyne UTS2 49 32 O=C(NC1CSC1)c1nc(C2CC2)n(-c2ccccc2Cl)n1 ZINC000880736197 EF On-Demand Anodyne CNR1 31 41 O=C(NC1CSC1)c1ccc(N2CCCC2)nn1 ZINC000880736217 CC On-Demand Anodyne SCD1 57 43 O=C(NC1CSC1)c1ccc(N2CCCC2)nn1 ZINC000880736217 CC On-Demand Anodyne SCD 46 40 O=C(COc1ccc([N+](=O)[O-])c(F)c1)NC1CSC1 ZINC000880736290 CD On-Demand Bother TRAR 29 41 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736291 GJ On-Demand Anodyne RBP4 85 51 COc1ccccc1[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736294 GJ On-Demand Anodyne RBP4 85 51 Cn1nccc1C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736350 FI On-Demand Anodyne RBP4 57 40 NC(=O)c1cn(CC(=O)NC2CSC2)c2ccccc12 ZINC000880736351 CC On-Demand Anodyne CNR2 23 40 COC(=O)N[C@H](CC(C)C)C(=O)NC1CSC1 ZINC000880736367 CC On-Demand Anodyne CTSK 29 45 COC(=O)N[C@H](CC(C)C)C(=O)NC1CSC1 ZINC000880736367 CC On-Demand Anodyne CAPNS1 53 33 COC(=O)N[C@H](CC(C)C)C(=O)NC1CSC1 ZINC000880736367 CC On-Demand Anodyne CAPN1 69 52 COC(=O)N[C@H](CC(C)C)C(=O)NC1CSC1 ZINC000880736367 CC On-Demand Anodyne CAPN2 82 40 COC(=O)N[C@H](CC(C)C)C(=O)NC1CSC1 ZINC000880736367 CC On-Demand Anodyne FPR1 44 34 O=C(CCCCC(=O)c1ccccc1)NC1CSC1 ZINC000880736378 CF On-Demand Anodyne HDAC8 40 48 O=C(CCCCC(=O)c1ccccc1)NC1CSC1 ZINC000880736378 CF On-Demand Anodyne HDAC1 15 56 O=C(CCCCC(=O)c1ccccc1)NC1CSC1 ZINC000880736378 CF On-Demand Anodyne CYP2J2 46 32 O=C(CCCOCc1ccccc1)NC1CSC1 ZINC000880736393 CE On-Demand Anodyne GRIN2B 21 43 O=C(CCCOCc1ccccc1)NC1CSC1 ZINC000880736393 CE On-Demand Anodyne SIGMAR1 15 40 O=C(CCCOCc1ccccc1)NC1CSC1 ZINC000880736393 CE On-Demand Anodyne NAAA 33 42 O=C(CCCOCc1ccccc1)NC1CSC1 ZINC000880736393 CE On-Demand Anodyne TNKS 46 31 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccc(Br)cc1 ZINC000880736394 FE On-Demand Anodyne PREP 31 48 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccc(Br)cc1 ZINC000880736396 FE On-Demand Anodyne PREP 31 48 O=C(NC1CSC1)c1cc2cccc([N+](=O)[O-])c2[nH]1 ZINC000880736412 CD On-Demand Bother PYGL 18 58 Cc1cc(C(=O)NC2CSC2)n(C)n1 ZINC000880736427 BC On-Demand Anodyne INHA 47 33 Cc1cc(C(=O)NC2CSC2)n(C)n1 ZINC000880736427 BC On-Demand Anodyne MAPK13 41 31 O=C(NC1CSC1)c1ccc(N2CCc3ccccc3C2)cc1 ZINC000880736434 DG On-Demand Anodyne NOD2 43 36 O=C(CNC(=O)c1cc(-c2ccccc2)on1)NC1CSC1 ZINC000880736435 DD On-Demand Anodyne HDAC10 16 53 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)N1CCCC[C@H]1C ZINC000880736450 FH On-Demand Anodyne ACE 21 40 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)N1CCCC[C@H]1C ZINC000880736450 FH On-Demand Anodyne CELA1 40 38 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880736451 FH On-Demand Anodyne ACE 21 40 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880736451 FH On-Demand Anodyne CELA1 40 38 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)N1CCCC[C@@H]1C ZINC000880736452 FH On-Demand Anodyne ACE 21 40 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)N1CCCC[C@@H]1C ZINC000880736452 FH On-Demand Anodyne CELA1 40 38 Cn1c(C(=O)NC2CSC2)cc2ccccc21 ZINC000880736476 BE On-Demand Anodyne GLRA1 17 45 Cn1c(C(=O)NC2CSC2)cc2ccccc21 ZINC000880736476 BE On-Demand Anodyne PYK 25 41 O=C(CNC(=O)c1ccc(F)c(F)c1)NC1CSC1 ZINC000880736484 CC On-Demand Anodyne CCR2 62 42 CCS(=O)(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736497 GE On-Demand Anodyne RBP4 53 34 O=C(NC1CSC1)C1CCCCCC1 ZINC000880736502 BE On-Demand Anodyne EPHX2 18 45 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736514 EF On-Demand Anodyne RBP4 52 34 C[C@H]1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CCN1C ZINC000880736519 EH On-Demand Anodyne EPHX2 35 41 CS(=O)(=O)c1ccc(OCCCCC(=O)NC2CSC2)cc1 ZINC000880736523 ED On-Demand Anodyne PLA2G4B 54 36 CS(=O)(=O)c1ccc(OCCCCC(=O)NC2CSC2)cc1 ZINC000880736523 ED On-Demand Anodyne MMP1 19 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccc2ccccc2c1O ZINC000880736524 FE On-Demand Anodyne PREP 44 37 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccc2ccccc2c1O ZINC000880736525 FE On-Demand Anodyne PREP 44 37 COC(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736529 EG On-Demand Anodyne RBP4 51 34 CS(=O)(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880736549 ED On-Demand Anodyne MMP13 36 40 CS(=O)(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880736549 ED On-Demand Anodyne MMP2 22 40 CS(=O)(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880736549 ED On-Demand Anodyne MMP3 22 40 CS(=O)(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880736549 ED On-Demand Anodyne PLA2G4B 44 34 CS(=O)(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880736549 ED On-Demand Anodyne MMP1 21 43 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne ACE 16 41 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne CELA1 18 40 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne PREP 28 47 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne LGMN 59 40 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne Q9NAW4_PLAFA 51 61 O=C(NC1CSC1)[C@@H]1C[C@@H](O)CN1C(=O)OCc1ccccc1 ZINC000880736563 EC On-Demand Anodyne VHL 51 35 O=C(NC1CCC(C(=O)NC2CSC2)CC1)C1CCCC1 ZINC000880736578 DE On-Demand Anodyne EPHX2 18 43 CN(C)C(=O)Nc1cccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880736590 GI On-Demand Anodyne TRPV1 17 41 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne ACE 62 37 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne MME 68 36 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne PAPA1_CARPA 41 36 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne CTSK 36 40 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne CAPNS1 58 33 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne CAPN1 67 38 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne CAPN2 87 37 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne NPR 77 34 C[C@@H](OCc1ccccc1)C(=O)NC1CSC1 ZINC000880736598 CD On-Demand Anodyne NAAA 48 38 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne DRD2 19 55 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne DRD4 40 31 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne ACHE 25 47 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne HRH2 39 47 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne CHRM3 24 43 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne SIGMAR1 31 55 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne SSTR5 47 43 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne CCR3 31 52 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne BDKRB1 44 52 O=C(NC1CSC1)c1cccc(CN2CCCC2)c1 ZINC000880736607 CE On-Demand Anodyne MCHR1 43 52 CCCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880736611 BE On-Demand Anodyne ECR 23 40 CCCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880736611 BE On-Demand Anodyne E3UJZ5_SPOLI 20 40 O=C(CSCc1cccnc1)NC1CSC1 ZINC000880736614 CD On-Demand Anodyne CHRNA7 50 39 CC(=O)N1CCc2cc(NC(=O)Nc3cccc(F)c3C(C)(F)F)ccc21 ZINC000880736619 GI On-Demand Anodyne P2RY1 64 37 CC(=O)N1CCc2cc(NC(=O)Nc3cccc(F)c3C(C)(F)F)ccc21 ZINC000880736619 GI On-Demand Anodyne HSD17B3 41 34 COC[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736620 EH On-Demand Anodyne RBP4 47 37 C[C@@H](Cn1cncn1)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880736623 EF On-Demand Anodyne HIS3 79 38 COCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736635 EH On-Demand Anodyne EPHX2 20 40 COCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736635 EH On-Demand Anodyne RBP4 46 42 O=C(NC1CSC1)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880736637 ED On-Demand Anodyne GRIN2B 18 40 O=C(NC1CSC1)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880736637 ED On-Demand Anodyne LTA4H 23 42 O=C(NC1CSC1)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880736637 ED On-Demand Anodyne CPT1A 98 36 O=C(NC1CSC1)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880736637 ED On-Demand Anodyne CPT2 44 34 O=C(NC1CSC1)C1CCN(C(=O)CCOc2ccccc2)CC1 ZINC000880736637 ED On-Demand Anodyne EPHX2 37 47 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880736657 CD On-Demand Anodyne ACE 44 38 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880736657 CD On-Demand Anodyne DRD4 19 41 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880736657 CD On-Demand Anodyne SIGMAR1 33 48 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880736657 CD On-Demand Anodyne HSD11B1 50 47 O=C(NC1CSC1)[C@@H]1CCCN1Cc1ccccc1 ZINC000880736657 CD On-Demand Anodyne PREP 77 37 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccccc1 ZINC000880736658 CD On-Demand Anodyne ACE 44 38 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccccc1 ZINC000880736658 CD On-Demand Anodyne DRD4 19 41 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccccc1 ZINC000880736658 CD On-Demand Anodyne SIGMAR1 33 48 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccccc1 ZINC000880736658 CD On-Demand Anodyne HSD11B1 50 47 O=C(NC1CSC1)[C@H]1CCCN1Cc1ccccc1 ZINC000880736658 CD On-Demand Anodyne PREP 77 37 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736659 GI On-Demand Anodyne RBP4 52 34 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880736660 GI On-Demand Anodyne RBP4 52 34 COCCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880736665 CE On-Demand Anodyne CNR1 34 60 COCCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880736665 CE On-Demand Anodyne CNR2 63 60 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880736668 DH On-Demand Anodyne RBP4 54 36 O=C(CNC(=O)c1cc(F)cc(F)c1)NC1CSC1 ZINC000880736671 CC On-Demand Anodyne CCR2 55 41 COCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880736672 CD On-Demand Anodyne DRD4 48 37 COCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880736672 CD On-Demand Anodyne MTNR1A 29 42 COCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880736672 CD On-Demand Anodyne MTNR1B 24 42 COCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880736672 CD On-Demand Anodyne PLA2G4B 43 43 COCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880736672 CD On-Demand Anodyne EPHX2 15 41 Cn1nc(C(C)(C)C)cc1C(=O)NC1CSC1 ZINC000880736678 CD On-Demand Anodyne CTSV 44 34 C=CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736679 EH On-Demand Mild EPHX2 41 42 C=CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736679 EH On-Demand Mild CXCR3 19 40 O=C(Cc1ccc2c(c1)OCO2)NC1CSC1 ZINC000880736680 CD On-Demand Anodyne NOS2 85 33 O=C(Cc1ccc2c(c1)OCO2)NC1CSC1 ZINC000880736680 CD On-Demand Anodyne MCHR1 24 52 O=C(Cc1ccc2c(c1)OCO2)NC1CSC1 ZINC000880736680 CD On-Demand Anodyne LUXR 46 49 O=C(CSCC(=O)NC1CSC1)Nc1cccc(Br)c1 ZINC000880736681 GE On-Demand Anodyne EGFR 20 42 CC(C)(C)OC(=O)N1CCC(n2cc(C(=O)NC3CSC3)nn2)CC1 ZINC000880736706 FD On-Demand Anodyne GPR119 40 39 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880736708 FI On-Demand Anodyne TRPV1 24 41 O=C(NC1CSC1)c1ccc(OCc2ccccc2)nc1 ZINC000880736711 DF On-Demand Anodyne SSTR5 20 40 O=C(NC1CSC1)c1ccc(OCc2ccccc2)nc1 ZINC000880736711 DF On-Demand Anodyne SLC6A5 37 41 O=C(NC1CSC1)c1ccc(OCc2ccccc2)nc1 ZINC000880736711 DF On-Demand Anodyne HPGDS 34 46 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne DRD4 27 48 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne CHRM3 20 42 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne SIGMAR1 21 51 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne SSTR5 44 40 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne CCR3 15 48 O=C(NC1CSC1)c1cccc(CN2CCS(=O)(=O)CC2)c1 ZINC000880736721 EC On-Demand Anodyne MCHR1 25 48 COCCCOc1ccc(C(=O)NC2CSC2)cn1 ZINC000880736723 CD On-Demand Anodyne HPGDS 32 40 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CTSB 51 46 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CYSP_TRYCR 46 39 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CTSK 31 46 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CTSL 40 44 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne PREP 21 46 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CAPNS1 61 35 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CTSS 18 46 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CAPN1 71 39 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne CAPN2 123 40 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne NPR 71 37 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne NAAA 55 46 O=C(CNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880736724 CD On-Demand Anodyne PSMB5 16 40 CS(=O)(=O)Nc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880736725 DD On-Demand Anodyne MAPK11 27 40 CS(=O)(=O)Nc1cc(C(=O)NC2CSC2)ccc1Cl ZINC000880736725 DD On-Demand Anodyne MAPK14 27 40 CCOC[C@H](O)CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736726 GE On-Demand Anodyne ABCB1 27 41 O=C(NC1CSC1)c1ccc(N2CCCC2)nc1 ZINC000880736732 CD On-Demand Anodyne HDAC1 18 41 O=C(NC1CSC1)c1ccc(N2CCCC2)nc1 ZINC000880736732 CD On-Demand Anodyne HPGDS 38 62 CC(C)(C)OC(=O)NCCCCCCC(=O)NC1CSC1 ZINC000880736737 DF On-Demand Anodyne EPHX2 15 43 O=C(Cc1cccc(Br)c1)NC1CSC1 ZINC000880736744 CE On-Demand Anodyne SIGMAR1 15 59 O=C(Cc1cccc(Br)c1)NC1CSC1 ZINC000880736744 CE On-Demand Anodyne LUXR 24 44 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne ACE 40 43 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne MME 83 36 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne ANPEP 53 36 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne PTAFR 21 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne FCER2 48 33 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTSB 35 43 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne PAPA1_CARPA 34 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CYSP_TRYCR 63 41 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTSK 15 43 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTSL 43 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne NPFFR2 41 38 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne TIMP3 62 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTRB1 23 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTSS 24 50 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne MMP9 17 44 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CAPN2 21 41 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne ACE2 51 34 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne CTSV 34 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne MMP7 15 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne MMP1 19 44 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne PSMB5 52 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne BLA1_STEMA 59 37 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne PSMB8 22 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne NPFFR1 50 38 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736764 ED On-Demand Anodyne GPR142 61 36 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne ACE 40 43 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne MME 83 36 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne ANPEP 53 36 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne PTAFR 21 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne FCER2 48 33 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTSB 35 43 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne PAPA1_CARPA 34 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CYSP_TRYCR 63 41 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTSK 15 43 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTSL 43 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne NPFFR2 41 38 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne TIMP3 62 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTRB1 23 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTSS 24 50 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne MMP9 17 44 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CAPN2 21 41 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne ACE2 51 34 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne CTSV 34 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne MMP7 15 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne MMP1 19 44 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne PSMB5 52 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne BLA1_STEMA 59 37 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne PSMB8 22 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne NPFFR1 50 38 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccnc1 ZINC000880736765 ED On-Demand Anodyne GPR142 61 36 COc1cc(I)c(C(=O)NC2CSC2)cc1OC ZINC000880736771 GE On-Demand Anodyne HTR4 26 41 N#Cc1ccccc1OCc1ccc(C(=O)NC2CSC2)o1 ZINC000880736806 DF On-Demand Mild ADRB1 44 35 N#Cc1ccccc1OCc1ccc(C(=O)NC2CSC2)o1 ZINC000880736806 DF On-Demand Mild EZH2 38 40 CN1CCC(CNC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736813 EG On-Demand Anodyne CCR3 45 42 CN1CCC(CNC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736813 EG On-Demand Anodyne CACNA1I 66 39 O=C(NC1CSC1)c1c[nH]c2ncccc12 ZINC000880736814 BD On-Demand Anodyne PIM1 40 35 CCCCNC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736821 GI On-Demand Anodyne ASAH1 46 32 COC(=O)C1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736823 FH On-Demand Anodyne EPHX2 48 46 C=C(C)CN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736834 FI On-Demand Mild EPHX2 41 44 C=C(C)CN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736834 FI On-Demand Mild CXCR3 20 41 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)c1ccc2c(c1)CCC(=O)N2 ZINC000880736838 GJ On-Demand Anodyne GRIN2B 15 42 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCS1 ZINC000880736847 DH On-Demand Anodyne RBP4 53 34 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne CHRM2 21 47 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne CHRM1 16 47 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne DRD2 30 54 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne DRD4 68 54 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne ACHE 52 47 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne DRD3 23 54 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne CHRM3 29 47 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne LTA4H 27 48 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne HRH3 15 49 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne SIGMAR1 85 74 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne CCR3 36 45 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne SLC18A3 20 40 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne EPHX2 28 51 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne MCHR1 43 47 O=C(NC1CSC1)C1CCN(Cc2ccccc2)CC1 ZINC000880736848 CE On-Demand Anodyne CACNA1G 46 51 COc1cccc([C@@H](C)C(=O)NC2CSC2)c1 ZINC000880736852 CE On-Demand Anodyne MTNR1A 37 42 COc1cccc([C@@H](C)C(=O)NC2CSC2)c1 ZINC000880736852 CE On-Demand Anodyne MTNR1B 37 42 COc1cccc([C@H](C)C(=O)NC2CSC2)c1 ZINC000880736853 CE On-Demand Anodyne MTNR1A 37 42 COc1cccc([C@H](C)C(=O)NC2CSC2)c1 ZINC000880736853 CE On-Demand Anodyne MTNR1B 37 42 CCc1nnc2n1CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)C2 ZINC000880736857 FG On-Demand Anodyne P2RX7 25 51 Cc1noc(C2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880736864 FI On-Demand Anodyne RBP4 47 39 Cc1noc(C2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880736864 FI On-Demand Anodyne SMO 43 49 Cc1noc(C2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880736864 FI On-Demand Anodyne ETHR 74 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1cccs1 ZINC000880736869 DD On-Demand Anodyne PREP 85 38 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1cccs1 ZINC000880736869 DD On-Demand Anodyne XIAP 24 43 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880736870 DD On-Demand Anodyne PREP 85 38 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1cccs1 ZINC000880736870 DD On-Demand Anodyne XIAP 24 43 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880736884 FH On-Demand Anodyne CACNA1H 64 35 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880736884 FH On-Demand Anodyne RBP4 40 37 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880736884 FH On-Demand Anodyne TRPM8 30 40 O=C(NC1CSC1)c1c[nH]c(C(=O)N2CCCC2)c1 ZINC000880736893 CD On-Demand Anodyne L3MBTL3 50 33 O=C(NC1CSC1)c1ccc(OCC2CC2)cc1 ZINC000880736897 CE On-Demand Anodyne GRIN2B 15 51 O=C(NC1CSC1)c1ccc(OCC2CC2)cc1 ZINC000880736897 CE On-Demand Anodyne SLC6A5 37 41 O=C(NC1CSC1)c1ccc(OCC2CC2)cc1 ZINC000880736897 CE On-Demand Anodyne PLAU 23 41 O=C(NC1CSC1)c1ccc(OCC2CC2)cc1 ZINC000880736897 CE On-Demand Anodyne ST14 20 41 O=C(NC1CSC1)c1ccc(OCC2CC2)cc1 ZINC000880736897 CE On-Demand Anodyne AOC3 15 48 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne DRD2 18 46 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne DRD4 42 46 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne ACHE 37 40 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne SLC6A1 163 42 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne DRD3 16 44 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne CHRM3 17 42 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne HRH3 15 40 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne SIGMAR1 58 58 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne CCR3 32 41 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne EPHX2 21 42 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne MCHR1 20 44 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne CACNA1G 20 41 O=C(NC1CSC1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880736900 CE On-Demand Anodyne BIRC2 29 45 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne DRD2 18 46 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne DRD4 42 46 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne ACHE 37 40 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne SLC6A1 163 42 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne DRD3 16 44 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne CHRM3 17 42 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne HRH3 15 40 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne SIGMAR1 58 58 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne CCR3 32 41 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne EPHX2 21 42 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne MCHR1 20 44 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne CACNA1G 20 41 O=C(NC1CSC1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880736901 CE On-Demand Anodyne BIRC2 29 45 CC(=O)c1cccc(OCCCC(=O)NC2CSC2)c1 ZINC000880736904 CE On-Demand Anodyne PLA2G4B 29 40 Cc1nc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cn1C ZINC000880736929 FC On-Demand Anodyne EPHX2 39 46 O=C(NC1CSC1)c1csc(-c2ccc3c(c2)OCO3)n1 ZINC000880736931 DE On-Demand Anodyne CLK4 48 34 COCCCOC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880736950 FH On-Demand Anodyne RBP4 32 40 O=C(NC1CSC1)c1ccccc1OCC1CC1 ZINC000880736954 CE On-Demand Anodyne HCN1 56 35 O=C(NC1CSC1)c1ccccc1OCC1CC1 ZINC000880736954 CE On-Demand Anodyne HCN4 45 35 NS(=O)(=O)Cc1ccc(C(=O)NC2CSC2)cc1 ZINC000880736955 CC On-Demand Anodyne CA2 18 40 NS(=O)(=O)Cc1ccc(C(=O)NC2CSC2)cc1 ZINC000880736955 CC On-Demand Anodyne CA14 15 40 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880736980 CD On-Demand Anodyne SLC6A1 75 34 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880736980 CD On-Demand Anodyne SIGMAR1 17 44 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccnc2)C1 ZINC000880736980 CD On-Demand Anodyne CHRNA7 46 37 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccnc2)C1 ZINC000880736981 CD On-Demand Anodyne SLC6A1 75 34 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccnc2)C1 ZINC000880736981 CD On-Demand Anodyne SIGMAR1 17 44 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccnc2)C1 ZINC000880736981 CD On-Demand Anodyne CHRNA7 46 37 O=C(Cc1csc(-c2ccc3c(c2)OCO3)n1)NC1CSC1 ZINC000880736983 EE On-Demand Anodyne TGFBR1 15 45 O=C(Cc1csc(-c2ccc3c(c2)OCO3)n1)NC1CSC1 ZINC000880736983 EE On-Demand Anodyne CLK2 45 38 O=C(Cc1csc(-c2ccc3c(c2)OCO3)n1)NC1CSC1 ZINC000880736983 EE On-Demand Anodyne CLK4 63 38 O=C(NC1CSC1)c1ccc(N2CCOCC2)cc1 ZINC000880736984 CD On-Demand Anodyne HPGDS 31 42 O=C(CCn1ccnc1)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737020 ED On-Demand Anodyne TBXAS1 41 41 O=C(CCn1ccnc1)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737020 ED On-Demand Anodyne KCNK3 60 36 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne SLC6A1 43 34 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne CYSLTR2 50 35 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne HRH3 15 44 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne CPT1A 101 39 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne CPT2 44 34 O=C(NC1CSC1)[C@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737036 ED On-Demand Anodyne EPHX2 20 42 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne SLC6A1 43 34 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne CYSLTR2 50 35 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne HRH3 15 44 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne CPT1A 101 39 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne CPT2 44 34 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)CCOc2ccccc2)C1 ZINC000880737037 ED On-Demand Anodyne EPHX2 20 42 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne KLK3 64 33 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CTSB 44 41 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CYSP_TRYCR 44 37 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CTSK 28 41 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CTSL 37 41 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne PREP 19 44 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CAPNS1 58 34 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CAPN1 66 47 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne CAPN2 113 47 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne NPR 68 38 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne NAAA 41 43 O=C(CCCNC(=O)OCc1ccccc1)NC1CSC1 ZINC000880737039 DD On-Demand Anodyne POLG_WNV 42 37 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737041 GJ On-Demand Anodyne LPL 42 33 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737041 GJ On-Demand Anodyne P2RY1 57 39 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737041 GJ On-Demand Anodyne RIPK1 40 32 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737041 GJ On-Demand Anodyne KCNK3 71 36 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737041 GJ On-Demand Anodyne KCNK9 63 36 CCOc1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880737043 CE On-Demand Anodyne PPO2 29 42 CCOc1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880737043 CE On-Demand Anodyne FFAR4 42 32 CN1C[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1=O ZINC000880737047 DE On-Demand Anodyne EPHX2 17 40 CN1C[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1=O ZINC000880737048 DE On-Demand Anodyne EPHX2 17 40 N#CCOc1ccccc1C(=O)NC1CSC1 ZINC000880737055 BD On-Demand Mild HCN1 51 31 N#CCOc1ccccc1C(=O)NC1CSC1 ZINC000880737055 BD On-Demand Mild HCN4 40 30 COc1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737056 CD On-Demand Anodyne DRD4 41 31 COc1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737056 CD On-Demand Anodyne MTNR1A 58 47 COc1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737056 CD On-Demand Anodyne MTNR1B 51 47 Cn1cc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880737063 DF On-Demand Anodyne TRPV1 17 41 Cn1cc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880737063 DF On-Demand Anodyne NAMPT 19 40 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)c1cccnc1 ZINC000880737070 DI On-Demand Anodyne KCNQ2 32 41 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne MTNR1A 55 36 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne MTNR1B 40 34 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne SSTR3 17 48 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne CA9 24 53 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne MCHR1 18 42 COc1ccc(CC(=O)NCc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880737073 FE On-Demand Anodyne PROKR1 58 32 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne F2 64 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne PLG 21 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne PRSS1 22 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne ACE 54 44 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne FKBP1A 45 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne OPRM1 28 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne MME 22 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne SIGMAR1 18 42 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne TRY1_BOVIN 73 36 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne CPT2 41 33 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne DPP4 22 45 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne PREP 120 44 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne LGMN 57 39 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne XIAP 53 39 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne BRCA1 53 33 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737075 DD On-Demand Anodyne TMPRSS11D 64 35 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne F2 64 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne PLG 21 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne PRSS1 22 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne ACE 54 44 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne FKBP1A 45 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne OPRM1 28 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne MME 22 41 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne SIGMAR1 18 42 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne TRY1_BOVIN 73 36 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne CPT2 41 33 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne DPP4 22 45 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne PREP 120 44 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne LGMN 57 39 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne XIAP 53 39 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne BRCA1 53 33 O=C(NC1CSC1)[C@H]1CCCN1C(=O)Cc1ccccc1 ZINC000880737076 DD On-Demand Anodyne TMPRSS11D 64 35 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne DRD4 24 45 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne SLC6A1 133 42 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne CHRM3 15 40 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne SIGMAR1 24 52 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne CCR3 72 45 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne MLNR 33 41 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne MCHR1 26 43 O=C(NC1CSC1)[C@@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737100 DE On-Demand Anodyne CACNA1G 29 43 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne DRD4 24 45 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne SLC6A1 133 42 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne CHRM3 15 40 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne SIGMAR1 24 52 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne CCR3 72 45 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne MLNR 33 41 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne MCHR1 26 43 O=C(NC1CSC1)[C@H]1CCCN(Cc2cccc(F)c2)C1 ZINC000880737101 DE On-Demand Anodyne CACNA1G 29 43 O=C(CCn1ccnc1)NC1CSC1 ZINC000880737121 BC On-Demand Anodyne TBXAS1 46 48 NC(=O)c1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880737122 CC On-Demand Anodyne HIF1A 16 43 NC(=O)c1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880737122 CC On-Demand Anodyne TRAR 33 40 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880737144 FG On-Demand Anodyne RBP4 59 41 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCCO1 ZINC000880737151 DH On-Demand Anodyne RBP4 52 34 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCCO1 ZINC000880737152 DH On-Demand Anodyne RBP4 52 34 CCC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737167 CD On-Demand Anodyne MAPK14 15 40 CCC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737167 CD On-Demand Anodyne EPHX2 18 43 CCC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737167 CD On-Demand Anodyne KCNK3 104 40 CCC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880737167 CD On-Demand Anodyne KCNK9 63 40 O=C(COc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880737181 CE On-Demand Anodyne PPARD 43 43 O=C(COc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880737181 CE On-Demand Anodyne SLC6A5 34 42 O=C(COc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880737181 CE On-Demand Anodyne MCHR1 17 48 O=C(COc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880737181 CE On-Demand Anodyne TRAR 47 46 C[C@H]1CN(c2ccc(C(=O)NC3CSC3)cn2)C[C@@H](C)O1 ZINC000880737193 DD On-Demand Anodyne HPGDS 31 44 C[C@H]1CN(c2ccc(C(=O)NC3CSC3)cn2)C[C@H](C)O1 ZINC000880737195 DD On-Demand Anodyne HPGDS 31 44 O=C(NC1CSC1)C1CCN(C(=O)CCc2ccccc2)CC1 ZINC000880737199 EE On-Demand Anodyne GRIN2B 22 53 O=C(NC1CSC1)C1CCN(C(=O)CCc2ccccc2)CC1 ZINC000880737199 EE On-Demand Anodyne SIGMAR1 18 49 O=C(NC1CSC1)C1CCN(C(=O)CCc2ccccc2)CC1 ZINC000880737199 EE On-Demand Anodyne C3AR1 45 45 O=C(NC1CSC1)C1CCN(C(=O)CCc2ccccc2)CC1 ZINC000880737199 EE On-Demand Anodyne PREP 57 45 O=C(NC1CSC1)C1CCN(C(=O)CCc2ccccc2)CC1 ZINC000880737199 EE On-Demand Anodyne EPHX2 36 47 Cc1cc(C(=O)NC2CSC2)nn1-c1ccccc1 ZINC000880737206 CE On-Demand Anodyne MAPK14 16 40 Cc1cc(C(=O)NC2CSC2)nn1-c1ccccc1 ZINC000880737206 CE On-Demand Anodyne FPR1 18 40 COC(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880737210 CD On-Demand Anodyne DRD4 40 31 CN(CC(=O)NC1CSC1)S(=O)(=O)c1ccccc1 ZINC000880737220 DC On-Demand Anodyne CCR5 20 40 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737232 GI On-Demand Anodyne HRH2 26 42 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737232 GI On-Demand Anodyne MTNR1A 25 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737232 GI On-Demand Anodyne MTNR1B 23 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880737232 GI On-Demand Anodyne EPHX2 22 40 O=C(CNC(=O)c1ccncc1)NC1CSC1 ZINC000880737245 CC On-Demand Anodyne CCR2 41 39 CCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880737248 CE On-Demand Anodyne DRD4 44 34 CCCOc1cccc(C(=O)NC2CSC2)c1 ZINC000880737248 CE On-Demand Anodyne PLA2G4B 65 47 N#Cc1ccc(C(=O)NCC(=O)NC2CSC2)cc1 ZINC000880737250 CC On-Demand Mild CCR2 30 40 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737260 FH On-Demand Anodyne RBP4 50 32 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737261 FH On-Demand Anodyne RBP4 50 32 COc1ccccc1[C@@H](O)CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880737297 FH On-Demand Anodyne SOAT1 22 41 O=C(CNS(=O)(=O)c1ccc(Cl)s1)NC1CSC1 ZINC000880737298 EC On-Demand Anodyne CCR4 43 33 O=C(NC1CSC1)c1c[nH]c2ccc([N+](=O)[O-])cc12 ZINC000880737299 CD On-Demand Bother GABRA1 21 60 O=C(NC1CSC1)c1c[nH]c2ccc([N+](=O)[O-])cc12 ZINC000880737299 CD On-Demand Bother GABRA5 17 60 O=C(NC1CSC1)c1c[nH]c2ccc([N+](=O)[O-])cc12 ZINC000880737299 CD On-Demand Bother GABRA2 20 60 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880737308 ED On-Demand Anodyne PREP 26 40 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880737308 ED On-Demand Anodyne TRPC6 40 38 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880737309 ED On-Demand Anodyne PREP 26 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccc2c(c1)OCO2 ZINC000880737309 ED On-Demand Anodyne TRPC6 40 38 O=C(CCc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880737312 CG On-Demand Anodyne SIGMAR1 21 46 O=C(CCc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880737312 CG On-Demand Anodyne LUXR 38 42 O=C(NC1CSC1)c1ccc2nncn2c1 ZINC000880737317 BC On-Demand Anodyne MAPK13 47 33 CC(=O)CCc1ccc(OCCC(=O)NC2CSC2)cc1 ZINC000880737319 DE On-Demand Anodyne PLA2G4B 43 35 CC(=O)CCc1ccc(OCCC(=O)NC2CSC2)cc1 ZINC000880737319 DE On-Demand Anodyne PPO2 30 41 CC(=O)CCc1ccc(OCCC(=O)NC2CSC2)cc1 ZINC000880737319 DE On-Demand Anodyne FFAR4 41 31 O=C(COCCc1ccccc1)NC1CSC1 ZINC000880737321 CD On-Demand Anodyne GRIN2B 15 40 O=C(COCCc1ccccc1)NC1CSC1 ZINC000880737321 CD On-Demand Anodyne NAAA 37 40 Cn1cc([C@@H]2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)C2)cn1 ZINC000880737325 FH On-Demand Anodyne RBP4 57 38 Cc1oc(-c2ccco2)nc1CC(=O)NC1CSC1 ZINC000880737328 CE On-Demand Anodyne PDE8B 42 30 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(Cl)s2)CC1 ZINC000880737360 EE On-Demand Anodyne EPHX2 21 49 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(Cl)s2)CC1 ZINC000880737360 EE On-Demand Anodyne L3MBTL3 32 45 O=C(CCCOc1ccc(Cl)cc1)NC1CSC1 ZINC000880737364 CF On-Demand Anodyne PLA2G4B 47 35 O=C(CCCOc1ccc(Cl)cc1)NC1CSC1 ZINC000880737364 CF On-Demand Anodyne TRAR 28 43 O=C(NC1CSC1)c1ccnc(OCc2ccccc2)c1 ZINC000880737389 DF On-Demand Anodyne KDM4E 33 44 CN1CCC(C(=O)NC2CSC2)CC1 ZINC000880737401 BC On-Demand Anodyne EPHX2 17 41 C[C@@H](Cc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880737426 CE On-Demand Anodyne ACE 27 43 C[C@@H](Cc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880737426 CE On-Demand Anodyne AVPR1A 31 40 C[C@@H](Cc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880737426 CE On-Demand Anodyne MME 53 43 C[C@@H](Cc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880737426 CE On-Demand Anodyne ACE2 58 40 C[C@@H](Cc1ccc(F)cc1)C(=O)NC1CSC1 ZINC000880737426 CE On-Demand Anodyne LEF 43 34 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880737434 ED On-Demand Anodyne CCR3 60 35 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880737434 ED On-Demand Anodyne MLNR 30 42 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880737435 ED On-Demand Anodyne CCR3 60 35 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccc(F)cc2)C1 ZINC000880737435 ED On-Demand Anodyne MLNR 30 42 O=C(CCCOCCc1ccccc1)NC1CSC1 ZINC000880737436 CE On-Demand Anodyne GRIN2B 21 45 O=C(CCCOCCc1ccccc1)NC1CSC1 ZINC000880737436 CE On-Demand Anodyne SIGMAR1 16 43 O=C(CCCOCCc1ccccc1)NC1CSC1 ZINC000880737436 CE On-Demand Anodyne NAAA 37 40 O=C(CCCOCCc1ccccc1)NC1CSC1 ZINC000880737436 CE On-Demand Anodyne TNKS 40 31 O=C(CCCc1ccc(Cl)cc1)NC1CSC1 ZINC000880737439 CF On-Demand Anodyne LUXR 19 46 Cc1ccc(C(=O)N2CCC[C@H](C(=O)NC3CSC3)C2)cc1 ZINC000880737443 DE On-Demand Anodyne EPHX2 23 62 Cc1ccc(C(=O)N2CCC[C@H](C(=O)NC3CSC3)C2)cc1 ZINC000880737443 DE On-Demand Anodyne L3MBTL3 69 40 O=C(C[C@H](NC(=O)c1ccc(O)cc1)c1ccccc1)NC1CSC1 ZINC000880737446 FE On-Demand Anodyne UTS2 45 36 O=C(C[C@@H](NC(=O)c1ccc(O)cc1)c1ccccc1)NC1CSC1 ZINC000880737447 FE On-Demand Anodyne UTS2 45 36 O=C(COc1cccc(NC(=O)C2CC2)c1)NC1CSC1 ZINC000880737448 DD On-Demand Anodyne EPHX2 27 46 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne GRIN2B 41 55 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne SIGMAR1 15 51 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne CTSK 16 43 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne CTSL 23 43 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne PREP 41 46 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne EPHX2 39 49 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne TGM2 42 46 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne DPP7 19 43 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne F13A1 47 46 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne CCR8 25 41 O=C(NC1CSC1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880737450 EE On-Demand Anodyne SLC12A5 49 37 O=C(Cc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880737451 CE On-Demand Anodyne CSNK1D 19 41 O=C(Cc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880737451 CE On-Demand Anodyne EPHX2 42 45 O=C(Cc1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880737451 CE On-Demand Anodyne TRAR 45 46 CN(C)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737469 DG On-Demand Anodyne RBP4 61 40 O=C(Cc1cc2ccccc2nc1O)NC1CSC1 ZINC000880737472 CD On-Demand Anodyne TNKS 60 33 O=C(CNC(=O)c1c[nH]c2ccccc2c1=O)NC1CSC1 ZINC000880737478 DC On-Demand Anodyne CFTR 41 47 COC(=O)[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880737485 EE On-Demand Anodyne RBP4 46 37 COC(=O)[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)CCO1 ZINC000880737486 EE On-Demand Anodyne RBP4 46 37 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CSC3)CC2)cc1 ZINC000880737489 FC On-Demand Anodyne EPHX2 21 49 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CSC3)CC2)cc1 ZINC000880737489 FC On-Demand Anodyne TGM2 74 39 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CSC3)CC2)cc1 ZINC000880737489 FC On-Demand Anodyne F13A1 72 39 COc1ccc(-c2nc(C)c(C(=O)NC3CSC3)s2)cc1OC ZINC000880737502 FF On-Demand Anodyne PPARD 21 44 C[C@@H](Oc1ccc(C(=O)NC2CSC2)cn1)c1ccccc1 ZINC000880737507 DG On-Demand Anodyne HPGDS 32 42 N#Cc1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737525 BD On-Demand Mild CHRNA10 17 44 N#Cc1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737525 BD On-Demand Mild TNKS 22 42 CN(CCN1CCOCC1)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880737529 EF On-Demand Anodyne CASR 53 40 O=C(CCOCc1ccccc1)NC1CSC1 ZINC000880737545 CD On-Demand Anodyne GRIN2B 19 43 Cn1cc(CN2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)cn1 ZINC000880737548 GG On-Demand Anodyne FAAH 23 42 O=C(Cn1ccc2ccc(Cl)cc21)NC1CSC1 ZINC000880737561 CF On-Demand Anodyne NPY5R 18 58 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880737572 EH On-Demand Anodyne RBP4 44 32 CC[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)O1 ZINC000880737573 EH On-Demand Anodyne RBP4 44 32 O=C(Nc1cccc(C(=O)NC2CSC2)c1)NC1CC1 ZINC000880737578 CD On-Demand Anodyne MAPK14 32 43 O=C(Nc1cccc(C(=O)NC2CSC2)c1)NC1CC1 ZINC000880737578 CD On-Demand Anodyne EPHX2 54 48 O=C(Nc1cccc(C(=O)NC2CSC2)c1)NC1CC1 ZINC000880737578 CD On-Demand Anodyne KCNK3 97 38 O=C(Nc1cccc(C(=O)NC2CSC2)c1)NC1CC1 ZINC000880737578 CD On-Demand Anodyne KCNK9 51 38 COc1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880737583 GG On-Demand Anodyne FAAH 23 45 COc1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)n1 ZINC000880737583 GG On-Demand Anodyne RBP4 26 43 COc1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)c1 ZINC000880737588 GH On-Demand Anodyne DRD4 41 33 COc1ccnc(N2CCN(C(=O)Nc3cccc(F)c3C(C)(F)F)CC2)c1 ZINC000880737588 GH On-Demand Anodyne RBP4 32 45 C[C@@H](Nc1ccc(C(=O)NC2CSC2)cc1[N+](=O)[O-])c1ccccn1 ZINC000880737613 FG On-Demand Bother TAAR1 16 40 O=C(NC1CSC1)C1CCN(C(=O)COc2ccccc2)CC1 ZINC000880737630 ED On-Demand Anodyne CPT1A 129 42 O=C(NC1CSC1)C1CCN(C(=O)COc2ccccc2)CC1 ZINC000880737630 ED On-Demand Anodyne CPT2 51 39 O=C(NC1CSC1)C1CCN(C(=O)COc2ccccc2)CC1 ZINC000880737630 ED On-Demand Anodyne EPHX2 42 50 O=C1CCCc2cc(C(=O)NC3CSC3)ccc2N1 ZINC000880737633 CD On-Demand Anodyne HDAC9 15 46 O=C(NC1CSC1)[C@H]1CCCN1C(=O)c1ccccc1O ZINC000880737637 DD On-Demand Anodyne PREP 66 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1O ZINC000880737638 DD On-Demand Anodyne PREP 66 40 O=C(Cc1cccs1)Nc1nc(CC(=O)NC2CSC2)cs1 ZINC000880737639 FE On-Demand Anodyne CA5B 32 44 O=C(Cc1cccs1)Nc1nc(CC(=O)NC2CSC2)cs1 ZINC000880737639 FE On-Demand Anodyne CA5A 32 44 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)NC1CSC1 ZINC000880737644 DE On-Demand Anodyne P2RX7 35 59 O=C(Cn1c(O)nc2ccccc21)NC1CSC1 ZINC000880737648 CC On-Demand Anodyne TNKS 57 33 O=C(Cn1c(O)nc2ccccc21)NC1CSC1 ZINC000880737648 CC On-Demand Anodyne IMDH_CRYPV 37 40 CN(C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1)S(C)(=O)=O ZINC000880737651 GF On-Demand Anodyne RBP4 59 44 CN(C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1)S(C)(=O)=O ZINC000880737651 GF On-Demand Anodyne SFRP1 46 35 C[C@H](NC(=O)Nc1cccc(F)c1C(C)(F)F)C(=O)NCc1ccccc1 ZINC000880737666 GH On-Demand Anodyne ANPEP 35 45 O=C(NC1CSC1)[C@H]1CC(c2ccccc2)=NO1 ZINC000880737669 CD On-Demand Anodyne LUCI_PHOPY 51 40 O=C(NC1CSC1)[C@@H]1CC(c2ccccc2)=NO1 ZINC000880737670 CD On-Demand Anodyne LUCI_PHOPY 51 40 O=C(COCCOc1ccccc1)NC1CSC1 ZINC000880737681 CD On-Demand Anodyne PLA2G4B 51 35 O=C(CCCc1nc(-c2cccs2)no1)NC1CSC1 ZINC000880737696 DE On-Demand Anodyne ETHR 37 42 O=C(CCCn1cncn1)NC1CSC1 ZINC000880737705 BC On-Demand Anodyne HIS3 66 36 O=C(NC1CSC1)c1nn(-c2ccc(F)c(F)c2)c2c1CCC2 ZINC000880737708 EE On-Demand Anodyne CNR1 51 32 C[C@@H](NC(=O)c1cccc(Cl)c1Cl)C(=O)NC1CSC1 ZINC000880737712 EE On-Demand Anodyne ECR 20 42 C[C@H](NC(=O)c1cccc(Cl)c1Cl)C(=O)NC1CSC1 ZINC000880737713 EE On-Demand Anodyne ECR 20 42 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737722 ED On-Demand Anodyne EPHX2 26 60 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737722 ED On-Demand Anodyne AKR1C3 19 55 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737722 ED On-Demand Anodyne SFRP1 107 39 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737722 ED On-Demand Anodyne WNT3 70 32 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737723 ED On-Demand Anodyne EPHX2 26 60 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737723 ED On-Demand Anodyne AKR1C3 19 55 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737723 ED On-Demand Anodyne SFRP1 107 39 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)c2ccccc2)C1 ZINC000880737723 ED On-Demand Anodyne WNT3 70 32 O=C(CCCc1nc(-c2ccc(F)cc2)no1)NC1CSC1 ZINC000880737728 DE On-Demand Anodyne SPHK1 33 40 O=C(NC1CSC1)c1cccn(Cc2ccccc2)c1=O ZINC000880737730 DD On-Demand Anodyne DRD4 19 45 O=C(NC1CSC1)c1cccn(Cc2ccccc2)c1=O ZINC000880737730 DD On-Demand Anodyne CNR2 19 74 O=C(NC1CSC1)c1cccn(Cc2ccccc2)c1=O ZINC000880737730 DD On-Demand Anodyne POLR1A 36 40 COc1cccc(OC)c1C(=O)NC1CSC1 ZINC000880737733 CD On-Demand Anodyne DRD2 21 42 C=CC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880737734 DI On-Demand Mild RBP4 49 40 O=C(CCc1ccc2ccccc2c1)NC1CSC1 ZINC000880737749 CG On-Demand Anodyne HCAR2 24 43 O=C(CCc1ccc2ccccc2c1)NC1CSC1 ZINC000880737749 CG On-Demand Anodyne LUXR 44 45 CN1CCC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737775 EG On-Demand Anodyne CCR3 51 40 CN1CCC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737775 EG On-Demand Anodyne CACNA1I 48 36 COC(=O)[C@@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737792 EF On-Demand Anodyne RBP4 53 37 COC(=O)[C@H]1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737793 EF On-Demand Anodyne RBP4 53 37 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne GRIN2B 19 48 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne SIGMAR1 26 46 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne PREP 41 40 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne MTNR1A 18 41 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne MTNR1B 16 41 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne FAAH 50 36 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne CES1 58 39 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne NAAA 34 47 O=C(CCCc1ccccc1)NC1CSC1 ZINC000880737802 BE On-Demand Anodyne TNKS 40 31 C[C@H](SCc1ccccc1)C(=O)NC1CSC1 ZINC000880737826 CF On-Demand Anodyne ACE 57 38 C[C@H](SCc1ccccc1)C(=O)NC1CSC1 ZINC000880737826 CF On-Demand Anodyne MME 64 38 O=C(NC1CSC1)c1ccc(OCC(F)(F)F)cc1 ZINC000880737830 CE On-Demand Anodyne SLC6A5 38 48 O=C(NC1CSC1)c1ccc(OCC(F)(F)F)cc1 ZINC000880737830 CE On-Demand Anodyne AOC3 18 47 O=C(CCc1nc(-c2ccccn2)no1)NC1CSC1 ZINC000880737831 CD On-Demand Anodyne FAAH 17 43 O=C(CCc1nc(-c2ccccn2)no1)NC1CSC1 ZINC000880737831 CD On-Demand Anodyne HCAR2 37 45 CCC(=O)N1CCC[C@@H](C(=O)NC2CSC2)C1 ZINC000880737850 CC On-Demand Anodyne EPHX2 23 46 CCC(=O)N1CCC[C@H](C(=O)NC2CSC2)C1 ZINC000880737851 CC On-Demand Anodyne EPHX2 23 46 O=C(NC1CSC1)c1cc(-c2cccnc2)on1 ZINC000880737854 CD On-Demand Anodyne CYP2E1 41 37 O=C(NC1CSC1)c1ccc(Cn2ccnc2)cc1 ZINC000880737861 CD On-Demand Anodyne CYP19A1 18 54 O=C(NC1CSC1)c1ccc(Cn2ccnc2)cc1 ZINC000880737861 CD On-Demand Anodyne CYP11B1 50 49 O=C(NC1CSC1)c1ccc(Cn2ccnc2)cc1 ZINC000880737861 CD On-Demand Anodyne TBXAS1 60 54 O=C(NC1CSC1)c1ccc(Cn2ccnc2)cc1 ZINC000880737861 CD On-Demand Anodyne CYP11B2 25 49 CC(C)c1cccc(OCC(=O)NC2CSC2)c1 ZINC000880737864 CE On-Demand Anodyne PDS 15 42 O=C(NC1CSC1)c1cccc(NC(=O)[C@@H]2Cc3ccccc3O2)c1 ZINC000880737869 FE On-Demand Anodyne KCNK3 65 36 O=C(NC1CSC1)c1cccc(NC(=O)[C@H]2Cc3ccccc3O2)c1 ZINC000880737870 FE On-Demand Anodyne KCNK3 65 36 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCC2)o1 ZINC000880737871 DC On-Demand Anodyne LPL 47 38 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737875 DE On-Demand Anodyne DRD4 22 45 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737875 DE On-Demand Anodyne UTS2R 18 40 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737875 DE On-Demand Anodyne MCHR1 16 41 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737875 DE On-Demand Anodyne NOD2 40 34 C[C@@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737876 DE On-Demand Anodyne DRD4 22 45 C[C@@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737876 DE On-Demand Anodyne UTS2R 18 40 C[C@@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737876 DE On-Demand Anodyne MCHR1 16 41 C[C@@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880737876 DE On-Demand Anodyne NOD2 40 34 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@H](C)O1 ZINC000880737877 DE On-Demand Anodyne DRD4 22 45 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@H](C)O1 ZINC000880737877 DE On-Demand Anodyne UTS2R 18 40 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@H](C)O1 ZINC000880737877 DE On-Demand Anodyne MCHR1 16 41 C[C@H]1CN(Cc2ccc(C(=O)NC3CSC3)cc2)C[C@H](C)O1 ZINC000880737877 DE On-Demand Anodyne NOD2 40 34 COC(=O)N1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737880 FG On-Demand Anodyne EPHX2 41 44 COC(=O)N1CCC[C@@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880737881 FG On-Demand Anodyne EPHX2 41 44 O=C(NC1CSC1)c1cn(-c2ccccc2)nn1 ZINC000880737894 CD On-Demand Anodyne ESRRA 24 47 O=C(NC1CSC1)c1ccc(OC2CCCC2)cc1 ZINC000880737895 CF On-Demand Anodyne EPHX2 28 46 O=C(NC1CSC1)c1ccc(OC2CCCC2)cc1 ZINC000880737895 CF On-Demand Anodyne PLAU 19 42 O=C(NC1CSC1)c1ccc(OC2CCCC2)cc1 ZINC000880737895 CF On-Demand Anodyne ST14 16 42 O=C(COc1cccc(NC(=O)c2ccco2)c1)NC1CSC1 ZINC000880737896 EE On-Demand Anodyne KISS1R 54 35 O=C(COc1cccc(NC(=O)c2ccco2)c1)NC1CSC1 ZINC000880737896 EE On-Demand Anodyne KCNK3 24 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737898 DD On-Demand Anodyne SLC6A1 49 34 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737898 DD On-Demand Anodyne SIGMAR1 18 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737898 DD On-Demand Anodyne PREP 56 39 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737898 DD On-Demand Anodyne EPHX2 23 44 O=C(NC1CSC1)[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737898 DD On-Demand Anodyne BIRC2 21 49 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737899 DD On-Demand Anodyne SLC6A1 49 34 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737899 DD On-Demand Anodyne SIGMAR1 18 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737899 DD On-Demand Anodyne PREP 56 39 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737899 DD On-Demand Anodyne EPHX2 23 44 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880737899 DD On-Demand Anodyne BIRC2 21 49 O=C(NC1CSC1)c1cccc(OCc2cccs2)c1 ZINC000880737900 DG On-Demand Anodyne PLG 16 42 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000880737905 EC On-Demand Anodyne EPHX2 42 57 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000880737905 EC On-Demand Anodyne TGM2 47 36 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000880737905 EC On-Demand Anodyne NAMPT 66 44 Cc1nn(-c2ccc(C(F)(F)F)cn2)c(C)c1CC(=O)NC1CSC1 ZINC000880737906 FF On-Demand Anodyne P2RX7 19 48 Cc1cc(C(=O)NC2CSC2)cc(C)c1OCc1cccnc1 ZINC000880737921 EG On-Demand Anodyne CHRNA7 44 38 Cc1cc(C(=O)NC2CSC2)cc(C)c1OCc1cccnc1 ZINC000880737921 EG On-Demand Anodyne SLC6A5 26 42 CCn1c(O)nc2cc(C(=O)NC3CSC3)ccc2c1=O ZINC000880737922 DC On-Demand Anodyne POLR1A 52 35 Cc1nn(-c2ccc(Cl)cc2)c(C)c1CC(=O)NC1CSC1 ZINC000880737923 EF On-Demand Anodyne P2RX7 36 59 CC(=O)Nc1ccc(CCNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880737926 GI On-Demand Anodyne TRPV1 15 45 CC(=O)Nc1ccc(CCNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880737926 GI On-Demand Anodyne RAF1 22 40 O=C(NC1CSC1)c1cccc(OCc2cccnc2)c1 ZINC000880737929 DF On-Demand Anodyne PLG 15 45 O=C(NC1CSC1)c1cccc(OCc2cccnc2)c1 ZINC000880737929 DF On-Demand Anodyne PTAFR 32 42 O=C(NC1CSC1)c1cccc(OCc2cccnc2)c1 ZINC000880737929 DF On-Demand Anodyne CHRNA7 46 42 O=C(NC1CSC1)c1cccc(OCc2cccnc2)c1 ZINC000880737929 DF On-Demand Anodyne SLC6A5 31 47 O=C(NC1CSC1)c1cccc(OCc2cccnc2)c1 ZINC000880737929 DF On-Demand Anodyne PLAU 15 45 O=C(CCCc1nnc(-c2ccccc2)o1)NC1CSC1 ZINC000880737938 DE On-Demand Anodyne CES1 15 40 O=C(CCCc1nnc(-c2ccccc2)o1)NC1CSC1 ZINC000880737938 DE On-Demand Anodyne TNKS 24 49 O=C(NC1CSC1)[C@H]1CC(c2cccc(F)c2)=NO1 ZINC000880737941 CD On-Demand Anodyne LUCI_PHOPY 24 45 O=C(NC1CSC1)[C@@H]1CC(c2cccc(F)c2)=NO1 ZINC000880737942 CD On-Demand Anodyne LUCI_PHOPY 24 45 O=C(Cc1csc2ccccc12)NC1CSC1 ZINC000880737948 CF On-Demand Anodyne FFAR2 50 33 CCOC(=O)N(C)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880737954 GI On-Demand Anodyne RBP4 42 39 O=C(NC1CSC1)[C@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880737955 CD On-Demand Anodyne INHA 24 54 O=C(NC1CSC1)[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880737956 CD On-Demand Anodyne INHA 24 54 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne HTR1A 19 50 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne HTR1D 56 50 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne HTR1B 48 50 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne NQO2 33 55 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne MPO 47 37 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne HTR1E 35 43 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne MTNR1A 81 56 COc1ccc2[nH]cc(CC(=O)NC3CSC3)c2c1 ZINC000880737959 CD On-Demand Anodyne MTNR1B 62 55 O=C(CCCc1nc(-c2ccc(Cl)cc2)no1)NC1CSC1 ZINC000880737962 EF On-Demand Anodyne SPHK1 33 40 O=C(Cc1ccc(-n2cccn2)cc1)NC1CSC1 ZINC000880737963 CD On-Demand Anodyne AMP1_PLAFQ 58 43 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NC1CSC1 ZINC000880737970 ED On-Demand Anodyne PREP 52 35 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NC1CSC1 ZINC000880737970 ED On-Demand Anodyne HCN1 58 39 CCOc1ccccc1C(=O)N1CCC[C@H]1C(=O)NC1CSC1 ZINC000880737970 ED On-Demand Anodyne HCN4 50 39 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NC1CSC1 ZINC000880737971 ED On-Demand Anodyne PREP 52 35 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NC1CSC1 ZINC000880737971 ED On-Demand Anodyne HCN1 58 39 CCOc1ccccc1C(=O)N1CCC[C@@H]1C(=O)NC1CSC1 ZINC000880737971 ED On-Demand Anodyne HCN4 50 39 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880737989 ED On-Demand Anodyne EPHX2 18 62 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1cccs1 ZINC000880737990 ED On-Demand Anodyne EPHX2 18 62 O=C(CCCc1nc2ccccc2[nH]1)NC1CSC1 ZINC000880737991 CE On-Demand Anodyne TNKS 59 35 Cc1cc(C(=O)NC2CSC2)ccc1-n1cnnn1 ZINC000880737994 CC On-Demand Anodyne MAPK14 44 37 Cc1cc(C(=O)NC2CSC2)ccc1-n1cnnn1 ZINC000880737994 CC On-Demand Anodyne MAPK13 69 37 O=C(NC1CSC1)C1CCN(C(=O)N2CCCC2)CC1 ZINC000880738008 CD On-Demand Anodyne EPHX2 19 44 CCOC(=O)N[C@@H](C(=O)NC1CSC1)C(C)C ZINC000880738015 CC On-Demand Anodyne HLA-DRB1 40 39 CCOC(=O)N[C@H](C(=O)NC1CSC1)C(C)C ZINC000880738016 CC On-Demand Anodyne HLA-DRB1 40 39 O=C(NC1CSC1)c1cccc(NC(=O)C2CCCCC2)c1 ZINC000880738021 DG On-Demand Anodyne EPHX2 26 42 O=C(NC1CSC1)c1cccc(NC(=O)C2CCCCC2)c1 ZINC000880738021 DG On-Demand Anodyne KCNK3 86 62 C[C@H](O)c1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880738023 FI On-Demand Anodyne ANPEP 20 40 C[C@H](O)c1ccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)cc1 ZINC000880738023 FI On-Demand Anodyne TRPV1 55 44 Cc1ccccc1[C@@H](CC(=O)NC1CSC1)NC(N)=O ZINC000880738028 CD On-Demand Anodyne CTSA 59 37 Cc1ccccc1[C@H](CC(=O)NC1CSC1)NC(N)=O ZINC000880738029 CD On-Demand Anodyne CTSA 59 37 O=C(Cc1cccc(F)c1)NCC(=O)NC1CSC1 ZINC000880738030 CC On-Demand Anodyne CCR2 44 38 C[C@@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738036 CE On-Demand Anodyne TYK2 18 42 C[C@@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738036 CE On-Demand Anodyne KCNK3 97 39 C[C@@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738036 CE On-Demand Anodyne KCNK9 52 39 C[C@@H]1C[C@@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738037 CE On-Demand Anodyne TYK2 18 42 C[C@@H]1C[C@@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738037 CE On-Demand Anodyne KCNK3 97 39 C[C@@H]1C[C@@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738037 CE On-Demand Anodyne KCNK9 52 39 C[C@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738038 CE On-Demand Anodyne TYK2 18 42 C[C@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738038 CE On-Demand Anodyne KCNK3 97 39 C[C@H]1C[C@H]1C(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880738038 CE On-Demand Anodyne KCNK9 52 39 CCCc1c(C(=O)NC2CSC2)cnn1Cc1ccccc1 ZINC000880738040 DF On-Demand Anodyne CNR2 21 42 O=C(CCCc1ncc(-c2ccccc2)o1)NC1CSC1 ZINC000880738047 DF On-Demand Anodyne FAAH 56 38 O=C(CCCc1ncc(-c2ccccc2)o1)NC1CSC1 ZINC000880738047 DF On-Demand Anodyne CES1 33 42 O=C(CCCc1ncc(-c2ccccc2)o1)NC1CSC1 ZINC000880738047 DF On-Demand Anodyne CES1D 44 30 COc1ccc2c(c1)C[C@H](C(=O)NC1CSC1)CO2 ZINC000880738072 CD On-Demand Anodyne MTNR1A 16 52 COc1ccc2c(c1)C[C@H](C(=O)NC1CSC1)CO2 ZINC000880738072 CD On-Demand Anodyne ROCK2 39 54 COc1ccc2c(c1)C[C@@H](C(=O)NC1CSC1)CO2 ZINC000880738073 CD On-Demand Anodyne MTNR1A 16 52 COc1ccc2c(c1)C[C@@H](C(=O)NC1CSC1)CO2 ZINC000880738073 CD On-Demand Anodyne ROCK2 39 54 O=C(COc1ccccc1C(F)(F)F)NC1CSC1 ZINC000880738089 CE On-Demand Anodyne SCD1 26 42 O=C(COc1ccccc1C(F)(F)F)NC1CSC1 ZINC000880738089 CE On-Demand Anodyne SCD 26 42 O=C(NC1CSC1)[C@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738093 EF On-Demand Anodyne TRPV1 34 51 O=C(NC1CSC1)[C@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738093 EF On-Demand Anodyne EPHX2 16 40 O=C(NC1CSC1)[C@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738093 EF On-Demand Anodyne SFRP1 74 36 O=C(NC1CSC1)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738094 EF On-Demand Anodyne TRPV1 34 51 O=C(NC1CSC1)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738094 EF On-Demand Anodyne EPHX2 16 40 O=C(NC1CSC1)[C@@H]1CCCN(c2ncccc2C(F)(F)F)C1 ZINC000880738094 EF On-Demand Anodyne SFRP1 74 36 CCOc1ccc(-c2nc(C)c(C(=O)NC3CSC3)s2)cc1 ZINC000880738099 EG On-Demand Anodyne PPARA 16 49 CCOc1ccc(-c2nc(C)c(C(=O)NC3CSC3)s2)cc1 ZINC000880738099 EG On-Demand Anodyne PPARD 19 42 O=C(NC1CSC1)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880738106 DD On-Demand Anodyne SLC18A3 15 45 O=C(NC1CSC1)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880738106 DD On-Demand Anodyne EPHX2 24 55 O=C(NC1CSC1)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880738106 DD On-Demand Anodyne SFRP1 20 44 O=C(NC1CSC1)C1CCN(C(=O)c2cccnc2)CC1 ZINC000880738106 DD On-Demand Anodyne L3MBTL3 68 37 C=CCOc1ccccc1C(=O)NC1CSC1 ZINC000880738107 BE On-Demand Mild HCN1 53 33 C=CCOc1ccccc1C(=O)NC1CSC1 ZINC000880738107 BE On-Demand Mild HCN4 40 31 C[C@@H](CNC(=O)Nc1cccc(F)c1C(C)(F)F)CN1CCCC1 ZINC000880738109 EH On-Demand Anodyne KCNQ2 45 36 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880738116 EG On-Demand Anodyne RBP4 52 34 CC(=O)N[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880738117 EG On-Demand Anodyne RBP4 52 34 NC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880738118 CC On-Demand Anodyne PLG 17 43 NC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880738118 CC On-Demand Anodyne DRD4 42 32 NC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880738118 CC On-Demand Anodyne PLAU 26 43 NC(=O)COc1cccc(C(=O)NC2CSC2)c1 ZINC000880738118 CC On-Demand Anodyne ST14 18 43 COCCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738122 FG On-Demand Anodyne CCR3 42 45 COCCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738122 FG On-Demand Anodyne EPHX2 46 41 COCCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738122 FG On-Demand Anodyne CXCR3 19 40 Cc1ccc2cc(C(=O)NC3CSC3)[nH]c2c1 ZINC000880738130 BE On-Demand Anodyne PYGL 35 44 Cc1ccc2cc(C(=O)NC3CSC3)[nH]c2c1 ZINC000880738130 BE On-Demand Anodyne PYGM 33 44 CC(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880738132 CE On-Demand Anodyne CYSLTR2 44 33 CC(=O)c1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880738132 CE On-Demand Anodyne PLA2G4B 71 36 O=C(NC1CSC1)c1c[nH]c2cc([N+](=O)[O-])ccc12 ZINC000880738144 CD On-Demand Bother GABRA1 18 49 O=C(NC1CSC1)c1c[nH]c2cc([N+](=O)[O-])ccc12 ZINC000880738144 CD On-Demand Bother GABRA2 17 49 CCOc1ccc(-c2noc(CCC(=O)NC3CSC3)n2)cc1 ZINC000880738148 EE On-Demand Anodyne HCAR2 22 42 Cc1cc([C@@H]2CCCN2C(=O)Nc2cccc(F)c2C(C)(F)F)on1 ZINC000880738156 FJ On-Demand Anodyne KCNA5 18 45 COCCn1cc(NC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880738163 EG On-Demand Anodyne P2RY1 40 35 COCCn1cc(NC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880738163 EG On-Demand Anodyne MAPK10 16 41 COCCn1cc(NC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880738163 EG On-Demand Anodyne PANC 50 33 O=C(NC1CSC1)c1c(F)cccc1F ZINC000880738164 BD On-Demand Anodyne DAC 22 41 COCCNS(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880738165 EC On-Demand Anodyne AKR1C3 24 48 O=C(NC1CSC1)c1ccc(OCc2cccnc2)cc1 ZINC000880738168 DF On-Demand Anodyne PTAFR 33 42 O=C(NC1CSC1)c1ccc(OCc2cccnc2)cc1 ZINC000880738168 DF On-Demand Anodyne CHRNA7 47 45 O=C(NC1CSC1)c1ccc(OCc2cccnc2)cc1 ZINC000880738168 DF On-Demand Anodyne ADAM17 28 41 O=C(NC1CSC1)c1ccc(OCc2cccnc2)cc1 ZINC000880738168 DF On-Demand Anodyne SLC6A5 40 58 O=C(NC1CSC1)c1ccc(OCc2cccnc2)cc1 ZINC000880738168 DF On-Demand Anodyne ACHP_LYMST 20 41 O=C(NC1CSC1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000880738193 BC On-Demand Anodyne INHA 19 45 O=C(NC1CSC1)[C@H]1CC(=O)N(C2CC2)C1 ZINC000880738194 BC On-Demand Anodyne INHA 19 45 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne ADRB2 15 41 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne ADRB1 16 41 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne ADRB3 23 41 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne PRTN3 45 33 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne CTSS 19 41 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)NC3CSC3)cc2)cc1 ZINC000880738198 GF On-Demand Anodyne LIMK2 26 42 O=C(NC1CSC1)[C@H]1COc2ccc(Cl)cc2C1 ZINC000880738202 CE On-Demand Anodyne ROCK2 25 51 O=C(NC1CSC1)[C@@H]1COc2ccc(Cl)cc2C1 ZINC000880738203 CE On-Demand Anodyne ROCK2 25 51 O=C(CCc1nc(-c2ccsc2)no1)NC1CSC1 ZINC000880738222 CD On-Demand Anodyne HCAR2 22 42 CCOc1ccccc1C(=O)NCCCC(=O)NC1CSC1 ZINC000880738234 DD On-Demand Anodyne KCNA3 42 43 CCOc1ccccc1C(=O)NCCCC(=O)NC1CSC1 ZINC000880738234 DD On-Demand Anodyne HCN1 80 42 CCOc1ccccc1C(=O)NCCCC(=O)NC1CSC1 ZINC000880738234 DD On-Demand Anodyne HCN4 61 41 CCOc1ccccc1C(=O)NCCCC(=O)NC1CSC1 ZINC000880738234 DD On-Demand Anodyne KCNK3 32 41 CCOc1ccccc1C(=O)NCCCC(=O)NC1CSC1 ZINC000880738234 DD On-Demand Anodyne KCNK9 29 41 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880738236 GJ On-Demand Anodyne ABCB1B 50 39 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880738236 GJ On-Demand Anodyne ABCB1 19 41 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc(F)c1C(C)(F)F)CC2 ZINC000880738236 GJ On-Demand Anodyne ABCG2 30 40 N#Cc1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880738252 BD On-Demand Mild FFAR1 22 40 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738280 GH On-Demand Anodyne MTNR1A 21 44 O=C(CCc1ccc(Cl)cc1)NC1CSC1 ZINC000880738290 CF On-Demand Anodyne LUXR 37 54 O=C(NC1CSC1)C1CCN(C(=O)/C=C\c2ccccc2)CC1 ZINC000880738303 EE On-Demand Anodyne CCR2 15 41 O=C(NC1CSC1)C1CCN(C(=O)/C=C\c2ccccc2)CC1 ZINC000880738303 EE On-Demand Anodyne EPHX2 20 47 O=C(NC1CSC1)C1CCN(C(=O)/C=C/c2ccccc2)CC1 ZINC000880738304 EE On-Demand Anodyne CCR2 15 41 O=C(NC1CSC1)C1CCN(C(=O)/C=C/c2ccccc2)CC1 ZINC000880738304 EE On-Demand Anodyne EPHX2 20 47 O=C(Cc1ccc(NS(=O)(=O)c2cccs2)cc1)NC1CSC1 ZINC000880738305 FE On-Demand Anodyne RORA 15 47 O=C(NC1CSC1)c1ccc(-n2cccn2)nc1 ZINC000880738309 CD On-Demand Anodyne HPGDS 33 40 O=C(NC1CSC1)c1cccc(S(=O)(=O)NC2CCCC2)c1 ZINC000880738314 ED On-Demand Anodyne AKR1C3 45 35 O=C(NC1CSC1)c1cccc(S(=O)(=O)NC2CCCC2)c1 ZINC000880738314 ED On-Demand Anodyne SFRP1 70 38 Cc1nc(SCC(=O)NC2CSC2)[nH]c1Cc1ccccc1 ZINC000880738315 EF On-Demand Anodyne ENPP1 61 33 O=C(NC1CSC1)c1cnn2cccnc12 ZINC000880738323 BC On-Demand Anodyne PIM1 40 35 O=C(NC1CSC1)c1cnn2cccnc12 ZINC000880738323 BC On-Demand Anodyne PIM3 44 35 O=C(CCc1cccc(Br)c1)NC1CSC1 ZINC000880738328 DF On-Demand Anodyne LUXR 39 58 C[C@@H](Oc1ccccc1Cl)C(=O)NC1CSC1 ZINC000880738336 CE On-Demand Anodyne IMDH_CRYPV 20 41 O=C(NC1CSC1)c1cn(Cc2ccccc2)nn1 ZINC000880738352 CD On-Demand Anodyne DRD4 21 40 O=C(NC1CSC1)c1cn(Cc2ccccc2)nn1 ZINC000880738352 CD On-Demand Anodyne SIGMAR1 21 40 Cc1oc(-c2cccs2)nc1CC(=O)NC1CSC1 ZINC000880738354 CE On-Demand Anodyne PPARG 23 42 Cc1oc(-c2cccs2)nc1CC(=O)NC1CSC1 ZINC000880738354 CE On-Demand Anodyne PPARA 39 43 Cc1oc(-c2cccs2)nc1CC(=O)NC1CSC1 ZINC000880738354 CE On-Demand Anodyne PDE8B 47 33 Cc1nn(C)c2ncc(C(=O)NC3CSC3)cc12 ZINC000880738355 CD On-Demand Anodyne MAPK13 48 31 CC[C@H](C)[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738358 CG On-Demand Anodyne KCNQ2 43 36 CC[C@H](C)[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738358 CG On-Demand Anodyne ACE2 43 36 CC[C@@H](C)[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738359 CG On-Demand Anodyne KCNQ2 43 36 CC[C@@H](C)[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738359 CG On-Demand Anodyne ACE2 43 36 O=C(CNS(=O)(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738362 ED On-Demand Anodyne F2 21 49 O=C(CNS(=O)(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738362 ED On-Demand Anodyne TRY2_BOVIN 66 49 NC(=O)COc1ccccc1C(=O)NC1CSC1 ZINC000880738363 CC On-Demand Anodyne HCN1 52 31 NC(=O)COc1ccccc1C(=O)NC1CSC1 ZINC000880738363 CC On-Demand Anodyne HCN4 40 31 O=C(Cc1ccccc1)NCCC(=O)NC1CSC1 ZINC000880738368 CC On-Demand Anodyne SIGMAR1 15 46 O=C(Cc1ccccc1)NCCC(=O)NC1CSC1 ZINC000880738368 CC On-Demand Anodyne CA5B 36 41 O=C(Cc1ccccc1)NCCC(=O)NC1CSC1 ZINC000880738368 CC On-Demand Anodyne CA5A 37 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA2 67 49 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA1 58 48 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA7 61 48 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA13 15 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA5B 53 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA4 63 49 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA5A 55 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA14 40 48 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA12 39 48 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA9 43 49 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CAH_METTE 35 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CYNT 33 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne CA15 23 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CSC2)c1 ZINC000880738369 DC On-Demand Anodyne P96878_MYCTU 40 38 CC[C@@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738370 BE On-Demand Anodyne KCNQ2 52 47 CC[C@H](C(=O)NC1CSC1)c1ccccc1 ZINC000880738371 BE On-Demand Anodyne KCNQ2 52 47 O=C(NC1CSC1)c1cnn(-c2cccc(C(F)(F)F)c2)c1C(F)(F)F ZINC000880738376 GH On-Demand Anodyne CCR2 51 35 O=C(NC1CSC1)C1CCN(C(=O)c2ccoc2)CC1 ZINC000880738381 CD On-Demand Anodyne EPHX2 20 52 O=C(NC1CSC1)C1CCN(C(=O)c2ccoc2)CC1 ZINC000880738381 CD On-Demand Anodyne L3MBTL3 70 37 O=C(COc1ccc(F)c(Cl)c1)NC1CSC1 ZINC000880738386 CE On-Demand Anodyne TRAR 30 44 C=CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738387 BE On-Demand Mild PLAU 22 41 C=CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738387 BE On-Demand Mild ST14 19 41 C=CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738387 BE On-Demand Mild AOC3 15 48 O=C(CCCNC(=O)NC1CCCCC1)NC1CSC1 ZINC000880738390 CD On-Demand Anodyne EPHX2 22 60 O=C(COc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880738391 CF On-Demand Anodyne TRAR 31 42 CCO[C@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880738393 EH On-Demand Anodyne RBP4 53 35 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2cccc3ccccc23)C1 ZINC000880738406 FF On-Demand Anodyne EPHX2 15 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2cccc3ccccc23)C1 ZINC000880738407 FF On-Demand Anodyne EPHX2 15 47 Cc1ccc(CCC(=O)NC2CSC2)cc1Cl ZINC000880738417 CF On-Demand Anodyne LUXR 33 40 O=C(CCn1c(=O)nc(O)c2ccccc21)NC1CSC1 ZINC000880738418 DC On-Demand Anodyne TNKS 65 36 CNC(=O)CN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738421 FE On-Demand Anodyne DRD4 21 41 CNC(=O)CN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738421 FE On-Demand Anodyne EPHX2 43 42 CNC(=O)CN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738421 FE On-Demand Anodyne CXCR3 19 40 O=C(NC1CSC1)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880738423 FF On-Demand Anodyne CHRM2 15 42 O=C(NC1CSC1)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880738423 FF On-Demand Anodyne EPHX2 23 56 O=C(NC1CSC1)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880738423 FF On-Demand Anodyne CCR8 41 31 O=C(NC1CSC1)C1CCN(C(=O)c2cccc3ccccc23)CC1 ZINC000880738423 FF On-Demand Anodyne L3MBTL3 45 44 O=C(CNS(=O)(=O)c1cccnc1)NC1CSC1 ZINC000880738429 CB On-Demand Anodyne TBXAS1 49 39 O=C(CNS(=O)(=O)c1cccnc1)NC1CSC1 ZINC000880738429 CB On-Demand Anodyne NAMPT 43 37 O=C(NC1CSC1)c1cnn(Cc2ccccc2Cl)c1 ZINC000880738434 DE On-Demand Anodyne PANC 42 34 CCn1c(S)nc2cc(C(=O)NC3CSC3)ccc2c1=O ZINC000880738444 DD On-Demand Anodyne POLR1A 50 34 COc1ncccc1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738448 EH On-Demand Anodyne TRPV1 36 42 COc1ncccc1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738448 EH On-Demand Anodyne P2RY1 52 42 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738452 FH On-Demand Anodyne TRPV1 22 40 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738453 FH On-Demand Anodyne TRPV1 22 40 O=C(CCNS(=O)(=O)c1ccc(F)c(F)c1)NC1CSC1 ZINC000880738459 EC On-Demand Anodyne TBXA2R 48 35 Cc1cc(C(=O)NC2CSC2)c2cnn(C(C)C)c2n1 ZINC000880738470 CE On-Demand Anodyne EZH2 16 44 O=C(CCn1nnc2ccccc2c1=O)NC1CSC1 ZINC000880738473 CC On-Demand Anodyne TNKS 64 36 O=C(CCN1c2ccccc2Sc2ccccc21)Nc1ccc(N2CCOCC2)cn1 ZINC000880738480 IJ On-Demand Anodyne STAT6 59 36 CC(=O)N1CCc2cc(C(=O)NC3CSC3)ccc21 ZINC000880738483 CD On-Demand Anodyne HSD17B3 48 32 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne ACE 82 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne OPRM1 65 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne OPRD1 58 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MME 155 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne ANPEP 84 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne TACR1 21 49 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne FCER2 95 38 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne RNPEP 33 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CTSB 54 44 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne PAPA1_CARPA 63 42 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CYSP_TRYCR 66 42 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CTSK 26 41 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CTSL 62 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CPA1 45 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne NPFFR2 67 38 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne TIMP3 84 41 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CAPNS1 69 34 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MMP2 17 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MMP3 24 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MMP8 20 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne GRIA1 52 38 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne HLA-DRB1 62 37 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CTSS 23 41 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CAPN1 83 43 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MMP9 26 41 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne CAPN2 59 44 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne ACE2 71 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne LAP3 41 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne MMP1 31 41 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne FPR1 67 54 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne AMP1_PLAFQ 35 40 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne BLA1_STEMA 65 36 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne POLG_WNV 45 31 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne QRFPR 47 35 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne NPFFR1 70 38 NC(=O)N[C@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738489 CC On-Demand Anodyne GPR142 42 33 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne ACE 82 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne OPRM1 65 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne OPRD1 58 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MME 155 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne ANPEP 84 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne TACR1 21 49 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne FCER2 95 38 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne RNPEP 33 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CTSB 54 44 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne PAPA1_CARPA 63 42 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CYSP_TRYCR 66 42 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CTSK 26 41 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CTSL 62 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CPA1 45 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne NPFFR2 67 38 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne TIMP3 84 41 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CAPNS1 69 34 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MMP2 17 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MMP3 24 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MMP8 20 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne GRIA1 52 38 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne HLA-DRB1 62 37 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CTSS 23 41 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CAPN1 83 43 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MMP9 26 41 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne CAPN2 59 44 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne ACE2 71 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne LAP3 41 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne MMP1 31 41 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne FPR1 67 54 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne AMP1_PLAFQ 35 40 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne BLA1_STEMA 65 36 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne POLG_WNV 45 31 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne QRFPR 47 35 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne NPFFR1 70 38 NC(=O)N[C@@H](Cc1ccccc1)C(=O)NC1CSC1 ZINC000880738490 CC On-Demand Anodyne GPR142 42 33 O=C(CCc1nc(-c2ccncc2)no1)NC1CSC1 ZINC000880738493 CD On-Demand Anodyne HCAR2 23 44 O=C(NC1CSC1)c1cc2cc(Cl)ccc2[nH]1 ZINC000880738499 CF On-Demand Anodyne CYP51A1 24 42 O=C(NC1CSC1)c1cc2cc(Cl)ccc2[nH]1 ZINC000880738499 CF On-Demand Anodyne PYGL 132 55 O=C(NC1CSC1)c1cc2cc(Cl)ccc2[nH]1 ZINC000880738499 CF On-Demand Anodyne PYGM 41 54 O=C(NC1CSC1)c1cc2cc(Cl)ccc2[nH]1 ZINC000880738499 CF On-Demand Anodyne PYK 23 41 O=C(CCc1nc2ccccc2oc1=O)NC1CSC1 ZINC000880738500 CD On-Demand Anodyne TNKS 47 33 O=C(CCNC(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738505 DE On-Demand Anodyne DRD4 15 45 O=C(CCNC(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738505 DE On-Demand Anodyne NMT1 24 40 CC(=O)NCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738510 FG On-Demand Anodyne EPHX2 26 40 CC(=O)NCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738510 FG On-Demand Anodyne RBP4 39 40 CC(=O)NCC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738510 FG On-Demand Anodyne CACNA1I 54 34 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880738511 DD On-Demand Anodyne PAPA1_CARPA 35 59 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880738511 DD On-Demand Anodyne CTSK 15 59 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CSC1 ZINC000880738511 DD On-Demand Anodyne FPR1 33 47 CCn1cc(NC(=O)Nc2cccc(F)c2C(C)(F)F)cn1 ZINC000880738528 DH On-Demand Anodyne MAPK10 16 40 O=C(CSc1nc2ccccc2o1)NC1CSC1 ZINC000880738529 CE On-Demand Anodyne TNKS 47 34 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2cccnc2Cl)CC1 ZINC000880738535 GD On-Demand Anodyne EPHX2 44 53 O=C(NC1CSC1)c1ccc(C(F)(F)F)nc1 ZINC000880738541 CD On-Demand Anodyne HPGDS 37 41 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild FABP3 32 42 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild FABP5 16 45 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild LUXR 39 51 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild TRAR 16 48 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild LASR 68 51 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild NOD1 49 38 CCCCCCCC(=O)NC1CSC1 ZINC000880738542 BF On-Demand Mild CQSS 59 36 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738551 GI On-Demand Anodyne EPHX2 49 50 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738551 GI On-Demand Anodyne CCR8 40 39 O=C(CCNS(=O)(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738598 FD On-Demand Anodyne F2 20 42 O=C(CCNS(=O)(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738598 FD On-Demand Anodyne HTR7 17 46 O=C(CCNS(=O)(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738598 FD On-Demand Anodyne TRY2_BOVIN 63 41 O=C(CCC(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738605 CG On-Demand Anodyne HDAC8 23 41 O=C(CCC(=O)c1ccc2ccccc2c1)NC1CSC1 ZINC000880738605 CG On-Demand Anodyne TNKS 40 30 N#Cc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880738606 FD On-Demand Mild EPHX2 42 57 N#Cc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880738606 FD On-Demand Mild TGM2 48 36 O=C(CCC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1)NC1CSC1 ZINC000880738610 GC On-Demand Anodyne TGM2 76 46 O=C(CCC(=O)N1CCN(S(=O)(=O)c2ccccc2)CC1)NC1CSC1 ZINC000880738610 GC On-Demand Anodyne F13A1 78 46 O=C(CCc1nc(-c2cccs2)no1)NC1CSC1 ZINC000880738612 CD On-Demand Anodyne ETHR 38 44 Cn1ncc2c(=O)n(CC(=O)NC3CSC3)cnc21 ZINC000880738624 CB On-Demand Anodyne Q9M629_MAIZE 43 34 O=C(NC1CSC1)c1cccc(S(=O)(=O)NCc2cccs2)c1 ZINC000880738626 FE On-Demand Anodyne AKR1C3 15 42 CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738628 EH On-Demand Anodyne DRD4 15 41 CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738628 EH On-Demand Anodyne CCR3 32 42 CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738628 EH On-Demand Anodyne EPHX2 51 45 CCN1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738628 EH On-Demand Anodyne CXCR3 22 42 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NC2CSC2)C1 ZINC000880738629 DD On-Demand Anodyne EPHX2 17 44 O=C(NC1CSC1)c1cc2ccccc2cc1NC(=O)C1CC1 ZINC000880738641 EG On-Demand Anodyne PYGL 39 40 O=C(NC1CSC1)c1sccc1S(=O)(=O)N1CCCCC1 ZINC000880738649 ED On-Demand Anodyne EPHX2 16 41 O=C(Cn1c(Cc2ccccc2)nc2ccccc21)NC1CSC1 ZINC000880738651 EF On-Demand Anodyne MAOA 15 45 O=C(Cn1c(Cc2ccccc2)nc2ccccc21)NC1CSC1 ZINC000880738651 EF On-Demand Anodyne PDE6D 52 33 O=C(Cn1c(Cc2ccccc2)nc2ccccc21)NC1CSC1 ZINC000880738651 EF On-Demand Anodyne TNKS 46 32 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)NC3CSC3)c2)cc1 ZINC000880738654 GF On-Demand Anodyne SSTR5 23 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)NC3CSC3)c2)cc1 ZINC000880738654 GF On-Demand Anodyne PRTN3 52 33 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)NC3CSC3)c2)cc1 ZINC000880738654 GF On-Demand Anodyne ALPL 16 46 O=C(COc1cc(Cl)ccc1Cl)NC1CSC1 ZINC000880738655 CF On-Demand Anodyne TRAR 27 40 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)NC1CSC1 ZINC000880738659 FD On-Demand Anodyne MMP2 22 43 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)NC1CSC1 ZINC000880738660 FD On-Demand Anodyne MMP2 22 43 COCC(=O)NC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738669 FF On-Demand Anodyne EPHX2 36 41 COCC(=O)NC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738669 FF On-Demand Anodyne RBP4 43 42 O=C(CCNS(=O)(=O)c1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880738670 GD On-Demand Anodyne MMP14 20 45 O=C(Cc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880738672 CE On-Demand Anodyne LUXR 34 53 O=C(Cc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880738672 CE On-Demand Anodyne TRPM8 32 40 O=C(Cc1ccc(C(F)(F)F)cc1)NC1CSC1 ZINC000880738672 CE On-Demand Anodyne TRAR 27 53 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(F)cc2F)CC1 ZINC000880738674 EE On-Demand Anodyne EPHX2 23 57 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(F)cc2F)CC1 ZINC000880738674 EE On-Demand Anodyne L3MBTL3 44 35 O=C(Cc1ccc2c(c1)CCO2)NC1CSC1 ZINC000880738675 BD On-Demand Anodyne LUXR 45 36 O=C(CCn1cnc2ccccc21)NC1CSC1 ZINC000880738678 CD On-Demand Anodyne TNKS 40 32 CCOC(=O)CC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738679 FI On-Demand Anodyne CCR8 40 38 Cn1cnnc1C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738682 FG On-Demand Anodyne RBP4 55 41 O=C(CCCOc1ccc(F)cc1)NC1CSC1 ZINC000880738688 CE On-Demand Anodyne PLA2G4B 47 35 Cc1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880738689 BE On-Demand Anodyne VIPR1 18 43 O=C(NC1CSC1)c1cnn(-c2ccccc2)c1C(F)(F)F ZINC000880738692 EF On-Demand Anodyne MST1R 43 41 COc1ccc2c(C)c(CCC(=O)NC3CSC3)c(=O)oc2c1 ZINC000880738700 EE On-Demand Anodyne MAOB 38 49 COc1ccc2c(C)c(CCC(=O)NC3CSC3)c(=O)oc2c1 ZINC000880738700 EE On-Demand Anodyne NQO1 50 47 CCCCSCC(=O)NC1CSC1 ZINC000880738724 BD On-Demand Anodyne CES1 17 42 CCCCSCC(=O)NC1CSC1 ZINC000880738724 BD On-Demand Anodyne EST1_PIG 49 42 O=C(NC1CSC1)c1ccc(S(=O)(=O)NCCc2cccs2)cc1 ZINC000880738737 GE On-Demand Anodyne ALOX15 16 41 Cc1cc(C(=O)NC2CSC2)c2cnn(Cc3cccs3)c2n1 ZINC000880738753 EF On-Demand Anodyne GPR142 46 29 O=C(NC1CSC1)c1cc([N+](=O)[O-])ccc1N1CCOCC1 ZINC000880738755 DD On-Demand Bother SLC6A9 15 52 CC(C)CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738764 EH On-Demand Anodyne RBP4 45 35 Cn1c(=O)n(CC(=O)NC2CSC2)c2ccccc21 ZINC000880738768 CC On-Demand Anodyne CALCRL 17 43 C[C@@H](Oc1ccccc1C#N)C(=O)NC1CSC1 ZINC000880738776 CD On-Demand Mild ADRB1 41 32 C[C@@H](Oc1ccccc1C#N)C(=O)NC1CSC1 ZINC000880738776 CD On-Demand Mild EZH2 35 40 CCN1CC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880738784 EG On-Demand Anodyne CCR3 57 41 CCN1CC[C@H](CNC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880738784 EG On-Demand Anodyne CACNA1I 63 37 Cc1oc(-c2ccccc2)nc1CC(=O)NC1CSC1 ZINC000880738788 CE On-Demand Anodyne PPARG 92 45 Cc1oc(-c2ccccc2)nc1CC(=O)NC1CSC1 ZINC000880738788 CE On-Demand Anodyne PPARA 99 47 Cc1oc(-c2ccccc2)nc1CC(=O)NC1CSC1 ZINC000880738788 CE On-Demand Anodyne PDE8B 74 42 CCOC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738797 FH On-Demand Anodyne EPHX2 56 48 CCOC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738797 FH On-Demand Anodyne CXCR3 15 41 CCOC(=O)N1CCC(NC(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738797 FH On-Demand Anodyne CCR8 70 44 O=C(CCc1ccc2c(c1)OCCO2)NC1CSC1 ZINC000880738798 CD On-Demand Anodyne LUXR 56 56 O=C(CCc1ccc2c(c1)OCCO2)NC1CSC1 ZINC000880738798 CD On-Demand Anodyne TRAR 23 40 O=C(Cc1ccccc1)NCC(=O)NC1CSC1 ZINC000880738799 CC On-Demand Anodyne SIGMAR1 15 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne ACE 67 49 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne OPRM1 25 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne OPRD1 24 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CELA1 23 58 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne ELANE 37 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne MME 72 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne ANPEP 42 35 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTSD 16 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CASP3 28 55 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne BMP1 22 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne KLK3 94 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTSB 89 53 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne PAPA1_CARPA 87 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CYSP_TRYCR 67 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTSK 57 56 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTSL 58 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne PGA 38 46 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne PREP 15 49 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CAPNS1 77 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne HLA-DRB1 79 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne REN 25 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne LGMN 17 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne MMP11 45 34 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTSS 34 51 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CAPN1 113 52 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CASP1 38 52 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CTRC 15 56 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CAPN2 166 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne ACE2 41 33 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne PLAU 20 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CASP6 21 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne CASP9 45 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne TPSAB1 25 49 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne NPR 93 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne NAAA 73 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne PSMB5 58 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne BIRC2 42 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne Q6PRC7_IXORI 60 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne SLC12A5 45 33 C[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CSC1 ZINC000880738806 CD On-Demand Anodyne Q9NAW4_PLAFA 38 41 O=C(CCc1ncc(-c2ccccc2)o1)NC1CSC1 ZINC000880738823 CF On-Demand Anodyne FAAH 46 41 O=C(CCc1ncc(-c2ccccc2)o1)NC1CSC1 ZINC000880738823 CF On-Demand Anodyne CES1 25 41 O=C(CCNS(=O)(=O)c1cccnc1)NC1CSC1 ZINC000880738831 DB On-Demand Anodyne TBXA2R 25 40 O=C(CCNS(=O)(=O)c1cccnc1)NC1CSC1 ZINC000880738831 DB On-Demand Anodyne TBXAS1 57 42 O=C(NC1CSC1)c1ccc(OCC(F)(F)F)nc1 ZINC000880738835 CD On-Demand Anodyne HPGDS 40 49 COCCOc1ncccc1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738838 GH On-Demand Anodyne TRPV1 27 40 COCCOc1ncccc1CNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738838 GH On-Demand Anodyne P2RY1 48 41 O=C(NC1CSC1)c1cnn(-c2ccc(F)cc2)c1C(F)(F)F ZINC000880738840 EF On-Demand Anodyne MAPK14 15 41 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738843 FH On-Demand Anodyne RBP4 45 36 O=C(CCn1cnc2sc3c(c2c1=O)CCCC3)NC1CSC1 ZINC000880738859 ED On-Demand Anodyne HTR1B 19 40 NC(=O)COc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738861 CC On-Demand Anodyne SLC6A5 35 40 NC(=O)COc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738861 CC On-Demand Anodyne PLAU 26 44 NC(=O)COc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738861 CC On-Demand Anodyne ST14 24 44 NC(=O)COc1ccc(C(=O)NC2CSC2)cc1 ZINC000880738861 CC On-Demand Anodyne AOC3 17 52 C#CCNS(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880738864 DC On-Demand Mild AKR1C3 21 44 CS(=O)(=O)Nc1ccccc1C(=O)NC1CSC1 ZINC000880738872 CC On-Demand Anodyne PLA2G7 29 40 CS(=O)(=O)Nc1ccccc1C(=O)NC1CSC1 ZINC000880738872 CC On-Demand Anodyne PRTN3 47 35 CS(=O)(=O)Nc1ccccc1C(=O)NC1CSC1 ZINC000880738872 CC On-Demand Anodyne DAC 21 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne F2 47 40 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne ACE 34 43 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne TRY1_BOVIN 47 36 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne PREP 94 51 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne XIAP 40 37 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne SFRP1 41 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne WNT3 45 41 O=C(NC1CSC1)[C@@H]1CCCN1C(=O)c1ccccc1 ZINC000880738883 CD On-Demand Anodyne TMPRSS11D 57 34 O=C(NC1CSC1)c1ccc(Cn2cccn2)cc1 ZINC000880738889 CD On-Demand Anodyne DRD4 18 43 O=C(NC1CSC1)c1ccc(Cn2cccn2)cc1 ZINC000880738889 CD On-Demand Anodyne SSTR5 42 36 Cc1cc(C)nc(-n2nc(C)c(CC(=O)NC3CSC3)c2C)n1 ZINC000880738892 ED On-Demand Anodyne P2RX7 22 49 CCOc1ccc(-c2nc(CC(=O)NC3CSC3)cs2)cc1 ZINC000880738897 EF On-Demand Anodyne PPARD 17 42 O=C(Cc1ccc(-n2cnnn2)cc1)NC1CSC1 ZINC000880738902 CC On-Demand Anodyne KCNJ1 56 44 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne FABP3 32 42 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne FABP5 16 45 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne LUXR 39 51 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne TRAR 16 48 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne LASR 68 51 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne NOD1 49 38 CCCCCCC(=O)NC1CSC1 ZINC000880738903 BE On-Demand Anodyne CQSS 59 36 CCCCCNC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738907 GI On-Demand Anodyne EPHX2 23 41 CCCCCNC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738907 GI On-Demand Anodyne ASAH1 70 35 O=C(CCc1ccc(S(=O)(=O)N2CCCC2)cc1)NC1CSC1 ZINC000880738911 FD On-Demand Anodyne TGM2 66 39 O=C(CCc1ccc(S(=O)(=O)N2CCCC2)cc1)NC1CSC1 ZINC000880738911 FD On-Demand Anodyne F13A1 61 41 O=C(CCc1ccc(S(=O)(=O)N2CCCC2)cc1)NC1CSC1 ZINC000880738911 FD On-Demand Anodyne NAMPT 38 41 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne CHRM2 15 43 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne DRD2 28 49 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne DRD4 85 49 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne ACHE 42 52 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne DRD3 20 49 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne CHRM3 17 43 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne LTA4H 22 45 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne SIGMAR1 80 60 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne FAAH 16 41 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne MCHR1 20 45 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne CACNA1G 23 44 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne CCR8 16 41 O=C(CN1CCN(Cc2ccccc2)CC1)NC1CSC1 ZINC000880738917 DD On-Demand Anodyne NPFFR1 42 37 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne DRD4 56 44 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne NQO2 15 41 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne CTSL 27 43 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne RAF1 25 41 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne CTSS 18 46 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne TAAR1 32 44 COc1cccc(C(=O)NCCNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880738923 GG On-Demand Anodyne KCNK3 37 43 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCc3sccc3C2)c1 ZINC000880738931 GE On-Demand Anodyne AKR1C3 86 73 C=CCNS(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880738951 DC On-Demand Mild AKR1C3 17 44 O=C(NC1CSC1)C1CCN(c2nc3ccccc3o2)CC1 ZINC000880738957 DE On-Demand Anodyne HTR3A 17 43 O=C(NC1CSC1)C1CCN(c2nc3ccccc3o2)CC1 ZINC000880738957 DE On-Demand Anodyne PTGES 40 53 O=C(NC1CSC1)c1cccn1Cc1ccccc1 ZINC000880738961 CE On-Demand Anodyne DRD4 21 41 O=C(NC1CSC1)c1cccn1Cc1ccccc1 ZINC000880738961 CE On-Demand Anodyne SIGMAR1 18 40 C[C@H](CN1CCOCC1)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880738973 EF On-Demand Anodyne EPHX2 17 40 O=C(CNS(=O)(=O)c1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880738975 FD On-Demand Anodyne CACNA1B 54 34 O=C(CNS(=O)(=O)c1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880738975 FD On-Demand Anodyne BDKRB1 21 40 O=C(CNS(=O)(=O)c1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880738975 FD On-Demand Anodyne CCR2 91 45 O=C(CNS(=O)(=O)c1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880738975 FD On-Demand Anodyne SFRP1 71 33 NC(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880738976 BC On-Demand Anodyne KCNK3 51 34 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne FKBP1A 20 53 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP13 46 45 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne ITGA4 36 49 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne CAPNS1 23 47 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP2 21 45 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP3 52 49 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP8 33 44 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne CAPN1 20 54 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP9 29 41 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne EPHX2 17 50 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP7 55 45 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne MMP1 51 49 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne SFRP1 115 36 O=C(NC1CSC1)[C@@H]1CCCN1S(=O)(=O)c1ccccc1 ZINC000880738982 ED On-Demand Anodyne WNT3 83 35 O=C(NC1CSC1)c1cc2cc(F)ccc2[nH]1 ZINC000880738985 CE On-Demand Anodyne PYGL 88 53 O=C(NC1CSC1)c1cc2cc(F)ccc2[nH]1 ZINC000880738985 CE On-Demand Anodyne PLD1 35 44 O=C(NC1CSC1)c1cc2cc(F)ccc2[nH]1 ZINC000880738985 CE On-Demand Anodyne PYGM 36 53 O=C(NC1CSC1)c1cc2cc(F)ccc2[nH]1 ZINC000880738985 CE On-Demand Anodyne PLD2 48 44 O=C(NC1CSC1)c1cc2cc(F)ccc2[nH]1 ZINC000880738985 CE On-Demand Anodyne PYK 27 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738991 GF On-Demand Anodyne CCR8 98 44 CCS(=O)(=O)NC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738991 GF On-Demand Anodyne SFRP1 118 38 CCS(=O)(=O)NC1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880738991 GF On-Demand Anodyne WNT3 83 38 O=C(NC1CSC1)c1cnn(-c2ccccc2F)c1C(F)(F)F ZINC000880738992 EF On-Demand Anodyne MAPK14 16 40 O=C(NC1CSC1)C1(c2ccc(F)cc2)CCCC1 ZINC000880738995 CF On-Demand Anodyne AVPR1A 33 44 O=C(CNS(=O)(=O)c1ccccc1C(F)(F)F)NC1CSC1 ZINC000880738999 FD On-Demand Anodyne SFRP1 97 34 O=C(CNS(=O)(=O)c1ccccc1C(F)(F)F)NC1CSC1 ZINC000880738999 FD On-Demand Anodyne WNT3 61 34 O=C(NC1CSC1)c1ccc(Cn2cncn2)cc1 ZINC000880739008 CD On-Demand Anodyne HIS3 65 33 CN1CCC[C@H](NC(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880739022 DG On-Demand Anodyne EPHX2 39 47 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCOCC2)ccc1F ZINC000880739027 FC On-Demand Anodyne PKM 42 37 O=C(NC1CSC1)c1cc2cc(Br)ccc2[nH]1 ZINC000880739038 DF On-Demand Anodyne PYGL 85 53 O=C(NC1CSC1)c1cc2cc(Br)ccc2[nH]1 ZINC000880739038 DF On-Demand Anodyne PYGM 33 53 O=C(NC1CSC1)c1cc2cc(Br)ccc2[nH]1 ZINC000880739038 DF On-Demand Anodyne PYK 63 45 O=C(NC1CSC1)c1c(F)cccc1Cl ZINC000880739041 BE On-Demand Anodyne PPIA 28 49 O=C(NC1CSC1)c1c(F)cccc1Cl ZINC000880739041 BE On-Demand Anodyne TYK2 23 49 O=C(NC1CSC1)c1cccc(S(=O)(=O)NCC2CC2)c1 ZINC000880739042 ED On-Demand Anodyne NPY5R 27 43 O=C(NC1CSC1)c1cccc(S(=O)(=O)NCC2CC2)c1 ZINC000880739042 ED On-Demand Anodyne AKR1C3 19 44 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA2 58 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA1 46 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA7 52 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA5B 52 35 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA4 46 40 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA5A 55 35 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA14 32 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA12 31 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne CA9 37 43 NS(=O)(=O)c1ccc(Br)c(C(=O)NC2CSC2)c1 ZINC000880739048 FC On-Demand Anodyne P96878_MYCTU 43 37 O=C(NC1CSC1)c1cccc(NC(=O)[C@H]2CCCO2)c1 ZINC000880739050 DD On-Demand Anodyne KCNK3 68 41 O=C(NC1CSC1)c1cccc(NC(=O)[C@@H]2CCCO2)c1 ZINC000880739051 DD On-Demand Anodyne KCNK3 68 41 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880739057 FF On-Demand Anodyne EPHX2 45 54 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880739057 FF On-Demand Anodyne MCHR1 20 40 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880739057 FF On-Demand Anodyne MLYCD 19 44 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880739057 FF On-Demand Anodyne SFRP1 38 45 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000880739057 FF On-Demand Anodyne L3MBTL3 83 41 Cc1nc2c3ccccc3nn2c(C)c1CCC(=O)NC1CSC1 ZINC000880739063 EF On-Demand Anodyne TNKS 57 32 COc1ccc(-c2nnc(SCC(=O)NC3CSC3)o2)cc1 ZINC000880739064 EE On-Demand Anodyne GSK3A 23 43 CC[C@H](C(=O)NC1CSC1)n1nnc(-c2ccc(Cl)cc2)n1 ZINC000880739065 EE On-Demand Anodyne SCARB1 32 46 CC[C@@H](C(=O)NC1CSC1)n1nnc(-c2ccc(Cl)cc2)n1 ZINC000880739067 EE On-Demand Anodyne SCARB1 32 46 O=C(CSc1ccc([N+](=O)[O-])cc1)NC1CSC1 ZINC000880739074 CD On-Demand Bother LUXR 17 41 O=C(CSc1ccc([N+](=O)[O-])cc1)NC1CSC1 ZINC000880739074 CD On-Demand Bother FAS 33 43 O=C(CSc1nc2ccccc2s1)NC1CSC1 ZINC000880739086 CF On-Demand Anodyne LTA4H 21 41 O=C(CSc1nc2ccccc2s1)NC1CSC1 ZINC000880739086 CF On-Demand Anodyne HMOX2 32 41 O=C(CSc1nc2ccccc2s1)NC1CSC1 ZINC000880739086 CF On-Demand Anodyne TNKS 56 32 O=C(CCc1cccc(Cl)c1)NC1CSC1 ZINC000880739089 CF On-Demand Anodyne LUXR 38 41 O=C(COc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880739092 CD On-Demand Bother CACNA1C 55 36 O=C(COc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880739092 CD On-Demand Bother CACNA1D 87 36 O=C(COc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880739092 CD On-Demand Bother ACR 15 44 O=C(COc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880739092 CD On-Demand Bother LUXR 16 41 O=C(COc1cccc([N+](=O)[O-])c1)NC1CSC1 ZINC000880739092 CD On-Demand Bother TRAR 35 45 O=C(CCc1nnc(-c2ccccc2)o1)NC1CSC1 ZINC000880739093 CD On-Demand Anodyne TNKS 27 47 O=C(CCn1cncn1)NC1CSC1 ZINC000880739099 BB On-Demand Anodyne HIS3 72 36 O=C(CCNS(=O)(=O)c1cccc(Cl)c1)NC1CSC1 ZINC000880739104 ED On-Demand Anodyne TBXA2R 42 34 O=C(Cn1nnc2ccccc2c1=O)NC1CSC1 ZINC000880739106 CC On-Demand Anodyne TNKS 59 34 O=C(NC1CSC1)c1csc(S(=O)(=O)N2CCc3ccccc3C2)c1 ZINC000880739112 GE On-Demand Anodyne MMP8 15 42 O=C(NC1CSC1)c1csc(S(=O)(=O)N2CCc3ccccc3C2)c1 ZINC000880739112 GE On-Demand Anodyne AKR1C3 73 51 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCCC2)ccc1Cl ZINC000880739131 FD On-Demand Anodyne EPHX2 19 40 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCCC2)ccc1Cl ZINC000880739131 FD On-Demand Anodyne TGM2 43 36 O=C(CCSc1ccccc1F)NC1CSC1 ZINC000880739141 CF On-Demand Anodyne TNKS 65 37 O=C(CCn1cnc2ccccc2c1=O)NC1CSC1 ZINC000880739143 CD On-Demand Anodyne TNKS 58 34 CS(=O)(=O)NCCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739145 DC On-Demand Anodyne A6YCJ1_9METZ 15 41 O=C(NC1CSC1)c1cc2cc(Cl)ccc2o1 ZINC000880739154 CF On-Demand Anodyne MCHR1 16 42 CN(C)C(=O)c1cccc(CNC(=O)Nc2cccc(F)c2C(C)(F)F)c1 ZINC000880739157 GH On-Demand Anodyne ROCK2 20 40 Cc1nnc(SCC(=O)NC2CSC2)n1Cc1ccccc1 ZINC000880739159 ED On-Demand Anodyne SIGMAR1 17 42 O=C(NC1CSC1)[C@@H]1COc2ccccc2C1 ZINC000880739166 BD On-Demand Anodyne ROCK2 23 47 O=C(NC1CSC1)[C@H]1COc2ccccc2C1 ZINC000880739167 BD On-Demand Anodyne ROCK2 23 47 CS(=O)(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739181 CC On-Demand Anodyne NR3C2 18 41 CS(=O)(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739181 CC On-Demand Anodyne KCNK3 67 35 COc1ccc(-c2noc(CCC(=O)NC3CSC3)n2)cc1 ZINC000880739185 DD On-Demand Anodyne HCAR2 22 44 C[C@@H]1Oc2ccccc2N(CC(=O)NC2CSC2)C1=O ZINC000880739188 CD On-Demand Anodyne ACE 15 42 O=C(NC1CSC1)c1ccc(N2CCOCC2)nc1 ZINC000880739201 CC On-Demand Anodyne DGAT1 19 42 O=C(NC1CSC1)c1ccc(N2CCOCC2)nc1 ZINC000880739201 CC On-Demand Anodyne HPGDS 45 64 O=C(CCCCCn1c(S)nc2ccccc2c1=O)NC1CSC1 ZINC000880739202 FE On-Demand Anodyne HTR7 21 40 O=C(CCCCCn1c(S)nc2ccccc2c1=O)NC1CSC1 ZINC000880739202 FE On-Demand Anodyne TNKS 64 36 O=C(CSc1nnc(C2CC2)n1Cc1ccccc1)NC1CSC1 ZINC000880739207 FF On-Demand Anodyne SIGMAR1 18 43 CCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880739222 CF On-Demand Anodyne CNR1 35 47 CCn1cc(C(=O)NC2CSC2)c2ccccc21 ZINC000880739222 CF On-Demand Anodyne CNR2 62 47 O=C(NC1CSC1)c1cccc(OCc2cscn2)c1 ZINC000880739225 DF On-Demand Anodyne PLAU 15 40 COc1ccc(-c2nc(C(=O)NC3CSC3)cs2)cc1OC ZINC000880739227 EF On-Demand Anodyne PPARD 15 41 COc1ccc(-c2nc(C(=O)NC3CSC3)cs2)cc1OC ZINC000880739227 EF On-Demand Anodyne STK17B 41 39 O=C(Cn1c(=O)nc(O)c2ccccc21)NC1CSC1 ZINC000880739235 CC On-Demand Anodyne TNKS 59 33 O=C(Cn1c(=O)ccn(Cc2ccccc2)c1=O)NC1CSC1 ZINC000880739248 EC On-Demand Anodyne SIGMAR1 19 45 O=C(Cc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739257 CE On-Demand Anodyne CSNK1D 29 49 O=C(Cc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739257 CE On-Demand Anodyne CCR2 106 44 O=C(Cc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739257 CE On-Demand Anodyne LUXR 28 47 O=C(Cc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739257 CE On-Demand Anodyne PDS 43 37 O=C(NC1CSC1)C1CCCC1 ZINC000880739263 AD On-Demand Anodyne EPHX2 16 42 O=C(CNC(=O)c1cccc(Cl)c1)NC1CSC1 ZINC000880739265 CD On-Demand Anodyne CCR2 69 49 O=C(CNC(=O)c1cccc(Cl)c1)NC1CSC1 ZINC000880739265 CD On-Demand Anodyne CACNA1I 42 44 CC(=O)N1CCc2ccccc2[C@@H]1CC(=O)NC1CSC1 ZINC000880739274 DD On-Demand Anodyne MTNR1B 15 55 O=C(Cn1c(S)nc2ccccc2c1=O)NC1CSC1 ZINC000880739278 DC On-Demand Anodyne TNKS 61 34 O=C(CNC(=O)c1ccccc1)NC1CSC1 ZINC000880739287 CC On-Demand Anodyne CTRB1 28 40 O=C(CNC(=O)c1ccccc1)NC1CSC1 ZINC000880739287 CC On-Demand Anodyne CCR2 61 45 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000880739293 ED On-Demand Anodyne EPHX2 20 59 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000880739293 ED On-Demand Anodyne AKR1C3 71 47 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000880739293 ED On-Demand Anodyne SFRP1 21 44 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000880739293 ED On-Demand Anodyne NAMPT 19 41 CCOc1ccc(C(=O)NCC(=O)NC2CSC2)cc1OCC ZINC000880739298 ED On-Demand Anodyne SSTR5 44 36 CCOc1ccc(C(=O)NCC(=O)NC2CSC2)cc1OCC ZINC000880739298 ED On-Demand Anodyne CCR2 60 40 O=C(CNC(=O)c1ccc2c(c1)OCO2)NC1CSC1 ZINC000880739299 CC On-Demand Anodyne CCR2 46 51 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne DRD4 58 44 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne MAPK11 24 42 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne MAPK14 17 46 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne MTNR1A 47 41 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne MTNR1B 40 41 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne MCHR1 16 53 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne LGALS3 15 40 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne TAAR1 32 42 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne AKR1C3 16 40 COc1cccc(C(=O)NC2CSC2)c1 ZINC000880739300 BD On-Demand Anodyne KCNK3 34 51 CC(=O)N1CCC[C@H](C(=O)NC2CSC2)C1 ZINC000880739307 BC On-Demand Anodyne EPHX2 21 46 O=C(CCc1nc(O)c2cnn(-c3ccccc3)c2n1)NC1CSC1 ZINC000880739312 FD On-Demand Anodyne TNKS 59 33 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000880739315 EC On-Demand Anodyne TGM2 29 40 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000880739315 EC On-Demand Anodyne AKR1C3 68 46 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000880739315 EC On-Demand Anodyne SFRP1 15 41 C[C@H]1CCC[C@H](C)N1C(=O)COc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739323 FF On-Demand Anodyne SLC6A5 37 43 O=C(CCn1c(S)nc2ccccc2c1=O)NC1CSC1 ZINC000880739326 DD On-Demand Anodyne TNKS 64 36 O=C(NC1CSC1)c1ccc(F)cc1Cl ZINC000880739329 BE On-Demand Anodyne P2RX7 34 42 O=C(NC1CSC1)c1ccc(F)cc1Cl ZINC000880739329 BE On-Demand Anodyne PYGL 16 46 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1 ZINC000880739331 GE On-Demand Anodyne CA7 17 44 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1 ZINC000880739331 GE On-Demand Anodyne EPHX2 42 55 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1 ZINC000880739331 GE On-Demand Anodyne AKR1C3 46 34 Cc1cc(C(=O)NC2CSC2)c(C)n1Cc1ccccc1 ZINC000880739339 DF On-Demand Anodyne DRD4 26 41 Cc1cc(C(=O)NC2CSC2)c(C)n1Cc1ccccc1 ZINC000880739339 DF On-Demand Anodyne CNR2 20 48 Cc1cc(C(=O)NC2CSC2)c(C)n1Cc1ccccc1 ZINC000880739339 DF On-Demand Anodyne SIGMAR1 19 42 Cc1cc(C(=O)NC2CSC2)c(C)n1Cc1ccccc1 ZINC000880739339 DF On-Demand Anodyne PLA2G2A 46 34 CC(=O)N1CCN(c2ccc(C(=O)NC3CSC3)cc2[N+](=O)[O-])CC1 ZINC000880739342 FD On-Demand Bother TAAR1 20 45 O=C(NC1CSC1)c1cccc(S(=O)(=O)NC2CC2)c1 ZINC000880739347 DC On-Demand Anodyne SFRP1 65 39 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000880739360 EC On-Demand Anodyne TGM2 56 52 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000880739360 EC On-Demand Anodyne MERTK 31 40 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000880739360 EC On-Demand Anodyne NAMPT 26 42 O=C(Cc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880739361 CF On-Demand Anodyne OPRK1 25 41 O=C(Cc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880739361 CF On-Demand Anodyne SIGMAR1 23 57 O=C(Cc1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880739361 CF On-Demand Anodyne LUXR 40 35 CCOC(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880739362 FG On-Demand Anodyne P2RY12 40 39 CCOC(=O)Nc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739366 CE On-Demand Anodyne MAPK14 15 41 CCOC(=O)Nc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739366 CE On-Demand Anodyne EPHX2 19 40 CCOC(=O)Nc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739366 CE On-Demand Anodyne ACR 44 33 O=C(CNC(=O)c1ccccc1OC(F)F)NC1CSC1 ZINC000880739371 DD On-Demand Anodyne HCN1 62 33 O=C(CNC(=O)c1ccccc1OC(F)F)NC1CSC1 ZINC000880739371 DD On-Demand Anodyne HCN4 46 30 Cc1nn(-c2ccccc2)c(C)c1CC(=O)NC1CSC1 ZINC000880739375 DE On-Demand Anodyne P2RX7 32 75 O=C(CCCNC(=O)c1ccccc1)NC1CSC1 ZINC000880739377 CD On-Demand Anodyne HDAC1 15 44 O=C(CCCNC(=O)c1ccccc1)NC1CSC1 ZINC000880739377 CD On-Demand Anodyne HDAC3 19 44 O=C(CCCNC(=O)c1ccccc1)NC1CSC1 ZINC000880739377 CD On-Demand Anodyne HDAC6 17 44 O=C(CCCNC(=O)c1ccccc1)NC1CSC1 ZINC000880739377 CD On-Demand Anodyne HDAC9 23 44 O=C(COc1ccc(Cl)cc1)NC1CSC1 ZINC000880739383 CD On-Demand Anodyne TRAR 36 57 O=C(Cc1ccc(Cl)cc1)NC1CSC1 ZINC000880739389 BE On-Demand Anodyne AVPR1A 35 46 O=C(Cc1ccc(Cl)cc1)NC1CSC1 ZINC000880739389 BE On-Demand Anodyne LUXR 35 40 CCN(CC)S(=O)(=O)c1ccc(C(=O)NCC(=O)NC2CSC2)cc1 ZINC000880739393 GC On-Demand Anodyne CA2 17 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne ACE 58 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne OPRM1 42 38 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne MME 124 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne ANPEP 79 37 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne FCER2 86 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CTSB 44 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne PAPA1_CARPA 47 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CYSP_TRYCR 63 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CTSK 19 48 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CTSL 50 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne NPFFR2 51 36 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne TIMP3 79 38 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CAPNS1 56 31 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne MMP3 17 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne ECE1 16 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne HLA-DRB1 51 32 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CTSS 24 45 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CAPN1 61 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne MMP9 20 58 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CAPN2 34 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne ACE2 69 37 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne CTSC 35 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne MMP7 17 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne MMP1 25 58 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne FPR1 53 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne BLA1_STEMA 66 35 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739396 EE On-Demand Anodyne NPFFR1 64 36 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne ACE 58 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne OPRM1 42 38 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne MME 124 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne ANPEP 79 37 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne FCER2 86 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CTSB 44 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne PAPA1_CARPA 47 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CYSP_TRYCR 63 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CTSK 19 48 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CTSL 50 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne NPFFR2 51 36 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne TIMP3 79 38 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CAPNS1 56 31 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne MMP3 17 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne ECE1 16 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne HLA-DRB1 51 32 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CTSS 24 45 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CAPN1 61 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne MMP9 20 58 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CAPN2 34 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne ACE2 69 37 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne CTSC 35 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne MMP7 17 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne MMP1 25 58 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne FPR1 53 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne BLA1_STEMA 66 35 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1cccs1 ZINC000880739397 EE On-Demand Anodyne NPFFR1 64 36 CC[C@H](C)NC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880739399 CH On-Demand Anodyne ANPEP 15 48 C[C@@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@@H](C)O1 ZINC000880739403 DH On-Demand Anodyne RBP4 55 35 C[C@H]1CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C[C@H](C)O1 ZINC000880739404 DH On-Demand Anodyne RBP4 55 35 O=C(CCc1ccc(S(=O)(=O)N2CCCCC2)cc1)NC1CSC1 ZINC000880739406 FE On-Demand Anodyne EPHX2 15 44 O=C(CCc1ccc(S(=O)(=O)N2CCCCC2)cc1)NC1CSC1 ZINC000880739406 FE On-Demand Anodyne TGM2 63 39 O=C(CCc1ccc(S(=O)(=O)N2CCCCC2)cc1)NC1CSC1 ZINC000880739406 FE On-Demand Anodyne F13A1 59 40 O=C(CCc1ccc(S(=O)(=O)N2CCCCC2)cc1)NC1CSC1 ZINC000880739406 FE On-Demand Anodyne NAMPT 39 43 O=C(CNC(=O)c1cccc(F)c1)NC1CSC1 ZINC000880739410 CC On-Demand Anodyne CCR2 89 48 COc1ccc(-c2nnc(S)n2CC(=O)NC2CSC2)cc1 ZINC000880739416 ED On-Demand Anodyne AVPR1B 33 40 O=C(CCc1nc(-c2ccc(Cl)cc2)no1)NC1CSC1 ZINC000880739419 DF On-Demand Anodyne HCAR2 22 45 O=C(NC1CSC1)c1ccc(OC(F)(F)F)cc1 ZINC000880739425 CE On-Demand Anodyne SLC6A5 33 40 O=C(NC1CSC1)c1ccc(OC(F)(F)F)cc1 ZINC000880739425 CE On-Demand Anodyne EPHX2 45 46 O=C(NC1CSC1)c1ccc(OC(F)(F)F)cc1 ZINC000880739425 CE On-Demand Anodyne GIPR 42 36 O=C(NC1CSC1)c1ccc(OC(F)(F)F)cc1 ZINC000880739425 CE On-Demand Anodyne SHH 48 45 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cn2)CC1 ZINC000880739428 EF On-Demand Anodyne EPHX2 27 45 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cn2)CC1 ZINC000880739428 EF On-Demand Anodyne PTGES 21 43 O=C(CCCCc1nc2ccccc2s1)NC1CSC1 ZINC000880739438 DG On-Demand Anodyne TNKS 46 32 CC(=O)N1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880739446 EF On-Demand Anodyne RBP4 53 37 COc1ccc(-c2nc(C(=O)NC3CSC3)cs2)cc1 ZINC000880739452 DF On-Demand Anodyne PDK1 40 34 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880739453 DI On-Demand Anodyne RBP4 69 41 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880739454 DI On-Demand Anodyne RBP4 69 41 O=C(COCc1nc2ccccc2s1)NC1CSC1 ZINC000880739457 CE On-Demand Anodyne LTA4H 20 40 CCOc1ccccc1C(=O)NCC(=O)NC1CSC1 ZINC000880739458 CD On-Demand Anodyne KCNA3 42 46 CCOc1ccccc1C(=O)NCC(=O)NC1CSC1 ZINC000880739458 CD On-Demand Anodyne HCN1 90 44 CCOc1ccccc1C(=O)NCC(=O)NC1CSC1 ZINC000880739458 CD On-Demand Anodyne HCN4 65 43 CCOc1ccccc1C(=O)NCC(=O)NC1CSC1 ZINC000880739458 CD On-Demand Anodyne KCNK3 34 44 CCOc1ccccc1C(=O)NCC(=O)NC1CSC1 ZINC000880739458 CD On-Demand Anodyne KCNK9 30 44 CCCCN(CC)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880739460 DJ On-Demand Anodyne SOAT1 19 42 O=C(CNC(=O)c1cccc(Br)c1)NC1CSC1 ZINC000880739465 ED On-Demand Anodyne CCR2 72 57 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne ACE 24 53 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne SSTR2 39 42 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne OPRM1 18 60 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne GHRHR 27 41 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MME 32 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne EDNRB 54 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne EDNRA 49 51 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne TACR1 39 57 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MC4R 58 51 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne CCKAR 134 48 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne CTSL 25 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne BRS3 32 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne TIMP3 28 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne NMBR 64 50 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MC3R 76 47 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MC5R 85 47 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP2 32 56 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP8 45 56 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP14 24 48 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne GRPR 99 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne ECE1 71 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne SSTR3 28 42 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP11 84 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne CCKBR 108 50 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne GHSR 72 58 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP9 31 56 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MC1R 111 51 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne C5AR1 42 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP7 19 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne MMP1 25 50 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne NPR 33 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne ADAM12 15 48 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne KISS1R 77 37 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne ERAP2 44 39 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne PSMB8 28 41 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CSC1 ZINC000880739478 DD On-Demand Anodyne HPN 23 46 Cc1nc2ccc(C(=O)NC3CSC3)cc2nc1C ZINC000880739480 CE On-Demand Anodyne MAPK14 40 38 CC(C)c1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880739482 CE On-Demand Anodyne TRAR 32 42 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne SIGMAR1 18 55 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP13 39 40 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne CSNK1D 15 45 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MTNR1A 54 38 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MTNR1B 40 38 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP3 46 40 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP8 26 40 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP9 42 38 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP12 17 40 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne CA9 20 45 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne MMP1 51 40 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne PROKR1 41 31 COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880739483 BD On-Demand Anodyne H9B8T9_CAPHI 18 40 O=C(Cc1ccc(Br)cc1)NC1CSC1 ZINC000880739484 CE On-Demand Anodyne LUXR 32 54 O=C(Cc1ccc(Br)cc1)NC1CSC1 ZINC000880739484 CE On-Demand Anodyne TRAR 31 50 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA2 134 54 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA6 23 44 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA1 113 48 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA7 85 46 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA13 30 44 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA5B 71 45 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA4 92 48 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA5A 76 45 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA14 78 46 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA12 89 46 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA9 95 50 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CAH_METTE 25 44 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CYNT 31 41 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne NCE103 28 54 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne CA15 15 44 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne MTCA1 38 40 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne P96878_MYCTU 50 41 NS(=O)(=O)c1ccc(CCC(=O)NC2CSC2)cc1 ZINC000880739489 DC On-Demand Anodyne A6YCJ1_9METZ 25 45 O=C(NC1CSC1)c1cc2cc(F)ccc2s1 ZINC000880739492 CF On-Demand Anodyne PIN1 22 40 C[C@@H]1CCCN(C(=O)Nc2cccc(F)c2C(C)(F)F)C1 ZINC000880739498 DI On-Demand Anodyne RBP4 57 39 CC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)NC3CSC3)cc2)CC1 ZINC000880739499 GC On-Demand Anodyne TGM2 84 46 CC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)NC3CSC3)cc2)CC1 ZINC000880739499 GC On-Demand Anodyne F13A1 72 39 O=C(CNC(=O)c1ccc(Br)cc1)NC1CSC1 ZINC000880739502 ED On-Demand Anodyne CCR2 40 42 COc1ccc(CN(C)C(=O)Nc2cccc(F)c2C(C)(F)F)cc1OC ZINC000880739509 GJ On-Demand Anodyne MT-ND1 20 46 CCOc1ccccc1OCC(=O)NC1CSC1 ZINC000880739513 CD On-Demand Anodyne HCN1 49 32 CCOc1ccccc1OCC(=O)NC1CSC1 ZINC000880739513 CD On-Demand Anodyne HCN4 42 32 O=C(Cc1ccccc1[N+](=O)[O-])NC1CSC1 ZINC000880739514 CD On-Demand Bother COLA 116 39 CCOc1ccc(C(=O)NCC(=O)NC2CSC2)cc1 ZINC000880739516 CD On-Demand Anodyne CCR2 41 38 CN(C)S(=O)(=O)c1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739517 FB On-Demand Anodyne CCR2 75 50 CCCCN(CCO)C(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880739518 DH On-Demand Anodyne SOAT1 21 41 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 ZINC000880739519 FE On-Demand Anodyne CNR1 15 59 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 ZINC000880739519 FE On-Demand Anodyne CNR2 20 80 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 ZINC000880739519 FE On-Demand Anodyne UTS2R 20 43 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 ZINC000880739519 FE On-Demand Anodyne EPHX2 28 45 O=C(NC1CSC1)c1ccccc1OCCOc1ccccc1 ZINC000880739521 EF On-Demand Anodyne CYSLTR2 19 44 O=C(NC1CSC1)c1ccccc1OCCOc1ccccc1 ZINC000880739521 EF On-Demand Anodyne KCNA3 44 36 O=C(NC1CSC1)c1ccccc1OCCOc1ccccc1 ZINC000880739521 EF On-Demand Anodyne HCN1 51 31 O=C(NC1CSC1)c1ccccc1OCCOc1ccccc1 ZINC000880739521 EF On-Demand Anodyne HCN4 40 30 CC(C)(C)OC(=O)N1CCC(C(=O)NC2CSC2)CC1 ZINC000880739523 DD On-Demand Anodyne EPHX2 20 53 CC(C)(C)OC(=O)N1CCC(C(=O)NC2CSC2)CC1 ZINC000880739523 DD On-Demand Anodyne GPR119 34 41 O=C(COc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739528 CE On-Demand Anodyne CCR2 77 41 O=C(COc1cccc(C(F)(F)F)c1)NC1CSC1 ZINC000880739528 CE On-Demand Anodyne PDS 49 45 COC(=O)c1cn(CC(=O)NC2CSC2)c2ccccc12 ZINC000880739540 DD On-Demand Anodyne CNR1 20 42 COC(=O)c1cn(CC(=O)NC2CSC2)c2ccccc12 ZINC000880739540 DD On-Demand Anodyne CNR2 32 42 O=C(Cc1ccc(Cl)cc1Cl)NC1CSC1 ZINC000880739541 CF On-Demand Anodyne P2RX7 47 44 O=C(Cc1ccc(Cl)cc1Cl)NC1CSC1 ZINC000880739541 CF On-Demand Anodyne EPHX2 18 43 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000880739545 ED On-Demand Anodyne EPHX2 19 53 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000880739545 ED On-Demand Anodyne TGM2 68 48 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000880739545 ED On-Demand Anodyne F13A1 53 44 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000880739545 ED On-Demand Anodyne NAMPT 31 45 O=C(CCc1nc2ccccc2o1)NC1CSC1 ZINC000880739547 CD On-Demand Anodyne FASN 17 41 O=C(CCc1nc2ccccc2o1)NC1CSC1 ZINC000880739547 CD On-Demand Anodyne TNKS 57 34 COc1cc(CNC(=O)/C=C\c2ccc(OC)c(OC)c2)on1 ZINC000880739552 DE On-Demand Anodyne TUBB1 41 36 COc1cc(CNC(=O)/C=C/c2ccc(OC)c(OC)c2)on1 ZINC000880739553 DE On-Demand Anodyne TUBB1 41 36 COc1cc(CNC(=O)CCn2c(S)nc3ccccc3c2=O)on1 ZINC000880739554 FD On-Demand Anodyne HTR7 18 41 O=C(CCSc1ccc(F)cc1)NC1CSC1 ZINC000880739559 CF On-Demand Anodyne TNKS 42 41 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP13 78 45 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne ADAM17 61 40 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP2 32 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP3 67 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP8 21 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP9 32 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne EPHX2 47 64 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne TGM2 53 39 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP7 66 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne MMP1 71 43 CCOc1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739561 GD On-Demand Anodyne F13A1 41 36 O=C(NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880739568 CF On-Demand Anodyne MAPK14 17 41 O=C(NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880739568 CF On-Demand Anodyne CCR2 92 49 O=C(NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880739568 CF On-Demand Anodyne AKR1C3 15 48 O=C(NC1CSC1)c1cccc(C(F)(F)F)c1 ZINC000880739568 CF On-Demand Anodyne KCNK3 20 51 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne FKBP1A 29 57 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP13 44 50 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne ITGA4 35 46 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne CAPNS1 23 48 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP2 19 45 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP3 49 50 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP8 28 42 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne CAPN1 19 50 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP9 28 41 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne EPHX2 23 55 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP7 52 50 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne MMP1 49 50 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne SFRP1 112 35 O=C(NC1CSC1)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739570 ED On-Demand Anodyne WNT3 82 35 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne FKBP1A 29 57 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP13 44 50 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne ITGA4 35 46 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne CAPNS1 23 48 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP2 19 45 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP3 49 50 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP8 28 42 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne CAPN1 19 50 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP9 28 41 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne EPHX2 23 55 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP7 52 50 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne MMP1 49 50 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne SFRP1 112 35 O=C(NC1CSC1)[C@H]1CCCCN1S(=O)(=O)c1ccccc1 ZINC000880739571 ED On-Demand Anodyne WNT3 82 35 COc1cc(CNC(=O)C2CCCCCCC2)on1 ZINC000880739577 CF On-Demand Anodyne STK17B 41 43 O=C(CCc1nc(O)c2ccccc2n1)NC1CSC1 ZINC000880739580 CD On-Demand Anodyne TNKS 85 45 O=C(CCc1nc(O)c2ccccc2n1)NC1CSC1 ZINC000880739580 CD On-Demand Anodyne TNKS2 26 45 O=C(NC1CSC1)C1(c2ccc(Cl)cc2)CC1 ZINC000880739583 CF On-Demand Anodyne AVPR1A 38 46 O=C(NC1CSC1)c1ccccc1Cl ZINC000880739586 BE On-Demand Anodyne ECR 47 41 O=C(NC1CSC1)c1ccccc1Cl ZINC000880739586 BE On-Demand Anodyne NR2E3 44 32 O=C(NC1CSC1)c1ccccc1Cl ZINC000880739586 BE On-Demand Anodyne SMO 18 44 CSCC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739588 FD On-Demand Anodyne MMP13 17 40 CSCC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739588 FD On-Demand Anodyne MMP2 25 42 CSCC[C@H](NS(=O)(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739589 FD On-Demand Anodyne MMP13 17 40 CSCC[C@H](NS(=O)(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739589 FD On-Demand Anodyne MMP2 25 42 O=C(Cc1cccs1)NC1CSC1 ZINC000880739590 BD On-Demand Anodyne CA5B 37 46 O=C(Cc1cccs1)NC1CSC1 ZINC000880739590 BD On-Demand Anodyne CA5A 36 46 O=C(Cc1cccs1)NC1CSC1 ZINC000880739590 BD On-Demand Anodyne SLC22A6 16 40 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CTSB 26 46 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CTSG 27 41 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CTSK 17 44 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CTSL 23 46 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CTRB1 41 45 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne CELA2A 24 45 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne ACE2 40 36 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739599 DE On-Demand Anodyne GAG-PRO 46 36 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CTSB 26 46 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CTSG 27 41 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CTSK 17 44 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CTSL 23 46 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CTRB1 41 45 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne CELA2A 24 45 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne ACE2 40 36 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739600 DE On-Demand Anodyne GAG-PRO 46 36 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CTSB 26 46 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CTSG 27 41 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CTSK 17 44 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CTSL 23 46 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CTRB1 41 45 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne CELA2A 24 45 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne ACE2 40 36 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739601 DE On-Demand Anodyne GAG-PRO 46 36 O=C(NC1CSC1)c1ccc(C(F)(F)F)cc1 ZINC000880739605 CF On-Demand Anodyne TRPV1 18 45 O=C(NC1CSC1)c1ccc(C(F)(F)F)cc1 ZINC000880739605 CF On-Demand Anodyne SLC6A5 35 44 O=C(NC1CSC1)c1ccccc1C(F)(F)F ZINC000880739607 CF On-Demand Anodyne RBP4 75 36 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880739608 FE On-Demand Anodyne AKR1C3 64 46 C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880739609 FE On-Demand Anodyne AKR1C3 64 46 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 ZINC000880739617 GE On-Demand Anodyne TRY2_BOVIN 55 38 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 ZINC000880739617 GE On-Demand Anodyne EPHX2 44 57 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 ZINC000880739617 GE On-Demand Anodyne PKM 18 45 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 ZINC000880739617 GE On-Demand Anodyne TGM2 47 43 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 ZINC000880739617 GE On-Demand Anodyne AKR1C3 18 60 COc1cc(CNC(=O)CC2C[C@@H]3CC[C@H](C2)N3C(=O)OC(C)(C)C)on1 ZINC000880739622 GF On-Demand Anodyne GPR119 15 40 O=C(CCc1ccc(-c2ccccc2)o1)NC1CSC1 ZINC000880739625 CG On-Demand Anodyne CYP2E1 17 40 O=C(NC1CSC1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880739628 CD On-Demand Anodyne INHA 23 52 COc1ccccc1N1C[C@@H](C(=O)NC2CSC2)CC1=O ZINC000880739631 DD On-Demand Anodyne HTR1A 46 42 COc1ccccc1N1C[C@@H](C(=O)NC2CSC2)CC1=O ZINC000880739631 DD On-Demand Anodyne DRD2 28 41 COc1ccccc1N1C[C@H](C(=O)NC2CSC2)CC1=O ZINC000880739632 DD On-Demand Anodyne HTR1A 46 42 COc1ccccc1N1C[C@H](C(=O)NC2CSC2)CC1=O ZINC000880739632 DD On-Demand Anodyne DRD2 28 41 O=C(NC1CSC1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880739633 CD On-Demand Anodyne INHA 23 52 CCCCCCn1nc(C(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739645 EF On-Demand Anodyne CNR1 15 40 CCCCCCn1nc(C(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739645 EF On-Demand Anodyne HTR3A 21 44 CCCCCCn1nc(C(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739645 EF On-Demand Anodyne CNR2 37 44 COc1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739646 CC On-Demand Anodyne DRD4 57 44 COc1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739646 CC On-Demand Anodyne MTNR1A 56 41 COc1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739646 CC On-Demand Anodyne MTNR1B 48 41 COc1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739646 CC On-Demand Anodyne CCR2 72 51 COc1cccc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739646 CC On-Demand Anodyne KCNK3 15 44 CCN(CC)S(=O)(=O)c1cc(C(=O)NC2CSC2)ccc1OC ZINC000880739650 FD On-Demand Anodyne CPT1A 63 36 CCN(CC)S(=O)(=O)c1cc(C(=O)NC2CSC2)ccc1OC ZINC000880739650 FD On-Demand Anodyne CPT1B 65 35 O=C(Cc1nnc(O)c2ccccc12)NC1CSC1 ZINC000880739651 CD On-Demand Anodyne TNKS 47 32 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880739662 FD On-Demand Anodyne CNR2 17 78 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880739662 FD On-Demand Anodyne UTS2R 20 43 O=C(NC1CSC1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880739662 FD On-Demand Anodyne EPHX2 27 43 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne ACE 79 49 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne OPRM1 41 38 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne MME 156 42 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne ANPEP 74 37 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTRA_BOVIN 15 53 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne FCER2 93 37 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTSB 63 51 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne PAPA1_CARPA 60 57 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CYSP_TRYCR 68 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTSK 28 51 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTSL 67 57 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CPA1 44 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne NPFFR2 54 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne TIMP3 83 41 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTRB1 47 49 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CAPNS1 65 32 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne MMP2 16 50 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne HLA-DRB1 50 32 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTSS 40 57 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CAPN1 69 45 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne MMP9 25 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CAPN2 39 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne ACE2 72 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTSV 42 47 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne PIN1 31 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne MMP1 30 46 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne FPR1 67 39 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne CTRB_BOVIN 47 35 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne BLA1_STEMA 78 40 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne KISS1R 47 33 O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739665 EE On-Demand Anodyne NPFFR1 68 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne ACE 79 49 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne OPRM1 41 38 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne MME 156 42 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne ANPEP 74 37 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTRA_BOVIN 15 53 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne FCER2 93 37 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTSB 63 51 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne PAPA1_CARPA 60 57 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CYSP_TRYCR 68 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTSK 28 51 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTSL 67 57 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CPA1 44 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne NPFFR2 54 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne TIMP3 83 41 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTRB1 47 49 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CAPNS1 65 32 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne MMP2 16 50 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne HLA-DRB1 50 32 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTSS 40 57 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CAPN1 69 45 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne MMP9 25 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CAPN2 39 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne ACE2 72 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTSV 42 47 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne PIN1 31 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne MMP1 30 46 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne FPR1 67 39 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne CTRB_BOVIN 47 35 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne BLA1_STEMA 78 40 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne KISS1R 47 33 O=C(N[C@H](Cc1ccccc1)C(=O)NC1CSC1)c1ccccc1 ZINC000880739666 EE On-Demand Anodyne NPFFR1 68 46 Cc1sc2ncnc(N3CCC(C(=O)NC4CSC4)CC3)c2c1C ZINC000880739670 FF On-Demand Anodyne SIRT3 57 36 Cc1sc2ncnc(N3CCC(C(=O)NC4CSC4)CC3)c2c1C ZINC000880739670 FF On-Demand Anodyne SIRT2 47 32 Cc1sc2ncnc(N3CCC(C(=O)NC4CSC4)CC3)c2c1C ZINC000880739670 FF On-Demand Anodyne SIRT1 45 32 O=C(NC1CSC1)c1ccc2c(c1)OCO2 ZINC000880739672 BD On-Demand Anodyne MCHR1 17 45 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCCC2)cc1 ZINC000880739681 FE On-Demand Anodyne EPHX2 19 53 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCCC2)cc1 ZINC000880739681 FE On-Demand Anodyne TGM2 68 48 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCCC2)cc1 ZINC000880739681 FE On-Demand Anodyne F13A1 53 44 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCCCC2)cc1 ZINC000880739681 FE On-Demand Anodyne NAMPT 31 45 O=C(NC1CSC1)c1cccc(Cl)c1Cl ZINC000880739682 CF On-Demand Anodyne ECR 25 43 CCOc1ccc(C(=O)NC2CSC2)cc1OCC ZINC000880739685 CE On-Demand Anodyne DRD4 15 40 CCOc1ccc(C(=O)NC2CSC2)cc1OCC ZINC000880739685 CE On-Demand Anodyne SSTR5 56 44 CCOc1ccc(C(=O)NC2CSC2)cc1OCC ZINC000880739685 CE On-Demand Anodyne EZH2 40 36 Cc1cc(C)cc(C(=O)NCC(=O)NC2CSC2)c1 ZINC000880739686 CD On-Demand Anodyne CCR2 44 39 Cc1nn(-c2ccc(F)cc2)c(C)c1C(=O)NC1CSC1 ZINC000880739689 DE On-Demand Anodyne MAPK14 15 45 CCOc1ccc(SCC(=O)NC2CSC2)cc1 ZINC000880739691 CE On-Demand Anodyne FAS 42 39 O=C(NC1CSC1)c1cccc(F)c1 ZINC000880739696 BD On-Demand Anodyne GRM5 15 67 O=C(NC1CSC1)c1cccc(F)c1 ZINC000880739696 BD On-Demand Anodyne KCNK3 27 48 O=C(NC1CSC1)c1cccc(F)c1 ZINC000880739696 BD On-Demand Anodyne KCNK9 15 44 O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)NC1CSC1 ZINC000880739700 DD On-Demand Anodyne CCR2 55 41 Cc1cc(C(=O)NC2CSC2)c2ccccc2n1 ZINC000880739701 CE On-Demand Anodyne ADAM17 83 42 CCOc1ccccc1C(=O)NC1CSC1 ZINC000880739703 BD On-Demand Anodyne KCNA3 41 45 CCOc1ccccc1C(=O)NC1CSC1 ZINC000880739703 BD On-Demand Anodyne HCN1 84 44 CCOc1ccccc1C(=O)NC1CSC1 ZINC000880739703 BD On-Demand Anodyne HCN4 64 43 CCOc1ccccc1C(=O)NC1CSC1 ZINC000880739703 BD On-Demand Anodyne KCNK3 55 49 CCOc1ccccc1C(=O)NC1CSC1 ZINC000880739703 BD On-Demand Anodyne KCNK9 46 49 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne SSTR5 42 37 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne PLA2G4B 62 37 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne SLC6A5 39 46 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne PLAU 22 40 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne ST14 18 40 CCOc1ccc(C(=O)NC2CSC2)cc1 ZINC000880739704 BD On-Demand Anodyne AOC3 15 47 O=C(NC1CSC1)[C@@H]1CCCN(S(=O)(=O)c2ccc(F)cc2)C1 ZINC000880739711 FD On-Demand Anodyne EPHX2 22 48 O=C(NC1CSC1)[C@H]1CCCN(S(=O)(=O)c2ccc(F)cc2)C1 ZINC000880739712 FD On-Demand Anodyne EPHX2 22 48 Cn1nc(CC(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739717 CC On-Demand Anodyne INHA 42 32 Cn1nc(CC(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739717 CC On-Demand Anodyne AKR1B1 40 37 Cn1nc(CC(=O)NC2CSC2)c2ccccc2c1=O ZINC000880739717 CC On-Demand Anodyne IMDH_CRYPV 40 58 O=C(CCc1ccc2ccccc2n1)NC1CSC1 ZINC000880739723 CE On-Demand Anodyne TNKS 58 33 O=C(COc1ccccc1)NC1CSC1 ZINC000880739724 BD On-Demand Anodyne CPT1A 49 34 O=C(COc1ccccc1)NC1CSC1 ZINC000880739724 BD On-Demand Anodyne TRAR 38 40 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000880739726 FE On-Demand Anodyne EPHX2 20 59 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000880739726 FE On-Demand Anodyne AKR1C3 71 47 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000880739726 FE On-Demand Anodyne SFRP1 21 44 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCCCCC2)c1 ZINC000880739726 FE On-Demand Anodyne NAMPT 19 41 O=C(NC1CSC1)c1cc(C2CC2)nc2ccccc12 ZINC000880739727 CF On-Demand Anodyne TACR3 21 50 O=C(NC1CSC1)c1cc(C2CC2)nc2ccccc12 ZINC000880739727 CF On-Demand Anodyne TNKS 59 35 CC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739730 CD On-Demand Anodyne MAPK14 21 40 CC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739730 CD On-Demand Anodyne EPHX2 18 44 CC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739730 CD On-Demand Anodyne AKR1C3 20 44 CC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739730 CD On-Demand Anodyne KCNK3 116 44 CC(=O)Nc1cccc(C(=O)NC2CSC2)c1 ZINC000880739730 CD On-Demand Anodyne KCNK9 71 44 O=C(Cc1ccc(F)cc1)NC1CSC1 ZINC000880739733 BD On-Demand Anodyne SIGMAR1 16 52 COc1ccc(CC(=O)NC2CSC2)cc1OC ZINC000880739734 CD On-Demand Anodyne HCRTR1 19 44 COc1ccc(CC(=O)NC2CSC2)cc1OC ZINC000880739734 CD On-Demand Anodyne ENPP1 54 30 C[C@H]1CN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)C[C@H](C)O1 ZINC000880739739 FD On-Demand Anodyne AKR1C3 62 42 C[C@H]1CN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)C[C@@H](C)O1 ZINC000880739740 FD On-Demand Anodyne AKR1C3 62 42 C[C@@H]1CN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)C[C@@H](C)O1 ZINC000880739741 FD On-Demand Anodyne AKR1C3 62 42 CCCCNC(=O)Nc1cccc(F)c1C(C)(F)F ZINC000880739745 CH On-Demand Anodyne ASAH1 61 33 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)CC1 ZINC000880739755 GC On-Demand Anodyne EPHX2 15 48 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)CC1 ZINC000880739755 GC On-Demand Anodyne TGM2 59 37 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)CC1 ZINC000880739755 GC On-Demand Anodyne F13A1 48 36 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)CC1 ZINC000880739755 GC On-Demand Anodyne AKR1C3 68 45 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)NC3CSC3)c2)CC1 ZINC000880739755 GC On-Demand Anodyne SFRP1 17 40 O=C(COc1ccc([N+](=O)[O-])cc1)NC1CSC1 ZINC000880739765 CD On-Demand Bother TRAR 41 60 O=C(COc1cccc(Br)c1)NC1CSC1 ZINC000880739767 DE On-Demand Anodyne TRAR 29 41 O=C(COc1cccc(Cl)c1)NC1CSC1 ZINC000880739772 CD On-Demand Anodyne MAOB 16 47 O=C(COc1cccc(Cl)c1)NC1CSC1 ZINC000880739772 CD On-Demand Anodyne PTPN22 19 40 O=C(COc1cccc(Cl)c1)NC1CSC1 ZINC000880739772 CD On-Demand Anodyne TRAR 29 41 COc1cc(CNC(=O)C2CCN(C(=O)OCC(C)C)CC2)on1 ZINC000880739773 ED On-Demand Anodyne SLC5A7 27 40 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1 ZINC000880739775 GD On-Demand Anodyne EPHX2 41 79 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1 ZINC000880739775 GD On-Demand Anodyne PKM 48 56 O=C(CCCOc1ccccc1)NC1CSC1 ZINC000880739780 CE On-Demand Anodyne LTA4H 33 41 O=C(CCCOc1ccccc1)NC1CSC1 ZINC000880739780 CE On-Demand Anodyne CYSLTR2 67 35 O=C(CCCOc1ccccc1)NC1CSC1 ZINC000880739780 CE On-Demand Anodyne PLA2G4B 70 36 O=C(CCCOc1ccccc1)NC1CSC1 ZINC000880739780 CE On-Demand Anodyne TNKS 54 33 O=C(Cc1ccc2ccccc2c1)NC1CSC1 ZINC000880739782 CF On-Demand Anodyne SIGMAR1 15 59 O=C(Cc1ccc2ccccc2c1)NC1CSC1 ZINC000880739782 CF On-Demand Anodyne CCR3 23 46 O=C(Cc1ccc2ccccc2c1)NC1CSC1 ZINC000880739782 CF On-Demand Anodyne LUXR 39 56 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739796 GE On-Demand Anodyne EPHX2 47 78 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739796 GE On-Demand Anodyne TGM2 52 38 O=C(NC1CSC1)c1cc2ccccc2s1 ZINC000880739802 BF On-Demand Anodyne PIN1 29 42 CN(C)S(=O)(=O)c1cccc(C(=O)NC2CSC2)c1 ZINC000880739812 DC On-Demand Anodyne AKR1C3 45 35 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880739820 GD On-Demand Anodyne TGM2 31 40 O=C(CCc1nc2ccccc2n1-c1ccccc1)NC1CSC1 ZINC000880739824 EG On-Demand Anodyne TNKS 57 32 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880739832 ED On-Demand Anodyne EPHX2 50 75 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880739832 ED On-Demand Anodyne TGM2 69 44 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880739832 ED On-Demand Anodyne F13A1 62 39 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880739832 ED On-Demand Anodyne AKR1C3 42 36 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880739832 ED On-Demand Anodyne SFRP1 61 43 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1 ZINC000880739836 CD On-Demand Anodyne DRD4 30 47 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1 ZINC000880739836 CD On-Demand Anodyne ACHE 18 41 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1 ZINC000880739836 CD On-Demand Anodyne SIGMAR1 21 45 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1 ZINC000880739836 CD On-Demand Anodyne ITK 15 44 O=C(NC1CSC1)c1cnn(Cc2ccccc2)c1 ZINC000880739836 CD On-Demand Anodyne PANC 48 39 C[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739837 CD On-Demand Anodyne CTSB 17 46 C[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739837 CD On-Demand Anodyne CTRB1 40 37 C[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739839 CD On-Demand Anodyne CTSB 17 46 C[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880739839 CD On-Demand Anodyne CTRB1 40 37 O=C(Cc1ccccc1Cl)NC1CSC1 ZINC000880739843 BE On-Demand Anodyne P2RX7 20 40 COc1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880739850 CE On-Demand Anodyne MMP13 19 40 COc1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880739850 CE On-Demand Anodyne PLA2G4B 64 37 O=C(COc1ccc(Br)cc1)NC1CSC1 ZINC000880739852 DE On-Demand Anodyne TRAR 48 57 Cc1cc(C)c(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)c(C)c1 ZINC000880739864 GE On-Demand Anodyne EPHX2 52 78 O=C(Cc1ccc2c(c1)OCCO2)NC1CSC1 ZINC000880739865 CD On-Demand Anodyne MCHR1 17 48 O=C(Cc1ccc2c(c1)OCCO2)NC1CSC1 ZINC000880739865 CD On-Demand Anodyne LUXR 58 45 CCOc1ccc(C(=O)CCC(=O)NC2CSC2)cc1OCC ZINC000880739866 EF On-Demand Anodyne SSTR5 43 35 O=C(NC1CSC1)c1cc(Cl)cc(Cl)c1 ZINC000880739868 CF On-Demand Anodyne CACNA1H 18 45 O=C(NC1CSC1)c1cc(Cl)cc(Cl)c1 ZINC000880739868 CF On-Demand Anodyne CACNA1I 57 37 COc1ccc(-c2nc(C)c(C(=O)NC3CSC3)s2)cc1 ZINC000880739869 DF On-Demand Anodyne PPARA 15 55 O=C(CCc1cccnc1)NC1CSC1 ZINC000880739877 BD On-Demand Anodyne TBXAS1 52 49 O=C(CCc1cccnc1)NC1CSC1 ZINC000880739877 BD On-Demand Anodyne CHRNA7 47 38 O=C(CCc1cccnc1)NC1CSC1 ZINC000880739877 BD On-Demand Anodyne C3AR1 44 47 O=C(CCc1cccnc1)NC1CSC1 ZINC000880739877 BD On-Demand Anodyne NAMPT 33 47 Cc1cc(C)cc(C(=O)NC2CSC2)c1 ZINC000880739881 BE On-Demand Anodyne MAPK13 40 30 O=C(NC1CSC1)c1cccc(OC(F)F)c1 ZINC000880739885 CE On-Demand Anodyne DRD4 41 31 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880739887 ED On-Demand Anodyne EPHX2 17 51 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880739887 ED On-Demand Anodyne TGM2 69 49 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880739887 ED On-Demand Anodyne F13A1 54 45 O=C(NC1CSC1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000880739887 ED On-Demand Anodyne NAMPT 33 43 CCOC(=O)N1CCC(C(=O)NCc2cc(OC)no2)CC1 ZINC000880739896 DD On-Demand Anodyne SLC5A7 31 40 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880739897 FE On-Demand Anodyne CPT1A 21 44 O=C(NC1CSC1)c1cccc(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880739897 FE On-Demand Anodyne AKR1C3 69 48 O=C(NC1CSC1)c1cc(Cl)ccc1Cl ZINC000880739908 CF On-Demand Anodyne CNR1 15 43 O=C(NC1CSC1)c1ccc(Cl)s1 ZINC000880739909 BE On-Demand Anodyne F10 18 42 CN1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880739910 DF On-Demand Anodyne RBP4 52 37 O=C(CCc1ccc(S(=O)(=O)N2CCOCC2)cc1)NC1CSC1 ZINC000880739920 FC On-Demand Anodyne TGM2 56 39 O=C(CCc1ccc(S(=O)(=O)N2CCOCC2)cc1)NC1CSC1 ZINC000880739920 FC On-Demand Anodyne F13A1 48 37 O=C(CCc1ccc(S(=O)(=O)N2CCOCC2)cc1)NC1CSC1 ZINC000880739920 FC On-Demand Anodyne NAMPT 37 43 COc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880739921 CD On-Demand Anodyne TRAR 34 41 O=C(CCc1nc2ccccc2[nH]1)NC1CSC1 ZINC000880739929 CD On-Demand Anodyne PARP3 24 42 O=C(CCc1nc2ccccc2[nH]1)NC1CSC1 ZINC000880739929 CD On-Demand Anodyne TNKS 60 35 CCOC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880739930 FH On-Demand Anodyne EPHX2 22 41 CCOC(=O)C1CCN(C(=O)Nc2cccc(F)c2C(C)(F)F)CC1 ZINC000880739930 FH On-Demand Anodyne CCR8 38 41 CCOc1ccccc1OCCCC(=O)NC1CSC1 ZINC000880739940 CE On-Demand Anodyne HCN1 47 31 CCOc1ccccc1OCCCC(=O)NC1CSC1 ZINC000880739940 CE On-Demand Anodyne HCN4 40 30 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000880739947 GF On-Demand Anodyne EPHX2 27 75 O=C(NC1CSC1)C1CCN(C(=O)c2ccc(Br)cc2)CC1 ZINC000880739947 GF On-Demand Anodyne L3MBTL3 89 43 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1 ZINC000880739954 GD On-Demand Anodyne CA7 17 44 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1 ZINC000880739954 GD On-Demand Anodyne EPHX2 42 55 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1 ZINC000880739954 GD On-Demand Anodyne AKR1C3 46 34 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne DRD2 28 54 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne DRD4 17 41 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne DRD3 15 56 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne KDR 26 43 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne KCNK3 34 40 COc1cccc(C(=O)NC2CSC2)c1OC ZINC000880739965 CD On-Demand Anodyne KCNK9 25 40 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl ZINC000880739966 FE On-Demand Anodyne CNR2 15 52 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl ZINC000880739966 FE On-Demand Anodyne EPHX2 20 42 O=C(NC1CSC1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl ZINC000880739966 FE On-Demand Anodyne TGM2 40 36 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2cc(F)ccc2F)CC1 ZINC000880739967 GD On-Demand Anodyne EPHX2 47 61 COc1cc(CNC(=O)C[C@H](C)[C@H]2CCCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880739972 GF On-Demand Anodyne GPR119 21 42 COc1cc(CNC(=O)C[C@@H](C)[C@H]2CCCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880739973 GF On-Demand Anodyne GPR119 21 42 COc1cc(CNC(=O)C[C@H](C)[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880739974 GF On-Demand Anodyne GPR119 21 42 COc1cc(CNC(=O)C[C@@H](C)[C@@H]2CCCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880739975 GF On-Demand Anodyne GPR119 21 42 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739976 GD On-Demand Anodyne EPHX2 45 77 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739976 GD On-Demand Anodyne TGM2 55 41 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)NC3CSC3)CC2)cc1 ZINC000880739976 GD On-Demand Anodyne F13A1 41 35 O=C(Cc1cccc2ccccc12)NC1CSC1 ZINC000880739978 CF On-Demand Anodyne TNKS 40 30 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne FKBP1A 19 40 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne GRIN2B 30 46 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne PREP 28 41 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne EPHX2 21 42 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne TGM2 32 40 COc1cc(CNC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880739982 FE On-Demand Anodyne F13A1 32 40 C[C@H]1CN(S(=O)(=O)c2ccc(C(=O)NC3CSC3)cc2)C[C@H](C)O1 ZINC000880739983 FD On-Demand Anodyne TGM2 30 41 C[C@H]1CN(S(=O)(=O)c2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880739984 FD On-Demand Anodyne TGM2 30 41 C[C@@H]1CN(S(=O)(=O)c2ccc(C(=O)NC3CSC3)cc2)C[C@@H](C)O1 ZINC000880739985 FD On-Demand Anodyne TGM2 30 41 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NC3CSC3)ccc21 ZINC000880740003 DC On-Demand Anodyne PLD1 53 32 O=C(COc1ccc(I)cc1)NC1CSC1 ZINC000880740014 ED On-Demand Anodyne TRAR 36 57 O=C(NC1CSC1)c1cccc(NC(=O)C2CC2)c1 ZINC000880740016 CD On-Demand Anodyne TYK2 52 40 O=C(NC1CSC1)c1cccc(NC(=O)C2CC2)c1 ZINC000880740016 CD On-Demand Anodyne KCNK3 98 52 O=C(NC1CSC1)c1cccc(NC(=O)C2CC2)c1 ZINC000880740016 CD On-Demand Anodyne KCNK9 51 38 C=CCc1cc(C(=O)NCc2cc(OC)no2)cc(OC)c1OC ZINC000880740017 EE On-Demand Mild SLC5A7 23 40 O=C(C[C@H](NC(=O)c1ccccc1)c1ccccc1)NC1CSC1 ZINC000880740020 EF On-Demand Anodyne UTS2 58 36 O=C(C[C@@H](NC(=O)c1ccccc1)c1ccccc1)NC1CSC1 ZINC000880740021 EF On-Demand Anodyne UTS2 58 36 Cc1nn(-c2ccccc2)c(C)c1C(=O)NC1CSC1 ZINC000880740037 CE On-Demand Anodyne FPR1 19 52 O=C(CCCc1cccs1)NC1CSC1 ZINC000880740038 BE On-Demand Anodyne PTPRF 20 46 O=C(NC1CSC1)c1cc([N+](=O)[O-])ccc1N1CCCCC1 ZINC000880740044 DE On-Demand Bother WDR5 35 40 CCOc1ccc(C(=O)NC2CSC2)cc1OC ZINC000880740056 CD On-Demand Anodyne DRD4 15 40 CCOc1ccc(C(=O)NC2CSC2)cc1OC ZINC000880740056 CD On-Demand Anodyne SSTR5 51 40 COc1ccc(CC(=O)NC2CSC2)cc1S(=O)(=O)N1CCOCC1 ZINC000880740061 GC On-Demand Anodyne CPT1A 49 37 COc1ccc(CC(=O)NC2CSC2)cc1S(=O)(=O)N1CCOCC1 ZINC000880740061 GC On-Demand Anodyne CPT1B 56 36 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740063 DD On-Demand Anodyne CTSK 17 43 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740063 DD On-Demand Anodyne CTSL 15 40 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740063 DD On-Demand Anodyne CTSS 18 40 CSCC[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740064 DD On-Demand Anodyne CTSK 17 43 CSCC[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740064 DD On-Demand Anodyne CTSL 15 40 CSCC[C@H](NC(=O)c1ccccc1)C(=O)NC1CSC1 ZINC000880740064 DD On-Demand Anodyne CTSS 18 40 O=C(COc1ccc2ccc(=O)oc2c1)NC1CSC1 ZINC000880740065 CD On-Demand Anodyne MAOA 46 44 O=C(COc1ccc2ccc(=O)oc2c1)NC1CSC1 ZINC000880740065 CD On-Demand Anodyne MAOB 25 47 O=C(COc1ccc2ccc(=O)oc2c1)NC1CSC1 ZINC000880740065 CD On-Demand Anodyne TRAR 33 40 CCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740066 CF On-Demand Mild MTNR1A 26 40 CCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740066 CF On-Demand Mild SOAT1 18 41 CCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740066 CF On-Demand Mild NOD1 46 33 O=C(NC1CSC1)c1cccc([N+](=O)[O-])c1 ZINC000880740067 BD On-Demand Bother CACNA1C 50 36 O=C(NC1CSC1)c1cccc([N+](=O)[O-])c1 ZINC000880740067 BD On-Demand Bother CACNA1D 78 34 O=C(NC1CSC1)c1cccc([N+](=O)[O-])c1 ZINC000880740067 BD On-Demand Bother AKR1C3 15 41 CCCOc1ccc(C(=O)NC2CSC2)cc1OCC ZINC000880740071 CF On-Demand Anodyne SSTR5 50 41 O=C(CNS(=O)(=O)c1ccc(Cl)cc1)NC1CSC1 ZINC000880740072 DC On-Demand Anodyne TBXA2R 52 38 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne GRIN2B 20 57 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne SIGMAR1 19 48 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne NAAA 36 55 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne VIPR1 21 40 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne FFAR1 22 40 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne LUXR 42 38 O=C(CCc1ccccc1)NC1CSC1 ZINC000880740076 BD On-Demand Anodyne TNKS 40 31 CCCOc1c(Cl)cc(C(=O)NC2CSC2)cc1OC ZINC000880740080 DF On-Demand Anodyne LPAR2 35 44 CCCOc1c(Cl)cc(C(=O)NC2CSC2)cc1OC ZINC000880740080 DF On-Demand Anodyne S1PR2 33 44 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cc2[N+](=O)[O-])CC1 ZINC000880740082 GG On-Demand Bother SERPINE1 20 48 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cc2[N+](=O)[O-])CC1 ZINC000880740082 GG On-Demand Bother EPHX2 22 43 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cc2[N+](=O)[O-])CC1 ZINC000880740082 GG On-Demand Bother LIPG 49 34 O=C(NC1CSC1)C1CCN(c2ccc(C(F)(F)F)cc2[N+](=O)[O-])CC1 ZINC000880740082 GG On-Demand Bother PTGES 20 42 O=C(NC1CSC1)C1CCN(c2ncc(C(F)(F)F)cc2Cl)CC1 ZINC000880740087 GG On-Demand Anodyne MPL 33 41 O=C(NC1CSC1)C1CCN(c2ncc(C(F)(F)F)cc2Cl)CC1 ZINC000880740087 GG On-Demand Anodyne EPHX2 25 45 O=C(NC1CSC1)C1CCN(c2ncc(C(F)(F)F)cc2Cl)CC1 ZINC000880740087 GG On-Demand Anodyne PTGES 30 41 O=C(CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880740093 FD On-Demand Anodyne MMP13 23 43 O=C(CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880740093 FD On-Demand Anodyne MMP2 27 43 O=C(CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880740093 FD On-Demand Anodyne MMP14 24 45 O=C(CNS(=O)(=O)c1ccc(OC(F)(F)F)cc1)NC1CSC1 ZINC000880740093 FD On-Demand Anodyne EPHX2 34 40 NC(=O)NCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880740095 CC On-Demand Anodyne SSTR3 24 42 NC(=O)NCc1ccc(C(=O)NC2CSC2)cc1 ZINC000880740095 CC On-Demand Anodyne TPSAB1 16 40 CC1CCN(c2ccc([N+](=O)[O-])cc2C(=O)NC2CSC2)CC1 ZINC000880740103 EF On-Demand Bother WDR5 35 40 O=C(Cc1cccc(F)c1)NC1CSC1 ZINC000880740110 BD On-Demand Anodyne SIGMAR1 17 59 O=C(Cc1cccc(F)c1)NC1CSC1 ZINC000880740110 BD On-Demand Anodyne HAO2 27 42 O=C(COc1ccc(Cl)cc1Cl)NC1CSC1 ZINC000880740120 CF On-Demand Anodyne MCHR2 21 41 O=C(COc1ccc(Cl)cc1Cl)NC1CSC1 ZINC000880740120 CF On-Demand Anodyne PTGDR2 33 40 O=C(COc1ccc(Cl)cc1Cl)NC1CSC1 ZINC000880740120 CF On-Demand Anodyne TRAR 27 41 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)NC1CSC1 ZINC000880740131 DF On-Demand Anodyne FPR1 17 48 COc1ccc(-c2nc(CC(=O)NC3CSC3)cs2)cc1OC ZINC000880740132 FF On-Demand Anodyne DCK 25 42 COc1ccc(-c2nc(CC(=O)NC3CSC3)cs2)cc1OC ZINC000880740132 FF On-Demand Anodyne PPARD 19 44 COc1ccc(-c2nc(CC(=O)NC3CSC3)cs2)cc1OC ZINC000880740132 FF On-Demand Anodyne ENPP1 48 30 CCCOc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880740134 CE On-Demand Anodyne MMP13 20 41 CCCOc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880740134 CE On-Demand Anodyne PLA2G4B 90 39 CCCOc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880740134 CE On-Demand Anodyne TRAR 33 40 O=C(NC1CSC1)c1ccc(Cl)cc1Cl ZINC000880740143 CF On-Demand Anodyne CNR1 18 46 O=C(NC1CSC1)c1ccc(Cl)cc1Cl ZINC000880740143 CF On-Demand Anodyne P2RX7 17 40 O=C(NC1CSC1)c1ccc(Cl)cc1Cl ZINC000880740143 CF On-Demand Anodyne PYGL 17 45 O=C(NC1CSC1)c1ccc(Cl)cc1Cl ZINC000880740143 CF On-Demand Anodyne SLC6A9 46 36 COc1cc(CNC(=O)/C=C(\C)c2ccccc2OC)on1 ZINC000880740147 DE On-Demand Anodyne KCNA3 40 37 COc1cc(CNC(=O)/C=C(\C)c2ccccc2OC)on1 ZINC000880740147 DE On-Demand Anodyne ALS 44 33 COc1cc(CNC(=O)/C=C(\C)c2ccccc2OC)on1 ZINC000880740147 DE On-Demand Anodyne MT-CYB 49 36 COc1cc(CNC(=O)/C=C(/C)c2ccccc2OC)on1 ZINC000880740148 DE On-Demand Anodyne KCNA3 40 37 COc1cc(CNC(=O)/C=C(/C)c2ccccc2OC)on1 ZINC000880740148 DE On-Demand Anodyne ALS 44 33 COc1cc(CNC(=O)/C=C(/C)c2ccccc2OC)on1 ZINC000880740148 DE On-Demand Anodyne MT-CYB 49 36 O=C(NC1CSC1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880740153 DD On-Demand Anodyne P2RX7 22 52 O=C(NC1CSC1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880740154 DD On-Demand Anodyne P2RX7 22 52 O=C(NC1CSC1)C1CCCCC1 ZINC000880740156 AD On-Demand Anodyne EPHX2 18 45 O=C(NC1CSC1)C1CCN(S(=O)(=O)c2ccccc2F)CC1 ZINC000880740159 FD On-Demand Anodyne EPHX2 47 77 CCOC(=O)N1CCC(C(=O)NC2CSC2)CC1 ZINC000880740163 CD On-Demand Anodyne EPHX2 19 42 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne ABCC9 15 40 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne ABAT 26 41 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne MAPK11 20 44 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne MAPK14 17 44 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne GRM5 15 67 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne KCNK3 25 48 O=C(NC1CSC1)c1cccc(Cl)c1 ZINC000880740171 BE On-Demand Anodyne KCNK9 15 44 O=C(NC1CSC1)[C@@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880740268 CD On-Demand Anodyne SIGMAR1 16 44 O=C(NC1CSC1)[C@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880740269 CD On-Demand Anodyne SIGMAR1 16 44 O=C(NC1CSC1)c1ccccn1 ZINC000880740277 AC On-Demand Anodyne GRM4 68 44 COc1ccc2c(CC(=O)NC3CSC3)coc2c1 ZINC000880740282 CE On-Demand Anodyne ALDH2 65 32 COc1ccc2c(CC(=O)NC3CSC3)coc2c1 ZINC000880740282 CE On-Demand Anodyne NQO2 34 46 COc1ccc2c(CC(=O)NC3CSC3)coc2c1 ZINC000880740282 CE On-Demand Anodyne MTNR1A 76 46 COc1ccc2c(CC(=O)NC3CSC3)coc2c1 ZINC000880740282 CE On-Demand Anodyne MTNR1B 57 46 COc1cc(CNC(=O)CC2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880740284 FE On-Demand Anodyne GPR119 50 42 O=C(NC1CSC1)c1ccc(Cl)c(Cl)c1 ZINC000880740296 CF On-Demand Anodyne MAPK14 33 40 O=C(NC1CSC1)c1ccc(Cl)c(Cl)c1 ZINC000880740296 CF On-Demand Anodyne UTS2R 23 42 O=C(NC1CSC1)c1ccc(Cl)c(Cl)c1 ZINC000880740296 CF On-Demand Anodyne MAPK13 41 36 O=C(NC1CSC1)c1ccc(Cl)c(Cl)c1 ZINC000880740296 CF On-Demand Anodyne SSTR3 17 41 CSCC[C@H](NC(=O)COc1ccccc1)C(=O)NC1CSC1 ZINC000880740306 FD On-Demand Anodyne CASP3 19 45 CSCC[C@@H](NC(=O)COc1ccccc1)C(=O)NC1CSC1 ZINC000880740307 FD On-Demand Anodyne CASP3 19 45 COc1cc(CNC(=O)C2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880740310 ED On-Demand Anodyne EPHX2 21 41 COc1cc(CNC(=O)C2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880740310 ED On-Demand Anodyne GPR119 48 41 C/C=C\c1ccc(OCC(=O)NC2CSC2)c(OC)c1 ZINC000880740314 CE On-Demand Anodyne TUBB1 46 36 C/C=C/c1ccc(OCC(=O)NC2CSC2)c(OC)c1 ZINC000880740315 CE On-Demand Anodyne TUBB1 46 36 O=C(CCNC(=O)c1ccc(Br)cc1)NC1CSC1 ZINC000880740316 ED On-Demand Anodyne HDAC9 15 43 O=C(COc1cccc2ccccc12)NC1CSC1 ZINC000880740321 CE On-Demand Anodyne CASP6 24 44 O=C(COc1cccc2ccccc12)NC1CSC1 ZINC000880740321 CE On-Demand Anodyne TNKS 40 31 O=C(NC1CSC1)c1ccccc1[N+](=O)[O-] ZINC000880740324 BD On-Demand Bother KCNMA1 17 40 O=C(NC1CSC1)c1ccccc1[N+](=O)[O-] ZINC000880740324 BD On-Demand Bother DAC 15 50 CCOC(=O)c1cc(C(=O)NC2CSC2)cc([N+](=O)[O-])c1 ZINC000880740325 DD On-Demand Bother CACNA1C 43 38 CCOC(=O)c1cc(C(=O)NC2CSC2)cc([N+](=O)[O-])c1 ZINC000880740325 DD On-Demand Bother CACNA1D 61 38 CCOc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880740331 CD On-Demand Anodyne PLA2G4B 46 38 O=C(NC1CSC1)c1ccc(-c2ccc3c(c2)OCCO3)s1 ZINC000880740336 EG On-Demand Anodyne MAPK11 22 41 Cc1noc(C)c1COc1ccc(CC(=O)NC2CSC2)cc1 ZINC000880740339 EF On-Demand Anodyne RORC 20 52 CCCOc1ccc(C(=O)CCC(=O)NC2CSC2)cc1 ZINC000880740342 DF On-Demand Anodyne PLA2G4B 80 37 Cn1nc(C(=O)NC2CSC2)c2ccccc2c1=O ZINC000880740343 CC On-Demand Anodyne HTR3A 16 49 Cn1nc(C(=O)NC2CSC2)c2ccccc2c1=O ZINC000880740343 CC On-Demand Anodyne INHA 54 33 CCOc1ccc(S(=O)(=O)NCCC(=O)NC2CSC2)cc1 ZINC000880740348 EC On-Demand Anodyne MMP13 26 49 CCOc1ccc(S(=O)(=O)NCCC(=O)NC2CSC2)cc1 ZINC000880740348 EC On-Demand Anodyne MMP2 17 45 CCOc1ccc(S(=O)(=O)NCCC(=O)NC2CSC2)cc1 ZINC000880740348 EC On-Demand Anodyne MMP14 17 45 CCOc1ccc(S(=O)(=O)NCCC(=O)NC2CSC2)cc1 ZINC000880740348 EC On-Demand Anodyne MMP1 15 49 Cc1oc(-c2ccccc2)nc1C(=O)NC1CSC1 ZINC000880740352 CE On-Demand Anodyne PPARG 48 40 Cc1oc(-c2ccccc2)nc1C(=O)NC1CSC1 ZINC000880740352 CE On-Demand Anodyne PPARA 51 41 Cc1oc(-c2ccccc2)nc1C(=O)NC1CSC1 ZINC000880740352 CE On-Demand Anodyne PDE8B 64 38 O=C(CSc1ccccc1)NC1CSC1 ZINC000880740356 BE On-Demand Anodyne FAS 49 43 O=C(CCCc1nc(O)c2ccccc2n1)NC1CSC1 ZINC000880740361 DD On-Demand Anodyne TNKS 83 44 O=C(CCCc1nc(O)c2ccccc2n1)NC1CSC1 ZINC000880740361 DD On-Demand Anodyne TNKS2 22 44 O=C(COc1ccc(F)cc1)NC1CSC1 ZINC000880740370 BD On-Demand Anodyne TRAR 34 42 O=C(NC1CSC1)c1ccc(N2CCCC2)c([N+](=O)[O-])c1 ZINC000880740382 DE On-Demand Bother TAAR1 40 53 COc1cc(CNC(=O)CN2CCN(C(=O)OCc3ccccc3)CC2)on1 ZINC000880740383 GD On-Demand Anodyne GRIN2B 19 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnn(-c2ccccc2)n1 ZINC000880740384 FD On-Demand Anodyne PRNP 30 41 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnn(-c2ccccc2)n1 ZINC000880740384 FD On-Demand Anodyne STAT6 55 37 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnn(-c2ccccc2)n1 ZINC000880740384 FD On-Demand Anodyne DGAT1 17 40 CCOc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880740400 CD On-Demand Anodyne PLA2G4B 52 33 CCOc1ccc(OCC(=O)NC2CSC2)cc1 ZINC000880740400 CD On-Demand Anodyne TRAR 34 41 C[C@@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740407 FE On-Demand Anodyne MMP13 25 42 C[C@@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740407 FE On-Demand Anodyne MMP3 24 42 C[C@@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740407 FE On-Demand Anodyne MMP7 31 42 C[C@@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740407 FE On-Demand Anodyne MMP1 31 42 C[C@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740408 FE On-Demand Anodyne MMP13 25 42 C[C@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740408 FE On-Demand Anodyne MMP3 24 42 C[C@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740408 FE On-Demand Anodyne MMP7 31 42 C[C@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)NC2CSC2)cc1 ZINC000880740408 FE On-Demand Anodyne MMP1 31 42 CCCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740414 CG On-Demand Mild MTNR1A 26 40 CCCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740414 CG On-Demand Mild SOAT1 18 41 CCCCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740414 CG On-Demand Mild NOD1 46 33 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccc(Cl)cc2)C1 ZINC000880740415 EE On-Demand Anodyne EPHX2 21 47 O=C(NC1CSC1)[C@@H]1CCCN(C(=O)c2ccc(Cl)cc2)C1 ZINC000880740415 EE On-Demand Anodyne L3MBTL3 63 40 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccc(Cl)cc2)C1 ZINC000880740416 EE On-Demand Anodyne EPHX2 21 47 O=C(NC1CSC1)[C@H]1CCCN(C(=O)c2ccc(Cl)cc2)C1 ZINC000880740416 EE On-Demand Anodyne L3MBTL3 63 40 O=C(NC1CSC1)c1ccc2[nH]c3c(c2c1)CCCC3 ZINC000880740429 CF On-Demand Anodyne PARP1 15 40 CCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740430 BE On-Demand Anodyne MTNR1A 26 40 CCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740430 BE On-Demand Anodyne SOAT1 18 41 CCCCCCC(=O)NCc1cc(OC)no1 ZINC000880740430 BE On-Demand Anodyne NOD1 46 33 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne F10 18 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne PRNP 55 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne MAPKAPK5 42 38 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne MAPK9 31 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne MAPK10 39 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne STAT6 73 38 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880740431 JF On-Demand Anodyne DGAT1 18 41 CCOc1ccc(OCCCC(=O)NC2CSC2)cc1 ZINC000880740437 CE On-Demand Anodyne PLA2G4B 82 40 O=C(CCNS(=O)(=O)c1ccccc1)NC1CSC1 ZINC000880740438 DC On-Demand Anodyne TBXA2R 32 48 O=C(NC1CSC1)C1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000880740439 DE On-Demand Bother EPHX2 16 51 CCSC1(CNC(=O)c2cc(-c3ccc(OC)cc3)on2)CC1 ZINC000880740460 EG On-Demand Anodyne PDK1 42 34 CCSC1(CNC(=O)Cc2ccccc2N2CCCC2=O)CC1 ZINC000880740469 EF On-Demand Anodyne KCNQ2 42 33 O=C(c1cccc2nsnc12)N1CC[C@@H]2C[C@H]2C1 ZINC000880740470 CE On-Demand Anodyne L3MBTL3 40 37 O=C(c1cccc2nsnc12)N1CC[C@H]2C[C@@H]2C1 ZINC000880740471 CE On-Demand Anodyne L3MBTL3 40 37 O=C(c1cccc2nsnc12)N1CC[C@H]2C[C@H]2C1 ZINC000880740472 CE On-Demand Anodyne L3MBTL3 40 37 O=C(c1cccc2nsnc12)N1CC[C@@H]2C[C@@H]2C1 ZINC000880740473 CE On-Demand Anodyne L3MBTL3 40 37 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CC[C@H]2C[C@@H]2C1 ZINC000880740474 CE On-Demand Anodyne L3MBTL3 43 32 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CC[C@@H]2C[C@H]2C1 ZINC000880740475 CE On-Demand Anodyne L3MBTL3 43 32 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CC[C@@H]2C[C@@H]2C1 ZINC000880740476 CE On-Demand Anodyne L3MBTL3 43 32 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CC[C@H]2C[C@H]2C1 ZINC000880740477 CE On-Demand Anodyne L3MBTL3 43 32 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2C[C@@H]2C1 ZINC000880740497 BE On-Demand Anodyne L3MBTL3 58 37 O=C(c1cnc2cc[nH]c2c1)N1CC[C@@H]2C[C@H]2C1 ZINC000880740498 BE On-Demand Anodyne L3MBTL3 58 37 O=C(c1cnc2cc[nH]c2c1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880740499 BE On-Demand Anodyne L3MBTL3 58 37 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2C[C@H]2C1 ZINC000880740500 BE On-Demand Anodyne L3MBTL3 58 37 COc1cc(CNC(=O)C[C@@H]2CCCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880740524 FF On-Demand Anodyne GPR119 44 40 COc1cc(CNC(=O)C[C@H]2CCCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880740525 FF On-Demand Anodyne GPR119 44 40 CCSC1(CNC(=O)c2cccn3nccc23)CC1 ZINC000880740540 CE On-Demand Anodyne HCN1 74 35 CCSC1(CNC(=O)c2cccn3nccc23)CC1 ZINC000880740540 CE On-Demand Anodyne HCN4 52 33 C[C@H]1CN(Cc2ccccc2)C[C@@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740599 EC On-Demand Reactive SIGMAR1 30 40 C[C@H]1CN(Cc2ccccc2)C[C@@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740599 EC On-Demand Reactive TIMP3 42 31 C[C@@H]1CN(Cc2ccccc2)C[C@@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740600 EC On-Demand Reactive SIGMAR1 30 40 C[C@@H]1CN(Cc2ccccc2)C[C@@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740600 EC On-Demand Reactive TIMP3 42 31 C[C@H]1CN(Cc2ccccc2)C[C@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740601 EC On-Demand Reactive SIGMAR1 30 40 C[C@H]1CN(Cc2ccccc2)C[C@H](C(=O)NNC(=O)COC2CC2)O1 ZINC000880740601 EC On-Demand Reactive TIMP3 42 31 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880740627 DG On-Demand Anodyne L3MBTL3 65 37 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@@H]2C[C@H]2C1 ZINC000880740628 DG On-Demand Anodyne L3MBTL3 65 37 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2C[C@@H]2C1 ZINC000880740629 DG On-Demand Anodyne L3MBTL3 65 37 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2C[C@H]2C1 ZINC000880740630 DG On-Demand Anodyne L3MBTL3 65 37 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H]3C[C@H]3C2)N1Cc1ccccc1 ZINC000880740636 ED On-Demand Anodyne PREP 44 37 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H]3C[C@H]3C2)N1Cc1ccccc1 ZINC000880740637 ED On-Demand Anodyne PREP 44 37 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H]3C[C@@H]3C2)N1Cc1ccccc1 ZINC000880740638 ED On-Demand Anodyne PREP 44 37 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H]3C[C@@H]3C2)N1Cc1ccccc1 ZINC000880740639 ED On-Demand Anodyne PREP 44 37 C#CCCOc1ccc(C(=O)NCc2cc(OC)no2)cc1 ZINC000880740664 DE On-Demand Mild SLC5A7 23 42 O=C(NCC1CCC(O)CC1)c1ncccc1-c1ccccn1 ZINC000880740713 DE On-Demand Anodyne GRIN2B 24 40 O=C(NCC1CCC(O)CC1)c1ncccc1-c1ccccn1 ZINC000880740713 DE On-Demand Anodyne MERTK 26 40 O=C(CN1C(=O)c2ccccc2S1(=O)=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880740716 HC On-Demand Anodyne STAT6 59 36 O=C(NCC1CCC(O)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880740744 DE On-Demand Anodyne GABRA1 19 51 O=C(NCC1CCC(O)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880740744 DE On-Demand Anodyne GRIN2B 17 45 O=C(NCC1CCC(O)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880740744 DE On-Demand Anodyne MPO 55 35 O=C(NCC1CCC(O)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880740744 DE On-Demand Anodyne GABRA2 17 51 O=C(Cc1ccccc1N1CCCC1=O)N(CCN1CCOCC1)CC1CC1 ZINC000880740745 GD On-Demand Anodyne CASR 42 35 COC(=O)c1ccc(CNC(=O)COC2CC2)c(F)c1 ZINC000880740781 CD On-Demand Anodyne BDKRB1 26 43 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H]4C[C@H]4C3)cc2)N1 ZINC000880740795 CE On-Demand Anodyne L3MBTL3 74 42 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H]4C[C@@H]4C3)cc2)N1 ZINC000880740796 CE On-Demand Anodyne L3MBTL3 74 42 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H]4C[C@@H]4C3)cc2)N1 ZINC000880740797 CE On-Demand Anodyne L3MBTL3 74 42 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H]4C[C@H]4C3)cc2)N1 ZINC000880740798 CE On-Demand Anodyne L3MBTL3 74 42 COc1cc(CNC(=O)CCc2cccnc2Cl)on1 ZINC000880740826 CD On-Demand Anodyne SUCNR1 41 42 CCSC1(CNC(=O)c2ccc(-c3ccccc3OC)nc2O)CC1 ZINC000880740829 FG On-Demand Anodyne KCNA3 50 43 CCSC1(CNC(=O)c2ccc(-c3ccccc3OC)nc2O)CC1 ZINC000880740829 FG On-Demand Anodyne HCN1 75 39 CCSC1(CNC(=O)c2ccc(-c3ccccc3OC)nc2O)CC1 ZINC000880740829 FG On-Demand Anodyne HCN4 52 39 C#CCC(CC#C)C(=O)NCc1cc(OC)no1 ZINC000880740834 BC On-Demand Mild SLC5A7 22 41 CCSC1(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740880 DG On-Demand Anodyne NQO2 26 40 CCSC1(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740880 DG On-Demand Anodyne MTNR1A 46 45 CCSC1(CNC(=O)[C@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740880 DG On-Demand Anodyne MTNR1B 41 45 CCSC1(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740881 DG On-Demand Anodyne NQO2 26 40 CCSC1(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740881 DG On-Demand Anodyne MTNR1A 46 45 CCSC1(CNC(=O)[C@@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880740881 DG On-Demand Anodyne MTNR1B 41 45 Cc1nc(C(C)C)ncc1C(=O)N[C@H](c1ccccc1)[C@@H](O)C(C)C ZINC000880740907 EG On-Demand Anodyne TACR3 19 42 Cc1nc(C(C)C)ncc1C(=O)N[C@H](c1ccccc1)[C@H](O)C(C)C ZINC000880740908 EG On-Demand Anodyne TACR3 19 42 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](c1ccccc1)[C@@H](O)C(C)C ZINC000880740909 EG On-Demand Anodyne TACR3 19 42 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](c1ccccc1)[C@H](O)C(C)C ZINC000880740910 EG On-Demand Anodyne TACR3 19 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(C)(C)CC1 ZINC000880740914 FE On-Demand Anodyne PAPA1_CARPA 40 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(C)(C)CC1 ZINC000880740915 FE On-Demand Anodyne PAPA1_CARPA 40 49 O=C(Nc1ccc(N2CCOCC2)cn1)c1cccnc1SC(F)F ZINC000880740947 FF On-Demand Anodyne PRNP 26 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cccnc1SC(F)F ZINC000880740947 FF On-Demand Anodyne STAT6 53 33 CC(C)(C(=O)NCC1CCC(O)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880740952 EH On-Demand Anodyne CACNA1I 50 40 CC(C)(C(=O)NCC1CCC(O)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880740952 EH On-Demand Anodyne LIPG 18 46 O=C(c1ccc(CN2CCOCC2)o1)N(CCN1CCOCC1)CC1CC1 ZINC000880740980 GD On-Demand Anodyne CASR 41 36 CCC(=O)c1cc(C(=O)NCc2cc(OC)no2)ccc1F ZINC000880740993 DE On-Demand Anodyne SLC5A7 23 41 O=C(c1cc2ccccc2cc1F)N1CC[C@H]2C[C@H]2C1 ZINC000880741003 CG On-Demand Anodyne L3MBTL3 60 40 O=C(c1cc2ccccc2cc1F)N1CC[C@@H]2C[C@H]2C1 ZINC000880741004 CG On-Demand Anodyne L3MBTL3 60 40 O=C(c1cc2ccccc2cc1F)N1CC[C@H]2C[C@@H]2C1 ZINC000880741005 CG On-Demand Anodyne L3MBTL3 60 40 O=C(c1cc2ccccc2cc1F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741006 CG On-Demand Anodyne L3MBTL3 60 40 COc1cc(CNC(=O)C#CC2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880741019 FD On-Demand Mild GPR119 40 40 COc1cc(CNC(=O)CCC2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880741024 FF On-Demand Anodyne GPR119 51 43 O=C(Cn1cnc2sc(-c3ccccc3)cc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880741048 IF On-Demand Anodyne PRKDC 46 36 O=C(Cn1cnc2sc(-c3ccccc3)cc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880741048 IF On-Demand Anodyne STAT6 48 34 O=C(c1cnc2cc[nH]c2c1)N(CCN1CCOCC1)CC1CC1 ZINC000880741085 ED On-Demand Anodyne CASR 49 36 C=CC(C)(C)CC(=O)NCc1ccc(C(=O)OC)cc1F ZINC000880741093 CF On-Demand Mild BDKRB1 27 43 O=C(NCC1CCC(O)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880741120 DD On-Demand Anodyne HTR4 39 40 O=C(NCC1CCC(O)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880741120 DD On-Demand Anodyne CACNA1I 63 41 O=C(c1cccn2nccc12)N(CCN1CCOCC1)CC1CC1 ZINC000880741144 ED On-Demand Anodyne CASR 48 39 O=C(c1cnc(CC2CC2)s1)N(CCN1CCOCC1)CC1CC1 ZINC000880741170 EE On-Demand Anodyne CASR 47 38 O=C(c1coc(-c2ccccn2)n1)N(CCN1CCOCC1)CC1CC1 ZINC000880741217 FD On-Demand Anodyne CASR 53 41 COC(=O)[C@@H]1CCN(C(=O)c2cnc(CC3CC3)s2)C[C@@H]1C ZINC000880741219 DE On-Demand Anodyne PTR1 48 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CCC(O)CC1 ZINC000880741221 ED On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1CCC(O)CC1 ZINC000880741223 ED On-Demand Anodyne PAPA1_CARPA 39 48 CCSC1(CNC(=O)c2cc(C)cnc2Cl)CC1 ZINC000880741238 CG On-Demand Anodyne SLC6A9 42 35 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne F2 20 41 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne ACE 15 40 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne CELA1 19 42 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne GRIN2B 28 44 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne PREP 29 42 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne LGMN 65 39 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne KLK5 40 40 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne SLC12A5 65 36 O=C(NCC1CCC(O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880741310 GE On-Demand Anodyne Q9NAW4_PLAFA 43 50 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741311 EH On-Demand Anodyne L3MBTL3 66 42 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741313 EH On-Demand Anodyne L3MBTL3 66 42 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741315 EH On-Demand Anodyne L3MBTL3 66 42 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@H]2C[C@H]2C1 ZINC000880741316 EH On-Demand Anodyne L3MBTL3 66 42 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne CELA1 20 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne GRIN2B 32 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne PREP 70 53 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne LGMN 50 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne TGM2 33 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne KLK5 22 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne F13A1 45 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne SLC12A5 46 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@H]2C1 ZINC000880741322 EF On-Demand Anodyne Q9NAW4_PLAFA 25 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne CELA1 20 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne GRIN2B 32 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne PREP 70 53 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne LGMN 50 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne TGM2 33 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne KLK5 22 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne F13A1 45 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne SLC12A5 46 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741324 EF On-Demand Anodyne Q9NAW4_PLAFA 25 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne CELA1 20 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne GRIN2B 32 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne PREP 70 53 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne LGMN 50 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne TGM2 33 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne KLK5 22 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne F13A1 45 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne SLC12A5 46 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741326 EF On-Demand Anodyne Q9NAW4_PLAFA 25 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne CELA1 20 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne GRIN2B 32 45 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne PREP 70 53 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne LGMN 50 38 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne TGM2 33 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne KLK5 22 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne F13A1 45 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne SLC12A5 46 36 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741328 EF On-Demand Anodyne Q9NAW4_PLAFA 25 40 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880741333 ED On-Demand Anodyne CASR 43 33 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880741335 ED On-Demand Anodyne CASR 43 33 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880741337 ED On-Demand Anodyne CASR 43 33 COc1cc(CNC(=O)C[C@@H](C)C2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880741363 GF On-Demand Anodyne GPR119 47 50 COc1cc(CNC(=O)C[C@H](C)C2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880741365 GF On-Demand Anodyne GPR119 47 50 COc1cc(CNC(=O)CC[C@@H]2CCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880741367 FE On-Demand Anodyne GPR119 42 39 COc1cc(CNC(=O)CC[C@H]2CCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880741369 FE On-Demand Anodyne GPR119 42 39 O=C(c1cc(Br)ccc1C1CC1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741388 DH On-Demand Anodyne L3MBTL3 44 36 O=C(c1cc(Br)ccc1C1CC1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741390 DH On-Demand Anodyne L3MBTL3 44 36 O=C(c1cc(Br)ccc1C1CC1)N1CC[C@H]2C[C@H]2C1 ZINC000880741392 DH On-Demand Anodyne L3MBTL3 44 36 O=C(c1cc(Br)ccc1C1CC1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741394 DH On-Demand Anodyne L3MBTL3 44 36 Cc1nc(C(C)C)ncc1C(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880741409 EE On-Demand Anodyne CASR 47 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H]2C[C@@H]2C1 ZINC000880741415 EG On-Demand Anodyne RBP4 80 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H]2C[C@H]2C1 ZINC000880741417 EG On-Demand Anodyne RBP4 80 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741418 EG On-Demand Anodyne RBP4 80 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H]2C[C@H]2C1 ZINC000880741420 EG On-Demand Anodyne RBP4 80 37 COC(=O)c1ccc(CNC(=O)CC[C@H]2CC(C)(C)CO2)c(F)c1 ZINC000880741426 EF On-Demand Anodyne BDKRB1 26 40 COC(=O)c1ccc(CNC(=O)CC[C@@H]2CC(C)(C)CO2)c(F)c1 ZINC000880741428 EF On-Demand Anodyne BDKRB1 26 40 COc1cc(CNC(=O)Cc2ccc(Cl)nc2C)on1 ZINC000880741473 CD On-Demand Anodyne P2RX7 48 42 COc1cc(CNC(=O)CSC2CCN(C(=O)OC(C)(C)C)CC2)on1 ZINC000880741542 GE On-Demand Anodyne GPR119 46 40 COc1cc(CNC(=O)Cc2cc(C)n(-c3ccccc3)c2C)on1 ZINC000880741550 EF On-Demand Clean P2RX7 26 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C(C)(C)C1(F)F)C2 ZINC000880741579 DG On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C(C)(C)C1(F)F)C2 ZINC000880741579 DG On-Demand Anodyne NQO2 33 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C(C)(C)C1(F)F)C2 ZINC000880741579 DG On-Demand Anodyne MTNR1A 49 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C(C)(C)C1(F)F)C2 ZINC000880741579 DG On-Demand Anodyne MTNR1B 44 45 Cn1nnc(C(=O)N(CCN2CCOCC2)CC2CC2)n1 ZINC000880741584 CB On-Demand Anodyne CASR 36 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1C(C)(C)C1(F)F)C2 ZINC000880741585 DG On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1C(C)(C)C1(F)F)C2 ZINC000880741585 DG On-Demand Anodyne NQO2 33 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1C(C)(C)C1(F)F)C2 ZINC000880741585 DG On-Demand Anodyne MTNR1A 49 45 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1C(C)(C)C1(F)F)C2 ZINC000880741585 DG On-Demand Anodyne MTNR1B 44 45 Cc1cnc(Cl)c(C(=O)NCC2(O)CCC(C)(C)CC2)c1 ZINC000880741604 DG On-Demand Anodyne P2RX7 15 54 CC(C)(C(=O)NCC1CCC(O)CC1)c1ccc(F)cc1F ZINC000880741638 DF On-Demand Anodyne CACNA1I 45 34 COC(=O)[C@@H]1CCN(C(=O)c2csc(-c3ncc[nH]3)n2)C[C@@H]1C ZINC000880741649 ED On-Demand Anodyne TRPC6 46 39 O=C(c1csc(-c2ncc[nH]2)n1)N(CCN1CCOCC1)CC1CC1 ZINC000880741653 FD On-Demand Anodyne CASR 43 38 COC(=O)c1ccc(CNC(=O)Cc2ccccc2N2CCCC2=O)c(F)c1 ZINC000880741657 GF On-Demand Anodyne P2RX7 50 41 COC(=O)[C@@H]1CCN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C[C@@H]1C ZINC000880741678 GG On-Demand Anodyne RBP4 49 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C(C)(C)C1(F)F ZINC000880741713 FE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1C(C)(C)C1(F)F ZINC000880741714 FE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1C(C)(C)C1(F)F ZINC000880741715 FE On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C(C)(C)C1(F)F ZINC000880741716 FE On-Demand Anodyne PAPA1_CARPA 39 47 COc1cc(CNC(=O)/C(C)=C\c2ccc(OC)c(F)c2)on1 ZINC000880741754 DF On-Demand Anodyne TUBB1 38 49 COc1cc(CNC(=O)/C(C)=C/c2ccc(OC)c(F)c2)on1 ZINC000880741755 DF On-Demand Anodyne TUBB1 38 49 O=C(Cc1csc(-c2sccc2Br)n1)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741781 GI On-Demand Anodyne ETHR 43 37 O=C(Cc1csc(-c2sccc2Br)n1)N1CC[C@H]2C[C@H]2C1 ZINC000880741782 GI On-Demand Anodyne ETHR 43 37 O=C(Cc1csc(-c2sccc2Br)n1)N1CC[C@H]2C[C@@H]2C1 ZINC000880741783 GI On-Demand Anodyne ETHR 43 37 O=C(Cc1csc(-c2sccc2Br)n1)N1CC[C@@H]2C[C@H]2C1 ZINC000880741784 GI On-Demand Anodyne ETHR 43 37 O=C(NCC1CCC(O)CC1)c1cc(Br)ccc1C1CC1 ZINC000880741838 FH On-Demand Anodyne CACNA1I 51 35 O=C(NCC1CCC(O)CC1)c1coc(-c2ccccn2)n1 ZINC000880741839 DE On-Demand Anodyne GRIN2B 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741860 FF On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741860 FF On-Demand Anodyne REN 29 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741860 FF On-Demand Anodyne FPR1 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741861 FF On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741861 FF On-Demand Anodyne REN 29 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741861 FF On-Demand Anodyne FPR1 41 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741862 FF On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741862 FF On-Demand Anodyne REN 29 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C1CCC(F)CC1 ZINC000880741862 FF On-Demand Anodyne FPR1 41 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741863 FF On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741863 FF On-Demand Anodyne REN 29 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)C1CCC(F)CC1 ZINC000880741863 FF On-Demand Anodyne FPR1 41 37 COC(=O)c1ccc(CNC(=O)CC(C)(C)CC(F)(F)F)c(F)c1 ZINC000880741864 EH On-Demand Anodyne BDKRB1 27 43 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MMP13 18 40 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MTNR1A 15 44 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MTNR1B 16 44 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MMP3 23 40 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MMP9 19 40 COC(=O)[C@@H]1CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741876 EE On-Demand Anodyne MMP1 20 40 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MMP13 18 40 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MTNR1A 15 44 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MTNR1B 16 44 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MMP3 23 40 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MMP9 19 40 COC(=O)[C@@H]1CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880741877 EE On-Demand Anodyne MMP1 20 40 O=C(NCC1CCC(O)CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880741878 EG On-Demand Anodyne PDE4D 34 53 O=C(NCC1CCC(O)CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880741878 EG On-Demand Anodyne CACNA1I 72 44 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne ACHE 21 44 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne GRIN2B 37 54 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne TBXAS1 21 40 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne CHRNA7 41 47 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne C3AR1 43 56 O=C(/C=C\c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741894 DH On-Demand Anodyne NAMPT 20 56 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne ACHE 21 44 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne GRIN2B 37 54 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne TBXAS1 21 40 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne CHRNA7 41 47 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne C3AR1 43 56 O=C(/C=C/c1cccnc1)N1CCC(CCc2ccccc2)CC1 ZINC000880741895 DH On-Demand Anodyne NAMPT 20 56 COc1cc(CNC(=O)Cc2ccc(C)nc2Cl)on1 ZINC000880741915 CD On-Demand Anodyne P2RX7 40 40 Cc1cc([C@@H]2CCN(C(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)C2)c(O)cc1Cl ZINC000880741918 GH On-Demand Anodyne L3MBTL3 53 35 Cc1cc([C@@H]2CCN(C(=O)c3ccc([C@H]4CCC(=O)N4)cc3)C2)c(O)cc1Cl ZINC000880741921 GH On-Demand Anodyne L3MBTL3 53 35 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CC[C@@H]2C[C@@H]2C1 ZINC000880741934 DE On-Demand Bother L3MBTL3 21 43 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CC[C@@H]2C[C@H]2C1 ZINC000880741935 DE On-Demand Bother L3MBTL3 21 43 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CC[C@H]2C[C@H]2C1 ZINC000880741936 DE On-Demand Bother L3MBTL3 21 43 O=C(c1cc2c(cc1[N+](=O)[O-])OCCCO2)N1CC[C@H]2C[C@@H]2C1 ZINC000880741937 DE On-Demand Bother L3MBTL3 21 43 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC[C@H]4C[C@@H]4C3)ccn2)CC1 ZINC000880741938 GF On-Demand Anodyne GPR119 57 57 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC[C@@H]4C[C@@H]4C3)ccn2)CC1 ZINC000880741939 GF On-Demand Anodyne GPR119 57 57 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC[C@H]4C[C@H]4C3)ccn2)CC1 ZINC000880741940 GF On-Demand Anodyne GPR119 57 57 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC[C@@H]4C[C@H]4C3)ccn2)CC1 ZINC000880741941 GF On-Demand Anodyne GPR119 57 57 O=C(N1CC[C@@H]2C[C@@H]2C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880741952 CF On-Demand Anodyne RBP4 59 35 O=C(N1CC[C@H]2C[C@H]2C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880741953 CF On-Demand Anodyne RBP4 59 35 O=C(N1CC[C@@H]2C[C@H]2C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880741954 CF On-Demand Anodyne RBP4 59 35 O=C(N1CC[C@H]2C[C@@H]2C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880741955 CF On-Demand Anodyne RBP4 59 35 CCSC1(CNC(=O)c2cccc3nsnc23)CC1 ZINC000880741972 CF On-Demand Anodyne HCN1 42 31 COc1cc(CNC(=O)C[C@H]2CCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880741979 ED On-Demand Anodyne GPR119 42 39 COc1cc(CNC(=O)C[C@@H]2CCN(C(=O)OC(C)(C)C)C2)on1 ZINC000880741980 ED On-Demand Anodyne GPR119 42 39 Cc1cnc(Cl)c(C(=O)N(CCN2CCOCC2)CC2CC2)c1 ZINC000880741987 EE On-Demand Anodyne CASR 51 39 COC(=O)c1ccc(CNC(=O)C2CCC(S(C)(=O)=O)CC2)c(F)c1 ZINC000880741999 FD On-Demand Anodyne EPHX2 18 45 COC(=O)[C@@H]1CCN(C(=O)CCCCc2ccc(OC)c(OC)c2)C[C@@H]1C ZINC000880742000 GG On-Demand Anodyne FKBP1A 46 42 Cc1cnc(Cl)c(C(=O)NCC2CCC(O)CC2)c1 ZINC000880742001 CE On-Demand Anodyne HTR4 18 41 Cc1cnc(Cl)c(C(=O)NCC2CCC(O)CC2)c1 ZINC000880742001 CE On-Demand Anodyne CACNA1I 63 41 C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CCC(F)CC1 ZINC000880742004 EG On-Demand Anodyne KCNQ2 49 33 COC(=O)c1ccc(CNC(=O)CC(C)(C)CC(F)F)c(F)c1 ZINC000880742006 EG On-Demand Anodyne BDKRB1 26 42 O=C(c1cccc2nsnc12)N(CCN1CCOCC1)CC1CC1 ZINC000880742010 ED On-Demand Anodyne CASR 51 40 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)(C)CC2)c(O)n1 ZINC000880742011 GH On-Demand Anodyne KCNA3 51 42 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)(C)CC2)c(O)n1 ZINC000880742011 GH On-Demand Anodyne HCN1 74 38 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)(C)CC2)c(O)n1 ZINC000880742011 GH On-Demand Anodyne HCN4 52 38 O=C(NCC1CCC(O)CC1)c1ccc(OC(F)F)c(Br)c1 ZINC000880742020 GG On-Demand Anodyne PDE4D 31 46 O=C(NCC1CCC(O)CC1)c1ccc(OC(F)F)c(Br)c1 ZINC000880742020 GG On-Demand Anodyne CACNA1I 65 38 COc1cccc(C2=NO[C@H](C(=O)NCc3cc(OC)no3)C2)c1 ZINC000880742063 ED On-Demand Anodyne LUCI_PHOPY 34 46 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCC(O)CC3)cc2)N1 ZINC000880742064 DD On-Demand Anodyne GRIN2B 17 45 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCC(O)CC3)cc2)N1 ZINC000880742064 DD On-Demand Anodyne CACNA1I 55 34 COc1cccc(C2=NO[C@@H](C(=O)NCc3cc(OC)no3)C2)c1 ZINC000880742065 ED On-Demand Anodyne LUCI_PHOPY 34 46 O=C1CC[C@H](c2ccc(C(=O)NCC3CCC(O)CC3)cc2)N1 ZINC000880742067 DD On-Demand Anodyne GRIN2B 17 45 O=C1CC[C@H](c2ccc(C(=O)NCC3CCC(O)CC3)cc2)N1 ZINC000880742067 DD On-Demand Anodyne CACNA1I 55 34 O=C(C(=O)N(CCN1CCOCC1)CC1CC1)c1c[nH]c2cc(F)ccc12 ZINC000880742069 FE On-Demand Anodyne CASR 41 37 COC(=O)[C@@H]1CCN(C(=O)C(C)(C)c2ccc(F)cc2F)C[C@@H]1C ZINC000880742106 EF On-Demand Anodyne PRCP 42 33 COc1cc(CNC(=O)C(F)F)on1 ZINC000880742113 BC On-Demand Anodyne ALS 44 31 COC(=O)c1ccc(CNC(=O)c2ccc(CN3CCOCC3)o2)c(F)c1 ZINC000880742128 GD On-Demand Anodyne BDKRB1 24 45 O=C(CC[C@H]1CCc2ccccc21)NCC1CCC(O)CC1 ZINC000880742143 DG On-Demand Anodyne NQO2 20 42 O=C(CC[C@H]1CCc2ccccc21)NCC1CCC(O)CC1 ZINC000880742143 DG On-Demand Anodyne MTNR1B 27 46 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCC(O)CC1 ZINC000880742144 DG On-Demand Anodyne NQO2 20 42 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCC(O)CC1 ZINC000880742144 DG On-Demand Anodyne MTNR1B 27 46 COC(=O)c1ccc(CNC(=O)[C@@H]2CCc3nncn3CC2)c(F)c1 ZINC000880742146 ED On-Demand Anodyne P2RX7 49 38 COC(=O)c1ccc(CNC(=O)[C@@H]2CCc3nncn3CC2)c(F)c1 ZINC000880742146 ED On-Demand Anodyne EPHX2 19 42 COC(=O)c1ccc(CNC(=O)[C@H]2CCc3nncn3CC2)c(F)c1 ZINC000880742147 ED On-Demand Anodyne P2RX7 49 38 COC(=O)c1ccc(CNC(=O)[C@H]2CCc3nncn3CC2)c(F)c1 ZINC000880742147 ED On-Demand Anodyne EPHX2 19 42 O=C(NCC1CCC(O)CC1)c1cccc2nsnc12 ZINC000880742155 CD On-Demand Anodyne ACACB 15 40 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCC(O)CC2)N1Cc1ccccc1 ZINC000880742184 FD On-Demand Anodyne F2 23 43 COC(=O)c1ccc(CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c(F)c1 ZINC000880742189 FE On-Demand Anodyne P2RX7 20 40 COC(=O)c1ccc(CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c(F)c1 ZINC000880742190 FE On-Demand Anodyne P2RX7 20 40 COC(=O)c1ccc(CNC(=O)Cc2c(Br)cnn2C)c(F)c1 ZINC000880742201 GD On-Demand Anodyne P2RX7 38 53 COC(=O)c1ccc(CNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)c(F)c1 ZINC000880742205 FD On-Demand Anodyne P2RX7 37 40 COc1ccccc1-c1ccc(C(=O)NCC2CCC(O)CC2)c(O)n1 ZINC000880742223 FF On-Demand Anodyne KCNA3 45 36 O=C(NCC1CCC(O)CC1)c1cnc2cc[nH]c2c1 ZINC000880742228 CD On-Demand Anodyne GRIN2B 20 46 O=C(NCC1CCC(O)CC1)c1cnc2cc[nH]c2c1 ZINC000880742228 CD On-Demand Anodyne CACNA1I 55 36 COC(=O)c1ccc(CNC(=O)C[C@@H]2C[C@H]2C2CC2)c(F)c1 ZINC000880742266 DF On-Demand Anodyne BDKRB1 21 41 O=C(NCC1CCC(O)CC1)c1cc2ccccc2cc1F ZINC000880742272 DG On-Demand Anodyne GRIN2B 19 48 O=C(NCC1CCC(O)CC1)c1cc2ccccc2cc1F ZINC000880742272 DG On-Demand Anodyne CACNA1I 48 33 Cc1cc(C)c2c(-n3cccc3)c(C(=O)Nc3ccc(N4CCOCC4)cn3)sc2n1 ZINC000880742292 II On-Demand Anodyne STAT6 46 30 COC(=O)[C@@H]1CCN(C(=O)c2cc(-c3ccc(OC)cc3)on2)C[C@@H]1C ZINC000880742315 FF On-Demand Anodyne PDK1 41 36 COC(=O)[C@@H]1CCN(C(=O)c2cc(-c3ccc(OC)cc3)on2)C[C@@H]1C ZINC000880742315 FF On-Demand Anodyne TRPC6 35 42 COC(=O)[C@@H]1CCN(C(=O)c2cc(-c3ccc(OC)cc3)on2)C[C@@H]1C ZINC000880742315 FF On-Demand Anodyne TRPC3 28 42 O=C(NCCNC(=O)c1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742336 EF On-Demand Anodyne NAMPT 36 40 O=C(NCCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742354 DH On-Demand Anodyne TBXAS1 42 46 O=C(NCCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742354 DH On-Demand Anodyne HMOX2 44 31 O=C(NCCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742354 DH On-Demand Anodyne QPCT 37 48 CNC(=O)CC1(CNC(=O)c2coc(-c3ccccn3)n2)CCCCC1 ZINC000880742355 FF On-Demand Anodyne HCN1 49 31 CNC(=O)CC1(CNC(=O)c2coc(-c3ccccn3)n2)CCCCC1 ZINC000880742355 FF On-Demand Anodyne HCN4 47 31 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742363 FH On-Demand Anodyne EPHX2 49 44 CS(=O)(=O)C1CCC(C(=O)NC[C@@H](O)c2ccc(Cl)c(Cl)c2)CC1 ZINC000880742364 GF On-Demand Anodyne ADRB3 22 41 CS(=O)(=O)C1CCC(C(=O)NC[C@H](O)c2ccc(Cl)c(Cl)c2)CC1 ZINC000880742365 GF On-Demand Anodyne ADRB3 22 41 CS(=O)(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742366 GG On-Demand Anodyne TRPV1 103 39 CS(=O)(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742366 GG On-Demand Anodyne ROCK2 15 48 CC(C)(C)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742371 EI On-Demand Anodyne EPHX2 41 43 O=C(CC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)NC1CCCC1 ZINC000880742411 GI On-Demand Anodyne DGAT1 17 41 CC(=O)Nc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880742413 EH On-Demand Anodyne TRPV1 21 48 CC(=O)Nc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880742413 EH On-Demand Anodyne IDO1 15 40 COc1ccccc1[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)c1nccn1C ZINC000880742417 GI On-Demand Anodyne P2RY1 17 41 CN(c1ccccc1)[C@H]1CCN(C(=O)CC(C)(C)CC(F)F)C1 ZINC000880742450 DH On-Demand Anodyne SFRP1 86 39 CN(c1ccccc1)[C@H]1CCN(C(=O)CC(C)(C)CC(F)F)C1 ZINC000880742450 DH On-Demand Anodyne WNT3 64 39 CN(c1ccccc1)[C@@H]1CCN(C(=O)CC(C)(C)CC(F)F)C1 ZINC000880742451 DH On-Demand Anodyne SFRP1 86 39 CN(c1ccccc1)[C@@H]1CCN(C(=O)CC(C)(C)CC(F)F)C1 ZINC000880742451 DH On-Demand Anodyne WNT3 64 39 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742458 GH On-Demand Anodyne CA2 30 45 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742458 GH On-Demand Anodyne CA1 29 44 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742458 GH On-Demand Anodyne TRPV1 93 37 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742458 GH On-Demand Anodyne CA4 34 45 O=C(NCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880742473 DE On-Demand Anodyne EPHX2 29 52 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880742480 FH On-Demand Anodyne NPY2R 24 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880742480 FH On-Demand Anodyne SLC18A3 17 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880742480 FH On-Demand Anodyne RBP4 57 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880742480 FH On-Demand Anodyne SMO 49 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880742480 FH On-Demand Anodyne L3MBTL3 44 35 CN(c1ccccc1)[C@@H]1CCN(C(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)C1 ZINC000880742483 FE On-Demand Anodyne CCR5 18 40 CN(c1ccccc1)[C@H]1CCN(C(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)C1 ZINC000880742484 FE On-Demand Anodyne CCR5 18 40 O=C(NNc1ccc(Cl)cn1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880742487 ED On-Demand Reactive F10 22 41 C#C[C@@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CCOCC1 ZINC000880742493 FD On-Demand Mild PAPA1_CARPA 34 41 C#C[C@H](NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C1CCOCC1 ZINC000880742494 FD On-Demand Mild PAPA1_CARPA 34 41 C#C[C@@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CCOCC1 ZINC000880742495 FD On-Demand Mild PAPA1_CARPA 34 41 C#C[C@H](NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C1CCOCC1 ZINC000880742496 FD On-Demand Mild PAPA1_CARPA 34 41 CCOC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742500 EH On-Demand Anodyne CACNA1H 40 32 CCOC(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742507 EG On-Demand Anodyne EPHX2 52 43 CCOC(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742507 EG On-Demand Anodyne CCR8 48 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2cccc(F)c2)CC1 ZINC000880742534 GI On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2cccc(F)c2)CC1 ZINC000880742534 GI On-Demand Anodyne HRH3 26 41 O=C(NCc1nnc2ccc(C(F)(F)F)cn12)Nc1ccc(C2CC2)cc1F ZINC000880742537 GI On-Demand Anodyne TRPV1 52 34 CS(=O)(=O)NCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742546 DD On-Demand Anodyne TRPV1 98 38 O=C(NCCOCC(F)(F)F)Nc1ccc(C2CC2)cc1F ZINC000880742549 DG On-Demand Anodyne TRPV1 54 34 O=C(Nc1ccc(C2CC2)cc1F)NC1CCOCC1 ZINC000880742554 CG On-Demand Anodyne EPHX2 21 47 O=C(NCCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742555 CG On-Demand Anodyne TRPV1 18 40 O=C(NCCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742555 CG On-Demand Anodyne CHRNA7 43 38 O=C(NCCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880742555 CG On-Demand Anodyne NAMPT 47 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@H](c2ccccc2)C1 ZINC000880742560 EI On-Demand Anodyne RBP4 57 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@H](c2ccccc2)C1 ZINC000880742561 EI On-Demand Anodyne RBP4 57 36 CNC(=O)CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880742569 EE On-Demand Anodyne HCN1 68 37 CNC(=O)CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880742569 EE On-Demand Anodyne HCN4 56 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880742570 GI On-Demand Anodyne HRH3 24 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880742570 GI On-Demand Anodyne L3MBTL3 62 38 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742578 EH On-Demand Anodyne TRPV1 19 40 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742579 EH On-Demand Anodyne TRPV1 19 40 CC(=O)NCC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742584 EG On-Demand Anodyne CACNA1I 51 31 CC(C)(C)C(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742594 EG On-Demand Anodyne CACNA1H 52 36 CC(C)(C)C(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742594 EG On-Demand Anodyne RBP4 41 37 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742601 GJ On-Demand Anodyne EPHX2 32 41 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742601 GJ On-Demand Anodyne RBP4 53 39 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742601 GJ On-Demand Anodyne DGAT1 28 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C2CC2)CC1 ZINC000880742610 DG On-Demand Anodyne EPHX2 40 44 O=C(CCNC(=O)Nc1ccc(C2CC2)cc1F)NC1CCCCC1 ZINC000880742618 EH On-Demand Anodyne EPHX2 18 47 CC(C)(C)N1C[C@H](CNC(=O)CC[C@H]2CCc3ccccc32)CC1=O ZINC000880742651 EG On-Demand Anodyne MTNR1A 15 42 CC(C)(C)N1C[C@@H](CNC(=O)CC[C@H]2CCc3ccccc32)CC1=O ZINC000880742652 EG On-Demand Anodyne MTNR1A 15 42 CC(C)(C)N1C[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)CC1=O ZINC000880742653 EG On-Demand Anodyne MTNR1A 15 42 CC(C)(C)N1C[C@@H](CNC(=O)CC[C@@H]2CCc3ccccc32)CC1=O ZINC000880742654 EG On-Demand Anodyne MTNR1A 15 42 O=C(NC[C@H](O)c1ccc(Cl)c(Cl)c1)c1c[nH]cc1C1CC1 ZINC000880742658 EH On-Demand Anodyne CCR3 16 42 O=C(NC[C@@H](O)c1ccc(Cl)c(Cl)c1)c1c[nH]cc1C1CC1 ZINC000880742659 EH On-Demand Anodyne CCR3 16 42 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742662 DF On-Demand Anodyne PLD1 46 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CC1)OCCO2 ZINC000880742664 DG On-Demand Anodyne CACNA1H 55 38 COCCn1cc(NC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880742665 DG On-Demand Anodyne PANC 53 37 CCC(=O)N1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742666 EG On-Demand Anodyne CACNA1H 41 34 CS(=O)(=O)NCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742675 ED On-Demand Anodyne TRPV1 94 38 CC(C)(C)N1C[C@@H](CNC(=O)c2cnc3cc[nH]c3c2)CC1=O ZINC000880742676 DD On-Demand Anodyne CACNA1I 62 37 CC(C)(C)N1C[C@H](CNC(=O)c2cnc3cc[nH]c3c2)CC1=O ZINC000880742677 DD On-Demand Anodyne CACNA1I 62 37 CCCN(CCO)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742679 CF On-Demand Anodyne SOAT1 24 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2sccc2C1 ZINC000880742694 DI On-Demand Anodyne TRPM8 15 40 CN(c1ccccc1)[C@H]1CCN(C(=O)CC(C)(C)CC(F)(F)F)C1 ZINC000880742702 EI On-Demand Anodyne SFRP1 86 39 CN(c1ccccc1)[C@H]1CCN(C(=O)CC(C)(C)CC(F)(F)F)C1 ZINC000880742702 EI On-Demand Anodyne WNT3 64 39 CN(c1ccccc1)[C@@H]1CCN(C(=O)CC(C)(C)CC(F)(F)F)C1 ZINC000880742703 EI On-Demand Anodyne SFRP1 86 39 CN(c1ccccc1)[C@@H]1CCN(C(=O)CC(C)(C)CC(F)(F)F)C1 ZINC000880742703 EI On-Demand Anodyne WNT3 64 39 CC[C@H]1CCC[C@]1(C)C(=O)Nc1cnn(C(C)(C)C(=O)OC)c1 ZINC000880742707 DF On-Demand Anodyne PANC 49 33 CC[C@@H]1CCC[C@@]1(C)C(=O)Nc1cnn(C(C)(C)C(=O)OC)c1 ZINC000880742708 DF On-Demand Anodyne PANC 49 33 CC[C@H]1CCC[C@@]1(C)C(=O)Nc1cnn(C(C)(C)C(=O)OC)c1 ZINC000880742709 DF On-Demand Anodyne PANC 49 33 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1ccc(C2CC2)cc1F ZINC000880742712 GI On-Demand Anodyne NPY1R 22 41 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1ccc(C2CC2)cc1F ZINC000880742712 GI On-Demand Anodyne NAMPT 16 40 CN(c1ccccc1)[C@@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742729 FE On-Demand Anodyne CCR5 32 40 CN(c1ccccc1)[C@@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742729 FE On-Demand Anodyne SFRP1 77 34 CN(c1ccccc1)[C@@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742729 FE On-Demand Anodyne WNT3 69 34 CN(c1ccccc1)[C@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742730 FE On-Demand Anodyne CCR5 32 40 CN(c1ccccc1)[C@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742730 FE On-Demand Anodyne SFRP1 77 34 CN(c1ccccc1)[C@H]1CCN(C(=O)C2CCC(S(C)(=O)=O)CC2)C1 ZINC000880742730 FE On-Demand Anodyne WNT3 69 34 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne DRD4 23 48 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne SIGMAR1 21 48 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne SSTR5 47 38 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne CCR3 45 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne CXCR3 28 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccncc2)CC1 ZINC000880742737 FH On-Demand Anodyne MCHR1 67 45 COc1ccc(-c2nnc(S)n2CCC(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880742744 IF On-Demand Anodyne STAT6 57 35 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccccc1 ZINC000880742745 GI On-Demand Anodyne DRD4 20 40 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccccc1 ZINC000880742745 GI On-Demand Anodyne CCR1 26 42 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccccc1 ZINC000880742745 GI On-Demand Anodyne EPHX2 37 42 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccccc1 ZINC000880742745 GI On-Demand Anodyne RBP4 53 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ccccn2)CC1 ZINC000880742759 EG On-Demand Anodyne EBP 28 46 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ccccn2)CC1 ZINC000880742759 EG On-Demand Anodyne RBP4 47 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ccccn2)CC1 ZINC000880742759 EG On-Demand Anodyne DGAT1 20 44 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccc(F)cc1 ZINC000880742762 GI On-Demand Anodyne CCR1 17 43 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccc(F)cc1 ZINC000880742762 GI On-Demand Anodyne CCR3 15 46 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)c1ccc(F)cc1 ZINC000880742762 GI On-Demand Anodyne MCHR1 18 44 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880742767 EG On-Demand Anodyne EPHX2 46 54 N#Cc1ccnc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)c1 ZINC000880742770 FG On-Demand Mild MAP3K12 47 35 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742771 FG On-Demand Anodyne ROCK2 21 50 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(N2CCCCC2)CC1 ZINC000880742772 EI On-Demand Anodyne CALCRL 48 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(N2CCCCC2)CC1 ZINC000880742772 EI On-Demand Anodyne L3MBTL3 113 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2cccnc2)CC1 ZINC000880742779 FG On-Demand Anodyne CHRNA7 47 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2cccnc2)CC1 ZINC000880742779 FG On-Demand Anodyne FAAH 32 48 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2cccnc2)CC1 ZINC000880742779 FG On-Demand Anodyne MCHR1 18 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880742781 FH On-Demand Anodyne DRD4 17 53 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880742781 FH On-Demand Anodyne SIGMAR1 17 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880742781 FH On-Demand Anodyne CCR3 31 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880742781 FH On-Demand Anodyne EPHX2 25 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(Cc2ccccn2)CC1 ZINC000880742781 FH On-Demand Anodyne MCHR1 45 41 NC(=O)c1ccc(CN(C(=O)Nc2ccc(C3CC3)cc2F)C2CC2)cc1 ZINC000880742785 FH On-Demand Anodyne GCGR 32 40 NC(=O)c1ccc(CN(C(=O)Nc2ccc(C3CC3)cc2F)C2CC2)cc1 ZINC000880742785 FH On-Demand Anodyne GIPR 56 41 CCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742797 DG On-Demand Anodyne CCR3 28 41 CCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742797 DG On-Demand Anodyne EPHX2 42 43 CCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742797 DG On-Demand Anodyne CXCR3 20 42 NC(=O)c1ccc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)nc1 ZINC000880742802 GF On-Demand Anodyne DGAT1 21 45 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)C1CC1 ZINC000880742810 EG On-Demand Anodyne EPHX2 34 42 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742823 EE On-Demand Anodyne DRD4 16 45 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742823 EE On-Demand Anodyne EPHX2 30 40 Cc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)n1 ZINC000880742838 CH On-Demand Anodyne TRPV1 21 41 CNC(=O)CC1(CNC(=O)c2ncccc2-c2ccccn2)CCCCC1 ZINC000880742839 FF On-Demand Anodyne HCN1 50 31 CNC(=O)CC1(CNC(=O)c2ncccc2-c2ccccn2)CCCCC1 ZINC000880742839 FF On-Demand Anodyne HCN4 47 31 O=C(Nc1ccc(C2CC2)cc1F)N1CCOc2ccccc2C1 ZINC000880742840 EI On-Demand Anodyne DGAT1 15 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](N2CCCC2)C1 ZINC000880742845 EH On-Demand Anodyne L3MBTL3 69 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](N2CCCC2)C1 ZINC000880742846 EH On-Demand Anodyne L3MBTL3 69 40 CC(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742847 EH On-Demand Anodyne TRPV1 17 42 CC(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742847 EH On-Demand Anodyne NPY1R 24 41 CC(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742847 EH On-Demand Anodyne CCR3 51 38 CC(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742847 EH On-Demand Anodyne ROCK2 21 45 CC(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742847 EH On-Demand Anodyne MCHR1 26 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccccc2F)CC1 ZINC000880742860 GI On-Demand Anodyne RBP4 54 38 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742861 EH On-Demand Anodyne SOAT1 24 40 COC(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742865 EG On-Demand Anodyne EPHX2 51 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880742868 FG On-Demand Anodyne GRM4 45 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880742868 FG On-Demand Anodyne RBP4 54 34 Cn1ncc2c(N3CCN(C(=O)Nc4ccc(C5CC5)cc4F)CC3)ncnc21 ZINC000880742869 GF On-Demand Anodyne PDGFRB 56 40 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne HTR1A 52 52 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne DRD2 51 45 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne DRD4 33 45 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne ADRA1D 53 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne HTR2A 49 45 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne HTR2C 28 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne ADRA1A 72 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne ADRA1B 46 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne DRD3 58 46 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne HTR7 53 39 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne CCR3 43 43 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc(C2CC2)cc1F ZINC000880742873 GF On-Demand Anodyne MCHR1 26 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880742875 FJ On-Demand Anodyne RBP4 53 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880742876 FJ On-Demand Anodyne RBP4 53 38 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742890 GI On-Demand Anodyne CCR1 34 40 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880742890 GI On-Demand Anodyne EPHX2 42 47 CN(C)C(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880742895 FH On-Demand Anodyne ROCK2 21 43 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)nc1 ZINC000880742898 FG On-Demand Mild FASN 41 46 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)nc1 ZINC000880742898 FG On-Demand Mild DGAT1 18 44 CC[C@H](C)NC(=O)CCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880742903 DG On-Demand Anodyne TRPV1 59 35 CN(Cc1cccc(C#N)c1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742915 DI On-Demand Mild MCHR1 29 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(CC(F)(F)F)CC1 ZINC000880742917 EG On-Demand Anodyne RBP4 44 36 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1ccc(C2CC2)cc1F ZINC000880742919 GI On-Demand Anodyne L3MBTL3 76 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1=CCCC1 ZINC000880742920 DE On-Demand Anodyne PAPA1_CARPA 44 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1=CCCC1 ZINC000880742920 DE On-Demand Anodyne FPR1 44 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1=CCCC1 ZINC000880742921 DE On-Demand Anodyne PAPA1_CARPA 44 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1=CCCC1 ZINC000880742921 DE On-Demand Anodyne FPR1 44 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCCC1 ZINC000880742922 BG On-Demand Anodyne RBP4 44 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2ccncc2)CC1 ZINC000880742930 FG On-Demand Anodyne FAAH 24 46 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2ccncc2)CC1 ZINC000880742930 FG On-Demand Anodyne MCHR1 30 44 Cc1ncc(CC(=O)NC[C@@H](O)c2ccc(Cl)c(Cl)c2)o1 ZINC000880742937 EF On-Demand Anodyne ADRB2 36 40 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ccc(Cl)cn1)C2 ZINC000880742938 EF On-Demand Reactive F10 47 31 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ccc(Cl)cn1)C2 ZINC000880742938 EF On-Demand Reactive FAAH 15 42 O=C(NCCCN1CCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880742943 DF On-Demand Anodyne ADRA1B 25 42 O=C(NCCCN1CCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880742943 DF On-Demand Anodyne CCR3 37 40 O=C(NCCCN1CCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880742943 DF On-Demand Anodyne TYRO3 21 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ncccn2)CC1 ZINC000880742944 EF On-Demand Anodyne FAAH 23 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ncccn2)CC1 ZINC000880742944 EF On-Demand Anodyne RBP4 45 33 Cc1ncc(CC(=O)NC[C@H](O)c2ccc(Cl)c(Cl)c2)o1 ZINC000880742950 EF On-Demand Anodyne ADRB2 36 40 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc(C3CC3)cc2F)on1 ZINC000880742951 EI On-Demand Anodyne KCNA5 18 44 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1ccc(C2CC2)cc1F ZINC000880742961 FH On-Demand Anodyne CACNA1I 50 34 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1ccc(C2CC2)cc1F ZINC000880742963 FH On-Demand Anodyne CACNA1I 50 34 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880742976 GI On-Demand Anodyne TNKS 51 32 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild CTRA_BOVIN 60 31 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild CTSG 41 31 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild CELA2A 49 31 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild LGMN 74 43 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild KLK5 41 41 C#C[C@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742983 GE On-Demand Mild Q9NAW4_PLAFA 41 47 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild CTRA_BOVIN 60 31 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild CTSG 41 31 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild CELA2A 49 31 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild LGMN 74 43 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild KLK5 41 41 C#C[C@@H](NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)C1CCOCC1 ZINC000880742984 GE On-Demand Mild Q9NAW4_PLAFA 41 47 CS(=O)(=O)C1CCC(C(=O)NNc2ccc(Cl)cn2)CC1 ZINC000880742987 ED On-Demand Reactive F10 31 44 CCCCN(CCO)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880743000 CG On-Demand Anodyne SOAT1 29 46 COc1ccc([C@@H](O)CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880743031 EH On-Demand Anodyne TRPV1 50 35 CCN1CC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743036 DG On-Demand Anodyne CCR3 55 37 CCN1CC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743036 DG On-Demand Anodyne CACNA1I 54 33 N#Cc1cccnc1NCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743038 EG On-Demand Mild ADRB1 41 33 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)c2ccccc2F)CC1 ZINC000880743040 GI On-Demand Anodyne EPHX2 38 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)c2ccccc2F)CC1 ZINC000880743040 GI On-Demand Anodyne CCR8 46 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743055 DE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743055 DE On-Demand Anodyne CTSK 15 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743055 DE On-Demand Anodyne POLG_HCV1 22 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743056 DE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743056 DE On-Demand Anodyne CTSK 15 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743056 DE On-Demand Anodyne POLG_HCV1 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743057 DE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743057 DE On-Demand Anodyne CTSK 15 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@]1(C)CC1(C)C ZINC000880743057 DE On-Demand Anodyne POLG_HCV1 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743058 DE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743058 DE On-Demand Anodyne CTSK 15 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@]1(C)CC1(C)C ZINC000880743058 DE On-Demand Anodyne POLG_HCV1 22 40 O=C(NCc1ccccc1CN1CCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880743061 GI On-Demand Anodyne TRPV1 42 35 CC(C)(C)NS(=O)(=O)CCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743065 FF On-Demand Anodyne TRPV1 56 36 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880743074 DG On-Demand Anodyne EPHX2 15 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880743075 DG On-Demand Anodyne EPHX2 15 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880743076 DG On-Demand Anodyne EPHX2 15 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880743077 DG On-Demand Anodyne EPHX2 15 40 COc1ccc2c(c1)CN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880743079 EI On-Demand Anodyne HDAC6 27 40 CS(=O)(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743080 ED On-Demand Anodyne RBP4 48 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880743081 GG On-Demand Anodyne RBP4 56 40 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743087 GF On-Demand Anodyne CACNA1H 53 35 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743108 FF On-Demand Anodyne EPHX2 17 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743108 FF On-Demand Anodyne CCR8 91 42 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743108 FF On-Demand Anodyne SFRP1 44 32 O=C(NCCNC(=O)c1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743120 EG On-Demand Anodyne DGAT1 29 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne GHRHR 52 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne P2RY12 183 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne CCKAR 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne AMY2 47 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne REN 48 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne FPR1 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne SFRP1 43 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743123 GF On-Demand Anodyne WNT3 41 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne GHRHR 52 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne P2RY12 183 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne PGC 50 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne CCKAR 22 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne AMY2 47 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne REN 48 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne FPR1 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne SFRP1 43 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](N(C)c2ccccc2)C1 ZINC000880743125 GF On-Demand Anodyne WNT3 41 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne GHRHR 52 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne P2RY12 183 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne PGC 50 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne CCKAR 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne AMY2 47 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne REN 48 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne FPR1 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne SFRP1 43 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743127 GF On-Demand Anodyne WNT3 41 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne GHRHR 52 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne P2RY12 183 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne PGC 50 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne CCKAR 22 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne AMY2 47 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne REN 48 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne FPR1 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne SFRP1 43 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](N(C)c2ccccc2)C1 ZINC000880743129 GF On-Demand Anodyne WNT3 41 33 NC(=O)[C@H](c1ccccc1)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743132 GG On-Demand Anodyne NPY2R 67 38 NC(=O)[C@H](c1ccccc1)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743132 GG On-Demand Anodyne RBP4 56 37 NC(=O)[C@@H](c1ccccc1)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743134 GG On-Demand Anodyne NPY2R 67 38 NC(=O)[C@@H](c1ccccc1)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743134 GG On-Demand Anodyne RBP4 56 37 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743146 DG On-Demand Anodyne TRPV1 42 35 O=C(NCc1ccc(C(=O)N2CCOCC2)cc1)Nc1ccc(C2CC2)cc1F ZINC000880743155 GG On-Demand Anodyne EPHX2 17 46 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743169 FG On-Demand Mild TRPV1 15 54 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743169 FG On-Demand Mild RBP4 24 41 Cc1coc(C(=O)NC[C@H]2CC(=O)N(C(C)(C)C)C2)c1 ZINC000880743181 CD On-Demand Anodyne CACNA1I 58 34 Cc1coc(C(=O)NC[C@@H]2CC(=O)N(C(C)(C)C)C2)c1 ZINC000880743182 CD On-Demand Anodyne CACNA1I 58 34 COCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743190 CF On-Demand Anodyne ADRA1D 17 41 COCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743190 CF On-Demand Anodyne ADRA1A 32 41 COCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743190 CF On-Demand Anodyne ADRA1B 18 41 CC(C)(C)N1C[C@@H](CNC(=O)c2cc3ccccc3cc2F)CC1=O ZINC000880743196 EG On-Demand Anodyne CACNA1I 52 35 CC(C)(C)N1C[C@H](CNC(=O)c2cc3ccccc3cc2F)CC1=O ZINC000880743197 EG On-Demand Anodyne CACNA1I 52 35 O=C(NCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743217 DG On-Demand Anodyne TBXAS1 44 44 O=C(NCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743217 DG On-Demand Anodyne HMOX2 44 31 O=C(NCCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743217 DG On-Demand Anodyne QPCT 38 51 CC(C)(C)N1C[C@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC1=O ZINC000880743225 FE On-Demand Anodyne CACNA1I 64 37 CC(C)(C)N1C[C@@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)CC1=O ZINC000880743226 FE On-Demand Anodyne CACNA1I 64 37 CC(C)(C)N1C[C@@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC1=O ZINC000880743227 FE On-Demand Anodyne CACNA1I 64 37 CC(C)(C)N1C[C@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)CC1=O ZINC000880743228 FE On-Demand Anodyne CACNA1I 64 37 CCN1CCC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743232 DG On-Demand Anodyne CCR3 41 40 CCN1CCC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743232 DG On-Demand Anodyne EPHX2 25 42 CCN1CCC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743233 DG On-Demand Anodyne CCR3 41 40 CCN1CCC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743233 DG On-Demand Anodyne EPHX2 25 42 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743270 FG On-Demand Anodyne TRPV1 42 41 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743270 FG On-Demand Anodyne PIK3CA 29 40 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743270 FG On-Demand Anodyne MTOR 44 40 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743270 FG On-Demand Anodyne PIK3CG 19 40 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743270 FG On-Demand Anodyne SCN10A 21 49 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880743271 FG On-Demand Anodyne MTOR 27 42 Cn1cnnc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743273 CE On-Demand Anodyne TRPV1 44 35 CCn1cc(NC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880743276 CH On-Demand Anodyne PANC 47 36 CN1CCC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743282 CF On-Demand Anodyne EPHX2 22 44 CCCCNC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743291 FH On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2[nH]c3ccccc3c2C1 ZINC000880743300 EJ On-Demand Anodyne SSTR4 52 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2[nH]c3ccccc3c2C1 ZINC000880743300 EJ On-Demand Anodyne SSTR5 42 35 O=C(COC1CC1)NC[C@@H](O)c1ccc(Cl)c(Cl)c1 ZINC000880743301 DE On-Demand Anodyne ADRB1 24 47 O=C(COC1CC1)NC[C@@H](O)c1ccc(Cl)c(Cl)c1 ZINC000880743301 DE On-Demand Anodyne ADRB3 28 44 O=C(COC1CC1)NC[C@H](O)c1ccc(Cl)c(Cl)c1 ZINC000880743302 DE On-Demand Anodyne ADRB1 24 47 O=C(COC1CC1)NC[C@H](O)c1ccc(Cl)c(Cl)c1 ZINC000880743302 DE On-Demand Anodyne ADRB3 28 44 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743306 EG On-Demand Anodyne ADRB2 26 44 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743306 EG On-Demand Anodyne ADRB1 63 50 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743306 EG On-Demand Anodyne ADRB3 34 40 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743306 EG On-Demand Anodyne PDS 41 33 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743307 EG On-Demand Anodyne ADRB2 26 44 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743307 EG On-Demand Anodyne ADRB1 63 50 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743307 EG On-Demand Anodyne ADRB3 34 40 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743307 EG On-Demand Anodyne PDS 41 33 COc1ncccc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743311 DG On-Demand Anodyne TRPV1 77 36 COc1ncccc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743311 DG On-Demand Anodyne P2RY1 37 47 O=C(NCc1nnc2n1CCC2)Nc1ccc(C2CC2)cc1F ZINC000880743313 DF On-Demand Anodyne TRPV1 46 33 C#C[C@@H](NC(=O)c1ccc(OC(F)F)c(Br)c1)C1CCOCC1 ZINC000880743342 GG On-Demand Mild PDE4D 17 41 C#C[C@H](NC(=O)c1ccc(OC(F)F)c(Br)c1)C1CCOCC1 ZINC000880743343 GG On-Demand Mild PDE4D 17 41 O=C(NCC1=CCCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880743354 CF On-Demand Anodyne GABRA1 18 55 O=C(NNc1ccc(Cl)cn1)c1ccc(CN2CCOCC2)o1 ZINC000880743382 ED On-Demand Reactive KLKB1 18 41 O=C(NNc1ccc(Cl)cn1)c1ccc(CN2CCOCC2)o1 ZINC000880743382 ED On-Demand Reactive F10 50 35 O=C(NNc1ccc(Cl)cn1)c1ccc(CN2CCOCC2)o1 ZINC000880743382 ED On-Demand Reactive DPOL_VZVD 24 42 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne ADRA1D 30 46 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne ADRA1A 53 46 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne ADRA1B 36 46 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne CCR3 46 45 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne CHRNA7 15 43 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne EPHX2 29 49 O=C(NCCCN1CCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880743387 DF On-Demand Anodyne MCHR1 26 43 C#C[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CCOCC1 ZINC000880743390 ED On-Demand Mild KCNQ2 44 34 C#C[C@@H](NC(=O)Cc1ccccc1N1CCCC1=O)C1CCOCC1 ZINC000880743391 ED On-Demand Mild KCNQ2 44 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne PGC 42 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne CTSK 19 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne REN 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne POLG_HCV1 25 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743399 EE On-Demand Anodyne FPR1 48 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne PGC 42 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne CTSK 19 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne REN 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne POLG_HCV1 25 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C1CC1 ZINC000880743400 EE On-Demand Anodyne FPR1 48 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne PGC 42 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne CTSK 19 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne REN 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne POLG_HCV1 25 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743401 EE On-Demand Anodyne FPR1 48 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne PGC 42 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne CTSK 19 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne REN 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne POLG_HCV1 25 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C(C)C)C1CC1 ZINC000880743402 EE On-Demand Anodyne FPR1 48 40 O=C(CN1CCCCS1(=O)=O)NNc1ccc(Cl)cn1 ZINC000880743426 DC On-Demand Reactive F10 32 41 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743433 GF On-Demand Anodyne ADRA1D 30 43 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743433 GF On-Demand Anodyne ADRA1A 52 43 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743433 GF On-Demand Anodyne ADRA1B 35 43 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743433 GF On-Demand Anodyne CCR3 43 43 NC(=O)C1CCN(CCCCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743433 GF On-Demand Anodyne MCHR1 28 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880743440 GI On-Demand Anodyne NPY2R 21 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880743440 GI On-Demand Anodyne RBP4 48 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880743440 GI On-Demand Anodyne L3MBTL3 53 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880743440 GI On-Demand Anodyne MAP3K12 29 40 O=C(NCC(=O)N1CCCCC1)Nc1ccc(C2CC2)cc1F ZINC000880743449 DF On-Demand Anodyne PRMT3 18 44 COCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743467 CG On-Demand Anodyne ADRA1D 15 41 COCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743467 CG On-Demand Anodyne ADRA1A 30 41 COCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880743467 CG On-Demand Anodyne ADRA1B 17 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCc2nc(O)ccc21 ZINC000880743468 EI On-Demand Anodyne TRPV1 20 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCc2nc(O)ccc21 ZINC000880743469 EI On-Demand Anodyne TRPV1 20 41 O=C(NCC(F)(F)F)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743470 GH On-Demand Anodyne RBP4 40 36 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1ccc(C2CC2)cc1F ZINC000880743482 EH On-Demand Anodyne PANC 51 36 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1ccc(C2CC2)cc1F ZINC000880743483 EH On-Demand Anodyne PANC 51 36 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(C2CC2)cc1F ZINC000880743486 FG On-Demand Anodyne MTOR 16 40 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc(C2CC2)cc1F ZINC000880743486 FG On-Demand Anodyne NAMPT 27 41 CNC(=O)CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880743488 EF On-Demand Anodyne HCN1 52 32 CNC(=O)CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880743488 EF On-Demand Anodyne HCN4 50 32 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2cscn2)CC1 ZINC000880743492 FH On-Demand Anodyne SCN5A 42 36 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880743498 GI On-Demand Anodyne EPHX2 48 52 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880743498 GI On-Demand Anodyne L3MBTL3 44 34 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880743499 FH On-Demand Anodyne EPHX2 35 41 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743506 GI On-Demand Anodyne EPHX2 16 41 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743506 GI On-Demand Anodyne ASAH1 60 36 O=C(CNC(=O)Nc1ccc(C2CC2)cc1F)NCc1ccccc1 ZINC000880743516 EG On-Demand Anodyne TRPV1 15 43 O=C(CNC(=O)Nc1ccc(C2CC2)cc1F)NCc1ccccc1 ZINC000880743516 EG On-Demand Anodyne CA5B 20 40 O=C(CNC(=O)Nc1ccc(C2CC2)cc1F)NCc1ccccc1 ZINC000880743516 EG On-Demand Anodyne CA5A 23 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC2CC2)CC1 ZINC000880743519 EH On-Demand Anodyne SIGMAR1 18 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC2CC2)CC1 ZINC000880743519 EH On-Demand Anodyne CCR3 40 39 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC2CC2)CC1 ZINC000880743519 EH On-Demand Anodyne EPHX2 41 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC2CC2)CC1 ZINC000880743519 EH On-Demand Anodyne CXCR3 19 48 CS(=O)(=O)Nc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880743521 GG On-Demand Anodyne TRPV1 105 60 O=C(NCc1ccc(Cl)nc1)Nc1ccc(C2CC2)cc1F ZINC000880743531 DI On-Demand Anodyne NAMPT 15 46 O=C(NCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743534 CG On-Demand Anodyne TRPV1 23 40 O=C(NCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743534 CG On-Demand Anodyne CHRNA7 40 38 O=C(NCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743534 CG On-Demand Anodyne ROCK2 19 45 O=C(NCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743534 CG On-Demand Anodyne NAMPT 81 48 O=C(Nc1ccc(C2CC2)cc1F)NC1CC1 ZINC000880743535 BF On-Demand Anodyne EPHX2 47 52 CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743538 CE On-Demand Anodyne RBP4 40 36 Cc1cnc(Cl)c(C(=O)NC[C@H]2CC(=O)N(C(C)(C)C)C2)c1 ZINC000880743554 DE On-Demand Anodyne CACNA1I 61 35 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC(=O)N(C(C)(C)C)C2)c1 ZINC000880743555 DE On-Demand Anodyne CACNA1I 61 35 O=C(NCc1ccncc1)Nc1ccc(C2CC2)cc1F ZINC000880743561 CG On-Demand Anodyne TRPV1 21 41 O=C(NCc1ccncc1)Nc1ccc(C2CC2)cc1F ZINC000880743561 CG On-Demand Anodyne FLT1 20 41 O=C(NCc1ccncc1)Nc1ccc(C2CC2)cc1F ZINC000880743561 CG On-Demand Anodyne NAMPT 42 34 CC(C)(C)N1C[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)CC1=O ZINC000880743577 FD On-Demand Anodyne CACNA1I 58 37 CC(C)(C)N1C[C@@H](CNC(=O)c2ccc(CN3CCOCC3)o2)CC1=O ZINC000880743578 FD On-Demand Anodyne CACNA1I 58 37 C#C[C@@H](NC(=O)c1cc2ccccc2cc1F)C1CCOCC1 ZINC000880743579 DG On-Demand Mild PYGL 16 43 C#C[C@H](NC(=O)c1cc2ccccc2cc1F)C1CCOCC1 ZINC000880743580 DG On-Demand Mild PYGL 16 43 CCOC(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743590 EG On-Demand Anodyne CACNA1H 46 33 CCOC(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743590 EG On-Demand Anodyne P2RY12 42 36 O=C(NC[C@H](O)c1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743629 DH On-Demand Anodyne TRPV1 15 41 O=C(NC[C@@H](O)c1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880743630 DH On-Demand Anodyne TRPV1 15 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880743636 EJ On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](C(F)(F)F)C1 ZINC000880743637 EJ On-Demand Anodyne RBP4 54 36 CN(c1ccccc1)[C@H]1CCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880743641 DF On-Demand Anodyne SFRP1 43 38 CN(c1ccccc1)[C@@H]1CCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880743642 DF On-Demand Anodyne SFRP1 43 38 O=C(NCCn1ccnc1)Nc1ccc(C2CC2)cc1F ZINC000880743702 CF On-Demand Anodyne QPCT 31 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2ccccc2C1 ZINC000880743703 DI On-Demand Anodyne RBP4 43 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2ccccc2C1 ZINC000880743703 DI On-Demand Anodyne TRPM8 33 44 CC(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743717 DE On-Demand Anodyne RBP4 41 36 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743732 GI On-Demand Anodyne CCR1 20 40 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743732 GI On-Demand Anodyne EPHX2 38 45 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743732 GI On-Demand Anodyne RBP4 44 37 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743742 FF On-Demand Anodyne NQO2 24 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743742 FF On-Demand Anodyne MTNR1A 33 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743742 FF On-Demand Anodyne MTNR1B 32 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743742 FF On-Demand Anodyne MMP3 16 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743745 FF On-Demand Anodyne NQO2 24 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743745 FF On-Demand Anodyne MTNR1A 33 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743745 FF On-Demand Anodyne MTNR1B 32 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1)C2 ZINC000880743745 FF On-Demand Anodyne MMP3 16 41 C#C[C@@H](NC(=O)CCCCc1ccc(OC)c(OC)c1)C1CCOCC1 ZINC000880743746 FF On-Demand Mild MMP2 44 30 C#C[C@H](NC(=O)CCCCc1ccc(OC)c(OC)c1)C1CCOCC1 ZINC000880743747 FF On-Demand Mild MMP2 44 30 C#C[C@@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1CCOCC1 ZINC000880743756 EG On-Demand Mild PDE4D 20 42 C#C[C@H](NC(=O)c1ccc(OC(F)F)c(Cl)c1)C1CCOCC1 ZINC000880743757 EG On-Demand Mild PDE4D 20 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1 ZINC000880743782 GD On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1 ZINC000880743783 GD On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC(=O)N(C(C)(C)C)C1 ZINC000880743784 GD On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CC(=O)N(C(C)(C)C)C1 ZINC000880743785 GD On-Demand Anodyne PAPA1_CARPA 37 43 CC(C)(C)N1C[C@H](CNC(=O)COC2CC2)CC1=O ZINC000880743798 CC On-Demand Anodyne CACNA1I 42 33 CC(C)(C)N1C[C@@H](CNC(=O)COC2CC2)CC1=O ZINC000880743799 CC On-Demand Anodyne CACNA1I 42 33 CC(C)(C)N1C[C@@H](CNC(=O)c2cnc(CC3CC3)s2)CC1=O ZINC000880743803 EE On-Demand Anodyne CACNA1I 43 33 CC(C)(C)N1C[C@H](CNC(=O)c2cnc(CC3CC3)s2)CC1=O ZINC000880743804 EE On-Demand Anodyne CACNA1I 43 33 CCN(Cc1ccncc1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880743832 DI On-Demand Anodyne SOAT1 17 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2=CCCC2)N1Cc1ccccc1 ZINC000880743837 ED On-Demand Anodyne P2RX7 25 40 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2=CCCC2)N1Cc1ccccc1 ZINC000880743837 ED On-Demand Anodyne TMPRSS11D 54 35 O=C(NCCCN1CCCCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880743862 EH On-Demand Anodyne CCR3 37 40 O=C(NCCCN1CCCCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880743862 EH On-Demand Anodyne TYRO3 20 40 O=C(NCCCN1C(=O)NC2(CCCC2)C1=O)Nc1ccc(C2CC2)cc1F ZINC000880743867 GG On-Demand Anodyne ADRA1D 24 40 O=C(NCCCN1C(=O)NC2(CCCC2)C1=O)Nc1ccc(C2CC2)cc1F ZINC000880743867 GG On-Demand Anodyne ADRA1A 42 40 O=C(NCCCN1C(=O)NC2(CCCC2)C1=O)Nc1ccc(C2CC2)cc1F ZINC000880743867 GG On-Demand Anodyne ADRA1B 26 40 CC(C)(C)N1C[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880743887 FG On-Demand Anodyne PDE4D 15 42 CC(C)(C)N1C[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880743887 FG On-Demand Anodyne CACNA1I 73 45 CC(C)(C)N1C[C@@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880743888 FG On-Demand Anodyne PDE4D 15 42 CC(C)(C)N1C[C@@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)CC1=O ZINC000880743888 FG On-Demand Anodyne CACNA1I 73 45 CN(c1ccccc1)[C@H]1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880743891 FF On-Demand Anodyne L3MBTL3 50 38 CN(c1ccccc1)[C@@H]1CCN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880743892 FF On-Demand Anodyne L3MBTL3 50 38 CN(c1ccccc1)[C@H]1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880743893 FF On-Demand Anodyne L3MBTL3 50 38 CN(c1ccccc1)[C@@H]1CCN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880743894 FF On-Demand Anodyne L3MBTL3 50 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccco2)CC1 ZINC000880743904 FG On-Demand Anodyne RBP4 33 44 O=C(NCc1cccs1)Nc1ccc(C2CC2)cc1F ZINC000880743926 CI On-Demand Anodyne CA5B 25 45 O=C(NCc1cccs1)Nc1ccc(C2CC2)cc1F ZINC000880743926 CI On-Demand Anodyne CA5A 29 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2nnc3ccccn23)CC1 ZINC000880743932 GI On-Demand Anodyne RBP4 51 38 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743956 FE On-Demand Anodyne ADRA1D 24 40 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743956 FE On-Demand Anodyne SLC6A1 107 35 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743956 FE On-Demand Anodyne ADRA1A 45 40 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743956 FE On-Demand Anodyne ADRA1B 28 41 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743956 FE On-Demand Anodyne CCR3 43 44 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743957 FE On-Demand Anodyne ADRA1D 24 40 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743957 FE On-Demand Anodyne SLC6A1 107 35 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743957 FE On-Demand Anodyne ADRA1A 45 40 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743957 FE On-Demand Anodyne ADRA1B 28 41 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880743957 FE On-Demand Anodyne CCR3 43 44 Cc1noc(C2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)n1 ZINC000880743959 EH On-Demand Anodyne SMO 41 49 Cc1noc(C2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)n1 ZINC000880743959 EH On-Demand Anodyne ETHR 63 38 CCOCCN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743960 EF On-Demand Anodyne ADRA1A 42 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](N2CCCC2)C1 ZINC000880743961 DG On-Demand Anodyne L3MBTL3 93 45 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](N2CCCC2)C1 ZINC000880743962 DG On-Demand Anodyne L3MBTL3 93 45 CN1CCC(CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743968 DG On-Demand Anodyne HTR1F 47 33 CN1CCC(CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743968 DG On-Demand Anodyne CCR3 42 37 CN1CCC(CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880743968 DG On-Demand Anodyne CACNA1I 59 35 O=C1CC[C@H](c2ccc(C(=O)NCCN3C[C@@H]4CCCCN4C3=O)cc2)N1 ZINC000880743972 FD On-Demand Anodyne PLD1 66 38 O=C1CC[C@H](c2ccc(C(=O)NCCN3C[C@@H]4CCCCN4C3=O)cc2)N1 ZINC000880743972 FD On-Demand Anodyne PLD2 75 38 O=C1CC[C@H](c2ccc(C(=O)NCCN3C[C@H]4CCCCN4C3=O)cc2)N1 ZINC000880743973 FD On-Demand Anodyne PLD1 66 38 O=C1CC[C@H](c2ccc(C(=O)NCCN3C[C@H]4CCCCN4C3=O)cc2)N1 ZINC000880743973 FD On-Demand Anodyne PLD2 75 38 O=C1CC[C@@H](c2ccc(C(=O)NCCN3C[C@@H]4CCCCN4C3=O)cc2)N1 ZINC000880743974 FD On-Demand Anodyne PLD1 66 38 O=C1CC[C@@H](c2ccc(C(=O)NCCN3C[C@@H]4CCCCN4C3=O)cc2)N1 ZINC000880743974 FD On-Demand Anodyne PLD2 75 38 O=C1CC[C@@H](c2ccc(C(=O)NCCN3C[C@H]4CCCCN4C3=O)cc2)N1 ZINC000880743975 FD On-Demand Anodyne PLD1 66 38 O=C1CC[C@@H](c2ccc(C(=O)NCCN3C[C@H]4CCCCN4C3=O)cc2)N1 ZINC000880743975 FD On-Demand Anodyne PLD2 75 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1c2ccccc2C[C@H]1O ZINC000880743990 EG On-Demand Anodyne PLM1_PLAFA 46 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1c2ccccc2C[C@H]1O ZINC000880743990 EG On-Demand Anodyne PLM2_PLAFA 30 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880743991 EG On-Demand Anodyne PLM1_PLAFA 46 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880743991 EG On-Demand Anodyne PLM2_PLAFA 30 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880743995 FG On-Demand Anodyne RBP4 65 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H]2COC[C@H]2C1 ZINC000880743996 FG On-Demand Anodyne RBP4 65 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H]2COC[C@@H]2C1 ZINC000880743997 FG On-Demand Anodyne RBP4 65 37 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@@H]2COC[C@H]2C1 ZINC000880743998 FG On-Demand Anodyne RBP4 65 37 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880744007 GH On-Demand Anodyne EPHX2 45 58 CCOCCN(CC)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744008 CH On-Demand Anodyne SOAT1 19 41 Cc1ncc(CN2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)s1 ZINC000880744020 FH On-Demand Anodyne MGEA5 38 47 O=C(NCCS(=O)(=O)c1ccccc1)Nc1ccc(C2CC2)cc1F ZINC000880744025 FG On-Demand Anodyne TRPV1 42 35 O=C(NCCc1ccc(O)cc1)Nc1ccc(C2CC2)cc1F ZINC000880744027 DH On-Demand Anodyne TRPV1 15 44 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CCO)CC1 ZINC000880744052 DE On-Demand Anodyne ADRA1B 15 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CCO)CC1 ZINC000880744052 DE On-Demand Anodyne SIGMAR1 15 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CCO)CC1 ZINC000880744052 DE On-Demand Anodyne CCR3 37 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CCO)CC1 ZINC000880744052 DE On-Demand Anodyne SLC6A5 16 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CCO)CC1 ZINC000880744052 DE On-Demand Anodyne EPHX2 34 42 O=C(NCCCN1C(=O)CNC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744056 ED On-Demand Anodyne ADRA1D 20 40 O=C(NCCCN1C(=O)CNC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744056 ED On-Demand Anodyne ADRA1A 36 40 O=C(NCCCN1C(=O)CNC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744056 ED On-Demand Anodyne ADRA1B 23 40 CN(CCN1CCOCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744060 DE On-Demand Anodyne CASR 51 38 CN(CCN1CCOCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744060 DE On-Demand Anodyne EPHX2 20 42 COc1ccnc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)n1 ZINC000880744100 FF On-Demand Anodyne FAAH 22 41 N#Cc1ccc(N2CCC(NC(=O)Nc3ccc(C4CC4)cc3F)CC2)nc1 ZINC000880744121 GH On-Demand Mild FASN 31 43 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744126 FE On-Demand Anodyne EPHX2 29 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCSCC1 ZINC000880744136 CH On-Demand Anodyne EPHX2 28 48 N#CCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744141 DF On-Demand Mild EPHX2 29 40 COc1ccc(-n2c(C)cc(C(=O)Nc3ccc(N4CCOCC4)cn3)c2C)cc1 ZINC000880744154 HH On-Demand Clean F10 51 35 COc1ccc(-n2c(C)cc(C(=O)Nc3ccc(N4CCOCC4)cn3)c2C)cc1 ZINC000880744154 HH On-Demand Clean EPHB4 54 36 COc1ccc(-n2c(C)cc(C(=O)Nc3ccc(N4CCOCC4)cn3)c2C)cc1 ZINC000880744154 HH On-Demand Clean LUCI_LUCLA 18 43 COc1ccc(-n2c(C)cc(C(=O)Nc3ccc(N4CCOCC4)cn3)c2C)cc1 ZINC000880744154 HH On-Demand Clean STAT6 53 35 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne CELA1 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne GRIN2B 24 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne PREP 62 50 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne TGM2 26 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne KLK5 32 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744161 GE On-Demand Anodyne F13A1 37 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne CELA1 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne GRIN2B 24 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne PREP 62 50 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne TGM2 26 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne KLK5 32 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744162 GE On-Demand Anodyne F13A1 37 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne CELA1 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne GRIN2B 24 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne PREP 62 50 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne TGM2 26 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne KLK5 32 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744163 GE On-Demand Anodyne F13A1 37 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne CELA1 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne GRIN2B 24 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne PREP 62 50 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne TGM2 26 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne KLK5 32 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744164 GE On-Demand Anodyne F13A1 37 41 CN(C)CCn1cc(NC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880744175 EG On-Demand Anodyne PANC 41 34 C[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744176 CH On-Demand Anodyne CSF1R 18 42 C[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744176 CH On-Demand Anodyne RBP4 47 34 C[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744176 CH On-Demand Anodyne TRPC6 28 40 C[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744177 CH On-Demand Anodyne CSF1R 18 42 C[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744177 CH On-Demand Anodyne RBP4 47 34 C[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744177 CH On-Demand Anodyne TRPC6 28 40 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744181 GG On-Demand Anodyne TRPV1 48 43 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744181 GG On-Demand Anodyne P2RY1 17 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880744187 EG On-Demand Anodyne CCR3 22 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880744188 EG On-Demand Anodyne CCR3 22 42 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744189 GD On-Demand Anodyne ADRA1A 40 39 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744189 GD On-Demand Anodyne TRPV1 62 37 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744189 GD On-Demand Anodyne CCR3 46 42 CS(=O)(=O)N1CCN(CCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744189 GD On-Demand Anodyne MCHR1 19 41 CC(C)(C(=O)N1CC[C@@H]2COC[C@H]2C1)c1ccc(C(F)(F)F)cc1 ZINC000880744198 EG On-Demand Anodyne EPHX2 30 41 CC(C)(C(=O)N1CC[C@@H]2COC[C@@H]2C1)c1ccc(C(F)(F)F)cc1 ZINC000880744199 EG On-Demand Anodyne EPHX2 30 41 CC(C)(C(=O)N1CC[C@H]2COC[C@H]2C1)c1ccc(C(F)(F)F)cc1 ZINC000880744200 EG On-Demand Anodyne EPHX2 30 41 CC(C)(C(=O)N1CC[C@H]2COC[C@@H]2C1)c1ccc(C(F)(F)F)cc1 ZINC000880744201 EG On-Demand Anodyne EPHX2 30 41 O=C(CNC(=O)Nc1ccc(C2CC2)cc1F)NC1CCCCC1 ZINC000880744202 EG On-Demand Anodyne EPHX2 17 48 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744209 EG On-Demand Anodyne L3MBTL3 42 33 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744210 EG On-Demand Anodyne L3MBTL3 42 33 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744211 EG On-Demand Anodyne L3MBTL3 42 33 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744212 EG On-Demand Anodyne L3MBTL3 42 33 CC(C)(C(=O)N1CC[C@@H]2COC[C@@H]2C1)c1ccc(F)cc1F ZINC000880744219 DF On-Demand Anodyne PRCP 40 36 CC(C)(C(=O)N1CC[C@H]2COC[C@H]2C1)c1ccc(F)cc1F ZINC000880744220 DF On-Demand Anodyne PRCP 40 36 CC(C)(C(=O)N1CC[C@H]2COC[C@@H]2C1)c1ccc(F)cc1F ZINC000880744221 DF On-Demand Anodyne PRCP 40 36 CC(C)(C(=O)N1CC[C@@H]2COC[C@H]2C1)c1ccc(F)cc1F ZINC000880744222 DF On-Demand Anodyne PRCP 40 36 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H]4COC[C@H]4C3)cc2)N1 ZINC000880744239 DD On-Demand Anodyne L3MBTL3 52 40 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H]4COC[C@H]4C3)cc2)N1 ZINC000880744240 DD On-Demand Anodyne L3MBTL3 52 40 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H]4COC[C@@H]4C3)cc2)N1 ZINC000880744241 DD On-Demand Anodyne L3MBTL3 52 40 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H]4COC[C@@H]4C3)cc2)N1 ZINC000880744242 DD On-Demand Anodyne L3MBTL3 52 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@H](CO)Cc1ccccc1 ZINC000880744254 EG On-Demand Anodyne MME 59 37 O=C(Nc1ccc(C2CC2)cc1F)N[C@H](CO)Cc1ccccc1 ZINC000880744254 EG On-Demand Anodyne ANPEP 49 31 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H](CO)Cc1ccccc1 ZINC000880744255 EG On-Demand Anodyne MME 59 37 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H](CO)Cc1ccccc1 ZINC000880744255 EG On-Demand Anodyne ANPEP 49 31 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne ADRA1D 24 42 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne ADRA1A 39 42 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne ADRA1B 27 42 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne CCR3 38 45 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne EPHX2 37 40 COCCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744259 EF On-Demand Anodyne MCHR1 41 41 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744291 FE On-Demand Anodyne RBP4 44 35 Cn1cc(CN2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)cn1 ZINC000880744307 FF On-Demand Anodyne MCHR1 25 42 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne ACE 42 37 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne OPRM1 49 41 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne OPRD1 37 40 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne MME 77 37 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne ANPEP 45 34 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne TACR1 22 48 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne FCER2 72 41 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne F2R 40 32 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne NPFFR2 73 37 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne TIMP3 73 34 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne HLA-DRB1 58 36 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne MMP11 40 31 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne MMP9 16 50 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne ACE2 49 34 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne MMP1 15 50 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne BLA1_STEMA 59 38 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne QRFPR 50 36 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744318 EF On-Demand Anodyne NPFFR1 74 40 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne ACE 42 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne OPRM1 49 41 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne OPRD1 37 40 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne MME 77 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne ANPEP 45 34 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne TACR1 22 48 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne FCER2 72 41 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne F2R 40 32 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne NPFFR2 73 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne TIMP3 73 34 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne HLA-DRB1 58 36 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne MMP11 40 31 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne MMP9 16 50 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne ACE2 49 34 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne MMP1 15 50 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne BLA1_STEMA 59 38 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne QRFPR 50 36 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744319 EF On-Demand Anodyne NPFFR1 74 40 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744330 GI On-Demand Anodyne EPHX2 35 53 CCOC(=O)C1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744331 EH On-Demand Anodyne EPHX2 40 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](C2OCCO2)C1 ZINC000880744333 EG On-Demand Anodyne RBP4 46 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](C2OCCO2)C1 ZINC000880744334 EG On-Demand Anodyne RBP4 46 34 CC[C@@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744337 CI On-Demand Anodyne CCR1 15 45 CC[C@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744338 CI On-Demand Anodyne CCR1 15 45 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744354 GI On-Demand Anodyne ACACB 15 42 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744354 GI On-Demand Anodyne CACNA1I 54 34 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744354 GI On-Demand Anodyne GPR119 23 41 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744355 GI On-Demand Anodyne ACACB 15 42 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744355 GI On-Demand Anodyne CACNA1I 54 34 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744355 GI On-Demand Anodyne GPR119 23 41 O=C(Nc1cnn(CCO)c1)Nc1ccc(C2CC2)cc1F ZINC000880744362 DF On-Demand Anodyne PANC 41 34 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880744375 FH On-Demand Anodyne EPHX2 40 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880744375 FH On-Demand Anodyne CXCR3 19 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880744375 FH On-Demand Anodyne MCHR1 15 40 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC(F)(F)F)CC1 ZINC000880744375 FH On-Demand Anodyne HPGDS 39 42 O=C(Nc1ccc(C2CC2)cc1F)N1Cc2ccccc2C1 ZINC000880744376 CI On-Demand Anodyne RBP4 48 36 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744384 GF On-Demand Anodyne RBP4 41 36 CC(C)(C)CN(CCCO)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744408 DH On-Demand Anodyne SOAT1 22 45 CNC(=O)CC1(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)CCCCC1 ZINC000880744424 FF On-Demand Anodyne MPO 32 41 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744447 GH On-Demand Anodyne CA2 18 43 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744447 GH On-Demand Anodyne CA1 17 40 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744447 GH On-Demand Anodyne CA4 24 43 CN(C(=O)Nc1ccc(C2CC2)cc1F)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880744450 GI On-Demand Anodyne L3MBTL3 42 36 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744452 FH On-Demand Anodyne CACNA1H 43 33 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(CC(F)F)CC1 ZINC000880744455 EH On-Demand Anodyne EPHX2 40 42 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744458 CF On-Demand Anodyne CCR1 25 40 CN(C)[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744458 CF On-Demand Anodyne RBP4 48 35 O=C(NCCCN1CCCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744476 EG On-Demand Anodyne CCR3 38 41 O=C(NCCCN1CCCCC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744476 EG On-Demand Anodyne TYRO3 20 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CCC1 ZINC000880744483 BG On-Demand Anodyne EPHX2 44 57 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744488 GJ On-Demand Anodyne CCR1 17 42 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744488 GJ On-Demand Anodyne CCR3 22 45 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744488 GJ On-Demand Anodyne EPHX2 64 52 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744488 GJ On-Demand Anodyne RBP4 51 38 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744488 GJ On-Demand Anodyne DGAT1 28 40 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744493 EG On-Demand Anodyne EPHX2 28 42 COC(=O)N1CCC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744494 EG On-Demand Anodyne EPHX2 28 42 O=C(NCc1cccc(CO)c1)Nc1ccc(C2CC2)cc1F ZINC000880744500 DH On-Demand Anodyne ROCK2 19 44 C[C@@H](Cn1cncn1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744503 DF On-Demand Anodyne HIS3 77 36 O=C(NCc1cccc(C(=O)N2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880744518 GG On-Demand Anodyne EPHX2 17 44 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744527 EH On-Demand Anodyne ACE 21 40 C[C@H](O)c1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880744559 EI On-Demand Anodyne TRPV1 99 42 CN1CCC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880744564 DG On-Demand Anodyne CCR3 49 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCCC[C@H]2C1 ZINC000880744576 DG On-Demand Anodyne HRH3 17 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCCC[C@H]2C1 ZINC000880744576 DG On-Demand Anodyne L3MBTL3 65 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCCC[C@@H]2C1 ZINC000880744577 DG On-Demand Anodyne HRH3 17 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCCC[C@@H]2C1 ZINC000880744577 DG On-Demand Anodyne L3MBTL3 65 38 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccc(C2CC2)cc1F ZINC000880744619 GH On-Demand Anodyne SIGMAR1 23 43 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccc(C2CC2)cc1F ZINC000880744619 GH On-Demand Anodyne CCR3 48 38 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccc(C2CC2)cc1F ZINC000880744619 GH On-Demand Anodyne MCHR1 41 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880744632 EF On-Demand Anodyne SLC18A3 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880744633 EF On-Demand Anodyne SLC18A3 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880744634 EF On-Demand Anodyne SLC18A3 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880744635 EF On-Demand Anodyne SLC18A3 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(CC(F)F)CC1 ZINC000880744644 EG On-Demand Anodyne CACNA1H 50 37 CS(=O)(=O)c1ccc(OCCNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880744688 GG On-Demand Anodyne TRPV1 96 36 CCN(Cc1ccc(C(=O)N(C)C)cc1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744690 GI On-Demand Anodyne GIPR 43 33 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](N2CCCCC2)C1 ZINC000880744698 EH On-Demand Anodyne L3MBTL3 91 44 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](N2CCCCC2)C1 ZINC000880744699 EH On-Demand Anodyne L3MBTL3 91 44 CCOC(=O)N1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744712 EG On-Demand Anodyne CACNA1H 40 32 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(Cc2cscn2)CC1 ZINC000880744727 FH On-Demand Anodyne SCN5A 41 35 O=C(NCCN1C[C@H]2CCCCN2C1=O)c1cnc2cc[nH]c2c1 ZINC000880744728 ED On-Demand Anodyne PLD1 60 44 O=C(NCCN1C[C@H]2CCCCN2C1=O)c1cnc2cc[nH]c2c1 ZINC000880744728 ED On-Demand Anodyne PLD2 69 44 O=C(NCCN1C[C@@H]2CCCCN2C1=O)c1cnc2cc[nH]c2c1 ZINC000880744729 ED On-Demand Anodyne PLD1 60 44 O=C(NCCN1C[C@@H]2CCCCN2C1=O)c1cnc2cc[nH]c2c1 ZINC000880744729 ED On-Demand Anodyne PLD2 69 44 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CCN2CCOCC2)CC1 ZINC000880744734 GH On-Demand Anodyne EPHX2 29 42 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744738 GF On-Demand Anodyne HDAC8 15 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744738 GF On-Demand Anodyne MTNR1A 18 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744738 GF On-Demand Anodyne MTNR1B 21 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744738 GF On-Demand Anodyne ROCK2 17 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744739 GF On-Demand Anodyne HDAC8 15 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744739 GF On-Demand Anodyne MTNR1A 18 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744739 GF On-Demand Anodyne MTNR1B 21 45 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc([C@H]3CC(=O)NC(=O)N3)cc1)C2 ZINC000880744739 GF On-Demand Anodyne ROCK2 17 41 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@@H]2COC[C@H]2C1 ZINC000880744761 GG On-Demand Anodyne L3MBTL3 41 38 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880744762 GG On-Demand Anodyne L3MBTL3 41 38 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@H]2COC[C@@H]2C1 ZINC000880744763 GG On-Demand Anodyne L3MBTL3 41 38 O=C(c1ccc(OC(F)F)c(Br)c1)N1CC[C@H]2COC[C@H]2C1 ZINC000880744764 GG On-Demand Anodyne L3MBTL3 41 38 CO[C@@H](C)CCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744771 CG On-Demand Anodyne TRPV1 46 34 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744888 EG On-Demand Anodyne RBP4 41 37 COC(=O)C1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744898 EH On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN(CC2CC2)C1 ZINC000880744904 DG On-Demand Anodyne CCR3 46 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN(CC2CC2)C1 ZINC000880744904 DG On-Demand Anodyne CCR2 19 44 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880744905 DG On-Demand Anodyne CCR3 46 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880744905 DG On-Demand Anodyne CCR2 19 44 CCCN(CC)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880744908 CH On-Demand Anodyne SOAT1 24 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCC[C@H]2C1 ZINC000880744913 DG On-Demand Anodyne L3MBTL3 47 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCN2CCC[C@@H]2C1 ZINC000880744914 DG On-Demand Anodyne L3MBTL3 47 36 O=C(NCCCN1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744925 DF On-Demand Anodyne ADRA1D 22 44 O=C(NCCCN1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744925 DF On-Demand Anodyne ADRA1A 40 44 O=C(NCCCN1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880744925 DF On-Demand Anodyne ADRA1B 25 44 C=CCN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744926 DG On-Demand Mild EPHX2 28 40 C=C(C)CN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744930 EH On-Demand Mild EPHX2 30 40 C=C(C)CN1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880744930 EH On-Demand Mild CXCR3 19 40 COC(=O)CCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744944 DH On-Demand Anodyne EPHX2 21 47 CN(C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)S(C)(=O)=O ZINC000880744953 FF On-Demand Anodyne RBP4 45 39 COCCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744956 CH On-Demand Anodyne ADRA1A 27 40 COCCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744956 CH On-Demand Anodyne ADRA1B 15 40 COCCCCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880744956 CH On-Demand Anodyne EPHX2 15 45 O=C(NC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)C1CCCCC1 ZINC000880744982 GI On-Demand Anodyne EPHX2 35 47 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2cccnn2)CC1 ZINC000880745003 EF On-Demand Anodyne FAAH 23 42 C[C@@H](Cc1ccncc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745023 DH On-Demand Anodyne TRPV1 41 34 C[C@@H](Cc1ccncc1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745023 DH On-Demand Anodyne CCR1 16 40 Cn1nnc(C(=O)NCCc2nsc3ccccc23)n1 ZINC000880745028 CC On-Demand Anodyne HTR1A 17 43 Cn1nnc(C(=O)NCCc2nsc3ccccc23)n1 ZINC000880745028 CC On-Demand Anodyne DRD2 21 43 O=C(NC[C@H]1CN(Cc2ccccc2)CC12CCC2)[C@H]1CCc2nncn2CC1 ZINC000880745036 GF On-Demand Anodyne CACNA1G 23 43 O=C(NC[C@H]1CN(Cc2ccccc2)CC12CCC2)[C@@H]1CCc2nncn2CC1 ZINC000880745038 GF On-Demand Anodyne CACNA1G 23 43 O=C(NC[C@@H]1CN(Cc2ccccc2)CC12CCC2)[C@H]1CCc2nncn2CC1 ZINC000880745039 GF On-Demand Anodyne CACNA1G 23 43 O=C(NC[C@@H]1CN(Cc2ccccc2)CC12CCC2)[C@@H]1CCc2nncn2CC1 ZINC000880745041 GF On-Demand Anodyne CACNA1G 23 43 CC(C)n1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)n1 ZINC000880745043 DH On-Demand Anodyne TRPV1 53 36 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880745069 DF On-Demand Anodyne EPHX2 36 50 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880745070 DF On-Demand Anodyne EPHX2 36 50 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745072 DG On-Demand Anodyne CCR1 17 44 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745073 DG On-Demand Anodyne CCR1 17 44 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745077 DE On-Demand Anodyne LGMN 56 34 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745096 EF On-Demand Anodyne CACNA1H 52 36 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745097 EF On-Demand Anodyne CACNA1H 52 36 O=C(NCC1SCCS1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880745102 DE On-Demand Anodyne GABRA1 18 51 O=C(NCC1SCCS1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880745102 DE On-Demand Anodyne MPO 55 35 O=C(NCC1SCCS1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880745102 DE On-Demand Anodyne GABRA2 16 51 O=C(CC[C@H]1CCc2ccccc21)NCC1SCCS1 ZINC000880745112 DG On-Demand Anodyne MTNR1A 20 46 O=C(CC[C@H]1CCc2ccccc21)NCC1SCCS1 ZINC000880745112 DG On-Demand Anodyne MTNR1B 22 46 O=C(CC[C@@H]1CCc2ccccc21)NCC1SCCS1 ZINC000880745113 DG On-Demand Anodyne MTNR1A 20 46 O=C(CC[C@@H]1CCc2ccccc21)NCC1SCCS1 ZINC000880745113 DG On-Demand Anodyne MTNR1B 22 46 CC(C)(C(N)=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745114 EE On-Demand Anodyne RBP4 43 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCC2)C1 ZINC000880745171 CI On-Demand Anodyne EPHX2 27 42 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880745178 GF On-Demand Anodyne EPHX2 36 54 O=C(Nc1ccc(C2CC2)cc1F)N1CCOC2(CCOCC2)C1 ZINC000880745203 EG On-Demand Anodyne EPHX2 18 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C2CCCC2)CC1 ZINC000880745226 EI On-Demand Anodyne EPHX2 35 48 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880745339 DG On-Demand Anodyne CACNA1H 47 37 O=C(NC[C@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)C1)c1ccccc1 ZINC000880745368 GI On-Demand Anodyne RBP4 45 34 O=C(NC[C@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)C1)c1ccccc1 ZINC000880745368 GI On-Demand Anodyne CACNA1I 52 33 C[C@@H](CCS(C)(=O)=O)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745387 EF On-Demand Anodyne TRPV1 63 35 C[C@H](CCS(C)(=O)=O)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745389 EF On-Demand Anodyne TRPV1 63 35 COC1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745419 DH On-Demand Anodyne CACNA1H 71 39 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880745426 GH On-Demand Anodyne SLC18A3 54 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880745426 GH On-Demand Anodyne EPHX2 36 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880745427 GH On-Demand Anodyne SLC18A3 54 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880745427 GH On-Demand Anodyne EPHX2 36 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880745429 GH On-Demand Anodyne SLC18A3 54 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880745429 GH On-Demand Anodyne EPHX2 36 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880745431 GH On-Demand Anodyne SLC18A3 54 46 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880745431 GH On-Demand Anodyne EPHX2 36 46 C[C@H]1c2ccccc2CN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745436 DJ On-Demand Anodyne TRPM8 26 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H](C4CCC4)C3)cc2)N1 ZINC000880745460 EG On-Demand Anodyne L3MBTL3 57 42 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H](C4CCC4)C3)cc2)N1 ZINC000880745461 EG On-Demand Anodyne L3MBTL3 57 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@H](C4CCC4)C3)cc2)N1 ZINC000880745462 EG On-Demand Anodyne L3MBTL3 57 42 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@H](C4CCC4)C3)cc2)N1 ZINC000880745463 EG On-Demand Anodyne L3MBTL3 57 42 CCC1(CO)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745489 DH On-Demand Anodyne CACNA1H 67 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCN(Cc2ccccn2)C1=O ZINC000880745517 GG On-Demand Anodyne CALCRL 16 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCN(Cc2ccccn2)C1=O ZINC000880745518 GG On-Demand Anodyne CALCRL 16 42 CN(C)CCCC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745528 EI On-Demand Anodyne CCR1 22 41 CN(C)c1nccc(CNC(=O)Nc2ccc(C3CC3)cc2F)n1 ZINC000880745529 EF On-Demand Anodyne TRPV1 24 40 O=C(CC1CC1)NNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745530 CF On-Demand Reactive DGAT1 36 40 CS(=O)(=O)C1CCC(C(=O)NCCc2nsc3ccccc23)CC1 ZINC000880745537 FF On-Demand Anodyne MTNR1A 21 46 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880745541 EG On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880745541 EG On-Demand Anodyne RBP4 42 33 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880745542 EG On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880745542 EG On-Demand Anodyne RBP4 42 33 O=C(NCC1SCCS1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880745554 EG On-Demand Anodyne PDE4D 18 46 O=C(NCC1SCCS1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880745554 EG On-Demand Anodyne CACNA1I 58 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CC[C@H](CO)CC1 ZINC000880745557 DG On-Demand Anodyne EPHX2 29 45 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880745558 DG On-Demand Anodyne EPHX2 29 45 C[C@@H](CNC(=O)Nc1ccc(C2CC2)cc1F)c1ccncc1 ZINC000880745568 DI On-Demand Anodyne TRPV1 53 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(N2CC=CC2)CC1 ZINC000880745599 EH On-Demand Anodyne L3MBTL3 46 32 CO[C@@H](C)c1nc(CNC(=O)Nc2ccc(C3CC3)cc2F)cs1 ZINC000880745609 EI On-Demand Anodyne TRPV1 62 36 O=C(Nc1ccc(C2CC2)cc1F)N(CCO)CCN1CCOCC1 ZINC000880745620 FD On-Demand Anodyne CASR 60 43 O=C(Nc1ccc(C2CC2)cc1F)N(CCO)CCN1CCOCC1 ZINC000880745620 FD On-Demand Anodyne EPHX2 18 41 O=C(NCCOc1ncccc1F)Nc1ccc(C2CC2)cc1F ZINC000880745622 EG On-Demand Anodyne P2RY1 23 42 C[C@@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)[S@@](C)=O ZINC000880745629 DF On-Demand Anodyne TRPV1 59 35 C[C@@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)[S@](C)=O ZINC000880745630 DF On-Demand Anodyne TRPV1 59 35 C[C@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)[S@@](C)=O ZINC000880745631 DF On-Demand Anodyne TRPV1 59 35 C[C@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)[S@](C)=O ZINC000880745632 DF On-Demand Anodyne TRPV1 59 35 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc(C2CC2)cc1F ZINC000880745641 GH On-Demand Anodyne EPHX2 19 47 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1ccc(C2CC2)cc1F ZINC000880745641 GH On-Demand Anodyne CACNA1I 42 33 CS(=O)(=O)N[C@@H]1CCC[C@H]1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745661 FF On-Demand Anodyne TRPV1 44 34 CS(=O)(=O)N[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745662 FF On-Demand Anodyne TRPV1 44 34 CS(=O)(=O)N[C@@H]1CCC[C@@H]1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745663 FF On-Demand Anodyne TRPV1 44 34 CS(=O)(=O)N[C@H]1CCC[C@H]1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880745664 FF On-Demand Anodyne TRPV1 44 34 CN1C(=O)N[C@]2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)C2)C1=O ZINC000880745668 ED On-Demand Anodyne CACNA1H 43 40 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)C2)C1=O ZINC000880745669 ED On-Demand Anodyne CACNA1H 43 40 O=C(Nc1ccc(C2CC2)cc1F)N(CCCO)Cc1ccccc1 ZINC000880745710 EI On-Demand Anodyne SOAT1 24 45 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880745711 FH On-Demand Anodyne EPHX2 34 43 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880745712 FH On-Demand Anodyne EPHX2 34 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880745716 FH On-Demand Anodyne RBP4 45 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880745717 FH On-Demand Anodyne RBP4 45 38 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880745725 DF On-Demand Anodyne CACNA1H 53 37 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880745743 FG On-Demand Anodyne SLC18A3 47 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880745743 FG On-Demand Anodyne EPHX2 36 44 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880745744 FG On-Demand Anodyne SLC18A3 47 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880745744 FG On-Demand Anodyne EPHX2 36 44 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880745745 FG On-Demand Anodyne SLC18A3 47 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880745745 FG On-Demand Anodyne EPHX2 36 44 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880745746 FG On-Demand Anodyne SLC18A3 47 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880745746 FG On-Demand Anodyne EPHX2 36 44 CS(=O)(=O)CC1(CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745748 EF On-Demand Anodyne TRPV1 61 36 O=C(NCCc1nsc2ccccc12)c1ccc(CN2CCOCC2)o1 ZINC000880745757 FF On-Demand Anodyne DRD2 16 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC(CC(F)(F)F)C1 ZINC000880745772 DI On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880745777 EH On-Demand Anodyne EPHX2 15 48 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880745777 EH On-Demand Anodyne RBP4 45 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880745778 EH On-Demand Anodyne EPHX2 15 48 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880745778 EH On-Demand Anodyne RBP4 45 32 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745786 FF On-Demand Anodyne CACNA1H 48 33 CC[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)C(=O)N1CCOCC1 ZINC000880745790 EE On-Demand Anodyne CCR1 31 48 COCCC(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745792 FF On-Demand Anodyne EPHX2 41 45 COCCC(=O)N1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880745792 FF On-Demand Anodyne CCR8 47 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C(=O)c2ccc(O)cc2)CC1 ZINC000880745797 GG On-Demand Anodyne L3MBTL3 50 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne PAPA1_CARPA 51 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne CTSK 23 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne CTSL 30 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne CTSS 22 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne SCN10A 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745813 GG On-Demand Anodyne FPR1 46 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne PAPA1_CARPA 51 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne CTSK 23 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne CTSL 30 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne CTSS 22 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne SCN10A 18 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccccc1C ZINC000880745814 GG On-Demand Anodyne FPR1 46 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745828 GF On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745828 GF On-Demand Anodyne CCKAR 40 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745828 GF On-Demand Anodyne FPR1 44 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745829 GF On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745829 GF On-Demand Anodyne CCKAR 40 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1nsc2ccccc12 ZINC000880745829 GF On-Demand Anodyne FPR1 44 38 C[C@H](CS(C)(=O)=O)N(C(=O)Nc1ccc(C2CC2)cc1F)C1CC1 ZINC000880745841 FG On-Demand Anodyne TRPV1 76 37 O=C(NCC[C@@H](O)C(F)(F)F)Nc1ccc(C2CC2)cc1F ZINC000880745872 DG On-Demand Anodyne TRPV1 48 34 O=C(NCC[C@H](O)C(F)(F)F)Nc1ccc(C2CC2)cc1F ZINC000880745873 DG On-Demand Anodyne TRPV1 48 34 C[S@](=O)c1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880745898 EH On-Demand Anodyne TRPV1 15 47 C[S@@](=O)c1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880745899 EH On-Demand Anodyne TRPV1 15 47 O=C(NCc1ccccc1CN1CCC(O)CC1)Nc1ccc(C2CC2)cc1F ZINC000880745943 GH On-Demand Anodyne SIGMAR1 17 41 O=C(NCc1ccccc1CN1CCC(O)CC1)Nc1ccc(C2CC2)cc1F ZINC000880745943 GH On-Demand Anodyne CCR3 38 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1SCCS1 ZINC000880745950 FD On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1SCCS1 ZINC000880745951 FD On-Demand Anodyne PAPA1_CARPA 39 48 O=C(Nc1ccc(C2CC2)cc1F)NC1CCS(=O)(=O)CC1 ZINC000880745953 EE On-Demand Anodyne EPHX2 17 46 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2ccccc2[C@@H]1CO ZINC000880745954 EH On-Demand Anodyne TRPM8 45 51 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2ccccc2[C@H]1CO ZINC000880745955 EH On-Demand Anodyne TRPM8 45 51 O=C(Nc1ccc(C2CC2)cc1F)N1CCOC2(CCCC2)C1 ZINC000880745958 DH On-Demand Anodyne EPHX2 17 44 C[S@@](=O)C[C@H](NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccc1 ZINC000880745968 FH On-Demand Anodyne NPY2R 48 37 C[S@](=O)C[C@H](NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccc1 ZINC000880745969 FH On-Demand Anodyne NPY2R 48 37 C[S@](=O)C[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccc1 ZINC000880745970 FH On-Demand Anodyne NPY2R 48 37 C[S@@](=O)C[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccc1 ZINC000880745971 FH On-Demand Anodyne NPY2R 48 37 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745977 EF On-Demand Anodyne TRPV1 41 35 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880745978 EF On-Demand Anodyne TRPV1 41 35 NC(=O)COc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880745993 FF On-Demand Anodyne ROCK2 19 49 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880745994 FF On-Demand Anodyne HTR2A 17 45 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880745994 FF On-Demand Anodyne PIK3CA 16 42 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880745994 FF On-Demand Anodyne MTOR 28 42 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880745994 FF On-Demand Anodyne EPHX2 28 49 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880745994 FF On-Demand Anodyne TBK1 24 44 O=C1CC[C@@H](c2ccc(C(=O)NCC(F)(F)c3ccc(F)cc3)cc2)N1 ZINC000880746016 FG On-Demand Anodyne PLD1 41 37 O=C1CC[C@H](c2ccc(C(=O)NCC(F)(F)c3ccc(F)cc3)cc2)N1 ZINC000880746017 FG On-Demand Anodyne PLD1 41 37 O=C(COC1CC1)NCCc1ccc(I)cc1 ZINC000880746019 EE On-Demand Anodyne LUXR 16 41 Cc1ccccc1[C@@H](CO)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880746023 EH On-Demand Anodyne CTSA 55 35 Cc1ccccc1[C@H](CO)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880746024 EH On-Demand Anodyne CTSA 55 35 CCC1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746035 DG On-Demand Anodyne CACNA1H 72 39 CCC1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746035 DG On-Demand Anodyne S1PR2 28 40 NC(=O)C1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746038 DF On-Demand Anodyne EPHX2 22 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2cccnc2)CC1 ZINC000880746065 EJ On-Demand Anodyne CACNA1H 42 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2cccnc2)CC1 ZINC000880746065 EJ On-Demand Anodyne CHRNA7 16 44 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2cccnc2)CC1 ZINC000880746065 EJ On-Demand Anodyne RBP4 44 37 CN(C)CC1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746070 EH On-Demand Anodyne EPHX2 31 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@H](CO)Cc1ccc(O)cc1 ZINC000880746074 EG On-Demand Anodyne YARS 63 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](O)C1 ZINC000880746096 CE On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](O)C1 ZINC000880746097 CE On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880746105 EI On-Demand Anodyne CCR3 58 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](Cc2ccncc2)C1 ZINC000880746106 EI On-Demand Anodyne CCR3 58 42 CCCCN(CCCO)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880746107 DH On-Demand Anodyne SOAT1 29 46 O=C1NC(=O)N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)C[C@H]12 ZINC000880746120 ED On-Demand Anodyne SMO 28 41 O=C1NC(=O)N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)C[C@@H]12 ZINC000880746121 ED On-Demand Anodyne SMO 28 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC=C(C(F)(F)F)CC1 ZINC000880746131 EI On-Demand Anodyne RBP4 48 35 CN1C(=O)NC2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)C1=O ZINC000880746153 FE On-Demand Anodyne CACNA1H 63 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCOCC1 ZINC000880746155 CG On-Demand Anodyne EPHX2 15 50 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCOCC1 ZINC000880746156 CG On-Demand Anodyne EPHX2 15 50 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(n2ccc(C(F)(F)F)n2)CC1 ZINC000880746245 GJ On-Demand Anodyne RBP4 48 36 O=C(NOCc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880746260 DG On-Demand Anodyne CHRNA7 42 41 NC(=O)c1cc(OC2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)ccn1 ZINC000880746274 GG On-Demand Anodyne EPHX2 17 40 Cc1csc([C@H](C)CNC(=O)Nc2ccc(C3CC3)cc2F)n1 ZINC000880746293 EI On-Demand Anodyne TRPV1 49 34 O=C1NC2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)CO1 ZINC000880746297 EF On-Demand Anodyne CACNA1H 60 37 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746312 FE On-Demand Anodyne TRPV1 42 34 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746313 FE On-Demand Anodyne TRPV1 42 34 COc1cc(NC(=O)[C@H](CNC(=O)OC(C)(C)C)OC)ccc1OC(F)F ZINC000880746333 GF On-Demand Anodyne ENPP1 54 30 O=C(NC[C@H](O)CO)Nc1ccc(C2CC2)cc1F ZINC000880746346 CD On-Demand Anodyne MAP2K1 15 41 O=C(NC[C@@H](O)CO)Nc1ccc(C2CC2)cc1F ZINC000880746348 CD On-Demand Anodyne MAP2K1 15 41 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@H](C2CCC2)C1 ZINC000880746350 DG On-Demand Anodyne MAP3K12 29 40 CN1CC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746351 CF On-Demand Anodyne CCR3 41 35 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@@H](C2CCC2)C1 ZINC000880746352 DG On-Demand Anodyne MAP3K12 29 40 CN1CC[C@@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746353 CF On-Demand Anodyne CCR3 41 35 CS(=O)(=O)C1CCC(C(=O)N2CC[C@@H](Oc3ccccc3)C2)CC1 ZINC000880746355 FE On-Demand Anodyne PRSS2 53 32 CS(=O)(=O)C1CCC(C(=O)N2CC[C@@H](Oc3ccccc3)C2)CC1 ZINC000880746355 FE On-Demand Anodyne EPHX2 19 42 CS(=O)(=O)C1CCC(C(=O)N2CC[C@@H](Oc3ccccc3)C2)CC1 ZINC000880746355 FE On-Demand Anodyne GPR119 28 41 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(C2CC2)cc1F ZINC000880746382 GG On-Demand Anodyne PIK3CA 18 40 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(C2CC2)cc1F ZINC000880746382 GG On-Demand Anodyne MTOR 34 40 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc(C2CC2)cc1F ZINC000880746382 GG On-Demand Anodyne STAT6 49 33 O=C(COC1CC1)N1CCC(c2ccon2)CC1 ZINC000880746393 CD On-Demand Anodyne ETHR 66 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2c([nH]c3ccccc23)C1 ZINC000880746396 EJ On-Demand Anodyne SSTR4 52 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2c([nH]c3ccccc23)C1 ZINC000880746396 EJ On-Demand Anodyne SSTR5 42 34 O=C(c1cncc2[nH]ccc12)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746397 EH On-Demand Anodyne ACACA 42 36 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880746407 EG On-Demand Anodyne PLM1_PLAFA 46 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880746407 EG On-Demand Anodyne PLM2_PLAFA 30 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880746408 EG On-Demand Anodyne PLM1_PLAFA 46 41 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880746408 EG On-Demand Anodyne PLM2_PLAFA 30 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCCC2(CC2)C1 ZINC000880746414 CI On-Demand Anodyne EPHX2 26 41 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746416 EG On-Demand Anodyne HDAC10 24 43 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746416 EG On-Demand Anodyne HDAC3 29 43 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746416 EG On-Demand Anodyne HDAC6 20 43 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746418 EG On-Demand Anodyne HDAC10 24 43 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746418 EG On-Demand Anodyne HDAC3 29 43 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCC(C)(C)CO3)c2)nn1 ZINC000880746418 EG On-Demand Anodyne HDAC6 20 43 COc1cc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)ccc1OC(F)F ZINC000880746437 GH On-Demand Anodyne ENPP1 66 32 COc1cc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)ccc1OC(F)F ZINC000880746439 GH On-Demand Anodyne ENPP1 66 32 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)F)c2)nn1 ZINC000880746451 DG On-Demand Anodyne HDAC10 33 43 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)F)c2)nn1 ZINC000880746451 DG On-Demand Anodyne HDAC2 15 43 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)F)c2)nn1 ZINC000880746451 DG On-Demand Anodyne HDAC3 36 43 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)F)c2)nn1 ZINC000880746451 DG On-Demand Anodyne HDAC6 30 43 C=CC(C)(C)CC(=O)Nc1ccc(OC(F)F)c(OC)c1 ZINC000880746494 CH On-Demand Mild ENPP1 78 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2ccccn2)CC1 ZINC000880746509 EJ On-Demand Anodyne CACNA1H 45 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2ccccn2)CC1 ZINC000880746509 EJ On-Demand Anodyne EPHX2 16 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2ccccn2)CC1 ZINC000880746509 EJ On-Demand Anodyne RBP4 60 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(C(F)F)CC1 ZINC000880746530 EG On-Demand Anodyne CACNA1H 67 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(F)(F)C1 ZINC000880746551 CH On-Demand Anodyne CACNA1H 62 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880746554 FI On-Demand Anodyne RBP4 52 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880746556 GI On-Demand Anodyne CACNA1H 64 39 COCC1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746559 DF On-Demand Anodyne CACNA1H 75 38 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880746637 FG On-Demand Anodyne CACNA1H 55 35 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880746639 FG On-Demand Anodyne CACNA1H 55 35 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880746642 FG On-Demand Anodyne CACNA1H 55 35 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880746644 FG On-Demand Anodyne CACNA1H 55 35 Cc1nc(C(C)C)ncc1C(=O)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746646 FH On-Demand Anodyne ACACA 64 39 Cc1nc(C(C)C)ncc1C(=O)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746646 FH On-Demand Anodyne ACACB 42 38 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746659 DE On-Demand Anodyne EPHX2 15 42 O=C(NCCCNC(=O)C1CCC1)Nc1ccc(C2CC2)cc1F ZINC000880746668 EG On-Demand Anodyne TBK1 75 42 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne HRH1 18 40 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne CHRM3 19 45 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne GRIN2B 18 42 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne PRSS2 42 32 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne CCR3 22 40 O=C(COC1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746685 CD On-Demand Anodyne EPHX2 23 46 C=CC(C)(C)CC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746699 CG On-Demand Mild CHRM3 25 47 C=CC(C)(C)CC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746699 CG On-Demand Mild EPHX2 20 42 CC1(CO)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746709 DG On-Demand Anodyne CACNA1H 71 39 C[C@H](NC(=O)OC(C)(C)C)[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746720 GI On-Demand Anodyne GPR119 19 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](C2CCOCC2)C1 ZINC000880746728 EH On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](C2CCOCC2)C1 ZINC000880746729 EH On-Demand Anodyne RBP4 47 35 O=C(c1ncccc1-c1ccccn1)N1CCC[C@H](C2CCC2)C1 ZINC000880746732 DH On-Demand Anodyne MAP3K12 29 40 O=C(c1ncccc1-c1ccccn1)N1CCC[C@@H](C2CCC2)C1 ZINC000880746733 DH On-Demand Anodyne MAP3K12 29 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CC[C@@H](O)CC1 ZINC000880746758 CG On-Demand Anodyne EPHX2 30 48 O=C(NCC(F)(F)F)[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746759 FG On-Demand Anodyne RBP4 46 34 O=C(NCC(F)(F)F)[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746761 FG On-Demand Anodyne RBP4 46 34 COc1cc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)ncn1 ZINC000880746780 FF On-Demand Anodyne PDGFRB 50 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCOC2(CCC2)C1 ZINC000880746788 DG On-Demand Anodyne EPHX2 18 46 O=C(CN1CCCCS1(=O)=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746800 ED On-Demand Anodyne CPT1A 57 34 O=C(CN1CCCCS1(=O)=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880746800 ED On-Demand Anodyne EPHX2 15 41 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne F10 30 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne GRM4 19 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne MAPK9 40 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne MAPK10 47 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne CCR2 16 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne EPHB3 21 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne STAT6 50 35 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne CREBBP 34 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne DGAT1 18 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1cc(S(=O)(=O)Nc2ccccc2F)ccc1Cl ZINC000880746802 JH On-Demand Anodyne BRD9 34 40 Cc1nc(CN2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)n[nH]1 ZINC000880746805 FE On-Demand Anodyne MCHR1 18 40 CN1CCC(N2CCC(NC(=O)Nc3ccc(C4CC4)cc3F)CC2)CC1 ZINC000880746844 FG On-Demand Anodyne HTR1F 45 33 CN1CCC(N2CCC(NC(=O)Nc3ccc(C4CC4)cc3F)CC2)CC1 ZINC000880746844 FG On-Demand Anodyne SLC6A5 17 41 CN1CCC(N2CCC(NC(=O)Nc3ccc(C4CC4)cc3F)CC2)CC1 ZINC000880746844 FG On-Demand Anodyne EPHX2 29 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]([C@H]2CCOC2)C1 ZINC000880746847 DH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]([C@H]2CCOC2)C1 ZINC000880746849 DH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]([C@@H]2CCOC2)C1 ZINC000880746852 DH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]([C@@H]2CCOC2)C1 ZINC000880746854 DH On-Demand Anodyne RBP4 46 35 COc1cc(NC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)ccc1OC(F)F ZINC000880746855 EG On-Demand Anodyne ENPP1 48 29 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1ccc(C2CC2)cc1F ZINC000880746856 GH On-Demand Anodyne MCHR1 23 41 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1ccc(C2CC2)cc1F ZINC000880746858 GH On-Demand Anodyne MCHR1 23 41 COCCO[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746860 DF On-Demand Anodyne LIPG 26 41 CCC1(O)CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746861 DH On-Demand Anodyne EPHX2 26 42 COCCO[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880746862 DF On-Demand Anodyne LIPG 26 41 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@@H](Oc4ccccc4)C3)cc2)N1 ZINC000880746864 FF On-Demand Anodyne L3MBTL3 47 35 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H](Oc4ccccc4)C3)cc2)N1 ZINC000880746865 FF On-Demand Anodyne L3MBTL3 47 35 O=C1NCC[C@H]1CC(=O)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746876 ED On-Demand Anodyne GHRL 48 32 O=C1NCC[C@@H]1CC(=O)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746877 ED On-Demand Anodyne GHRL 48 32 O=C(NCc1nc(C(F)(F)F)n[nH]1)Nc1ccc(C2CC2)cc1F ZINC000880746879 EG On-Demand Anodyne TRPV1 62 35 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H](CN3CCCC3=O)C2)N1Cc1ccccc1 ZINC000880746880 GC On-Demand Anodyne ACHE 15 45 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H](CN3CCCC3=O)C2)N1Cc1ccccc1 ZINC000880746881 GC On-Demand Anodyne ACHE 15 45 Cc1nc(C(C)C)ncc1C(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880746893 EF On-Demand Anodyne KCNK3 43 35 Cc1nc(C(C)C)ncc1C(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880746893 EF On-Demand Anodyne KCNK9 43 35 COc1cc(NC(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)ccc1OC(F)F ZINC000880746901 FG On-Demand Anodyne ENPP1 70 33 COc1cc(NC(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)ccc1OC(F)F ZINC000880746902 FG On-Demand Anodyne ENPP1 70 33 CC(C)(CS(C)(=O)=O)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880746914 EF On-Demand Anodyne TRPV1 69 38 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](C2CC2)C1 ZINC000880746924 CH On-Demand Anodyne RBP4 57 38 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](C2CC2)C1 ZINC000880746925 CH On-Demand Anodyne RBP4 57 38 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880746926 ED On-Demand Anodyne CCR1 33 40 COc1cc(NC(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)ccc1OC(F)F ZINC000880746930 FG On-Demand Anodyne ENPP1 70 33 COc1cc(NC(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)ccc1OC(F)F ZINC000880746932 FG On-Demand Anodyne ENPP1 70 33 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746944 EH On-Demand Anodyne ACACA 89 51 O=C(c1cnc2cc[nH]c2c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880746944 EH On-Demand Anodyne ACACB 60 51 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H](O)[C@H](O)C1 ZINC000880746951 CD On-Demand Anodyne RBP4 48 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2ccccn2)CC1 ZINC000880746990 FG On-Demand Anodyne FAAH 18 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(Cc2ccccn2)CC1 ZINC000880746990 FG On-Demand Anodyne RBP4 50 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccon2)CC1 ZINC000880746993 FE On-Demand Anodyne P2RY12 129 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccon2)CC1 ZINC000880746994 FE On-Demand Anodyne P2RY12 129 36 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747038 EE On-Demand Anodyne EPHX2 16 45 O=C(Nc1ccc(C2CC2)cc1F)NC1CCC(F)(F)CC1 ZINC000880747041 DI On-Demand Anodyne EPHX2 26 46 COc1cc(NC(=O)c2ncsc2C2CC2)ccc1OC(F)F ZINC000880747056 EH On-Demand Anodyne MAP1 62 38 COc1cc(NC(=O)c2ncsc2C2CC2)ccc1OC(F)F ZINC000880747056 EH On-Demand Anodyne ENPP1 70 35 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(C2CC2)cc1F ZINC000880747058 FG On-Demand Anodyne PIK3CA 22 42 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(C2CC2)cc1F ZINC000880747058 FG On-Demand Anodyne MTOR 23 42 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(C2CC2)cc1F ZINC000880747058 FG On-Demand Anodyne PIK3CG 19 42 O=C(NCc1cccc(N2CCOCC2)n1)Nc1ccc(C2CC2)cc1F ZINC000880747058 FG On-Demand Anodyne PIK3CB 53 36 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747064 EG On-Demand Anodyne CCR3 46 38 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747065 EG On-Demand Anodyne CCR3 46 38 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747066 EG On-Demand Anodyne CCR3 46 38 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747067 EG On-Demand Anodyne CCR3 46 38 N#C[C@@]1(F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880747076 CG On-Demand Mild CACNA1H 41 37 N#C[C@]1(F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880747077 CG On-Demand Mild CACNA1H 41 37 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(c2ccon2)CC1 ZINC000880747093 FF On-Demand Anodyne ETHR 63 36 O=C(c1cnc(CC2CC2)s1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747098 EG On-Demand Anodyne GRIN2B 50 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne GHRHR 53 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne P2RY12 174 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne PGC 51 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne CCKAR 26 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne REN 65 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747101 GF On-Demand Anodyne FPR1 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne GHRHR 53 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne P2RY12 174 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne PGC 51 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne CCKAR 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne REN 65 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747102 GF On-Demand Anodyne FPR1 46 36 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@@H](C2CCC2)C1 ZINC000880747103 CG On-Demand Anodyne JAK3 15 40 O=C(c1cnc2cc[nH]c2c1)N1CCC[C@H](C2CCC2)C1 ZINC000880747104 CG On-Demand Anodyne JAK3 15 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCC(c2ccon2)CC1 ZINC000880747109 DH On-Demand Anodyne ETHR 69 40 O=C(CC[C@H]1CCc2ccccc21)N1CCC(c2ccon2)CC1 ZINC000880747111 DH On-Demand Anodyne ETHR 69 40 Cn1nnc(C(=O)N2CCC3(CCc4ccccc4O3)CC2)n1 ZINC000880747113 DD On-Demand Anodyne ACACA 68 36 Cn1nnc(C(=O)N2CCC3(CCc4ccccc4O3)CC2)n1 ZINC000880747113 DD On-Demand Anodyne ACACB 45 36 Cn1nnc(C(=O)N2CCC3(CCc4ccccc4O3)CC2)n1 ZINC000880747113 DD On-Demand Anodyne SCD 18 41 Cn1cc(-c2cccc(NC(=O)[C@H]3C[C@@H]4CC[C@H](C3)S4(=O)=O)c2)nn1 ZINC000880747115 FD On-Demand Anodyne HDAC10 20 42 Cn1cc(-c2cccc(NC(=O)[C@H]3C[C@@H]4CC[C@H](C3)S4(=O)=O)c2)nn1 ZINC000880747115 FD On-Demand Anodyne HDAC3 23 42 Cn1cc(-c2cccc(NC(=O)[C@H]3C[C@@H]4CC[C@H](C3)S4(=O)=O)c2)nn1 ZINC000880747115 FD On-Demand Anodyne HDAC6 16 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747118 GI On-Demand Anodyne CCR3 22 40 CO[C@@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)C(F)(F)F ZINC000880747121 EH On-Demand Anodyne TRPV1 57 34 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747122 GI On-Demand Anodyne CCR3 22 40 C[C@@](O)(C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1)C(F)(F)F ZINC000880747127 FI On-Demand Anodyne RBP4 42 38 C[C@@H](CNC(=O)Nc1ccc(C2CC2)cc1F)S(C)(=O)=O ZINC000880747128 DE On-Demand Anodyne TRPV1 97 38 O=C(C[C@@H]1C[C@H]1C1CC1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747133 CG On-Demand Anodyne EPHX2 16 45 O=C(CCn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880747147 HD On-Demand Anodyne HTR7 17 42 O=C(CCn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880747147 HD On-Demand Anodyne PRKDC 41 33 O=C(CCn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880747147 HD On-Demand Anodyne STAT6 58 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(c2ncccc2F)CC1 ZINC000880747156 FH On-Demand Anodyne TRPV1 15 52 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(c2ncccc2F)CC1 ZINC000880747156 FH On-Demand Anodyne RBP4 28 48 O=C1NCC[C@H]1CC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747170 CD On-Demand Anodyne GRIN2B 20 42 O=C1NCC[C@@H]1CC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747171 CD On-Demand Anodyne GRIN2B 20 42 O=C1NCC2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)O1 ZINC000880747178 EF On-Demand Anodyne CACNA1H 63 38 Cn1cc(-c2cccc(NC(=O)CN3CCCCS3(=O)=O)c2)nn1 ZINC000880747181 EC On-Demand Anodyne HDAC10 31 44 Cn1cc(-c2cccc(NC(=O)CN3CCCCS3(=O)=O)c2)nn1 ZINC000880747181 EC On-Demand Anodyne HDAC2 15 44 Cn1cc(-c2cccc(NC(=O)CN3CCCCS3(=O)=O)c2)nn1 ZINC000880747181 EC On-Demand Anodyne HDAC3 36 44 Cn1cc(-c2cccc(NC(=O)CN3CCCCS3(=O)=O)c2)nn1 ZINC000880747181 EC On-Demand Anodyne HDAC6 27 44 CN(CCO)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747198 EF On-Demand Anodyne CCR1 25 42 CC(C)(C(=O)N1CCC(c2ccon2)CC1)c1ccc(F)cc1F ZINC000880747219 EH On-Demand Anodyne PRCP 45 36 C#C[C@@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747227 BF On-Demand Mild TRPV1 54 36 C#C[C@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747228 BF On-Demand Mild TRPV1 54 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCC(c2ccon2)CC1 ZINC000880747229 GH On-Demand Anodyne RBP4 46 41 C[C@H](C#N)Oc1ccccc1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747251 EJ On-Demand Mild P2RY1 21 41 C[C@@H](C#N)Oc1ccccc1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747252 EJ On-Demand Mild P2RY1 21 41 O=C(COC1CC1)N1CC[C@H](c2ccccc2)[C@H](NC(=O)C(F)(F)F)C1 ZINC000880747255 FE On-Demand Anodyne EPHX2 25 42 COC(=O)C1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747267 EE On-Demand Anodyne CACNA1H 71 38 Cn1nnc(C(=O)N2CC[C@@H](Oc3ccccc3)C2)n1 ZINC000880747341 CC On-Demand Anodyne GRIN2B 18 43 Cn1nnc(C(=O)N2CC[C@@H](Oc3ccccc3)C2)n1 ZINC000880747341 CC On-Demand Anodyne EPHX2 15 42 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC(c2ccon2)CC1 ZINC000880747343 CF On-Demand Anodyne ETHR 62 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880747352 GI On-Demand Anodyne CACNA1H 60 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880747352 GI On-Demand Anodyne S1PR2 28 40 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880747353 EG On-Demand Anodyne CCR1 22 40 O=C(c1cc2ccccc2cc1F)N1CCC(c2ccon2)CC1 ZINC000880747359 DH On-Demand Anodyne ETHR 42 34 COc1cc(NC(=O)c2c3c(nn2C)CCSC3)ccc1OC(F)F ZINC000880747383 FG On-Demand Anodyne ENPP1 66 31 O=C(NOCCO)Nc1ccc(C2CC2)cc1F ZINC000880747410 CD On-Demand Anodyne MAP2K1 28 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(C(F)(F)F)CC1 ZINC000880747411 EH On-Demand Anodyne CACNA1H 56 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(C(F)(F)F)CC1 ZINC000880747411 EH On-Demand Anodyne RBP4 47 36 Cc1cncc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880747421 CH On-Demand Anodyne NAMPT 28 48 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880747435 FI On-Demand Anodyne CACNA1H 63 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(c2ccccc2)CC1 ZINC000880747435 FI On-Demand Anodyne RBP4 55 37 CN(Cc1ccc(S(C)(=O)=O)cc1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880747482 GH On-Demand Anodyne TRPV1 55 36 O=C(Nc1ccc(C2CC2)cc1F)N(CCO)CCCO ZINC000880747486 CD On-Demand Anodyne SOAT1 24 40 O=C(Nc1cnn(CC(F)F)c1)Nc1ccc(C2CC2)cc1F ZINC000880747490 DH On-Demand Anodyne PANC 41 34 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H](C(F)(F)F)O1 ZINC000880747492 EH On-Demand Anodyne RBP4 45 34 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C(F)(F)F)O1 ZINC000880747493 EH On-Demand Anodyne RBP4 45 34 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C(F)(F)F)O1 ZINC000880747494 EH On-Demand Anodyne RBP4 45 34 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H](C(F)(F)F)O1 ZINC000880747495 EH On-Demand Anodyne RBP4 45 34 NC(=O)c1cccnc1N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747496 GF On-Demand Anodyne TRPV1 15 48 NC(=O)c1cccnc1N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747496 GF On-Demand Anodyne RBP4 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C2CC2)CC1 ZINC000880747500 DG On-Demand Anodyne L3MBTL3 43 32 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747507 EI On-Demand Anodyne TRPV1 20 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCn2c(nnc2-c2ccccc2)C1 ZINC000880747519 GI On-Demand Anodyne P2RX7 28 48 O=C(Nc1ccc(C2CC2)cc1F)N1CCn2c(nnc2-c2ccccc2)C1 ZINC000880747519 GI On-Demand Anodyne RBP4 45 32 Cn1cc(CN2CCCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)cn1 ZINC000880747537 FG On-Demand Anodyne MCHR1 17 44 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880747567 EF On-Demand Anodyne CCR3 58 39 Cn1nc2c(c1C(=O)N1CCC3(CCc4ccccc4O3)CC1)CSCC2 ZINC000880747591 GG On-Demand Anodyne ACACA 43 33 C=CC(C)(C)CC(=O)N1CCC(c2ccon2)CC1 ZINC000880747593 CF On-Demand Mild ETHR 65 35 O=C(c1ccc(CN2CCOCC2)o1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880747600 FE On-Demand Anodyne GRIN2B 17 41 O=C(NCCN1CCCOCC1)Nc1ccc(C2CC2)cc1F ZINC000880747607 DF On-Demand Anodyne EPHX2 26 51 O=C(Cn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880747608 GD On-Demand Anodyne STAT6 68 38 COc1cc(NC(=O)c2nnn(C)n2)ccc1OC(F)F ZINC000880747614 CD On-Demand Anodyne ENPP1 83 40 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747628 FG On-Demand Anodyne RBP4 49 37 COC(=O)C1=NOC2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)C1 ZINC000880747629 GG On-Demand Anodyne CACNA1H 45 34 O=C1CC[C@@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5O4)CC3)cc2)N1 ZINC000880747642 GH On-Demand Anodyne ACACA 64 38 O=C1CC[C@@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5O4)CC3)cc2)N1 ZINC000880747642 GH On-Demand Anodyne ACACB 40 37 O=C1CC[C@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5O4)CC3)cc2)N1 ZINC000880747643 GH On-Demand Anodyne ACACA 64 38 O=C1CC[C@H](c2ccc(C(=O)N3CCC4(CCc5ccccc5O4)CC3)cc2)N1 ZINC000880747643 GH On-Demand Anodyne ACACB 40 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880747662 FH On-Demand Anodyne CACNA1H 54 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880747663 FH On-Demand Anodyne CACNA1H 54 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880747664 GI On-Demand Anodyne CACNA1H 65 41 Cn1nccc1C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747713 EH On-Demand Anodyne CACNA1H 43 33 C[C@H](CS(C)(=O)=O)N(C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880747724 EF On-Demand Anodyne TRPV1 63 36 CNC(=O)CC1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880747737 EG On-Demand Anodyne CCR1 23 40 CCCCCN(CCO)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880747746 DH On-Demand Anodyne SOAT1 35 49 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2ncc[nH]2)CC1 ZINC000880747781 EH On-Demand Anodyne HTR2B 18 41 CC1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880747784 CH On-Demand Anodyne CACNA1H 68 41 COc1cc(NC(=O)[C@H]2CCc3nncn3CC2)ccc1OC(F)F ZINC000880747787 FE On-Demand Anodyne ENPP1 61 31 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1OC(F)F ZINC000880747793 FH On-Demand Anodyne JUN 15 41 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1OC(F)F ZINC000880747793 FH On-Demand Anodyne ENPP1 75 36 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1OC(F)F ZINC000880747793 FH On-Demand Anodyne KCNK3 50 39 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)ccc1OC(F)F ZINC000880747793 FH On-Demand Anodyne KCNK9 43 39 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1C ZINC000880747796 CH On-Demand Anodyne RBP4 46 35 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)ccc1OC(F)F ZINC000880747798 GF On-Demand Anodyne ENPP1 67 33 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H]1C ZINC000880747800 CH On-Demand Anodyne RBP4 46 35 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H]1C ZINC000880747804 CH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@]2(CCOC2)C1 ZINC000880747819 DF On-Demand Anodyne EPHX2 16 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@]2(CCOC2)C1 ZINC000880747820 DF On-Demand Anodyne EPHX2 16 41 O=C(NCC(F)(F)c1ccc(F)cc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880747826 FE On-Demand Anodyne CACNA1G 39 45 Cn1cc(-c2cccc(NC(=O)C3CCC(S(C)(=O)=O)CC3)c2)nn1 ZINC000880747831 FE On-Demand Anodyne HDAC10 20 42 Cn1cc(-c2cccc(NC(=O)C3CCC(S(C)(=O)=O)CC3)c2)nn1 ZINC000880747831 FE On-Demand Anodyne HDAC3 23 42 Cn1cc(-c2cccc(NC(=O)C3CCC(S(C)(=O)=O)CC3)c2)nn1 ZINC000880747831 FE On-Demand Anodyne HDAC6 16 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](Nc2ccc3nccn3n2)C1 ZINC000880747841 GG On-Demand Anodyne RBP4 44 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Nc2ccc3nccn3n2)C1 ZINC000880747842 GG On-Demand Anodyne RBP4 44 32 CC(C)(C(=O)N1CCC(c2ccon2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880747843 FI On-Demand Anodyne ETHR 61 33 O=C(C(=O)N1CC[C@H](CN2CCCC2=O)C1)c1c[nH]c2cc(F)ccc12 ZINC000880747844 FD On-Demand Anodyne GRIN2B 16 55 O=C(C(=O)N1CC[C@@H](CN2CCCC2=O)C1)c1c[nH]c2cc(F)ccc12 ZINC000880747845 FD On-Demand Anodyne GRIN2B 16 55 Cn1nnc(C(=O)N[C@H](CO)c2cccc(Cl)c2Cl)n1 ZINC000880747855 DC On-Demand Anodyne CTSA 27 42 Cn1nnc(C(=O)N[C@@H](CO)c2cccc(Cl)c2Cl)n1 ZINC000880747856 DC On-Demand Anodyne CTSA 27 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880747857 EG On-Demand Anodyne CCR8 57 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880747858 EG On-Demand Anodyne CCR8 57 40 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(c4ccon4)CC3)cc2)N1 ZINC000880747864 EF On-Demand Anodyne L3MBTL3 48 35 O=C1CC[C@H](c2ccc(C(=O)N3CCC(c4ccon4)CC3)cc2)N1 ZINC000880747865 EF On-Demand Anodyne L3MBTL3 48 35 Cc1cnc(Cl)c(C(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880747870 DG On-Demand Anodyne HRH1 29 45 Cc1cnc(Cl)c(C(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880747870 DG On-Demand Anodyne HCRTR1 21 42 Cc1cnc(Cl)c(C(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880747870 DG On-Demand Anodyne CCR3 34 45 Cc1cnc(Cl)c(C(=O)N2CC[C@@H](Oc3ccccc3)C2)c1 ZINC000880747870 DG On-Demand Anodyne EPHX2 16 42 O=C(CN1CCCCS1(=O)=O)N1CCC(c2ccon2)CC1 ZINC000880747878 EC On-Demand Anodyne ETHR 46 32 COc1ccccc1-c1ccc(C(=O)NC[C@H](OC)C2CCCC2)c(O)n1 ZINC000880747902 FG On-Demand Anodyne KCNA3 40 38 COc1ccccc1-c1ccc(C(=O)NC[C@@H](OC)C2CCCC2)c(O)n1 ZINC000880747903 FG On-Demand Anodyne KCNA3 40 38 COc1ccc(O)c(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880747951 EH On-Demand Clean MTNR1A 27 41 COc1ccc(O)c(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880747951 EH On-Demand Clean MTNR1B 19 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C2CCCC2)CC1 ZINC000880747966 EI On-Demand Anodyne HRH3 25 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCCN(C2CCCC2)CC1 ZINC000880747966 EI On-Demand Anodyne L3MBTL3 63 36 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CCCC1 ZINC000880747986 EF On-Demand Anodyne GABRA1 18 45 CO[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)C1CCCC1 ZINC000880747986 EF On-Demand Anodyne GABRA2 16 45 O=C(NCC(F)(F)c1ccc(F)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880747999 FF On-Demand Anodyne CACNA1G 40 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@H](C(F)(F)F)C1 ZINC000880748014 EG On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@H](C(F)(F)F)C1 ZINC000880748015 EG On-Demand Anodyne RBP4 47 35 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748028 GH On-Demand Anodyne CACNA1H 63 37 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748028 GH On-Demand Anodyne RBP4 55 37 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880748041 EH On-Demand Anodyne HTR3A 32 43 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880748041 EH On-Demand Anodyne EPHX2 16 42 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880748048 FF On-Demand Mild ADRA1A 22 40 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880748048 FF On-Demand Mild CASR 56 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748049 GF On-Demand Anodyne PAPA1_CARPA 50 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748049 GF On-Demand Anodyne CTSK 20 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748049 GF On-Demand Anodyne CTSL 22 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748049 GF On-Demand Anodyne CTSS 15 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748049 GF On-Demand Anodyne FPR1 44 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748050 GF On-Demand Anodyne PAPA1_CARPA 50 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748050 GF On-Demand Anodyne CTSK 20 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748050 GF On-Demand Anodyne CTSL 22 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748050 GF On-Demand Anodyne CTSS 15 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)c1ccc(F)cc1 ZINC000880748050 GF On-Demand Anodyne FPR1 44 39 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(C3CC3)cc1F)CC2 ZINC000880748057 EH On-Demand Anodyne CACNA1H 65 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C2CCC2)CC1 ZINC000880748075 DG On-Demand Anodyne HRH3 24 44 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(C2CCC2)CC1 ZINC000880748075 DG On-Demand Anodyne L3MBTL3 51 33 O=C1CC2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)CN1 ZINC000880748077 EF On-Demand Anodyne CACNA1H 55 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCOCC2)C1 ZINC000880748089 DH On-Demand Anodyne EPHX2 26 41 C[S@@](=O)CCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748105 CF On-Demand Anodyne CCR3 33 41 O=C1NCCN(C(=O)Nc2ccc(C3CC3)cc2F)[C@H]1c1cccs1 ZINC000880748106 FG On-Demand Anodyne TRPM8 32 41 O=C1NCCN(C(=O)Nc2ccc(C3CC3)cc2F)[C@@H]1c1cccs1 ZINC000880748107 FG On-Demand Anodyne TRPM8 32 41 O=C(Nc1ccc(C2CC2)cc1F)N1[C@H]2CC[C@H]1c1ccccc12 ZINC000880748110 DK On-Demand Anodyne RBP4 54 34 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880748136 ED On-Demand Anodyne CCR8 67 35 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880748137 ED On-Demand Anodyne CCR8 67 35 CCS(=O)(=O)C[C@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748164 EF On-Demand Anodyne TRPV1 55 35 CCS(=O)(=O)C[C@@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748165 EF On-Demand Anodyne TRPV1 55 35 O=C(Nc1ccc(C2CC2)cc1F)N(CCO)CCc1ccccc1 ZINC000880748274 EH On-Demand Anodyne SOAT1 21 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880748275 FI On-Demand Anodyne ETHR 54 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880748276 FI On-Demand Anodyne ETHR 54 42 C[C@@H](O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748282 DG On-Demand Anodyne CACNA1H 45 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880748287 FG On-Demand Anodyne RBP4 48 34 COC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748299 DG On-Demand Anodyne RBP4 38 40 CN(C)C(=O)Nc1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880748302 FI On-Demand Anodyne ROCK2 19 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880748303 FH On-Demand Anodyne RBP4 44 32 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880748304 FH On-Demand Anodyne RBP4 44 32 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2cncnc2C1 ZINC000880748305 DG On-Demand Anodyne MAPK1 51 36 COc1cccc([C@H](CO)NC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880748307 EH On-Demand Anodyne ROCK2 17 41 CS(=O)(=O)C1CCC(C(=O)NCC(F)(F)c2ccc(F)cc2)CC1 ZINC000880748318 FF On-Demand Anodyne CACNA1G 44 49 C[C@H](CS(C)(=O)=O)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748325 DE On-Demand Anodyne TRPV1 70 36 O=C(Nc1ccc(O[C@H]2CC2(F)F)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880748329 GG On-Demand Anodyne EPHX2 27 41 O=C(Nc1ccc(O[C@@H]2CC2(F)F)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880748330 GG On-Demand Anodyne EPHX2 27 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CC(N2CCCCC2)C1 ZINC000880748345 EH On-Demand Anodyne EPHX2 16 44 O=C(Nc1cc(C2CCOCC2)[nH]n1)Nc1ccc(C2CC2)cc1F ZINC000880748396 EH On-Demand Anodyne CDK2 15 47 O=C(Nc1cc(C2CCOCC2)[nH]n1)Nc1ccc(C2CC2)cc1F ZINC000880748396 EH On-Demand Anodyne PKNB 47 36 O=C(Nc1ccc(C2CC2)cc1F)N(CCCO)Cc1ccccn1 ZINC000880748406 EH On-Demand Anodyne SOAT1 25 41 O=C(Nc1ccc(C2CC2)cc1F)NC1CC(F)(F)C1 ZINC000880748412 CH On-Demand Anodyne EPHX2 17 44 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880748419 EH On-Demand Anodyne EPHX2 18 47 C[C@H](O)CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748432 DE On-Demand Anodyne CACNA1H 49 39 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](N2CCOCC2)C1 ZINC000880748437 EF On-Demand Anodyne L3MBTL3 45 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](N2CCOCC2)C1 ZINC000880748438 EF On-Demand Anodyne L3MBTL3 45 36 O=C(NCCOc1cccnc1)Nc1ccc(C2CC2)cc1F ZINC000880748443 DG On-Demand Anodyne CHRNA7 15 46 O=C(Nc1cnn(CC(=O)N2CCOCC2)c1)Nc1ccc(C2CC2)cc1F ZINC000880748444 GE On-Demand Anodyne EPHX2 18 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(C(F)(F)F)CC1 ZINC000880748460 EJ On-Demand Anodyne RBP4 54 40 N#Cc1cc(NC(=O)Nc2ccc(C3CC3)cc2F)ccc1N1CCC(O)CC1 ZINC000880748461 GI On-Demand Mild CSF1R 24 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(Nc2cccnn2)CC1 ZINC000880748462 FH On-Demand Anodyne FAAH 23 42 O=C(CCNC(=O)Nc1ccc(C2CC2)cc1F)Nc1ccccc1 ZINC000880748491 EH On-Demand Anodyne CCR3 31 41 O=C(CCNC(=O)Nc1ccc(C2CC2)cc1F)Nc1ccccc1 ZINC000880748491 EH On-Demand Anodyne DGAT1 24 42 O=C(NCC(F)(F)c1ccc(F)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880748541 EE On-Demand Anodyne CACNA1G 45 50 O=C(NCC(F)(F)c1ccc(F)cc1)[C@H]1CCc2nncn2CC1 ZINC000880748543 EE On-Demand Anodyne CACNA1G 45 50 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880748597 FI On-Demand Anodyne EPHX2 22 52 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880748597 FI On-Demand Anodyne RBP4 42 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880748598 FI On-Demand Anodyne EPHX2 22 52 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880748598 FI On-Demand Anodyne RBP4 42 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC(C2CCOCC2)C1 ZINC000880748607 DH On-Demand Anodyne RBP4 54 36 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccc(C2CC2)cc1F ZINC000880748608 DH On-Demand Anodyne CDK2 17 53 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccc(C2CC2)cc1F ZINC000880748608 DH On-Demand Anodyne PKNB 68 40 C[C@]1(O)CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748619 DG On-Demand Anodyne CACNA1H 64 38 C=CC(C)(C)CC(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880748624 CG On-Demand Mild HDAC10 35 46 C=CC(C)(C)CC(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880748624 CG On-Demand Mild HDAC2 17 46 C=CC(C)(C)CC(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880748624 CG On-Demand Mild HDAC3 38 46 C=CC(C)(C)CC(=O)Nc1cccc(-c2cn(C)nn2)c1 ZINC000880748624 CG On-Demand Mild HDAC6 32 46 CC1CN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880748651 BG On-Demand Anodyne RBP4 56 37 Cn1cc(-c2cccc(NC(=O)C[C@@H]3C[C@H]3C3CC3)c2)nn1 ZINC000880748666 CF On-Demand Anodyne HDAC10 31 46 Cn1cc(-c2cccc(NC(=O)C[C@@H]3C[C@H]3C3CC3)c2)nn1 ZINC000880748666 CF On-Demand Anodyne HDAC2 16 46 Cn1cc(-c2cccc(NC(=O)C[C@@H]3C[C@H]3C3CC3)c2)nn1 ZINC000880748666 CF On-Demand Anodyne HDAC3 35 46 Cn1cc(-c2cccc(NC(=O)C[C@@H]3C[C@H]3C3CC3)c2)nn1 ZINC000880748666 CF On-Demand Anodyne HDAC6 26 46 O=C(Nc1cnn(Cc2nnc3n2CCCC3)c1)Nc1ccc(C2CC2)cc1F ZINC000880748671 GH On-Demand Anodyne PANC 52 35 C[C@@H]1CN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)CCCO1 ZINC000880748673 EG On-Demand Anodyne ADRA1D 25 45 C[C@@H]1CN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)CCCO1 ZINC000880748673 EG On-Demand Anodyne ADRA1A 46 45 C[C@@H]1CN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)CCCO1 ZINC000880748673 EG On-Demand Anodyne ADRA1B 30 45 C[C@@H]1CN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)CCCO1 ZINC000880748673 EG On-Demand Anodyne CCR3 47 44 C[C@@H]1CN(CCCNC(=O)Nc2ccc(C3CC3)cc2F)CCCO1 ZINC000880748673 EG On-Demand Anodyne MCHR1 21 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880748698 GH On-Demand Anodyne CACNA1I 40 32 O=C(NCCOC(F)(F)F)Nc1ccc(C2CC2)cc1F ZINC000880748706 DG On-Demand Anodyne TRPV1 48 33 CC(C)(C)OC(=O)N1CC2CC1(CNC(=O)c1cccn3nccc13)C2 ZINC000880748721 FE On-Demand Anodyne HCN1 68 31 CC(C)(C)OC(=O)N1CC2CC1(CNC(=O)c1cccn3nccc13)C2 ZINC000880748721 FE On-Demand Anodyne HCN4 47 30 O=C(NCc1ccc(S(=O)(=O)CCO)cc1)Nc1ccc(C2CC2)cc1F ZINC000880748724 GF On-Demand Anodyne TRPV1 41 34 O=C(NCc1ccc(S(=O)(=O)CCO)cc1)Nc1ccc(C2CC2)cc1F ZINC000880748724 GF On-Demand Anodyne NAMPT 41 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCO2)CC1 ZINC000880748728 DG On-Demand Anodyne CACNA1H 55 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(Oc2ncccc2F)CC1 ZINC000880748729 FI On-Demand Anodyne EPHX2 18 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(Oc2ncccc2F)CC1 ZINC000880748729 FI On-Demand Anodyne CALCRL 41 39 O=C(Nc1ccc(C2CC2)cc1F)N(CCc1ccccn1)Cc1cccnc1 ZINC000880748734 GJ On-Demand Anodyne SOAT1 15 43 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(c2nccs2)CC1 ZINC000880748742 FH On-Demand Anodyne EPHX2 28 40 N#C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1c1ccccc1 ZINC000880748749 EI On-Demand Mild RBP4 53 35 Cn1cc(-c2cccc(NC(=O)[C@@H]3C[C@]3(C)c3ccccc3)c2)nn1 ZINC000880748769 EG On-Demand Anodyne HDAC10 21 40 Cn1cc(-c2cccc(NC(=O)[C@@H]3C[C@]3(C)c3ccccc3)c2)nn1 ZINC000880748769 EG On-Demand Anodyne HDAC3 26 40 Cn1cc(-c2cccc(NC(=O)[C@@H]3C[C@]3(C)c3ccccc3)c2)nn1 ZINC000880748769 EG On-Demand Anodyne HDAC6 18 40 CN(C(=O)Nc1ccc(C2CC2)cc1F)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880748810 EH On-Demand Anodyne SLC6A4 18 41 CN(C(=O)Nc1ccc(C2CC2)cc1F)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880748810 EH On-Demand Anodyne SLC6A3 47 41 O=C(Nc1ccc(C2CC2)cc1F)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880748821 EH On-Demand Anodyne EPHX2 56 50 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(Oc2cnccn2)CC1 ZINC000880748822 FH On-Demand Anodyne EPHX2 16 54 O=C(Nc1ccc(C2CC2)cc1F)N1CCOC[C@@H](C2CCC2)C1 ZINC000880748849 EH On-Demand Anodyne RBP4 45 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCOC[C@H](C2CCC2)C1 ZINC000880748851 EH On-Demand Anodyne RBP4 45 34 Cn1cc(-c2cccc(NC(=O)CC[C@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748898 EG On-Demand Anodyne HDAC10 33 45 Cn1cc(-c2cccc(NC(=O)CC[C@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748898 EG On-Demand Anodyne HDAC2 16 45 Cn1cc(-c2cccc(NC(=O)CC[C@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748898 EG On-Demand Anodyne HDAC3 37 45 Cn1cc(-c2cccc(NC(=O)CC[C@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748898 EG On-Demand Anodyne HDAC6 29 45 Cn1cc(-c2cccc(NC(=O)CC[C@@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748899 EG On-Demand Anodyne HDAC10 33 45 Cn1cc(-c2cccc(NC(=O)CC[C@@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748899 EG On-Demand Anodyne HDAC2 16 45 Cn1cc(-c2cccc(NC(=O)CC[C@@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748899 EG On-Demand Anodyne HDAC3 37 45 Cn1cc(-c2cccc(NC(=O)CC[C@@H]3CC(C)(C)CO3)c2)nn1 ZINC000880748899 EG On-Demand Anodyne HDAC6 29 45 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880748902 EG On-Demand Anodyne CCR3 41 37 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880748903 EG On-Demand Anodyne CCR3 41 37 Cn1cc(-c2cccc(NC(=O)c3cnc(CC4CC4)s3)c2)nn1 ZINC000880748908 EG On-Demand Anodyne PTPN2 48 31 Cn1cc(-c2cccc(NC(=O)c3cnc(CC4CC4)s3)c2)nn1 ZINC000880748908 EG On-Demand Anodyne PTPN1 42 31 Cn1ncc(Br)c1CC(=O)Nc1ccc(O[C@@H]2CC2(F)F)cc1 ZINC000880748924 GG On-Demand Anodyne HTR2A 19 40 Cn1ncc(Br)c1CC(=O)Nc1ccc(O[C@H]2CC2(F)F)cc1 ZINC000880748925 GG On-Demand Anodyne HTR2A 19 40 CS(=O)(=O)c1cccnc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748939 FF On-Demand Anodyne TRPV1 79 36 CC(=O)Nc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880748940 EG On-Demand Anodyne TRPV1 16 43 O=C(c1cc2ccccc2cc1F)N1CCC2(COC2)C1 ZINC000880748942 CF On-Demand Anodyne EPHX2 15 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC([C@@H]2CCOC2)C1 ZINC000880748959 DG On-Demand Anodyne RBP4 47 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC([C@H]2CCOC2)C1 ZINC000880748960 DG On-Demand Anodyne RBP4 47 36 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748969 FE On-Demand Anodyne TRPV1 60 35 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748969 FE On-Demand Anodyne HLA-DRB1 55 34 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748970 FE On-Demand Anodyne TRPV1 60 35 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748970 FE On-Demand Anodyne HLA-DRB1 55 34 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880748982 DI On-Demand Anodyne CACNA1H 61 37 CS(=O)(=O)C1(CNC(=O)Nc2ccc(C3CC3)cc2F)CCC1 ZINC000880748986 EF On-Demand Anodyne TRPV1 40 35 CS(=O)(=O)NC[C@@H]1CCC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880748990 FF On-Demand Anodyne TRPV1 43 34 CN(C)S(=O)(=O)C[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)C(F)(F)F ZINC000880749011 GF On-Demand Anodyne TRPV1 44 34 CN(C)S(=O)(=O)C[C@H](NC(=O)Nc1ccc(C2CC2)cc1F)C(F)(F)F ZINC000880749012 GF On-Demand Anodyne TRPV1 44 34 CS(=O)(=O)C1(CNC(=O)Nc2ccc(C3CC3)cc2F)CCCC1 ZINC000880749018 FG On-Demand Anodyne TRPV1 40 35 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(F)(F)CC2)c(O)n1 ZINC000880749052 GG On-Demand Anodyne KCNA3 50 41 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(F)(F)CC2)c(O)n1 ZINC000880749052 GG On-Demand Anodyne HCN1 73 39 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(F)(F)CC2)c(O)n1 ZINC000880749052 GG On-Demand Anodyne HCN4 51 39 NC(=O)Cc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880749053 EG On-Demand Anodyne TRPV1 15 46 CCC[C@]1(CO)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880749060 DH On-Demand Anodyne CACNA1H 44 36 C[C@@H](F)CCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749067 CH On-Demand Anodyne TRPV1 55 35 Cc1cnc(Cl)c(C(=O)NCC2(O)CCC(F)(F)CC2)c1 ZINC000880749077 DF On-Demand Anodyne P2RX7 15 56 CN(C)S(=O)(=O)CCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749078 ED On-Demand Anodyne TRPV1 43 34 C[C@@]1(C#N)CCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880749080 CD On-Demand Mild ACACA 16 50 C[C@]1(C#N)CCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880749081 CD On-Demand Mild ACACA 16 50 CS(=O)(=O)NC[C@H]1CCC[C@@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749091 FF On-Demand Anodyne TRPV1 43 34 CS(=O)(=O)NC[C@H]1CCC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749092 FF On-Demand Anodyne TRPV1 43 34 CS(=O)(=O)NC[C@@H]1CCC[C@@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749093 FF On-Demand Anodyne TRPV1 43 34 O=C(Nc1ccc(O[C@@H]2CC2(F)F)cc1)c1ncsc1C1CC1 ZINC000880749106 EI On-Demand Anodyne MAP1 43 36 O=C(Nc1ccc(O[C@H]2CC2(F)F)cc1)c1ncsc1C1CC1 ZINC000880749107 EI On-Demand Anodyne MAP1 43 36 Cn1cc(-c2cccc(NC(=O)c3ccc(CN4CCOCC4)o3)c2)nn1 ZINC000880749113 FE On-Demand Anodyne CASR 31 40 Cn1cc(-c2cccc(NC(=O)c3ccc(CN4CCOCC4)o3)c2)nn1 ZINC000880749113 FE On-Demand Anodyne HDAC10 23 40 Cn1cc(-c2cccc(NC(=O)c3ccc(CN4CCOCC4)o3)c2)nn1 ZINC000880749113 FE On-Demand Anodyne HDAC3 26 41 Cn1cc(-c2cccc(NC(=O)c3ccc(CN4CCOCC4)o3)c2)nn1 ZINC000880749113 FE On-Demand Anodyne HDAC6 21 41 Cn1cc(-c2cccc(NC(=O)c3ccc(CN4CCOCC4)o3)c2)nn1 ZINC000880749113 FE On-Demand Anodyne EPHX2 18 40 CCn1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1=O ZINC000880749138 EG On-Demand Anodyne P2RX7 47 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCOCC2)CC1 ZINC000880749160 EI On-Demand Anodyne CACNA1H 53 38 Cn1cc(-c2cccc(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)c2)nn1 ZINC000880749161 FG On-Demand Anodyne HDAC10 25 41 Cn1cc(-c2cccc(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)c2)nn1 ZINC000880749161 FG On-Demand Anodyne HDAC3 31 41 Cn1cc(-c2cccc(NC(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)c2)nn1 ZINC000880749161 FG On-Demand Anodyne HDAC6 22 41 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880749190 FH On-Demand Anodyne CACNA1H 40 36 O=C(NCC1(O)CCC(F)(F)CC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880749196 FH On-Demand Anodyne PDE4D 16 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880749203 FI On-Demand Anodyne CACNA1H 62 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880749203 FI On-Demand Anodyne RBP4 57 38 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CCC1(F)F ZINC000880749217 DI On-Demand Anodyne CACNA1H 43 37 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CCC1(F)F ZINC000880749218 DI On-Demand Anodyne CACNA1H 43 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880749248 FI On-Demand Anodyne EPHX2 20 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](c2ccccn2)C1 ZINC000880749252 EI On-Demand Anodyne RBP4 57 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](c2ccccn2)C1 ZINC000880749254 EI On-Demand Anodyne RBP4 57 36 C[C@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749266 FE On-Demand Mild PREP 42 45 C[C@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749266 FE On-Demand Mild LGMN 67 38 C[C@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749266 FE On-Demand Mild SLC12A5 67 35 C[C@@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749269 FE On-Demand Mild PREP 42 45 C[C@@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749269 FE On-Demand Mild LGMN 67 38 C[C@@]1(C#N)CCN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880749269 FE On-Demand Mild SLC12A5 67 35 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880749270 EI On-Demand Mild FKBP1A 24 41 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(C4CC4)cc3F)C2)C1 ZINC000880749287 DG On-Demand Anodyne CACNA1H 40 40 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749355 DH On-Demand Anodyne CCR1 18 42 CN(C)[C@@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749355 DH On-Demand Anodyne RBP4 40 37 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC2(COC2)C1 ZINC000880749361 FD On-Demand Anodyne CELA1 18 40 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC2(COC2)C1 ZINC000880749361 FD On-Demand Anodyne PREP 42 46 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCC2(COC2)C1 ZINC000880749361 FD On-Demand Anodyne SLC12A5 65 36 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)(F)F)c2)nn1 ZINC000880749366 EH On-Demand Anodyne HDAC10 33 46 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)(F)F)c2)nn1 ZINC000880749366 EH On-Demand Anodyne HDAC2 16 46 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)(F)F)c2)nn1 ZINC000880749366 EH On-Demand Anodyne HDAC3 37 46 Cn1cc(-c2cccc(NC(=O)CC(C)(C)CC(F)(F)F)c2)nn1 ZINC000880749366 EH On-Demand Anodyne HDAC6 30 46 Cn1cc(-c2cccc(NC(=O)COC3CC3)c2)nn1 ZINC000880749370 CD On-Demand Anodyne TIMP3 40 31 Cn1cc(-c2cccc(NC(=O)COC3CC3)c2)nn1 ZINC000880749370 CD On-Demand Anodyne HDAC10 40 51 Cn1cc(-c2cccc(NC(=O)COC3CC3)c2)nn1 ZINC000880749370 CD On-Demand Anodyne HDAC2 20 51 Cn1cc(-c2cccc(NC(=O)COC3CC3)c2)nn1 ZINC000880749370 CD On-Demand Anodyne HDAC3 44 51 Cn1cc(-c2cccc(NC(=O)COC3CC3)c2)nn1 ZINC000880749370 CD On-Demand Anodyne HDAC6 36 51 COC1(CO)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749373 DF On-Demand Anodyne CACNA1H 61 37 Cn1cc(-c2cccc(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)c2)nn1 ZINC000880749424 DE On-Demand Anodyne HDAC10 19 40 Cn1cc(-c2cccc(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)c2)nn1 ZINC000880749424 DE On-Demand Anodyne HDAC3 22 40 Cn1cc(-c2cccc(NC(=O)[C@@H]3OC[C@@H]4CCC[C@@H]43)c2)nn1 ZINC000880749424 DE On-Demand Anodyne HDAC6 15 40 N#CC1(c2ccccn2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749450 FI On-Demand Mild CACNA1H 57 40 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCNC3=O)c2)nn1 ZINC000880749460 CC On-Demand Anodyne HDAC10 33 44 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCNC3=O)c2)nn1 ZINC000880749460 CC On-Demand Anodyne HDAC2 17 44 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCNC3=O)c2)nn1 ZINC000880749460 CC On-Demand Anodyne HDAC3 38 44 Cn1cc(-c2cccc(NC(=O)C[C@H]3CCNC3=O)c2)nn1 ZINC000880749460 CC On-Demand Anodyne HDAC6 28 44 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCNC3=O)c2)nn1 ZINC000880749461 CC On-Demand Anodyne HDAC10 33 44 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCNC3=O)c2)nn1 ZINC000880749461 CC On-Demand Anodyne HDAC2 17 44 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCNC3=O)c2)nn1 ZINC000880749461 CC On-Demand Anodyne HDAC3 38 44 Cn1cc(-c2cccc(NC(=O)C[C@@H]3CCNC3=O)c2)nn1 ZINC000880749461 CC On-Demand Anodyne HDAC6 28 44 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(F)(F)CC1 ZINC000880749463 CH On-Demand Anodyne CACNA1H 75 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(F)(F)CC1 ZINC000880749463 CH On-Demand Anodyne RBP4 44 34 O=C1N[C@H]2CCN(C(=O)Nc3ccc(C4CC4)cc3F)C[C@@H]2CO1 ZINC000880749478 EF On-Demand Anodyne RBP4 46 35 CC(C)(C(=O)N1CCC2(COC2)C1)c1ccc(C(F)(F)F)cc1 ZINC000880749513 EG On-Demand Anodyne EPHX2 32 42 O=C(c1cnc2cc[nH]c2c1)N1CCC2(COC2)C1 ZINC000880749515 CD On-Demand Anodyne ACACA 27 55 O=C(c1cnc2cc[nH]c2c1)N1CCC2(COC2)C1 ZINC000880749515 CD On-Demand Anodyne ACACB 17 55 Nc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880749533 DG On-Demand Anodyne NAMPT 17 46 CC1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CCS1(=O)=O ZINC000880749545 FG On-Demand Anodyne CACNA1H 49 37 C[C@@H](O)CCCNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880749556 CF On-Demand Anodyne TRPV1 75 36 CS(=O)(=O)C1(CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749565 EE On-Demand Anodyne TRPV1 70 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CC(F)(F)F)CC1 ZINC000880749569 EJ On-Demand Anodyne RBP4 45 38 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](C(=O)N2CCCC2)C1 ZINC000880749592 EG On-Demand Anodyne RBP4 45 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](C(=O)N2CCCC2)C1 ZINC000880749593 EG On-Demand Anodyne RBP4 45 32 C[S@@](=O)Cc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880749605 FH On-Demand Anodyne TRPV1 16 47 C[S@](=O)Cc1ccc(CNC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880749606 FH On-Demand Anodyne TRPV1 16 47 N#Cc1ccncc1N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749616 FG On-Demand Mild CSF1R 33 41 O=C(NCC1(O)CCC(F)(F)CC1)c1cccn2nccc12 ZINC000880749622 DE On-Demand Anodyne HCN1 65 32 O=C(NCC1(O)CCC(F)(F)CC1)c1cccn2nccc12 ZINC000880749622 DE On-Demand Anodyne HCN4 48 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880749628 FH On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880749629 FH On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](C(F)(F)F)[C@H](CO)C1 ZINC000880749630 FH On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](C(F)(F)F)[C@H](CO)C1 ZINC000880749631 FH On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880749632 FI On-Demand Anodyne CACNA1H 41 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880749632 FI On-Demand Anodyne RBP4 43 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880749633 FI On-Demand Anodyne CACNA1H 41 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880749633 FI On-Demand Anodyne RBP4 43 36 COC(=O)C[C@](C)(NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccn1 ZINC000880749701 FH On-Demand Anodyne P2RY1 23 40 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(C2CC2)cc1F)c1ccccn1 ZINC000880749702 FH On-Demand Anodyne P2RY1 23 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC(C2CC2)C1 ZINC000880749790 CH On-Demand Anodyne RBP4 58 39 CS(=O)(=O)CC1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880749799 FG On-Demand Anodyne EPHX2 22 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880749804 FH On-Demand Anodyne CACNA1H 61 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880749804 FH On-Demand Anodyne EPHX2 23 44 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880749804 FH On-Demand Anodyne RBP4 40 34 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880749805 FH On-Demand Anodyne CACNA1H 61 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880749805 FH On-Demand Anodyne EPHX2 23 44 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880749805 FH On-Demand Anodyne RBP4 40 34 CC(C)(C)OC(=O)N[C@@H]1CCCCC[C@@H]1C(=O)N1CC[C@@](C)(C#N)C1 ZINC000880749818 EG On-Demand Mild CTSK 21 40 CC(C)(C)OC(=O)N[C@@H]1CCCCC[C@@H]1C(=O)N1CC[C@](C)(C#N)C1 ZINC000880749819 EG On-Demand Mild CTSK 21 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880749902 GF On-Demand Clean GABRA1 18 61 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880749910 DG On-Demand Anodyne RBP4 65 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1csc(-c2ncc[nH]2)n1 ZINC000880749917 GE On-Demand Clean NAMPT 28 41 CC(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880749932 EI On-Demand Anodyne TRPV1 15 42 CC(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880749932 EI On-Demand Anodyne CCR3 33 41 CC(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880749932 EI On-Demand Anodyne ROCK2 23 44 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1C[C@H](O)C1 ZINC000880749936 CE On-Demand Anodyne EPHX2 18 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(N3CCC(O)CC3)cc1)C2 ZINC000880749962 GG On-Demand Clean DRD4 45 36 CN(CC(=O)N1CCCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880749969 DF On-Demand Anodyne CCR1 17 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(COC2)C1 ZINC000880749972 CF On-Demand Anodyne CACNA1H 53 38 CN(CCN1CCCCC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880749973 DH On-Demand Anodyne ADRA1A 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H]1C[C@@H](C(=O)OC)C1 ZINC000880749978 FD On-Demand Anodyne CTSK 15 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)[C@H]1C[C@@H](C(=O)OC)C1 ZINC000880749979 FD On-Demand Anodyne CTSK 15 45 O=C(NCC1(O)CCC(F)(F)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880749988 FF On-Demand Anodyne GABRA1 15 49 O=C(NCC1(O)CCC(F)(F)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880749988 FF On-Demand Anodyne MPO 44 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC(O)(c2ccccc2)C1 ZINC000880749993 EG On-Demand Anodyne RBP4 47 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(F)(F)CC1 ZINC000880750007 GD On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(F)(F)CC1 ZINC000880750008 GD On-Demand Anodyne PAPA1_CARPA 39 48 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1c[nH]cc1C1CC1 ZINC000880750088 EF On-Demand Clean HTR1F 47 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@]2(C1)CC2(F)F ZINC000880750096 DH On-Demand Anodyne CACNA1H 41 38 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@]2(C1)CC2(F)F ZINC000880750097 DH On-Demand Anodyne CACNA1H 41 38 O=C1CC[C@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@H]2N1 ZINC000880750110 EF On-Demand Anodyne RBP4 54 36 O=C1CC[C@@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@@H]2N1 ZINC000880750111 EF On-Demand Anodyne RBP4 54 36 O=C1CC[C@@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@H]2N1 ZINC000880750112 EF On-Demand Anodyne RBP4 54 36 O=C1CC[C@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@@H]2N1 ZINC000880750113 EF On-Demand Anodyne RBP4 54 36 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ccc2c(O)ncnc2c1 ZINC000880750118 GE On-Demand Clean NAMPT 28 42 C=CC(C)(C)CC(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880750127 DF On-Demand Mild STAT6 16 41 Cn1nnc(C(=O)NCc2ccc(N3CCC(O)CC3)cc2)n1 ZINC000880750130 DC On-Demand Clean NAMPT 24 40 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CC[C@@H](C)O1 ZINC000880750133 DH On-Demand Anodyne RBP4 40 34 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc2cc[nH]c2c1 ZINC000880750154 FE On-Demand Clean CXCR3 18 43 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc2cc[nH]c2c1 ZINC000880750154 FE On-Demand Clean NAMPT 70 53 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880750158 CH On-Demand Anodyne RBP4 67 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2C[C@H]2C1 ZINC000880750159 CH On-Demand Anodyne RBP4 67 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2C[C@@H]2C1 ZINC000880750160 CH On-Demand Anodyne RBP4 67 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2C[C@H]2C1 ZINC000880750161 CH On-Demand Anodyne RBP4 67 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2cc(Cl)nnc2C1 ZINC000880750164 EH On-Demand Anodyne MAPK1 42 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@]2(CCCOC2)C1 ZINC000880750190 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@]2(CCCOC2)C1 ZINC000880750191 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](n2cccn2)C1 ZINC000880750200 DG On-Demand Anodyne RBP4 45 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](n2cccn2)C1 ZINC000880750201 DG On-Demand Anodyne RBP4 45 32 C[C@@]1(C#N)CCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880750213 CG On-Demand Mild EBP 18 42 C[C@@]1(C#N)CCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880750213 CG On-Demand Mild SSTR1 38 40 C[C@@]1(C#N)CCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880750214 CG On-Demand Mild EBP 18 42 C[C@@]1(C#N)CCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880750214 CG On-Demand Mild SSTR1 38 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(C#N)C1 ZINC000880750224 ED On-Demand Mild PAPA1_CARPA 31 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(C#N)C1 ZINC000880750225 ED On-Demand Mild PAPA1_CARPA 31 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@](C)(C#N)C1 ZINC000880750226 ED On-Demand Mild PAPA1_CARPA 31 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@](C)(C#N)C1 ZINC000880750227 ED On-Demand Mild PAPA1_CARPA 31 41 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CC1)OCCCO2 ZINC000880750241 EG On-Demand Anodyne CACNA1H 47 37 O=C(NCCS(=O)(=O)CC(F)(F)F)Nc1ccc(C2CC2)cc1F ZINC000880750272 FF On-Demand Anodyne TRPV1 88 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880750273 FJ On-Demand Anodyne CACNA1H 65 40 O=C(NCc1cnc(C(F)(F)F)nc1)Nc1ccc(C2CC2)cc1F ZINC000880750278 FH On-Demand Anodyne TRPV1 55 35 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750283 DF On-Demand Anodyne EPHX2 15 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(O)(CO)CC1 ZINC000880750296 DE On-Demand Anodyne CACNA1H 64 38 CC(C)(C)N1CC[C@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750322 EH On-Demand Anodyne CACNA1I 46 33 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750323 EH On-Demand Anodyne CACNA1I 46 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CC1)CC2(F)F ZINC000880750324 DI On-Demand Anodyne CACNA1H 60 39 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc2ccccc2cc1F ZINC000880750349 GH On-Demand Clean STAT6 51 31 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc2ccccc2cc1F ZINC000880750349 GH On-Demand Clean NAMPT 24 41 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880750364 DH On-Demand Anodyne CACNA1H 48 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CO)(CO)C1 ZINC000880750366 DD On-Demand Anodyne CACNA1H 47 38 O=C(Nc1ccc(C2CC2)cc1F)N(CCO)CCOCCO ZINC000880750375 ED On-Demand Anodyne SOAT1 15 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](F)C1 ZINC000880750382 CG On-Demand Anodyne DPP4 20 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](F)C1 ZINC000880750382 CG On-Demand Anodyne RBP4 48 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](F)C1 ZINC000880750383 CG On-Demand Anodyne DPP4 20 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](F)C1 ZINC000880750383 CG On-Demand Anodyne RBP4 48 36 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880750409 DG On-Demand Anodyne RBP4 65 40 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880750410 DG On-Demand Anodyne RBP4 65 40 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880750411 DG On-Demand Anodyne RBP4 65 40 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880750412 DG On-Demand Anodyne RBP4 65 40 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880750413 DG On-Demand Anodyne CHRNA10 54 36 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880750413 DG On-Demand Anodyne ACKR3 67 34 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880750414 DG On-Demand Anodyne CHRNA10 54 36 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880750414 DG On-Demand Anodyne ACKR3 67 34 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2[C@H]3C=C[C@@H](C3)[C@H]2C1 ZINC000880750417 DH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(S)n1-c1ccc(F)cc1 ZINC000880750418 GF On-Demand Anodyne STAT6 56 35 Cc1ccncc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880750426 CH On-Demand Anodyne NAMPT 16 47 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(S)n1-c1ccccc1 ZINC000880750435 GF On-Demand Anodyne PRNP 25 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1cnc(S)n1-c1ccccc1 ZINC000880750435 GF On-Demand Anodyne STAT6 54 36 COc1cccc(C2(NC(=O)CN3CCCCS3(=O)=O)CCC2)c1 ZINC000880750438 FD On-Demand Anodyne DRD4 40 31 O=C(NC[C@H]1CCCN1CCCO)Nc1ccc(C2CC2)cc1F ZINC000880750441 EF On-Demand Anodyne CCR3 17 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCN(CCCO)C1 ZINC000880750442 EF On-Demand Anodyne CCR3 42 43 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCN(CCCO)C1 ZINC000880750443 EF On-Demand Anodyne CCR3 42 43 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1C[C@H](O)C1 ZINC000880750444 CE On-Demand Anodyne EPHX2 18 45 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCC(O)CC2)CC1 ZINC000880750445 EI On-Demand Anodyne CACNA1H 56 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1COCc2ccccc21 ZINC000880750463 EI On-Demand Anodyne TRPV1 16 45 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1COCc2ccccc21 ZINC000880750464 EI On-Demand Anodyne TRPV1 16 45 O=C(NCc1ccc(CO)cc1)Nc1ccc(C2CC2)cc1F ZINC000880750473 DH On-Demand Anodyne TRPV1 16 48 COc1cccc(C2(NC(=O)[C@H]3CCc4nncn4CC3)CCC2)c1 ZINC000880750501 EE On-Demand Anodyne DRD4 41 32 COc1cccc(C2(NC(=O)[C@@H]3CCc4nncn4CC3)CCC2)c1 ZINC000880750502 EE On-Demand Anodyne DRD4 41 32 CC1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC[S@]1=O ZINC000880750524 EG On-Demand Anodyne CACNA1H 53 37 CC1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC[S@@]1=O ZINC000880750525 EG On-Demand Anodyne CACNA1H 53 37 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCc2nnnn2CC1 ZINC000880750536 EE On-Demand Anodyne EPHX2 19 40 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCc2nnnn2CC1 ZINC000880750538 EE On-Demand Anodyne EPHX2 19 40 O=C(NCc1cc(F)cnc1Cl)Nc1ccc(C2CC2)cc1F ZINC000880750543 EI On-Demand Anodyne P2RX7 45 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880750554 FG On-Demand Anodyne L3MBTL3 72 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880750555 FG On-Demand Anodyne L3MBTL3 72 39 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750557 ED On-Demand Anodyne EPHX2 34 47 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750558 ED On-Demand Anodyne EPHX2 34 47 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880750564 EG On-Demand Anodyne RBP4 45 32 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880750565 EG On-Demand Anodyne RBP4 45 32 O=C(NCc1nccc(C(F)(F)F)n1)Nc1ccc(C2CC2)cc1F ZINC000880750572 FH On-Demand Anodyne TRPV1 99 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc(C(F)F)[nH]n1 ZINC000880750586 FE On-Demand Clean NAMPT 27 42 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ncsc1C1CC1 ZINC000880750600 FF On-Demand Clean VHL 42 34 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C)N1CC#N ZINC000880750619 EG On-Demand Mild RBP4 48 36 NC(=O)[C@@H]1CC[C@@H](CNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880750624 EG On-Demand Anodyne VCP 35 41 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C)N1CC#N ZINC000880750626 EG On-Demand Mild RBP4 48 36 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H](C)N1CC#N ZINC000880750628 EG On-Demand Mild RBP4 48 36 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750661 DF On-Demand Anodyne CACNA1H 43 34 COc1cccc(C2(NC(=O)c3nnn(C)n3)CCC2)c1 ZINC000880750662 CD On-Demand Anodyne DRD4 40 31 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCOC1=O ZINC000880750676 CE On-Demand Anodyne LUXR 79 46 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCOC1=O ZINC000880750676 CE On-Demand Anodyne TRAR 92 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCOC1=O ZINC000880750676 CE On-Demand Anodyne LASR 61 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(C2(O)CC2)CC1 ZINC000880750678 DG On-Demand Anodyne CACNA1H 41 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2COC[C@@H]2C1 ZINC000880750690 DG On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880750691 DG On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2COC[C@H]2C1 ZINC000880750692 DG On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2COC[C@H]2C1 ZINC000880750693 DG On-Demand Anodyne RBP4 54 36 COc1cccc(C2(NC(=O)C3CCC(S(C)(=O)=O)CC3)CCC2)c1 ZINC000880750704 FF On-Demand Anodyne MTNR1A 31 42 COc1cccc(C2(NC(=O)C3CCC(S(C)(=O)=O)CC3)CCC2)c1 ZINC000880750704 FF On-Demand Anodyne MTNR1B 26 42 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc(C2CC2)o1 ZINC000880750731 EE On-Demand Clean NAMPT 37 41 O=C1CC(c2ccc(NC(=O)Nc3ccc(C4CC4)cc3F)cc2)CC(=O)N1 ZINC000880750760 GH On-Demand Anodyne DGAT1 17 41 CCN1CC[C@H](N(CC)C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750775 DH On-Demand Anodyne CCR5 16 40 CCN1CC[C@@H](N(CC)C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750777 DH On-Demand Anodyne CCR5 16 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc(CC2CC2)s1 ZINC000880750779 FF On-Demand Clean SIRT3 41 33 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc(CC2CC2)s1 ZINC000880750779 FF On-Demand Clean SIRT1 41 33 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc(CC2CC2)s1 ZINC000880750779 FF On-Demand Clean STAT6 18 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cnc(CC2CC2)s1 ZINC000880750779 FF On-Demand Clean NAMPT 36 43 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750797 DF On-Demand Anodyne EPHX2 15 42 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](c2cccnc2)C1 ZINC000880750812 EI On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](c2cccnc2)C1 ZINC000880750814 EI On-Demand Anodyne RBP4 47 35 C[C@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)N(C)C ZINC000880750827 CG On-Demand Anodyne TRPV1 44 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](O)[C@H](C2CCCC2)C1 ZINC000880750828 EI On-Demand Anodyne RBP4 42 33 C[C@@H](CCNC(=O)Nc1ccc(C2CC2)cc1F)N(C)C ZINC000880750829 CG On-Demand Anodyne TRPV1 44 35 O=C(Nc1ccc(C2CC2)cc1F)NC1CCN(C2CCC2)CC1 ZINC000880750834 EH On-Demand Anodyne EPHX2 38 45 CCN1C[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)CC1=O ZINC000880750843 DE On-Demand Anodyne EPHX2 17 40 COCC1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880750845 DI On-Demand Anodyne EPHX2 33 42 NC(=O)[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1c1ccccc1 ZINC000880750848 FG On-Demand Anodyne RBP4 54 36 NC(=O)[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1c1ccccc1 ZINC000880750848 FG On-Demand Anodyne SMO 29 40 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880750861 GH On-Demand Anodyne RBP4 72 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880750862 GH On-Demand Anodyne RBP4 72 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880750863 GH On-Demand Anodyne RBP4 72 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880750864 GH On-Demand Anodyne RBP4 72 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880750866 DG On-Demand Anodyne SLC6A4 21 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880750866 DG On-Demand Anodyne SLC6A3 55 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880750866 DG On-Demand Anodyne EPHX2 18 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc(C3CC3)cc1F)C2 ZINC000880750866 DG On-Demand Anodyne GLRA1 41 30 COC(=O)[C@@H]1C[C@H](N(C)C(=O)c2cnc(CC3CC3)s2)C1 ZINC000880750872 DE On-Demand Anodyne PTR1 45 33 CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CCC1=O ZINC000880750878 DE On-Demand Anodyne CACNA1H 53 39 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2OCC[C@@H]2C1 ZINC000880750924 DG On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2ccc3cccnc3n2)CC1 ZINC000880750925 GK On-Demand Anodyne SUCNR1 60 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCCC2=O)CC1 ZINC000880750927 EI On-Demand Anodyne CACNA1H 65 38 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880750929 FF On-Demand Clean MERTK 17 41 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880750929 FF On-Demand Clean STAT6 37 42 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880750929 FF On-Demand Clean NAMPT 30 40 Cc1nc(C(C)C)ncc1C(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880750929 FF On-Demand Clean VHL 40 32 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1coc(-c2ccccn2)n1 ZINC000880750950 GF On-Demand Clean METAP1 41 35 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1coc(-c2ccccn2)n1 ZINC000880750950 GF On-Demand Clean STAT6 19 41 COc1ccc(-c2nnc(S)n2CC(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880750954 IE On-Demand Anodyne AVPR1B 35 41 COc1ccc(-c2nnc(S)n2CC(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880750954 IE On-Demand Anodyne MTOR 43 35 COc1ccc(-c2nnc(S)n2CC(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880750954 IE On-Demand Anodyne STAT6 63 36 C[C@H]1C[C@H](CO)CN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880750983 DG On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCSC2(CCC2)CC1 ZINC000880750995 EJ On-Demand Anodyne CACNA1H 45 36 CN1CCC(CNC(=O)Nc2ccc(C3CC3)cc2F)(N2CCOCC2)CC1 ZINC000880751003 GF On-Demand Anodyne HCN1 43 32 O=C1C[C@@H](Oc2cccc(NC(=O)Nc3ccc(C4CC4)cc3F)c2)N1 ZINC000880751014 FH On-Demand Anodyne CCR3 28 40 O=C1C[C@H](Oc2cccc(NC(=O)Nc3ccc(C4CC4)cc3F)c2)N1 ZINC000880751015 FH On-Demand Anodyne CCR3 28 40 COc1cccc(C2(NC(=O)c3cccn4nccc34)CCC2)c1 ZINC000880751023 DG On-Demand Anodyne DRD4 41 31 CCn1cc([C@H](C)NC(=O)Nc2ccc(C3CC3)cc2F)cn1 ZINC000880751027 DH On-Demand Anodyne TRPV1 66 35 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880751034 GI On-Demand Anodyne LPL 41 32 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880751034 GI On-Demand Anodyne CA1 24 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880751034 GI On-Demand Anodyne CA12 20 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880751034 GI On-Demand Anodyne CA9 20 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880751034 GI On-Demand Anodyne P96878_MYCTU 41 36 COc1cccc(C2(NC(=O)c3ccc(CN4CCOCC4)o3)CCC2)c1 ZINC000880751049 FF On-Demand Anodyne DRD4 42 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880751065 EH On-Demand Anodyne CPT1A 46 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880751066 EH On-Demand Anodyne CPT1A 46 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880751069 FI On-Demand Anodyne RBP4 54 35 CS(=O)(=O)CC1(CCNC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751095 FG On-Demand Anodyne TRPV1 43 35 CO[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CCO1 ZINC000880751097 CF On-Demand Anodyne RBP4 40 38 O=C1CC[C@@H](c2ccc(C(=O)NCc3ccc(N4CCC(O)CC4)cc3)cc2)N1 ZINC000880751099 GF On-Demand Clean NAMPT 22 44 O=C1CC[C@H](c2ccc(C(=O)NCc3ccc(N4CCC(O)CC4)cc3)cc2)N1 ZINC000880751100 GF On-Demand Clean NAMPT 22 44 CN(C(=O)Nc1ccc(C2CC2)cc1F)[C@H](CO)Cc1ccccc1 ZINC000880751102 EH On-Demand Anodyne NPY5R 23 41 CN(C(=O)Nc1ccc(C2CC2)cc1F)[C@@H](CO)Cc1ccccc1 ZINC000880751103 EH On-Demand Anodyne NPY5R 23 41 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc(C(F)(F)F)ccn1 ZINC000880751109 GF On-Demand Clean CCR2 71 38 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc(C(F)(F)F)ccn1 ZINC000880751109 GF On-Demand Clean LIPG 48 36 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cc(C(F)(F)F)ccn1 ZINC000880751109 GF On-Demand Clean NAMPT 42 39 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ncccc1-c1ccccn1 ZINC000880751113 GG On-Demand Clean METAP1 41 35 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ncccc1-c1ccccn1 ZINC000880751113 GG On-Demand Clean MERTK 22 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ncccc1-c1ccccn1 ZINC000880751113 GG On-Demand Clean STAT6 17 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880751130 EH On-Demand Anodyne RBP4 42 33 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880751131 EH On-Demand Anodyne RBP4 42 33 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cccn2nccc12 ZINC000880751150 FE On-Demand Clean STAT6 24 41 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1cccn2nccc12 ZINC000880751150 FE On-Demand Clean NAMPT 54 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC(CC2CC2)C1 ZINC000880751158 CH On-Demand Anodyne RBP4 46 35 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880751173 CH On-Demand Anodyne EPHX2 15 46 O=C(Nc1ccc(C2CC2)cc1F)NC1C[C@@H]2C[C@H]2C1 ZINC000880751174 CH On-Demand Anodyne EPHX2 15 46 O=C(Nc1ccc(C2CC2)cc1F)NC1C[C@H]2C[C@@H]2C1 ZINC000880751175 CH On-Demand Anodyne EPHX2 15 46 CC(C)(C[C@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)C1)C(N)=O ZINC000880751190 FH On-Demand Anodyne RBP4 44 32 CC(C)(C[C@@H]1CCCN(C(=O)Nc2ccc(C3CC3)cc2F)C1)C(N)=O ZINC000880751191 FH On-Demand Anodyne RBP4 44 32 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880751219 CH On-Demand Anodyne RBP4 48 36 CS(=O)(=O)CC1(CNC(=O)Nc2ccc(C3CC3)cc2F)CCC1 ZINC000880751288 FG On-Demand Anodyne TRPV1 53 35 COc1cccc(C2(NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)CCC2)c1 ZINC000880751290 FG On-Demand Anodyne DRD4 40 31 COc1cccc(C2(NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)CCC2)c1 ZINC000880751291 FG On-Demand Anodyne DRD4 40 31 CN1CCC[C@@H](CCNC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751303 DH On-Demand Anodyne CCR3 51 39 O=C(Nc1ccc(C2CC2)cc1F)NC1CCC(OC(F)F)CC1 ZINC000880751307 EI On-Demand Anodyne EPHX2 33 43 COc1cccc(C2(NC(=O)c3c4c(nn3C)CCSC4)CCC2)c1 ZINC000880751315 FG On-Demand Anodyne DRD4 40 30 CCOC(=O)C1([S@@](C)=O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751331 GG On-Demand Anodyne CACNA1H 53 34 CCOC(=O)C1([S@](C)=O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751332 GG On-Demand Anodyne CACNA1H 53 34 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751336 FG On-Demand Anodyne CACNA1H 54 35 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751336 FG On-Demand Anodyne RBP4 54 34 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751337 FG On-Demand Anodyne CACNA1H 54 35 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751337 FG On-Demand Anodyne RBP4 54 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880751342 GG On-Demand Bother TRPV1 15 55 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880751342 GG On-Demand Bother RBP4 20 41 CC[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)[C@H](O)C(C)C ZINC000880751345 DH On-Demand Anodyne TRPV1 43 35 CC[C@@H](NC(=O)Nc1ccc(C2CC2)cc1F)[C@@H](O)C(C)C ZINC000880751348 DH On-Demand Anodyne TRPV1 43 35 NC(=O)C1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751351 DD On-Demand Anodyne CACNA1H 68 38 CC[C@@H](CNS(C)(=O)=O)NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880751357 EE On-Demand Anodyne TRPV1 45 35 O=C1C[C@@H](Oc2ccc(NC(=O)Nc3ccc(C4CC4)cc3F)cc2)N1 ZINC000880751385 FH On-Demand Anodyne DGAT1 19 41 O=C1C[C@H](Oc2ccc(NC(=O)Nc3ccc(C4CC4)cc3F)cc2)N1 ZINC000880751386 FH On-Demand Anodyne DGAT1 19 41 C[C@H]1C[C@H](O)CN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751401 CF On-Demand Anodyne RBP4 48 36 C[C@@H]1C[C@H](O)CN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751403 CF On-Demand Anodyne RBP4 48 36 COc1cccc(C2(NC(=O)c3cc(C)cnc3Cl)CCC2)c1 ZINC000880751478 EH On-Demand Anodyne DRD4 41 32 CN(C)C1CCC(NC(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751484 DH On-Demand Anodyne EPHX2 37 44 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880751485 GE On-Demand Clean DPOL_VZVD 23 40 O=C(NCc1ccc(N2CCC(O)CC2)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880751485 GE On-Demand Clean NAMPT 27 40 CS(=O)(=O)c1ccccc1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880751498 FG On-Demand Anodyne TRPV1 95 38 COC[C@@]1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751507 DH On-Demand Anodyne CACNA1H 53 36 COC[C@]1(C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751508 DH On-Demand Anodyne CACNA1H 53 36 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@H](CC(F)(F)F)C1 ZINC000880751536 EJ On-Demand Anodyne RBP4 47 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC[C@@H](CC(F)(F)F)C1 ZINC000880751537 EJ On-Demand Anodyne RBP4 47 34 COC[C@]1(CO)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880751585 DF On-Demand Anodyne CACNA1H 54 37 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880751588 FH On-Demand Anodyne CHRNA4 26 45 CN1C(=O)CC[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1=O ZINC000880751597 DD On-Demand Anodyne NPY1R 20 42 CN1C(=O)CC[C@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1=O ZINC000880751598 DD On-Demand Anodyne NPY1R 20 42 COc1cccc(C2(NC(=O)COC3CC3)CCC2)c1 ZINC000880751603 CE On-Demand Anodyne MTNR1B 40 37 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880751615 GI On-Demand Anodyne TRPM8 32 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880751616 GI On-Demand Anodyne TRPM8 32 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880751617 GI On-Demand Anodyne TRPM8 32 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880751618 GI On-Demand Anodyne TRPM8 32 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC(C(F)(F)F)C1 ZINC000880751620 DH On-Demand Anodyne RBP4 57 38 NC(=O)[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1C(F)(F)F ZINC000880751624 FF On-Demand Anodyne RBP4 46 35 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751627 FI On-Demand Anodyne CACNA1H 65 37 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751627 FI On-Demand Anodyne RBP4 46 39 CS(=O)(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880751632 FG On-Demand Anodyne TRPV1 72 35 CS(=O)(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880751632 FG On-Demand Anodyne ROCK2 15 43 CS(=O)(=O)c1cccc(CNC(=O)Nc2ccc(C3CC3)cc2F)c1 ZINC000880751632 FG On-Demand Anodyne NAMPT 33 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCCC(F)(F)CC1 ZINC000880751638 DI On-Demand Anodyne CACNA1H 64 38 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@@H](CO)[C@H](C(F)(F)F)C1 ZINC000880751642 EG On-Demand Anodyne RBP4 46 35 N#CCCN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751643 DF On-Demand Mild CSF1R 22 43 O=C(NCCO)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751644 EE On-Demand Anodyne EPHX2 15 42 C[C@@H](CNC(=O)Nc1ccc(C2CC2)cc1F)c1ccc(S(C)(=O)=O)cc1 ZINC000880751658 GI On-Demand Anodyne TRPV1 109 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCSCC2)CC1 ZINC000880751678 EJ On-Demand Anodyne CACNA1H 62 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880751694 FE On-Demand Anodyne RBP4 48 36 O=C(NCCC[C@@H]1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880751697 DG On-Demand Anodyne LUXR 53 37 O=C(NCCC[C@@H]1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880751697 DG On-Demand Anodyne TRAR 60 31 O=C(NCCC[C@H]1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880751698 DG On-Demand Anodyne LUXR 53 37 O=C(NCCC[C@H]1CCOC1=O)Nc1ccc(C2CC2)cc1F ZINC000880751698 DG On-Demand Anodyne TRAR 60 31 O=C(CC[C@@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751702 DH On-Demand Anodyne NQO2 21 46 O=C(CC[C@@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751702 DH On-Demand Anodyne MTNR1A 18 43 O=C(CC[C@@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751702 DH On-Demand Anodyne MTNR1B 18 41 O=C(CC[C@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751703 DH On-Demand Anodyne NQO2 21 46 O=C(CC[C@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751703 DH On-Demand Anodyne MTNR1A 18 43 O=C(CC[C@H]1CCc2ccccc21)NCCC1SCCS1 ZINC000880751703 DH On-Demand Anodyne MTNR1B 18 41 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2COC[C@H]2C1 ZINC000880751706 CF On-Demand Anodyne RBP4 56 38 CC(=O)C1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751716 DH On-Demand Anodyne RBP4 40 37 O=C(NCCCc1ccco1)[C@@H]1CCc2nncn2CC1 ZINC000880751721 CD On-Demand Anodyne TBK1 55 32 O=C(NCCCc1ccco1)[C@H]1CCc2nncn2CC1 ZINC000880751722 CD On-Demand Anodyne TBK1 55 32 CS(=O)(=O)C1CCC(C(=O)NCCCc2ccco2)CC1 ZINC000880751735 DD On-Demand Anodyne MTNR1A 23 43 CS(=O)(=O)C1CCC(C(=O)NCCCc2ccco2)CC1 ZINC000880751735 DD On-Demand Anodyne MTNR1B 18 43 O=C(NCCC1SCCS1)c1cnc(CC2CC2)s1 ZINC000880751741 DG On-Demand Anodyne SIRT3 42 35 O=C(NCCC1SCCS1)c1cnc(CC2CC2)s1 ZINC000880751741 DG On-Demand Anodyne SIRT2 45 35 O=C(NCCC1SCCS1)c1cnc(CC2CC2)s1 ZINC000880751741 DG On-Demand Anodyne SIRT1 42 35 CN1CCN(C2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)CC1 ZINC000880751758 FF On-Demand Anodyne L3MBTL3 70 41 Cn1ncc(Br)c1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880751759 FH On-Demand Anodyne HTR2A 18 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CCF)CC1 ZINC000880751777 DI On-Demand Anodyne RBP4 54 40 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880751786 GJ On-Demand Anodyne SMO 39 43 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880751786 GJ On-Demand Anodyne ETHR 65 48 C[S@](=N)(=O)N1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751791 EE On-Demand Anodyne RBP4 49 38 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880751800 FF On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880751801 FF On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880751802 FF On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880751803 FF On-Demand Anodyne RBP4 47 35 CCC1(N2CCOCC2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751841 GH On-Demand Anodyne CACNA1H 50 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880751881 FH On-Demand Anodyne ETHR 59 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880751882 FH On-Demand Anodyne ETHR 59 37 O=C1OC[C@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)C[C@@H]12 ZINC000880751902 DE On-Demand Anodyne RBP4 40 34 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CCO)(CCO)CC1 ZINC000880751907 FG On-Demand Anodyne CACNA1H 63 38 NC(=O)C1(N2CCCCC2)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880751920 GG On-Demand Anodyne CACNA1H 40 36 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CC[C@@H](C(F)(F)F)O1 ZINC000880751926 FI On-Demand Anodyne RBP4 43 35 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CC[C@@H](C(F)(F)F)O1 ZINC000880751927 FI On-Demand Anodyne RBP4 43 35 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CC[C@H](C(F)(F)F)O1 ZINC000880751928 FI On-Demand Anodyne RBP4 43 35 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)CC[C@H](C(F)(F)F)O1 ZINC000880751929 FI On-Demand Anodyne RBP4 43 35 CC(C)c1cc(NC(=O)Nc2ccn(CCF)n2)ccc1O ZINC000880751933 DG On-Demand Anodyne THRA 58 35 CC(C)c1cc(NC(=O)Nc2ccn(CCF)n2)ccc1O ZINC000880751933 DG On-Demand Anodyne THRB 58 38 COc1ccc(CN(CCO)C(=O)Nc2ccn(CCF)n2)cc1 ZINC000880751968 ED On-Demand Anodyne ROCK2 15 41 O=C(CN1CCCCS1(=O)=O)NNc1nc2ccc(Cl)cc2s1 ZINC000880752004 FD On-Demand Reactive CSNK1D 37 41 COc1ccc(CN(CCO)C(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880752029 FH On-Demand Anodyne ROCK2 20 41 COc1ccc(CN(CCO)C(=O)Nc2ccc(C3CC3)cc2F)cc1 ZINC000880752029 FH On-Demand Anodyne SOAT1 16 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC(CNC(=O)C(F)(F)F)C1 ZINC000880752038 FF On-Demand Anodyne RBP4 46 34 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752042 EG On-Demand Anodyne SLC6A4 35 44 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752042 EG On-Demand Anodyne SLC6A3 66 44 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752043 EG On-Demand Anodyne SLC6A4 35 44 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752043 EG On-Demand Anodyne SLC6A3 66 44 CO[C@@H]1C[C@@H](NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880752074 CG On-Demand Anodyne EPHX2 28 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCN(c2nccnn2)CC1 ZINC000880752094 EE On-Demand Anodyne FAAH 24 44 CS(=O)(=O)N[C@@H]1CCCC[C@H]1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880752095 FF On-Demand Anodyne TRPV1 63 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CO)(CO)CC1 ZINC000880752097 DE On-Demand Anodyne CACNA1H 66 39 O=C(Nc1ccc(C2CC2)cc1F)N1CCC(CO)(CO)CC1 ZINC000880752097 DE On-Demand Anodyne RBP4 41 34 CN1CC[C@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@H]21 ZINC000880752103 DG On-Demand Anodyne RBP4 47 35 CN1CC[C@H]2CN(C(=O)Nc3ccc(C4CC4)cc3F)CC[C@@H]21 ZINC000880752104 DG On-Demand Anodyne RBP4 47 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCC1SCCS1 ZINC000880752118 FE On-Demand Anodyne PAPA1_CARPA 38 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCC1SCCS1 ZINC000880752119 FE On-Demand Anodyne PAPA1_CARPA 38 47 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)OCc1ccccc1 ZINC000880752175 GF On-Demand Anodyne CTSL 16 47 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)OCc1ccccc1 ZINC000880752175 GF On-Demand Anodyne TGM2 21 43 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)OCc1ccccc1 ZINC000880752175 GF On-Demand Anodyne F13A1 23 43 O=C(COC1CC1)NNc1nc2ccc(Cl)cc2s1 ZINC000880752202 CF On-Demand Reactive LCK 24 43 O=C(COC1CC1)NNc1nc2ccc(Cl)cc2s1 ZINC000880752202 CF On-Demand Reactive CSNK1D 46 48 O=C(COC1CC1)NNc1nc2ccc(Cl)cc2s1 ZINC000880752202 CF On-Demand Reactive ITK 19 43 O=C(Nc1ccc(C2CC2)cc1F)N1CC(c2ccccc2)C1 ZINC000880752265 DI On-Demand Anodyne RBP4 75 41 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752278 FH On-Demand Anodyne ACKR3 44 30 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)c1 ZINC000880752290 GJ On-Demand Anodyne CACNA1H 41 33 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880752299 EJ On-Demand Anodyne CACNA1H 43 38 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880752299 EJ On-Demand Anodyne RBP4 42 34 O=C(Nc1ccc(C2CC2)cc1F)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880752323 DI On-Demand Anodyne RBP4 56 38 O=C(/C=C\c1ccc2c(c1)OCO2)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880752353 HG On-Demand Anodyne ITGAL 20 41 O=C(/C=C\c1ccc2c(c1)OCO2)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880752353 HG On-Demand Anodyne DYRK2 41 32 COC[C@@H]1CCCN1C(=O)Nc1ccc(C2CC2)cc1F ZINC000880752358 CG On-Demand Anodyne ACKR3 44 30 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880752363 FH On-Demand Anodyne TRPV1 43 33 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1ccc(C2CC2)cc1F ZINC000880752363 FH On-Demand Anodyne P2RX7 22 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1Cc2ccccc2NC1=O ZINC000880752365 EG On-Demand Anodyne PYGM 15 45 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1Cc2ccccc2NC1=O ZINC000880752367 EG On-Demand Anodyne PYGM 15 45 COCC1CC(NC(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880752426 CG On-Demand Anodyne EPHX2 15 40 O=C1CC[C@@H](c2ccc(C(=O)NCc3cc(F)ccc3OC(F)F)cc2)N1 ZINC000880752436 GG On-Demand Anodyne PPARD 15 42 O=C1CC[C@H](c2ccc(C(=O)NCc3cc(F)ccc3OC(F)F)cc2)N1 ZINC000880752437 GG On-Demand Anodyne PPARD 15 42 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2ccn(CCF)n2)C3)c1 ZINC000880752441 FC On-Demand Anodyne P2RX7 24 40 O=C(NCc1cc(F)ccc1OC(F)F)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880752482 GE On-Demand Anodyne P2RX7 26 40 CN1CCN(C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)CC1 ZINC000880752499 ED On-Demand Anodyne L3MBTL3 57 40 COc1ccccc1[C@H]1CCCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880752537 FH On-Demand Anodyne RBP4 41 42 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880752539 FH On-Demand Anodyne RBP4 41 42 Cc1ccccc1[C@@H](C)NC(=O)Nc1ccn(CCF)n1 ZINC000880752544 CG On-Demand Anodyne CTSA 54 37 CC(C)(C)OC(=O)N1[C@H]2CC[C@@H]1C[C@H](CNC(=O)Nc1ccn(CCF)n1)C2 ZINC000880752574 GG On-Demand Anodyne GPR119 20 40 C[C@H](NC(=O)Nc1ccn(CCF)n1)c1nc2cc(Cl)c(Cl)cc2[nH]1 ZINC000880752578 GH On-Demand Anodyne PRCP 30 49 O=C(C[C@H]1CCNC1=O)NNc1nc2ccc(Cl)cc2s1 ZINC000880752594 DD On-Demand Reactive CSNK1D 40 41 O=C(C[C@@H]1CCNC1=O)NNc1nc2ccc(Cl)cc2s1 ZINC000880752596 DD On-Demand Reactive CSNK1D 40 41 O=C(NCCN1CC[C@@H](O)C1)Nc1ccc(C2CC2)cc1F ZINC000880752603 DD On-Demand Anodyne MCHR1 21 43 O=C(NCCN1CC[C@H](O)C1)Nc1ccc(C2CC2)cc1F ZINC000880752605 DD On-Demand Anodyne MCHR1 21 43 CN1CCN(C(=O)Nc2ccc(C3CC3)cc2F)CCC1(C)C ZINC000880752687 DH On-Demand Anodyne CACNA1H 66 41 O=C(NCC[C@@H](O)COCc1ccccc1)Nc1ccn(CCF)n1 ZINC000880752690 FD On-Demand Anodyne ADRB1 41 32 O=C(Nc1ccc(C2CC2)cc1F)N1CCc2nc(C3CC3)ncc2C1 ZINC000880752693 FH On-Demand Anodyne MAPK1 44 34 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880752705 EE On-Demand Anodyne CACNA1H 45 37 N#Cc1ccc(N2CCN(C(=O)Nc3ccc(C4CC4)cc3F)CC2)cn1 ZINC000880752720 FG On-Demand Mild CSF1R 48 37 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880752730 EH On-Demand Anodyne RBP4 44 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880752731 EH On-Demand Anodyne RBP4 44 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752761 FF On-Demand Reactive PAPA1_CARPA 38 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752761 FF On-Demand Reactive CTSK 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752761 FF On-Demand Reactive CTSL 22 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752763 FF On-Demand Reactive PAPA1_CARPA 38 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752763 FF On-Demand Reactive CTSK 22 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(C)c(F)c1 ZINC000880752763 FF On-Demand Reactive CTSL 22 43 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880752804 GE On-Demand Anodyne UTS2R 17 43 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880752804 GE On-Demand Anodyne NPFFR1 45 39 C[C@H](NC(=O)Nc1ccn(CCF)n1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880752814 GG On-Demand Anodyne GPR119 43 42 CS(=O)(=O)C1CCC(C(=O)NNc2nc3ccc(Cl)cc3s2)CC1 ZINC000880752823 GF On-Demand Reactive LCK 29 47 CS(=O)(=O)C1CCC(C(=O)NNc2nc3ccc(Cl)cc3s2)CC1 ZINC000880752823 GF On-Demand Reactive CSNK1D 29 40 C#CCC1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880752828 DG On-Demand Mild CACNA1H 48 36 O=C(NCC1CCN(CC2CC2)CC1)Nc1ccn(CCF)n1 ZINC000880752846 DE On-Demand Anodyne CACNA1I 58 35 O=C(CCCCCn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880752847 JG On-Demand Anodyne HTR7 31 43 O=C(CCCCCn1c(S)nc2ccccc2c1=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880752847 JG On-Demand Anodyne STAT6 52 35 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CC[C@H](O)CC1 ZINC000880752873 CG On-Demand Anodyne EPHX2 30 48 O=C(Nc1ccc(C2CC2)cc1F)N1CCn2cnc(C(F)(F)F)c2C1 ZINC000880752892 FH On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc(NC2CCCC2)c1)Nc1ccn(CCF)n1 ZINC000880752986 EH On-Demand Anodyne CCKBR 51 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880753006 DH On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880753007 DH On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@H]2CSC[C@H]2C1 ZINC000880753009 DH On-Demand Anodyne RBP4 54 36 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880753010 DH On-Demand Anodyne RBP4 54 36 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H]1c1ccc(O)cc1 ZINC000880753015 GH On-Demand Anodyne SLC6A3 42 41 O=C(NCCC1SCCS1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880753066 EF On-Demand Anodyne GABRA1 17 49 O=C(NCCC1SCCS1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880753066 EF On-Demand Anodyne MPO 41 35 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2ccc(C4CC4)cc2F)C3)c1 ZINC000880753087 GF On-Demand Anodyne P2RX7 21 41 CCC1(N(C)C)CCN(C(=O)Nc2ccc(C3CC3)cc2F)CC1 ZINC000880753096 EI On-Demand Anodyne CACNA1H 66 38 COC[C@@H]1CCCN1NC(=O)Nc1ccc(C2CC2)cc1F ZINC000880753117 DF On-Demand Anodyne CASP7 45 35 O=C(NCCC1SCCS1)c1ccc2c(O)ncnc2c1 ZINC000880753131 DE On-Demand Anodyne SIRT3 43 36 O=C(NCCC1SCCS1)c1ccc2c(O)ncnc2c1 ZINC000880753131 DE On-Demand Anodyne SIRT2 47 36 O=C(NCCC1SCCS1)c1ccc2c(O)ncnc2c1 ZINC000880753131 DE On-Demand Anodyne SIRT1 43 36 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2ccc(N3CCOCC3)cn2)C1 ZINC000880753152 GF On-Demand Anodyne MTOR 23 40 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2ccc(N3CCOCC3)cn2)C1 ZINC000880753152 GF On-Demand Anodyne MAPK10 16 40 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2ccc(N3CCOCC3)cn2)C1 ZINC000880753152 GF On-Demand Anodyne GPR119 39 43 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)Nc2ccc(N3CCOCC3)cn2)C1 ZINC000880753152 GF On-Demand Anodyne STAT6 51 31 Cn1ncc(Br)c1CC(=O)NCc1cc(F)ccc1OC(F)F ZINC000880753164 GF On-Demand Anodyne HTR2A 19 41 Cn1ncc(Br)c1CC(=O)NCc1cc(F)ccc1OC(F)F ZINC000880753164 GF On-Demand Anodyne P2RX7 48 52 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccn(CCF)n1 ZINC000880753166 DD On-Demand Anodyne SLC6A4 25 41 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccn(CCF)n1 ZINC000880753166 DD On-Demand Anodyne SLC6A3 50 41 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccn(CCF)n1 ZINC000880753167 DD On-Demand Anodyne SLC6A4 25 41 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1ccn(CCF)n1 ZINC000880753167 DD On-Demand Anodyne SLC6A3 50 41 O=C(Cc1ccccc1N1CCCC1=O)NCc1cc(F)ccc1OC(F)F ZINC000880753168 GG On-Demand Anodyne HTR7 18 40 O=C(Cc1ccccc1N1CCCC1=O)NCc1cc(F)ccc1OC(F)F ZINC000880753168 GG On-Demand Anodyne P2RX7 55 44 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880753173 FG On-Demand Anodyne SLC18A2 47 34 O=C(NC[C@H]1CCCN(CC2CC2)C1)Nc1ccn(CCF)n1 ZINC000880753174 DE On-Demand Anodyne CCR3 73 44 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880753175 FG On-Demand Anodyne SLC18A2 47 34 Cc1nc(C(C)C)ncc1C(=O)NNc1nc2ccc(Cl)cc2s1 ZINC000880753203 FH On-Demand Reactive CSNK1D 27 40 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1ccn(CCF)n1 ZINC000880753252 DG On-Demand Anodyne TRPM8 18 41 Cn1nnc(C(=O)NCc2cc(F)ccc2OC(F)F)n1 ZINC000880753268 DC On-Demand Anodyne P2RX7 40 38 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CC1)COCCO2 ZINC000880753273 EG On-Demand Anodyne CACNA1H 46 37 COc1ccccc1-c1ccc(C(=O)NC[C@H](OC)C2CCCCC2)c(O)n1 ZINC000880753330 GH On-Demand Anodyne NTSR2 18 41 COc1ccccc1-c1ccc(C(=O)NC[C@@H](OC)C2CCCCC2)c(O)n1 ZINC000880753331 GH On-Demand Anodyne NTSR2 18 41 O=C(Nc1ccc(C2CC2)cc1F)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880753341 CD On-Demand Anodyne RBP4 47 34 C[C@@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C)C1(F)F ZINC000880753358 EI On-Demand Anodyne RBP4 47 35 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@@H](C)C1(F)F ZINC000880753360 EI On-Demand Anodyne RBP4 47 35 C[C@H]1CN(C(=O)Nc2ccc(C3CC3)cc2F)C[C@H](C)C1(F)F ZINC000880753362 EI On-Demand Anodyne RBP4 47 35 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCNC2=O)CC1 ZINC000880753366 EF On-Demand Anodyne CACNA1H 70 42 O=C(Nc1ccc(C2CC2)cc1F)N1CCC2(CCNC2=O)CC1 ZINC000880753366 EF On-Demand Anodyne CALCRL 15 46 O=C(NNc1nc2ccc(Cl)cc2s1)c1ccc(CN2CCOCC2)o1 ZINC000880753380 GG On-Demand Reactive CASR 15 47 O=C(NNc1nc2ccc(Cl)cc2s1)c1ccc(CN2CCOCC2)o1 ZINC000880753380 GG On-Demand Reactive LCK 28 47 O=C(NNc1nc2ccc(Cl)cc2s1)c1ccc(CN2CCOCC2)o1 ZINC000880753380 GG On-Demand Reactive DPOL_VZVD 23 42 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880753400 ED On-Demand Anodyne GPR119 40 36 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880753502 DD On-Demand Anodyne CACNA1H 47 37 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C3CC3)cc2F)C1 ZINC000880753520 EH On-Demand Anodyne CACNA1H 55 36 CC1C[C@@H]2CC[C@H](C1)N2C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880753620 DG On-Demand Anodyne MPO 41 33 O=C1C[C@]2(CCCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880753621 FF On-Demand Anodyne EPHX2 17 42 O=C1C[C@@]2(CCCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880753622 FF On-Demand Anodyne EPHX2 17 42 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880753697 GF On-Demand Anodyne CCR3 40 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880753697 GF On-Demand Anodyne EPHX2 27 49 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880753698 GF On-Demand Anodyne CCR3 40 38 O=C(Nc1ccc(C2CC2)cc1F)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880753698 GF On-Demand Anodyne EPHX2 27 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](C(=O)NC(C)C)C1 ZINC000880753723 GD On-Demand Anodyne SSTR2 41 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H](C(=O)NC(C)C)C1 ZINC000880753724 GD On-Demand Anodyne SSTR2 41 38 CC1C[C@@H]2CC[C@H](C1)N2C(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880753752 FE On-Demand Anodyne KCNH2 29 41 CC(C)(C)OC(=O)N1C[C@H](C(=O)N2CCc3nccnc3C2)C(C)(C)C1 ZINC000880753789 FE On-Demand Anodyne GPR119 23 42 CC(C)(C)OC(=O)N1C[C@@H](C(=O)N2CCc3nccnc3C2)C(C)(C)C1 ZINC000880753791 FE On-Demand Anodyne GPR119 23 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](C(=O)NC(C)C)C1 ZINC000880753833 GD On-Demand Anodyne SSTR2 41 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H](C(=O)NC(C)C)C1 ZINC000880753834 GD On-Demand Anodyne SSTR2 41 38 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(c2ccccc2)CC1 ZINC000880753918 FF On-Demand Anodyne KCNA3 47 38 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(c2ccccc2)CC1 ZINC000880753918 FF On-Demand Anodyne SOAT1 17 44 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(OC)c1 ZINC000880754040 GE On-Demand Clean HTR1A 38 44 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(OC)c1 ZINC000880754040 GE On-Demand Clean HTR1D 15 44 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(OC)c1 ZINC000880754040 GE On-Demand Clean HTR1B 17 44 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(OC)c1 ZINC000880754040 GE On-Demand Clean DRD3 41 36 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(OC)c1 ZINC000880754040 GE On-Demand Clean PDGFRB 77 43 COC(=O)c1ccc(CNC(=O)Nc2ccn(CCF)n2)c(F)c1 ZINC000880754190 EE On-Demand Anodyne BDKRB1 27 40 C[C@@](CO)(Cc1ccc(Cl)cc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880754270 FF On-Demand Anodyne PTGES2 55 31 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne DRD4 25 45 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne SIGMAR1 17 40 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne SSTR5 44 35 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne CCR3 32 45 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne UTS2R 22 41 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne CCR2 15 44 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754335 EF On-Demand Anodyne MCHR1 33 47 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne DRD4 25 45 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne SIGMAR1 17 40 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne SSTR5 44 35 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne CCR3 32 45 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne UTS2R 22 41 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne CCR2 15 44 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc1 ZINC000880754336 EF On-Demand Anodyne MCHR1 33 47 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCc2nccnc2C1 ZINC000880754467 GE On-Demand Anodyne GRIN2B 19 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCc2nccnc2C1 ZINC000880754467 GE On-Demand Anodyne PREP 55 47 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCc2nccnc2C1 ZINC000880754467 GE On-Demand Anodyne SLC12A5 50 32 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne DRD2 17 45 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne DRD4 35 45 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne ACHE 61 57 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne HTR4 27 42 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne SIGMAR1 43 43 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne BCHE 18 46 O=C(NCCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880754593 FG On-Demand Anodyne CCR3 60 45 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880754599 DD On-Demand Anodyne HCRTR1 19 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880754618 FH On-Demand Anodyne RBP4 65 32 CC1C[C@@H]2CC[C@H](C1)N2C(=O)c1cnc2cc[nH]c2c1 ZINC000880754705 CF On-Demand Anodyne GLRA1 26 41 Cc1cc(F)ccc1C[C@@H](C)NC(=O)Nc1ccn(CCF)n1 ZINC000880754760 DG On-Demand Anodyne CCR3 40 34 Cc1cc(F)ccc1C[C@H](C)NC(=O)Nc1ccn(CCF)n1 ZINC000880754761 DG On-Demand Anodyne CCR3 40 34 O=C(c1ncsc1C1CC1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880754864 DD On-Demand Anodyne L3MBTL3 65 37 O=C(c1ncsc1C1CC1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880754865 DD On-Demand Anodyne L3MBTL3 65 37 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne P2RY12 167 40 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne KLK3 76 42 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CTSB 55 39 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne TRY2_BOVIN 58 32 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne PAPA1_CARPA 51 35 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CYSP_TRYCR 54 37 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CTSK 32 41 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CTSL 45 36 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CAPNS1 55 33 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne HDAC2 15 43 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne MMP11 43 31 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CAPN1 71 44 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne CAPN2 112 38 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne TGM2 31 47 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne TPSAB1 43 43 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne NPR 46 31 NC(=O)CC[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880754883 JE On-Demand Anodyne Q6PRC7_IXORI 43 35 O=C(c1c[nH]cc1C1CC1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880754904 DD On-Demand Anodyne L3MBTL3 84 42 O=C(c1c[nH]cc1C1CC1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880754905 DD On-Demand Anodyne L3MBTL3 84 42 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880754964 EF On-Demand Anodyne CHRM2 48 40 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880754964 EF On-Demand Anodyne CCR3 32 41 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880754964 EF On-Demand Anodyne L3MBTL3 90 48 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880754965 EF On-Demand Anodyne CHRM2 48 40 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880754965 EF On-Demand Anodyne CCR3 32 41 O=C(c1cc2ccccc2cc1F)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880754965 EF On-Demand Anodyne L3MBTL3 90 48 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880755009 ED On-Demand Anodyne GPR119 40 36 CS(=O)(=O)C1CCC(C(=O)NC2CCC(C3CCC3)CC2)CC1 ZINC000880755018 EG On-Demand Anodyne EPHX2 18 50 O=C(CCn1c(S)nc2ccccc2c1=O)Nc1cc(-c2nnc3n2CCCCC3)ccc1F ZINC000880755023 JH On-Demand Anodyne Q8MHZ5_SHEEP 40 30 O=C(c1cnc(CC2CC2)s1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880755031 ED On-Demand Anodyne CCR3 17 41 O=C(c1cnc(CC2CC2)s1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880755031 ED On-Demand Anodyne L3MBTL3 71 42 O=C(c1cnc(CC2CC2)s1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880755032 ED On-Demand Anodyne CCR3 17 41 O=C(c1cnc(CC2CC2)s1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880755032 ED On-Demand Anodyne L3MBTL3 71 42 O=C(NCc1cccnc1N1CCCC1)Nc1ccn(CCF)n1 ZINC000880755115 EE On-Demand Anodyne SCN2A 17 42 O=C(NCc1cccnc1N1CCCC1)Nc1ccn(CCF)n1 ZINC000880755115 EE On-Demand Anodyne SCN10A 18 42 O=C(N1CCC(N2CC[C@H](O)C2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880755136 EE On-Demand Anodyne L3MBTL3 53 36 O=C(N1CCC(N2CC[C@@H](O)C2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880755137 EE On-Demand Anodyne L3MBTL3 53 36 O=C(c1sc2cccc(F)c2c1Cl)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880755146 GG On-Demand Anodyne L3MBTL3 66 37 O=C(c1sc2cccc(F)c2c1Cl)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880755147 GG On-Demand Anodyne L3MBTL3 66 37 CCN1CC[C@@H](N(CC)C(=O)Nc2ccn(CCF)n2)C1 ZINC000880755189 CD On-Demand Anodyne CCR5 18 44 CCN1CC[C@H](N(CC)C(=O)Nc2ccn(CCF)n2)C1 ZINC000880755190 CD On-Demand Anodyne CCR5 18 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880755203 FH On-Demand Anodyne F10 35 51 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880755203 FH On-Demand Anodyne MAPK14 18 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880755203 FH On-Demand Anodyne PIK3CA 15 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880755203 FH On-Demand Anodyne PRNP 49 45 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880755203 FH On-Demand Anodyne STAT6 53 34 Cc1cnc(Cl)c(C(=O)N2CCC(N3CC[C@@H](O)C3)CC2)c1 ZINC000880755214 DD On-Demand Anodyne L3MBTL3 73 44 Cc1cnc(Cl)c(C(=O)N2CCC(N3CC[C@H](O)C3)CC2)c1 ZINC000880755215 DD On-Demand Anodyne L3MBTL3 73 44 COC(=O)[C@@H]1CN(C(=O)Nc2ccn(CCF)n2)C[C@H]1c1ccc(Cl)cc1 ZINC000880755277 GF On-Demand Anodyne SLC6A4 22 47 COC(=O)[C@@H]1CN(C(=O)Nc2ccn(CCF)n2)C[C@H]1c1ccc(Cl)cc1 ZINC000880755277 GF On-Demand Anodyne SLC6A3 40 47 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880755312 FD On-Demand Anodyne L3MBTL3 76 38 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880755313 FD On-Demand Anodyne L3MBTL3 76 38 CN(C(=O)Nc1ccn(CCF)n1)[C@H](CO)Cc1ccccc1 ZINC000880755327 DD On-Demand Anodyne NPY5R 27 42 CN(C(=O)Nc1ccn(CCF)n1)[C@@H](CO)Cc1ccccc1 ZINC000880755328 DD On-Demand Anodyne NPY5R 27 42 O=C(c1cc(Br)ccc1C1CC1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880755360 GF On-Demand Anodyne L3MBTL3 84 43 O=C(c1cc(Br)ccc1C1CC1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880755361 GF On-Demand Anodyne L3MBTL3 84 43 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880755366 FE On-Demand Anodyne ACHE 22 42 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880755366 FE On-Demand Anodyne HTR4 34 40 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880755366 FE On-Demand Anodyne SIGMAR1 19 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880755366 FE On-Demand Anodyne CCR3 35 44 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880755366 FE On-Demand Anodyne CACNA1I 60 38 O=C(N1CCC(N2CC[C@H](O)C2)CC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880755420 FE On-Demand Anodyne L3MBTL3 43 32 O=C(N1CCC(N2CC[C@@H](O)C2)CC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880755421 FE On-Demand Anodyne L3MBTL3 43 32 C=CC[C@@H]1CCCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880755423 CG On-Demand Mild CCR3 26 43 C=CC[C@@H]1CCCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880755424 CG On-Demand Mild CCR3 26 43 C=CC[C@H]1CCCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880755425 CG On-Demand Mild CCR3 26 43 C=CC[C@H]1CCCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880755426 CG On-Demand Mild CCR3 26 43 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880755428 EE On-Demand Anodyne EPHX2 44 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCOC1(C)C)C2 ZINC000880755637 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCOC1(C)C)C2 ZINC000880755637 DF On-Demand Anodyne MTNR1A 42 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCOC1(C)C)C2 ZINC000880755639 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCOC1(C)C)C2 ZINC000880755639 DF On-Demand Anodyne MTNR1A 42 44 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880755748 FC On-Demand Anodyne HCN1 61 39 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880755748 FC On-Demand Anodyne HCN4 46 30 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880755788 IF On-Demand Anodyne HTR7 15 40 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880755788 IF On-Demand Anodyne PRNP 41 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880755788 IF On-Demand Anodyne STAT6 53 34 O=C1C[C@@]2(CCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880755823 FE On-Demand Anodyne NPY5R 17 42 O=C1C[C@@]2(CCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880755823 FE On-Demand Anodyne EPHX2 16 46 O=C1C[C@]2(CCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880755824 FE On-Demand Anodyne NPY5R 17 42 O=C1C[C@]2(CCN(C(=O)Nc3ccn(CCF)n3)C2)Oc2ccccc21 ZINC000880755824 FE On-Demand Anodyne EPHX2 16 46 CC[C@@H](NC(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880755833 CG On-Demand Anodyne TACR3 53 42 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccn(CCF)n1)C2 ZINC000880755838 CD On-Demand Anodyne HTR3A 32 40 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(N2CCOCC2)CC1 ZINC000880755950 FC On-Demand Anodyne HCN1 69 37 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(N2CCOCC2)CC1 ZINC000880755950 FC On-Demand Anodyne HCN4 47 30 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880755983 GE On-Demand Anodyne NPFFR2 41 42 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880755983 GE On-Demand Anodyne UTS2R 15 41 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880755983 GE On-Demand Anodyne NPFFR1 51 42 O=C(Cc1ccc([N+](=O)[O-])cc1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880756037 GG On-Demand Bother SSTR1 15 40 O=C(Cc1ccc([N+](=O)[O-])cc1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880756037 GG On-Demand Bother KCNJ1 58 47 CC(C)(C(=O)N1CCC(N2CC[C@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756074 GG On-Demand Anodyne SLC6A5 15 40 CC(C)(C(=O)N1CCC(N2CC[C@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756074 GG On-Demand Anodyne MCHR1 18 45 CC(C)(C(=O)N1CCC(N2CC[C@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756074 GG On-Demand Anodyne L3MBTL3 51 34 CC(C)(C(=O)N1CCC(N2CC[C@@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756075 GG On-Demand Anodyne SLC6A5 15 40 CC(C)(C(=O)N1CCC(N2CC[C@@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756075 GG On-Demand Anodyne MCHR1 18 45 CC(C)(C(=O)N1CCC(N2CC[C@@H](O)C2)CC1)c1ccc(C(F)(F)F)cc1 ZINC000880756075 GG On-Demand Anodyne L3MBTL3 51 34 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2ccccc2C(F)(F)F)n1 ZINC000880756078 FE On-Demand Anodyne SLC16A1 42 35 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2ccccc2C(F)(F)F)n1 ZINC000880756078 FE On-Demand Anodyne SLC12A5 41 36 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2ccccc2C(F)(F)F)n1 ZINC000880756080 FE On-Demand Anodyne SLC16A1 42 35 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2ccccc2C(F)(F)F)n1 ZINC000880756080 FE On-Demand Anodyne SLC12A5 41 36 CN(C(=O)Nc1ccn(CCF)n1)c1ccc2c(c1)OCO2 ZINC000880756161 DE On-Demand Anodyne NOS2 65 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCOC1(C)C ZINC000880756271 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCOC1(C)C ZINC000880756272 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCOC1(C)C ZINC000880756273 ED On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCOC1(C)C ZINC000880756274 ED On-Demand Anodyne PAPA1_CARPA 35 43 C[C@@H](CCCc1cccnc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880756293 DF On-Demand Anodyne PTAFR 34 45 COC(=O)[C@@H]1CN(C(=O)Nc2ccn(CCF)n2)C[C@@H]1c1ccccc1 ZINC000880756332 FE On-Demand Anodyne SLC6A3 19 45 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCOC2(C)C)c(O)n1 ZINC000880756382 FG On-Demand Anodyne KCNA3 41 35 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCOC2(C)C)c(O)n1 ZINC000880756383 FG On-Demand Anodyne KCNA3 41 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880756392 GF On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880756393 GF On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@H]21 ZINC000880756394 GF On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1[C@@H]2c3ccc(F)cc3C[C@H]21 ZINC000880756395 GF On-Demand Anodyne PAPA1_CARPA 33 42 C[C@H](NC(=O)Nc1ccn(CCF)n1)C(=O)NCCc1ccccc1 ZINC000880756401 ED On-Demand Anodyne BRS3 25 40 C[C@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880756461 FF On-Demand Anodyne MLNR 50 37 C[C@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880756461 FF On-Demand Anodyne FAAH 20 42 C[C@@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880756462 FF On-Demand Anodyne MLNR 50 37 C[C@@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880756462 FF On-Demand Anodyne FAAH 20 42 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880756487 FF On-Demand Anodyne KCNQ2 34 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@H]21 ZINC000880756488 FF On-Demand Anodyne KCNQ2 34 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880756489 FF On-Demand Anodyne KCNQ2 34 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1[C@@H]2c3ccc(F)cc3C[C@H]21 ZINC000880756490 FF On-Demand Anodyne KCNQ2 34 41 CN1CCC[C@H](NC(=O)Nc2ccn(CCF)n2)c2ccccc21 ZINC000880756537 EF On-Demand Anodyne CCKBR 44 35 C[C@@H](Cc1cccc(F)c1)N(C)C(=O)Nc1ccn(CCF)n1 ZINC000880756565 DG On-Demand Anodyne NPY5R 19 40 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)nc1 ZINC000880756590 ED On-Demand Anodyne PDGFRB 55 38 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)nc1 ZINC000880756590 ED On-Demand Anodyne DGAT1 25 44 C[C@H](NC(=O)Nc1ccn(CCF)n1)C(=O)N1c2ccccc2C[C@H]1C ZINC000880756663 FE On-Demand Anodyne TPP2 61 37 C[C@H](NC(=O)Nc1ccn(CCF)n1)C(=O)N1c2ccccc2C[C@@H]1C ZINC000880756665 FE On-Demand Anodyne TPP2 61 37 O=C(Nc1ccc(Nc2ccccc2)cn1)[C@H]1CCc2nncn2CC1 ZINC000880756670 EG On-Demand Anodyne MAPK10 18 40 O=C(Nc1ccc(Nc2ccccc2)cn1)[C@@H]1CCc2nncn2CC1 ZINC000880756671 EG On-Demand Anodyne MAPK10 18 40 COc1ccc(CN(C)C(=O)Nc2ccn(CCF)n2)cc1Cl ZINC000880756682 EG On-Demand Anodyne PDE6A 46 35 O=C(NC[C@H]1CCCCN1C(=O)C(F)(F)F)Nc1ccn(CCF)n1 ZINC000880756688 FD On-Demand Anodyne HCRTR1 19 46 CCn1c(S)nc2cc(C(=O)Nc3ccc(N4CCOCC4)cn3)ccc2c1=O ZINC000880756701 HE On-Demand Anodyne STAT6 51 31 O=C(NCc1ccc2c(c1)OC(F)(F)O2)Nc1ccn(CCF)n1 ZINC000880756708 EE On-Demand Anodyne KIT 23 44 O=C(NCc1ccc2c(c1)OC(F)(F)O2)Nc1ccn(CCF)n1 ZINC000880756708 EE On-Demand Anodyne BRAF 20 44 O=C(NC[C@H](O)Cc1ccccc1)Nc1ccn(CCF)n1 ZINC000880756717 DD On-Demand Anodyne ADRB1 40 32 O=C(NC[C@@H](O)Cc1ccccc1)Nc1ccn(CCF)n1 ZINC000880756719 DD On-Demand Anodyne ADRB1 40 32 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880756760 FF On-Demand Anodyne CCR3 26 43 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880756760 FF On-Demand Anodyne L3MBTL3 95 44 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880756763 FF On-Demand Anodyne CCR3 26 43 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880756763 FF On-Demand Anodyne L3MBTL3 95 44 CCCN(CCN1CCCCC1)C(=O)Nc1ccn(CCF)n1 ZINC000880756765 EF On-Demand Anodyne CASR 47 37 O=C(NC[C@H]1CCCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880756841 FG On-Demand Anodyne DRD4 20 41 O=C(NC[C@H]1CCCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880756841 FG On-Demand Anodyne SLC6A1 102 34 O=C(NC[C@H]1CCCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880756841 FG On-Demand Anodyne SIGMAR1 22 43 O=C(NC[C@H]1CCCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880756841 FG On-Demand Anodyne CCR3 53 45 O=C(c1cccn2nccc12)N1CCCC[C@H]1CC1CCC1 ZINC000880756898 CH On-Demand Anodyne HCRTR1 24 40 O=C(c1cccn2nccc12)N1CCCC[C@@H]1CC1CCC1 ZINC000880756899 CH On-Demand Anodyne HCRTR1 24 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H](CO)c1ccc(F)cc1F ZINC000880756911 FE On-Demand Anodyne KCNQ2 50 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@H](CO)c1ccc(F)cc1F ZINC000880756912 FE On-Demand Anodyne KCNQ2 50 40 Cc1cc(F)ccc1C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880756968 EH On-Demand Anodyne HTR1F 44 34 O=C(c1ncccc1-c1ccccn1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880756999 FD On-Demand Anodyne CCR3 15 40 O=C(c1ncccc1-c1ccccn1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880756999 FD On-Demand Anodyne L3MBTL3 72 39 O=C(c1ncccc1-c1ccccn1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880757002 FD On-Demand Anodyne CCR3 15 40 O=C(c1ncccc1-c1ccccn1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880757002 FD On-Demand Anodyne L3MBTL3 72 39 COc1cccc([C@H](CO)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880757065 DD On-Demand Anodyne ROCK1 19 45 C=C[C@H](CO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880757073 CD On-Demand Mild NQO2 26 40 C=C[C@H](CO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880757074 CD On-Demand Mild NQO2 26 40 CN(CCN1CCN(Cc2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880757078 GE On-Demand Anodyne ACHE 20 40 C=C[C@H](CO)NC(=O)[C@H]1CCCCC[C@H]1NC(=O)OC(C)(C)C ZINC000880757290 EE On-Demand Mild CTSK 15 47 C=C[C@H](CO)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880757300 DC On-Demand Mild PAPA1_CARPA 36 44 C=C[C@H](CO)NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880757300 DC On-Demand Mild CTSK 18 54 C=C[C@H](CO)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880757301 DC On-Demand Mild PAPA1_CARPA 36 44 C=C[C@H](CO)NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880757301 DC On-Demand Mild CTSK 18 54 C=C[C@H](CO)NC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)c1 ZINC000880757305 GD On-Demand Mild GPR119 32 43 CC(C)(C)OC(=O)N1CCC(CCNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880757338 GG On-Demand Anodyne GPR119 46 44 O=C(COC1CC1)Nc1ccc(Nc2ccccc2)cn1 ZINC000880757348 CF On-Demand Anodyne TIMP3 75 35 CN(C[C@H]1CCCN1C)C(=O)Nc1ccn(CCF)n1 ZINC000880757382 CD On-Demand Anodyne CHRNA10 45 32 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccn(CCF)n1 ZINC000880757383 CD On-Demand Anodyne CHRNA10 45 32 Cc1nc(C(C)C)ncc1C(=O)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880757426 ED On-Demand Anodyne L3MBTL3 68 40 Cc1nc(C(C)C)ncc1C(=O)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880757427 ED On-Demand Anodyne L3MBTL3 68 40 CC(C)(C(=O)N1CCC(N2CC[C@H](O)C2)CC1)c1ccc(F)cc1F ZINC000880757441 FE On-Demand Anodyne L3MBTL3 45 34 CC(C)(C(=O)N1CCC(N2CC[C@@H](O)C2)CC1)c1ccc(F)cc1F ZINC000880757442 FE On-Demand Anodyne L3MBTL3 45 34 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880757460 FD On-Demand Anodyne L3MBTL3 55 36 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880757461 FD On-Demand Anodyne L3MBTL3 55 36 CCCN(CCN1CCCCCC1)C(=O)Nc1ccn(CCF)n1 ZINC000880757490 EF On-Demand Anodyne CASR 47 37 CCCN(CCN1CCCC1)C(=O)Nc1ccn(CCF)n1 ZINC000880757528 DE On-Demand Anodyne CASR 49 38 C=C[C@H](CO)NC(=O)C(C)(C)[C@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880757539 EE On-Demand Mild CTSK 18 43 C=C[C@H](CO)NC(=O)C(C)(C)[C@@H](NC(=O)OC(C)(C)C)C(C)C ZINC000880757541 EE On-Demand Mild CTSK 18 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@]1(C)OC ZINC000880757632 DD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@]1(C)OC ZINC000880757634 DD On-Demand Anodyne PAPA1_CARPA 35 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@]1(C)OC)C2 ZINC000880757636 CE On-Demand Anodyne MTNR1A 43 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)c1ccc(F)cc1F ZINC000880757640 GE On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)c1ccc(F)cc1F ZINC000880757640 GE On-Demand Anodyne FPR1 43 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)c1ccc(F)cc1F ZINC000880757642 GE On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CO)c1ccc(F)cc1F ZINC000880757642 GE On-Demand Anodyne FPR1 43 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)c1ccc(F)cc1F ZINC000880757643 GE On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)c1ccc(F)cc1F ZINC000880757643 GE On-Demand Anodyne FPR1 43 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)c1ccc(F)cc1F ZINC000880757644 GE On-Demand Anodyne PAPA1_CARPA 38 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)c1ccc(F)cc1F ZINC000880757644 GE On-Demand Anodyne FPR1 43 36 N#Cc1cccc(CN2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757740 FF On-Demand Mild DRD4 21 48 N#Cc1cccc(CN2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757740 FF On-Demand Mild SIGMAR1 19 43 N#Cc1cccc(CN2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757740 FF On-Demand Mild SSTR5 45 37 N#Cc1cccc(CN2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757740 FF On-Demand Mild CCR3 42 47 N#Cc1cccc(CN2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757740 FF On-Demand Mild MCHR1 53 48 Cc1cccc(C(C)C)c1NNC(=O)Nc1ccn(CCF)n1 ZINC000880757778 DG On-Demand Reactive SOAT1 40 36 COc1cccc(C2(CNC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757815 EF On-Demand Anodyne KCNA3 43 36 COc1cccc(C2(CNC(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880757815 EF On-Demand Anodyne SOAT1 23 51 COC(=O)Nc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880757826 EE On-Demand Anodyne ROCK2 29 41 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild CTRA_BOVIN 52 31 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild KLK3 61 33 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild PREP 25 43 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild CELA2A 40 31 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild LGMN 73 42 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild CAPN1 45 43 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild TGM2 49 39 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild F13A1 46 39 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild PSMB5 24 40 C=C[C@H](CO)NC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880757834 ED On-Demand Mild Q9NAW4_PLAFA 44 53 O=C(c1cncc2[nH]ccc12)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880757907 DD On-Demand Anodyne L3MBTL3 76 39 O=C(c1cncc2[nH]ccc12)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880757908 DD On-Demand Anodyne L3MBTL3 76 39 CS(=O)(=O)C1CCC(C(=O)Nc2ccc(Nc3ccccc3)cn2)CC1 ZINC000880757945 FG On-Demand Anodyne NPY5R 19 42 O=C(CCC/N=C1/NS(=O)(=O)c2ccccc21)Nc1ccc(N2CCOCC2)cn1 ZINC000880757962 ID On-Demand Mild PRKDC 44 33 COC(=O)[C@@H]1CN(C(=O)Nc2ccn(CCF)n2)C[C@H]1c1ccccc1 ZINC000880757967 FE On-Demand Anodyne SLC6A3 19 45 O=C(c1coc(-c2ccccn2)n1)N1CCCC[C@H]1CC1CCC1 ZINC000880758016 EH On-Demand Anodyne CPT1A 57 40 O=C(c1coc(-c2ccccn2)n1)N1CCCC[C@@H]1CC1CCC1 ZINC000880758017 EH On-Demand Anodyne CPT1A 57 40 Cn1nnc(C(=O)N2CCC[C@@]2(C)Cc2cccc3ccccc23)n1 ZINC000880758020 EF On-Demand Anodyne SLC12A5 44 32 Cn1nnc(C(=O)N2CCC[C@]2(C)Cc2cccc3ccccc23)n1 ZINC000880758021 EF On-Demand Anodyne SLC12A5 44 32 CCN(CC)S(=O)(=O)c1cc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)ccc1F ZINC000880758046 JG On-Demand Anodyne CCR8 31 40 CC(C)(C)C(F)(F)CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880758068 EG On-Demand Anodyne KCNQ2 54 36 CC(C)(C)OC(=O)NC[C@@H]1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880758105 GG On-Demand Anodyne ACACB 15 41 O=C(CC[C@@H]1CCc2ccccc21)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758213 EF On-Demand Anodyne L3MBTL3 45 35 O=C(CC[C@H]1CCc2ccccc21)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758214 EF On-Demand Anodyne L3MBTL3 45 35 O=C(CC[C@H]1CCc2ccccc21)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758215 EF On-Demand Anodyne L3MBTL3 45 35 O=C(CC[C@@H]1CCc2ccccc21)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758216 EF On-Demand Anodyne L3MBTL3 45 35 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880758322 DC On-Demand Anodyne EPHX2 27 46 O=C(NCc1cc(F)cnc1Cl)Nc1ccn(CCF)n1 ZINC000880758363 DE On-Demand Anodyne P2RX7 40 40 CC(C)(C)C(F)(F)CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880758393 FE On-Demand Anodyne CACNA1G 27 44 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880758396 DC On-Demand Anodyne EPHX2 27 46 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880758399 FE On-Demand Anodyne EPHX2 16 43 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880758402 FE On-Demand Anodyne EPHX2 16 43 CNC(=O)COc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880758439 ED On-Demand Anodyne ROCK2 31 40 Cn1nnc(C(=O)N[C@@H]2CCCCc3cc(Br)ccc32)n1 ZINC000880758445 FE On-Demand Anodyne BDKRB1 50 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758446 FF On-Demand Anodyne PAPA1_CARPA 41 51 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758446 FF On-Demand Anodyne CTSK 16 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758446 FF On-Demand Anodyne POLG_HCV1 21 40 Cn1nnc(C(=O)N[C@H]2CCCCc3cc(Br)ccc32)n1 ZINC000880758447 FE On-Demand Anodyne BDKRB1 50 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758448 FF On-Demand Anodyne PAPA1_CARPA 41 51 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758448 FF On-Demand Anodyne CTSK 16 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(F)(F)C(C)(C)C ZINC000880758448 FF On-Demand Anodyne POLG_HCV1 21 40 C=C[C@H](CO)NC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758470 GF On-Demand Mild PAPA1_CARPA 33 43 C=C[C@H](CO)NC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758470 GF On-Demand Mild CTSK 16 40 C=C[C@H](CO)NC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758470 GF On-Demand Mild AMP1_PLAFQ 19 44 C=C[C@H](CO)NC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758472 GF On-Demand Mild PAPA1_CARPA 33 43 C=C[C@H](CO)NC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758472 GF On-Demand Mild CTSK 16 40 C=C[C@H](CO)NC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccc(Br)cc1 ZINC000880758472 GF On-Demand Mild AMP1_PLAFQ 19 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NS(=O)(=O)/C=C\c2ccccc2)cc1 ZINC000880758517 JH On-Demand Anodyne F10 15 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NS(=O)(=O)/C=C\c2ccccc2)cc1 ZINC000880758517 JH On-Demand Anodyne PRNP 56 43 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NS(=O)(=O)/C=C\c2ccccc2)cc1 ZINC000880758517 JH On-Demand Anodyne FLT3 15 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NS(=O)(=O)/C=C\c2ccccc2)cc1 ZINC000880758517 JH On-Demand Anodyne STAT6 58 36 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(NS(=O)(=O)/C=C\c2ccccc2)cc1 ZINC000880758517 JH On-Demand Anodyne DGAT1 20 41 CC[C@@H](NC(=O)Nc1ccn(CCF)n1)c1ccc(OC)c(OC)c1 ZINC000880758556 FG On-Demand Anodyne ENPP1 65 32 O=C(C[C@H]1CCNC1=O)N[C@H]1CCCCc2cc(Br)ccc21 ZINC000880758739 FF On-Demand Anodyne BDKRB1 65 49 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCCCc2cc(Br)ccc21 ZINC000880758740 FF On-Demand Anodyne BDKRB1 65 49 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCCCc2cc(Br)ccc21 ZINC000880758742 FF On-Demand Anodyne BDKRB1 65 49 O=C(C[C@@H]1CCNC1=O)N[C@H]1CCCCc2cc(Br)ccc21 ZINC000880758744 FF On-Demand Anodyne BDKRB1 65 49 O=C1CC[C@@H](c2ccc(C(=O)N[C@H](CO)c3ccc(F)cc3F)cc2)N1 ZINC000880758757 FE On-Demand Anodyne PLD1 44 36 O=C1CC[C@H](c2ccc(C(=O)N[C@H](CO)c3ccc(F)cc3F)cc2)N1 ZINC000880758758 FE On-Demand Anodyne PLD1 44 36 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H](CO)c3ccc(F)cc3F)cc2)N1 ZINC000880758760 FE On-Demand Anodyne PLD1 44 36 O=C1CC[C@H](c2ccc(C(=O)N[C@@H](CO)c3ccc(F)cc3F)cc2)N1 ZINC000880758762 FE On-Demand Anodyne PLD1 44 36 O=C(c1cccn2nccc12)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758817 DD On-Demand Anodyne L3MBTL3 84 47 O=C(c1cccn2nccc12)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758819 DD On-Demand Anodyne L3MBTL3 84 47 O=C(c1cnc2cc[nH]c2c1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758895 DD On-Demand Anodyne CCR3 20 46 O=C(c1cnc2cc[nH]c2c1)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758895 DD On-Demand Anodyne L3MBTL3 95 45 O=C(c1cnc2cc[nH]c2c1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758896 DD On-Demand Anodyne CCR3 20 46 O=C(c1cnc2cc[nH]c2c1)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758896 DD On-Demand Anodyne L3MBTL3 95 45 O=C(c1cccc2nsnc12)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880758919 ED On-Demand Anodyne L3MBTL3 84 45 O=C(c1cccc2nsnc12)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880758920 ED On-Demand Anodyne L3MBTL3 84 45 O=C(NCCCCCN1CCCC1)Nc1ccn(CCF)n1 ZINC000880758949 DE On-Demand Anodyne DRD3 41 36 O=C(NCCCCCN1CCCC1)Nc1ccn(CCF)n1 ZINC000880758949 DE On-Demand Anodyne CHRNA7 22 50 O=C(NCCCCCN1CCCC1)Nc1ccn(CCF)n1 ZINC000880758949 DE On-Demand Anodyne HNMT 48 35 O=C(NC[C@H]1CCCCN1CCO)Nc1ccn(CCF)n1 ZINC000880758964 DC On-Demand Anodyne HCRTR1 15 43 O=C(NCc1ccccc1N1CCCC1)Nc1ccn(CCF)n1 ZINC000880759034 EF On-Demand Anodyne KCNQ2 70 40 O=C(NCc1ccccc1N1CCCC1)Nc1ccn(CCF)n1 ZINC000880759034 EF On-Demand Anodyne SCN2A 17 41 CCSCCCNC(=O)Nc1ccn(CCF)n1 ZINC000880759078 CE On-Demand Anodyne DOT1L 42 33 Cc1ccccc1[C@@]1(F)CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880759120 EG On-Demand Anodyne NPY5R 31 40 CS(=O)(=O)c1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880759172 ED On-Demand Anodyne CARM1 22 43 Cn1nnc(C(=O)N[C@H](CO)c2ccc(F)cc2F)n1 ZINC000880759196 CB On-Demand Anodyne CTSA 44 34 Cn1nnc(C(=O)N[C@@H](CO)c2ccc(F)cc2F)n1 ZINC000880759197 CB On-Demand Anodyne CTSA 44 34 COC(=O)c1ccc(CCNC(=O)Nc2ccn(CCF)n2)c(OC)c1 ZINC000880759217 FE On-Demand Anodyne NQO2 24 40 O=C(NCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759253 EF On-Demand Anodyne HTR1A 18 54 O=C(NCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759253 EF On-Demand Anodyne HTR1D 57 41 O=C(NCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759253 EF On-Demand Anodyne HTR1B 46 54 O=C(NCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759253 EF On-Demand Anodyne SLC6A4 21 48 O=C(NCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759253 EF On-Demand Anodyne MPO 105 48 O=C(c1ccc(CN2CCOCC2)o1)N(CCC1CC1)CC1CC1 ZINC000880759259 EF On-Demand Anodyne ACHE 15 42 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)cc1 ZINC000880759303 JK On-Demand Anodyne HDAC1 28 41 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2cc(-c3nnc4n3CCCCC4)ccc2F)cc1 ZINC000880759303 JK On-Demand Anodyne HDAC2 23 41 COc1cnccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880759342 ED On-Demand Anodyne HTR1A 29 43 COc1cnccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880759342 ED On-Demand Anodyne HTR1D 15 43 COc1cnccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880759342 ED On-Demand Anodyne HTR1B 16 43 COc1cnccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880759342 ED On-Demand Anodyne PDGFRB 56 43 Cc1cnc(Cl)c(C(=O)N(CCC2CC2)CC2CC2)c1 ZINC000880759440 CH On-Demand Anodyne CACNA1I 45 34 Cn1cc(CN(Cc2ccc(Cl)cc2)C(=O)Nc2ccn(CCF)n2)cn1 ZINC000880759539 GG On-Demand Anodyne PLA2G7 64 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccnn1C(C)(C)C)C2 ZINC000880759553 EG On-Demand Anodyne FAAH 15 43 O=C(NCCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759592 EG On-Demand Anodyne HTR1A 22 52 O=C(NCCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759592 EG On-Demand Anodyne HTR1D 70 39 O=C(NCCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759592 EG On-Demand Anodyne HTR1B 61 52 O=C(NCCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759592 EG On-Demand Anodyne SLC6A4 25 52 O=C(NCCCc1c[nH]c2ccc(F)cc12)Nc1ccn(CCF)n1 ZINC000880759592 EG On-Demand Anodyne MPO 111 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccnn1C(C)(C)C ZINC000880759629 FF On-Demand Anodyne CTSK 15 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccnn1C(C)(C)C ZINC000880759629 FF On-Demand Anodyne FPR1 42 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccnn1C(C)(C)C ZINC000880759630 FF On-Demand Anodyne CTSK 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccnn1C(C)(C)C ZINC000880759630 FF On-Demand Anodyne FPR1 42 36 O=C(NCCc1cccc(OCC(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880759717 FG On-Demand Anodyne HRH2 30 40 COC[C@@H](O)CNC(=O)Nc1ccn(CCF)n1 ZINC000880759739 CB On-Demand Anodyne ADRB1 41 34 COc1cc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)ccc1F ZINC000880759812 FE On-Demand Anodyne PDGFRB 51 37 COc1cc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)ccc1F ZINC000880759812 FE On-Demand Anodyne CCR1 25 40 C[C@@]1(CNC(=O)Nc2ccn(CCF)n2)CCN(Cc2ccccc2)C1 ZINC000880759837 FF On-Demand Anodyne NPFFR1 43 37 Cc1ccccc1[C@@H](CC(F)(F)F)NC(=O)Nc1ccn(CCF)n1 ZINC000880760100 FH On-Demand Anodyne CTSA 54 38 Cc1ccccc1[C@H](CC(F)(F)F)NC(=O)Nc1ccn(CCF)n1 ZINC000880760101 FH On-Demand Anodyne CTSA 54 38 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880760108 FD On-Demand Anodyne KCNJ1 40 33 N#Cc1ccc(OC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880760166 FF On-Demand Mild EPHX2 15 49 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne DRD4 32 46 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne ACHE 44 44 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne HTR4 48 46 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne SIGMAR1 35 41 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne CCR3 65 41 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760170 EE On-Demand Anodyne CACNA1I 40 36 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne DRD4 32 46 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne ACHE 44 44 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne HTR4 48 46 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne SIGMAR1 35 41 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne CCR3 65 41 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760171 EE On-Demand Anodyne CACNA1I 40 36 COC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880760176 DD On-Demand Anodyne EPHX2 44 44 O=C(NCCc1ccccc1OC(F)F)Nc1ccn(CCF)n1 ZINC000880760313 EF On-Demand Anodyne ADRB1 40 32 O=C(Nc1cc(C2CCCC2)[nH]n1)Nc1ccn(CCF)n1 ZINC000880760345 DF On-Demand Anodyne PKNB 57 35 O=C(Nc1cc(C2CCCCC2)[nH]n1)Nc1ccn(CCF)n1 ZINC000880760361 DG On-Demand Anodyne PKNB 52 36 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccn(CCF)n1 ZINC000880760380 CE On-Demand Anodyne CDK2 15 52 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccn(CCF)n1 ZINC000880760380 CE On-Demand Anodyne PKNB 71 35 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880760412 FG On-Demand Anodyne SLC18A3 32 42 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880760412 FG On-Demand Anodyne WNT3A 48 36 O=C(NCC1(N2CCOCC2)CC1)Nc1ccn(CCF)n1 ZINC000880760419 DC On-Demand Anodyne HCN1 61 36 O=C(NCC1(N2CCOCC2)CC1)Nc1ccn(CCF)n1 ZINC000880760419 DC On-Demand Anodyne HCN4 47 30 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1ccn(CCF)n1 ZINC000880760421 EF On-Demand Anodyne NPY5R 20 42 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1ccn(CCF)n1 ZINC000880760422 EF On-Demand Anodyne NPY5R 20 42 O=C(Nc1cc(C2CCOCC2)[nH]n1)Nc1ccn(CCF)n1 ZINC000880760441 DE On-Demand Anodyne PKNB 42 31 O=C(NC[C@H]1CCCN(c2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880760524 EF On-Demand Anodyne SLC6A1 62 31 O=C(NCCCc1cccc(Cl)c1)Nc1ccn(CCF)n1 ZINC000880760685 DG On-Demand Anodyne HRH2 21 40 O=C(NCCCc1cccc(Cl)c1)Nc1ccn(CCF)n1 ZINC000880760685 DG On-Demand Anodyne SLC6A5 15 40 O=C1NCC2(CCN(C(=O)Nc3ccn(CCF)n3)CC2)O1 ZINC000880760732 DC On-Demand Anodyne NPY5R 17 44 O=C(c1cc2cc(F)ccc2[nH]c1=O)N1CCC(N2CCOC2=O)CC1 ZINC000880760742 FD On-Demand Anodyne L3MBTL3 52 34 NC(=O)CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880760762 DD On-Demand Anodyne HCN1 62 36 NC(=O)CC1(CNC(=O)c2cccn3nccc23)CCCCC1 ZINC000880760762 DD On-Demand Anodyne HCN4 54 35 C[C@H]1c2ccccc2CCN1C(=O)Nc1ccn(CCF)n1 ZINC000880760821 DG On-Demand Anodyne TRPM8 29 41 O=C(NCCc1c[nH]c2cc(F)ccc12)Nc1ccn(CCF)n1 ZINC000880760831 EF On-Demand Anodyne MPO 83 39 O=C(c1cc(Br)ccc1C1CC1)N1CCC(N2CCOC2=O)CC1 ZINC000880760947 GG On-Demand Anodyne L3MBTL3 49 37 CC(C)c1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880760978 DG On-Demand Anodyne CARM1 44 33 O=C(c1cc2ccccc2cc1F)N1CCC(N2CCOC2=O)CC1 ZINC000880760996 EG On-Demand Anodyne OXTR 37 41 O=C(c1cc2ccccc2cc1F)N1CCC(N2CCOC2=O)CC1 ZINC000880760996 EG On-Demand Anodyne L3MBTL3 54 40 O=C(c1ccc(CN2CCOCC2)o1)N1CCC(N2CCOC2=O)CC1 ZINC000880761027 FD On-Demand Anodyne L3MBTL3 23 43 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1ccn(CCF)n1 ZINC000880761061 FE On-Demand Anodyne CACNA1I 56 37 CC(C)(C)OC(=O)N1CCC[C@@H](NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880761069 FF On-Demand Anodyne GPR119 44 37 CC(C)(C)OC(=O)N1CCC[C@H](NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880761070 FF On-Demand Anodyne GPR119 44 37 NC(=O)CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880761081 EE On-Demand Anodyne HCN1 51 31 NC(=O)CC1(CNC(=O)c2cccc3nsnc23)CCCCC1 ZINC000880761081 EE On-Demand Anodyne HCN4 48 31 Cc1cccc2c1CCC[C@@H]2NC(=O)CN1CCCCS1(=O)=O ZINC000880761101 ED On-Demand Anodyne BDKRB1 54 36 Cc1cccc2c1CCC[C@H]2NC(=O)CN1CCCCS1(=O)=O ZINC000880761102 ED On-Demand Anodyne BDKRB1 54 36 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880761118 DD On-Demand Anodyne CCR8 42 39 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880761119 DD On-Demand Anodyne CCR8 42 39 COc1cccc(C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880761120 EG On-Demand Anodyne MCHR1 27 41 Cc1cccc2c1CCC[C@@H]2NC(=O)COC1CC1 ZINC000880761164 CF On-Demand Anodyne BDKRB1 46 39 Cc1cccc2c1CCC[C@H]2NC(=O)COC1CC1 ZINC000880761165 CF On-Demand Anodyne BDKRB1 46 39 O=C(NC[C@H]1CCCCN1C(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880761185 FF On-Demand Anodyne HCRTR1 28 57 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@H](C4CCCCC4)C3)cc2)N1 ZINC000880761236 FI On-Demand Anodyne L3MBTL3 53 41 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H](C4CCCCC4)C3)cc2)N1 ZINC000880761237 FI On-Demand Anodyne L3MBTL3 53 41 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@H](C4CCCCC4)C3)cc2)N1 ZINC000880761238 FI On-Demand Anodyne L3MBTL3 53 41 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H](C4CCCCC4)C3)cc2)N1 ZINC000880761239 FI On-Demand Anodyne L3MBTL3 53 41 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(N2CCOC2=O)CC1 ZINC000880761264 FD On-Demand Anodyne OXTR 20 46 Cc1cccc2c1CCC[C@@H]2NC(=O)C[C@H]1CCNC1=O ZINC000880761308 CE On-Demand Anodyne BDKRB1 44 46 Cc1cccc2c1CCC[C@H]2NC(=O)C[C@H]1CCNC1=O ZINC000880761309 CE On-Demand Anodyne BDKRB1 44 46 Cc1cccc2c1CCC[C@H]2NC(=O)C[C@@H]1CCNC1=O ZINC000880761310 CE On-Demand Anodyne BDKRB1 44 46 Cc1cccc2c1CCC[C@@H]2NC(=O)C[C@@H]1CCNC1=O ZINC000880761311 CE On-Demand Anodyne BDKRB1 44 46 O=C(NCCCNC(=O)C1CCC1)Nc1ccn(CCF)n1 ZINC000880761378 DD On-Demand Anodyne TBK1 77 35 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCC(N2CCOC2=O)CC1 ZINC000880761385 FF On-Demand Anodyne L3MBTL3 69 38 Cc1cnc(Cl)c(C(=O)NCC2(CC(N)=O)CCCCC2)c1 ZINC000880761389 DF On-Demand Anodyne P2RX7 17 53 Cc1cnc(Cl)c(C(=O)NCC2(CC(N)=O)CCCCC2)c1 ZINC000880761389 DF On-Demand Anodyne HCN1 48 30 Cc1cnc(Cl)c(C(=O)NCC2(CC(N)=O)CCCCC2)c1 ZINC000880761389 DF On-Demand Anodyne HCN4 46 30 O=C(NCCN1CCCOCC1)Nc1ccn(CCF)n1 ZINC000880761414 CC On-Demand Anodyne EPHX2 18 43 CC[C@H]1c2ccccc2CCN1C(=O)Nc1ccn(CCF)n1 ZINC000880761425 DG On-Demand Anodyne TRPM8 27 40 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1ccn(CCF)n1 ZINC000880761426 DG On-Demand Anodyne TRPM8 27 40 O=C(c1c[nH]cc1C1CC1)N1CCC(N2CCOC2=O)CC1 ZINC000880761427 DD On-Demand Anodyne L3MBTL3 47 35 CN1CCC(N2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)CC1 ZINC000880761437 FD On-Demand Anodyne SLC6A5 21 43 O=C(c1cccn2nccc12)N1CCC(N2CCOC2=O)CC1 ZINC000880761454 DD On-Demand Anodyne L3MBTL3 46 40 O=C(c1cccc2nsnc12)N1CCC(N2CCOC2=O)CC1 ZINC000880761492 ED On-Demand Anodyne L3MBTL3 60 39 Cc1noc(C2(C)CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880761536 EE On-Demand Anodyne NPY5R 17 40 CC(C)(C)OC(=O)C1(CNC(=O)c2cccn3nccc23)CCC1 ZINC000880761577 EF On-Demand Anodyne HCN1 73 34 CC(C)(C)OC(=O)C1(CNC(=O)c2cccn3nccc23)CCC1 ZINC000880761577 EF On-Demand Anodyne HCN4 51 33 CCCC[C@@H](NC(=O)Nc1ccn(CCF)n1)C(=O)OC(C)(C)C ZINC000880761585 EF On-Demand Anodyne SSTR2 51 33 CCCC[C@@H](NC(=O)Nc1ccn(CCF)n1)C(=O)OC(C)(C)C ZINC000880761585 EF On-Demand Anodyne CTSK 20 41 CCCC[C@H](NC(=O)Nc1ccn(CCF)n1)C(=O)OC(C)(C)C ZINC000880761586 EF On-Demand Anodyne SSTR2 51 33 CCCC[C@H](NC(=O)Nc1ccn(CCF)n1)C(=O)OC(C)(C)C ZINC000880761586 EF On-Demand Anodyne CTSK 20 41 O=C(c1cnc2cc[nH]c2c1)N1CCC(N2CCOC2=O)CC1 ZINC000880761668 DD On-Demand Anodyne L3MBTL3 67 38 O=C(COc1cccc(C(F)(F)F)c1)NNC(=O)Nc1ccn(CCF)n1 ZINC000880761733 GE On-Demand Reactive PDS 41 36 CC(C)(C)OC(=O)N1CC[C@H]2CC[C@@H](C1)N2C(=O)Nc1ccn(CCF)n1 ZINC000880761734 GF On-Demand Anodyne GPR119 45 36 C[C@@H](CCC1CC1)NC(=O)Nc1ccn(CCF)n1 ZINC000880761822 CF On-Demand Anodyne CCR3 41 35 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccn(CCF)n1 ZINC000880761845 FD On-Demand Anodyne STAT6 43 32 CC[C@@H](NC(=O)Nc1ccn(CCF)n1)c1ncc(-c2ccccc2)[nH]1 ZINC000880761890 FH On-Demand Anodyne HDAC1 15 41 O=C(NCc1ccc(N2CCCS2(=O)=O)cc1)Nc1ccn(CCF)n1 ZINC000880761998 GD On-Demand Anodyne CDK1 17 42 O=C(NCc1cccc(N2CCCS2(=O)=O)c1)Nc1ccn(CCF)n1 ZINC000880762079 GD On-Demand Anodyne CDK1 17 43 Cc1ccccc1[C@@H]1CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880762095 DH On-Demand Anodyne CCR8 45 33 CCN1CCC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880762102 CD On-Demand Anodyne CCR3 29 42 CCN1CCC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880762103 CD On-Demand Anodyne CCR3 29 42 O=C(NCCNC(=O)c1ccccc1F)Nc1ccn(CCF)n1 ZINC000880762138 ED On-Demand Anodyne POLR1A 40 32 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762149 GF On-Demand Anodyne SSTR3 28 41 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762150 GF On-Demand Anodyne SSTR3 28 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762151 GF On-Demand Anodyne SSTR3 28 41 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762152 GF On-Demand Anodyne SSTR3 28 41 CC1(CO)CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880762287 CD On-Demand Anodyne NPY5R 15 41 C[C@H](NC(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880762321 FF On-Demand Anodyne DRD4 26 41 C[C@H](NC(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880762321 FF On-Demand Anodyne SIGMAR1 26 42 C[C@H](NC(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880762323 FF On-Demand Anodyne DRD4 26 41 C[C@H](NC(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880762323 FF On-Demand Anodyne SIGMAR1 26 42 C[C@H]1CN(Cc2ccccc2)C[C@H](C)C1NC(=O)Nc1ccn(CCF)n1 ZINC000880762419 FG On-Demand Anodyne DRD4 17 42 C[C@@H]1CN(Cc2ccccc2)C[C@@H](C)C1NC(=O)Nc1ccn(CCF)n1 ZINC000880762420 FG On-Demand Anodyne DRD4 17 42 C[C@H]1CN(Cc2ccccc2)C[C@@H](C)[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880762421 FG On-Demand Anodyne DRD4 17 42 COC(=O)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880762424 CD On-Demand Anodyne PTR1 45 33 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne ESR1 45 36 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne HRH2 41 41 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne LTA4H 52 45 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne HRH3 47 46 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne PSMB2 41 42 O=C(NCCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880762582 GF On-Demand Anodyne PSMB1 44 42 O=C(N[C@@H]1CCCC[C@H]1NC(=O)[C@@H]1CCc2nncn2CC1)c1ccccc1 ZINC000880762809 GE On-Demand Anodyne SSTR3 28 44 O=C(N[C@@H]1CCCC[C@H]1NC(=O)[C@H]1CCc2nncn2CC1)c1ccccc1 ZINC000880762810 GE On-Demand Anodyne SSTR3 28 44 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762823 ED On-Demand Anodyne SSTR3 32 46 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762825 ED On-Demand Anodyne SSTR3 32 46 CSc1nccnc1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880762835 FF On-Demand Anodyne SSTR3 32 46 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880762935 EE On-Demand Clean PDGFRB 52 37 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763006 FE On-Demand Anodyne CACNA1I 61 35 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763008 FE On-Demand Anodyne CACNA1I 61 35 CC[C@@H](C(=O)NNC(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880763014 EE On-Demand Reactive KCNQ2 43 39 O=C(CCNS(=O)(=O)/C=C\c1ccccc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880763071 HD On-Demand Anodyne STAT6 52 35 O=C(CCNS(=O)(=O)/C=C/c1ccccc1)Nc1ccc(N2CCOCC2)cn1 ZINC000880763073 HD On-Demand Anodyne STAT6 52 35 O=C(COC1CC1)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880763092 DE On-Demand Anodyne SSTR3 35 50 O=C(NCCNc1cccc(Br)c1)Nc1ccn(CCF)n1 ZINC000880763093 FF On-Demand Anodyne EGFR 43 35 CCOC(=O)[C@@]1(C)CCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880763107 DE On-Demand Anodyne JAK3 20 46 CCOC(=O)[C@@]1(C)CCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880763107 DE On-Demand Anodyne JAK1 16 46 CCOC(=O)[C@@]1(C)CCC[C@H]1NC(=O)c1cccn2nccc12 ZINC000880763107 DE On-Demand Anodyne TYK2 24 46 CCOC(=O)[C@@]1(C)CCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880763116 DE On-Demand Anodyne JAK3 20 46 CCOC(=O)[C@@]1(C)CCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880763116 DE On-Demand Anodyne JAK1 16 46 CCOC(=O)[C@@]1(C)CCC[C@@H]1NC(=O)c1cccn2nccc12 ZINC000880763116 DE On-Demand Anodyne TYK2 24 46 O=C(CN1CCCCS1(=O)=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1 ZINC000880763117 GD On-Demand Anodyne SSTR3 31 47 O=C1NCCN(C(=O)Nc2ccn(CCF)n2)[C@H]1c1ccccc1C(F)(F)F ZINC000880763157 GF On-Demand Anodyne RBP4 80 36 O=C1NCCN(C(=O)Nc2ccn(CCF)n2)[C@H]1c1ccccc1C(F)(F)F ZINC000880763157 GF On-Demand Anodyne TRPM8 31 41 O=C1NCCN(C(=O)Nc2ccn(CCF)n2)[C@@H]1c1ccccc1C(F)(F)F ZINC000880763158 GF On-Demand Anodyne RBP4 80 36 O=C1NCCN(C(=O)Nc2ccn(CCF)n2)[C@@H]1c1ccccc1C(F)(F)F ZINC000880763158 GF On-Demand Anodyne TRPM8 31 41 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880763176 HI On-Demand Anodyne OPRK1 24 42 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880763176 HI On-Demand Anodyne SIGMAR1 15 53 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880763176 HI On-Demand Anodyne CCR3 25 49 Cc1cncc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880763191 CD On-Demand Anodyne NAMPT 21 48 O=C(NCc1ccccc1N1CCCCC1)Nc1ccn(CCF)n1 ZINC000880763202 EG On-Demand Anodyne KCNQ2 69 39 O=C(NCc1ccccc1N1CCCCC1)Nc1ccn(CCF)n1 ZINC000880763202 EG On-Demand Anodyne SCN2A 18 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne HTR1A 73 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne DRD2 58 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne ADRA1D 55 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne ADRA1A 50 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne ADRA1B 45 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne DRD3 66 38 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763308 EE On-Demand Anodyne HTR7 54 38 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne HTR1A 73 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne DRD2 58 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne ADRA1D 55 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne ADRA1A 50 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne ADRA1B 45 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne DRD3 66 38 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763310 EE On-Demand Anodyne HTR7 54 38 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1ccn(CCF)n1 ZINC000880763344 DF On-Demand Anodyne NPY5R 19 41 O=C(NCC1(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880763354 DF On-Demand Anodyne NPFFR2 19 41 O=C(NCC1(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880763354 DF On-Demand Anodyne NPFFR1 23 41 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA2 17 47 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne F10 42 47 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA6 19 41 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA1 17 47 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA7 20 41 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne PRNP 30 40 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA13 35 41 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne CA4 15 47 NS(=O)(=O)c1cc(C(=O)Nc2ccc(N3CCOCC3)cn2)ccc1Cl ZINC000880763423 GD On-Demand Anodyne STAT6 56 37 Cc1ccccc1C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880763448 EH On-Demand Anodyne HTR1F 49 38 Cc1ccccc1C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880763448 EH On-Demand Anodyne RBP4 50 42 Cc1ccccc1C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880763448 EH On-Demand Anodyne CCR8 49 33 C[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)[C@@H]1C ZINC000880763567 CF On-Demand Anodyne TRPC6 48 35 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880763568 CF On-Demand Anodyne TRPC6 48 35 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccn(CCF)n3)C2)CC1 ZINC000880763582 GG On-Demand Anodyne EPHX2 23 41 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3ccn(CCF)n3)C2)CC1 ZINC000880763582 GG On-Demand Anodyne GPR119 22 42 CC(C)CN1CCC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763593 EE On-Demand Anodyne CCR3 55 43 CC(C)CN1CCC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763595 EE On-Demand Anodyne CCR3 55 43 Cc1coc(C(=O)N[C@@H]2CCCC[C@H]2NC(=O)c2ccccc2)c1 ZINC000880763613 EG On-Demand Anodyne ADAM17 37 42 Cc1coc(C(=O)N[C@@H]2CCCC[C@H]2NC(=O)c2ccccc2)c1 ZINC000880763613 EG On-Demand Anodyne SSTR3 34 52 Cc1coc(C(=O)N[C@@H]2CCCC[C@H]2NC(=O)c2ccccc2)c1 ZINC000880763613 EG On-Demand Anodyne KCNK3 49 38 COCCCOc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880763622 FF On-Demand Anodyne HRH2 47 41 COCCCOc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880763622 FF On-Demand Anodyne ROCK2 37 47 COc1cc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)ncn1 ZINC000880763696 ED On-Demand Anodyne PDGFRB 72 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763730 EE On-Demand Anodyne DRD4 16 46 C[C@H]1CN(Cc2ccccc2)C[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763731 EE On-Demand Anodyne DRD4 16 46 C[C@H]1CN(Cc2ccccc2)C[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763732 EE On-Demand Anodyne DRD4 16 46 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763733 EE On-Demand Anodyne DRD4 16 46 CC1(C)CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880763734 CF On-Demand Anodyne NPY5R 21 41 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880763738 EE On-Demand Anodyne CAPNS1 51 31 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880763738 EE On-Demand Anodyne CAPN1 47 37 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880763738 EE On-Demand Anodyne CAPN2 65 32 C[C@H](CC(=O)OCc1ccccc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880763738 EE On-Demand Anodyne NPR 55 32 O=C(NCCCc1ccc2c(c1)OCCO2)Nc1ccn(CCF)n1 ZINC000880763868 EE On-Demand Anodyne NOS2 65 33 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880763869 DD On-Demand Anodyne SLC6A1 53 32 CCC(=O)N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763883 CC On-Demand Anodyne EPHX2 33 48 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880763884 CC On-Demand Anodyne EPHX2 33 48 Cn1nc2c(c1C(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1ccccc1)CSCC2 ZINC000880763928 GF On-Demand Anodyne SSTR3 25 41 Cc1coc(C(=O)NC[C@H]2CN(C)CCN2Cc2ccccc2)c1 ZINC000880763929 EE On-Demand Anodyne DRD2 15 42 Cc1coc(C(=O)NC[C@H]2CN(C)CCN2Cc2ccccc2)c1 ZINC000880763929 EE On-Demand Anodyne SIGMAR1 22 42 Cc1coc(C(=O)NC[C@@H]2CN(C)CCN2Cc2ccccc2)c1 ZINC000880763930 EE On-Demand Anodyne DRD2 15 42 Cc1coc(C(=O)NC[C@@H]2CN(C)CCN2Cc2ccccc2)c1 ZINC000880763930 EE On-Demand Anodyne SIGMAR1 22 42 COc1cccc(OCCN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880763940 GE On-Demand Anodyne DRD4 46 35 COc1cccc(OCCN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880763940 GE On-Demand Anodyne PDGFRB 61 38 COc1cccc(OCCN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880763940 GE On-Demand Anodyne FAAH 19 42 COc1cccc(OCCN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880763940 GE On-Demand Anodyne EPHX2 17 41 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763972 ED On-Demand Anodyne CCR3 33 41 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763973 ED On-Demand Anodyne CCR3 33 41 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763974 ED On-Demand Anodyne CCR3 33 41 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880763975 ED On-Demand Anodyne CCR3 33 41 CCc1nc2ccccc2n1C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880764001 GH On-Demand Anodyne FPR2 26 46 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880764069 EF On-Demand Anodyne SLC6A1 42 30 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880764069 EF On-Demand Anodyne LTA4H 17 43 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880764069 EF On-Demand Anodyne SIGMAR1 37 43 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880764069 EF On-Demand Anodyne CCR5 37 47 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880764069 EF On-Demand Anodyne MCHR1 23 41 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880764070 EF On-Demand Anodyne SLC6A1 42 30 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880764070 EF On-Demand Anodyne LTA4H 17 43 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880764070 EF On-Demand Anodyne SIGMAR1 37 43 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880764070 EF On-Demand Anodyne CCR5 37 47 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880764070 EF On-Demand Anodyne MCHR1 23 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764100 FD On-Demand Anodyne HTR1A 47 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764100 FD On-Demand Anodyne CCKAR 39 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764100 FD On-Demand Anodyne CCKBR 57 38 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764101 FD On-Demand Anodyne HTR1A 47 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764101 FD On-Demand Anodyne CCKAR 39 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccn(CCF)n2)C1=O ZINC000880764101 FD On-Demand Anodyne CCKBR 57 38 COCCC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880764102 ED On-Demand Anodyne EPHX2 35 46 COCCC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880764102 ED On-Demand Anodyne CCR8 45 37 COc1cccc(C=C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880764131 FH On-Demand Anodyne DRD4 42 32 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764138 FE On-Demand Anodyne CCR3 17 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764139 FE On-Demand Anodyne CCR3 17 40 CCOc1cc(Cl)ccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880764150 EG On-Demand Anodyne P2RX7 52 39 CCCOc1cccc(CCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764165 EG On-Demand Anodyne HRH2 47 43 CCCOc1cccc(CCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764165 EG On-Demand Anodyne MTNR1A 37 41 COc1cc(CN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc(OC)c1 ZINC000880764224 GE On-Demand Anodyne FAAH 27 48 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880764243 ED On-Demand Anodyne P2RY14 40 32 CC(C)(C)OC(=O)N1CCN(CCCNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880764288 GD On-Demand Anodyne DRD2 23 42 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880764297 FF On-Demand Anodyne SLC6A1 127 34 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880764297 FF On-Demand Anodyne LTA4H 16 42 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880764297 FF On-Demand Anodyne SIGMAR1 31 41 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880764297 FF On-Demand Anodyne CCR5 34 44 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(Cc2ccccc2)C1 ZINC000880764297 FF On-Demand Anodyne BIRC2 19 42 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880764298 FF On-Demand Anodyne SLC6A1 127 34 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880764298 FF On-Demand Anodyne LTA4H 16 42 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880764298 FF On-Demand Anodyne SIGMAR1 31 41 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880764298 FF On-Demand Anodyne CCR5 34 44 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000880764298 FF On-Demand Anodyne BIRC2 19 42 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(N2CCCCC2)CC1 ZINC000880764343 FD On-Demand Anodyne HCN1 79 42 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)(N2CCCCC2)CC1 ZINC000880764343 FD On-Demand Anodyne HCN4 54 35 O=C(NCC1(c2cccc(F)c2)CC1)Nc1ccn(CCF)n1 ZINC000880764354 DF On-Demand Anodyne SOAT1 15 44 Cc1cc(F)ccc1CCNC(=O)Nc1ccn(CCF)n1 ZINC000880764430 DF On-Demand Anodyne P2RX7 33 41 Cc1ccc(CNC(=O)C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880764457 GF On-Demand Anodyne EPHX2 17 41 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764504 EC On-Demand Mild CASR 60 45 C[C@H]1C[C@H](NC(=O)Nc2ccn(CCF)n2)C(=O)N1c1ccccc1 ZINC000880764536 EE On-Demand Anodyne CCKBR 47 35 CC(C)(C)OC(=O)N[C@@H](CNC(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880764557 GG On-Demand Anodyne SOAT1 24 56 C[C@H](NC(=O)Nc1ccn(CCF)n1)c1cccc(N2CCCC2)c1 ZINC000880764643 EG On-Demand Anodyne KCNQ2 43 39 C[C@H]1C[C@H](NC(=O)Nc2ccn(CCF)n2)CCN1Cc1ccccc1 ZINC000880764661 FG On-Demand Anodyne DRD4 17 42 C[C@H]1C[C@H](NC(=O)Nc2ccn(CCF)n2)CCN1Cc1ccccc1 ZINC000880764661 FG On-Demand Anodyne SIGMAR1 19 43 Cc1ccccc1[C@@H](CO)NC(=O)Nc1ccn(CCF)n1 ZINC000880764684 DE On-Demand Anodyne CTSA 56 38 Cc1ccccc1[C@H](CO)NC(=O)Nc1ccn(CCF)n1 ZINC000880764685 DE On-Demand Anodyne CTSA 56 38 COc1ccc(O[C@H](C)CNC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880764784 EE On-Demand Anodyne MTNR1A 18 40 COc1ccc(O[C@@H](C)CNC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880764785 EE On-Demand Anodyne MTNR1A 18 40 CN(CCNC(=O)Nc1ccn(CCF)n1)Cc1ccc(F)cc1 ZINC000880764814 EE On-Demand Anodyne CCR3 16 43 COc1cc(NC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc(OC)c1 ZINC000880764824 GF On-Demand Anodyne PDGFRB 42 34 CC[C@@H]1CCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764845 CF On-Demand Anodyne CCR3 29 45 CC[C@@H]1CCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764846 CF On-Demand Anodyne CCR3 29 45 CC[C@H]1CCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764847 CF On-Demand Anodyne CCR3 29 45 CC[C@H]1CCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880764848 CF On-Demand Anodyne CCR3 29 45 Cc1ccc(C[C@@H](C)N(C)C(=O)Nc2ccn(CCF)n2)cc1 ZINC000880764894 DG On-Demand Anodyne NPY5R 19 41 O=C(Nc1ccc(NC[C@H]2CCCO2)c(F)c1)Nc1ccn(CCF)n1 ZINC000880764938 FG On-Demand Anodyne TNK2 31 41 O=C(Nc1ccc(NC[C@@H]2CCCO2)c(F)c1)Nc1ccn(CCF)n1 ZINC000880764939 FG On-Demand Anodyne TNK2 31 41 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne HTR1A 47 42 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne DRD2 27 42 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne DRD4 24 42 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne DRD3 35 42 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne CASR 48 37 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1ccn(CCF)n1 ZINC000880764947 FE On-Demand Anodyne HTR7 65 46 CCN(Cc1cccc(-c2ccncc2)c1)C(=O)Nc1ccn(CCF)n1 ZINC000880764950 FH On-Demand Anodyne FSHR 42 33 CCN(Cc1cccc(-c2ccncc2)c1)C(=O)Nc1ccn(CCF)n1 ZINC000880764950 FH On-Demand Anodyne ROCK2 16 41 COc1cccc(O[C@H](C)CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764960 EE On-Demand Anodyne MTNR1A 43 53 COc1cccc(O[C@H](C)CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764960 EE On-Demand Anodyne MTNR1B 42 53 COc1cccc(O[C@@H](C)CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764961 EE On-Demand Anodyne MTNR1A 43 53 COc1cccc(O[C@@H](C)CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880764961 EE On-Demand Anodyne MTNR1B 42 53 C[C@H]1CN(Cc2ccccc2)CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880764987 FF On-Demand Anodyne SLC6A1 66 33 C[C@@H]1CN(Cc2ccccc2)CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880764988 FF On-Demand Anodyne SLC6A1 66 33 O=C(NCCNc1ccccc1)Nc1ccn(CCF)n1 ZINC000880765020 CE On-Demand Anodyne ADRB1 40 32 COc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1F ZINC000880765083 FE On-Demand Clean PDGFRB 50 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765103 DD On-Demand Anodyne PGC 46 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765103 DD On-Demand Anodyne PAPA1_CARPA 36 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765103 DD On-Demand Anodyne REN 45 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765104 DD On-Demand Anodyne PGC 46 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765104 DD On-Demand Anodyne PAPA1_CARPA 36 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NOCC1CCC1 ZINC000880765104 DD On-Demand Anodyne REN 45 42 COc1ccc2c(c1)CC[C@H](C(=O)NOCC1CCC1)C2 ZINC000880765105 CF On-Demand Anodyne NQO2 25 41 COc1ccc2c(c1)CC[C@H](C(=O)NOCC1CCC1)C2 ZINC000880765105 CF On-Demand Anodyne MTNR1A 36 41 CC(=O)N(CC(=O)NOCC1CCC1)c1ccccc1 ZINC000880765126 CD On-Demand Anodyne AMY2 44 30 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765129 FD On-Demand Anodyne NPFFR2 40 41 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765129 FD On-Demand Anodyne UTS2R 15 40 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765129 FD On-Demand Anodyne NPFFR1 50 41 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765130 FD On-Demand Anodyne NPFFR2 40 41 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765130 FD On-Demand Anodyne UTS2R 15 40 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765130 FD On-Demand Anodyne NPFFR1 50 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne PAPA1_CARPA 45 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne CCKAR 41 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne CTSK 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne CTSL 24 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne CTSS 16 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765143 FF On-Demand Anodyne FPR1 46 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne PAPA1_CARPA 45 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne CCKAR 41 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne CTSK 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne CTSL 24 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne CTSS 16 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccc(OC)c1C ZINC000880765144 FF On-Demand Anodyne FPR1 46 37 O=C(NOCC1CCC1)c1cccn2nccc12 ZINC000880765156 BD On-Demand Anodyne JAK3 18 41 O=C(NOCC1CCC1)c1cccn2nccc12 ZINC000880765156 BD On-Demand Anodyne TYK2 21 41 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1ccn(CCF)n1 ZINC000880765171 FF On-Demand Anodyne ACHE 43 43 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1ccn(CCF)n1 ZINC000880765171 FF On-Demand Anodyne SIGMAR1 35 42 C[C@@H]1CN(Cc2ccccc2)CCN1C(=O)Nc1ccn(CCF)n1 ZINC000880765196 EF On-Demand Anodyne CCR1 21 40 O=C(NC[C@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1)c1ccccc1 ZINC000880765240 FF On-Demand Anodyne SLC6A1 40 31 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne DRD4 25 42 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne SIGMAR1 15 41 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne SSTR5 52 38 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne CCR3 37 46 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne UTS2R 23 40 COc1cc(CN2CC[C@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765246 GE On-Demand Anodyne MCHR1 27 48 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne DRD4 25 42 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne SIGMAR1 15 41 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne SSTR5 52 38 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne CCR3 37 46 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne UTS2R 23 40 COc1cc(CN2CC[C@@H](NC(=O)Nc3ccn(CCF)n3)C2)cc(OC)c1 ZINC000880765247 GE On-Demand Anodyne MCHR1 27 48 O=C(c1ccc(F)cc1)[C@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880765313 FG On-Demand Anodyne SLC6A1 45 33 O=C(c1ccc(F)cc1)[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880765314 FG On-Demand Anodyne SLC6A1 45 33 C[C@H]1[C@H](C)N(C(=O)c2c[nH]cc2C2CC2)CCN1C(=O)c1c[nH]cc1C1CC1 ZINC000880765320 GG On-Demand Anodyne HTR1F 40 33 C[C@@H]1[C@@H](C)N(C(=O)c2c[nH]cc2C2CC2)CCN1C(=O)c1c[nH]cc1C1CC1 ZINC000880765322 GG On-Demand Anodyne HTR1F 40 33 O=C(NCC(=O)N1CCC(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880765435 GE On-Demand Anodyne IL2RA 50 31 O=C(NCC(=O)N1CCC(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880765435 GE On-Demand Anodyne GRIN2B 65 39 O=C(NCC(=O)N1CCC(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880765435 GE On-Demand Anodyne CCR3 54 45 C[C@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765457 FF On-Demand Anodyne DRD4 33 47 C[C@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765457 FF On-Demand Anodyne SIGMAR1 28 41 C[C@@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765458 FF On-Demand Anodyne DRD4 33 47 C[C@@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765458 FF On-Demand Anodyne SIGMAR1 28 41 C[C@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765459 FF On-Demand Anodyne DRD4 33 47 C[C@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765459 FF On-Demand Anodyne SIGMAR1 28 41 C[C@@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765460 FF On-Demand Anodyne DRD4 33 47 C[C@@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880765460 FF On-Demand Anodyne SIGMAR1 28 41 CC(C)(C)NC(=O)CN1CCC(CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880765461 GD On-Demand Anodyne CACNA1I 68 48 O=C(NCCc1c[nH]c2ccc(Cl)cc12)Nc1ccn(CCF)n1 ZINC000880765569 EG On-Demand Anodyne HTR1D 57 42 O=C(NCCc1c[nH]c2ccc(Cl)cc12)Nc1ccn(CCF)n1 ZINC000880765569 EG On-Demand Anodyne HTR1B 42 44 O=C(NCCc1c[nH]c2ccc(Cl)cc12)Nc1ccn(CCF)n1 ZINC000880765569 EG On-Demand Anodyne MPO 73 36 O=C(NCCc1c[nH]c2ccc(Cl)cc12)Nc1ccn(CCF)n1 ZINC000880765569 EG On-Demand Anodyne MAPT 15 46 COc1ccc(-n2cc(CNC(=O)Nc3ccn(CCF)n3)nn2)cc1 ZINC000880765604 FD On-Demand Anodyne MMP8 32 40 COc1ccc(-n2cc(CNC(=O)Nc3ccn(CCF)n3)nn2)cc1 ZINC000880765604 FD On-Demand Anodyne MMP9 17 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1CC(C)(C)C1 ZINC000880765616 DE On-Demand Anodyne PAPA1_CARPA 36 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1CC(C)(C)C1 ZINC000880765617 DE On-Demand Anodyne PAPA1_CARPA 36 44 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880765663 FF On-Demand Anodyne GPR119 43 38 O=C(NOCC1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880765782 CE On-Demand Anodyne GABRA1 18 44 O=C(NOCC1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880765782 CE On-Demand Anodyne MPO 44 36 O=C(NOCC1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880765782 CE On-Demand Anodyne GABRA2 15 44 CCCCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880765859 DE On-Demand Anodyne SSTR5 41 36 CCCCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880765859 DE On-Demand Anodyne EPHX2 32 40 Cn1ccnc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1=O ZINC000880765876 EC On-Demand Anodyne PDGFRB 44 35 C[C@@H](CNC(=O)Nc1ccn(CCF)n1)Oc1ccc(F)cc1 ZINC000880765887 DF On-Demand Anodyne GCK 15 42 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccn(CCF)n1)C2 ZINC000880765897 DD On-Demand Anodyne HTR3A 38 46 CCCOc1ccc([C@@H](C)NC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880765898 EH On-Demand Anodyne ACACA 22 49 CCCOc1ccc([C@@H](C)NC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880765898 EH On-Demand Anodyne ACACB 23 49 CCCOc1ccc([C@H](C)NC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880765899 EH On-Demand Anodyne ACACA 22 49 CCCOc1ccc([C@H](C)NC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880765899 EH On-Demand Anodyne ACACB 23 49 O=C(NC[C@H]1CCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765908 FF On-Demand Anodyne DRD4 21 41 O=C(NC[C@H]1CCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765908 FF On-Demand Anodyne SLC6A1 107 34 O=C(NC[C@H]1CCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765908 FF On-Demand Anodyne SIGMAR1 23 45 O=C(NC[C@H]1CCCN(Cc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880765908 FF On-Demand Anodyne CCR3 61 47 O=C(NC1CCCCC1)NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880765917 GE On-Demand Anodyne EPHX2 40 45 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880765997 FF On-Demand Anodyne ACACB 15 41 Cc1cccc2c1CCN(C(=O)Nc1ccn(CCF)n1)C2 ZINC000880766007 DF On-Demand Anodyne P2RY14 46 35 Cc1noc(C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880766019 DD On-Demand Anodyne SMO 40 42 Cc1noc(C2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880766019 DD On-Demand Anodyne ETHR 61 36 C[C@H](NC(=O)Nc1ccn(CCF)n1)c1cccnc1 ZINC000880766057 CE On-Demand Anodyne KCNA5 17 41 COc1ccnc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880766085 ED On-Demand Anodyne PDGFRB 46 36 COc1ccnc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880766085 ED On-Demand Anodyne FAAH 23 42 CC(=O)N1CCN(c2ccccc2CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766106 GD On-Demand Anodyne HTR7 27 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne HTR2A 17 40 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne TNF 35 42 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne MAPK14 18 42 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne EPHX2 24 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne MAPK12 20 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne STK10 22 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne EPHA8 16 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne EPHA5 18 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne EPHA4 17 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne TIE1 20 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne DDR2 19 41 O=C(NCc1ccccc1OCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880766125 GD On-Demand Anodyne CDK8 22 41 O=C(NCc1ccc2c(c1)OCCCO2)Nc1ccn(CCF)n1 ZINC000880766142 EE On-Demand Anodyne NOS2 92 37 O=C(Nc1ccc(F)cc1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766146 GF On-Demand Anodyne EPHX2 15 40 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766157 DD On-Demand Anodyne CCR3 15 41 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccn(CCF)n1 ZINC000880766209 GE On-Demand Anodyne SIGMAR1 18 41 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccn(CCF)n1 ZINC000880766209 GE On-Demand Anodyne MCHR1 15 43 CN1CCC(CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766259 CD On-Demand Anodyne CACNA1I 47 35 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne HTR1A 92 43 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne DRD2 76 47 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne DRD4 45 42 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne ADRA1D 77 47 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne HTR1D 15 43 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne HTR1B 18 43 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne ADRA1A 69 47 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne ADRA1B 59 47 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne DRD3 79 43 COc1ccccc1N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766323 FF On-Demand Anodyne HTR7 63 40 C[C@H](CN1CCOCC1)N(Cc1ccccc1)C(=O)Nc1ccn(CCF)n1 ZINC000880766361 GF On-Demand Anodyne CASR 51 38 C[C@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1ccn(CCF)n1 ZINC000880766373 EF On-Demand Anodyne NOS2 98 39 C[C@@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1ccn(CCF)n1 ZINC000880766374 EF On-Demand Anodyne NOS2 98 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne HTR1A 70 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne DRD2 51 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne ADRA1D 46 37 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne ADRA1A 42 36 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne DRD3 61 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766376 FF On-Demand Anodyne HTR7 51 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne HTR1A 70 40 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne DRD2 51 40 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne ADRA1D 46 37 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne ADRA1A 42 36 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne DRD3 61 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766377 FF On-Demand Anodyne HTR7 51 39 O=C(NCCCCCc1ccccc1)Nc1ccn(CCF)n1 ZINC000880766390 DG On-Demand Anodyne FAAH 48 38 O=C(NCCCCCc1ccccc1)Nc1ccn(CCF)n1 ZINC000880766390 DG On-Demand Anodyne CES1 46 35 CC(C)(C)OC(=O)N1CC[C@@H](CCNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766410 FF On-Demand Anodyne GPR119 34 41 CC(C)(C)OC(=O)N1CC[C@H](CCNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880766411 FF On-Demand Anodyne GPR119 34 41 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766412 EE On-Demand Anodyne ADRB1 23 41 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766412 EE On-Demand Anodyne HRH2 45 44 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766412 EE On-Demand Anodyne MTNR1A 27 42 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766412 EE On-Demand Anodyne MTNR1B 22 42 COc1ccc(O)c([C@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766428 DE On-Demand Clean THRA 46 34 COc1ccc(O)c([C@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766428 DE On-Demand Clean THRB 56 35 COc1ccc(O)c([C@@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766429 DE On-Demand Clean THRA 46 34 COc1ccc(O)c([C@@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880766429 DE On-Demand Clean THRB 56 35 Cc1nnc(CN(C)C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)s1 ZINC000880766548 GF On-Demand Anodyne PREP 21 40 COc1ccccc1C[C@@H]1CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880766581 EG On-Demand Anodyne ACKR3 65 33 COc1ccccc1C[C@H]1CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880766582 EG On-Demand Anodyne ACKR3 65 33 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766609 FF On-Demand Anodyne CCR3 16 44 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766609 FF On-Demand Anodyne CCKBR 54 35 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766609 FF On-Demand Anodyne EPHX2 47 47 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766621 FE On-Demand Anodyne EPHX2 42 41 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766621 FE On-Demand Anodyne GPR119 47 38 CC(C)(CNC(=O)Nc1ccn(CCF)n1)c1ccc(F)cc1 ZINC000880766627 DG On-Demand Anodyne CACNA1G 23 41 Cc1cnc(Cl)c(C(=O)N2CCn3c(nnc3C(C)(C)C)C2)c1 ZINC000880766641 EF On-Demand Anodyne P2RX7 44 44 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne DRD4 19 41 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne HTR1D 20 40 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne HTR1B 15 40 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne HTR4 33 47 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne SIGMAR1 23 40 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766644 FF On-Demand Anodyne CCR3 54 45 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne DRD4 19 41 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne HTR1D 20 40 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne HTR1B 15 40 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne HTR4 33 47 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne SIGMAR1 23 40 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1ccn(CCF)n1 ZINC000880766645 FF On-Demand Anodyne CCR3 54 45 COc1ccnc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880766658 ED On-Demand Anodyne PDGFRB 55 38 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne ESR1 72 36 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne HRH2 33 40 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne ESR2 50 36 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne LTA4H 54 45 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne HRH3 55 45 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne FLT3 16 42 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne PSMB2 42 44 O=C(NCc1ccc(OCCN2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880766660 GF On-Demand Anodyne PSMB1 46 44 O=C(NCCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880766661 EG On-Demand Anodyne CCKAR 42 38 O=C(NCCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880766661 EG On-Demand Anodyne MPO 63 35 O=C(NCCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880766661 EG On-Demand Anodyne NMBR 32 40 O=C(NCCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880766661 EG On-Demand Anodyne MC1R 40 36 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccn(CCF)n1 ZINC000880766666 FE On-Demand Anodyne BMP1 46 35 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccn(CCF)n1 ZINC000880766666 FE On-Demand Anodyne NOS2 75 34 O=C(Nc1ccc(N2CCOCC2)cn1)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880766667 JF On-Demand Anodyne EPHX2 20 46 O=C(Nc1ccc(N2CCOCC2)cn1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880766668 JF On-Demand Anodyne EPHX2 20 46 O=C(NC[C@H](O)COc1ccc(F)c(F)c1)Nc1ccn(CCF)n1 ZINC000880766681 FD On-Demand Anodyne ADRB1 46 34 O=C(NC[C@@H](O)COc1ccc(F)c(F)c1)Nc1ccn(CCF)n1 ZINC000880766682 FD On-Demand Anodyne ADRB1 46 34 COc1ccc(N2CCC(NC(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880766716 FF On-Demand Clean PDK1 43 31 CCOc1ccccc1CCNC(=O)Nc1ccn(CCF)n1 ZINC000880766736 DF On-Demand Anodyne HCN1 47 33 N#Cc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(F)c1 ZINC000880766752 FE On-Demand Mild SLC6A9 15 42 CCN(Cc1ccc(OC)cc1OC)C(=O)Nc1ccn(CCF)n1 ZINC000880766769 FF On-Demand Anodyne PDGFRB 33 43 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766791 FE On-Demand Anodyne ACACB 15 42 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766791 FE On-Demand Anodyne CACNA1I 52 33 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766792 FE On-Demand Anodyne ACACB 15 42 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766792 FE On-Demand Anodyne CACNA1I 52 33 CN(Cc1ccc(F)cc1Cl)C(=O)Nc1ccn(CCF)n1 ZINC000880766827 EG On-Demand Anodyne P2RX7 43 42 Cc1nc(C(C)C)ncc1C(=O)N1CCn2c(nnc2C(C)(C)C)C1 ZINC000880766853 EE On-Demand Anodyne P2RX7 37 40 O=C(Nc1ccc(F)cc1)N[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766860 GE On-Demand Anodyne CCR3 41 45 O=C(Nc1ccc(F)cc1)N[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766860 GE On-Demand Anodyne EPHX2 39 42 O=C(Nc1ccc(F)cc1)N[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766861 GE On-Demand Anodyne CCR3 41 45 O=C(Nc1ccc(F)cc1)N[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880766861 GE On-Demand Anodyne EPHX2 39 42 C[C@@H](Cn1cncn1)NC(=O)Nc1ccn(CCF)n1 ZINC000880766877 CC On-Demand Anodyne HIS3 85 39 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880766881 ED On-Demand Anodyne HCN1 63 38 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880766881 ED On-Demand Anodyne HCN4 49 31 CN(CCN1CCOCC1)C(=O)Nc1ccn(CCF)n1 ZINC000880766894 CC On-Demand Anodyne CASR 55 41 COCCN(Cc1ccc(F)cc1Cl)C(=O)Nc1ccn(CCF)n1 ZINC000880766896 FG On-Demand Anodyne P2RX7 37 43 O=C(NCc1cccc(OCC(F)F)c1)Nc1ccn(CCF)n1 ZINC000880766899 EF On-Demand Anodyne PDS 73 37 CN(CC1=CCSC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880766972 DF On-Demand Anodyne MPO 45 34 CC(C)(C)OC(=O)N1CCC(CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766980 FF On-Demand Anodyne CACNA1I 45 37 CC(C)(C)OC(=O)N1CCC(CNC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880766980 FF On-Demand Anodyne GPR119 46 41 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne HTR1A 57 54 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne DRD2 59 47 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne DRD1 15 43 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne DRD4 31 47 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne ADRA1D 22 41 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne HTR2A 33 47 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne HTR2C 19 46 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne ADRA1A 25 41 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne DRD3 77 44 O=C(NCCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880767039 GD On-Demand Anodyne HTR7 43 39 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne HTR1A 41 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne DRD2 35 43 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne HTR2A 30 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne DRD3 52 43 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne HTR7 41 36 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1ccn(CCF)n1 ZINC000880767148 GD On-Demand Anodyne CCR3 22 43 O=C(NC[C@H]1CCN1Cc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880767256 FD On-Demand Anodyne SIGMAR1 26 45 O=C(NC[C@H]1CCN1Cc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880767256 FD On-Demand Anodyne CACNA1G 21 40 O=C(NC[C@@H]1CCN1Cc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880767257 FD On-Demand Anodyne SIGMAR1 26 45 O=C(NC[C@@H]1CCN1Cc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880767257 FD On-Demand Anodyne CACNA1G 21 40 N#Cc1cccc(OC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880767274 FF On-Demand Mild CCR3 24 43 N#Cc1cccc(OC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c1 ZINC000880767274 FF On-Demand Mild EPHX2 17 52 COc1ccc(O)c(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880767291 DD On-Demand Clean MTNR1A 38 40 COc1ccc(O)c(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880767291 DD On-Demand Clean MTNR1B 27 40 Cn1nc2c(c1C(=O)NC[C@@H]1CCN1Cc1ccccc1)CSCC2 ZINC000880767299 FE On-Demand Anodyne DRD2 17 44 Cn1nc2c(c1C(=O)NC[C@H]1CCN1Cc1ccccc1)CSCC2 ZINC000880767301 FE On-Demand Anodyne DRD2 17 44 O=C(C[C@@H]1C[C@H]1C1CC1)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767314 CF On-Demand Anodyne SIGMAR1 27 41 O=C(C[C@@H]1C[C@H]1C1CC1)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767316 CF On-Demand Anodyne SIGMAR1 27 41 COc1ccc(N2CCCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880767332 FF On-Demand Clean PDGFRB 48 36 CN(CCN1CCN(C(=O)Nc2ccn(CCF)n2)CC1)Cc1ccccc1 ZINC000880767333 GE On-Demand Anodyne FAAH 18 40 CCOc1ccccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880767367 DF On-Demand Anodyne HCN1 50 35 CCOc1ccccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880767367 DF On-Demand Anodyne HCN4 41 32 O=C(NC[C@@H](O)c1cccc(Cl)c1)Nc1ccn(CCF)n1 ZINC000880767387 EE On-Demand Anodyne ADRB3 38 40 O=C(NC[C@H](O)c1cccc(Cl)c1)Nc1ccn(CCF)n1 ZINC000880767388 EE On-Demand Anodyne ADRB3 38 40 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1ccn(CCF)n1 ZINC000880767412 GD On-Demand Anodyne P2RX3 27 42 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCN2Cc2ccccc2)CC1 ZINC000880767413 FD On-Demand Anodyne SIGMAR1 27 46 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2CCN2Cc2ccccc2)CC1 ZINC000880767413 FD On-Demand Anodyne CACNA1G 30 43 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCN2Cc2ccccc2)CC1 ZINC000880767414 FD On-Demand Anodyne SIGMAR1 27 46 CS(=O)(=O)C1CCC(C(=O)NC[C@H]2CCN2Cc2ccccc2)CC1 ZINC000880767414 FD On-Demand Anodyne CACNA1G 30 43 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767420 FF On-Demand Anodyne DRD2 20 45 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767420 FF On-Demand Anodyne ACHE 16 42 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767420 FF On-Demand Anodyne SIGMAR1 20 44 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767420 FF On-Demand Anodyne PLD1 46 35 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767421 FF On-Demand Anodyne DRD2 20 45 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767421 FF On-Demand Anodyne ACHE 16 42 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767421 FF On-Demand Anodyne SIGMAR1 20 44 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767421 FF On-Demand Anodyne PLD1 46 35 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767422 FF On-Demand Anodyne DRD2 20 45 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767422 FF On-Demand Anodyne ACHE 16 42 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767422 FF On-Demand Anodyne SIGMAR1 20 44 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767422 FF On-Demand Anodyne PLD1 46 35 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767423 FF On-Demand Anodyne DRD2 20 45 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767423 FF On-Demand Anodyne ACHE 16 42 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767423 FF On-Demand Anodyne SIGMAR1 20 44 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCN3Cc3ccccc3)cc2)N1 ZINC000880767423 FF On-Demand Anodyne PLD1 46 35 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne HTR1A 17 49 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne HTR1D 60 47 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne HTR1B 45 49 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne NQO2 34 45 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne MPO 68 38 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne HTR1E 15 40 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne MTNR1A 89 66 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne MTNR1B 70 59 COc1ccc2[nH]cc(CCNC(=O)Nc3ccn(CCF)n3)c2c1 ZINC000880767435 EF On-Demand Anodyne ABCG2 26 43 O=C(Cc1ccccc1N1CCCC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767442 GF On-Demand Anodyne DRD2 17 41 O=C(Cc1ccccc1N1CCCC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767442 GF On-Demand Anodyne SIGMAR1 19 41 O=C(Cc1ccccc1N1CCCC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767442 GF On-Demand Anodyne MBTPS1 40 31 O=C(Cc1ccccc1N1CCCC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767443 GF On-Demand Anodyne DRD2 17 41 O=C(Cc1ccccc1N1CCCC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767443 GF On-Demand Anodyne SIGMAR1 19 41 O=C(Cc1ccccc1N1CCCC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767443 GF On-Demand Anodyne MBTPS1 40 31 O=C(NCc1ccnc(OC2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880767468 FE On-Demand Anodyne MAPK1 42 31 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cncc2[nH]ccc12 ZINC000880767470 DF On-Demand Anodyne DRD2 28 48 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cncc2[nH]ccc12 ZINC000880767471 DF On-Demand Anodyne DRD2 28 48 O=C(NCCn1cncn1)Nc1ccn(CCF)n1 ZINC000880767526 CC On-Demand Anodyne HIS3 43 31 O=C(NC[C@@H](O)COCC1CC1)Nc1ccn(CCF)n1 ZINC000880767596 DC On-Demand Anodyne ADRB1 40 31 O=C(NC[C@H](O)COCC1CC1)Nc1ccn(CCF)n1 ZINC000880767597 DC On-Demand Anodyne ADRB1 40 31 O=C(NC[C@H]1CCN1Cc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880767695 ED On-Demand Anodyne CACNA1G 22 40 O=C(NC[C@H]1CCN1Cc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880767696 ED On-Demand Anodyne CACNA1G 22 40 O=C(NC[C@@H]1CCN1Cc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880767697 ED On-Demand Anodyne CACNA1G 22 40 O=C(NC[C@@H]1CCN1Cc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880767698 ED On-Demand Anodyne CACNA1G 22 40 O=C(C[C@H]1CCNC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767708 DC On-Demand Anodyne SIGMAR1 22 40 O=C(C[C@H]1CCNC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767708 DC On-Demand Anodyne MBTPS1 41 32 O=C(C[C@@H]1CCNC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767709 DC On-Demand Anodyne SIGMAR1 22 40 O=C(C[C@@H]1CCNC1=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767709 DC On-Demand Anodyne MBTPS1 41 32 O=C(C[C@H]1CCNC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767710 DC On-Demand Anodyne SIGMAR1 22 40 O=C(C[C@H]1CCNC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767710 DC On-Demand Anodyne MBTPS1 41 32 O=C(C[C@@H]1CCNC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767711 DC On-Demand Anodyne SIGMAR1 22 40 O=C(C[C@@H]1CCNC1=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767711 DC On-Demand Anodyne MBTPS1 41 32 O=C(COC1CC1)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767713 CD On-Demand Anodyne DRD2 21 46 O=C(COC1CC1)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767713 CD On-Demand Anodyne SIGMAR1 38 45 O=C(COC1CC1)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767713 CD On-Demand Anodyne MBTPS1 51 36 O=C(COC1CC1)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767714 CD On-Demand Anodyne DRD2 21 46 O=C(COC1CC1)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767714 CD On-Demand Anodyne SIGMAR1 38 45 O=C(COC1CC1)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767714 CD On-Demand Anodyne MBTPS1 51 36 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne DRD2 15 42 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne DRD4 39 42 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne ACHE 46 42 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne LTA4H 18 41 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne SIGMAR1 47 48 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne CCR3 23 42 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne CCR5 32 48 CN(C(=O)Nc1ccn(CCF)n1)C1CCN(Cc2ccccc2)CC1 ZINC000880767731 FF On-Demand Anodyne CACNA1G 25 40 COc1cc(C)nc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880767767 FD On-Demand Anodyne PDGFRB 43 34 CCOc1cc(CNC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880767768 EF On-Demand Anodyne PDGFRB 16 42 CCOc1cc(CNC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880767768 EF On-Demand Anodyne ROCK2 15 45 CCOc1cc(CNC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880767768 EF On-Demand Anodyne QPCT 15 40 CCOc1cc(CNC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880767768 EF On-Demand Anodyne DRTS_TRYCR 48 35 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cc2c(cc1[N+](=O)[O-])OCCCO2 ZINC000880767774 GF On-Demand Bother DRD2 33 45 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cc2c(cc1[N+](=O)[O-])OCCCO2 ZINC000880767775 GF On-Demand Bother DRD2 33 45 Cn1nnc(C(=O)NC[C@H]2CCN2Cc2ccccc2)n1 ZINC000880767779 CC On-Demand Anodyne DRD2 27 48 Cn1nnc(C(=O)NC[C@H]2CCN2Cc2ccccc2)n1 ZINC000880767779 CC On-Demand Anodyne ACHE 25 41 Cn1nnc(C(=O)NC[C@H]2CCN2Cc2ccccc2)n1 ZINC000880767779 CC On-Demand Anodyne DRD3 15 46 Cn1nnc(C(=O)NC[C@H]2CCN2Cc2ccccc2)n1 ZINC000880767779 CC On-Demand Anodyne HTR4 36 41 Cn1nnc(C(=O)NC[C@H]2CCN2Cc2ccccc2)n1 ZINC000880767779 CC On-Demand Anodyne SIGMAR1 36 46 Cn1nnc(C(=O)NC[C@@H]2CCN2Cc2ccccc2)n1 ZINC000880767780 CC On-Demand Anodyne DRD2 27 48 Cn1nnc(C(=O)NC[C@@H]2CCN2Cc2ccccc2)n1 ZINC000880767780 CC On-Demand Anodyne ACHE 25 41 Cn1nnc(C(=O)NC[C@@H]2CCN2Cc2ccccc2)n1 ZINC000880767780 CC On-Demand Anodyne DRD3 15 46 Cn1nnc(C(=O)NC[C@@H]2CCN2Cc2ccccc2)n1 ZINC000880767780 CC On-Demand Anodyne HTR4 36 41 Cn1nnc(C(=O)NC[C@@H]2CCN2Cc2ccccc2)n1 ZINC000880767780 CC On-Demand Anodyne SIGMAR1 36 46 CCN(Cc1ccc(OC)cc1)C(=O)Nc1ccn(CCF)n1 ZINC000880767787 DF On-Demand Anodyne TSPO 27 41 NC(=O)c1cc(NC(=O)COC2CC2)nc2ccccc12 ZINC000880767799 CD On-Demand Anodyne TNKS 59 33 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880767819 GD On-Demand Anodyne PDGFRB 46 36 CN(C)S(=O)(=O)c1ccc(CNC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880767831 FD On-Demand Anodyne NAMPT 52 39 COc1cccc(OC)c1OC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880767861 GF On-Demand Anodyne EPHX2 16 41 COc1cccc(OC)c1OC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880767861 GF On-Demand Anodyne SCD1 17 44 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880767862 EC On-Demand Anodyne CCR8 90 38 CC(C)(C)OC(=O)N1CCCC[C@@H]1CNC(=O)Nc1ccn(CCF)n1 ZINC000880767865 FF On-Demand Anodyne HCRTR1 18 43 CC(C)(C)OC(=O)N1CCCC[C@H]1CNC(=O)Nc1ccn(CCF)n1 ZINC000880767866 FF On-Demand Anodyne HCRTR1 18 43 O=C(NCCNc1nc2ccccc2s1)Nc1ccn(CCF)n1 ZINC000880767874 EF On-Demand Anodyne CSNK1D 22 40 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne HTR1A 95 55 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne DRD2 78 51 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne DRD1 15 40 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne DRD4 46 46 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne ADRA1D 34 43 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne HTR2A 65 51 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne HTR2C 33 48 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne SLC6A4 15 40 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne ADRA1A 40 45 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne ADRA1B 22 45 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne DRD3 101 51 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne DRD5 17 40 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne HTR7 103 43 O=C(NCCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880767884 GF On-Demand Anodyne CCR3 23 40 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767890 DE On-Demand Anodyne DRD2 25 46 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767890 DE On-Demand Anodyne DRD4 15 43 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767890 DE On-Demand Anodyne SIGMAR1 18 46 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767891 DE On-Demand Anodyne DRD2 25 46 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767891 DE On-Demand Anodyne DRD4 15 43 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cccn2nccc12 ZINC000880767891 DE On-Demand Anodyne SIGMAR1 18 46 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880767894 FD On-Demand Anodyne NPY5R 26 42 O=C(c1ncsc1C1CC1)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880767904 DF On-Demand Anodyne ETHR 43 34 O=C(c1ncsc1C1CC1)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880767905 DF On-Demand Anodyne ETHR 43 34 O=C(NCCc1ccc(F)cc1Cl)Nc1ccn(CCF)n1 ZINC000880767916 EG On-Demand Anodyne P2RX7 50 46 Cc1nc(C(C)C)ncc1C(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767925 EF On-Demand Anodyne DRD2 23 45 Cc1nc(C(C)C)ncc1C(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880767925 EF On-Demand Anodyne HTR4 29 40 Cc1nc(C(C)C)ncc1C(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767926 EF On-Demand Anodyne DRD2 23 45 Cc1nc(C(C)C)ncc1C(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880767926 EF On-Demand Anodyne HTR4 29 40 COc1ccc(C)cc1NC(=O)[C@@H]1CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880767930 GF On-Demand Anodyne HCRTR2 17 40 COc1ccc(C)cc1NC(=O)[C@H]1CCCN1C(=O)Nc1ccn(CCF)n1 ZINC000880767931 GF On-Demand Anodyne HCRTR2 17 40 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768039 DD On-Demand Anodyne NQO2 24 41 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768039 DD On-Demand Anodyne MTNR1A 35 43 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768039 DD On-Demand Anodyne MTNR1B 33 40 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768039 DD On-Demand Anodyne MMP1 18 40 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768040 DD On-Demand Anodyne NQO2 24 41 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768040 DD On-Demand Anodyne MTNR1A 35 43 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768040 DD On-Demand Anodyne MTNR1B 33 40 COC(=O)[C@@H]1C[C@@H](NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880768040 DD On-Demand Anodyne MMP1 18 40 COc1ccc(OC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880768053 FF On-Demand Anodyne PRSS2 47 33 COc1ccc(OC2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880768053 FF On-Demand Anodyne EPHX2 21 47 O=C(NCCOc1cccc(Cl)c1)Nc1ccn(CCF)n1 ZINC000880768060 EF On-Demand Anodyne HRH2 36 46 CCOc1ccnc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)n1 ZINC000880768089 FD On-Demand Anodyne FAAH 22 41 O=C(NC[C@@H]1CCN1Cc1ccccc1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880768092 DE On-Demand Anodyne SIGMAR1 23 40 O=C(NC[C@H]1CCN1Cc1ccccc1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880768093 DE On-Demand Anodyne SIGMAR1 23 40 O=C(NC[C@H]1CCCN1Cc1ccccc1)Nc1ccn(CCF)n1 ZINC000880768099 EF On-Demand Anodyne DRD2 35 47 O=C(NC[C@H]1CCCN1Cc1ccccc1)Nc1ccn(CCF)n1 ZINC000880768099 EF On-Demand Anodyne SIGMAR1 18 45 COc1ccccc1[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880768112 EF On-Demand Anodyne RBP4 50 40 COc1ccccc1[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880768113 EF On-Demand Anodyne RBP4 50 40 COc1cccc(OCCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768121 EE On-Demand Anodyne DRD4 40 31 COc1cccc(OCCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768121 EE On-Demand Anodyne HRH2 50 49 COc1cccc(OCCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768121 EE On-Demand Anodyne MTNR1A 63 48 COc1cccc(OCCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768121 EE On-Demand Anodyne MTNR1B 61 48 COc1cc2c(cc1OC)CCN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880768204 FF On-Demand Anodyne PDGFRB 44 38 COc1cc2c(cc1OC)CCN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880768204 FF On-Demand Anodyne ABCB1B 49 37 O=C(NCCOc1cccc(Br)c1)Nc1ccn(CCF)n1 ZINC000880768273 FF On-Demand Anodyne HRH2 41 42 O=C(NCCOc1cccc(Br)c1)Nc1ccn(CCF)n1 ZINC000880768273 FF On-Demand Anodyne HMOX2 21 43 O=C(NCCCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880768309 EF On-Demand Anodyne HRH2 27 40 O=C(NCCCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880768309 EF On-Demand Anodyne CHRNA7 22 52 O=C(NCCCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880768309 EF On-Demand Anodyne HNMT 64 37 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880768343 DC On-Demand Anodyne CCR8 69 35 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880768344 DC On-Demand Anodyne CCR8 69 35 O=C(NCCNC(=O)c1ccccc1Cl)Nc1ccn(CCF)n1 ZINC000880768406 FE On-Demand Anodyne POLR1A 40 32 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne HTR1A 61 44 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne DRD2 46 43 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne DRD4 25 43 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne ADRA1D 37 42 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne HTR1D 17 43 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne HTR1B 24 43 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne ADRA1A 35 42 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne DRD3 55 43 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne PDGFRB 53 45 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne HTR7 52 44 CCOc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768418 FF On-Demand Anodyne HCN1 47 32 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1ccn(CCF)n1 ZINC000880768430 EE On-Demand Anodyne MAPK13 70 33 COC(=O)[C@@H]1C[C@@H](NC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880768463 DF On-Demand Anodyne NQO2 20 41 COC(=O)[C@@H]1C[C@@H](NC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880768464 DF On-Demand Anodyne NQO2 20 41 COC(=O)[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880768469 EF On-Demand Anodyne PDE4D 20 42 COC(=O)[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880768469 EF On-Demand Anodyne EZH2 43 41 COC(=O)[C@@H]1C[C@@H](NC(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880768477 EE On-Demand Anodyne PDK1 49 40 N#Cc1ccccc1CSCCNC(=O)Nc1ccn(CCF)n1 ZINC000880768482 EF On-Demand Mild ADRB1 44 35 Cn1ncc(Br)c1CC(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880768492 GE On-Demand Anodyne DRD2 15 44 Cn1ncc(Br)c1CC(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880768492 GE On-Demand Anodyne SIGMAR1 23 47 Cn1ncc(Br)c1CC(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880768493 GE On-Demand Anodyne DRD2 15 44 Cn1ncc(Br)c1CC(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880768493 GE On-Demand Anodyne SIGMAR1 23 47 O=C(CN1CCCCS1(=O)=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880768496 FC On-Demand Anodyne SIGMAR1 21 41 O=C(CN1CCCCS1(=O)=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880768497 FC On-Demand Anodyne SIGMAR1 21 41 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cnc2cc[nH]c2c1 ZINC000880768521 DF On-Demand Anodyne SIGMAR1 15 42 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1cnc2cc[nH]c2c1 ZINC000880768521 DF On-Demand Anodyne CXCR3 19 40 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cnc2cc[nH]c2c1 ZINC000880768522 DF On-Demand Anodyne SIGMAR1 15 42 O=C(NC[C@H]1CCN1Cc1ccccc1)c1cnc2cc[nH]c2c1 ZINC000880768522 DF On-Demand Anodyne CXCR3 19 40 C=CC(C)(C)CC(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880768529 CF On-Demand Mild DRD2 15 41 C=CC(C)(C)CC(=O)NC[C@@H]1CCN1Cc1ccccc1 ZINC000880768529 CF On-Demand Mild SIGMAR1 27 42 C=CC(C)(C)CC(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880768530 CF On-Demand Mild DRD2 15 41 C=CC(C)(C)CC(=O)NC[C@H]1CCN1Cc1ccccc1 ZINC000880768530 CF On-Demand Mild SIGMAR1 27 42 O=C(NCC1(N2CCSCC2)CCCCC1)Nc1ccn(CCF)n1 ZINC000880768551 FF On-Demand Anodyne HCN1 62 40 O=C(NCC1(N2CCSCC2)CCCCC1)Nc1ccn(CCF)n1 ZINC000880768551 FF On-Demand Anodyne HCN4 57 37 Cc1nc(CN2CCC(CNC(=O)Nc3ccn(CCF)n3)CC2)oc1C ZINC000880768561 GE On-Demand Anodyne HTR4 47 39 Cc1nc(CN2CCC(CNC(=O)Nc3ccn(CCF)n3)CC2)oc1C ZINC000880768561 GE On-Demand Anodyne CACNA1I 51 37 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1ncsc1C1CC1 ZINC000880768568 EG On-Demand Anodyne SIGMAR1 17 43 O=C(NC[C@H]1CCN1Cc1ccccc1)c1ncsc1C1CC1 ZINC000880768569 EG On-Demand Anodyne SIGMAR1 17 43 CN1CCC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880768585 CD On-Demand Anodyne CCR3 19 41 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880768589 CD On-Demand Anodyne TBXAS1 43 37 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne HTR1A 16 49 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne HTR1D 45 49 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne HTR1B 40 49 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne HTR1F 97 44 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne MTNR1A 15 50 COc1ccc2[nH]cc(C3CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880768605 GH On-Demand Anodyne CCR2 27 47 O=C(Cc1ccc(Cl)cc1)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768629 GE On-Demand Anodyne KCNJ1 40 33 O=C(NCC(=O)N1CCCc2ccccc21)Nc1ccn(CCF)n1 ZINC000880768640 ED On-Demand Anodyne AVPR2 35 40 O=C(NCCCS(=O)(=O)c1ccccc1)Nc1ccn(CCF)n1 ZINC000880768648 FD On-Demand Anodyne NAMPT 15 40 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880768654 FF On-Demand Anodyne EPHX2 34 48 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768674 GG On-Demand Anodyne ADRB3 17 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768674 GG On-Demand Anodyne NQO2 26 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768674 GG On-Demand Anodyne MTNR1A 29 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768674 GG On-Demand Anodyne MTNR1B 26 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768675 GG On-Demand Anodyne ADRB3 17 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768675 GG On-Demand Anodyne NQO2 26 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768675 GG On-Demand Anodyne MTNR1A 29 44 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)c1cc(F)c(F)c(F)c1)C2 ZINC000880768675 GG On-Demand Anodyne MTNR1B 26 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)C1)C2 ZINC000880768677 CD On-Demand Anodyne NQO2 24 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)C1)C2 ZINC000880768677 CD On-Demand Anodyne MTNR1A 35 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1C[C@H](O)C1)C2 ZINC000880768677 CD On-Demand Anodyne MTNR1B 33 40 COC(=O)[C@@H]1C[C@@H](NC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880768695 ED On-Demand Anodyne KCNQ2 65 37 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)Nc1ccn(CCF)n1 ZINC000880768747 GD On-Demand Anodyne NAMPT 99 56 COC(=O)[C@@H]1C[C@@H](NC(=O)c2ccc(-c3ccccc3OC)nc2O)C1 ZINC000880768758 FE On-Demand Anodyne HTR3A 22 45 O=C(NCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880768809 CD On-Demand Anodyne CHRNA7 18 44 O=C(NCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880768809 CD On-Demand Anodyne HNMT 46 32 Cc1cccc(C(C)(C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768827 DG On-Demand Anodyne IMDH_CRYPV 62 36 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880768831 CD On-Demand Anodyne SLC6A1 62 32 CN(C(=O)Nc1ccn(CCF)n1)[C@H]1CCCN(c2ccccc2)C1 ZINC000880768836 EF On-Demand Anodyne SLC6A1 78 31 CN(C(=O)Nc1ccn(CCF)n1)[C@@H]1CCCN(c2ccccc2)C1 ZINC000880768839 EF On-Demand Anodyne SLC6A1 78 31 CCOc1ccccc1Oc1ccc(CNC(=O)Nc2ccn(CCF)n2)cn1 ZINC000880768848 GH On-Demand Anodyne HCN1 47 32 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1ccn(CCF)n1 ZINC000880768851 EE On-Demand Clean STAT6 51 33 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne DRD2 41 51 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne DRD4 27 41 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne ACHE 17 42 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne DRD3 17 50 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne HTR4 18 40 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne SIGMAR1 22 50 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2Cc2ccccc2)c1 ZINC000880768852 EG On-Demand Anodyne CACNA1I 51 39 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne DRD2 41 51 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne DRD4 27 41 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne ACHE 17 42 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne DRD3 17 50 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne HTR4 18 40 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne SIGMAR1 22 50 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2Cc2ccccc2)c1 ZINC000880768854 EG On-Demand Anodyne CACNA1I 51 39 C#CCCN(CCOC)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880768870 DD On-Demand Mild MPO 58 34 O=C(N[C@H]1C[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880768878 CE On-Demand Anodyne HTR4 25 40 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccccc1 ZINC000880768879 FE On-Demand Anodyne DRD4 21 43 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccccc1 ZINC000880768879 FE On-Demand Anodyne MAPK13 47 33 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccccc1 ZINC000880768879 FE On-Demand Anodyne MCHR1 15 43 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccccc1 ZINC000880768879 FE On-Demand Anodyne CCR8 49 35 O=C(NCCCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880768891 CD On-Demand Anodyne TBXAS1 54 49 O=C(NCCCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880768891 CD On-Demand Anodyne QPCT 43 53 O=C(CC[C@H]1CCc2ccccc21)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880768921 EH On-Demand Anodyne ETHR 50 37 O=C(CC[C@@H]1CCc2ccccc21)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880768922 EH On-Demand Anodyne ETHR 50 37 O=C(CC[C@H]1CCc2ccccc21)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880768924 EH On-Demand Anodyne ETHR 50 37 O=C(CC[C@@H]1CCc2ccccc21)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880768926 EH On-Demand Anodyne ETHR 50 37 CCOc1cc(CCCNC(=O)Nc2ccn(CCF)n2)ccc1OC ZINC000880768982 FG On-Demand Anodyne QPCT 23 44 O=C(NC[C@H]1CCN1Cc1ccccc1)c1ccc(CN2CCOCC2)o1 ZINC000880768983 FE On-Demand Anodyne DRD2 20 46 O=C(NC[C@H]1CCN1Cc1ccccc1)c1ccc(CN2CCOCC2)o1 ZINC000880768983 FE On-Demand Anodyne SIGMAR1 44 44 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1ccc(CN2CCOCC2)o1 ZINC000880768984 FE On-Demand Anodyne DRD2 20 46 O=C(NC[C@@H]1CCN1Cc1ccccc1)c1ccc(CN2CCOCC2)o1 ZINC000880768984 FE On-Demand Anodyne SIGMAR1 44 44 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880768999 FG On-Demand Anodyne CARM1 45 33 O=C(NCCOc1cccc(F)c1)Nc1ccn(CCF)n1 ZINC000880769038 DE On-Demand Anodyne HRH2 37 42 CC[C@@H](CNC(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880769060 DG On-Demand Anodyne SOAT1 26 40 COc1cccc(C(=O)NCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769083 ED On-Demand Anodyne DRD4 58 44 COc1cccc(C(=O)NCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769083 ED On-Demand Anodyne DRD3 20 46 COc1cccc(C(=O)NCCNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769083 ED On-Demand Anodyne NQO2 17 42 O=C(N[C@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880769088 EE On-Demand Anodyne EZH2 27 40 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769123 GE On-Demand Anodyne HCN1 60 39 CCOc1ccccc1C(=O)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769123 GE On-Demand Anodyne HCN4 46 36 CN(C)CCOc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769129 EE On-Demand Anodyne HRH2 40 38 CN(C)CCOc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769129 EE On-Demand Anodyne ROCK2 37 49 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne CELA1 19 40 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne GRIN2B 18 40 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne PREP 28 44 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne LGMN 60 39 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne SLC12A5 68 36 O=C(N[C@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880769144 ED On-Demand Anodyne Q9NAW4_PLAFA 45 52 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2ccn(CCF)n2)c1 ZINC000880769152 EG On-Demand Anodyne ROCK2 42 36 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2ccn(CCF)n2)c1 ZINC000880769152 EG On-Demand Anodyne ACKR3 46 32 CCN1CC[C@H](CNC(=O)Nc2ccn(CCF)n2)C1 ZINC000880769164 CD On-Demand Anodyne CACNA1I 50 34 Cc1ccccc1CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769171 FF On-Demand Anodyne DRD4 20 55 Cc1ccccc1CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769171 FF On-Demand Anodyne SIGMAR1 18 46 Cc1ccccc1CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769171 FF On-Demand Anodyne SSTR5 46 38 Cc1ccccc1CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769171 FF On-Demand Anodyne MCHR1 31 41 Cc1ccccc1CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769171 FF On-Demand Anodyne CCR8 52 32 N#Cc1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)nc1 ZINC000880769212 ED On-Demand Mild PDGFRB 18 41 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne HRH2 49 42 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne TNF 34 41 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne MAPK14 17 41 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne ROCK2 24 44 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne EPHX2 30 46 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne FLT3 22 44 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne MAPK12 19 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne AURKA 15 48 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne STK10 21 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne EPHA8 15 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne EPHA5 17 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne EPHA4 16 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne TIE1 19 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne DDR2 18 40 O=C(NCc1cccc(OCCN2CCOCC2)c1)Nc1ccn(CCF)n1 ZINC000880769215 GD On-Demand Anodyne CDK8 21 40 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@H]1CCc2nncn2CC1 ZINC000880769216 GF On-Demand Anodyne EPHX2 17 43 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@H]1CCc2nncn2CC1 ZINC000880769216 GF On-Demand Anodyne SFRP1 104 35 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@H]1CCc2nncn2CC1 ZINC000880769216 GF On-Demand Anodyne WNT3 59 34 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@H]1CCc2nncn2CC1 ZINC000880769216 GF On-Demand Anodyne NAMPT 31 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccn(CCF)n2)C1 ZINC000880769236 EC On-Demand Anodyne EPHX2 27 40 COC(=O)[C@@H]1C[C@@H](NC(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880769240 EE On-Demand Anodyne FKBP1A 41 44 COC(=O)[C@@H]1C[C@@H](NC(=O)CCCCc2ccc(OC)c(OC)c2)C1 ZINC000880769240 EE On-Demand Anodyne MTNR1B 29 44 COC(=O)[C@@H]1C[C@@H](NC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880769292 CD On-Demand Anodyne PTR1 44 32 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)C1CCCCC1 ZINC000880769301 FF On-Demand Anodyne EPHX2 34 44 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1ccn(CCF)n1 ZINC000880769303 EE On-Demand Anodyne TSPO 37 41 COC(=O)[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880769315 DD On-Demand Anodyne GABRA1 19 42 COC(=O)[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880769315 DD On-Demand Anodyne MPO 43 33 COC(=O)[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880769315 DD On-Demand Anodyne GABRA2 17 42 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880769321 GF On-Demand Anodyne EPHX2 17 43 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880769321 GF On-Demand Anodyne SFRP1 104 35 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880769321 GF On-Demand Anodyne WNT3 59 34 O=C(Nc1cccc(S(=O)(=O)c2ccccc2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880769321 GF On-Demand Anodyne NAMPT 31 40 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2C[C@H](O)C2)N1Cc1ccccc1 ZINC000880769369 DC On-Demand Anodyne SIGMAR1 20 42 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1ccn(CCF)n1 ZINC000880769392 ED On-Demand Anodyne ADRB1 51 39 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1ccn(CCF)n1 ZINC000880769393 ED On-Demand Anodyne ADRB1 51 39 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)Nc1ccn(CCF)n1 ZINC000880769414 GF On-Demand Anodyne ADRB1 52 38 O=C(NC[C@@H](O)COc1cccc(Cl)c1Cl)Nc1ccn(CCF)n1 ZINC000880769415 GF On-Demand Anodyne ADRB1 52 38 O=C(NCc1ccc(N2CCCCCC2)nc1)Nc1ccn(CCF)n1 ZINC000880769429 FF On-Demand Anodyne NAMPT 23 40 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne DRD2 19 47 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne DRD4 42 47 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne ACHE 56 47 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne HRH1 19 40 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne HTR4 61 49 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne SIGMAR1 52 43 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne BCHE 18 43 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne CCR3 64 45 O=C(NCC1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769442 FF On-Demand Anodyne CACNA1I 61 41 COc1cccc([C@@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769443 DF On-Demand Anodyne ROCK1 17 48 COc1cccc([C@@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769443 DF On-Demand Anodyne ROCK2 25 41 COc1cccc([C@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769444 DF On-Demand Anodyne ROCK1 17 48 COc1cccc([C@H](C)NC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769444 DF On-Demand Anodyne ROCK2 25 41 O=C(Cc1ccccc1N1CCCC1=O)NC[C@H](O)c1cc(F)c(F)c(F)c1 ZINC000880769452 GF On-Demand Anodyne KCNQ2 51 36 O=C(Cc1ccccc1N1CCCC1=O)NC[C@@H](O)c1cc(F)c(F)c(F)c1 ZINC000880769453 GF On-Demand Anodyne KCNQ2 51 36 COc1ccccc1-c1ccc(C(=O)N[C@H]2C[C@H](O)C2)c(O)n1 ZINC000880769455 DD On-Demand Anodyne HTR3A 20 46 CC(=O)N[C@@H](CC(=O)N1CCN(Cc2cccc3cccnc23)CC1)c1ccc(Br)cc1 ZINC000880769457 JH On-Demand Anodyne PTAFR 20 47 O=C(N[C@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880769482 CD On-Demand Anodyne GABRA1 19 45 O=C(N[C@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880769482 CD On-Demand Anodyne MPO 45 36 O=C(N[C@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880769482 CD On-Demand Anodyne GABRA2 17 45 O=C(N[C@H]1C[C@H](O)C1)c1cccn2nccc12 ZINC000880769492 BC On-Demand Anodyne JAK3 17 40 O=C(N[C@H]1C[C@H](O)C1)c1cccn2nccc12 ZINC000880769492 BC On-Demand Anodyne TYK2 20 40 O=C(N[C@H]1C[C@H](O)C1)c1cccn2nccc12 ZINC000880769492 BC On-Demand Anodyne EPHB3 32 40 COCCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769505 DD On-Demand Anodyne DRD4 16 42 COCCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769505 DD On-Demand Anodyne SSTR5 43 37 COCCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769505 DD On-Demand Anodyne SLC6A5 28 40 O=C(NC[C@@H](O)COc1ccc(C(F)(F)F)cc1)Nc1ccn(CCF)n1 ZINC000880769515 GE On-Demand Anodyne ADRB1 42 35 O=C(NC[C@H](O)COc1ccc(C(F)(F)F)cc1)Nc1ccn(CCF)n1 ZINC000880769516 GE On-Demand Anodyne ADRB1 42 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)C1 ZINC000880769538 DC On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)C1 ZINC000880769538 DC On-Demand Anodyne CTSK 15 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)C1 ZINC000880769539 DC On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1C[C@H](O)C1 ZINC000880769539 DC On-Demand Anodyne CTSK 15 49 O=C(N[C@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880769546 CE On-Demand Anodyne PDE4D 18 44 O=C(N[C@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880769546 CE On-Demand Anodyne EZH2 43 40 C[C@@H](Cc1ccc(O)cc1)NC(=O)Nc1ccn(CCF)n1 ZINC000880769569 DE On-Demand Anodyne GRIA1 40 32 O=C(N[C@H]1C[C@H](O)C1)c1ncccc1-c1ccccn1 ZINC000880769592 CD On-Demand Anodyne MERTK 24 43 O=C(Nc1ccc(Cl)cn1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769602 GF On-Demand Anodyne F10 25 44 O=C(NC[C@@H](O)COc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880769603 GE On-Demand Anodyne ADRB1 46 37 O=C(NC[C@@H](O)COc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880769603 GE On-Demand Anodyne PDS 46 40 O=C(NC[C@H](O)COc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880769604 GE On-Demand Anodyne ADRB1 46 37 O=C(NC[C@H](O)COc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880769604 GE On-Demand Anodyne PDS 46 40 N#Cc1ccc(CN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880769625 FE On-Demand Mild MLNR 21 41 N#Cc1ccc(CN2CCN(C(=O)Nc3ccn(CCF)n3)CC2)cc1 ZINC000880769625 FE On-Demand Mild FAAH 17 42 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769633 FE On-Demand Anodyne EPHX2 37 46 O=C(N[C@H]1C[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880769640 CC On-Demand Anodyne PLD2 40 37 O=C(Nc1ccc(Cl)cn1)[C@@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880769649 GF On-Demand Anodyne F10 19 41 O=C(Nc1ccc(Cl)cn1)[C@H]1CCCN(C(=O)Nc2ccn(CCF)n2)C1 ZINC000880769650 GF On-Demand Anodyne F10 19 41 COc1ccc(CN(C)C(=O)Nc2ccn(CCF)n2)c(OC)c1 ZINC000880769657 EF On-Demand Anodyne PDGFRB 36 41 CC(C)(C)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769661 DE On-Demand Anodyne EPHX2 34 40 COc1ccc(OCCCNC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880769670 EE On-Demand Anodyne HRH2 25 43 CCC(=O)Nc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880769671 EF On-Demand Anodyne ROCK2 21 41 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N[C@H]3C[C@H](O)C3)ccn2)CC1 ZINC000880769676 GD On-Demand Anodyne GPR119 48 47 Cc1ccccc1[C@H](C)NC(=O)Nc1ccn(CCF)n1 ZINC000880769699 CG On-Demand Anodyne CTSA 54 37 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne HTR1A 20 47 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne DRD2 23 41 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne DRD4 32 41 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne ACHE 29 40 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne DRD3 25 41 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne SIGMAR1 37 47 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne CCR3 25 40 O=C(NCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880769703 FD On-Demand Anodyne UTS2R 17 41 N#Cc1cccnc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769725 ED On-Demand Mild PDGFRB 40 39 Cc1ccccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880769730 CE On-Demand Anodyne P2RX7 22 40 Cc1ccccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880769730 CE On-Demand Anodyne MT-CYB 40 32 O=C(NCCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880769768 CD On-Demand Anodyne TBXAS1 55 49 O=C(NCCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880769768 CD On-Demand Anodyne QPCT 47 56 O=C(NC[C@H]1CN(Cc2ccccc2)CCO1)Nc1ccn(CCF)n1 ZINC000880769774 FD On-Demand Anodyne DRD4 21 44 O=C(NC[C@@H]1CN(Cc2ccccc2)CCO1)Nc1ccn(CCF)n1 ZINC000880769775 FD On-Demand Anodyne DRD4 21 44 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne HTR1A 56 52 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne DRD2 56 47 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne DRD4 31 47 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne ADRA1D 27 41 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne HTR2A 40 48 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne HTR2C 25 48 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne ADRA1A 29 41 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne DRD3 68 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccn(CCF)n1 ZINC000880769779 GC On-Demand Anodyne HTR7 49 39 CN(CCOc1ccccc1)C(=O)Nc1ccn(CCF)n1 ZINC000880769811 DE On-Demand Anodyne LTA4H 20 40 CC(=O)c1ccc(N2CCN(C(=O)Nc3ccn(CCF)n3)CC2)c(F)c1 ZINC000880769818 GF On-Demand Anodyne NPY2R 82 37 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccn(CCF)n1 ZINC000880769840 DE On-Demand Anodyne NOS2 80 35 O=C(NCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880769841 CC On-Demand Anodyne TBXAS1 58 41 O=C(NCCn1ccnc1)Nc1ccn(CCF)n1 ZINC000880769841 CC On-Demand Anodyne QPCT 33 47 O=C(NCCc1ccc(Cl)cc1Cl)Nc1ccn(CCF)n1 ZINC000880769849 EH On-Demand Anodyne CNR1 22 45 O=C(NCCc1ccc(Cl)cc1Cl)Nc1ccn(CCF)n1 ZINC000880769849 EH On-Demand Anodyne P2RX7 41 40 O=C(NCCNc1ccccn1)Nc1ccn(CCF)n1 ZINC000880769880 CD On-Demand Anodyne ADRB1 40 32 O=C(COC1CC1)NCC1CCN(CC2CC2)CC1 ZINC000880769894 CD On-Demand Anodyne CACNA1I 60 38 COc1cccc([C@H](CNC(=O)Nc2ccn(CCF)n2)N2CCCC2)c1 ZINC000880769911 GF On-Demand Anodyne DRD4 41 31 O=C(NCC1CCN(CC2CC2)CC1)C1(c2cccnc2)CC2(CCC2)C1 ZINC000880769923 FH On-Demand Anodyne CACNA1I 25 40 CCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769926 CD On-Demand Anodyne SSTR5 43 38 CCN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880769926 CD On-Demand Anodyne EPHX2 36 40 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769934 DD On-Demand Anodyne ADRB2 29 40 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769934 DD On-Demand Anodyne ADRB1 55 39 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769934 DD On-Demand Anodyne ADRB3 27 41 O=C(NC[C@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769940 DD On-Demand Anodyne ADRB2 29 40 O=C(NC[C@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769940 DD On-Demand Anodyne ADRB1 55 39 O=C(NC[C@H](O)COc1ccccc1)Nc1ccn(CCF)n1 ZINC000880769940 DD On-Demand Anodyne ADRB3 27 41 O=C(NC1CC1)c1ccc(CN(C(=O)Nc2ccn(CCF)n2)C2CC2)cc1 ZINC000880769962 GF On-Demand Anodyne MAPK13 61 31 O=C(NC1CC1)c1ccc(CN(C(=O)Nc2ccn(CCF)n2)C2CC2)cc1 ZINC000880769962 GF On-Demand Anodyne SLC6A5 30 40 O=C(NCc1cccc(N2CCCC2=O)c1)Nc1ccn(CCF)n1 ZINC000880769966 EE On-Demand Anodyne CARM1 40 33 O=C(NCC1CCN(CC2CC2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880769995 FD On-Demand Anodyne HTR4 59 44 O=C(NCC1CCN(CC2CC2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880769995 FD On-Demand Anodyne TACR2 25 40 O=C(NCC1CCN(CC2CC2)CC1)c1ccc(CN2CCOCC2)o1 ZINC000880769995 FD On-Demand Anodyne CACNA1I 73 45 O=C(NC[C@@H](c1ccccc1)N1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770022 FE On-Demand Anodyne CASR 44 36 O=C(NC[C@H](c1ccccc1)N1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770024 FE On-Demand Anodyne CASR 44 36 C[C@@H]1CCCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770029 CF On-Demand Anodyne CCR3 16 42 C[C@@H]1CCCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770031 CF On-Demand Anodyne CCR3 16 42 COc1ccc(CN(C)C(=O)Nc2ccn(CCF)n2)cc1OC ZINC000880770051 EF On-Demand Anodyne MT-ND1 17 42 O=C(NCCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770080 CC On-Demand Anodyne CHRNA7 15 47 O=C(NCCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770080 CC On-Demand Anodyne EPHX2 22 42 O=C(NCC1(c2ccccc2)CCC1)Nc1ccn(CCF)n1 ZINC000880770083 DG On-Demand Anodyne KCNA3 46 38 O=C(NCC1(c2ccccc2)CCC1)Nc1ccn(CCF)n1 ZINC000880770083 DG On-Demand Anodyne SOAT1 15 48 NC(=O)c1cccc2c1CCN(C(=O)c1ccc([C@H]3CCC(=O)N3)cc1)C2 ZINC000880770094 FD On-Demand Anodyne PARP2 33 42 NC(=O)c1cccc2c1CCN(C(=O)c1ccc([C@H]3CCC(=O)N3)cc1)C2 ZINC000880770094 FD On-Demand Anodyne PARP1 15 42 NC(=O)c1cccc2c1CCN(C(=O)c1ccc([C@@H]3CCC(=O)N3)cc1)C2 ZINC000880770095 FD On-Demand Anodyne PARP2 33 42 NC(=O)c1cccc2c1CCN(C(=O)c1ccc([C@@H]3CCC(=O)N3)cc1)C2 ZINC000880770095 FD On-Demand Anodyne PARP1 15 42 CC1(C)CC[C@@H](CC(=O)NCC2CCN(CC3CC3)CC2)OC1 ZINC000880770096 DF On-Demand Anodyne CACNA1I 54 33 COc1ccc(CC(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1F ZINC000880770109 GG On-Demand Anodyne MLNR 25 40 COc1ccc(CC(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1F ZINC000880770109 GG On-Demand Anodyne KCNJ1 42 37 CCN1CC[C@@H]1CNC(=O)Nc1ccccc1C(F)(F)CC ZINC000880770114 DG On-Demand Anodyne RBP4 75 36 O=C(NCc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880770128 EG On-Demand Anodyne SCD1 22 48 O=C(NCc1cccc(C(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880770128 EG On-Demand Anodyne CARM1 48 34 O=C(NCC1(c2ccccc2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880770131 EF On-Demand Anodyne KCNA3 43 39 O=C(NCC1(c2ccccc2)CCOCC1)Nc1ccn(CCF)n1 ZINC000880770131 EF On-Demand Anodyne SOAT1 16 44 CC[C@H]1CCC[C@]1(C)C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770135 DG On-Demand Anodyne CACNA1I 47 36 CC[C@@H]1CCC[C@@]1(C)C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770140 DG On-Demand Anodyne CACNA1I 47 36 CCCCCNC(=O)Nc1ccn(CCF)n1 ZINC000880770141 BE On-Demand Anodyne ASAH1 84 39 CC[C@@H]1CCC[C@]1(C)C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770143 DG On-Demand Anodyne CACNA1I 47 36 CC[C@H]1CCC[C@@]1(C)C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770145 DG On-Demand Anodyne CACNA1I 47 36 O=C(CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1)Nc1ccccc1 ZINC000880770148 GE On-Demand Anodyne DRD4 25 52 O=C(CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1)Nc1ccccc1 ZINC000880770148 GE On-Demand Anodyne SIGMAR1 15 43 O=C(CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1)Nc1ccccc1 ZINC000880770148 GE On-Demand Anodyne CCR3 19 43 O=C(CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1)Nc1ccccc1 ZINC000880770148 GE On-Demand Anodyne EPHX2 32 41 Cc1coc(C(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880770151 CE On-Demand Anodyne HTR4 65 45 Cc1coc(C(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880770151 CE On-Demand Anodyne CACNA1I 89 48 O=C(NCCN1CCc2ccccc2C1)Nc1ccn(CCF)n1 ZINC000880770157 EE On-Demand Anodyne NOD2 42 35 Cc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880770159 CE On-Demand Anodyne ROCK2 20 48 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne DRD2 22 55 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne DRD4 29 55 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne ACHE 16 43 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne HRH1 25 40 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne DRD3 19 42 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne HTR4 79 46 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne GRIN2B 34 47 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne SIGMAR1 33 47 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne CCR3 84 39 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne MCHR1 15 40 O=C(NCC1CCN(CC2CC2)CC1)c1cc2ccccc2cc1F ZINC000880770164 EH On-Demand Anodyne CACNA1I 79 41 COc1ccc([C@@H]2CCCCCN2C(=O)Nc2ccn(CCF)n2)cc1 ZINC000880770175 FI On-Demand Anodyne CPT1A 31 40 CC(C)CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770176 DE On-Demand Anodyne EPHX2 32 41 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770183 FE On-Demand Anodyne HTR4 55 40 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770183 FE On-Demand Anodyne GRIN2B 17 44 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770183 FE On-Demand Anodyne PLD1 54 35 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770183 FE On-Demand Anodyne CACNA1I 73 42 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770185 FE On-Demand Anodyne HTR4 55 40 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770185 FE On-Demand Anodyne GRIN2B 17 44 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770185 FE On-Demand Anodyne PLD1 54 35 O=C1CC[C@H](c2ccc(C(=O)NCC3CCN(CC4CC4)CC3)cc2)N1 ZINC000880770185 FE On-Demand Anodyne CACNA1I 73 42 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne HTR1A 65 50 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne DRD2 48 50 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne DRD4 44 36 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne ADRA1D 22 41 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne HTR2A 37 43 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne HTR2C 18 41 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne ADRA1A 21 41 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne DRD3 64 45 O=C(NCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770204 FD On-Demand Anodyne HTR7 66 42 COc1ccc(OCCNC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880770207 DE On-Demand Anodyne HRH2 16 40 O=C(NCc1cccc(OCC(F)(F)F)c1)Nc1ccn(CCF)n1 ZINC000880770208 FG On-Demand Anodyne PDS 42 36 CNC(=O)CN1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770209 EC On-Demand Anodyne DRD4 15 44 C=CC(C)(C)CC(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770213 CF On-Demand Mild CACNA1I 60 41 Cc1nn(-c2ccccc2)c(C)c1CNC(=O)Nc1ccn(CCF)n1 ZINC000880770219 FF On-Demand Anodyne P2RX7 26 52 O=C(CN1CCN(C(=O)Nc2ccn(CCF)n2)CC1)NCc1ccccc1 ZINC000880770227 GD On-Demand Anodyne HTR7 20 40 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne HTR1A 104 54 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne DRD2 75 46 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne DRD1 21 41 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne DRD4 42 46 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne ADRA1D 75 43 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne HTR1D 23 54 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne HTR1B 26 54 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne HTR2A 25 43 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne ADRA1A 70 43 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne ADRA1B 58 43 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne DRD3 83 44 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne PDGFRB 68 42 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne HTR7 71 47 COc1ccccc1N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770247 EE On-Demand Anodyne RBP4 22 45 O=C(CN1CCN(C(=O)Nc2ccn(CCF)n2)CC1)Nc1ccccc1 ZINC000880770307 FD On-Demand Anodyne FAAH 15 45 O=C(NCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880770312 CD On-Demand Anodyne HRH2 29 41 O=C(NCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880770312 CD On-Demand Anodyne CCR3 24 40 O=C(NCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880770312 CD On-Demand Anodyne CHRNA7 23 50 O=C(NCCCN1CCCCC1)Nc1ccn(CCF)n1 ZINC000880770312 CD On-Demand Anodyne HNMT 62 34 O=C(NCC1(N2CCOCC2)CCCCC1)Nc1ccn(CCF)n1 ZINC000880770330 FE On-Demand Anodyne HCN1 66 40 O=C(NCC1(N2CCOCC2)CCCCC1)Nc1ccn(CCF)n1 ZINC000880770330 FE On-Demand Anodyne HCN4 56 36 O=C(NCCCCc1ccccc1)Nc1ccn(CCF)n1 ZINC000880770342 DF On-Demand Anodyne FAAH 29 49 CCOC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770346 ED On-Demand Anodyne SSTR5 40 36 CCOC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770346 ED On-Demand Anodyne EPHX2 44 43 CCOC(=O)N1CCC(NC(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770346 ED On-Demand Anodyne CCR8 37 40 Cn1ncc2c(N3CCN(C(=O)Nc4ccn(CCF)n4)CC3)ncnc21 ZINC000880770355 FC On-Demand Anodyne PDGFRB 64 38 O=C(NCCc1ccc2c(c1)OCO2)Nc1ccn(CCF)n1 ZINC000880770358 DD On-Demand Anodyne NOS2 97 41 NC(=O)c1cccc2c1CCN(C(=O)COC1CC1)C2 ZINC000880770385 CC On-Demand Anodyne PARP1 17 54 Cn1nc2c(c1C(=O)NCC1CCN(CC3CC3)CC1)CSCC2 ZINC000880770407 EE On-Demand Anodyne CACNA1I 66 38 O=C(NCc1cccnc1N1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770408 ED On-Demand Anodyne SCN10A 20 45 O=C(Cc1ccccc1N1CCCC1=O)NCC1CCN(CC2CC2)CC1 ZINC000880770416 FF On-Demand Anodyne HTR4 46 38 O=C(Cc1ccccc1N1CCCC1=O)NCC1CCN(CC2CC2)CC1 ZINC000880770416 FF On-Demand Anodyne CACNA1I 61 41 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne GABRA1 18 46 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne HTR4 33 40 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne GRIN2B 19 48 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne CCR3 46 39 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne GABRA2 16 46 O=C(NCC1CCN(CC2CC2)CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880770420 FF On-Demand Anodyne CACNA1I 56 35 O=C(NCCCOc1ccccc1)Nc1ccn(CCF)n1 ZINC000880770422 DE On-Demand Anodyne HRH2 43 43 O=C(NCc1ccc2c(c1)OCCO2)Nc1ccn(CCF)n1 ZINC000880770425 DD On-Demand Anodyne NOS2 91 37 CCCCCNC(=O)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770430 FE On-Demand Anodyne ASAH1 41 34 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne HTR4 55 42 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne GRIN2B 26 44 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne SSTR5 43 33 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne CCR3 32 41 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne PLD1 26 40 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne PLD2 33 40 O=C(NCC1CCN(CC2CC2)CC1)c1cnc2cc[nH]c2c1 ZINC000880770431 DE On-Demand Anodyne CACNA1I 81 43 O=C(NCC1CCN(CC2CC2)CC1)c1cc2c(cc1[N+](=O)[O-])OCCCO2 ZINC000880770436 GF On-Demand Bother HTR4 61 45 O=C(NCC1CCN(CC2CC2)CC1)c1cc2c(cc1[N+](=O)[O-])OCCCO2 ZINC000880770436 GF On-Demand Bother CACNA1I 60 37 O=C(NCC1(N2CCSCC2)CCCC1)Nc1ccn(CCF)n1 ZINC000880770438 FE On-Demand Anodyne HCN1 68 39 O=C(NCC1(N2CCSCC2)CCCC1)Nc1ccn(CCF)n1 ZINC000880770438 FE On-Demand Anodyne HCN4 55 35 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770445 FE On-Demand Anodyne EPHX2 26 43 O=C(NCc1ccc(N2CCCC2)nc1)Nc1ccn(CCF)n1 ZINC000880770457 EE On-Demand Anodyne NAMPT 21 40 C=C1c2ccccc2C(=O)N1CC(=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880770527 FD On-Demand Anodyne PRKDC 46 37 C=C1c2ccccc2C(=O)N1CC(=O)Nc1ccc(N2CCOCC2)cn1 ZINC000880770527 FD On-Demand Anodyne STAT6 70 38 O=C(NCCN1CCOCC1)Nc1ccn(CCF)n1 ZINC000880770545 CC On-Demand Anodyne EPHX2 21 46 COc1ccc(C)cc1CN1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770546 GF On-Demand Anodyne SLC9A1 58 34 O=C(NCC1(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770574 DF On-Demand Anodyne KCNA3 47 39 O=C(NCC1(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770574 DF On-Demand Anodyne SOAT1 16 45 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne HTR1A 93 52 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne DRD2 76 53 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne DRD1 15 40 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne DRD4 45 48 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne ADRA1D 39 48 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne HTR2A 69 48 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne HTR2C 37 46 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne SLC6A4 17 42 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne ADRA1A 49 48 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne ADRA1B 27 48 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne DRD3 95 53 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne DRD5 15 40 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne HTR7 107 45 O=C(NCCCN1CCN(c2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770628 FE On-Demand Anodyne CCR3 28 42 O=C(c1ccccc1)C1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770637 EF On-Demand Anodyne SLC18A3 38 40 O=C(NCCCN1CCc2ccccc2C1)Nc1ccn(CCF)n1 ZINC000880770642 EE On-Demand Anodyne DRD3 16 46 O=C(NCCCN1CCc2ccccc2C1)Nc1ccn(CCF)n1 ZINC000880770642 EE On-Demand Anodyne NOD2 40 34 COc1ccc2cc(CN(C)C(=O)Nc3ccn(CCF)n3)ccc2c1 ZINC000880770645 FH On-Demand Anodyne ROCK1 15 41 COc1ccc2cc(CN(C)C(=O)Nc3ccn(CCF)n3)ccc2c1 ZINC000880770645 FH On-Demand Anodyne ROCK2 20 41 C[C@H](NC(=O)Nc1ccn(CCF)n1)c1ccc(-n2cncn2)cc1 ZINC000880770652 EE On-Demand Anodyne AMP1_PLAFQ 44 32 CC[C@@H]1CCCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770657 CF On-Demand Anodyne CCR3 32 47 CC[C@H]1CCCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770658 CF On-Demand Anodyne CCR3 32 47 CC[C@H]1CCCC[C@@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770659 CF On-Demand Anodyne CCR3 32 47 CC[C@@H]1CCCC[C@H]1NC(=O)Nc1ccn(CCF)n1 ZINC000880770660 CF On-Demand Anodyne CCR3 32 47 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne HTR1A 30 49 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne DRD2 21 49 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne DRD4 25 50 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne HTR2A 16 41 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne DRD3 28 41 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne HTR7 30 40 O=C(NCCN1CCN(c2ccc(F)cc2)CC1)Nc1ccn(CCF)n1 ZINC000880770661 GD On-Demand Anodyne SLC27A1 36 41 O=C(NCc1ccc(N2CCCCC2)nc1)Nc1ccn(CCF)n1 ZINC000880770671 EF On-Demand Anodyne NAMPT 23 40 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770680 EH On-Demand Anodyne ACHE 17 45 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770680 EH On-Demand Anodyne CHRM4 16 41 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770680 EH On-Demand Anodyne SIGMAR1 21 47 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770680 EH On-Demand Anodyne MTNR1A 17 43 O=C(CC[C@@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770680 EH On-Demand Anodyne CACNA1I 57 36 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770681 EH On-Demand Anodyne ACHE 17 45 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770681 EH On-Demand Anodyne CHRM4 16 41 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770681 EH On-Demand Anodyne SIGMAR1 21 47 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770681 EH On-Demand Anodyne MTNR1A 17 43 O=C(CC[C@H]1CCc2ccccc21)NCC1CCN(CC2CC2)CC1 ZINC000880770681 EH On-Demand Anodyne CACNA1I 57 36 NC(=O)[C@H](c1ccccc1)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770685 FD On-Demand Anodyne NPY2R 42 34 NC(=O)[C@@H](c1ccccc1)N1CCN(C(=O)Nc2ccn(CCF)n2)CC1 ZINC000880770686 FD On-Demand Anodyne NPY2R 42 34 COc1cccc([C@H](CNC(=O)Nc2ccn(CCF)n2)N(C)C)c1 ZINC000880770708 EE On-Demand Anodyne ROCK2 41 35 CCC[C@H](NC(=O)Nc1ccn(CCF)n1)c1ccccc1 ZINC000880770711 DH On-Demand Anodyne TACR3 39 41 O=C(NCCc1cccnc1)Nc1ccn(CCF)n1 ZINC000880770718 CD On-Demand Anodyne NAMPT 41 46 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccn(CCF)n1 ZINC000880770766 EF On-Demand Anodyne NOS2 77 34 CN(Cc1ccc(Cl)nc1)C(=O)Nc1ccn(CCF)n1 ZINC000880770774 DF On-Demand Anodyne NACHRBETA2 23 40 O=C(NCCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770777 DE On-Demand Anodyne HRH2 29 41 O=C(NCCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770777 DE On-Demand Anodyne CCR3 24 40 O=C(NCCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770777 DE On-Demand Anodyne CHRNA7 23 50 O=C(NCCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770777 DE On-Demand Anodyne HNMT 62 34 O=C(NCC1CCN(CC2CC2)CC1)c1cccc2nsnc12 ZINC000880770793 EF On-Demand Anodyne HTR4 69 52 O=C(NCC1CCN(CC2CC2)CC1)c1cccc2nsnc12 ZINC000880770793 EF On-Demand Anodyne CACNA1I 62 37 O=C(NCC1CCN(CC2CC2)CC1)c1ncsc1C1CC1 ZINC000880770817 DF On-Demand Anodyne HTR4 50 42 O=C(NCC1CCN(CC2CC2)CC1)c1ncsc1C1CC1 ZINC000880770817 DF On-Demand Anodyne CACNA1I 64 40 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880770845 FD On-Demand Anodyne MTNR1A 25 42 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne F2 22 43 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne DRD4 24 42 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne ACHE 42 42 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne HTR4 46 41 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne SIGMAR1 48 42 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CCN(CC3CC3)CC2)N1Cc1ccccc1 ZINC000880770853 GD On-Demand Anodyne CACNA1I 55 37 CCN(Cc1ccccc1)C(=O)Nc1ccn(CCF)n1 ZINC000880770893 CF On-Demand Anodyne TSPO 49 41 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccc(F)cc1 ZINC000880770915 GE On-Demand Anodyne DRD4 15 45 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccc(F)cc1 ZINC000880770915 GE On-Demand Anodyne MAPK13 54 34 O=C(NC1CCN(C(=O)Nc2ccn(CCF)n2)CC1)c1ccc(F)cc1 ZINC000880770915 GE On-Demand Anodyne MCHR1 16 44 CN(Cc1ccc(Cl)cc1Cl)C(=O)Nc1ccn(CCF)n1 ZINC000880770918 EH On-Demand Anodyne P2RX7 26 44 O=C(C[C@@H]1CCNC1=O)NCC1CCN(CC2CC2)CC1 ZINC000880770919 CC On-Demand Anodyne CACNA1I 50 35 O=C(C[C@H]1CCNC1=O)NCC1CCN(CC2CC2)CC1 ZINC000880770920 CC On-Demand Anodyne CACNA1I 50 35 Cn1nnc(C(=O)NCC2CCN(CC3CC3)CC2)n1 ZINC000880770921 CC On-Demand Anodyne HTR4 58 44 Cn1nnc(C(=O)NCC2CCN(CC3CC3)CC2)n1 ZINC000880770921 CC On-Demand Anodyne CACNA1I 72 42 O=C(NCc1ccc(F)cc1C(F)(F)F)Nc1ccn(CCF)n1 ZINC000880770922 EG On-Demand Anodyne P2RX7 46 46 COCc1ccccc1CNC(=O)Nc1ccn(CCF)n1 ZINC000880770923 DE On-Demand Anodyne MT-CYB 42 32 COc1cc2c(cc1OC)CN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880770929 EE On-Demand Anodyne ABCB1B 62 39 COc1cc2c(cc1OC)CN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880770929 EE On-Demand Anodyne ABCB1 21 43 COc1cc2c(cc1OC)CN(C(=O)Nc1ccn(CCF)n1)CC2 ZINC000880770929 EE On-Demand Anodyne ABCG2 36 40 C[C@@H](Sc1nc(CC(=O)NCC2CCN(CC3CC3)CC2)cs1)C(N)=O ZINC000880770942 GD On-Demand Anodyne CACNA1I 53 36 C[C@H](Sc1nc(CC(=O)NCC2CCN(CC3CC3)CC2)cs1)C(N)=O ZINC000880770943 GD On-Demand Anodyne CACNA1I 53 36 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne HTR1A 36 42 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne DRD2 49 40 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne DRD4 37 40 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne ACHE 27 42 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne HRH2 42 41 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne HTR2A 34 43 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne DRD3 67 40 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne HTR7 39 45 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne SIGMAR1 38 42 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne BCHE 15 42 O=C(NCCCN1CCN(Cc2ccccc2)CC1)Nc1ccn(CCF)n1 ZINC000880770946 GE On-Demand Anodyne CCR3 37 48 COc1ccc2[nH]cc(C3=CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880770947 GH On-Demand Anodyne HTR1A 15 45 COc1ccc2[nH]cc(C3=CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880770947 GH On-Demand Anodyne HTR1D 23 47 COc1ccc2[nH]cc(C3=CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880770947 GH On-Demand Anodyne HTR1B 20 47 COc1ccc2[nH]cc(C3=CCN(C(=O)Nc4ccn(CCF)n4)CC3)c2c1 ZINC000880770947 GH On-Demand Anodyne SLC6A4 15 54 O=C(NCC1CCN(CC2CC2)CC1)c1csc(-c2ncc[nH]2)n1 ZINC000880770955 EE On-Demand Anodyne CACNA1I 62 35 O=C(NCC1CCN(CC2CC2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880770956 EG On-Demand Anodyne ACHE 15 41 O=C(NCC1CCN(CC2CC2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880770956 EG On-Demand Anodyne HTR4 44 36 O=C(NCC1CCN(CC2CC2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880770956 EG On-Demand Anodyne SIGMAR1 34 46 O=C(NCC1CCN(CC2CC2)CC1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880770956 EG On-Demand Anodyne CACNA1I 60 47 O=C(NCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770959 CD On-Demand Anodyne CHRNA7 18 44 O=C(NCCN1CCCCCC1)Nc1ccn(CCF)n1 ZINC000880770959 CD On-Demand Anodyne HNMT 46 32 O=C(NCC1CCN(CC2CC2)CC1)c1coc(-c2ccccn2)n1 ZINC000880770961 EF On-Demand Anodyne HTR4 60 39 O=C(NCC1CCN(CC2CC2)CC1)c1coc(-c2ccccn2)n1 ZINC000880770961 EF On-Demand Anodyne CACNA1I 59 35 O=C(NCC1CCN(CC2CC2)CC1)c1cccn2nccc12 ZINC000880770965 DE On-Demand Anodyne HTR4 71 46 O=C(NCC1CCN(CC2CC2)CC1)c1cccn2nccc12 ZINC000880770965 DE On-Demand Anodyne CACNA1I 66 38 O=C(NCC1CCN(CC2CC2)CC1)c1cccn2nccc12 ZINC000880770965 DE On-Demand Anodyne HCN1 47 32 O=C(NCC1CCN(CC2CC2)CC1)c1cccn2nccc12 ZINC000880770965 DE On-Demand Anodyne HCN4 41 32 O=C(NCC1CCN(CC2CC2)CC1)c1cncc2[nH]ccc12 ZINC000880770975 DE On-Demand Anodyne HTR4 66 45 O=C(NCC1CCN(CC2CC2)CC1)c1cncc2[nH]ccc12 ZINC000880770975 DE On-Demand Anodyne CCR3 21 42 O=C(NCC1CCN(CC2CC2)CC1)c1cncc2[nH]ccc12 ZINC000880770975 DE On-Demand Anodyne CACNA1I 64 37 O=C(NCCc1ccc2c(c1)OCCO2)Nc1ccn(CCF)n1 ZINC000880770981 ED On-Demand Anodyne NOS2 73 37 CS(=O)(=O)C1CCC(C(=O)NCC2CCN(CC3CC3)CC2)CC1 ZINC000880770989 FD On-Demand Anodyne CACNA1I 46 33 O=C(C[C@@H]1C[C@H]1C1CC1)NCC1CCN(CC2CC2)CC1 ZINC000880770990 CF On-Demand Anodyne CACNA1I 45 34 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880770999 EE On-Demand Anodyne CACNA1I 49 32 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771000 EE On-Demand Anodyne CACNA1I 49 32 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771001 EE On-Demand Anodyne CACNA1I 49 32 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771002 EE On-Demand Anodyne CACNA1I 49 32 C[C@H](NC(=O)Nc1ccn(CCF)n1)c1ccc2c(c1)OCO2 ZINC000880771006 DE On-Demand Anodyne KCNQ2 21 42 O=C(NCC1CCN(CC2CC2)CC1)c1cnc(CC2CC2)s1 ZINC000880771020 EF On-Demand Anodyne HTR4 50 40 O=C(NCC1CCN(CC2CC2)CC1)c1cnc(CC2CC2)s1 ZINC000880771020 EF On-Demand Anodyne CACNA1I 69 42 O=C(NCC1CCN(CC2CC2)CC1)c1ncccc1-c1ccccn1 ZINC000880771024 FF On-Demand Anodyne HTR4 65 44 O=C(NCC1CCN(CC2CC2)CC1)c1ncccc1-c1ccccn1 ZINC000880771024 FF On-Demand Anodyne CACNA1I 62 37 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne DRD2 48 49 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne DRD4 32 49 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne ACHE 15 42 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne DRD3 48 42 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne HTR4 80 47 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne HTR7 31 41 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne CCR3 27 41 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne CACNA1I 63 34 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne HCN1 62 33 COc1ccccc1-c1ccc(C(=O)NCC2CCN(CC3CC3)CC2)c(O)n1 ZINC000880771029 GG On-Demand Anodyne HCN4 51 33 O=C(NCCOc1ccccc1F)Nc1ccn(CCF)n1 ZINC000880771030 DE On-Demand Anodyne ADRB1 41 35 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne HTR1B 16 40 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne CCKAR 36 42 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne BRS3 27 41 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne NMBR 51 44 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne GHSR 45 39 O=C(NCCc1c[nH]c2ccccc12)Nc1ccn(CCF)n1 ZINC000880771072 DF On-Demand Anodyne MMP9 15 51 CCOc1ccc([C@@H](C)NC(=O)Nc2ccn(CCF)n2)cc1 ZINC000880771073 DG On-Demand Anodyne ACACB 21 45 Cc1cnc(Cl)c(C(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880771079 DF On-Demand Anodyne HTR4 72 51 Cc1cnc(Cl)c(C(=O)NCC2CCN(CC3CC3)CC2)c1 ZINC000880771079 DF On-Demand Anodyne CACNA1I 94 49 O=C(NCC1CCN(CC2CC2)CC1)[C@H]1CCc2nncn2CC1 ZINC000880771082 ED On-Demand Anodyne CACNA1I 51 37 O=C(NCC1CCN(CC2CC2)CC1)[C@@H]1CCc2nncn2CC1 ZINC000880771083 ED On-Demand Anodyne CACNA1I 51 37 Cn1ncc(Br)c1CC(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771088 FD On-Demand Anodyne HTR4 42 39 Cn1ncc(Br)c1CC(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771088 FD On-Demand Anodyne CACNA1I 69 44 CC(=O)Nc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880771099 DE On-Demand Anodyne HTR1D 17 40 CC(=O)Nc1cccc(CNC(=O)Nc2ccn(CCF)n2)c1 ZINC000880771099 DE On-Demand Anodyne ROCK2 22 47 O=C(NCc1cccc(CN2CCCC2)c1)Nc1ccn(CCF)n1 ZINC000880771104 EF On-Demand Anodyne HRH2 49 44 O=C(NCc1cccc(CN2CCCC2)c1)Nc1ccn(CCF)n1 ZINC000880771104 EF On-Demand Anodyne ROCK2 21 40 C#C[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771119 DI On-Demand Mild RBP4 85 46 C#C[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771119 DI On-Demand Mild SMO 17 41 C#C[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771119 DI On-Demand Mild WNT3 48 34 C#C[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771120 DI On-Demand Mild RBP4 85 46 C#C[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771120 DI On-Demand Mild SMO 17 41 C#C[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771120 DI On-Demand Mild WNT3 48 34 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771129 EF On-Demand Anodyne HTR4 57 49 Cc1nc(C(C)C)ncc1C(=O)NCC1CCN(CC2CC2)CC1 ZINC000880771129 EF On-Demand Anodyne CACNA1I 69 38 CCc1nccn1C[C@H]1CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880771189 GJ On-Demand Anodyne RBP4 42 34 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771223 DH On-Demand Anodyne TIMP3 47 32 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771223 DH On-Demand Anodyne EPHX2 39 41 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771223 DH On-Demand Anodyne RBP4 49 33 CCN1CC[C@H](N(CC)C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771276 EI On-Demand Anodyne CCR5 24 44 CCN1CC[C@H](N(CC)C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771276 EI On-Demand Anodyne RBP4 75 38 CCN1CC[C@@H](N(CC)C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771277 EI On-Demand Anodyne CCR5 24 44 CCN1CC[C@@H](N(CC)C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771277 EI On-Demand Anodyne RBP4 75 38 C#CC[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771367 DI On-Demand Mild RBP4 87 47 C#CC[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771368 DI On-Demand Mild RBP4 87 47 C#CCNS(=O)(=O)c1ccc(C(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880771401 HD On-Demand Mild F10 27 42 C#CCNS(=O)(=O)c1ccc(C(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880771401 HD On-Demand Mild PRNP 48 43 C#CCNS(=O)(=O)c1ccc(C(=O)Nc2ccc(N3CCOCC3)cn2)cc1 ZINC000880771401 HD On-Demand Mild STAT6 51 31 CCc1noc([C@]2(O)CCN(C(=O)Nc3ccccc3C(F)(F)CC)C2)n1 ZINC000880771425 GG On-Demand Anodyne RBP4 52 32 CCc1noc([C@@]2(O)CCN(C(=O)Nc3ccccc3C(F)(F)CC)C2)n1 ZINC000880771426 GG On-Demand Anodyne RBP4 52 32 C#CC1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880771624 DI On-Demand Mild RBP4 95 47 C#CC1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880771624 DI On-Demand Mild SMO 19 42 C#CC1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880771624 DI On-Demand Mild WNT3 45 34 CCN1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1=O ZINC000880771885 EF On-Demand Anodyne RBP4 62 35 CCN1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1=O ZINC000880771887 EF On-Demand Anodyne RBP4 62 35 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CC12COC2 ZINC000880771908 GG On-Demand Anodyne RBP4 64 37 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771976 FH On-Demand Anodyne RBP4 82 41 C=CC[C@@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771978 DJ On-Demand Mild RBP4 89 43 C=CC[C@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771980 DJ On-Demand Mild RBP4 89 43 CCC(=O)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880771993 EG On-Demand Anodyne RBP4 78 42 CCn1c(O)nnc1C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880772065 GH On-Demand Anodyne RBP4 85 46 CCn1c(O)nnc1C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880772065 GH On-Demand Anodyne SMO 19 45 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880772074 GI On-Demand Anodyne KCNQ2 42 33 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880772074 GI On-Demand Anodyne RBP4 86 42 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1ccccc1C(F)(F)CC ZINC000880772075 DJ On-Demand Mild RBP4 64 37 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880772089 FH On-Demand Anodyne RBP4 82 41 CC[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)C(N)=O ZINC000880772096 CF On-Demand Anodyne ANPEP 20 54 CC[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)C(N)=O ZINC000880772096 CF On-Demand Anodyne NPFFR1 44 31 CCN1C[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)CC1=O ZINC000880772162 EF On-Demand Anodyne EPHX2 21 42 CC[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)C(=O)NC ZINC000880772225 DF On-Demand Anodyne ANPEP 19 54 CCO[C@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880772371 DH On-Demand Anodyne TIMP3 47 32 CCO[C@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880772371 DH On-Demand Anodyne EPHX2 39 41 CCO[C@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880772371 DH On-Demand Anodyne RBP4 49 33 CC[C@H](C)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880772389 EI On-Demand Anodyne RBP4 86 41 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccc(N2CCOCC2)nc1 ZINC000880772418 IG On-Demand Anodyne HDAC1 23 42 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccc(N2CCOCC2)nc1 ZINC000880772418 IG On-Demand Anodyne DGAT1 32 43 O=C(Nc1cc(-c2nnc3n2CCCCC3)ccc1F)c1ccc(N2CCOCC2)nc1 ZINC000880772418 IG On-Demand Anodyne HPGDS 18 42 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880772449 EI On-Demand Anodyne TIMP3 63 32 CC[C@H]1C[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880772509 EI On-Demand Anodyne EPHX2 19 41 CC[C@@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880772511 EI On-Demand Anodyne EPHX2 19 41 CC[C@H]1C[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880772512 EI On-Demand Anodyne EPHX2 19 41 C#CC1(F)CN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880772632 CG On-Demand Mild RBP4 68 39 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772790 EG On-Demand Anodyne MTNR1A 34 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772790 EG On-Demand Anodyne MTNR1B 36 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772790 EG On-Demand Anodyne FAAH 15 45 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772792 EG On-Demand Anodyne MTNR1A 34 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772792 EG On-Demand Anodyne MTNR1B 36 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@H](C)O)C2 ZINC000880772792 EG On-Demand Anodyne FAAH 15 45 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772794 EG On-Demand Anodyne MTNR1A 34 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772794 EG On-Demand Anodyne MTNR1B 36 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772794 EG On-Demand Anodyne FAAH 15 45 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772797 EG On-Demand Anodyne MTNR1A 34 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772797 EG On-Demand Anodyne MTNR1B 36 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](c1ccccc1)[C@@H](C)O)C2 ZINC000880772797 EG On-Demand Anodyne FAAH 15 45 CCOC(=O)[C@@]1(C)CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880772927 FG On-Demand Anodyne RBP4 53 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CTSD 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne PGC 58 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne KLK3 71 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CTSB 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne PAPA1_CARPA 56 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CYSP_TRYCR 44 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CCKAR 46 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CTSK 35 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CTSL 28 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne PGA 42 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne TACR3 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CAPNS1 54 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne HLA-DRB1 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne REN 75 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne REN1 28 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CTSS 18 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CAPN1 64 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne CAPN2 97 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@H](C)O ZINC000880773136 FE On-Demand Anodyne FPR1 78 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CTSD 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne PGC 58 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne KLK3 71 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CTSB 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne PAPA1_CARPA 56 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CYSP_TRYCR 44 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CCKAR 46 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CTSK 35 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CTSL 28 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne PGA 42 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne TACR3 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CAPNS1 54 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne HLA-DRB1 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne REN 75 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne REN1 28 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CTSS 18 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CAPN1 64 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne CAPN2 97 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@H](C)O ZINC000880773137 FE On-Demand Anodyne FPR1 78 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CTSD 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne PGC 58 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne KLK3 71 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CTSB 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne PAPA1_CARPA 56 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CYSP_TRYCR 44 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CCKAR 46 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CTSK 35 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CTSL 28 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne PGA 42 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne TACR3 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CAPNS1 54 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne HLA-DRB1 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne REN 75 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne REN1 28 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CTSS 18 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CAPN1 64 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne CAPN2 97 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccc1)[C@@H](C)O ZINC000880773138 FE On-Demand Anodyne FPR1 78 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CTSD 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne PGC 58 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne KLK3 71 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CTSB 41 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne PAPA1_CARPA 56 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CYSP_TRYCR 44 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CCKAR 46 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CTSK 35 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CTSL 28 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne PGA 42 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne TACR3 20 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CAPNS1 54 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne HLA-DRB1 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne REN 75 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne REN1 28 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CTSS 18 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CAPN1 64 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne CAPN2 97 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne POLG_HCV1 24 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccc1)[C@@H](C)O ZINC000880773140 FE On-Demand Anodyne FPR1 78 48 C#C[C@@H]1COCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773153 DG On-Demand Mild RBP4 59 36 C#C[C@H]1COCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773156 DG On-Demand Mild RBP4 59 36 C#CCC1(O)CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880773205 EH On-Demand Mild RBP4 61 39 CCn1cc([C@@H]2OCC[C@H]2NC(=O)Nc2ccccc2C(F)(F)CC)cn1 ZINC000880773218 GI On-Demand Anodyne RBP4 41 32 CC[C@@H]1CN(C)CCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773247 EH On-Demand Anodyne RBP4 75 40 CC[C@H]1CN(C)CCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773250 EH On-Demand Anodyne RBP4 75 40 C#CCN(C(=O)Nc1ccccc1C(F)(F)CC)C1CC1 ZINC000880773299 CH On-Demand Mild RBP4 72 35 CC[C@H]1[C@@H](CO)CCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773311 EH On-Demand Anodyne RBP4 74 37 CCOC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880773342 EG On-Demand Anodyne RBP4 73 41 CC[C@@H]1[C@H](CO)CCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773413 EH On-Demand Anodyne RBP4 74 37 CC[C@H]1[C@H](CO)CCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773414 EH On-Demand Anodyne RBP4 74 37 CCOC[C@H]1CCCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773447 EJ On-Demand Anodyne RBP4 63 37 C#CCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880773654 FG On-Demand Mild RBP4 83 45 C#CCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880773654 FG On-Demand Mild CACNA1G 36 41 NC(=O)NCCCCCC(=O)N1CCC(c2ccc(F)cn2)CC1 ZINC000880773694 EE On-Demand Anodyne ETHR 41 33 CCC[C@H](NC(=O)Nc1ccccc1C(F)(F)CC)C(N)=O ZINC000880773706 DF On-Demand Anodyne ANPEP 15 52 C=C[C@@H]1CCCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773777 DJ On-Demand Mild RBP4 68 38 C=C[C@H]1CCCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880773778 DJ On-Demand Mild RBP4 68 38 CCC[C@]1(CO)CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880773784 EI On-Demand Anodyne RBP4 89 40 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H](C)S1(=O)=O ZINC000880773931 FH On-Demand Anodyne RBP4 80 44 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@H](C)S1(=O)=O ZINC000880773933 FH On-Demand Anodyne RBP4 80 44 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCCO1 ZINC000880773967 EI On-Demand Anodyne RBP4 90 47 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCCO1 ZINC000880773967 EI On-Demand Anodyne SMO 25 43 O=C(c1c[nH]cc1C1CC1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880773974 DG On-Demand Anodyne HTR1F 58 37 O=C(c1c[nH]cc1C1CC1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880773974 DG On-Demand Anodyne RBP4 26 40 Cc1nn(CC(=O)N2CCC(c3ccc(F)cn3)CC2)c(=O)o1 ZINC000880774053 DD On-Demand Anodyne ETHR 40 32 C#C[C@H](CC)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880774122 CH On-Demand Mild KCNQ2 40 37 C#C[C@@H](CC)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880774123 CH On-Demand Mild KCNQ2 40 37 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(c4ccc(F)cn4)CC3)cc2)N1 ZINC000880774189 FG On-Demand Anodyne L3MBTL3 43 34 O=C1CC[C@H](c2ccc(C(=O)N3CCC(c4ccc(F)cn4)CC3)cc2)N1 ZINC000880774190 FG On-Demand Anodyne L3MBTL3 43 34 CCC1(O)CN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880774210 CG On-Demand Anodyne RBP4 73 41 O=C(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880774283 FH On-Demand Bother L3MBTL3 40 44 CCn1ccnc1[C@H]1CCCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880774319 GK On-Demand Anodyne RBP4 46 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccc(F)cn2)CC1 ZINC000880774326 GF On-Demand Anodyne P2RY12 134 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(c2ccc(F)cn2)CC1 ZINC000880774327 GF On-Demand Anodyne P2RY12 134 37 C[C@@H]1[C@@H](C(=O)N2CCC(c3ccc(F)cn3)CC2)CCN1C ZINC000880774378 DE On-Demand Anodyne PRCP 51 36 C[C@H]1[C@H](C(=O)N2CCC(c3ccc(F)cn3)CC2)CCN1C ZINC000880774379 DE On-Demand Anodyne PRCP 51 36 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne F10 22 47 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne PRNP 54 46 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne HDAC1 21 42 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne STAT6 55 34 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne DGAT1 24 44 O=C(Nc1ccc(N2CCOCC2)cn1)c1ccc(N2CCOCC2)nc1 ZINC000880774464 FD On-Demand Anodyne HPGDS 22 49 Cc1cnc(Cl)c(C(=O)N2CCC(c3ccc(F)cn3)CC2)c1 ZINC000880774549 EH On-Demand Anodyne PRCP 47 34 CCn1cccc(CNC(=O)Nc2ccccc2C(F)(F)CC)c1=O ZINC000880774585 EH On-Demand Anodyne P2RX7 42 38 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880774640 GF On-Demand Anodyne HLA-DRB1 70 37 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880774642 GF On-Demand Anodyne HLA-DRB1 70 37 CCOC(=O)[C@@]1(COC)CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880774675 GI On-Demand Anodyne RBP4 53 34 CCOC(=O)[C@]1(COC)CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880774676 GI On-Demand Anodyne RBP4 53 34 NS(=O)(=O)c1cc(CNC(=O)COC2CC2)ccc1F ZINC000880774806 DC On-Demand Anodyne CA2 22 41 NS(=O)(=O)c1cc(CNC(=O)COC2CC2)ccc1F ZINC000880774806 DC On-Demand Anodyne CA1 21 41 NS(=O)(=O)c1cc(CNC(=O)COC2CC2)ccc1F ZINC000880774806 DC On-Demand Anodyne CA9 20 41 CCN1CC[C@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)[C@H](C)C1 ZINC000880774836 FI On-Demand Anodyne RBP4 46 34 CCN1CC[C@@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)[C@H](C)C1 ZINC000880774837 FI On-Demand Anodyne RBP4 46 34 CC[C@@H](C(=O)N1CCC(c2ccc(F)cn2)CC1)[C@@H](C)O ZINC000880774838 CE On-Demand Anodyne CCR1 26 40 CCN1CC[C@@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)[C@@H](C)C1 ZINC000880774839 FI On-Demand Anodyne RBP4 46 34 CC[C@H](C(=O)N1CCC(c2ccc(F)cn2)CC1)[C@H](C)O ZINC000880774840 CE On-Demand Anodyne CCR1 26 40 CCN1CC[C@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)[C@@H](C)C1 ZINC000880774841 FI On-Demand Anodyne RBP4 46 34 CC[C@H](C(=O)N1CCC(c2ccc(F)cn2)CC1)[C@@H](C)O ZINC000880774843 CE On-Demand Anodyne CCR1 26 40 CC[C@@H](C(=O)N1CCC(c2ccc(F)cn2)CC1)[C@H](C)O ZINC000880774844 CE On-Demand Anodyne CCR1 26 40 C=CCN(C(=O)Nc1ccccc1C(F)(F)CC)C1CC1 ZINC000880774930 CI On-Demand Mild RBP4 66 35 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880774941 GF On-Demand Anodyne RBP4 86 44 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880774943 GF On-Demand Anodyne RBP4 86 44 O=C(CCCCCc1ccc(O)cc1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880774954 FI On-Demand Anodyne ETHR 41 33 CCc1nnc2n1C[C@H](NC(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775115 FG On-Demand Anodyne EPHX2 23 41 CCc1nnc2n1C[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775116 FG On-Demand Anodyne EPHX2 23 41 CNc1nc(C(=O)N2CCC(c3ccc(F)cn3)CC2)cs1 ZINC000880775161 DF On-Demand Anodyne TRPC6 66 47 CNc1nc(C(=O)N2CCC(c3ccc(F)cn3)CC2)cs1 ZINC000880775161 DF On-Demand Anodyne TRPC3 58 47 CCn1cc([C@@H]2CN(C(=O)Nc3ccccc3C(F)(F)CC)CCO2)cn1 ZINC000880775162 GI On-Demand Anodyne RBP4 68 39 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775227 GH On-Demand Anodyne RBP4 68 38 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775228 GH On-Demand Anodyne RBP4 68 38 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775229 GH On-Demand Anodyne RBP4 68 38 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880775230 GH On-Demand Anodyne RBP4 68 38 CCC1(CO)CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880775277 EI On-Demand Anodyne RBP4 92 43 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(F)c(S(N)(=O)=O)c1)C2 ZINC000880775317 GD On-Demand Anodyne CA12 17 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(F)c(S(N)(=O)=O)c1)C2 ZINC000880775317 GD On-Demand Anodyne CA9 19 41 C#CCN(C)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880775400 CG On-Demand Mild RBP4 21 42 CCOCCOC1CN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775478 EG On-Demand Anodyne RBP4 81 41 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@H]1N1CCOCC1 ZINC000880775486 GH On-Demand Anodyne RBP4 78 42 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H]1N1CCOCC1 ZINC000880775488 GH On-Demand Anodyne RBP4 78 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775502 GI On-Demand Anodyne EPHX2 32 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775502 GI On-Demand Anodyne RBP4 58 34 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775503 GI On-Demand Anodyne EPHX2 32 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775503 GI On-Demand Anodyne RBP4 58 34 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775529 EG On-Demand Anodyne EPHX2 50 53 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775529 EG On-Demand Anodyne RBP4 71 36 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775529 EG On-Demand Anodyne CCR8 49 36 CCC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775530 EG On-Demand Anodyne EPHX2 50 53 CCC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775530 EG On-Demand Anodyne RBP4 71 36 CCC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775530 EG On-Demand Anodyne CCR8 49 36 CC[C@@H](C)C(=O)NNC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775607 DG On-Demand Reactive ANPEP 15 51 O=C(/C=C\c1cccnc1)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000880775612 FH On-Demand Anodyne MCHR1 17 41 O=C(CCc1cn[nH]c1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880775662 DE On-Demand Anodyne C3AR1 35 40 O=C(CCc1cn[nH]c1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880775662 DE On-Demand Anodyne ETHR 40 32 CCN1CCC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775695 EH On-Demand Anodyne KCNQ2 50 33 CCN1CCC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775695 EH On-Demand Anodyne CCR3 33 41 CCN1CCC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775695 EH On-Demand Anodyne EPHX2 40 46 CCN1CCC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775695 EH On-Demand Anodyne RBP4 75 38 CCN1CCC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775696 EH On-Demand Anodyne KCNQ2 50 33 CCN1CCC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775696 EH On-Demand Anodyne CCR3 33 41 CCN1CCC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775696 EH On-Demand Anodyne EPHX2 40 46 CCN1CCC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880775696 EH On-Demand Anodyne RBP4 75 38 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775773 FH On-Demand Anodyne RBP4 71 36 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775774 FH On-Demand Anodyne RBP4 71 36 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775775 FH On-Demand Anodyne RBP4 71 36 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775776 FH On-Demand Anodyne RBP4 71 36 CCN(C)C(=O)[C@@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775827 EG On-Demand Anodyne ANPEP 15 51 CCN(C)C(=O)[C@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880775828 EG On-Demand Anodyne ANPEP 15 51 C=CCN(C)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880775892 CH On-Demand Mild RBP4 17 42 O=C(c1ccc2nc(Cl)ccc2c1)N1CCC(c2ccc(F)cn2)CC1 ZINC000880775924 FI On-Demand Anodyne L3MBTL3 48 39 C=CC(C)(C)CC(=O)NCc1ccc(F)c(S(N)(=O)=O)c1 ZINC000880775932 DD On-Demand Mild CA2 20 41 C=CC(C)(C)CC(=O)NCc1ccc(F)c(S(N)(=O)=O)c1 ZINC000880775932 DD On-Demand Mild CA1 19 41 C=CC(C)(C)CC(=O)NCc1ccc(F)c(S(N)(=O)=O)c1 ZINC000880775932 DD On-Demand Mild TRPV1 20 41 C=CC(C)(C)CC(=O)NCc1ccc(F)c(S(N)(=O)=O)c1 ZINC000880775932 DD On-Demand Mild CA9 15 41 CCC1(O)CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880775945 EI On-Demand Anodyne EPHX2 38 46 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776005 FH On-Demand Anodyne EPHX2 52 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776005 FH On-Demand Anodyne RBP4 74 35 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776005 FH On-Demand Anodyne CCR8 82 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776005 FH On-Demand Anodyne SFRP1 67 33 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776005 FH On-Demand Anodyne WNT3 43 32 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776007 FH On-Demand Anodyne EPHX2 52 42 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776007 FH On-Demand Anodyne RBP4 74 35 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776007 FH On-Demand Anodyne CCR8 82 42 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776007 FH On-Demand Anodyne SFRP1 67 33 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776007 FH On-Demand Anodyne WNT3 43 32 CCC[C@]1(CO)CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880776087 EI On-Demand Anodyne RBP4 73 38 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)c1cnc(C2CC2)o1 ZINC000880776110 EF On-Demand Anodyne GPR119 29 42 O=C(NCCOCCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880776113 FD On-Demand Anodyne CELA1 19 42 O=C(NCCOCCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880776113 FD On-Demand Anodyne PREP 27 42 O=C(NCCOCCF)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880776113 FD On-Demand Anodyne Q9NAW4_PLAFA 38 45 C=CCNC(=O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880776114 GF On-Demand Mild RBP4 61 37 CCc1nccn1[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776122 GJ On-Demand Anodyne RBP4 75 41 CCc1nccn1[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776123 GJ On-Demand Anodyne RBP4 75 41 Cc1ncc(CC(=O)N2[C@H]3CC[C@H]2CN(C(=O)OC(C)(C)C)C3)o1 ZINC000880776129 EE On-Demand Anodyne GPR119 37 41 COC(=O)c1cnc([C@@H]2CCCN(C(=O)c3coc(-c4ccccn4)n3)C2)s1 ZINC000880776217 GF On-Demand Anodyne MAP3K12 31 41 COC(=O)c1cnc([C@H]2CCCN(C(=O)c3coc(-c4ccccn4)n3)C2)s1 ZINC000880776220 GF On-Demand Anodyne MAP3K12 31 41 CCC[C@H]1C(=O)NCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880776317 EG On-Demand Anodyne RBP4 72 35 CCC[C@@H]1C(=O)NCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880776318 EG On-Demand Anodyne RBP4 72 35 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880776325 GJ On-Demand Anodyne EPHX2 27 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880776325 GJ On-Demand Anodyne RBP4 64 34 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880776327 GJ On-Demand Anodyne EPHX2 27 42 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880776327 GJ On-Demand Anodyne RBP4 64 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)C[C@H]1CC1(C)C ZINC000880776339 EE On-Demand Anodyne CTSK 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)C[C@H]1CC1(C)C ZINC000880776340 EE On-Demand Anodyne CTSK 15 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)C[C@@H]1CC1(C)C ZINC000880776342 EE On-Demand Anodyne CTSK 15 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)C[C@@H]1CC1(C)C ZINC000880776343 EE On-Demand Anodyne CTSK 15 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC2CC1(c1ccccc1)C2 ZINC000880776353 FG On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC2CC1(c1ccccc1)C2 ZINC000880776353 FG On-Demand Anodyne FPR1 46 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2CC1(c1ccccc1)C2 ZINC000880776355 FG On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC2CC1(c1ccccc1)C2 ZINC000880776355 FG On-Demand Anodyne FPR1 46 35 CCc1cnc(CN(C)C(=O)Nc2ccccc2C(F)(F)CC)s1 ZINC000880776417 FJ On-Demand Anodyne RBP4 17 40 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880776467 EI On-Demand Anodyne RBP4 53 40 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880776469 EI On-Demand Anodyne RBP4 53 40 CC[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)c1nnc2n1CCCCC2 ZINC000880776472 GJ On-Demand Anodyne KCNQ2 48 33 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776486 FH On-Demand Anodyne RBP4 79 44 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776486 FH On-Demand Anodyne SFRP1 47 33 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776486 FH On-Demand Anodyne WNT3 43 33 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880776545 FF On-Demand Anodyne RBP4 74 41 O=C1CC[C@H](c2ccc(C(=O)NCCOCCF)cc2)N1 ZINC000880776548 CD On-Demand Anodyne PLD1 47 37 O=C1CC[C@H](c2ccc(C(=O)NCCOCCF)cc2)N1 ZINC000880776548 CD On-Demand Anodyne PLD2 41 35 O=C1CC[C@@H](c2ccc(C(=O)NCCOCCF)cc2)N1 ZINC000880776549 CD On-Demand Anodyne PLD1 47 37 O=C1CC[C@@H](c2ccc(C(=O)NCCOCCF)cc2)N1 ZINC000880776549 CD On-Demand Anodyne PLD2 41 35 O=C(NCCOCCF)c1cc2cc(F)ccc2[nH]c1=O ZINC000880776588 CD On-Demand Anodyne CNR2 35 41 O=C(NCCOCCF)c1cc2cc(F)ccc2[nH]c1=O ZINC000880776588 CD On-Demand Anodyne PLD2 42 38 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)c1coc(-c2ccccn2)n1 ZINC000880776589 GF On-Demand Anodyne GPR119 19 42 CC[C@H](O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880776625 FG On-Demand Anodyne RBP4 80 40 CC[C@@H](O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880776626 FG On-Demand Anodyne RBP4 80 40 CCC[C@@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880776655 EI On-Demand Anodyne RBP4 87 43 CCC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880776658 EI On-Demand Anodyne RBP4 87 43 C=CC(C)(C)CC(=O)N1CCC(NC(=O)OC)CC1 ZINC000880776739 CD On-Demand Mild EPHX2 21 40 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NCCOCCF)ccn2)CC1 ZINC000880776808 GD On-Demand Anodyne DRD4 40 31 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NCCOCCF)ccn2)CC1 ZINC000880776808 GD On-Demand Anodyne GPR119 33 42 CCOCCN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880776861 FG On-Demand Anodyne RBP4 68 39 CCN(CC)C(=O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880776899 GG On-Demand Anodyne RBP4 73 41 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H]1O ZINC000880776935 DG On-Demand Anodyne RBP4 96 46 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@H]1O ZINC000880776937 DG On-Demand Anodyne RBP4 96 46 CC[C@H]1CCC[C@@]1(C)C(=O)N1CCC(NC(=O)OC)CC1 ZINC000880776963 CF On-Demand Anodyne EPHX2 15 40 CC[C@H]1CCC[C@]1(C)C(=O)N1CCC(NC(=O)OC)CC1 ZINC000880776964 CF On-Demand Anodyne EPHX2 15 40 CC[C@@H]1CCC[C@@]1(C)C(=O)N1CCC(NC(=O)OC)CC1 ZINC000880776965 CF On-Demand Anodyne EPHX2 15 40 CC[C@@H]1CCC[C@]1(C)C(=O)N1CCC(NC(=O)OC)CC1 ZINC000880776966 CF On-Demand Anodyne EPHX2 15 40 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880776979 GG On-Demand Anodyne RBP4 54 33 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccccc1C(F)(F)CC)CC2 ZINC000880776979 GG On-Demand Anodyne P2RY14 47 33 CCN1CC[C@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)C[C@H]1C ZINC000880776981 FJ On-Demand Anodyne RBP4 76 38 CCN1CC[C@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H]1C ZINC000880776982 FJ On-Demand Anodyne RBP4 76 38 CCN1CC[C@@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)C[C@H]1C ZINC000880776983 FJ On-Demand Anodyne RBP4 76 38 CCN1CC[C@@H](N(C)C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H]1C ZINC000880776984 FJ On-Demand Anodyne RBP4 76 38 CCOC[C@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880776996 EI On-Demand Anodyne RBP4 90 46 O=C(Nc1ccc(N2CCOCC2)cn1)C1=CC=CN2CCS(=O)(=O)N=C12 ZINC000880777024 GC On-Demand Anodyne STAT6 51 31 CCC1(O)CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880777030 EH On-Demand Anodyne RBP4 79 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCOCCF)C2 ZINC000880777145 CD On-Demand Anodyne NQO2 39 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCOCCF)C2 ZINC000880777145 CD On-Demand Anodyne MTNR1A 59 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCOCCF)C2 ZINC000880777145 CD On-Demand Anodyne MTNR1B 50 41 CC[C@@H](NC(=O)Nc1ccccc1C(F)(F)CC)c1ccncc1 ZINC000880777169 EJ On-Demand Anodyne TACR3 40 38 CC[C@@H]1CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777189 CJ On-Demand Anodyne RBP4 79 41 CC[C@@H]1CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777189 CJ On-Demand Anodyne WNT3 40 34 CC[C@H]1CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777190 CJ On-Demand Anodyne RBP4 79 41 CC[C@H]1CCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777190 CJ On-Demand Anodyne WNT3 40 34 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCN1C[C@@H](C)O ZINC000880777279 FG On-Demand Anodyne RBP4 78 41 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCN1C[C@H](C)O ZINC000880777280 FG On-Demand Anodyne RBP4 78 41 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)c1cc(C(F)(F)F)ccn1 ZINC000880777325 GG On-Demand Anodyne GPR119 44 39 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCS1 ZINC000880777430 EJ On-Demand Anodyne RBP4 89 44 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)c1cnc2cc[nH]c2c1 ZINC000880777471 FF On-Demand Anodyne GPR119 46 42 CCN(C)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777488 CH On-Demand Anodyne RBP4 18 45 O=C(NCCOCCF)c1cc2ccccc2cc1F ZINC000880777578 CF On-Demand Anodyne POLR1A 45 31 O=C(CC[C@@H]1CCc2ccccc21)NCCOCCF ZINC000880777627 CF On-Demand Anodyne NQO2 21 44 O=C(CC[C@H]1CCc2ccccc21)NCCOCCF ZINC000880777629 CF On-Demand Anodyne NQO2 21 44 CN(C[C@@H]1CC1(C)C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880777672 DF On-Demand Anodyne MPO 64 35 CC[C@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880777697 CI On-Demand Anodyne RBP4 99 47 CCCN(C)C[C@@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880777729 FI On-Demand Anodyne RBP4 93 42 CCOC[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880777840 EI On-Demand Anodyne RBP4 78 44 CCCN(C)C[C@H]1CCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880777855 FI On-Demand Anodyne RBP4 93 42 CC[C@@H]1COCCN1C(=O)Nc1ccccc1C(F)(F)CC ZINC000880777886 DH On-Demand Anodyne RBP4 60 37 CC(C)(C)OC(=O)N1C[C@@H]2CC[C@H](C1)N2C(=O)c1ncccc1-c1ccccn1 ZINC000880777893 GG On-Demand Anodyne GPR119 27 45 C=CC1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880777906 DJ On-Demand Mild RBP4 95 47 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@@H](C)O1 ZINC000880777957 EI On-Demand Anodyne RBP4 78 42 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)C[C@H](C)O1 ZINC000880777959 EI On-Demand Anodyne RBP4 78 42 CC[C@H](C[C@H](C)CO)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880778008 EI On-Demand Anodyne ANPEP 17 50 CCc1nc([C@H]2CCCN2C(=O)Nc2ccccc2C(F)(F)CC)no1 ZINC000880778106 FJ On-Demand Anodyne CPT1A 42 39 CCc1nc([C@H]2CCCN2C(=O)Nc2ccccc2C(F)(F)CC)no1 ZINC000880778106 FJ On-Demand Anodyne SMO 15 40 O=C(NCCOCCF)c1coc(-c2ccccn2)n1 ZINC000880778174 CD On-Demand Anodyne TBXA2R 19 41 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778225 GF On-Demand Anodyne ABCB1 46 42 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778225 GF On-Demand Anodyne RBP4 66 37 CCc1nnc2n1CCN(C(=O)Nc1ccccc1C(F)(F)CC)C2 ZINC000880778235 EG On-Demand Anodyne P2RX7 28 56 CCc1nnc2n1CCN(C(=O)Nc1ccccc1C(F)(F)CC)C2 ZINC000880778235 EG On-Demand Anodyne RBP4 58 38 O=C(CC[C@H]1CCc2ccccc21)NC[C@@H]1CCCN(CC2CC2)C1 ZINC000880778253 EH On-Demand Anodyne CHRM4 15 54 O=C(CC[C@@H]1CCc2ccccc21)NC[C@@H]1CCCN(CC2CC2)C1 ZINC000880778254 EH On-Demand Anodyne CHRM4 15 54 O=C(CC[C@@H]1CCc2ccccc21)NC[C@H]1CCCN(CC2CC2)C1 ZINC000880778255 EH On-Demand Anodyne CHRM4 15 54 O=C(CC[C@H]1CCc2ccccc21)NC[C@H]1CCCN(CC2CC2)C1 ZINC000880778256 EH On-Demand Anodyne CHRM4 15 54 CC[C@H]1CN(C(=O)Nc2ccccc2C(F)(F)CC)CCO1 ZINC000880778272 DH On-Demand Anodyne RBP4 91 45 C=CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778286 EH On-Demand Mild CCR3 23 40 C=CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778286 EH On-Demand Mild EPHX2 48 43 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1ncsc1C1CC1 ZINC000880778370 DF On-Demand Anodyne CCR3 15 45 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cccc2nsnc12 ZINC000880778373 EF On-Demand Anodyne HTR4 46 41 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cccc2nsnc12 ZINC000880778373 EF On-Demand Anodyne CCR3 23 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCN(CC3CC3)C1)C2 ZINC000880778382 FG On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCN(CC3CC3)C1)C2 ZINC000880778382 FG On-Demand Anodyne SIGMAR1 15 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCN(CC3CC3)C1)C2 ZINC000880778382 FG On-Demand Anodyne EBP 22 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCN(CC3CC3)C1)C2 ZINC000880778383 FG On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCN(CC3CC3)C1)C2 ZINC000880778383 FG On-Demand Anodyne SIGMAR1 15 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCN(CC3CC3)C1)C2 ZINC000880778383 FG On-Demand Anodyne EBP 22 43 O=C(NCCOCCF)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880778397 CD On-Demand Anodyne GABRA1 15 52 O=C(NCCOCCF)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880778397 CD On-Demand Anodyne MPO 61 37 Cn1nnc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)n1 ZINC000880778434 CC On-Demand Anodyne CCR3 55 37 Cn1nnc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)n1 ZINC000880778434 CC On-Demand Anodyne CACNA1I 40 31 Cn1nnc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)n1 ZINC000880778435 CC On-Demand Anodyne CCR3 55 37 Cn1nnc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)n1 ZINC000880778435 CC On-Demand Anodyne CACNA1I 40 31 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778450 GD On-Demand Anodyne F2 43 42 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778450 GD On-Demand Anodyne CHRM4 17 50 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778450 GD On-Demand Anodyne SIGMAR1 22 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778450 GD On-Demand Anodyne CCR3 33 43 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778450 GD On-Demand Anodyne TMPRSS11D 57 35 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778451 GD On-Demand Anodyne F2 43 42 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778451 GD On-Demand Anodyne CHRM4 17 50 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778451 GD On-Demand Anodyne SIGMAR1 22 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778451 GD On-Demand Anodyne CCR3 33 43 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN(CC3CC3)C2)N1Cc1ccccc1 ZINC000880778451 GD On-Demand Anodyne TMPRSS11D 57 35 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cccn2nccc12 ZINC000880778458 DE On-Demand Anodyne HTR4 48 36 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880778607 FH On-Demand Anodyne RBP4 85 44 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880778608 FH On-Demand Anodyne RBP4 85 44 CCOC(=O)N1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778641 FH On-Demand Anodyne P2RY12 46 39 CCOC(=O)N1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778641 FH On-Demand Anodyne KCNQ2 41 31 CCOC(=O)N1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778641 FH On-Demand Anodyne RBP4 77 43 CCCCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778661 GI On-Demand Anodyne RBP4 84 44 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cnc2cc[nH]c2c1 ZINC000880778664 DE On-Demand Anodyne CCR3 38 46 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cnc2cc[nH]c2c1 ZINC000880778664 DE On-Demand Anodyne CACNA1I 57 35 CCCO[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778675 FK On-Demand Anodyne RBP4 79 42 CCCO[C@@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778676 FK On-Demand Anodyne RBP4 79 42 O=C(Cc1ccccc1N1CCCC1=O)NC[C@H]1CCCN(CC2CC2)C1 ZINC000880778683 FF On-Demand Anodyne CHRM4 18 50 O=C(Cc1ccccc1N1CCCC1=O)NC[C@@H]1CCCN(CC2CC2)C1 ZINC000880778684 FF On-Demand Anodyne CHRM4 18 50 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne DRD4 15 45 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne SLC6A1 55 34 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne HTR4 48 36 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne CHRM4 15 46 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne CCR3 96 39 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cc2ccccc2cc1F ZINC000880778715 EH On-Demand Anodyne CACNA1I 48 32 C=C(C)CN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778773 FI On-Demand Mild CCR3 22 40 C=C(C)CN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778773 FI On-Demand Mild EPHX2 45 43 C=C(C)CN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778773 FI On-Demand Mild CXCR3 20 41 O=C(NC[C@H]1CCCN(CC2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880778776 FF On-Demand Anodyne GABRA1 15 45 O=C(NC[C@H]1CCCN(CC2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880778776 FF On-Demand Anodyne CCR3 85 37 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne DRD2 48 42 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne DRD4 28 43 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne DRD3 49 41 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne HTR4 56 42 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne CCR3 26 45 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne HCN1 50 33 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778801 GG On-Demand Anodyne HCN4 48 33 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne DRD2 48 42 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne DRD4 28 43 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne DRD3 49 41 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne HTR4 56 42 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne CCR3 26 45 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne HCN1 50 33 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c(O)n1 ZINC000880778802 GG On-Demand Anodyne HCN4 48 33 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1coc(-c2ccccn2)n1 ZINC000880778857 EF On-Demand Anodyne CCR3 19 46 Cc1cnc(Cl)c(C(=O)NCC2(O)CCC(C)CC2)c1 ZINC000880778881 CF On-Demand Anodyne P2RX7 18 53 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880778886 GI On-Demand Anodyne RBP4 91 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(C)CC1 ZINC000880778892 FD On-Demand Anodyne PAPA1_CARPA 39 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1(O)CCC(C)CC1 ZINC000880778893 FD On-Demand Anodyne PAPA1_CARPA 39 47 CC[C@H]1CCC[C@@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779004 DG On-Demand Anodyne KCNA3 41 35 CC[C@H]1CCC[C@@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779004 DG On-Demand Anodyne TIMP3 51 32 CC[C@H]1CCC[C@@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779004 DG On-Demand Anodyne HCN1 51 32 CC[C@H]1CCC[C@@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779004 DG On-Demand Anodyne HCN4 49 32 CC[C@H]1CCC[C@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779005 DG On-Demand Anodyne KCNA3 41 35 CC[C@H]1CCC[C@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779005 DG On-Demand Anodyne TIMP3 51 32 CC[C@H]1CCC[C@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779005 DG On-Demand Anodyne HCN1 51 32 CC[C@H]1CCC[C@]1(C)C(=O)NC[C@@H](O)c1ccccc1OC ZINC000880779005 DG On-Demand Anodyne HCN4 49 32 O=C(NC[C@H]1CCCN(CC2CC2)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880779015 EG On-Demand Anodyne CCR3 41 38 CCN(CC)C(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779033 GI On-Demand Anodyne RBP4 86 45 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCCN(CC4CC4)C3)cc2)N1 ZINC000880779042 FE On-Demand Anodyne CACNA1I 52 33 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCCN(CC4CC4)C3)cc2)N1 ZINC000880779043 FE On-Demand Anodyne CACNA1I 52 33 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCCN(CC4CC4)C3)cc2)N1 ZINC000880779044 FE On-Demand Anodyne CACNA1I 52 33 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCCN(CC4CC4)C3)cc2)N1 ZINC000880779045 FE On-Demand Anodyne CACNA1I 52 33 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c1 ZINC000880779046 DF On-Demand Anodyne CCR3 35 43 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c1 ZINC000880779046 DF On-Demand Anodyne CACNA1I 71 39 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c1 ZINC000880779047 DF On-Demand Anodyne CCR3 35 43 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c1 ZINC000880779047 DF On-Demand Anodyne CACNA1I 71 39 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1ncccc1-c1ccccn1 ZINC000880779067 FF On-Demand Anodyne CHRM4 15 44 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1ncccc1-c1ccccn1 ZINC000880779067 FF On-Demand Anodyne CCR3 22 46 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1ccc(CN2CCOCC2)o1 ZINC000880779077 FD On-Demand Anodyne CCR3 37 40 Cc1coc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c1 ZINC000880779085 CE On-Demand Anodyne CCR3 59 36 Cc1coc(C(=O)NC[C@@H]2CCCN(CC3CC3)C2)c1 ZINC000880779085 CE On-Demand Anodyne CACNA1I 59 38 Cc1coc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c1 ZINC000880779086 CE On-Demand Anodyne CCR3 59 36 Cc1coc(C(=O)NC[C@H]2CCCN(CC3CC3)C2)c1 ZINC000880779086 CE On-Demand Anodyne CACNA1I 59 38 O=C(NCc1cnccc1C(F)(F)F)c1ccc(CN2CCOCC2)o1 ZINC000880779159 FE On-Demand Anodyne NAMPT 42 43 O=C(C[C@H]1CCNC1=O)NCc1cnccc1C(F)(F)F ZINC000880779163 DD On-Demand Anodyne P2RX7 42 36 O=C(C[C@@H]1CCNC1=O)NCc1cnccc1C(F)(F)F ZINC000880779164 DD On-Demand Anodyne P2RX7 42 36 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)CC2)c(O)n1 ZINC000880779203 FG On-Demand Anodyne KCNA3 51 41 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)CC2)c(O)n1 ZINC000880779203 FG On-Demand Anodyne HCN1 72 37 COc1ccccc1-c1ccc(C(=O)NCC2(O)CCC(C)CC2)c(O)n1 ZINC000880779203 FG On-Demand Anodyne HCN4 52 37 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cnc(CC2CC2)s1 ZINC000880779215 EF On-Demand Anodyne CCR3 41 35 O=C(NC[C@H]1CCCN(CC2CC2)C1)c1cncc2[nH]ccc12 ZINC000880779228 DE On-Demand Anodyne CCR3 51 37 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779262 GJ On-Demand Anodyne EPHX2 55 54 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779262 GJ On-Demand Anodyne RBP4 61 35 CCCCCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779461 GJ On-Demand Anodyne EPHX2 26 43 CCCCCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779461 GJ On-Demand Anodyne RBP4 76 43 CCCCCNC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779461 GJ On-Demand Anodyne ASAH1 63 34 CCN1CC[C@H](CNC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880779518 EH On-Demand Anodyne CCR3 53 48 CCN1CC[C@H](CNC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880779518 EH On-Demand Anodyne RBP4 57 35 CCN1CC[C@H](CNC(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880779518 EH On-Demand Anodyne CACNA1I 62 36 CC(C)CN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880779549 EF On-Demand Anodyne EPHX2 35 41 O=C(Nc1cccc2nccnc12)N1CCC[C@H](C(F)(F)F)C1 ZINC000880779551 DG On-Demand Anodyne RBP4 62 40 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880779552 DG On-Demand Anodyne RBP4 62 40 CC[C@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880779568 CI On-Demand Anodyne ANPEP 18 54 CC[C@H](C)NC(=O)Nc1ccccc1C(F)(F)CC ZINC000880779568 CI On-Demand Anodyne KCNQ2 48 34 CNC(=O)CN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880779572 EC On-Demand Anodyne DRD4 19 45 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880779574 FE On-Demand Anodyne PIK3CA 29 41 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880779574 FE On-Demand Anodyne PIK3CD 20 41 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880779574 FE On-Demand Anodyne MTOR 30 41 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880779574 FE On-Demand Anodyne PIK3CG 20 41 O=C1CC[C@H](c2ccc(C(=O)N3CCC[C@@H]4CCCC[C@@H]43)cc2)N1 ZINC000880779576 EG On-Demand Anodyne PREP 17 40 O=C1CC[C@@H](c2ccc(C(=O)N3CCC[C@@H]4CCCC[C@@H]43)cc2)N1 ZINC000880779577 EG On-Demand Anodyne PREP 17 40 O=C(NCc1ccc(C(=O)N2CCCCC2)cc1)Nc1cccc2nccnc12 ZINC000880779587 GH On-Demand Anodyne NAMPT 33 54 O=C(NCCN1CCc2ccccc2C1)Nc1cccc2nccnc12 ZINC000880779588 EF On-Demand Anodyne UTS2R 18 42 O=C(NCCN1CCc2ccccc2C1)Nc1cccc2nccnc12 ZINC000880779588 EF On-Demand Anodyne ABCB1B 28 41 O=C(NCCN1CCc2ccccc2C1)Nc1cccc2nccnc12 ZINC000880779588 EF On-Demand Anodyne ABCG2 20 41 O=C(NCCN1CCc2ccccc2C1)Nc1cccc2nccnc12 ZINC000880779588 EF On-Demand Anodyne NOD2 40 34 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880779590 GG On-Demand Anodyne RBP4 74 38 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne EGFR 16 40 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne CASR 40 38 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne HRP1_PLAFA 44 37 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne CCR3 24 43 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne UTS2R 15 40 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne HNMT 68 37 O=C(NCCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880779599 DD On-Demand Anodyne EPHX2 28 44 CS(=O)(=O)C1CCC(C(=O)NCc2cnccc2C(F)(F)F)CC1 ZINC000880779611 FE On-Demand Anodyne P2RX7 41 36 O=C(Nc1cccc2nccnc12)N1C2CCC1CC2 ZINC000880779612 CF On-Demand Anodyne WNT3 15 40 CCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880779618 CE On-Demand Anodyne SSTR5 41 32 CCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880779618 CE On-Demand Anodyne EPHX2 40 41 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cccc2nccnc12 ZINC000880779633 GG On-Demand Clean PIK3CA 17 41 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cccc2nccnc12 ZINC000880779633 GG On-Demand Clean MTOR 17 41 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cccc2nccnc12 ZINC000880779633 GG On-Demand Clean EPHB4 62 36 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880779646 FH On-Demand Anodyne RBP4 77 42 C[C@H]1c2ccccc2OCCN1C(=O)C[C@H]1CCNC1=O ZINC000880779701 CD On-Demand Anodyne GHRL 60 35 C[C@H]1c2ccccc2OCCN1C(=O)C[C@@H]1CCNC1=O ZINC000880779702 CD On-Demand Anodyne GHRL 60 35 O=C(Nc1cccc2nccnc12)N1C[C@@H](C(F)(F)F)C[C@@H](C(F)(F)F)C1 ZINC000880779749 GI On-Demand Anodyne RBP4 75 39 O=C(Nc1cccc2nccnc12)N1C[C@H](C(F)(F)F)C[C@@H](C(F)(F)F)C1 ZINC000880779750 GI On-Demand Anodyne RBP4 75 39 O=C(Nc1cccc2nccnc12)N1C[C@@H](C(F)(F)F)C[C@H](C(F)(F)F)C1 ZINC000880779751 GI On-Demand Anodyne RBP4 75 39 O=C(NC1CCCCC1)NC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880779755 GG On-Demand Anodyne EPHX2 44 51 O=C(NCc1ccnc(N2CCCCC2)c1)Nc1cccc2nccnc12 ZINC000880779760 FG On-Demand Anodyne KCNQ2 47 32 O=C(NCc1ccnc(N2CCCCC2)c1)Nc1cccc2nccnc12 ZINC000880779760 FG On-Demand Anodyne HNMT 40 33 CCC(CC)(CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)c1ccc(F)cc1 ZINC000880779771 GG On-Demand Anodyne CACNA1G 51 60 CC(C)(C)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880779785 EG On-Demand Anodyne EPHX2 37 43 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne HTR1A 65 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne DRD2 47 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne ADRA1D 46 38 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne ADRA1A 42 38 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne DRD3 55 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne PDE3A 41 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne HTR7 47 37 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779786 GG On-Demand Anodyne PDE3B 44 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne HTR1A 65 40 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne DRD2 47 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne ADRA1D 46 38 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne ADRA1A 42 38 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne DRD3 55 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne PDE3A 41 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne HTR7 47 37 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880779787 GG On-Demand Anodyne PDE3B 44 41 O=C(CNC(=O)Nc1cccc2nccnc12)NC1CCCCC1 ZINC000880779789 EE On-Demand Anodyne EPHX2 15 44 COc1ccnc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)n1 ZINC000880779792 FD On-Demand Anodyne FAAH 22 40 O=C(Nc1cccc2nccnc12)N1CCn2c(nnc2C2CC2)C1 ZINC000880779797 EE On-Demand Anodyne P2RX7 22 48 COc1ccc([C@@H]2CCN(C(=O)Nc3cccc4nccnc34)C2)cc1 ZINC000880779807 EH On-Demand Anodyne RBP4 42 39 COc1ccc([C@@H]2CCN(C(=O)Nc3cccc4nccnc34)C2)cc1 ZINC000880779807 EH On-Demand Anodyne SMO 29 41 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cccc2nccnc12 ZINC000880779809 FE On-Demand Anodyne HCN1 53 38 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cccc2nccnc12 ZINC000880779809 FE On-Demand Anodyne HCN4 48 31 O=C(Nc1cccc2nccnc12)N1CCN(Cc2cscn2)CC1 ZINC000880779820 FE On-Demand Anodyne FAAH 15 44 O=C(Nc1cccc2nccnc12)N1CCN(Cc2cscn2)CC1 ZINC000880779820 FE On-Demand Anodyne SCN5A 41 33 O=C(Nc1cccc2nccnc12)NC1CCN(c2ccccc2)CC1 ZINC000880779847 EG On-Demand Anodyne EPHX2 31 48 CN(CCN1CCOCC1)C(=O)Nc1cccc2nccnc12 ZINC000880779849 DD On-Demand Anodyne CASR 56 43 CN(CCN1CCOCC1)C(=O)Nc1cccc2nccnc12 ZINC000880779849 DD On-Demand Anodyne EPHX2 17 43 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne TRPV1 17 58 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne PIK3CA 42 46 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne PIK3CD 15 46 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne MTOR 49 46 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne PIK3CG 23 46 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880779945 FE On-Demand Anodyne SCN10A 21 47 COCCCNC(=O)Nc1cccc2nccnc12 ZINC000880779951 CD On-Demand Anodyne HRH2 23 42 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880779965 GG On-Demand Anodyne HPGD 47 42 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880779965 GG On-Demand Anodyne KCNK3 40 37 O=C(Nc1cccc2nccnc12)NC1CCN(C(=O)C2CC2)CC1 ZINC000880779966 EE On-Demand Anodyne EPHX2 42 50 CCCCNC(=O)Nc1ccccc1C(F)(F)CC ZINC000880779968 CI On-Demand Anodyne ASAH1 41 33 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne HRH2 33 46 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne DRD3 42 39 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne HRP1_PLAFA 53 39 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne HRH3 43 48 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne CCR3 30 45 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne CHRNA7 23 52 O=C(NCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880779969 DF On-Demand Anodyne HNMT 117 48 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccco2)CC1 ZINC000880779975 EF On-Demand Anodyne FAAH 15 43 CCOC(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880779976 EE On-Demand Anodyne CCR8 22 42 CCOC(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880779976 EE On-Demand Anodyne PTR1 47 34 O=C(Nc1cccc2nccnc12)N1CCN(C2CCCC2)CC1 ZINC000880779980 EF On-Demand Anodyne HRH3 20 46 O=C(Nc1cccc2nccnc12)N1CCN(C2CCCC2)CC1 ZINC000880779980 EF On-Demand Anodyne L3MBTL3 41 35 C[C@@H](NC(=O)C[C@H]1CCNC1=O)c1ccc2c(c1)CCCO2 ZINC000880780016 DD On-Demand Anodyne GHRL 46 34 C[C@H](NC(=O)C[C@@H]1CCNC1=O)c1ccc2c(c1)CCCO2 ZINC000880780018 DD On-Demand Anodyne GHRL 46 34 C[C@@H](NC(=O)C[C@@H]1CCNC1=O)c1ccc2c(c1)CCCO2 ZINC000880780019 DD On-Demand Anodyne GHRL 46 34 O=C(NCc1ccnc(N2CCCC2)c1)Nc1cccc2nccnc12 ZINC000880780020 EF On-Demand Anodyne KCNQ2 50 33 C[C@H](NC(=O)C[C@H]1CCNC1=O)c1ccc2c(c1)CCCO2 ZINC000880780021 DD On-Demand Anodyne GHRL 46 34 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cnccc1C(F)(F)F)C2 ZINC000880780036 FH On-Demand Anodyne NQO2 26 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cnccc1C(F)(F)F)C2 ZINC000880780036 FH On-Demand Anodyne RAF1 15 44 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)N3CC4CC3(C)C4)ccn2)CC1 ZINC000880780047 GF On-Demand Anodyne GPR119 38 46 O=C(NC1CCN(C(=O)Nc2cccc3nccnc23)CC1)C1CC1 ZINC000880780054 EE On-Demand Anodyne EPHX2 35 42 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000880780064 DH On-Demand Anodyne CPT1A 46 39 O=C(CN1CCN(C(=O)Nc2cccc3nccnc23)CC1)N1CCCCC1 ZINC000880780085 GD On-Demand Anodyne HNMT 40 34 O=C(Cc1ccccc1N1CCCC1=O)NCc1cnccc1C(F)(F)F ZINC000880780101 GG On-Demand Anodyne P2RX7 47 39 Cn1ncc(Br)c1CC(=O)NCc1cnccc1C(F)(F)F ZINC000880780102 GE On-Demand Anodyne P2RX7 37 53 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HTR1A 67 53 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne DRD2 56 44 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne DRD4 34 44 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne ADRA1D 25 40 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HTR2A 49 48 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HTR2C 34 48 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne ADRA1A 28 40 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne DRD3 73 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HRP1_PLAFA 53 38 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HTR7 54 44 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne CCR3 23 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cccc2nccnc12 ZINC000880780109 GD On-Demand Anodyne HNMT 60 36 CCOC(=O)CC1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780126 FI On-Demand Anodyne RBP4 82 45 Cc1cc([C@@H]2CCCN2C(=O)Nc2cccc3nccnc23)no1 ZINC000880780129 DG On-Demand Anodyne CPT1A 44 41 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880780142 FG On-Demand Anodyne ABCB1B 71 42 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880780142 FG On-Demand Anodyne ABCB1 28 45 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880780142 FG On-Demand Anodyne ABCG2 43 42 O=C(NCc1ccccc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880780144 EH On-Demand Anodyne KCNQ2 83 46 O=C(NCc1ccccc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880780144 EH On-Demand Anodyne SCN2A 18 42 O=C(NCc1ccccc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880780144 EH On-Demand Anodyne SCN10A 15 42 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cccc2nccnc12 ZINC000880780149 EI On-Demand Anodyne TRPM8 16 53 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cccc2nccnc12 ZINC000880780150 EI On-Demand Anodyne TRPM8 16 53 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780153 GG On-Demand Anodyne EPHX2 34 51 Cn1cc(CN2CCN(C(=O)Nc3cccc4nccnc34)CC2)cn1 ZINC000880780155 FD On-Demand Anodyne FAAH 27 44 COc1ccc(N2CCC(NC(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880780157 GG On-Demand Clean EPHX2 31 44 O=C(Nc1cccc2nccnc12)N1CCC[C@H](N2CCCC2)C1 ZINC000880780164 EF On-Demand Anodyne L3MBTL3 64 39 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](N2CCCC2)C1 ZINC000880780165 EF On-Demand Anodyne L3MBTL3 64 39 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cccc2nccnc12 ZINC000880780166 FF On-Demand Clean PIK3CA 25 44 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cccc2nccnc12 ZINC000880780166 FF On-Demand Clean MTOR 31 44 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cccc2nccnc12 ZINC000880780166 FF On-Demand Clean PIK3CG 17 44 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cccc2nccnc12 ZINC000880780166 FF On-Demand Clean STAT6 60 36 O=C(Nc1cccc2nccnc12)N1CCCO[C@@H](c2ccccc2)C1 ZINC000880780175 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cccc2nccnc12)N1CCCO[C@H](c2ccccc2)C1 ZINC000880780176 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne DRD4 25 57 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne SIGMAR1 24 57 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne SSTR5 59 36 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne CCR3 39 40 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne EPHX2 28 42 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne CXCR3 21 41 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccncc2)CC1 ZINC000880780177 FF On-Demand Anodyne MCHR1 43 41 O=C(NC[C@H](O)C1CCCCC1)Nc1cccc2nccnc12 ZINC000880780181 DF On-Demand Anodyne PRMT3 26 48 O=C(NC[C@@H](O)C1CCCCC1)Nc1cccc2nccnc12 ZINC000880780182 DF On-Demand Anodyne PRMT3 26 48 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccccn2)CC1 ZINC000880780194 FF On-Demand Anodyne SIGMAR1 15 51 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccccn2)CC1 ZINC000880780194 FF On-Demand Anodyne CCR3 22 40 O=C(Nc1cccc2nccnc12)NC1CCN(Cc2ccccn2)CC1 ZINC000880780194 FF On-Demand Anodyne EPHX2 26 42 O=C(NC1CCN(C(=O)Nc2cccc3nccnc23)CC1)C1CCCCC1 ZINC000880780203 GG On-Demand Anodyne EPHX2 33 47 O=C(Nc1cccc2nccnc12)N1CCN2CCCC[C@@H]2C1 ZINC000880780205 DE On-Demand Anodyne HRH3 17 40 O=C(Nc1cccc2nccnc12)N1CCN2CCCC[C@@H]2C1 ZINC000880780205 DE On-Demand Anodyne L3MBTL3 55 38 O=C(Nc1cccc2nccnc12)N1CCN2CCCC[C@H]2C1 ZINC000880780206 DE On-Demand Anodyne HRH3 17 40 O=C(Nc1cccc2nccnc12)N1CCN2CCCC[C@H]2C1 ZINC000880780206 DE On-Demand Anodyne L3MBTL3 55 38 CCC(CC)(CNC(=O)C1CCC(S(C)(=O)=O)CC1)c1ccc(F)cc1 ZINC000880780209 GH On-Demand Anodyne CACNA1G 54 63 CCOC(=O)N1CCCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780211 EE On-Demand Anodyne P2RY12 43 42 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780215 GG On-Demand Anodyne ACACB 16 43 N#CCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780217 DD On-Demand Mild EPHX2 30 42 O=C(Nc1cccc2nccnc12)N1CCCN(c2ccccc2)CC1 ZINC000880780229 EG On-Demand Anodyne PDGFRB 21 42 O=C(Nc1cccc2nccnc12)N1CCCN(c2ccccc2)CC1 ZINC000880780229 EG On-Demand Anodyne FAAH 18 45 Cc1noc(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)n1 ZINC000880780230 EF On-Demand Anodyne SMO 49 55 Cc1noc(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)n1 ZINC000880780230 EF On-Demand Anodyne ETHR 62 36 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880780238 EI On-Demand Anodyne HCRTR1 25 41 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880780238 EI On-Demand Anodyne HCRTR2 22 41 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880780239 EI On-Demand Anodyne HCRTR1 25 41 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880780239 EI On-Demand Anodyne HCRTR2 22 41 CCOC(=O)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780299 FG On-Demand Anodyne P2RY12 53 41 CCOC(=O)N1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780299 FG On-Demand Anodyne RBP4 84 42 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccncc2)CC1 ZINC000880780349 EE On-Demand Anodyne FAAH 34 49 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne DRD4 18 45 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne CHRM3 20 41 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne SIGMAR1 15 48 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne CCR3 31 43 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne EPHX2 56 46 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne CXCR3 21 42 CCN1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780369 EH On-Demand Anodyne RBP4 57 34 O=C(Nc1cccc2nccnc12)N1CCN(Cc2cccnc2)CC1 ZINC000880780373 EE On-Demand Anodyne FAAH 36 49 O=C(NCc1cnccc1C(F)(F)F)[C@H]1CCc2nncn2CC1 ZINC000880780391 ED On-Demand Anodyne P2RX7 40 38 O=C(NCc1cnccc1C(F)(F)F)[C@H]1CCc2nncn2CC1 ZINC000880780391 ED On-Demand Anodyne EPHX2 15 45 O=C(NCc1cnccc1C(F)(F)F)[C@@H]1CCc2nncn2CC1 ZINC000880780394 ED On-Demand Anodyne P2RX7 40 38 O=C(NCc1cnccc1C(F)(F)F)[C@@H]1CCc2nncn2CC1 ZINC000880780394 ED On-Demand Anodyne EPHX2 15 45 CCC(=O)N1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880780395 FH On-Demand Anodyne RBP4 79 44 CCCN(CC1CC1)C(=O)Nc1ccccc1C(F)(F)CC ZINC000880780425 DJ On-Demand Anodyne RBP4 53 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000880780437 FG On-Demand Anodyne PLG 16 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000880780437 FG On-Demand Anodyne CELA1 40 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000880780438 FG On-Demand Anodyne PLG 16 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000880780438 FG On-Demand Anodyne CELA1 40 41 O=C(NCc1ccccc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880780451 FF On-Demand Anodyne KCNQ2 62 37 O=C(NCc1ccccc1N1CCOCC1)Nc1cccc2nccnc12 ZINC000880780451 FF On-Demand Anodyne SCN10A 15 45 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780453 FG On-Demand Anodyne ACACB 17 44 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780454 FG On-Demand Anodyne ACACB 17 44 O=C(CCCNC(=O)Nc1cccc2nccnc12)NC1CC1 ZINC000880780461 DD On-Demand Anodyne TNKS 46 33 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880780462 EE On-Demand Anodyne CCR3 17 41 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880780462 EE On-Demand Anodyne EPHX2 30 42 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880780462 EE On-Demand Anodyne HPGDS 38 42 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880780463 EE On-Demand Anodyne CCR3 17 41 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880780463 EE On-Demand Anodyne EPHX2 30 42 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880780463 EE On-Demand Anodyne HPGDS 38 42 C[C@@H](CNC(=O)Nc1cccc2nccnc12)N1CCCCC1 ZINC000880780467 DF On-Demand Anodyne KCNQ2 41 32 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cccc2nccnc12 ZINC000880780468 GF On-Demand Anodyne DRD4 16 42 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cccc2nccnc12 ZINC000880780468 GF On-Demand Anodyne SIGMAR1 20 44 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cccc2nccnc12 ZINC000880780468 GF On-Demand Anodyne CCR3 41 37 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cccc2nccnc12 ZINC000880780468 GF On-Demand Anodyne MCHR1 22 40 O=C(Nc1cccc2nccnc12)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880780474 GF On-Demand Anodyne EPHX2 45 56 O=C(Nc1cccc2nccnc12)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880780474 GF On-Demand Anodyne CCR8 41 34 O=C(Nc1cccc2nccnc12)N1CCN(CC(F)F)CC1 ZINC000880780476 DE On-Demand Anodyne FAAH 18 40 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne ACE 42 44 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne OPRM1 21 46 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne MME 61 44 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne MC4R 48 37 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne TRY2_BOVIN 60 36 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne CACNA1B 19 41 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne F2R 40 31 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne PREP 17 54 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne ACE2 66 34 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne BLA1_STEMA 40 36 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne PSMB8 40 34 O=C(Nc1cccc2nccnc12)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780477 GF On-Demand Anodyne GPR142 73 33 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne ACE 42 44 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne OPRM1 21 46 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne MME 61 44 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne MC4R 48 37 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne TRY2_BOVIN 60 36 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne CACNA1B 19 41 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne F2R 40 31 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne PREP 17 54 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne ACE2 66 34 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne BLA1_STEMA 40 36 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne PSMB8 40 34 O=C(Nc1cccc2nccnc12)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880780478 GF On-Demand Anodyne GPR142 73 33 CCC(CC)(CNC(=O)C[C@H]1CCNC1=O)c1ccc(F)cc1 ZINC000880780485 DF On-Demand Anodyne CACNA1G 41 48 CCC(CC)(CNC(=O)C[C@@H]1CCNC1=O)c1ccc(F)cc1 ZINC000880780486 DF On-Demand Anodyne CACNA1G 41 48 O=C(NCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780511 CE On-Demand Anodyne HRH2 28 43 O=C(NCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780511 CE On-Demand Anodyne HRH3 21 46 O=C(NCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780511 CE On-Demand Anodyne CHRNA7 15 46 O=C(NCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780511 CE On-Demand Anodyne UTS2R 19 44 O=C(NCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780511 CE On-Demand Anodyne HNMT 109 46 C[C@H]1C[C@H]1NC(=O)Nc1cccc2nccnc12 ZINC000880780516 BE On-Demand Anodyne TRPV1 15 46 C[C@@H]1C[C@@H]1NC(=O)Nc1cccc2nccnc12 ZINC000880780517 BE On-Demand Anodyne TRPV1 15 46 C[C@@H]1C[C@H]1NC(=O)Nc1cccc2nccnc12 ZINC000880780519 BE On-Demand Anodyne TRPV1 15 46 O=C(Nc1cccc2nccnc12)N1CCN(CC2CC2)CC1 ZINC000880780522 DE On-Demand Anodyne FAAH 15 44 O=C(Nc1cccc2nccnc12)N1CCN(CCCOCC(F)(F)F)CC1 ZINC000880780535 GF On-Demand Anodyne HNMT 42 36 O=C(Nc1cccc2nccnc12)N1CCN(CCCOCC(F)(F)F)CC1 ZINC000880780535 GF On-Demand Anodyne RBP4 40 35 CCN1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880780536 CE On-Demand Anodyne CCR3 46 36 CCN1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880780536 CE On-Demand Anodyne CACNA1I 46 32 CC(C)(C)OC(=O)NC[C@@H]1CCCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780542 GG On-Demand Anodyne ACACB 16 42 CC(C)(C)OC(=O)NC[C@H]1CCCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780543 GG On-Demand Anodyne ACACB 16 42 CCO[C@H]1CCCN(C(=O)Nc2ccccc2C(F)(F)CC)C1 ZINC000880780544 EI On-Demand Anodyne RBP4 96 48 O=C(Nc1cccc2nccnc12)N1CCC(O)CC1 ZINC000880780595 CD On-Demand Anodyne RBP4 40 39 O=C(Nc1cccc2nccnc12)N[C@@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000880780607 EH On-Demand Anodyne EPHX2 15 47 O=C(Nc1cccc2nccnc12)N[C@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000880780609 EH On-Demand Anodyne EPHX2 15 47 O=C(Nc1cccc2nccnc12)N[C@H]1CCC[C@H](C(F)(F)F)C1 ZINC000880780612 EH On-Demand Anodyne EPHX2 15 47 O=C(Nc1cccc2nccnc12)N[C@@H]1CCC[C@H](C(F)(F)F)C1 ZINC000880780614 EH On-Demand Anodyne EPHX2 15 47 CCOC(=O)N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780632 ED On-Demand Anodyne P2RY12 55 43 CCOC(=O)N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780632 ED On-Demand Anodyne FAAH 15 49 CCOC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780640 EE On-Demand Anodyne GRIN2B 22 40 CCOC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780640 EE On-Demand Anodyne SSTR5 42 33 CCOC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780640 EE On-Demand Anodyne EPHX2 48 44 CCOC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780640 EE On-Demand Anodyne CCR8 66 45 CCCCCNC(=O)Nc1cccc2nccnc12 ZINC000880780654 CF On-Demand Anodyne ASAH1 57 32 COc1cc(C)c(CN(C)C(=O)Nc2cccc3nccnc23)cc1OC ZINC000880780681 FH On-Demand Anodyne KDR 50 37 COc1cc(C)c(CN(C)C(=O)Nc2cccc3nccnc23)cc1OC ZINC000880780681 FH On-Demand Anodyne PDGFRA 52 40 CC(=O)NCCCNC(=O)Nc1cccc2nccnc12 ZINC000880780685 CD On-Demand Anodyne MTNR1A 48 45 CC(=O)NCCCNC(=O)Nc1cccc2nccnc12 ZINC000880780685 CD On-Demand Anodyne MTNR1B 46 45 CCn1cc(NC(=O)Nc2ccccc2C(F)(F)CC)cn1 ZINC000880780724 DI On-Demand Anodyne P2RY1 58 36 CCn1cc(NC(=O)Nc2ccccc2C(F)(F)CC)cn1 ZINC000880780724 DI On-Demand Anodyne MAPK10 15 40 CCn1cc(NC(=O)Nc2ccccc2C(F)(F)CC)cn1 ZINC000880780724 DI On-Demand Anodyne PANC 50 33 COc1ccc([C@@H]2CCCN2C(=O)Nc2cccc3nccnc23)c(OC)c1 ZINC000880780725 GI On-Demand Anodyne PDGFRA 46 36 O=C(Nc1cccc2nccnc12)N1CCN(CC(F)(F)F)CC1 ZINC000880780737 EE On-Demand Anodyne FAAH 18 40 O=C(Nc1cccc2nccnc12)N1CCN(CC(F)(F)F)CC1 ZINC000880780737 EE On-Demand Anodyne RBP4 47 36 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne HTR1A 28 41 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne DRD2 30 41 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne HRH2 37 45 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne DRD3 57 41 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne HRH3 40 51 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne CCR3 24 42 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne CHRNA7 22 53 O=C(NCCCCCN1CCCCC1)Nc1cccc2nccnc12 ZINC000880780753 EG On-Demand Anodyne HNMT 119 51 CCOCCN1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780758 ED On-Demand Anodyne HNMT 45 33 Cc1nc(CN2CCN(C(=O)Nc3cccc4nccnc34)CC2)oc1C ZINC000880780763 FF On-Demand Anodyne FAAH 17 43 CN(C)[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780766 CD On-Demand Anodyne RBP4 54 37 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780768 FG On-Demand Anodyne EPHX2 41 45 CCc1nc(CN2CCN(C(=O)Nc3cccc4nccnc34)CC2)cs1 ZINC000880780771 GF On-Demand Anodyne FAAH 16 42 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780783 FG On-Demand Anodyne EPHX2 46 42 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780783 FG On-Demand Anodyne CCR8 33 43 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780783 FG On-Demand Anodyne GPR119 46 45 O=C(NCCCCn1ccnc1)Nc1cccc2nccnc12 ZINC000880780792 DE On-Demand Anodyne TBXAS1 50 47 O=C(NCCCCn1ccnc1)Nc1cccc2nccnc12 ZINC000880780792 DE On-Demand Anodyne HMOX2 49 40 O=C(NCCCCn1ccnc1)Nc1cccc2nccnc12 ZINC000880780792 DE On-Demand Anodyne QPCT 45 49 C[C@H]1CN(c2ccc(CNC(=O)Nc3cccc4nccnc34)cn2)C[C@@H](C)O1 ZINC000880780804 GF On-Demand Anodyne NAMPT 26 43 C[C@H]1CN(c2ccc(CNC(=O)Nc3cccc4nccnc34)cn2)C[C@H](C)O1 ZINC000880780805 GF On-Demand Anodyne NAMPT 26 43 COC(=O)C1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780809 EE On-Demand Anodyne EPHX2 27 41 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cccc2nccnc12 ZINC000880780819 FF On-Demand Anodyne CCR3 37 40 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cccc2nccnc12 ZINC000880780820 FF On-Demand Anodyne CCR3 37 40 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne HTR1A 79 42 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne DRD2 63 55 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne DRD4 38 44 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne ADRA1D 69 55 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne HTR1B 20 42 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne ADRA1A 61 55 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne ADRA1B 53 55 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne DRD3 66 42 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne HTR7 54 38 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne KCNQ2 55 34 COc1ccccc1N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880780823 GG On-Demand Anodyne PDGFRA 38 40 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](C2OCCO2)C1 ZINC000880780826 EE On-Demand Anodyne RBP4 52 32 O=C(Nc1cccc2nccnc12)N1CCC[C@H](C2OCCO2)C1 ZINC000880780827 EE On-Demand Anodyne RBP4 52 32 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780852 CF On-Demand Anodyne RBP4 47 36 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880780853 CF On-Demand Anodyne RBP4 47 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780882 GF On-Demand Anodyne PAPA1_CARPA 39 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780882 GF On-Demand Anodyne SCN10A 26 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780882 GF On-Demand Anodyne FPR1 40 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780883 GF On-Demand Anodyne PAPA1_CARPA 39 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780883 GF On-Demand Anodyne SCN10A 26 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cnccc1C(F)(F)F ZINC000880780883 GF On-Demand Anodyne FPR1 40 35 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cccc2nccnc12 ZINC000880780911 FH On-Demand Anodyne ROCK2 24 42 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cccc2nccnc12 ZINC000880780911 FH On-Demand Anodyne ENPP1 44 31 O=C(NCCCN1CCCC1=O)Nc1cccc2nccnc12 ZINC000880780913 DD On-Demand Anodyne TYRO3 20 41 O=C(Nc1cccc2nccnc12)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880780921 FH On-Demand Anodyne RBP4 52 38 O=C(Nc1cccc2nccnc12)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880780922 FH On-Demand Anodyne RBP4 52 38 O=C(Nc1cccc2nccnc12)N1CCC(OCc2ccccc2)CC1 ZINC000880780948 FH On-Demand Anodyne GRIN2B 46 44 O=C(Nc1cccc2nccnc12)N1CCC(OCc2ccccc2)CC1 ZINC000880780948 FH On-Demand Anodyne RBP4 55 42 Cn1cc(CN2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cn1 ZINC000880780961 FE On-Demand Anodyne FAAH 24 42 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780971 GG On-Demand Anodyne EPHX2 30 43 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880780971 GG On-Demand Anodyne SCD 15 41 O=C(CN1CCN(C(=O)Nc2cccc3nccnc23)CC1)N1CCCCCC1 ZINC000880780976 GE On-Demand Anodyne HNMT 40 34 O=C(NCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880780983 DD On-Demand Anodyne CASR 40 39 O=C(NCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880780983 DD On-Demand Anodyne UTS2R 18 45 O=C(NCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880780983 DD On-Demand Anodyne EPHX2 24 46 O=C(NCCN1CCOCC1)Nc1cccc2nccnc12 ZINC000880780983 DD On-Demand Anodyne HPGDS 24 43 CC[C@@H](O)CN1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781001 ED On-Demand Anodyne ACOX1 51 37 CC[C@H](O)CN1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781002 ED On-Demand Anodyne ACOX1 51 37 O=C(Nc1cccc2nccnc12)NC1CC1 ZINC000880781003 BD On-Demand Anodyne TRPV1 15 46 O=C(Nc1cccc2nccnc12)NC1CC1 ZINC000880781003 BD On-Demand Anodyne EPHX2 33 49 O=C(Nc1cccc2nccnc12)N1CCC[C@H](Oc2ccccc2)C1 ZINC000880781014 EH On-Demand Anodyne RBP4 46 33 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](Oc2ccccc2)C1 ZINC000880781016 EH On-Demand Anodyne RBP4 46 33 N#Cc1ccc(CN2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781032 GG On-Demand Mild FAAH 24 44 O=C(Nc1cccc2nccnc12)N1CC[C@H](COCc2ccccc2)C1 ZINC000880781051 FH On-Demand Anodyne GRIN2B 53 42 O=C(Nc1cccc2nccnc12)N1CC[C@H](COCc2ccccc2)C1 ZINC000880781051 FH On-Demand Anodyne RBP4 52 36 CCOC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781052 FH On-Demand Anodyne PDE6D 50 33 CCOC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781052 FH On-Demand Anodyne RBP4 87 47 CCOC(=O)C1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781052 FH On-Demand Anodyne CCR8 23 42 O=C(Nc1cccc2nccnc12)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880781054 FH On-Demand Anodyne GRIN2B 53 42 O=C(Nc1cccc2nccnc12)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880781054 FH On-Demand Anodyne RBP4 52 36 COc1ccccc1[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781057 EH On-Demand Anodyne RBP4 68 45 COc1ccccc1[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781057 EH On-Demand Anodyne SMO 30 46 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781058 EH On-Demand Anodyne RBP4 68 45 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781058 EH On-Demand Anodyne SMO 30 46 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880781061 GF On-Demand Anodyne DRD4 27 47 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880781061 GF On-Demand Anodyne SIGMAR1 23 47 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880781062 GF On-Demand Anodyne DRD4 27 47 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880781062 GF On-Demand Anodyne SIGMAR1 23 47 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880781064 GF On-Demand Anodyne DRD4 27 47 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880781064 GF On-Demand Anodyne SIGMAR1 23 47 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880781065 GF On-Demand Anodyne DRD4 27 47 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880781065 GF On-Demand Anodyne SIGMAR1 23 47 CCOC[C@H](O)CN1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781068 FD On-Demand Anodyne ACOX1 55 40 CCOC[C@H](O)CN1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781068 FD On-Demand Anodyne ABCB1 45 42 CCNC(=O)CN1CCN(C(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781081 FE On-Demand Anodyne RBP4 72 40 O=C(Nc1cccc2nccnc12)NC1CCN(CC(F)F)CC1 ZINC000880781092 EE On-Demand Anodyne EPHX2 36 43 O=C(NCC(F)(F)F)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781096 GF On-Demand Anodyne RBP4 49 39 CN1CCN(c2ncccc2CNC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781100 GE On-Demand Anodyne TRPV1 22 60 CN(C1CCN(C(=O)Nc2cccc3nccnc23)CC1)S(C)(=O)=O ZINC000880781108 FD On-Demand Anodyne RBP4 41 41 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](OCC(F)(F)F)C1 ZINC000880781111 FG On-Demand Anodyne RBP4 57 38 O=C(Nc1cccc2nccnc12)N1CCC[C@H](OCC(F)(F)F)C1 ZINC000880781112 FG On-Demand Anodyne RBP4 57 38 CCC(CC)(CNC(=O)c1cn(C[C@@H]2CNC(=O)O2)nn1)c1ccc(F)cc1 ZINC000880781113 GE On-Demand Anodyne CACNA1G 36 42 CCC(CC)(CNC(=O)c1cn(C[C@H]2CNC(=O)O2)nn1)c1ccc(F)cc1 ZINC000880781115 GE On-Demand Anodyne CACNA1G 36 42 COc1ccc(CN(CCO)C(=O)Nc2cccc3nccnc23)c(OC)c1 ZINC000880781116 GF On-Demand Anodyne ROCK2 29 46 COc1ccc(CN(CCO)C(=O)Nc2cccc3nccnc23)c(OC)c1 ZINC000880781116 GF On-Demand Anodyne PDGFRA 41 37 O=C(Nc1cccc2nccnc12)N1CCC(Oc2ccc(F)cc2F)CC1 ZINC000880781123 GH On-Demand Anodyne SCD1 40 47 O=C(Nc1cccc2nccnc12)N1CCC(Oc2ccc(F)cc2F)CC1 ZINC000880781123 GH On-Demand Anodyne SCD 35 40 C[C@@H]1CCCCN1CCNC(=O)Nc1cccc2nccnc12 ZINC000880781127 DF On-Demand Anodyne HRH3 42 38 C[C@H]1CCCCN1CCNC(=O)Nc1cccc2nccnc12 ZINC000880781129 DF On-Demand Anodyne HRH3 42 38 O=C(NCCCN1CCCCC1=O)Nc1cccc2nccnc12 ZINC000880781135 EE On-Demand Anodyne TYRO3 19 40 CC(C)(C)NC(=O)CCNC(=O)Nc1cccc2nccnc12 ZINC000880781158 DE On-Demand Anodyne TRPV1 15 44 O=C(Nc1cccc2nccnc12)NC1CCC1 ZINC000880781163 BE On-Demand Anodyne EPHX2 25 51 O=C(Nc1cccc2nccnc12)N1CC[C@H](N2CCCCC2)C1 ZINC000880781164 EF On-Demand Anodyne L3MBTL3 91 43 O=C(Nc1cccc2nccnc12)N1CC[C@@H](N2CCCCC2)C1 ZINC000880781166 EF On-Demand Anodyne L3MBTL3 91 43 Cc1nc(CN2CCN(C(=O)Nc3cccc4nccnc34)CC2)cs1 ZINC000880781171 FF On-Demand Anodyne FAAH 17 44 COC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781204 ED On-Demand Anodyne EPHX2 46 43 CCc1nnc2n1CCN(C(=O)Nc1cccc3nccnc13)C2 ZINC000880781205 DD On-Demand Anodyne P2RX7 24 48 C[C@@H](CNC(=O)Nc1cccc2nccnc12)CN1CCCCC1 ZINC000880781206 EF On-Demand Anodyne HNMT 46 34 O=C(Nc1cccc2nccnc12)N(CCO)CCN1CCOCC1 ZINC000880781249 EC On-Demand Anodyne CASR 66 51 O=C(Nc1cccc2nccnc12)N(CCO)CCN1CCOCC1 ZINC000880781249 EC On-Demand Anodyne PRKDC 45 35 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cccc3nccnc13)C2 ZINC000880781255 EF On-Demand Anodyne HTR3A 39 47 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cccc3nccnc13)C2 ZINC000880781255 EF On-Demand Anodyne GLRA1 43 35 CCCCCN(CCO)C(=O)Nc1cccc2nccnc12 ZINC000880781269 DF On-Demand Anodyne SOAT1 29 40 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cccc2nccnc12 ZINC000880781286 GF On-Demand Anodyne EPHX2 17 46 COCCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781331 ED On-Demand Anodyne DRD4 20 44 COCCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781331 ED On-Demand Anodyne LTA4H 17 42 COCCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781331 ED On-Demand Anodyne CCR3 29 44 COCCN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781331 ED On-Demand Anodyne EPHX2 41 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781336 FF On-Demand Clean PDGFRB 51 42 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781336 FF On-Demand Clean CCKAR 25 42 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781336 FF On-Demand Clean FAAH 22 42 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781336 FF On-Demand Clean RBP4 24 41 COCCCCN(Cc1ccccc1)C(=O)Nc1cccc2nccnc12 ZINC000880781337 FI On-Demand Anodyne ROCK2 17 41 O=C(Nc1cccc2nccnc12)NC1CCN(C2CC2)CC1 ZINC000880781338 DE On-Demand Anodyne EPHX2 32 42 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cccc2nccnc12 ZINC000880781348 EF On-Demand Anodyne KCNQ2 42 33 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cccc2nccnc12 ZINC000880781348 EF On-Demand Anodyne NAMPT 45 41 O=C(Nc1cccc2nccnc12)N1CCC(OCCc2ccccc2)CC1 ZINC000880781364 GH On-Demand Anodyne GRIN2B 27 42 O=C(Nc1cccc2nccnc12)N1CCN(Cc2cccs2)CC1 ZINC000880781365 FG On-Demand Anodyne FAAH 18 43 CCC(CC)(CNC(=O)c1nnn(C)n1)c1ccc(F)cc1 ZINC000880781369 DD On-Demand Anodyne CACNA1G 42 48 Cc1cc([C@@H]2CCCN2C(=O)Nc2cccc3nccnc23)on1 ZINC000880781389 DG On-Demand Anodyne KCNA5 15 44 COc1ccc(OC2CCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781394 GH On-Demand Anodyne EPHX2 22 50 O=C(Nc1cccc2nccnc12)NC1CCN(CC(F)(F)F)CC1 ZINC000880781396 FF On-Demand Anodyne EPHX2 40 46 O=C(Nc1cccc2nccnc12)NC1CCN(CC(F)(F)F)CC1 ZINC000880781396 FF On-Demand Anodyne HPGDS 43 47 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccccc2)CC1 ZINC000880781399 EF On-Demand Anodyne DRD2 16 43 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccccc2)CC1 ZINC000880781399 EF On-Demand Anodyne PDGFRB 17 40 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccccc2)CC1 ZINC000880781399 EF On-Demand Anodyne SIGMAR1 38 41 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccccc2)CC1 ZINC000880781399 EF On-Demand Anodyne FAAH 45 53 O=C(NCCCN1CCCCCC1=O)Nc1cccc2nccnc12 ZINC000880781404 EF On-Demand Anodyne HNMT 60 35 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne HTR1A 96 54 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne DRD2 70 46 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne DRD1 19 41 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne DRD4 40 45 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne ADRA1D 72 43 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne HTR1D 22 54 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne HTR1B 28 54 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne HTR2A 24 43 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne ADRA1A 67 42 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne ADRA1B 56 42 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne DRD3 77 46 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne PDGFRB 66 51 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne HTR7 62 47 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne KCNQ2 55 34 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne PDGFRA 31 43 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne RBP4 36 52 COc1ccccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781406 FF On-Demand Anodyne SMO 20 41 O=C(Nc1cccc2nccnc12)NC1CCN(CC2CC2)CC1 ZINC000880781423 EF On-Demand Anodyne SIGMAR1 19 47 O=C(Nc1cccc2nccnc12)NC1CCN(CC2CC2)CC1 ZINC000880781423 EF On-Demand Anodyne EPHX2 34 40 O=C(Nc1cccc2nccnc12)NC1CCN(CC2CC2)CC1 ZINC000880781423 EF On-Demand Anodyne CXCR3 15 43 Cn1cnnc1C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781426 EE On-Demand Anodyne SMO 18 42 CCOC(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781428 FH On-Demand Anodyne EPHX2 67 45 CCOC(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781428 FH On-Demand Anodyne CXCR3 15 42 CCOC(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781428 FH On-Demand Anodyne RBP4 70 38 CCOC(=O)N1CCC(NC(=O)Nc2ccccc2C(F)(F)CC)CC1 ZINC000880781428 FH On-Demand Anodyne CCR8 67 44 CN1CCC(CNC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781435 CE On-Demand Anodyne HTR1F 54 37 CN1CCC(CNC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781435 CE On-Demand Anodyne CACNA1I 47 34 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cccc2nccnc12 ZINC000880781437 GG On-Demand Anodyne BMP1 51 35 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HTR1A 69 45 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne DRD2 53 43 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne DRD4 32 40 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne ADRA1D 26 41 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HTR2A 54 45 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HTR2C 36 43 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne ADRA1A 29 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne DRD3 77 45 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HRP1_PLAFA 44 37 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HTR7 73 39 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne CCR3 27 41 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880781453 GE On-Demand Anodyne HNMT 62 35 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781463 FF On-Demand Anodyne EPHX2 44 44 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1cccc2nccnc12 ZINC000880781466 DF On-Demand Anodyne TRPV1 20 44 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne PDGFRB 52 41 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne KDR 53 37 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne ABCB1B 63 40 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne ABCB1 23 41 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne PDGFRA 43 38 COc1cc2c(cc1OC)CCN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781467 GG On-Demand Anodyne RBP4 27 41 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1cccc2nccnc12 ZINC000880781468 DF On-Demand Anodyne TRPV1 20 44 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne CHRM2 15 43 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne DRD4 44 59 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne CHRM3 21 43 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne LTA4H 20 41 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne SIGMAR1 35 59 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne SSTR5 47 34 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne CCR3 50 49 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne CCR2 15 43 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne EPHX2 15 44 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne MCHR1 31 50 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880781482 EG On-Demand Anodyne BIRC2 27 42 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne CHRM2 15 43 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne DRD4 44 59 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne CHRM3 21 43 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne LTA4H 20 41 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne SIGMAR1 35 59 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne SSTR5 47 34 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne CCR3 50 49 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne CCR2 15 43 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne EPHX2 15 44 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne MCHR1 31 50 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880781484 EG On-Demand Anodyne BIRC2 27 42 O=C(NC[C@@H](O)C(F)(F)F)Nc1cccc2nccnc12 ZINC000880781487 DD On-Demand Anodyne TRPV1 15 46 O=C(NC[C@H](O)C(F)(F)F)Nc1cccc2nccnc12 ZINC000880781489 DD On-Demand Anodyne TRPV1 15 46 O=C(Nc1cccc2nccnc12)NC1CCC(C(F)(F)F)CC1 ZINC000880781515 EH On-Demand Anodyne TRPV1 15 47 O=C(Nc1cccc2nccnc12)NC1CCC(C(F)(F)F)CC1 ZINC000880781515 EH On-Demand Anodyne EPHX2 37 50 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccsc2)CC1 ZINC000880781526 FG On-Demand Anodyne FAAH 27 47 CCCCNC(=O)Nc1cccc2nccnc12 ZINC000880781556 BF On-Demand Anodyne MTNR1A 24 40 CCCCNC(=O)Nc1cccc2nccnc12 ZINC000880781556 BF On-Demand Anodyne MTNR1B 21 40 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccc2)CC1 ZINC000880781557 EI On-Demand Anodyne SLC18A3 39 40 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccc2)CC1 ZINC000880781557 EI On-Demand Anodyne EPHX2 22 40 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccc2)CC1 ZINC000880781557 EI On-Demand Anodyne RBP4 65 46 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccc2)CC1 ZINC000880781557 EI On-Demand Anodyne SMO 53 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781558 FF On-Demand Anodyne GPR119 39 43 CCCn1cc(CN2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cn1 ZINC000880781582 GF On-Demand Anodyne FAAH 21 40 O=C(Nc1cccc2nccnc12)N1CCC2(CCOCC2)C1 ZINC000880781589 DF On-Demand Anodyne EPHX2 25 42 CC[C@H](CN1CCCC1)NC(=O)Nc1cccc2nccnc12 ZINC000880781599 DF On-Demand Anodyne KCNQ2 45 34 CC[C@@H](CN1CCCC1)NC(=O)Nc1cccc2nccnc12 ZINC000880781600 DF On-Demand Anodyne KCNQ2 45 34 Cn1nccc1C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781605 EF On-Demand Anodyne SMO 26 42 O=C(Nc1cccc2nccnc12)N1CCC(C(F)(F)F)CC1 ZINC000880781607 DG On-Demand Anodyne RBP4 67 43 O=C(Nc1cccc2nccnc12)N1CCC(C(F)(F)F)CC1 ZINC000880781607 DG On-Demand Anodyne SMO 18 41 CCn1nc2c(cc1=O)CN(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880781616 FD On-Demand Anodyne P2RY14 49 35 O=C(NCC(=O)N1CCCCC1)Nc1cccc2nccnc12 ZINC000880781629 DD On-Demand Anodyne PRMT3 18 47 O=C(CCNC(=O)Nc1cccc2nccnc12)NC1CCCCC1 ZINC000880781635 EF On-Demand Anodyne EPHX2 15 43 COC(=O)[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781659 DD On-Demand Anodyne PTR1 45 32 COC(=O)[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880781661 DD On-Demand Anodyne PTR1 45 32 CCc1nc([C@H]2CCCN2C(=O)Nc2cccc3nccnc23)no1 ZINC000880781668 EF On-Demand Anodyne CPT1A 51 41 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](c2ccccc2)O1 ZINC000880781677 EH On-Demand Anodyne RBP4 47 34 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](c2ccccc2)O1 ZINC000880781677 EH On-Demand Anodyne TNKS 15 40 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](c2ccccc2)O1 ZINC000880781679 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](c2ccccc2)O1 ZINC000880781679 EH On-Demand Anodyne TNKS 15 40 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](c2ccccc2)O1 ZINC000880781681 EH On-Demand Anodyne RBP4 47 34 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](c2ccccc2)O1 ZINC000880781681 EH On-Demand Anodyne TNKS 15 40 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](c2ccccc2)O1 ZINC000880781682 EH On-Demand Anodyne RBP4 47 34 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](c2ccccc2)O1 ZINC000880781682 EH On-Demand Anodyne TNKS 15 40 COc1ccc(N2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781683 GG On-Demand Clean PDGFRB 46 40 COc1ccc(N2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781683 GG On-Demand Clean CCKAR 22 40 COc1ccc(N2CCCN(C(=O)Nc3cccc4nccnc34)CC2)cc1 ZINC000880781683 GG On-Demand Clean RBP4 21 44 C[C@H](NC(=O)Nc1cccc2nccnc12)c1ccc(N2CCOCC2)cc1 ZINC000880781697 GG On-Demand Clean PIK3CA 17 41 C[C@H](NC(=O)Nc1cccc2nccnc12)c1ccc(N2CCOCC2)cc1 ZINC000880781697 GG On-Demand Clean MTOR 15 41 O=C(NCc1ccc(N2CCCCC2)nc1)Nc1cccc2nccnc12 ZINC000880781718 FG On-Demand Anodyne NAMPT 46 40 Cc1nc(CN2CCC(CNC(=O)Nc3cccc4nccnc34)CC2)oc1C ZINC000880781728 GG On-Demand Anodyne HTR4 44 36 Cc1nc(CN2CCC(CNC(=O)Nc3cccc4nccnc34)CC2)oc1C ZINC000880781728 GG On-Demand Anodyne CACNA1I 46 32 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880781744 GF On-Demand Anodyne HRH2 27 40 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880781744 GF On-Demand Anodyne AURKB 17 43 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880781744 GF On-Demand Anodyne DDR2 22 43 O=C(Nc1cccc2nccnc12)N1CC[C@@H](N2CCCC2)C1 ZINC000880781748 DE On-Demand Anodyne L3MBTL3 93 44 O=C(Nc1cccc2nccnc12)N1CC[C@H](N2CCCC2)C1 ZINC000880781749 DE On-Demand Anodyne L3MBTL3 93 44 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781755 FG On-Demand Anodyne GPR119 34 41 CCC(CC)(CNC(=O)[C@H]1CCc2nncn2CC1)c1ccc(F)cc1 ZINC000880781758 FG On-Demand Anodyne CACNA1G 55 64 CCC(CC)(CNC(=O)[C@@H]1CCc2nncn2CC1)c1ccc(F)cc1 ZINC000880781759 FG On-Demand Anodyne CACNA1G 55 64 Cc1ncc(CN2CCN(C(=O)Nc3cccc4nccnc34)CC2)s1 ZINC000880781760 FF On-Demand Anodyne FAAH 17 43 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781771 GD On-Demand Anodyne RBP4 41 38 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880781771 GD On-Demand Anodyne CCR8 50 36 O=C(Nc1cccc2nccnc12)N1CCCN(C2CCCC2)CC1 ZINC000880781798 EG On-Demand Anodyne HRH3 24 44 O=C(Nc1cccc2nccnc12)N1CCCN(C2CCCC2)CC1 ZINC000880781798 EG On-Demand Anodyne L3MBTL3 53 36 CC(C)(C)NC(=O)CN1CCC(CNC(=O)Nc2cccc3nccnc23)CC1 ZINC000880781817 GE On-Demand Anodyne CACNA1I 63 49 O=C(Nc1cccc2nccnc12)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880781819 EE On-Demand Anodyne EPHX2 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880781819 EE On-Demand Anodyne RBP4 40 33 O=C(Nc1cccc2nccnc12)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880781820 EE On-Demand Anodyne EPHX2 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880781820 EE On-Demand Anodyne RBP4 40 33 O=C(NCCCC1CC1)Nc1cccc2nccnc12 ZINC000880781830 CF On-Demand Anodyne CCR3 19 40 O=C(Nc1cccc2nccnc12)NC1CCN(C2CCCC2)CC1 ZINC000880781831 EG On-Demand Anodyne EPHX2 32 46 O=C(NCC1CCN(C(=O)c2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880781868 GG On-Demand Anodyne GRIN2B 62 37 O=C(NCC1CCN(C(=O)c2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880781868 GG On-Demand Anodyne EPHX2 15 52 O=C(Nc1cccc2nccnc12)N1CC[C@]2(CCOC2)C1 ZINC000880781878 CE On-Demand Anodyne EPHX2 26 40 O=C(Nc1cccc2nccnc12)N1CC[C@@]2(CCOC2)C1 ZINC000880781879 CE On-Demand Anodyne EPHX2 26 40 O=C(NCCCC(F)(F)F)Nc1cccc2nccnc12 ZINC000880781900 CG On-Demand Anodyne TRPV1 15 47 O=C(Nc1cccc2nccnc12)N1CCC2(CCCCC2)C1 ZINC000880781936 DH On-Demand Anodyne EPHX2 25 44 O=C(Nc1cccc2nccnc12)N1CCC(Nc2cccnn2)CC1 ZINC000880781948 EF On-Demand Anodyne FAAH 22 41 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880781958 GG On-Demand Anodyne FAAH 31 48 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880781958 GG On-Demand Anodyne NACHRBETA2 41 34 O=C(Nc1cccc2nccnc12)N1CCOC2(CCCCC2)C1 ZINC000880782033 EG On-Demand Anodyne EPHX2 15 43 O=C(Nc1cccc2nccnc12)N1CCC2(CCCC2)C1 ZINC000880782042 CG On-Demand Anodyne EPHX2 25 44 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880782059 FG On-Demand Anodyne SMO 42 43 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880782059 FG On-Demand Anodyne ETHR 52 37 O=C(Nc1cccc2nccnc12)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880782060 FG On-Demand Anodyne SMO 42 43 O=C(Nc1cccc2nccnc12)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880782060 FG On-Demand Anodyne ETHR 52 37 O=C(Nc1cccc2nccnc12)N1CC[C@H](O)C1 ZINC000880782079 CD On-Demand Anodyne RBP4 47 36 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cccc2nccnc12 ZINC000880782088 EF On-Demand Anodyne TRPV1 22 42 CC(C)[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880782103 CG On-Demand Anodyne RBP4 45 34 C[C@H](N1CCN(C(=O)Nc2cccc3nccnc23)CC1)C(F)(F)F ZINC000880782111 FF On-Demand Anodyne RBP4 41 35 O=C(Nc1cccc2nccnc12)N1CCC(C(F)(F)F)(C(F)(F)F)C1 ZINC000880782116 GH On-Demand Anodyne EPHX2 30 42 O=C(Nc1cccc2nccnc12)N1CCC(C(F)(F)F)(C(F)(F)F)C1 ZINC000880782116 GH On-Demand Anodyne RBP4 47 34 O=C(Nc1cccc2nccnc12)N1CCN(CCO)CC1 ZINC000880782127 DC On-Demand Anodyne FAAH 17 43 COC(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880782130 DE On-Demand Anodyne RBP4 38 40 COC(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880782130 DE On-Demand Anodyne PTR1 48 34 CC[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCN1C[C@H](C)O ZINC000880782138 ED On-Demand Anodyne LCK 29 40 CC[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCN1C[C@@H](C)O ZINC000880782139 ED On-Demand Anodyne LCK 29 40 O=C(NCCN1CCSCC1)Nc1cccc2nccnc12 ZINC000880782165 DD On-Demand Anodyne UTS2R 20 47 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cccc2nccnc12 ZINC000880782172 GH On-Demand Anodyne ACHE 42 43 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cccc2nccnc12 ZINC000880782172 GH On-Demand Anodyne SIGMAR1 33 41 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cccc2nccnc12 ZINC000880782172 GH On-Demand Anodyne CCR3 42 37 O=C(Nc1cccc2nccnc12)N1CCC(c2ncc[nH]2)CC1 ZINC000880782217 DF On-Demand Anodyne HTR2B 18 40 CN(c1ccccc1)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880782227 FH On-Demand Anodyne RBP4 66 42 CN(c1ccccc1)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880782227 FH On-Demand Anodyne SMO 43 40 C[C@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cccc2nccnc12 ZINC000880782235 EI On-Demand Anodyne RBP4 53 35 C[C@@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cccc2nccnc12 ZINC000880782236 EI On-Demand Anodyne RBP4 53 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C(F)(F)F)O1 ZINC000880782245 EF On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C(F)(F)F)O1 ZINC000880782246 EF On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C(F)(F)F)O1 ZINC000880782247 EF On-Demand Anodyne RBP4 54 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C(F)(F)F)O1 ZINC000880782248 EF On-Demand Anodyne RBP4 54 35 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880782260 CD On-Demand Anodyne UL80 24 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880782260 CD On-Demand Anodyne LGMN 65 33 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880782260 CD On-Demand Anodyne XIAP 27 46 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880782267 FD On-Demand Anodyne MAPK10 20 47 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880782267 FD On-Demand Anodyne EPHX2 27 45 CN(C[C@H](O)CN1CCOCC1)C(=O)Nc1cccc2nccnc12 ZINC000880782320 EC On-Demand Anodyne CASR 41 37 C[C@@H](CNC(=O)Nc1cccc2nccnc12)CN1CCN(C)CC1 ZINC000880782326 ED On-Demand Anodyne ACOX1 40 34 O=C(NCc1ccccc1CN1CCC(O)CC1)Nc1cccc2nccnc12 ZINC000880782328 GF On-Demand Anodyne CCR3 24 41 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne DRD2 16 48 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne DRD4 48 48 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne ACHE 44 42 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne LTA4H 23 41 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne SIGMAR1 43 48 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne CCR3 28 40 CN(C(=O)Nc1cccc2nccnc12)C1CCN(Cc2ccccc2)CC1 ZINC000880782355 GH On-Demand Anodyne CCR5 15 43 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H]1C ZINC000880782356 CF On-Demand Anodyne RBP4 53 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782357 CF On-Demand Anodyne RBP4 53 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782358 CF On-Demand Anodyne RBP4 53 35 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](C(F)(F)F)C1 ZINC000880782359 EE On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CCO[C@H](C(F)(F)F)C1 ZINC000880782360 EE On-Demand Anodyne RBP4 57 37 CN1CCC(CNC(=O)Nc2cccc3nccnc23)(N2CCCCC2)CC1 ZINC000880782364 GF On-Demand Anodyne HCN1 77 41 CN1CCC(CNC(=O)Nc2cccc3nccnc23)(N2CCCCC2)CC1 ZINC000880782364 GF On-Demand Anodyne HCN4 53 34 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cccc2nccnc12 ZINC000880782368 GE On-Demand Anodyne DRD4 28 40 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cccc2nccnc12 ZINC000880782368 GE On-Demand Anodyne P2RX3 27 40 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cccc2nccnc12 ZINC000880782368 GE On-Demand Anodyne SLC27A1 17 40 O=C(Nc1cccc2nccnc12)N1CC=C(C(F)(F)F)CC1 ZINC000880782397 DG On-Demand Anodyne RBP4 55 35 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782477 CG On-Demand Anodyne RBP4 40 35 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782477 CG On-Demand Anodyne SMO 24 40 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@H]1C ZINC000880782478 CG On-Demand Anodyne RBP4 40 35 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@H]1C ZINC000880782478 CG On-Demand Anodyne SMO 24 40 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782479 CG On-Demand Anodyne RBP4 40 35 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1C ZINC000880782479 CG On-Demand Anodyne SMO 24 40 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H]1C ZINC000880782480 CG On-Demand Anodyne RBP4 40 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H]1C ZINC000880782480 CG On-Demand Anodyne SMO 24 40 O=C(Nc1cccc2nccnc12)NC12CCC(CC1)C2 ZINC000880782498 CG On-Demand Anodyne EPHX2 45 45 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@H]1F ZINC000880782501 CF On-Demand Anodyne RBP4 41 37 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1F ZINC000880782502 CF On-Demand Anodyne RBP4 41 37 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1F ZINC000880782503 CF On-Demand Anodyne RBP4 41 37 C[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@H]1F ZINC000880782504 CF On-Demand Anodyne RBP4 41 37 CCC1(O)CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880782529 DF On-Demand Anodyne EPHX2 20 40 COC[C@@H](O)CCNC(=O)Nc1cccc2nccnc12 ZINC000880782544 CD On-Demand Anodyne ADRB1 42 32 O=C(Nc1cccc2nccnc12)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880782546 FE On-Demand Anodyne EPHX2 26 42 O=C(Nc1cccc2nccnc12)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880782547 FE On-Demand Anodyne EPHX2 26 42 O=C(Nc1cccc2nccnc12)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880782548 FE On-Demand Anodyne EPHX2 26 42 O=C(Nc1cccc2nccnc12)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880782549 FE On-Demand Anodyne EPHX2 26 42 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cccc2nccnc12 ZINC000880782552 CG On-Demand Anodyne TRPC6 50 36 C[C@@H]1CCCN(C(=O)Nc2cccc3nccnc23)[C@@H]1C ZINC000880782555 CG On-Demand Anodyne TRPC6 50 36 O=C(Nc1cccc2nccnc12)N1CC(CC(F)(F)F)C1 ZINC000880782561 DG On-Demand Anodyne RBP4 58 39 O=C(Nc1cccc2nccnc12)N1CCC(O)(C(F)(F)F)CC1 ZINC000880782571 EF On-Demand Anodyne RBP4 48 36 O=C(Nc1cccc2nccnc12)N1CCOC2(CCCCCC2)C1 ZINC000880782586 EH On-Demand Anodyne EPHX2 15 43 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880782616 GH On-Demand Anodyne CCR8 56 36 O=C(Nc1cccc2nccnc12)N1CCC2(CC1)OCc1ccccc12 ZINC000880782618 FH On-Demand Anodyne NPY5R 36 42 COc1cccc([C@H]2CN(C(=O)Nc3cccc4nccnc34)CCO2)c1 ZINC000880782632 FG On-Demand Anodyne SMO 19 42 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1cccc2nccnc12 ZINC000880782642 EF On-Demand Anodyne HTR1F 41 32 O=C(Nc1cccc2nccnc12)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880782644 EG On-Demand Anodyne GRIN2B 55 36 O=C(Nc1cccc2nccnc12)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880782644 EG On-Demand Anodyne CCR3 41 40 O=C(Nc1cccc2nccnc12)N1CC[C@H](Cc2ccncc2)C1 ZINC000880782645 EG On-Demand Anodyne GRIN2B 55 36 O=C(Nc1cccc2nccnc12)N1CC[C@H](Cc2ccncc2)C1 ZINC000880782645 EG On-Demand Anodyne CCR3 41 40 O=C(Nc1cccc2nccnc12)N1CCC2(CCC2)C1 ZINC000880782648 CG On-Demand Anodyne EPHX2 25 44 O=C(Nc1cccc2nccnc12)N1CCC(n2ccc(C(F)(F)F)n2)CC1 ZINC000880782659 GH On-Demand Anodyne RBP4 64 40 O=C(Nc1cccc2nccnc12)N1CCCC[C@H]1c1cn[nH]c1 ZINC000880782665 DG On-Demand Anodyne CPT1A 45 34 O=C(Nc1cccc2nccnc12)N1CCCC[C@@H]1c1cn[nH]c1 ZINC000880782666 DG On-Demand Anodyne CPT1A 45 34 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880782676 FF On-Demand Anodyne EPHX2 31 40 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880782677 FF On-Demand Anodyne EPHX2 31 40 O=C(/C=C\c1cccnc1)NCc1ccc(COCC(F)(F)F)cc1 ZINC000880782712 FG On-Demand Anodyne NAMPT 22 42 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccn2)CC1 ZINC000880782723 EG On-Demand Anodyne RBP4 56 43 O=C(Nc1cccc2nccnc12)N1CCC(c2ccccn2)CC1 ZINC000880782723 EG On-Demand Anodyne SMO 48 42 CN(C)CC1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880782755 EF On-Demand Anodyne EPHX2 20 40 O=C(Nc1cccc2nccnc12)N1CCN(C2CCCCC2)CC1 ZINC000880782756 EG On-Demand Anodyne HRH3 20 45 COCCC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880782761 FD On-Demand Anodyne C3AR1 40 39 COCCC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880782761 FD On-Demand Anodyne EPHX2 40 43 COCCC(=O)N1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880782761 FD On-Demand Anodyne CCR8 59 38 O=C(Nc1cccc2nccnc12)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880782772 GH On-Demand Anodyne GRIN2B 32 43 O=C(Nc1cccc2nccnc12)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880782772 GH On-Demand Anodyne RBP4 41 38 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](c2cc(C(F)(F)F)n[nH]2)C1 ZINC000880782891 GH On-Demand Anodyne RBP4 62 38 O=C(Nc1cccc2nccnc12)N1CCC[C@H](c2cc(C(F)(F)F)n[nH]2)C1 ZINC000880782892 GH On-Demand Anodyne RBP4 62 38 O=C(Nc1cccc2nccnc12)N1CC[C@H](C2CCOCC2)C1 ZINC000880782898 EF On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1CC[C@@H](C2CCOCC2)C1 ZINC000880782899 EF On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1CCC(CCCn2ccnc2)CC1 ZINC000880782980 FH On-Demand Anodyne TBXAS1 38 41 O=C(Nc1cccc2nccnc12)N[C@@H]1CC[C@@H](O)CC1 ZINC000880783002 CE On-Demand Anodyne EPHX2 16 45 O=C(Nc1cccc2nccnc12)N1CCOC2(CCCC2)C1 ZINC000880783018 DF On-Demand Anodyne EPHX2 15 44 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](n2ccc(C(F)(F)F)n2)C1 ZINC000880783028 GH On-Demand Anodyne RBP4 54 35 O=C(Nc1cccc2nccnc12)N1CCC[C@H](n2ccc(C(F)(F)F)n2)C1 ZINC000880783029 GH On-Demand Anodyne RBP4 54 35 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783078 GF On-Demand Anodyne GRIN2B 28 45 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783078 GF On-Demand Anodyne C3AR1 46 44 O=C(Nc1cccc2nccnc12)N[C@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783078 GF On-Demand Anodyne CCR8 41 34 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783079 GF On-Demand Anodyne GRIN2B 28 45 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783079 GF On-Demand Anodyne C3AR1 46 44 O=C(Nc1cccc2nccnc12)N[C@@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880783079 GF On-Demand Anodyne CCR8 41 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H](O)C1 ZINC000880783080 CD On-Demand Anodyne RBP4 47 36 CS(=O)(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880783118 ED On-Demand Anodyne RBP4 35 40 O=C(Nc1cccc2nccnc12)N1CCC(C(F)F)CC1 ZINC000880783130 DG On-Demand Anodyne RBP4 52 39 O=C(Nc1cccc2nccnc12)N1CCC(OCc2ccccc2F)CC1 ZINC000880783141 GH On-Demand Anodyne RBP4 44 37 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783149 FG On-Demand Anodyne CACNA1I 47 33 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783149 FG On-Demand Anodyne CCR8 46 40 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783149 FG On-Demand Anodyne GPR119 42 39 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783150 FG On-Demand Anodyne CACNA1I 47 33 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783150 FG On-Demand Anodyne CCR8 46 40 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3nccnc23)C1 ZINC000880783150 FG On-Demand Anodyne GPR119 42 39 O=C(Nc1cccc2nccnc12)N1CCC(Cc2cccnc2)CC1 ZINC000880783161 EH On-Demand Anodyne GRIN2B 60 40 O=C(Nc1cccc2nccnc12)N1CCC(Cc2cccnc2)CC1 ZINC000880783161 EH On-Demand Anodyne CCR3 25 42 O=C(Nc1cccc2nccnc12)N1CCC(Cc2cccnc2)CC1 ZINC000880783161 EH On-Demand Anodyne CHRNA7 53 40 O=C(Nc1cccc2nccnc12)N1CCC(Cc2cccnc2)CC1 ZINC000880783161 EH On-Demand Anodyne C3AR1 41 42 O=C(Nc1cccc2nccnc12)N1CC[C@H](COc2ccccc2)C1 ZINC000880783167 EH On-Demand Anodyne GRIN2B 41 41 O=C(Nc1cccc2nccnc12)N1CC[C@H](COc2ccccc2)C1 ZINC000880783167 EH On-Demand Anodyne CPT1A 42 33 O=C(Nc1cccc2nccnc12)N1CC[C@H](COc2ccccc2)C1 ZINC000880783167 EH On-Demand Anodyne RBP4 46 35 O=C(Nc1cccc2nccnc12)N1CC[C@@H](COc2ccccc2)C1 ZINC000880783168 EH On-Demand Anodyne GRIN2B 41 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H](COc2ccccc2)C1 ZINC000880783168 EH On-Demand Anodyne CPT1A 42 33 O=C(Nc1cccc2nccnc12)N1CC[C@@H](COc2ccccc2)C1 ZINC000880783168 EH On-Demand Anodyne RBP4 46 35 O=C(Nc1cccc2nccnc12)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880783185 FG On-Demand Anodyne RBP4 62 42 O=C(Nc1cccc2nccnc12)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880783185 FG On-Demand Anodyne SMO 18 40 O=C(Nc1cccc2nccnc12)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880783190 FG On-Demand Anodyne EPHX2 19 40 O=C(Nc1cccc2nccnc12)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880783201 EF On-Demand Anodyne HNMT 40 34 O=C(Nc1cccc2nccnc12)N1CC[C@H](CN2CCCCC2)C1 ZINC000880783202 EF On-Demand Anodyne HNMT 40 34 Cc1noc(C2CN(C(=O)Nc3cccc4nccnc34)C2)n1 ZINC000880783221 DD On-Demand Anodyne SMO 39 44 O=C(Nc1cccc2nccnc12)N1CCC([C@@H]2CCCO2)CC1 ZINC000880783227 EG On-Demand Anodyne SMO 32 40 O=C(Nc1cccc2nccnc12)N1CCC([C@H]2CCCO2)CC1 ZINC000880783228 EG On-Demand Anodyne SMO 32 40 COc1cc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)ncn1 ZINC000880783243 FD On-Demand Anodyne PDGFRB 61 43 COc1cc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)ncn1 ZINC000880783243 FD On-Demand Anodyne RBP4 24 42 O=C(Nc1cccc2nccnc12)N1CC(C2CCOCC2)C1 ZINC000880783248 DF On-Demand Anodyne RBP4 54 34 CC(C)(C)OC(=O)N1CC[C@]2(CCN(C(=O)Nc3cccc4nccnc34)C2)C1 ZINC000880783262 GG On-Demand Anodyne EPHX2 24 42 CC(C)(C)OC(=O)N1CC[C@@]2(CCN(C(=O)Nc3cccc4nccnc34)C2)C1 ZINC000880783263 GG On-Demand Anodyne EPHX2 24 42 O=C(Nc1cccc2nccnc12)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880783378 EH On-Demand Anodyne RBP4 53 34 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880783379 EH On-Demand Anodyne RBP4 53 34 O=C(Nc1cccc2nccnc12)N1CCC(c2cccnc2)CC1 ZINC000880783421 EG On-Demand Anodyne RBP4 41 38 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CCN1CC(F)(F)F ZINC000880783454 FF On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCN1CC(F)(F)F ZINC000880783455 FF On-Demand Anodyne RBP4 54 35 Cc1ccncc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880783495 EF On-Demand Anodyne HTR1B 21 40 Cc1ccncc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880783495 EF On-Demand Anodyne PDGFRB 21 42 O=C(Nc1cccc2nccnc12)N1CCCN(c2ncccc2F)CC1 ZINC000880783497 FF On-Demand Anodyne TRPV1 15 45 O=C(Nc1cccc2nccnc12)N1CCCN(c2ncccc2F)CC1 ZINC000880783497 FF On-Demand Anodyne RBP4 19 49 O=C(Nc1cccc2nccnc12)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880783501 GG On-Demand Anodyne UTS2R 16 48 C[C@]1(O)CCCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880783502 CE On-Demand Anodyne EPHX2 15 41 O=C(Nc1cccc2nccnc12)NC1CC(N2CCC(C(F)(F)F)CC2)C1 ZINC000880783520 GH On-Demand Anodyne EPHX2 20 41 O=C(Nc1cccc2nccnc12)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880783521 FF On-Demand Anodyne EPHX2 27 44 O=C(Nc1cccc2nccnc12)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880783524 FF On-Demand Anodyne EPHX2 27 44 O=C(Nc1cccc2nccnc12)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880783527 FF On-Demand Anodyne EPHX2 27 44 O=C(Nc1cccc2nccnc12)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880783530 FF On-Demand Anodyne EPHX2 27 44 O=C(Nc1cccc2nccnc12)N1CCCC2(CCCC2)C1 ZINC000880783555 DH On-Demand Anodyne EPHX2 24 40 O=C(Nc1cccc2nccnc12)N1CCC[C@H](F)C1 ZINC000880783603 CF On-Demand Anodyne RBP4 53 34 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](F)C1 ZINC000880783604 CF On-Demand Anodyne RBP4 53 34 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880783614 CD On-Demand Anodyne RBP4 54 36 C[C@H]1C[C@H](O)CN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880783615 CD On-Demand Anodyne RBP4 54 36 O=C(Nc1cccc2nccnc12)N1C[C@H](O)[C@H](O)C1 ZINC000880783675 CC On-Demand Anodyne RBP4 55 35 C[C@@H](CCNC(=O)Nc1cccc2nccnc12)N1CCCCC1 ZINC000880783690 EG On-Demand Anodyne HRH2 22 40 C[C@H](CCNC(=O)Nc1cccc2nccnc12)N1CCCCC1 ZINC000880783691 EG On-Demand Anodyne HRH2 22 40 O=C(Nc1cccc2nccnc12)N1CCOC2(CCC2)C1 ZINC000880783700 CE On-Demand Anodyne EPHX2 15 44 O=C(Nc1cccc2nccnc12)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880783701 FF On-Demand Anodyne RBP4 62 41 O=C(Nc1cccc2nccnc12)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880783701 FF On-Demand Anodyne SMO 26 41 O=C(Nc1cccc2nccnc12)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880783702 FF On-Demand Anodyne RBP4 62 41 O=C(Nc1cccc2nccnc12)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880783702 FF On-Demand Anodyne SMO 26 41 O=C(Nc1cccc2nccnc12)N1CCN2C(=O)OC[C@@H]2C1 ZINC000880783704 DD On-Demand Anodyne RBP4 43 31 O=C(Nc1cccc2nccnc12)N1CCN2C(=O)OC[C@H]2C1 ZINC000880783705 DD On-Demand Anodyne RBP4 43 31 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cccc2nccnc12 ZINC000880783783 EG On-Demand Anodyne CPT1A 44 33 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cccc2nccnc12 ZINC000880783784 EG On-Demand Anodyne CPT1A 44 33 O=C(Nc1cccc2nccnc12)N1CCN(Cc2ccccn2)CC1 ZINC000880783829 EE On-Demand Anodyne FAAH 23 48 CN(C)CCc1ccc(CNC(=O)Nc2cccc3nccnc23)cc1 ZINC000880783844 EG On-Demand Anodyne ROCK2 15 41 O=C(Nc1cccc2nccnc12)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880783846 GH On-Demand Anodyne NPY5R 34 43 O=C1N[C@H]2CCN(C(=O)Nc3cccc4nccnc34)C[C@@H]2CO1 ZINC000880783847 ED On-Demand Anodyne RBP4 52 33 O=C(NCC(F)(F)F)[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880783859 FE On-Demand Anodyne RBP4 55 37 O=C(NCC(F)(F)F)[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880783860 FE On-Demand Anodyne RBP4 55 37 O=C(Nc1cccc2nccnc12)N1CCC(F)(F)CC1 ZINC000880783870 CF On-Demand Anodyne RBP4 40 34 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)nc1 ZINC000880783947 FE On-Demand Anodyne PDGFRB 57 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)nc1 ZINC000880783947 FE On-Demand Anodyne FAAH 21 40 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)nc1 ZINC000880783947 FE On-Demand Anodyne DGAT1 26 47 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)nc1 ZINC000880783947 FE On-Demand Anodyne NPBWR1 48 35 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne F10 44 61 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne MAPK14 20 43 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne PIK3CA 26 41 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne PRNP 64 52 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne NR1H4 15 41 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne HDAC1 21 43 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne PTK2 18 43 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne MAPK9 34 42 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne MAPK10 42 42 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne FLT3 19 41 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne AURKA 21 47 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne LUCI_LUCLA 38 46 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne EPHB3 29 45 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne STAT6 64 38 O=C(Nc1ccccc1C(=O)Nc1ccc(N2CCOCC2)cn1)c1ccccc1 ZINC000880783950 HG On-Demand Anodyne DGAT1 24 41 O=C(Nc1cccc2nccnc12)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880783965 CE On-Demand Anodyne RBP4 54 34 O=C(Nc1cccc2nccnc12)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880783966 CE On-Demand Anodyne RBP4 54 34 O=C(Nc1cccc2nccnc12)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880783967 CE On-Demand Anodyne RBP4 54 34 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880783983 GG On-Demand Anodyne ACHE 30 45 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880783983 GG On-Demand Anodyne HTR4 41 38 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880783983 GG On-Demand Anodyne SIGMAR1 27 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880783983 GG On-Demand Anodyne CCR3 57 44 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2nccnc12 ZINC000880783983 GG On-Demand Anodyne CACNA1I 52 39 CN(C(=O)Nc1cccc2nccnc12)C1CCN(CC(F)(F)F)CC1 ZINC000880783999 FG On-Demand Anodyne HPGDS 35 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cccc2nccnc12 ZINC000880784001 GF On-Demand Anodyne MCHR1 18 42 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cccc2nccnc12 ZINC000880784002 GF On-Demand Anodyne MCHR1 18 42 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784006 GH On-Demand Anodyne SIRT3 52 35 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784006 GH On-Demand Anodyne SIRT2 55 43 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784006 GH On-Demand Anodyne SIRT1 52 35 O=C(Nc1cccc2nccnc12)N1CC(C2CCCC2)C1 ZINC000880784030 CG On-Demand Anodyne RBP4 56 36 O=C(Nc1cccc2nccnc12)N1CCCC2(CC2)C1 ZINC000880784032 CG On-Demand Anodyne EPHX2 24 40 O=C(NCCN1CCCOCC1)Nc1cccc2nccnc12 ZINC000880784038 DD On-Demand Anodyne UTS2R 18 43 O=C(NCCN1CCCOCC1)Nc1cccc2nccnc12 ZINC000880784038 DD On-Demand Anodyne HNMT 86 39 O=C(NCCN1CCCOCC1)Nc1cccc2nccnc12 ZINC000880784038 DD On-Demand Anodyne EPHX2 22 43 O=C(NCCN1CCCOCC1)Nc1cccc2nccnc12 ZINC000880784038 DD On-Demand Anodyne HPGDS 23 43 O=C(Nc1cccc2nccnc12)N1CC(CO)C1 ZINC000880784044 CD On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc2nccnc12)N1CCC(c2ccsc2)CC1 ZINC000880784045 EI On-Demand Anodyne RBP4 37 40 CN1CCC(N2CCC(NC(=O)Nc3cccc4nccnc34)CC2)CC1 ZINC000880784063 FE On-Demand Anodyne HTR1F 58 34 CN1CCC(N2CCC(NC(=O)Nc3cccc4nccnc34)CC2)CC1 ZINC000880784063 FE On-Demand Anodyne SLC6A5 19 41 C[C@@](O)(C1CCN(C(=O)Nc2cccc3nccnc23)CC1)C(F)(F)F ZINC000880784093 FG On-Demand Anodyne RBP4 63 40 O=C(Nc1cccc2nccnc12)N1C[C@@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880784122 DG On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880784123 DG On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@@H]2C1 ZINC000880784124 DG On-Demand Anodyne RBP4 56 35 O=C(CCCNS(=O)(=O)c1ccc(F)cc1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784129 JF On-Demand Anodyne HTR2A 17 41 O=C(CCCNS(=O)(=O)c1ccc(F)cc1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784129 JF On-Demand Anodyne HTR7 41 42 O=C(CCCNS(=O)(=O)c1ccc(F)cc1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784129 JF On-Demand Anodyne HTR6 15 41 O=C(Nc1cccc2nccnc12)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880784146 FE On-Demand Anodyne CHRNA4 26 48 O=C(Nc1cccc2nccnc12)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880784148 DG On-Demand Anodyne CPT1A 80 40 O=C(Nc1cccc2nccnc12)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880784149 DG On-Demand Anodyne CPT1A 80 40 COC(=O)/C=C\c1ccc(OC(=O)c2cnc3ccccc3c2C(F)(F)F)c(OC)c1 ZINC000880784175 IJ On-Demand Anodyne CYSP_PLAFA 25 41 COC(=O)/C=C\c1ccc(OC(=O)c2ccc(-c3nnc(-c4cccc(C)c4)o3)cc2)c(OC)c1 ZINC000880784180 JK On-Demand Anodyne NR1H4 44 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H](C2CCC2)C1 ZINC000880784223 CG On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1CC[C@H](C2CCC2)C1 ZINC000880784224 CG On-Demand Anodyne RBP4 56 35 CC(C)(C)OC(=O)N1C[C@@H]2CCN(C(=O)Nc3cccc4nccnc34)[C@@H]2C1 ZINC000880784228 GG On-Demand Anodyne GPR119 27 43 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880784236 DE On-Demand Anodyne RBP4 53 36 CN(C)C1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880784266 DF On-Demand Anodyne EPHX2 20 45 CC(=O)NCCN(C)C(=O)Nc1cccc2nccnc12 ZINC000880784295 CD On-Demand Anodyne MTNR1A 25 43 CC(=O)NCCN(C)C(=O)Nc1cccc2nccnc12 ZINC000880784295 CD On-Demand Anodyne MTNR1B 22 43 O=C(Nc1cccc2nccnc12)N1CC[C@@H](O)[C@H](C2CCCC2)C1 ZINC000880784306 EG On-Demand Anodyne RBP4 40 35 CN1CCC(CNC(=O)Nc2cccc3nccnc23)(N2CCOCC2)CC1 ZINC000880784314 GD On-Demand Anodyne HCN1 63 36 CN1CCC(CNC(=O)Nc2cccc3nccnc23)(N2CCOCC2)CC1 ZINC000880784314 GD On-Demand Anodyne HCN4 46 30 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@@H]1O ZINC000880784346 CD On-Demand Anodyne SMO 24 40 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H]1O ZINC000880784347 CD On-Demand Anodyne SMO 24 40 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@@H]1O ZINC000880784348 CD On-Demand Anodyne SMO 24 40 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H]1O ZINC000880784349 CD On-Demand Anodyne SMO 24 40 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne HTR1A 40 45 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne HTR1D 18 46 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne HTR1B 22 46 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne PDGFRB 65 50 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne HTR7 33 42 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne PDGFRA 16 41 COc1cnccc1N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784358 FE On-Demand Anodyne RBP4 23 44 CCOC(=O)N1CCC([C@@H](C)NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880784369 FG On-Demand Anodyne P2RY12 41 33 CCOC(=O)N1CCC([C@H](C)NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880784370 FG On-Demand Anodyne P2RY12 41 33 C[C@@H](C1CC1)n1cc(NC(=O)Nc2cccc3nccnc23)cn1 ZINC000880784383 DG On-Demand Anodyne MAPK10 15 42 CCSCCCNC(=O)Nc1cccc2nccnc12 ZINC000880784388 CF On-Demand Anodyne DOT1L 43 38 CN(C[C@@]1(O)CCN(Cc2ccccc2)C1)C(=O)Nc1cccc2nccnc12 ZINC000880784392 GF On-Demand Anodyne UTS2R 15 40 O=C(NCC1(C(F)(F)F)CC1)Nc1cccc2nccnc12 ZINC000880784451 DG On-Demand Anodyne TRPV1 18 52 O=C(Nc1cccc2nccnc12)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880784470 FG On-Demand Anodyne EPHX2 16 51 O=C(Nc1cccc2nccnc12)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880784471 FG On-Demand Anodyne EPHX2 16 51 CC(C)(C)OC(=O)N1CC[C@@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@@H]21 ZINC000880784481 GG On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CC[C@@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@H]21 ZINC000880784484 GG On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@H]21 ZINC000880784486 GG On-Demand Anodyne GPR119 25 43 CC(C)(C)OC(=O)N1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@@H]21 ZINC000880784488 GG On-Demand Anodyne GPR119 25 43 O=C(Nc1cccc2nccnc12)N1CC(C2CCCCC2)C1 ZINC000880784501 DH On-Demand Anodyne RBP4 56 35 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCCc3n[nH]cc3C2)N1Cc1ccccc1 ZINC000880784512 FD On-Demand Anodyne PREP 77 37 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1CCCc2n[nH]cc2C1 ZINC000880784516 GE On-Demand Anodyne PREP 78 49 O=C(Nc1cccc2nccnc12)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880784532 EF On-Demand Anodyne EPHX2 17 43 O=C(Nc1cccc2nccnc12)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880784534 EF On-Demand Anodyne EPHX2 17 43 O=C(Nc1cccc2nccnc12)N1CCC(c2cn[nH]c2)CC1 ZINC000880784601 DF On-Demand Anodyne RBP4 40 37 O=C(Nc1cccc2nccnc12)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880784652 GF On-Demand Anodyne RBP4 45 39 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3cccc4nccnc34)C[C@@H]2C1 ZINC000880784672 GF On-Demand Anodyne RBP4 55 36 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3cccc4nccnc34)C[C@@H]2C1 ZINC000880784672 GF On-Demand Anodyne GPR119 24 40 C/C=C/C=C\C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784702 DF On-Demand Anodyne CYP1A1 16 41 C/C=C/C=C\C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784702 DF On-Demand Anodyne TUBB1 53 39 C/C=C/C=C\C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784702 DF On-Demand Anodyne ABCG2 17 45 C/C=C/C=C\C(=O)Oc1ccc(/C=C/C(=O)OC)cc1OC ZINC000880784703 DF On-Demand Anodyne CYP1A1 16 41 C/C=C/C=C\C(=O)Oc1ccc(/C=C/C(=O)OC)cc1OC ZINC000880784703 DF On-Demand Anodyne TUBB1 53 39 C/C=C/C=C\C(=O)Oc1ccc(/C=C/C(=O)OC)cc1OC ZINC000880784703 DF On-Demand Anodyne ABCG2 17 45 C/C=C/C=C/C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784704 DF On-Demand Anodyne CYP1A1 16 41 C/C=C/C=C/C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784704 DF On-Demand Anodyne TUBB1 53 39 C/C=C/C=C/C(=O)Oc1ccc(/C=C\C(=O)OC)cc1OC ZINC000880784704 DF On-Demand Anodyne ABCG2 17 45 O=C(Nc1cccc2nccnc12)N1CCOC[C@@H](C2CCC2)C1 ZINC000880784706 EF On-Demand Anodyne RBP4 52 32 O=C(Nc1cccc2nccnc12)N1CCOC[C@H](C2CCC2)C1 ZINC000880784707 EF On-Demand Anodyne RBP4 52 32 O=C(Nc1cccc2nccnc12)N1C[C@H]2[C@H]3C=C[C@@H](C3)[C@H]2C1 ZINC000880784767 DF On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1C[C@H]2[C@H]3C=C[C@@H](C3)[C@H]2C1 ZINC000880784767 DF On-Demand Anodyne WNT3 18 41 O=C(Nc1cccc2nccnc12)N1CCC(CC(F)(F)F)CC1 ZINC000880784782 EH On-Demand Anodyne RBP4 61 41 O=C(Nc1cccc2nccnc12)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880784801 FF On-Demand Anodyne EPHX2 19 41 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](c2ncc(C(F)(F)F)[nH]2)C1 ZINC000880784804 GH On-Demand Anodyne RBP4 72 43 O=C(Nc1cccc2nccnc12)N1CCC[C@H](c2ncc(C(F)(F)F)[nH]2)C1 ZINC000880784805 GH On-Demand Anodyne RBP4 72 43 O=C(Nc1cc(C2CCCC2)[nH]n1)Nc1cccc2nccnc12 ZINC000880784806 DH On-Demand Anodyne CDK2 15 49 O=C(Nc1cc(C2CCCC2)[nH]n1)Nc1cccc2nccnc12 ZINC000880784806 DH On-Demand Anodyne PKNB 64 39 O=C(NCC1(N2CCOCC2)CC1)Nc1cccc2nccnc12 ZINC000880784821 ED On-Demand Anodyne HCN1 51 36 O=C(NCC1(N2CCOCC2)CC1)Nc1cccc2nccnc12 ZINC000880784821 ED On-Demand Anodyne HCN4 47 30 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3nccnc23)C1 ZINC000880784829 ED On-Demand Anodyne EPHX2 33 41 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3nccnc23)C1 ZINC000880784829 ED On-Demand Anodyne CCR8 76 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3nccnc23)C1 ZINC000880784830 ED On-Demand Anodyne EPHX2 33 41 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3nccnc23)C1 ZINC000880784830 ED On-Demand Anodyne CCR8 76 44 O=C(Nc1cccc2nccnc12)N1CCC(CCCN2CCOCC2)CC1 ZINC000880784853 GF On-Demand Anodyne EPHX2 23 41 CC[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCCO1 ZINC000880784864 DF On-Demand Anodyne SMO 48 40 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2nccnc12 ZINC000880784867 EE On-Demand Anodyne MTNR1A 17 41 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2nccnc12 ZINC000880784867 EE On-Demand Anodyne MTNR1B 15 41 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2nccnc12 ZINC000880784867 EE On-Demand Anodyne IKBKE 41 40 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2nccnc12 ZINC000880784867 EE On-Demand Anodyne TBK1 84 40 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880784875 FE On-Demand Anodyne RBP4 41 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)S1(=O)=O ZINC000880784913 ED On-Demand Anodyne RBP4 45 33 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)S1(=O)=O ZINC000880784914 ED On-Demand Anodyne RBP4 45 33 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C)S1(=O)=O ZINC000880784915 ED On-Demand Anodyne RBP4 45 33 O=C(O)c1ccc(C(=O)Nc2ccc(N3CCOCC3)cn2)s1 ZINC000880784916 ED On-Demand Anodyne MAPKAPK5 41 38 O=C(O)c1ccc(C(=O)Nc2ccc(N3CCOCC3)cn2)s1 ZINC000880784916 ED On-Demand Anodyne STAT6 55 36 O=C(Nc1cccc2nccnc12)N1CC[C@@H](F)C1 ZINC000880784921 CE On-Demand Anodyne RBP4 56 38 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cccc2nccnc12 ZINC000880784950 GE On-Demand Anodyne PIK3CA 33 41 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cccc2nccnc12 ZINC000880784950 GE On-Demand Anodyne MTOR 36 41 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cccc2nccnc12 ZINC000880784950 GE On-Demand Anodyne PIK3CG 18 41 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cccc2nccnc12 ZINC000880784950 GE On-Demand Anodyne STAT6 54 34 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cccc2nccnc12 ZINC000880784973 FG On-Demand Anodyne CCR3 35 41 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cccc2nccnc12 ZINC000880784973 FG On-Demand Anodyne CACNA1I 55 35 O=C(COc1cccc(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784995 GH On-Demand Anodyne HTR1D 17 47 O=C(COc1cccc(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784995 GH On-Demand Anodyne HTR1B 18 47 O=C(COc1cccc(Cl)c1)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880784995 GH On-Demand Anodyne FAAH 27 44 O=C(Nc1cccc2nccnc12)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880785002 GG On-Demand Anodyne CACNA1H 50 34 O=C(Nc1cccc2nccnc12)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880785002 GG On-Demand Anodyne UTS2R 16 41 O=C(Nc1cccc2nccnc12)N1CCN(c2cc(C3CC3)[nH]n2)CC1 ZINC000880785006 FF On-Demand Anodyne PKNB 43 35 C[C@@H]1CN(CCCNC(=O)Nc2cccc3nccnc23)CCCO1 ZINC000880785009 EE On-Demand Anodyne HNMT 69 36 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cccc2nccnc12 ZINC000880785012 FE On-Demand Anodyne PIK3CA 29 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cccc2nccnc12 ZINC000880785012 FE On-Demand Anodyne PIK3CD 23 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cccc2nccnc12 ZINC000880785012 FE On-Demand Anodyne MTOR 30 40 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cccc2nccnc12 ZINC000880785012 FE On-Demand Anodyne PIK3CG 22 40 CCOC(=O)c1csc([C@@H]2CCCN2C(=O)Nc2cccc3nccnc23)n1 ZINC000880785014 GH On-Demand Anodyne CPT1A 32 42 CCOC(=O)c1csc([C@H]2CCCN2C(=O)Nc2cccc3nccnc23)n1 ZINC000880785015 GH On-Demand Anodyne CPT1A 32 42 O=C(Nc1cccc2nccnc12)N1CC[C@H](F)C1 ZINC000880785024 CE On-Demand Anodyne RBP4 56 38 COC[C@@H](O)CNC(=O)Nc1cccc2nccnc12 ZINC000880785031 CC On-Demand Anodyne ADRB1 43 33 Cn1ncc2c1CC(C)(C)CN(C(=O)CC[C@@H]1CCc3ccccc31)C2 ZINC000880785038 FH On-Demand Anodyne EBP 17 41 Cn1ncc2c1CC(C)(C)CN(C(=O)CC[C@H]1CCc3ccccc31)C2 ZINC000880785039 FH On-Demand Anodyne EBP 17 41 O=C(Nc1cccc2nccnc12)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880785064 FE On-Demand Anodyne L3MBTL3 63 39 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880785066 FE On-Demand Anodyne L3MBTL3 63 39 O=C(Nc1cccc2nccnc12)N1C[C@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880785079 FF On-Demand Anodyne RBP4 46 32 O=C(Nc1cccc2nccnc12)N1C[C@@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880785080 FF On-Demand Anodyne RBP4 46 32 O=C(Nc1cccc2nccnc12)N1C[C@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880785081 FF On-Demand Anodyne RBP4 46 32 O=C(Nc1cccc2nccnc12)N1C[C@@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880785082 FF On-Demand Anodyne RBP4 46 32 O=C(Nc1cccc2nccnc12)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880785100 FF On-Demand Anodyne RBP4 40 36 O=C(Nc1cccc2nccnc12)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880785101 FF On-Demand Anodyne RBP4 40 36 CN1CC[C@@]2(CCN(C(=O)Nc3cccc4nccnc34)C2)C1 ZINC000880785144 DE On-Demand Anodyne EPHX2 22 41 COC(=O)/C=C\c1ccc(OC(=O)[C@H]2CCCCN2C(=O)c2cccs2)c(OC)c1 ZINC000880785166 IH On-Demand Anodyne FKBP1A 45 38 COC(=O)/C=C\c1ccc(OC(=O)[C@@H]2CCCCN2C(=O)c2cccs2)c(OC)c1 ZINC000880785168 IH On-Demand Anodyne FKBP1A 45 38 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880785170 FF On-Demand Anodyne PIK3CA 22 43 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880785170 FF On-Demand Anodyne MTOR 24 43 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cccc2nccnc12 ZINC000880785170 FF On-Demand Anodyne STAT6 45 37 O=C(Nc1cccc2nccnc12)N1CCC[C@H](CNC(=O)C(F)(F)F)C1 ZINC000880785192 GF On-Demand Anodyne RBP4 52 33 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](CNC(=O)C(F)(F)F)C1 ZINC000880785193 GF On-Demand Anodyne RBP4 52 33 O=C(Nc1cccc2nccnc12)N1C[C@H]2COC[C@@H](C1)O2 ZINC000880785196 DD On-Demand Anodyne RBP4 45 31 O=C(Nc1cccc2nccnc12)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880785206 EF On-Demand Anodyne EPHX2 55 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCCc2n[nH]cc2C1 ZINC000880785230 FD On-Demand Anodyne P2RY12 48 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCCc2n[nH]cc2C1 ZINC000880785231 FD On-Demand Anodyne P2RY12 48 36 O=C(Nc1cccc2nccnc12)N1C[C@@H](CO)[C@@H](CO)C1 ZINC000880785266 DC On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc2nccnc12)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880785267 DC On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc2nccnc12)N[C@@H]1C[C@H]1C(F)(F)F ZINC000880785314 CF On-Demand Anodyne TRPV1 17 46 O=C(CNC(=O)Nc1cccc2nccnc12)NCCN1CCCCCC1 ZINC000880785364 FD On-Demand Anodyne UTS2R 16 41 O=C(CNC(=O)Nc1cccc2nccnc12)NCCN1CCCCCC1 ZINC000880785364 FD On-Demand Anodyne HNMT 100 43 O=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cccc2nccnc12 ZINC000880785367 CE On-Demand Anodyne WNT3 15 41 O=C(Nc1cccc2nccnc12)N1CC(C(F)(F)F)C1 ZINC000880785384 CF On-Demand Anodyne RBP4 71 41 O=C(Nc1cccc2nccnc12)N[C@@H]1CCCN(CCCO)C1 ZINC000880785385 ED On-Demand Anodyne CCR3 22 42 O=C(Nc1cccc2nccnc12)N[C@@H]1CCCN(CCCO)C1 ZINC000880785385 ED On-Demand Anodyne HNMT 53 34 O=C(Nc1cccc2nccnc12)N[C@H]1CCCN(CCCO)C1 ZINC000880785386 ED On-Demand Anodyne CCR3 22 42 O=C(Nc1cccc2nccnc12)N[C@H]1CCCN(CCCO)C1 ZINC000880785386 ED On-Demand Anodyne HNMT 53 34 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880785443 GH On-Demand Anodyne SLC18A2 45 33 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880785443 GH On-Demand Anodyne HCRTR1 15 41 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880785444 GH On-Demand Anodyne SLC18A2 45 33 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cccc3nccnc13)CC2 ZINC000880785444 GH On-Demand Anodyne HCRTR1 15 41 CN1CCN(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)CC1 ZINC000880785475 FD On-Demand Anodyne HTR1F 47 33 CN1CCN(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)CC1 ZINC000880785475 FD On-Demand Anodyne SMO 31 40 CN1CCN(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)CC1 ZINC000880785475 FD On-Demand Anodyne L3MBTL3 63 40 O=C1OC[C@H]2CN(C(=O)Nc3cccc4nccnc34)C[C@@H]12 ZINC000880785480 CD On-Demand Anodyne RBP4 46 33 O=C(NCC1(C(F)(F)F)CCCC1)Nc1cccc2nccnc12 ZINC000880785519 EH On-Demand Anodyne TRPV1 15 51 O=C(Nc1cccc2nccnc12)N1CCC(CCF)CC1 ZINC000880785522 DG On-Demand Anodyne RBP4 61 41 O=C(Nc1cccc2nccnc12)N1CCC2(COC2)C1 ZINC000880785525 CD On-Demand Anodyne EPHX2 24 42 O=C(Nc1cccc2nccnc12)N1CC(CNC(=O)C(F)(F)F)C1 ZINC000880785526 FD On-Demand Anodyne RBP4 55 34 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](CC(F)(F)F)O1 ZINC000880785530 FG On-Demand Anodyne RBP4 52 34 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](CC(F)(F)F)O1 ZINC000880785531 FG On-Demand Anodyne RBP4 52 34 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](CC(F)(F)F)O1 ZINC000880785532 FG On-Demand Anodyne RBP4 52 34 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](CC(F)(F)F)O1 ZINC000880785533 FG On-Demand Anodyne RBP4 52 34 CN(C(=O)Nc1cccc2nccnc12)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880785550 EF On-Demand Anodyne GLRA1 47 38 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCC1(F)F ZINC000880785566 DG On-Demand Anodyne RBP4 40 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CCC1(F)F ZINC000880785567 DG On-Demand Anodyne RBP4 40 35 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880785574 FF On-Demand Anodyne EPHX2 28 40 O=C(NCC1(c2ccccn2)CCC1)Nc1cccc2nccnc12 ZINC000880785577 EG On-Demand Anodyne NMBR 44 40 O=C(Nc1cccc2nccnc12)N[C@@H]1CCCN(C(=O)CCC(F)(F)F)C1 ZINC000880785603 GG On-Demand Anodyne EPHX2 24 41 O=C(Nc1cccc2nccnc12)N[C@@H]1CCCN(C(=O)CCC(F)(F)F)C1 ZINC000880785603 GG On-Demand Anodyne ETHR 57 37 CN(C)CCCOc1cnccc1CNC(=O)Nc1cccc2nccnc12 ZINC000880785613 GF On-Demand Anodyne ROCK2 17 43 O=C(Nc1cccc2nccnc12)N1CC(C2CC2)C1 ZINC000880785628 CF On-Demand Anodyne RBP4 58 37 O=C(Nc1cccc2nccnc12)N1CC[C@@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880785643 FF On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880785644 FF On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@H](C(F)(F)F)[C@H](CO)C1 ZINC000880785645 FF On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@@H](C(F)(F)F)[C@H](CO)C1 ZINC000880785646 FF On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880785662 EH On-Demand Anodyne NPY5R 37 41 O=C(Nc1cccc2nccnc12)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880785663 EH On-Demand Anodyne NPY5R 37 41 COC(=O)c1cnc(C2CCN(C(=O)Nc3cccc4nccnc34)CC2)s1 ZINC000880785671 GG On-Demand Anodyne RBP4 43 45 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cccc2nccnc12 ZINC000880785677 EE On-Demand Anodyne HCRTR1 31 42 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cccc2nccnc12 ZINC000880785677 EE On-Demand Anodyne HCRTR2 21 42 O=C(NCC1CCN(CC2CC2)CC1)Nc1cccc2nccnc12 ZINC000880785678 EF On-Demand Anodyne HTR4 34 41 O=C(NCC1CCN(CC2CC2)CC1)Nc1cccc2nccnc12 ZINC000880785678 EF On-Demand Anodyne CCR3 49 37 O=C(NCC1CCN(CC2CC2)CC1)Nc1cccc2nccnc12 ZINC000880785678 EF On-Demand Anodyne CACNA1I 53 35 O=C(Nc1cccc2nccnc12)N1CCN(CCc2cnccn2)CC1 ZINC000880785688 FD On-Demand Anodyne FAAH 15 40 O=C(Nc1cccc2nccnc12)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880785691 EH On-Demand Anodyne RBP4 66 38 O=C(Nc1cccc2nccnc12)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880785691 EH On-Demand Anodyne SMO 35 41 O=C(Nc1cccc2nccnc12)N1C[C@@H](CO)[C@H](C(F)(F)F)C1 ZINC000880785694 EE On-Demand Anodyne RBP4 56 37 O=C(Nc1cccc2nccnc12)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880785697 FG On-Demand Anodyne RBP4 40 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@@H](C(F)(F)F)O1 ZINC000880785731 FG On-Demand Anodyne RBP4 56 36 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H](C(F)(F)F)O1 ZINC000880785732 FG On-Demand Anodyne RBP4 56 36 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@@H](C(F)(F)F)O1 ZINC000880785733 FG On-Demand Anodyne RBP4 56 36 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@H](C(F)(F)F)O1 ZINC000880785734 FG On-Demand Anodyne RBP4 56 36 COc1ccc([C@@H]2CCCN2C(=O)Nc2cccc3nccnc23)cc1F ZINC000880785735 FI On-Demand Anodyne RBP4 19 40 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne CYP1B1 15 42 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne CYP1A1 15 42 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne NR1H4 44 37 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne TUBB1 42 36 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne ABCG2 15 40 COC(=O)/C=C\c1ccc(OC(=O)/C=C\c2cccnc2)c(OC)c1 ZINC000880785826 EF On-Demand Anodyne CYSP_PLAFA 20 40 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne CYP1B1 15 42 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne CYP1A1 15 42 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne NR1H4 44 37 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne TUBB1 42 36 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne ABCG2 15 40 COC(=O)/C=C\c1ccc(OC(=O)/C=C/c2cccnc2)c(OC)c1 ZINC000880785827 EF On-Demand Anodyne CYSP_PLAFA 20 40 O=C(Nc1cccc2nccnc12)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880785854 DF On-Demand Anodyne CPT1A 78 38 O=C(Nc1cccc2nccnc12)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880785855 DF On-Demand Anodyne CPT1A 78 38 CC(C)[C@H]1CN(C(=O)Nc2cccc3nccnc23)CCN1C ZINC000880785893 DE On-Demand Anodyne LCK 33 47 O=C(Nc1cccc2nccnc12)N1CC2(CCC2)[C@@H]1c1ccccc1 ZINC000880785898 EI On-Demand Anodyne TNKS 15 41 O=C(Nc1cccc2nccnc12)N1CC2(CCC2)[C@H]1c1ccccc1 ZINC000880785903 EI On-Demand Anodyne TNKS 15 41 O=C(Nc1cccc2nccnc12)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880785907 CF On-Demand Anodyne RBP4 54 34 COc1ccccc1[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CCO1 ZINC000880785923 FG On-Demand Anodyne RBP4 43 38 COc1ccccc1[C@@H]1CN(C(=O)Nc2cccc3nccnc23)CCO1 ZINC000880785923 FG On-Demand Anodyne SMO 21 41 O=C(NCCN1CC[C@@H](O)C1)Nc1cccc2nccnc12 ZINC000880785931 DC On-Demand Anodyne UTS2R 17 41 O=C(NCCN1CC[C@H](O)C1)Nc1cccc2nccnc12 ZINC000880785933 DC On-Demand Anodyne UTS2R 17 41 O=C(NCC[C@@H](O)COCc1ccccc1)Nc1cccc2nccnc12 ZINC000880785934 FF On-Demand Anodyne ADRB1 41 32 O=C(NC[C@H]1CCCCN1C(=O)C(F)(F)F)Nc1cccc2nccnc12 ZINC000880785946 GF On-Demand Anodyne HCRTR1 26 41 O=C(NC[C@H]1CCCCN1C(=O)C(F)(F)F)Nc1cccc2nccnc12 ZINC000880785946 GF On-Demand Anodyne HCRTR2 15 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880785992 CC On-Demand Anodyne RBP4 53 37 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786008 CD On-Demand Anodyne CCR8 43 32 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786011 CD On-Demand Anodyne CCR8 43 32 O=C(Nc1cccc2nccnc12)N1CCC[C@H](C2CCC2)C1 ZINC000880786012 DH On-Demand Anodyne RBP4 55 35 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](C2CCC2)C1 ZINC000880786014 DH On-Demand Anodyne RBP4 55 35 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)C1O ZINC000880786031 DE On-Demand Anodyne RBP4 45 33 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)[C@@H]1O ZINC000880786032 DE On-Demand Anodyne RBP4 45 33 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C)C1O ZINC000880786033 DE On-Demand Anodyne RBP4 45 33 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786035 EG On-Demand Anodyne RBP4 67 39 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786036 EG On-Demand Anodyne RBP4 67 39 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880786039 EF On-Demand Anodyne RBP4 54 35 O=C(Nc1cccc2nccnc12)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880786040 EF On-Demand Anodyne RBP4 54 35 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)N1CC#N ZINC000880786058 DE On-Demand Mild RBP4 54 36 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)N1CC#N ZINC000880786059 DE On-Demand Mild RBP4 54 36 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C)N1CC#N ZINC000880786060 DE On-Demand Mild RBP4 54 36 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cccc2nccnc12 ZINC000880786075 EH On-Demand Anodyne PTAFR 35 47 O=C(Nc1cccc2nccnc12)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880786081 GH On-Demand Anodyne SMO 47 49 O=C(Nc1cccc2nccnc12)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880786081 GH On-Demand Anodyne ETHR 63 43 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](C(F)F)CC1 ZINC000880786082 DF On-Demand Anodyne RBP4 43 37 O=C(Nc1cccc2nccnc12)N1CCO[C@H](C(F)F)CC1 ZINC000880786083 DF On-Demand Anodyne RBP4 43 37 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786088 DG On-Demand Anodyne EPHX2 28 40 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786088 DG On-Demand Anodyne RBP4 40 34 O=C(Nc1cccc2nccnc12)N1CC(CC2CC2)C1 ZINC000880786095 CF On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1C[C@H]2COC[C@H]2C1 ZINC000880786138 CD On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880786145 ED On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880786146 ED On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880786149 ED On-Demand Anodyne RBP4 53 33 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880786151 ED On-Demand Anodyne RBP4 53 33 CC(=O)C1CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880786170 CE On-Demand Anodyne SMO 27 40 O=C(Nc1cccc2nccnc12)N1CCC(F)CC1 ZINC000880786176 CF On-Demand Anodyne RBP4 57 41 CCOC(=O)[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H]1C(F)(F)F ZINC000880786178 GF On-Demand Anodyne RBP4 52 35 COC1(C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)CC1 ZINC000880786203 FG On-Demand Anodyne RBP4 41 38 O=C(Nc1cccc2nccnc12)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880786216 FH On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc2nccnc12)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880786217 FH On-Demand Anodyne RBP4 45 32 O=C(Nc1cccc2nccnc12)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880786223 DE On-Demand Anodyne RBP4 65 38 O=C(Nc1cccc2nccnc12)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880786224 DE On-Demand Anodyne RBP4 65 38 O=C(Nc1cccc2nccnc12)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880786225 DE On-Demand Anodyne RBP4 65 38 O=C(Nc1cccc2nccnc12)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880786226 DE On-Demand Anodyne RBP4 65 38 O=C(Nc1cccc2nccnc12)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880786227 DE On-Demand Anodyne RBP4 65 38 CS(=O)(=O)C1CN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786230 DC On-Demand Anodyne RBP4 42 33 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786247 GF On-Demand Anodyne HRH2 25 40 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786247 GF On-Demand Anodyne SIGMAR1 34 42 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786247 GF On-Demand Anodyne NPFFR2 41 42 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786247 GF On-Demand Anodyne UTS2R 19 48 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786247 GF On-Demand Anodyne NPFFR1 52 42 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1cccc2nccnc12 ZINC000880786254 FD On-Demand Anodyne HCN1 47 39 O=C(Nc1cccc2nccnc12)N1CC[C@H](C2CCCC2)C1 ZINC000880786257 DH On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1CC[C@@H](C2CCCC2)C1 ZINC000880786258 DH On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1CCC2(CC1)OCCc1ccccc12 ZINC000880786262 FH On-Demand Anodyne NPY5R 31 41 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)CC[C@@H](C)O1 ZINC000880786301 DF On-Demand Anodyne SMO 28 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2C[C@@H]2C1 ZINC000880786302 CF On-Demand Anodyne RBP4 62 40 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2C[C@H]2C1 ZINC000880786303 CF On-Demand Anodyne RBP4 62 40 O=C(Nc1cccc2nccnc12)N1CC[C@H]2C[C@H]2C1 ZINC000880786304 CF On-Demand Anodyne RBP4 62 40 O=C(Nc1cccc2nccnc12)N1CC[C@H]2C[C@@H]2C1 ZINC000880786305 CF On-Demand Anodyne RBP4 62 40 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880786306 EF On-Demand Anodyne RBP4 61 42 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880786306 EF On-Demand Anodyne SMO 16 41 O=C(Nc1cccc2nccnc12)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880786307 EF On-Demand Anodyne RBP4 61 42 O=C(Nc1cccc2nccnc12)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880786307 EF On-Demand Anodyne SMO 16 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean HTR1A 47 49 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean DRD4 40 32 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean HTR1D 17 49 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean HTR1B 19 49 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean DRD3 46 39 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean PDGFRB 81 51 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean HTR7 38 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean KDR 67 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean MET 15 41 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean PDGFRA 51 44 COc1ccc(N2CCN(C(=O)Nc3cccc4nccnc34)CC2)c(OC)c1 ZINC000880786313 GG On-Demand Clean RBP4 24 45 O=C(Nc1cccc2nccnc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880786329 FH On-Demand Anodyne FAAH 19 42 O=C(Nc1cccc2nccnc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880786329 FH On-Demand Anodyne EPHX2 21 40 O=C(Nc1cccc2nccnc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880786329 FH On-Demand Anodyne SCD1 23 43 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786354 FE On-Demand Anodyne EPHX2 25 40 O=C(Nc1cccc2nccnc12)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880786359 CG On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CCO[C@H](CCF)C1 ZINC000880786362 DE On-Demand Anodyne RBP4 50 32 O=C(Nc1cccc2nccnc12)N1CCO[C@@H](CCF)C1 ZINC000880786363 DE On-Demand Anodyne RBP4 50 32 O=C(Nc1cccc2nccnc12)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880786372 FD On-Demand Anodyne RBP4 48 37 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880786377 CE On-Demand Anodyne RBP4 55 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2OCC[C@@H]2C1 ZINC000880786388 CE On-Demand Anodyne RBP4 53 34 O=C(Nc1cccc2nccnc12)N(CCN1CCOCC1)Cc1ccco1 ZINC000880786389 GF On-Demand Anodyne CASR 57 45 C[C@@]1(CNC(=O)Nc2cccc3nccnc23)CC1(Cl)Cl ZINC000880786399 EG On-Demand Anodyne G2YM83_BOTF4 58 32 O=C(Nc1cccc2nccnc12)N1CC[C@](O)(Cc2ccc(F)cc2)C1 ZINC000880786400 FF On-Demand Anodyne UTS2R 15 45 O=C(Nc1cccc2nccnc12)N1CC[C@@](O)(Cc2ccc(F)cc2)C1 ZINC000880786401 FF On-Demand Anodyne UTS2R 15 45 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc3nccnc13)C2 ZINC000880786402 DE On-Demand Anodyne HTR3A 35 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc3nccnc13)C2 ZINC000880786402 DE On-Demand Anodyne GLRA1 48 39 O=C(Nc1cccc2nccnc12)N1CCC(C2CCC2)CC1 ZINC000880786423 DH On-Demand Anodyne RBP4 40 38 O=C(Nc1cccc2nccnc12)N1C[C@H]2CCCC[C@H]2C1 ZINC000880786424 CG On-Demand Anodyne RBP4 57 37 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880786443 GF On-Demand Anodyne RBP4 88 41 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880786444 GF On-Demand Anodyne RBP4 88 41 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880786445 GF On-Demand Anodyne RBP4 88 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880786446 GF On-Demand Anodyne RBP4 88 41 O=C(Nc1cccc2nccnc12)NC1CCN(C2CCC2)CC1 ZINC000880786459 EF On-Demand Anodyne EPHX2 31 43 O=C(Nc1cccc2nccnc12)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880786466 GG On-Demand Anodyne TRPM8 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880786467 GG On-Demand Anodyne TRPM8 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880786468 GG On-Demand Anodyne TRPM8 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880786469 GG On-Demand Anodyne TRPM8 26 41 O=C(Nc1cccc2nccnc12)N1CC[C@H]2COC[C@H]2C1 ZINC000880786478 CE On-Demand Anodyne RBP4 55 34 O=C(Nc1cccc2nccnc12)N1CC[C@H]2COC[C@@H]2C1 ZINC000880786479 CE On-Demand Anodyne RBP4 55 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2COC[C@H]2C1 ZINC000880786480 CE On-Demand Anodyne RBP4 55 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880786509 DF On-Demand Anodyne RBP4 54 34 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CSC[C@H]2C1 ZINC000880786510 DF On-Demand Anodyne RBP4 54 34 O=C(Nc1cccc2nccnc12)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880786511 DF On-Demand Anodyne RBP4 54 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880786512 DF On-Demand Anodyne RBP4 54 34 C[C@@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)C1(F)F ZINC000880786529 DG On-Demand Anodyne RBP4 55 36 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@@H](C)C1(F)F ZINC000880786530 DG On-Demand Anodyne RBP4 55 36 C[C@H]1CN(C(=O)Nc2cccc3nccnc23)C[C@H](C)C1(F)F ZINC000880786531 DG On-Demand Anodyne RBP4 55 36 O=C(Nc1cccc2nccnc12)N1CCC(c2ccon2)CC1 ZINC000880786544 DG On-Demand Anodyne SMO 43 44 O=C(NCCC1(O)CCN(c2ccccc2)CC1)Nc1cccc2nccnc12 ZINC000880786550 GG On-Demand Anodyne UTS2R 18 45 O=C1CC[C@@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@@H]2N1 ZINC000880786562 ED On-Demand Anodyne RBP4 54 35 O=C1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@H]2N1 ZINC000880786563 ED On-Demand Anodyne RBP4 54 35 O=C1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@@H]2N1 ZINC000880786564 ED On-Demand Anodyne RBP4 54 35 O=C1CC[C@@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@H]2N1 ZINC000880786565 ED On-Demand Anodyne RBP4 54 35 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880786580 EF On-Demand Anodyne KCNQ2 60 37 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880786580 EF On-Demand Anodyne TRPV1 23 61 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880786580 EF On-Demand Anodyne SCN2A 18 44 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2nccnc12 ZINC000880786580 EF On-Demand Anodyne SCN10A 23 44 CN(CCN1CCCCC1)C(=O)Nc1cccc2nccnc12 ZINC000880786600 DF On-Demand Anodyne HRH3 25 48 CN(CCN1CCCCC1)C(=O)Nc1cccc2nccnc12 ZINC000880786600 DF On-Demand Anodyne HNMT 93 48 C[C@@H]1CN(CC(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786618 FF On-Demand Anodyne RBP4 54 35 O=C(Nc1cccc2nccnc12)N1CCC(OC2CCC2)CC1 ZINC000880786638 EG On-Demand Anodyne EPHX2 15 40 CC(C)(C)C1CN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786640 CG On-Demand Anodyne RBP4 54 35 O=C(Nc1cccc2nccnc12)N1CCC[C@H](CC(F)(F)F)C1 ZINC000880786648 EH On-Demand Anodyne RBP4 56 35 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](CC(F)(F)F)C1 ZINC000880786649 EH On-Demand Anodyne RBP4 56 35 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild DRD4 21 51 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild HRH2 27 41 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild SIGMAR1 19 45 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild SSTR5 59 35 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild CCR3 48 50 N#Cc1cccc(CN2CCC(NC(=O)Nc3cccc4nccnc34)CC2)c1 ZINC000880786653 GG On-Demand Mild MCHR1 50 49 CC(C)(C)N1CC[C@@H](NC(=O)Nc2cccc3nccnc23)C1=O ZINC000880786660 EE On-Demand Anodyne TRPV1 17 48 CC(C)(C)N1CC[C@@H](NC(=O)Nc2cccc3nccnc23)C1=O ZINC000880786660 EE On-Demand Anodyne CCKBR 15 40 CC(C)(C)N1CC[C@H](NC(=O)Nc2cccc3nccnc23)C1=O ZINC000880786661 EE On-Demand Anodyne TRPV1 17 48 CC(C)(C)N1CC[C@H](NC(=O)Nc2cccc3nccnc23)C1=O ZINC000880786661 EE On-Demand Anodyne CCKBR 15 40 O=C(Nc1cccc2nccnc12)N1CCC[C@H](CCF)C1 ZINC000880786679 DG On-Demand Anodyne RBP4 51 33 O=C(Nc1cccc2nccnc12)N1CCC[C@@H](CCF)C1 ZINC000880786680 DG On-Demand Anodyne RBP4 51 33 CN1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@H]21 ZINC000880786683 DE On-Demand Anodyne RBP4 53 34 CN1CC[C@H]2CN(C(=O)Nc3cccc4nccnc34)CC[C@@H]21 ZINC000880786684 DE On-Demand Anodyne RBP4 53 34 O=C(Nc1cccc2nccnc12)N1CC[C@@H](c2nccs2)C1 ZINC000880786696 EG On-Demand Anodyne RBP4 40 37 O=C(Nc1cccc2nccnc12)N1CC[C@H](c2nccs2)C1 ZINC000880786697 EG On-Demand Anodyne RBP4 40 37 COc1ccc([C@@H]2CCN(C(=O)Nc3cccc4nccnc34)C2)cc1F ZINC000880786723 FH On-Demand Anodyne RBP4 54 44 COc1ccc([C@@H]2CCN(C(=O)Nc3cccc4nccnc34)C2)cc1F ZINC000880786723 FH On-Demand Anodyne SMO 23 41 O=C(Nc1cccc2nccnc12)N1CC[C@@H](CF)C1 ZINC000880786736 CE On-Demand Anodyne RBP4 47 36 O=C(Nc1cccc2nccnc12)N1CC[C@H](CF)C1 ZINC000880786737 CE On-Demand Anodyne RBP4 47 36 CC(C)(C)OC(=O)CN1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880786742 GF On-Demand Anodyne EPHX2 38 40 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cccc3nccnc23)C1 ZINC000880786750 EF On-Demand Anodyne EPHX2 28 40 C[C@@H]1CCN(C(=O)Nc2cccc3nccnc23)C[C@@H]1NC(=O)C(F)(F)F ZINC000880786761 GF On-Demand Anodyne RBP4 54 38 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)Nc3cccc4nccnc34)CC2)C1 ZINC000880786869 GG On-Demand Anodyne EPHX2 21 40 COCC1CCC(NC(=O)Nc2cccc3nccnc23)CC1 ZINC000880786870 DF On-Demand Anodyne EPHX2 18 40 CN(C[C@H]1CCCN1C)C(=O)Nc1cccc2nccnc12 ZINC000880786881 CE On-Demand Anodyne CHRNA10 61 35 CN(C[C@H]1CCCN1C)C(=O)Nc1cccc2nccnc12 ZINC000880786881 CE On-Demand Anodyne ACKR3 49 31 CN(C[C@@H]1CCCN1C)C(=O)Nc1cccc2nccnc12 ZINC000880786882 CE On-Demand Anodyne CHRNA10 61 35 CN(C[C@@H]1CCCN1C)C(=O)Nc1cccc2nccnc12 ZINC000880786882 CE On-Demand Anodyne ACKR3 49 31 O=C(Nc1cccc2nccnc12)NC1CCC(OC(F)F)CC1 ZINC000880786937 EG On-Demand Anodyne EPHX2 26 42 COC[C@@H]1CCCCN1C(=O)Nc1cccc2nccnc12 ZINC000880786942 DF On-Demand Anodyne CPT1A 75 35 O=C(Nc1cccc2nccnc12)N1C[C@@H]2OCCN(Cc3ccccc3)[C@@H]2C1 ZINC000880786960 GF On-Demand Anodyne RBP4 44 31 COc1ccc(CN(CCO)C(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880787075 GF On-Demand Anodyne ROCK2 15 45 COC(=O)[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C1CCCCC1 ZINC000880787216 GG On-Demand Anodyne PRMT3 34 42 COC(=O)[C@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C1CCCCC1 ZINC000880787217 GG On-Demand Anodyne PRMT3 34 42 O=C(Nc1cccc2nccnc12)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880787223 GD On-Demand Anodyne EPHX2 24 48 O=C(Nc1cccc2nccnc12)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880787224 GD On-Demand Anodyne EPHX2 24 48 N#CC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCCC1 ZINC000880787423 EG On-Demand Mild PRMT3 53 35 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787429 GG On-Demand Anodyne DRD4 28 46 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787429 GG On-Demand Anodyne CCR3 51 46 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787429 GG On-Demand Anodyne CCR2 17 41 Cc1ccc(CN2CC[C@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787429 GG On-Demand Anodyne MCHR1 25 46 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787430 GG On-Demand Anodyne DRD4 28 46 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787430 GG On-Demand Anodyne CCR3 51 46 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787430 GG On-Demand Anodyne CCR2 17 41 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)cc1 ZINC000880787430 GG On-Demand Anodyne MCHR1 25 46 C[S@@](=O)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880787491 DD On-Demand Anodyne PRMT3 51 32 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880787510 GF On-Demand Anodyne EPHX2 52 44 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880787510 GF On-Demand Anodyne CXCR3 18 46 CN1CCN(C2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)CC1 ZINC000880787566 GD On-Demand Anodyne L3MBTL3 49 38 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880787585 FH On-Demand Anodyne EPHX2 33 40 COCC(C)(C)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880787594 EF On-Demand Anodyne PRMT3 43 34 Cc1cncc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)n1 ZINC000880787735 EE On-Demand Anodyne PRMT3 58 32 N#CCc1cccc2c1CCN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)C2 ZINC000880787766 GG On-Demand Mild P2RY14 45 36 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@@H]1Br ZINC000880787890 FG On-Demand Reactive EPHX2 18 40 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@@H]1Br ZINC000880787890 FG On-Demand Reactive PRMT3 58 32 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@H]1Br ZINC000880787891 FG On-Demand Reactive EPHX2 18 40 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@H]1Br ZINC000880787891 FG On-Demand Reactive PRMT3 58 32 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880787965 FH On-Demand Anodyne TRPM8 18 43 CCN(CC)C(=O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880787983 ED On-Demand Anodyne PRMT3 45 32 CC1CC(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880787994 DF On-Demand Anodyne PRMT3 58 32 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880788014 GG On-Demand Anodyne P2RY14 47 33 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@@H]2C[C@@H]2C1 ZINC000880788136 EG On-Demand Anodyne EPHX2 19 41 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C[C@@H]2C[C@@H]2C1 ZINC000880788136 EG On-Demand Anodyne PRMT3 43 30 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788172 FI On-Demand Anodyne TRPM8 29 47 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880788197 GF On-Demand Anodyne EPHX2 43 39 CC[C@@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788221 CD On-Demand Anodyne PRMT3 60 36 CC(C)(C)OC(=O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCC1 ZINC000880788222 GG On-Demand Anodyne PRMT3 43 31 CCNC(=O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788255 DC On-Demand Anodyne PRMT3 61 33 COC1CC(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880788286 EF On-Demand Anodyne PRMT3 16 40 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880788318 DE On-Demand Anodyne EPHX2 42 34 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1(F)F ZINC000880788348 EF On-Demand Anodyne PRMT3 51 31 CO[C@]1(CO)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880788366 FD On-Demand Anodyne EPHX2 16 40 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)C2 ZINC000880788378 GG On-Demand Anodyne P2RY14 42 31 CO[C@@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788432 CD On-Demand Anodyne PRMT3 61 35 N#CC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880788452 EF On-Demand Mild PRMT3 52 33 COc1cccc([C@]2(C)CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)C2)c1 ZINC000880788497 GH On-Demand Anodyne EPHX2 28 41 COc1ccccc1-c1ccnc(C2CCN(C(=O)Cc3cnc(C)o3)CC2)n1 ZINC000880788507 GG On-Demand Anodyne ETHR 40 30 Cc1cc(F)ccc1C1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880788550 GJ On-Demand Anodyne HTR1D 15 43 CCCN(CCN1CCCCC1)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788568 GG On-Demand Anodyne CASR 41 37 CCCN(CCN1CCCC1)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788574 FG On-Demand Anodyne CASR 43 37 Cc1ccncc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880788575 GF On-Demand Anodyne HTR1B 15 43 C[C@@H]1CN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CCc2ccc(F)cc21 ZINC000880788656 GI On-Demand Anodyne TRPM8 15 41 C[C@H]1CN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CCc2ccc(F)cc21 ZINC000880788657 GI On-Demand Anodyne TRPM8 15 41 Cn1ncc(C2CC2)c1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788690 FF On-Demand Anodyne PRMT3 44 31 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@H](CO)Cc1ccccc1 ZINC000880788828 FF On-Demand Anodyne NPY5R 34 46 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@@H](CO)Cc1ccccc1 ZINC000880788830 FF On-Demand Anodyne NPY5R 34 46 COCC[C@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788863 DF On-Demand Anodyne PRMT3 51 33 COCC[C@@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788865 DF On-Demand Anodyne PRMT3 51 33 C[C@H]1CN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CCN1Cc1ccccc1 ZINC000880788884 GG On-Demand Anodyne P2RY14 42 33 C[C@@H]1CN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CCN1Cc1ccccc1 ZINC000880788886 GG On-Demand Anodyne P2RY14 42 33 Cc1cnc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c(C)c1 ZINC000880788944 FG On-Demand Anodyne PRMT3 60 34 C[C@@H](F)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880788971 CF On-Demand Anodyne PRMT3 44 32 Cc1nnc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)s1 ZINC000880789027 EE On-Demand Anodyne PRMT3 63 35 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880789032 GF On-Demand Anodyne EPHX2 43 39 COc1cnccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789069 GE On-Demand Anodyne HTR1A 17 49 COc1cnccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789069 GE On-Demand Anodyne HTR1D 15 49 COc1cnccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789069 GE On-Demand Anodyne HTR1B 20 49 COc1cnccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789069 GE On-Demand Anodyne PDGFRB 58 47 CC(C)(C)C(C)(C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789092 EH On-Demand Anodyne PRMT3 58 31 Cc1ncsc1CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789143 EF On-Demand Anodyne PRMT3 59 33 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1(Cl)Cl ZINC000880789168 FG On-Demand Anodyne PRMT3 50 30 C=CC(C)(C)CC(=O)N1CCC(c2nccc(-c3ccccc3OC)n2)CC1 ZINC000880789177 GI On-Demand Mild ETHR 40 31 CN1CCC[C@@H](CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880789180 EF On-Demand Anodyne CCR3 56 38 CN1CCC[C@@H](CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880789180 EF On-Demand Anodyne PRMT3 33 43 O=C(CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)NCC(F)F ZINC000880789189 ED On-Demand Anodyne F7 17 40 O=C(CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)NCC(F)F ZINC000880789189 ED On-Demand Anodyne PRMT3 40 35 CN1CC[C@@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)[C@@H]1c1cccnc1 ZINC000880789205 GF On-Demand Anodyne NAMPT 40 37 CC/C=C\CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789221 CF On-Demand Anodyne PRMT3 50 32 CC/C=C/CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789223 CF On-Demand Anodyne PRMT3 50 32 CC1(C)CCC[C@]1(O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789253 EF On-Demand Anodyne PRMT3 42 29 CN1CCC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)c2ccccc21 ZINC000880789254 GH On-Demand Anodyne CCKAR 30 40 CN1CCC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)c2ccccc21 ZINC000880789254 GH On-Demand Anodyne CCKBR 56 40 CC1(C)CCC[C@@]1(O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789255 EF On-Demand Anodyne PRMT3 42 29 COCC1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789262 EG On-Demand Anodyne EPHX2 43 37 C[C@@H]1CCC[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789411 DG On-Demand Anodyne PRMT3 65 36 C[C@H]1CCC[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789413 DG On-Demand Anodyne PRMT3 65 36 C[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789415 DG On-Demand Anodyne PRMT3 65 36 N#CC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789583 DE On-Demand Mild PRMT3 59 33 COc1cccc(C2(CNC(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)c1 ZINC000880789604 GH On-Demand Anodyne MTNR1B 27 40 COc1cccc(C2(CNC(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)c1 ZINC000880789604 GH On-Demand Anodyne SOAT1 17 46 CC(C)(C#N)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789616 DE On-Demand Mild PRMT3 60 31 COCC(C)(C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789657 DF On-Demand Anodyne PRMT3 58 31 CCc1nnc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)s1 ZINC000880789665 EE On-Demand Anodyne PRMT3 62 34 CCOC(=O)C1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789727 GF On-Demand Anodyne EPHX2 45 38 N#CC1(c2ccccn2)CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880789746 GG On-Demand Mild CACNA1H 32 40 COC[C@@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789849 DC On-Demand Anodyne ADRB1 41 32 COC[C@@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880789849 DC On-Demand Anodyne PRMT3 60 36 CCC[C@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)OC ZINC000880789902 DF On-Demand Anodyne PRMT3 51 33 CCC[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)OC ZINC000880789904 DF On-Demand Anodyne PRMT3 51 33 O=C(c1c[nH]cc1C1CC1)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880789984 GJ On-Demand Anodyne HTR1F 62 39 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880789988 FF On-Demand Anodyne EPHX2 19 40 Cc1cnc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cn1 ZINC000880789997 EE On-Demand Anodyne PRMT3 59 33 C[C@H]1c2ccccc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790168 FH On-Demand Anodyne TRPM8 38 41 N#CCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790183 CD On-Demand Mild PRMT3 58 33 C[C@@H](CCCc1cccnc1)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790200 FH On-Demand Anodyne PTAFR 35 46 C[C@@H]1CN(CCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCO1 ZINC000880790227 GE On-Demand Anodyne CCR3 42 42 CN(C)C1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880790230 EF On-Demand Anodyne EPHX2 40 38 N#CC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCC1 ZINC000880790240 DF On-Demand Mild PRMT3 52 33 O=C(COC1CC1)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790254 FG On-Demand Anodyne CPT1A 15 40 O=C(COC1CC1)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790254 FG On-Demand Anodyne MAPK1 55 39 O=C(COC1CC1)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790254 FG On-Demand Anodyne ETHR 38 44 COc1ccc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)nc1 ZINC000880790257 GE On-Demand Anodyne PDGFRB 56 40 COc1ccc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)nc1 ZINC000880790257 GE On-Demand Anodyne FAAH 15 42 COc1ccc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)nc1 ZINC000880790257 GE On-Demand Anodyne DGAT1 23 42 C=CCC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880790276 EH On-Demand Mild PRMT3 44 31 O=C1NCC[C@H]1CC(=O)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790283 GF On-Demand Anodyne ETHR 38 43 O=C1NCC[C@@H]1CC(=O)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790285 GF On-Demand Anodyne ETHR 38 43 COC(=O)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880790322 FE On-Demand Anodyne EPHX2 56 44 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790355 GG On-Demand Anodyne NPY5R 33 46 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790356 GG On-Demand Anodyne NPY5R 33 46 C[C@@H](C1CC1)n1cc(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)cn1 ZINC000880790385 FH On-Demand Anodyne ITK 41 32 CCC1(c2ccccc2)CN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880790388 FH On-Demand Anodyne EPHX2 15 43 O=C(c1cnc(C2CC2)o1)N1CCC(c2nccc(-c3cccc(F)c3)n2)CC1 ZINC000880790445 GI On-Demand Anodyne ETHR 17 41 CCO[C@H]1C[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880790490 DE On-Demand Anodyne EPHX2 42 34 C=C(CC)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790512 CF On-Demand Mild PRMT3 53 33 Cn1cnc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880790689 ED On-Demand Anodyne PRMT3 58 32 Cn1nc2c(cc1=O)CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880790710 FD On-Demand Anodyne P2RY14 42 31 Cc1ncc(CC(=O)N2CCC(c3nccc(-c4cccc(F)c4)n3)CC2)o1 ZINC000880790719 GH On-Demand Anodyne ETHR 47 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880790720 FE On-Demand Anodyne EPHX2 44 43 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880790721 FE On-Demand Anodyne EPHX2 44 43 CC[C@H]1c2ccccc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790739 FI On-Demand Anodyne TRPM8 36 41 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790740 FI On-Demand Anodyne TRPM8 36 41 Cn1cnc2c(c1=O)CCN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)C2 ZINC000880790746 FD On-Demand Anodyne P2RY14 47 33 Cc1cc(C)c2c(c1)CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880790770 FH On-Demand Anodyne P2RY14 40 33 O=C(c1cncc2[nH]ccc12)N1CCC(c2nccc(N3CCOCC3)n2)CC1 ZINC000880790771 GE On-Demand Anodyne ATR 48 36 CC[C@@H]1CCC[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790812 EH On-Demand Anodyne PRMT3 68 38 CC[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790813 EH On-Demand Anodyne PRMT3 68 38 CC[C@H]1CCC[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790814 EH On-Demand Anodyne PRMT3 68 38 CC[C@@H]1CCC[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790815 EH On-Demand Anodyne PRMT3 68 38 CSC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCC1 ZINC000880790840 EG On-Demand Anodyne PRMT3 44 31 CSC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880790844 DF On-Demand Anodyne PRMT3 50 31 C[C@H]1CCC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880790854 EH On-Demand Anodyne EPHX2 40 42 C[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)N(C)C ZINC000880790870 DD On-Demand Anodyne PRMT3 43 33 C[C@@H](Cc1cccc(F)c1)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790874 FH On-Demand Anodyne NPY5R 29 46 Cn1cc(-c2ccnc(C3CCN(C(=O)c4c[nH]cc4C4CC4)CC3)n2)cn1 ZINC000880790888 GG On-Demand Anodyne HTR1F 61 33 C[C@]1(O)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880790889 EE On-Demand Anodyne EPHX2 15 40 CN(C)CCc1ccc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880790928 GG On-Demand Anodyne PRMT3 54 40 COCCC[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790983 GH On-Demand Anodyne TACR2 40 33 COCCC[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880790984 GH On-Demand Anodyne TACR2 40 33 CN(CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C1CCCCC1 ZINC000880791136 FG On-Demand Anodyne PRMT3 41 39 COc1cccc(C2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)c1 ZINC000880791153 GI On-Demand Anodyne MCHR1 18 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791173 FE On-Demand Anodyne CCR3 40 37 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791175 FE On-Demand Anodyne CCR3 40 37 Cc1nn(CC(=O)N2CCC(c3nccc(-c4cccc(F)c4)n3)CC2)c(=O)o1 ZINC000880791177 GE On-Demand Anodyne ETHR 43 43 C=C(C)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791211 CF On-Demand Mild PRMT3 50 32 O=C(c1cnc2cc[nH]c2c1)N1CCC(c2nccc(N3CCOCC3)n2)CC1 ZINC000880791253 GE On-Demand Anodyne MTOR 22 41 O=C(c1cnc2cc[nH]c2c1)N1CCC(c2nccc(N3CCOCC3)n2)CC1 ZINC000880791253 GE On-Demand Anodyne FASN 35 41 O=C(c1cnc2cc[nH]c2c1)N1CCC(c2nccc(N3CCOCC3)n2)CC1 ZINC000880791253 GE On-Demand Anodyne ATR 47 37 COC(=O)CCCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791410 FF On-Demand Anodyne EPHX2 19 42 Cn1cc(-c2ccnc(C3CCN(C(=O)CC[C@@H]4CC(C)(C)CO4)CC3)n2)cn1 ZINC000880791449 GG On-Demand Anodyne ETHR 51 33 Cn1cc(-c2ccnc(C3CCN(C(=O)CC[C@H]4CC(C)(C)CO4)CC3)n2)cn1 ZINC000880791450 GG On-Demand Anodyne ETHR 51 33 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791452 GD On-Demand Anodyne CCR3 55 37 CO[C@@]1(C)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791462 EF On-Demand Anodyne EPHX2 20 40 CCNC(=O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCC1 ZINC000880791616 FE On-Demand Anodyne PRMT3 59 32 O=C(NCC1(C(=O)NCCc2cnoc2)CCCC1)OCc1ccccc1 ZINC000880791658 FF On-Demand Anodyne CAPN2 68 36 O=C(NCC1(C(=O)NCCc2cnoc2)CCCC1)OCc1ccccc1 ZINC000880791658 FF On-Demand Anodyne NPR 56 37 O=C(NCC1(C(=O)NCCc2cnoc2)CCCC1)OCc1ccccc1 ZINC000880791658 FF On-Demand Anodyne SLC12A5 41 32 CCC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880791662 EH On-Demand Anodyne PRMT3 58 30 CNC(C)(C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791729 DD On-Demand Anodyne PRMT3 50 30 CC(C)(C)OC(=O)N1CC[C@H](CC(=O)NCCc2cnoc2)C1 ZINC000880791756 DD On-Demand Anodyne GPR119 41 38 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791770 ED On-Demand Anodyne EPHX2 40 53 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791771 ED On-Demand Anodyne EPHX2 40 53 CC(C)CN1CCC[C@@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791793 GG On-Demand Anodyne CCR3 60 40 CC(C)CN1CCC[C@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791794 GG On-Demand Anodyne CCR3 60 40 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCO1 ZINC000880791811 DE On-Demand Anodyne PRMT3 44 31 CS[C@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791882 DF On-Demand Anodyne PRMT3 43 33 C[C@H](NC(=O)Nc1ccc2c(c1)SCC(=O)N2)c1cccc(N2CCCC2)c1 ZINC000880791891 GI On-Demand Anodyne KCNQ2 16 40 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880791908 GG On-Demand Anodyne ACHE 27 40 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880791908 GG On-Demand Anodyne SIGMAR1 30 42 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880791908 GG On-Demand Anodyne MCHR1 27 42 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880791909 GG On-Demand Anodyne ACHE 27 40 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880791909 GG On-Demand Anodyne SIGMAR1 30 42 CN(C(=O)Nc1ccc2c(c1)SCC(=O)N2)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880791909 GG On-Demand Anodyne MCHR1 27 42 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880791921 FH On-Demand Anodyne NPY5R 25 45 COCC1(O)CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880791949 FD On-Demand Anodyne S1PR2 28 40 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](F)C(=O)NCCc2cnoc2)C1 ZINC000880791953 ED On-Demand Anodyne GPR119 39 43 CC(C)(C)OC(=O)N1CC[C@@H]([C@H](F)C(=O)NCCc2cnoc2)C1 ZINC000880791954 ED On-Demand Anodyne GPR119 39 43 CC(C)(C)OC(=O)N1CC[C@H]([C@@H](F)C(=O)NCCc2cnoc2)C1 ZINC000880791955 ED On-Demand Anodyne GPR119 39 43 CC(C)(C)OC(=O)N1CC[C@H]([C@H](F)C(=O)NCCc2cnoc2)C1 ZINC000880791956 ED On-Demand Anodyne GPR119 39 43 CCN1CCC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791973 EE On-Demand Anodyne CCR3 35 41 CCN1CCC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880791974 EE On-Demand Anodyne CCR3 35 41 Cc1nc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)sc1C ZINC000880792018 FG On-Demand Anodyne PRMT3 59 33 Cc1ncc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)s1 ZINC000880792065 EF On-Demand Anodyne PRMT3 59 33 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCS1 ZINC000880792121 EG On-Demand Anodyne PRMT3 42 29 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCc2cnoc2)CC1 ZINC000880792184 EE On-Demand Anodyne TBK1 44 31 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCc2cnoc2)CC1 ZINC000880792184 EE On-Demand Anodyne GPR119 41 40 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCc2cnoc2)CC1 ZINC000880792185 EE On-Demand Anodyne TBK1 44 31 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCc2cnoc2)CC1 ZINC000880792185 EE On-Demand Anodyne GPR119 41 40 Cc1noc(C)c1CCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792191 FG On-Demand Anodyne PRMT3 50 32 COCCC(=O)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880792212 GD On-Demand Anodyne EPHX2 52 47 C=C(Cl)C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880792252 EE On-Demand Mild FPR1 44 37 C=C(Cl)C[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880792253 EE On-Demand Mild FPR1 44 37 COc1ccc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)cc1 ZINC000880792263 GG On-Demand Clean HTR1B 16 50 COc1ccc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)cc1 ZINC000880792263 GG On-Demand Clean PDGFRB 50 39 O=C(NCCc1cnoc1)[C@@H]1CC(c2ccc(Cl)cc2Cl)=NO1 ZINC000880792267 FF On-Demand Anodyne ALPL 40 33 O=C(NCCc1cnoc1)[C@H]1CC(c2ccc(Cl)cc2Cl)=NO1 ZINC000880792268 FF On-Demand Anodyne ALPL 40 33 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880792295 GD On-Demand Anodyne P2RY14 50 35 CCC1(O)CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880792341 EE On-Demand Anodyne S1PR2 29 41 O=C(CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)NCC1CC1 ZINC000880792355 ED On-Demand Anodyne PRMT3 47 35 N#CCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792448 CE On-Demand Mild PRMT3 44 32 Cc1nc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cs1 ZINC000880792471 EF On-Demand Anodyne PRMT3 60 33 O=C(CN1CCCC[C@@H](OCc2ccccc2)C1=O)NCCc1cnoc1 ZINC000880792482 FD On-Demand Anodyne PREP 50 34 O=C(CN1CCCC[C@H](OCc2ccccc2)C1=O)NCCc1cnoc1 ZINC000880792483 FD On-Demand Anodyne PREP 50 34 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792580 FH On-Demand Anodyne CFTR 56 32 C[C@H]1Cc2ccccc2CN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792581 FH On-Demand Anodyne CFTR 56 32 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792590 GD On-Demand Mild CASR 60 49 C[C@@H](CCc1cccn1C)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792592 FG On-Demand Anodyne CCR3 43 32 CCC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCC1 ZINC000880792619 DG On-Demand Anodyne PRMT3 43 30 CC(C)(C)OC(=O)N1CCC([C@@H]2C[C@H]2C(=O)NCCc2cnoc2)CC1 ZINC000880792633 FF On-Demand Anodyne GPR119 40 42 O=C(NCCc1cnoc1)c1ccccc1OC1CC1 ZINC000880792638 CE On-Demand Anodyne KCNA3 40 40 O=C(NCCc1cnoc1)c1ccccc1OC1CC1 ZINC000880792638 CE On-Demand Anodyne HCN1 55 33 O=C(NCCc1cnoc1)c1ccccc1OC1CC1 ZINC000880792638 CE On-Demand Anodyne HCN4 41 33 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792665 ED On-Demand Anodyne UL80 40 39 C[C@@H]1CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)[C@@H]1C ZINC000880792676 DG On-Demand Anodyne TRPC6 49 38 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792677 DG On-Demand Anodyne TRPC6 49 38 COC[C@@H](O)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792689 ED On-Demand Anodyne ADRB1 40 32 COC[C@@H](O)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792689 ED On-Demand Anodyne PRMT3 51 32 COc1cccc(C(C)(C)C(=O)NCCc2cnoc2)c1 ZINC000880792749 CE On-Demand Anodyne MTNR1A 63 40 COc1cccc(C(C)(C)C(=O)NCCc2cnoc2)c1 ZINC000880792749 CE On-Demand Anodyne MTNR1B 58 40 COc1ccc2c(c1)CC[C@H]2C(=O)NCCc1cnoc1 ZINC000880792755 CE On-Demand Anodyne NQO2 39 40 COc1ccc2c(c1)CC[C@H]2C(=O)NCCc1cnoc1 ZINC000880792755 CE On-Demand Anodyne MTNR1A 74 44 COc1ccc2c(c1)CC[C@H]2C(=O)NCCc1cnoc1 ZINC000880792755 CE On-Demand Anodyne MTNR1B 62 36 CN(C)CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880792791 ED On-Demand Anodyne PAPA1_CARPA 38 42 CN(C)CC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880792792 ED On-Demand Anodyne PAPA1_CARPA 38 42 CC[C@@H](Nc1cccnc1Cl)C(=O)NCCc1cnoc1 ZINC000880792798 DE On-Demand Anodyne G2YM83_BOTF4 62 31 CC[C@H](Nc1cccnc1Cl)C(=O)NCCc1cnoc1 ZINC000880792799 DE On-Demand Anodyne G2YM83_BOTF4 62 31 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne HTR1A 53 45 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne DRD2 40 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne ADRA1D 54 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne HTR1B 15 45 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne ADRA1A 46 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne ADRA1B 43 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792817 GG On-Demand Anodyne DRD3 44 38 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne HTR1A 53 45 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne DRD2 40 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne ADRA1D 54 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne HTR1B 15 45 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne ADRA1A 46 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne ADRA1B 43 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880792818 GG On-Demand Anodyne DRD3 44 38 CC(C)(C)OC(=O)N[C@@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880792867 EF On-Demand Anodyne PAPA1_CARPA 36 42 CC(C)(C)OC(=O)N[C@@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880792867 EF On-Demand Anodyne TACR3 19 40 CC(C)(C)OC(=O)N[C@@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880792867 EF On-Demand Anodyne FPR1 47 37 CC(C)(C)OC(=O)N[C@@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880792867 EF On-Demand Anodyne Q82323_9DELA 63 30 C[C@@H]1CN(Cc2ccccc2)CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792901 GG On-Demand Anodyne CCR1 22 41 C[C@@](O)(CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)c1cccs1 ZINC000880792936 FF On-Demand Anodyne PRMT3 44 31 CN(CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2)Cc1ccc(F)cc1 ZINC000880792941 GG On-Demand Anodyne CCR3 28 42 CC(C)(C)OC(=O)N[C@@H](c1ccccc1)C(C)(C)C(=O)NCCc1cnoc1 ZINC000880792942 GH On-Demand Anodyne CMA1 23 40 CC(C)(C)OC(=O)N[C@@H](c1ccccc1)C(C)(C)C(=O)NCCc1cnoc1 ZINC000880792942 GH On-Demand Anodyne PAPA1_CARPA 32 40 CC(C)(C)OC(=O)N[C@@H](c1ccccc1)C(C)(C)C(=O)NCCc1cnoc1 ZINC000880792942 GH On-Demand Anodyne TACR3 19 42 CC(C)(C)OC(=O)N[C@@H](c1ccccc1)C(C)(C)C(=O)NCCc1cnoc1 ZINC000880792942 GH On-Demand Anodyne FPR1 43 35 COc1ccccc1C[C@@H](C)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792948 GH On-Demand Anodyne NPY5R 33 43 COc1ccccc1C[C@H](C)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880792950 GH On-Demand Anodyne NPY5R 33 43 CCC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880792985 DG On-Demand Anodyne PRMT3 57 30 O=C(CCC1CCCCC1)NNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880793056 GG On-Demand Reactive PRMT3 25 40 O=C(NCCc1cnoc1)c1cccn(C2CC2)c1=O ZINC000880793057 CD On-Demand Anodyne POLR1A 50 32 CN(C)CC1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880793077 FF On-Demand Anodyne PRMT3 43 30 COC(=O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880793149 FF On-Demand Anodyne PRMT3 59 31 COCCCOc1cccc(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880793171 GH On-Demand Anodyne EPHX2 28 44 CC(C)(C)OC(=O)N[C@@H](C(=O)NCCc1cnoc1)c1c(F)cccc1F ZINC000880793236 GF On-Demand Anodyne PAPA1_CARPA 31 40 C[C@H](CCc1ccc(F)cc1)C(=O)NCCc1cnoc1 ZINC000880793266 CF On-Demand Anodyne LEF 46 37 C[C@@H](CCc1ccc(F)cc1)C(=O)NCCc1cnoc1 ZINC000880793267 CF On-Demand Anodyne LEF 46 37 COC[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)OC ZINC000880793279 ED On-Demand Anodyne PRMT3 58 33 CC[C@]1(C)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880793346 EH On-Demand Anodyne EPHX2 18 41 C[C@@H](CNC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880793362 CD On-Demand Anodyne FPR1 41 34 CCc1cnc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)s1 ZINC000880793392 EG On-Demand Anodyne PRMT3 51 31 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC[C@H]1O ZINC000880793396 EF On-Demand Anodyne PRMT3 46 33 C[C@@]1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC[C@@H]1O ZINC000880793399 EF On-Demand Anodyne PRMT3 46 33 Cc1nc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)sc1C ZINC000880793529 EG On-Demand Anodyne PRMT3 51 32 CCCCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880793536 FG On-Demand Anodyne EPHX2 50 42 CCCCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880793536 FG On-Demand Anodyne CXCR3 21 42 O=C(/C=C\c1cccnc1)Nc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000880793562 EE On-Demand Anodyne TGM2 41 43 O=C(/C=C\c1cccnc1)Nc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000880793562 EE On-Demand Anodyne F13A1 64 44 O=C(/C=C\c1cccnc1)Nc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000880793562 EE On-Demand Anodyne SFRP1 40 37 O=C(/C=C\c1cccnc1)Nc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000880793562 EE On-Demand Anodyne NAMPT 64 67 CC(C)(C)C(=O)NCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880793581 FE On-Demand Anodyne PRMT3 51 36 CC(C)(C)OC(=O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880793603 EE On-Demand Anodyne PRMT3 46 32 CC(C)(C)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880793632 CF On-Demand Anodyne IMDH_CRYPV 44 33 COc1cccc(O[C@H](C)CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880793641 GG On-Demand Anodyne MTNR1A 25 50 COc1cccc(O[C@H](C)CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880793641 GG On-Demand Anodyne MTNR1B 29 50 COc1cccc(O[C@@H](C)CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880793642 GG On-Demand Anodyne MTNR1A 25 50 COc1cccc(O[C@@H](C)CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880793642 GG On-Demand Anodyne MTNR1B 29 50 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)NCCc2cnoc2)C1 ZINC000880793740 DD On-Demand Anodyne GPBAR1 23 42 O=C(NCCc1cnoc1)c1ccnc(C(F)(F)F)c1 ZINC000880793766 CE On-Demand Anodyne KDM4E 26 48 CC(C)(C)OC(=O)N1CSC[C@H]1C(=O)NCCc1cnoc1 ZINC000880793768 ED On-Demand Anodyne CACNA1B 17 43 CO[C@H]1CCC[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880793860 EF On-Demand Anodyne PRMT3 62 35 O=C(NCCc1cnoc1)[C@@H](Cc1cccnc1)C1CCCC1 ZINC000880793910 DF On-Demand Anodyne C3AR1 44 44 O=C(NCCc1cnoc1)[C@H](Cc1cccnc1)C1CCCC1 ZINC000880793911 DF On-Demand Anodyne C3AR1 44 44 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CTSB 37 42 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne PAPA1_CARPA 43 34 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CTSK 42 44 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CTSL 36 44 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CAPNS1 58 42 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne HLA-DRB1 46 34 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CTSS 26 44 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CAPN1 90 43 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne CAPN2 129 42 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne FPR1 56 35 COC(=O)N[C@@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880793934 CD On-Demand Anodyne NPR 78 41 O=C(NCCc1cnoc1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794004 FD On-Demand Anodyne CELA1 19 43 O=C(NCCc1cnoc1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794004 FD On-Demand Anodyne PREP 39 43 O=C(NCCc1cnoc1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794004 FD On-Demand Anodyne LGMN 59 38 O=C(NCCc1cnoc1)[C@@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794004 FD On-Demand Anodyne KLK5 40 41 O=C(NCCc1cnoc1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794005 FD On-Demand Anodyne CELA1 19 43 O=C(NCCc1cnoc1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794005 FD On-Demand Anodyne PREP 39 43 O=C(NCCc1cnoc1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794005 FD On-Demand Anodyne LGMN 59 38 O=C(NCCc1cnoc1)[C@H]1COCCN1C(=O)OCc1ccccc1 ZINC000880794005 FD On-Demand Anodyne KLK5 40 41 CN(C)C(=O)c1cccc(CCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880794047 GF On-Demand Anodyne PRMT3 52 32 C[C@]1(O)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880794120 DE On-Demand Anodyne EPHX2 19 43 C[C@@]1(C#N)CCCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880794132 EF On-Demand Mild EPHX2 15 40 Cn1nccc1CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794153 ED On-Demand Anodyne PRMT3 61 33 CC(C)[C@H](O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794223 EF On-Demand Anodyne PRMT3 60 32 NS(=O)(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1 ZINC000880794231 HD On-Demand Anodyne CA2 19 41 NS(=O)(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1 ZINC000880794231 HD On-Demand Anodyne CA7 17 41 NS(=O)(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1 ZINC000880794231 HD On-Demand Anodyne CA13 16 41 NS(=O)(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1 ZINC000880794231 HD On-Demand Anodyne CCR8 35 41 COC(=O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCCC1 ZINC000880794247 GF On-Demand Anodyne PRMT3 60 32 CN(C)S(=O)(=O)c1cc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)ccc1Cl ZINC000880794278 JG On-Demand Anodyne CCR8 30 40 C[C@H]1c2c(F)cccc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794403 FI On-Demand Anodyne TRPM8 32 45 CCC(CC)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794404 DG On-Demand Anodyne PRMT3 59 34 CN1CCC(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794408 EE On-Demand Anodyne CACNA1I 42 32 CN(CCN1CCOCC1)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794419 FD On-Demand Anodyne CASR 54 42 CC(C)(C)OC(=O)N1CC[C@@H](C(=O)NCCc2cnoc2)C1 ZINC000880794502 DD On-Demand Anodyne GPR119 42 38 CC(C)(C)OC(=O)N1CC[C@H](C(=O)NCCc2cnoc2)C1 ZINC000880794503 DD On-Demand Anodyne GPR119 42 38 C[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C(C)(C)C ZINC000880794506 DH On-Demand Anodyne PRMT3 44 33 CC(C)(C)OC(=O)N1CC[C@@H](CC(=O)NCCc2cnoc2)C1 ZINC000880794514 DD On-Demand Anodyne GPR119 41 38 CCc1nc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cs1 ZINC000880794517 EG On-Demand Anodyne PRMT3 50 32 CC(C)(C)[C@@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794538 DE On-Demand Anodyne PRMT3 62 37 COC(=O)C1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794562 FF On-Demand Anodyne EPHX2 42 38 CC(C)(C)OC(=O)N1CCC(SCC(=O)NCCc2cnoc2)CC1 ZINC000880794563 FE On-Demand Anodyne GPR119 45 40 CC1(C)C[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794567 DF On-Demand Anodyne PRMT3 58 30 Cc1noc(C)c1CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794591 EF On-Demand Anodyne PRMT3 58 32 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)C(F)(F)F ZINC000880794602 DC On-Demand Anodyne F2 23 41 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)C(F)(F)F ZINC000880794603 DC On-Demand Anodyne F2 23 41 O=C(NCCc1cnoc1)c1coc(C2CCOCC2)n1 ZINC000880794661 CD On-Demand Anodyne TBXA2R 30 42 CC(C)(O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794721 CD On-Demand Anodyne PRMT3 59 31 CC(C)(C)OC(=O)N1CCC[C@H](CC(=O)NCCc2cnoc2)CC1 ZINC000880794736 FF On-Demand Anodyne GPR119 43 38 CC(C)(C)OC(=O)N1CCC[C@@H](CC(=O)NCCc2cnoc2)CC1 ZINC000880794737 FF On-Demand Anodyne GPR119 43 38 CC(C)n1ccc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)n1 ZINC000880794747 EF On-Demand Anodyne PRMT3 59 32 CN1CCC[C@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880794765 EE On-Demand Anodyne CCR3 49 39 C[C@@H](Cc1ccc(Cl)cc1)N(C)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880794778 GI On-Demand Anodyne NPY5R 25 44 CC(C)(C)OC(=O)NCc1cccc(C(=O)NCCc2cnoc2)c1 ZINC000880794782 EF On-Demand Anodyne KDM4E 21 42 C[C@@]1(C(=O)NCCc2cnoc2)CCN(C(=O)OCc2ccccc2)C1 ZINC000880794786 FE On-Demand Anodyne SLC12A5 52 35 Cc1ccc(C[C@@H](C)N(C)C(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880794798 FI On-Demand Anodyne NPY5R 25 45 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794806 GD On-Demand Anodyne ACOX1 51 36 COc1cccc(C2=NO[C@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794808 DD On-Demand Anodyne MTNR1A 54 37 COc1cccc(C2=NO[C@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794808 DD On-Demand Anodyne MTNR1B 46 37 COc1cccc(C2=NO[C@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794808 DD On-Demand Anodyne LUCI_PHOPY 37 46 COc1cccc(C2=NO[C@@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794809 DD On-Demand Anodyne MTNR1A 54 37 COc1cccc(C2=NO[C@@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794809 DD On-Demand Anodyne MTNR1B 46 37 COc1cccc(C2=NO[C@@H](C(=O)NCCc3cnoc3)C2)c1 ZINC000880794809 DD On-Demand Anodyne LUCI_PHOPY 37 46 CN(C)C(=O)C1(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)CCCC1 ZINC000880794830 GF On-Demand Anodyne PRMT3 58 31 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880794848 CD On-Demand Anodyne PAPA1_CARPA 41 44 CC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880794848 CD On-Demand Anodyne FPR1 43 34 Cc1cccc2c1CCN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)C2 ZINC000880794858 FH On-Demand Anodyne P2RY14 52 37 CN(CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C1CCCC1 ZINC000880794873 EF On-Demand Anodyne PRMT3 46 38 O=C(NCCc1cnoc1)[C@H](F)CC1CCCCC1 ZINC000880794876 CF On-Demand Anodyne MMP2 57 33 O=C(NCCc1cnoc1)[C@@H](F)CC1CCCCC1 ZINC000880794877 CF On-Demand Anodyne MMP2 57 33 CC(C)(C)OC(=O)N1CCc2cc(C(=O)NCCc3cnoc3)ccc21 ZINC000880794932 FF On-Demand Anodyne DRD4 40 32 C=C(C)CN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794944 FF On-Demand Mild EPHX2 38 41 C=C(C)CN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880794944 FF On-Demand Mild CXCR3 21 40 COc1cccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880794953 GG On-Demand Anodyne HRH2 41 51 COc1cccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880794953 GG On-Demand Anodyne CCR3 15 42 COc1cccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880794953 GG On-Demand Anodyne MTNR1A 33 46 COc1cccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880794953 GG On-Demand Anodyne MTNR1B 38 46 CC(C)(C)OC(=O)N1CCC(OCC(=O)NCCc2cnoc2)CC1 ZINC000880794989 FD On-Demand Anodyne GPR119 47 42 CCC(CC)[C@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795130 EF On-Demand Anodyne PRMT3 60 36 CCC(CC)[C@@H](O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795131 EF On-Demand Anodyne PRMT3 60 36 COc1ccccc1[C@@H]1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880795133 GH On-Demand Anodyne RBP4 26 41 COc1ccccc1[C@H]1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880795134 GH On-Demand Anodyne RBP4 26 41 O=C(NCCc1cnoc1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880795150 ED On-Demand Anodyne GRIN2B 29 47 O=C(NCCc1cnoc1)[C@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880795150 ED On-Demand Anodyne PREP 36 42 O=C(NCCc1cnoc1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880795151 ED On-Demand Anodyne GRIN2B 29 47 O=C(NCCc1cnoc1)[C@@H]1CCN(C(=O)OCc2ccccc2)C1 ZINC000880795151 ED On-Demand Anodyne PREP 36 42 CC(C)(C)OC(=O)N1CCCc2c(C(=O)NCCc3cnoc3)cccc21 ZINC000880795174 FG On-Demand Anodyne PANC 45 35 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne F2 73 43 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne PRSS1 22 40 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne ACE 33 45 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne FKBP1A 60 44 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne OPRM1 31 45 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne OPRD1 18 44 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne CELA1 28 56 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne ELANE 41 43 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne CTRA_BOVIN 63 34 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne TRY1_BOVIN 90 40 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne CTSG 43 34 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne DPP4 15 41 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne PREP 98 56 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne CELA2A 51 34 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne LGMN 91 51 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne KLK5 38 50 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne XIAP 43 48 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795211 EE On-Demand Anodyne TMPRSS11D 70 40 CCOc1cc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)ccc1OC ZINC000880795266 GG On-Demand Anodyne ROCK2 22 48 CCOc1cc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)ccc1OC ZINC000880795266 GG On-Demand Anodyne ENPP1 55 32 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne CTSD 15 42 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne PAPA1_CARPA 39 44 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne CTSL 16 44 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne TACR3 15 42 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne REN 58 38 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)Cc1ccccc1 ZINC000880795300 FF On-Demand Anodyne FPR1 49 39 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795315 ED On-Demand Anodyne PAPA1_CARPA 43 43 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795315 ED On-Demand Anodyne POLG_HCV1 33 44 CC(C)(C)OC(=O)N[C@@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795315 ED On-Demand Anodyne FPR1 47 36 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795316 ED On-Demand Anodyne PAPA1_CARPA 43 43 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795316 ED On-Demand Anodyne POLG_HCV1 33 44 CC(C)(C)OC(=O)N[C@H](CC(F)F)C(=O)NCCc1cnoc1 ZINC000880795316 ED On-Demand Anodyne FPR1 47 36 O=C(OCc1ccccc1)N1CC[C@](F)(C(=O)NCCc2cnoc2)C1 ZINC000880795350 FE On-Demand Anodyne SLC12A5 50 33 O=C(OCc1ccccc1)N1CC[C@@](F)(C(=O)NCCc2cnoc2)C1 ZINC000880795351 FE On-Demand Anodyne SLC12A5 50 33 CC(C)(C)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795355 DG On-Demand Anodyne PRMT3 58 35 COCCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880795359 FD On-Demand Anodyne EPHX2 52 40 COCCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880795359 FD On-Demand Anodyne CXCR3 21 41 COCCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795386 DF On-Demand Anodyne EPHX2 15 40 COCCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795386 DF On-Demand Anodyne PRMT3 58 33 O=C(NCCc1cnoc1)c1cc(S(=O)(=O)N2CCC2)ccc1Cl ZINC000880795437 FD On-Demand Anodyne NAMPT 37 42 COc1ccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880795446 GG On-Demand Anodyne ADRB1 17 42 COc1ccc(OCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880795446 GG On-Demand Anodyne HRH2 23 47 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880795464 ED On-Demand Anodyne PAPA1_CARPA 39 55 CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880795464 ED On-Demand Anodyne FPR1 50 47 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NCCc1cnoc1 ZINC000880795504 FD On-Demand Anodyne GRIN2B 18 43 O=C(CN1CCN(C(=O)OCc2ccccc2)CC1)NCCc1cnoc1 ZINC000880795504 FD On-Demand Anodyne TGM2 37 41 O=C(NCCc1cnoc1)[C@H](F)Cc1ccccc1 ZINC000880795509 CD On-Demand Anodyne MME 65 39 O=C(NCCc1cnoc1)[C@H](F)Cc1ccccc1 ZINC000880795509 CD On-Demand Anodyne ANPEP 30 40 O=C(NCCc1cnoc1)[C@H](F)Cc1ccccc1 ZINC000880795509 CD On-Demand Anodyne AMP1_PLAFQ 39 47 O=C(NCCc1cnoc1)[C@@H](F)Cc1ccccc1 ZINC000880795510 CD On-Demand Anodyne MME 65 39 O=C(NCCc1cnoc1)[C@@H](F)Cc1ccccc1 ZINC000880795510 CD On-Demand Anodyne ANPEP 30 40 O=C(NCCc1cnoc1)[C@@H](F)Cc1ccccc1 ZINC000880795510 CD On-Demand Anodyne AMP1_PLAFQ 39 47 O=C(NCCc1cnoc1)[C@H]1CCN(C2CCCCC2)C1 ZINC000880795520 CD On-Demand Anodyne GPBAR1 21 44 O=C(NCCc1cnoc1)[C@@H]1CCN(C2CCCCC2)C1 ZINC000880795521 CD On-Demand Anodyne GPBAR1 21 44 CC(C)(C)OC(=O)NC[C@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880795525 FF On-Demand Anodyne FPR1 45 35 CC(C)(C)OC(=O)NC[C@@H](C(=O)NCCc1cnoc1)c1ccccc1 ZINC000880795526 FF On-Demand Anodyne FPR1 45 35 C[C@@H]1CCCC[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795535 EH On-Demand Anodyne PRMT3 66 38 C[C@@H]1CCCC[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795538 EH On-Demand Anodyne PRMT3 66 38 CNC(=O)CCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795547 DC On-Demand Anodyne PRMT3 58 33 O=C(CC1CCCCC1)NCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795565 GF On-Demand Anodyne PRMT3 35 44 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne MME 85 38 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne ANPEP 43 31 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSD 21 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne PGC 63 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CMA1 43 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne FCER2 76 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSB 59 43 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne PAPA1_CARPA 93 62 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CYSP_TRYCR 69 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CCKAR 61 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSK 33 61 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSL 74 62 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne PGA 36 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne TIMP3 47 34 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne TACR3 28 55 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CAPNS1 64 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne MMP3 28 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne GRIA1 46 36 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne HLA-DRB1 61 47 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne REN 94 50 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne REN1 31 45 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CCKBR 22 49 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSS 33 62 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CAPN1 76 55 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne MMP9 19 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CAPN2 99 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne ACE2 42 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne SCN10A 19 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTSV 48 34 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne MMP1 27 41 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne FPR1 83 50 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne CTRB_BOVIN 30 42 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne NPR 50 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne AMP1_PLAFQ 29 40 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne PSMB5 43 35 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880795602 FE On-Demand Anodyne NPFFR1 44 31 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795612 GI On-Demand Anodyne TSHR 41 31 COc1ccccc1[C@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795613 GI On-Demand Anodyne TSHR 41 31 CC(C)(C)OC(=O)N[C@@H](CC(=O)NCCc1cnoc1)c1ccccc1 ZINC000880795639 FF On-Demand Anodyne FPR1 40 34 CC(C)(C)OC(=O)N[C@H](CC(=O)NCCc1cnoc1)c1ccccc1 ZINC000880795640 FF On-Demand Anodyne FPR1 40 34 COc1ccnc(N2CCN(C(=O)Nc3ccc4c(c3)SCC(=O)N4)CC2)c1 ZINC000880795651 GE On-Demand Anodyne PDGFRB 51 40 C[C@@H](CC(=O)NCCc1cnoc1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880795653 FG On-Demand Anodyne GPR119 44 47 C[C@H](CC(=O)NCCc1cnoc1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880795654 FG On-Demand Anodyne GPR119 44 47 CC(C)(C)OC(=O)N1CCC(CCC(=O)NCCc2cnoc2)CC1 ZINC000880795664 FF On-Demand Anodyne GPR119 49 42 Cc1noc(C)c1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795686 EF On-Demand Anodyne PRMT3 50 32 C[C@@H](CNC(=O)Nc1ccc2c(c1)SCC(=O)N2)C1CC1 ZINC000880795689 DF On-Demand Anodyne PRMT3 54 38 COc1ccccc1C[C@@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795703 GH On-Demand Anodyne TSHR 50 33 COc1ccccc1C[C@@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795703 GH On-Demand Anodyne ACKR3 63 33 COc1ccccc1C[C@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795704 GH On-Demand Anodyne TSHR 50 33 COc1ccccc1C[C@H]1CCCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795704 GH On-Demand Anodyne ACKR3 63 33 C[C@H](Sc1nc2ccccc2s1)C(=O)NCCc1cnoc1 ZINC000880795706 EG On-Demand Anodyne ST14 42 37 C[C@H](Sc1nc2ccccc2s1)C(=O)NCCc1cnoc1 ZINC000880795706 EG On-Demand Anodyne TMPRSS6 60 37 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCCc1cnoc1 ZINC000880795707 EG On-Demand Anodyne ST14 42 37 C[C@@H](Sc1nc2ccccc2s1)C(=O)NCCc1cnoc1 ZINC000880795707 EG On-Demand Anodyne TMPRSS6 60 37 CCN(Cc1ccc(OC)cc1)C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795729 FH On-Demand Anodyne ROCK2 15 43 COC[C@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795782 DE On-Demand Anodyne PRMT3 59 34 COC[C@@H](C)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795783 DE On-Demand Anodyne PRMT3 59 34 C[C@@H]1C[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795813 CF On-Demand Anodyne PRMT3 61 32 C[C@H]1C[C@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795815 CF On-Demand Anodyne PRMT3 61 32 C[C@@H]1C[C@@H]1CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795816 CF On-Demand Anodyne PRMT3 61 32 COC(=O)CCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880795872 FF On-Demand Anodyne EPHX2 19 42 O=C(NCCc1cnoc1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795873 FE On-Demand Anodyne GRIN2B 20 44 O=C(NCCc1cnoc1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795873 FE On-Demand Anodyne PREP 60 47 O=C(NCCc1cnoc1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795873 FE On-Demand Anodyne DPP7 55 40 O=C(NCCc1cnoc1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795873 FE On-Demand Anodyne GPBAR1 21 44 O=C(NCCc1cnoc1)[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795873 FE On-Demand Anodyne BIRC2 15 45 O=C(NCCc1cnoc1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795874 FE On-Demand Anodyne GRIN2B 20 44 O=C(NCCc1cnoc1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795874 FE On-Demand Anodyne PREP 60 47 O=C(NCCc1cnoc1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795874 FE On-Demand Anodyne DPP7 55 40 O=C(NCCc1cnoc1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795874 FE On-Demand Anodyne GPBAR1 21 44 O=C(NCCc1cnoc1)[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000880795874 FE On-Demand Anodyne BIRC2 15 45 C[C@H]1CCC[C@@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880795886 DG On-Demand Anodyne EPHX2 27 41 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne F2 73 43 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne PRSS1 22 40 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne ACE 33 45 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne FKBP1A 60 44 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne OPRM1 31 45 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne OPRD1 18 44 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne CELA1 28 56 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne ELANE 41 43 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne CTRA_BOVIN 63 34 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne TRY1_BOVIN 90 40 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne CTSG 43 34 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne DPP4 15 41 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne PREP 98 56 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne CELA2A 51 34 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne LGMN 91 51 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne KLK5 38 50 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne XIAP 43 48 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000880795953 EE On-Demand Anodyne TMPRSS11D 70 40 N#CCOc1cccc(CC(=O)NCCc2cnoc2)c1 ZINC000880795978 CD On-Demand Mild CRTM 41 37 O=C(Cc1ccc(S(=O)(=O)CC(F)(F)F)cc1)NCCc1cnoc1 ZINC000880796007 GD On-Demand Anodyne CA1 15 45 O=C(Cc1ccc(S(=O)(=O)CC(F)(F)F)cc1)NCCc1cnoc1 ZINC000880796007 GD On-Demand Anodyne CA5B 24 45 O=C(Cc1ccc(S(=O)(=O)CC(F)(F)F)cc1)NCCc1cnoc1 ZINC000880796007 GD On-Demand Anodyne CA5A 21 45 O=C(Cc1ccc(S(=O)(=O)CC(F)(F)F)cc1)NCCc1cnoc1 ZINC000880796007 GD On-Demand Anodyne CA9 18 41 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796036 EE On-Demand Anodyne CTSD 23 42 CC[C@@H](C)[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796036 EE On-Demand Anodyne ECE1 38 42 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796038 EE On-Demand Anodyne CTSD 23 42 CC[C@@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796038 EE On-Demand Anodyne ECE1 38 42 CC[C@H]1c2ccsc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796049 FI On-Demand Anodyne TRPM8 17 55 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796050 FI On-Demand Anodyne TRPM8 17 55 O=C(CCCn1ccnc1)NCCc1cnoc1 ZINC000880796060 BD On-Demand Anodyne TBXAS1 49 42 C/C(=C/C(=O)NCCc1cnoc1)c1cccc(C(F)(F)F)c1 ZINC000880796065 DG On-Demand Anodyne CCR2 40 33 CCOCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796073 DF On-Demand Anodyne EPHX2 15 40 CC(C)(C)OC(=O)N1CCC(n2cccc2C(=O)NCCc2cnoc2)CC1 ZINC000880796077 GG On-Demand Anodyne GPR119 42 39 COc1ccc([C@@H]2CCCN2C(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880796207 GI On-Demand Anodyne TSHR 40 30 O=C(Cc1ccncc1)NCCc1cnoc1 ZINC000880796225 BC On-Demand Anodyne CA5B 20 54 O=C(Cc1ccncc1)NCCc1cnoc1 ZINC000880796225 BC On-Demand Anodyne CA5A 18 54 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc3c(c2)SCC(=O)N3)on1 ZINC000880796232 FG On-Demand Anodyne KCNA5 17 43 O=C(NCCc1cnoc1)[C@@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880796244 ED On-Demand Anodyne LGMN 70 38 O=C(NCCc1cnoc1)[C@H]1CCCN1C(=O)OCC(F)(F)F ZINC000880796245 ED On-Demand Anodyne LGMN 70 38 O=C(NCCCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796269 DD On-Demand Anodyne FAAH 68 38 O=C(NCCCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796269 DD On-Demand Anodyne CES1 65 37 O=C(NCCCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796269 DD On-Demand Anodyne AMP1_PLAFQ 26 45 O=C(NCCCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796269 DD On-Demand Anodyne CRTM 34 41 O=C(Cc1csc(NC(=O)Cc2cccs2)n1)NCCc1cnoc1 ZINC000880796290 GE On-Demand Anodyne CA5B 39 46 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCc1cnoc1 ZINC000880796314 DD On-Demand Anodyne F2 30 41 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCc1cnoc1 ZINC000880796314 DD On-Demand Anodyne FKBP1A 28 42 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCc1cnoc1 ZINC000880796314 DD On-Demand Anodyne CMA1 27 40 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCc1cnoc1 ZINC000880796314 DD On-Demand Anodyne PREP 40 46 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCCc1cnoc1 ZINC000880796314 DD On-Demand Anodyne LGMN 54 34 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCc1cnoc1 ZINC000880796315 DD On-Demand Anodyne F2 30 41 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCc1cnoc1 ZINC000880796315 DD On-Demand Anodyne FKBP1A 28 42 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCc1cnoc1 ZINC000880796315 DD On-Demand Anodyne CMA1 27 40 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCc1cnoc1 ZINC000880796315 DD On-Demand Anodyne PREP 40 46 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCCc1cnoc1 ZINC000880796315 DD On-Demand Anodyne LGMN 54 34 CCOC(=O)N[C@@H](C(=O)NCCc1cnoc1)C(C)C ZINC000880796343 CD On-Demand Anodyne HLA-DRB1 63 40 CCOC(=O)N[C@H](C(=O)NCCc1cnoc1)C(C)C ZINC000880796344 CD On-Demand Anodyne HLA-DRB1 63 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne OPRD1 17 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CASP3 17 52 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne BMP1 26 58 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne KLK3 78 37 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CTSB 77 52 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne PAPA1_CARPA 86 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CYSP_TRYCR 55 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CTSK 42 56 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CTSL 53 52 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne PGA 22 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CAPNS1 71 46 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne HLA-DRB1 42 34 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne REN 17 41 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CTSS 20 56 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CAPN1 99 53 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CASP1 29 45 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CAPN2 155 50 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CASP6 15 42 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CASP9 33 42 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne TPSAB1 46 37 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne NPR 86 44 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne CASP10 34 40 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne PSMB5 55 46 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne F2RL1 71 36 CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880796374 FF On-Demand Anodyne Q6PRC7_IXORI 23 42 CN1CCC[C@H](NC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880796472 DD On-Demand Anodyne EPHX2 31 41 CC(=O)NCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796517 DD On-Demand Anodyne PRMT3 58 33 CCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796519 EE On-Demand Anodyne EPHX2 49 44 CCN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796519 EE On-Demand Anodyne CXCR3 22 41 O=C(NCCc1cnoc1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880796577 FE On-Demand Anodyne PREP 28 43 O=C(NCCc1cnoc1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880796577 FE On-Demand Anodyne Q9NAW4_PLAFA 38 44 C[C@@H](Cc1ccc(F)cc1)C(=O)NCCc1cnoc1 ZINC000880796584 CE On-Demand Anodyne LEF 45 33 CCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796598 CG On-Demand Anodyne EPHX2 15 51 CCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796598 CG On-Demand Anodyne ASAH1 61 33 CCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796598 CG On-Demand Anodyne PRMT3 58 33 CCOC(=O)N1CCC[C@@H](C(=O)NCCc2cnoc2)C1 ZINC000880796610 CD On-Demand Anodyne GPBAR1 23 43 CCOC(=O)N1CCC[C@H](C(=O)NCCc2cnoc2)C1 ZINC000880796611 CD On-Demand Anodyne GPBAR1 23 43 O=C(NCCc1cnoc1)[C@@H]1CC(c2cccc(F)c2)=NO1 ZINC000880796653 DD On-Demand Anodyne LUCI_PHOPY 24 44 O=C(NCCc1cnoc1)[C@H]1CC(c2cccc(F)c2)=NO1 ZINC000880796654 DD On-Demand Anodyne LUCI_PHOPY 24 44 COc1ccc2c(C)c(CCC(=O)NCCc3cnoc3)c(=O)oc2c1 ZINC000880796658 FE On-Demand Anodyne MAOB 38 45 COc1ccc2c(C)c(CCC(=O)NCCc3cnoc3)c(=O)oc2c1 ZINC000880796658 FE On-Demand Anodyne RAF1 22 40 COc1ccc2c(C)c(CCC(=O)NCCc3cnoc3)c(=O)oc2c1 ZINC000880796658 FE On-Demand Anodyne MTNR1A 62 43 COc1ccc2c(C)c(CCC(=O)NCCc3cnoc3)c(=O)oc2c1 ZINC000880796658 FE On-Demand Anodyne MTNR1B 54 43 COc1ccc2c(C)c(CCC(=O)NCCc3cnoc3)c(=O)oc2c1 ZINC000880796658 FE On-Demand Anodyne NQO1 30 44 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796660 ED On-Demand Anodyne PAPA1_CARPA 39 55 CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796660 ED On-Demand Anodyne FPR1 50 47 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796676 DE On-Demand Anodyne PAPA1_CARPA 41 54 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796676 DE On-Demand Anodyne CTSK 23 41 CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880796676 DE On-Demand Anodyne FPR1 43 36 CC(C)(C)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796684 FG On-Demand Anodyne EPHX2 46 42 CN1CC[C@H](C(=O)NCCc2cnoc2)C1 ZINC000880796712 BC On-Demand Anodyne GPBAR1 25 42 CN1CC[C@@H](C(=O)NCCc2cnoc2)C1 ZINC000880796713 BC On-Demand Anodyne GPBAR1 25 42 CCOC(=O)N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796755 FE On-Demand Anodyne TGM2 17 41 CCOC(=O)N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796755 FE On-Demand Anodyne F13A1 33 41 O=C(CCn1c(S)nnc1-c1cccs1)NCCc1cnoc1 ZINC000880796783 EE On-Demand Anodyne GPR142 40 31 COCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880796818 CD On-Demand Anodyne PRMT3 60 34 O=C(NCCc1cnoc1)c1ccc(N2CCCS2(=O)=O)cc1Cl ZINC000880796866 FD On-Demand Anodyne CDK1 16 40 CCCNC(=O)c1cccc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880796880 GG On-Demand Anodyne ROCK2 24 45 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA2 15 47 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA1 17 47 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA5B 28 46 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA5A 26 46 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA12 15 47 O=C(Cc1ccc(S(=O)(=O)C(F)F)cc1)NCCc1cnoc1 ZINC000880796903 ED On-Demand Anodyne CA9 19 42 COc1ccc(CN(C)C(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1OC ZINC000880796920 GG On-Demand Anodyne MT-ND1 17 40 COc1ccc(CN(C)C(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1OC ZINC000880796920 GG On-Demand Anodyne ENPP1 61 32 CC(C)CN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796942 FF On-Demand Anodyne EPHX2 43 43 CC(C)CN1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880796942 FF On-Demand Anodyne CXCR3 21 42 C[C@H]1C[C@@H](C)CN(CCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880796946 GH On-Demand Anodyne CCR3 36 40 C[C@@H]1C[C@@H](C)CN(CCCCNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880796948 GH On-Demand Anodyne CCR3 36 40 O=C(COc1cccc(C(F)(F)F)c1)NCCc1cnoc1 ZINC000880796970 DE On-Demand Anodyne PDS 49 47 O=C1CCCc2cc(C(=O)NCCc3cnoc3)ccc2N1 ZINC000880796986 CD On-Demand Anodyne HDAC9 18 48 O=C(NCCc1cnoc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl ZINC000880796987 GE On-Demand Anodyne NAMPT 39 46 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnoc1)C2 ZINC000880796990 DE On-Demand Anodyne NQO2 39 43 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnoc1)C2 ZINC000880796990 DE On-Demand Anodyne MTNR1A 79 45 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnoc1)C2 ZINC000880796990 DE On-Demand Anodyne MTNR1B 66 41 CC(C)(C)OC(=O)N1CCC(CC(=O)NCCc2cnoc2)CC1 ZINC000880797010 EE On-Demand Anodyne GPR119 48 41 CCCCCCCC(=O)NCCc1cnoc1 ZINC000880797011 BF On-Demand Mild NOD1 54 40 CCCCCCCC(=O)NCCc1cnoc1 ZINC000880797011 BF On-Demand Mild CQSS 41 31 O=C(NCCc1cnoc1)c1cc2ccccc2cc1NC(=O)C1CC1 ZINC000880797048 EG On-Demand Anodyne NMT1 35 40 CCOC(=O)CCCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880797062 GG On-Demand Anodyne EPHX2 18 45 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880797093 GG On-Demand Anodyne ABCB1 15 41 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc3c(c1)SCC(=O)N3)CC2 ZINC000880797093 GG On-Demand Anodyne ABCG2 24 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797114 GF On-Demand Anodyne TGM1 15 45 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797114 GF On-Demand Anodyne F13A1 25 45 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797114 GF On-Demand Anodyne GPR119 23 41 COCCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880797116 DE On-Demand Anodyne PRMT3 59 33 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880797144 EE On-Demand Anodyne QPCT 19 40 CNC(=O)CNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880797147 CC On-Demand Anodyne PRMT3 62 34 CCOc1ccc([C@@H](C)NC(=O)Nc2ccc3c(c2)SCC(=O)N3)cc1 ZINC000880797159 FI On-Demand Anodyne ACACB 19 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne ACE 21 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne OPRM1 22 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne OPRD1 27 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CELA1 16 55 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne MME 38 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CASP3 17 49 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne BMP1 20 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne KLK3 81 39 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CTSB 80 50 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne PAPA1_CARPA 83 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CYSP_TRYCR 58 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CTSK 46 50 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CTSL 54 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne PGA 29 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CAPNS1 74 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne MMP3 15 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne HLA-DRB1 68 38 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CTSS 26 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CAPN1 100 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CASP1 36 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CAPN2 157 48 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CASP6 15 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne CASP9 30 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne TPSAB1 46 49 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne NPR 93 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne NAAA 54 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne PSMB5 61 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)NCCc1cnoc1 ZINC000880797254 DD On-Demand Anodyne Q6PRC7_IXORI 43 39 O=C(NCCc1cnoc1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880797278 EE On-Demand Anodyne P2RX7 15 52 O=C(NCCc1cnoc1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880797279 EE On-Demand Anodyne P2RX7 15 52 CCCOc1ccc(OCC(=O)NCCc2cnoc2)cc1 ZINC000880797287 DE On-Demand Anodyne MTNR1A 34 42 CCCOc1ccc(OCC(=O)NCCc2cnoc2)cc1 ZINC000880797287 DE On-Demand Anodyne PLA2G4B 79 35 O=C(CCCNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797298 EE On-Demand Anodyne CAPN1 36 46 O=C(CCCNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797298 EE On-Demand Anodyne CAPN2 66 46 O=C(CCCNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797298 EE On-Demand Anodyne NPR 60 39 O=C(NCCc1cnoc1)c1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 ZINC000880797307 GE On-Demand Anodyne NAMPT 27 42 O=C(NCCc1cnoc1)c1cc(S(=O)(=O)N2CCCC2)ccc1Cl ZINC000880797309 GE On-Demand Anodyne NAMPT 38 44 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880797333 GF On-Demand Anodyne MTNR1B 29 41 O=C(Cc1cccs1)NCCc1cnoc1 ZINC000880797380 BD On-Demand Anodyne CA5B 45 58 O=C(Cc1cccs1)NCCc1cnoc1 ZINC000880797380 BD On-Demand Anodyne CA5A 43 45 CCN1CC[C@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880797395 EE On-Demand Anodyne CCR3 54 36 CCN1CC[C@H](CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)C1 ZINC000880797395 EE On-Demand Anodyne CACNA1I 41 31 CCOC(=O)N1CCC(NC(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797431 GE On-Demand Anodyne EPHX2 60 46 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@@H](N2CCOCC2)C1 ZINC000880797445 GE On-Demand Anodyne L3MBTL3 47 38 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@H](N2CCOCC2)C1 ZINC000880797447 GE On-Demand Anodyne L3MBTL3 47 38 CCN(CC)Cc1cccc(CNC(=O)Nc2ccc3c(c2)SCC(=O)N3)c1 ZINC000880797468 GH On-Demand Anodyne ROCK2 22 41 CC(C)(C)OC(=O)N1CCC[C@H](C(=O)NCCc2cnoc2)C1 ZINC000880797471 DD On-Demand Anodyne GPBAR1 23 42 C[C@H](NC(=O)OC(C)(C)C)C(=O)NCCc1cnoc1 ZINC000880797490 CD On-Demand Anodyne FPR1 37 40 O=C(NCCc1cnoc1)[C@@H]1CC(c2ccccc2)=NO1 ZINC000880797616 CD On-Demand Anodyne LUCI_PHOPY 51 39 O=C(NCCc1cnoc1)[C@H]1CC(c2ccccc2)=NO1 ZINC000880797619 CD On-Demand Anodyne LUCI_PHOPY 51 39 CCCCNC(=O)Nc1ccc2c(c1)SCC(=O)N2 ZINC000880797666 CF On-Demand Anodyne PRMT3 59 33 CC(C)(C)OC(=O)N1CCC(C(=O)NCCc2cnoc2)CC1 ZINC000880797679 DD On-Demand Anodyne GPR119 47 42 CCCCSCC(=O)NCCc1cnoc1 ZINC000880797702 BD On-Demand Anodyne EST1_PIG 40 34 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CTSB 37 42 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne PAPA1_CARPA 43 34 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CTSK 42 44 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CTSL 36 44 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CAPNS1 58 42 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne HLA-DRB1 46 34 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CTSS 26 44 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CAPN1 90 43 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne CAPN2 129 42 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne FPR1 56 35 COC(=O)N[C@H](CC(C)C)C(=O)NCCc1cnoc1 ZINC000880797704 CD On-Demand Anodyne NPR 78 41 O=C(NCCc1cnoc1)c1ccc(N2CCOCC2)nc1 ZINC000880797720 DC On-Demand Anodyne HPGDS 33 50 CCCCCCCCC(=O)NCCc1cnoc1 ZINC000880797724 CG On-Demand Mild NOD1 54 40 CCCCCCCCC(=O)NCCc1cnoc1 ZINC000880797724 CG On-Demand Mild CQSS 41 31 O=C(NCCc1cnoc1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880797821 FE On-Demand Anodyne GRIN2B 27 48 O=C(NCCc1cnoc1)C1CCN(C(=O)OCc2ccccc2)CC1 ZINC000880797821 FE On-Demand Anodyne PREP 41 43 Cc1cc(C(=O)NCCc2cnoc2)cc(C)c1OCc1cccnc1 ZINC000880797825 FG On-Demand Anodyne TBXAS1 21 43 Cc1cc(C(=O)NCCc2cnoc2)cc(C)c1OCc1cccnc1 ZINC000880797825 FG On-Demand Anodyne PTAFR 21 47 CN1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797844 DD On-Demand Anodyne HTR1B 16 46 O=C(NCCc1cnoc1)[C@@H]1CC(=O)N(C2CCCC2)C1 ZINC000880797848 CD On-Demand Anodyne INHA 20 45 O=C(NCCc1cnoc1)[C@H]1CC(=O)N(C2CCCC2)C1 ZINC000880797849 CD On-Demand Anodyne INHA 20 45 O=C(NCC(=O)N1CCN(Cc2cccc3cccnc23)CC1)c1ccccc1OC(F)F ZINC000880797865 JF On-Demand Anodyne SCD 20 40 O=C(NCC(=O)N1CCN(Cc2cccc3cccnc23)CC1)c1ccccc1OC(F)F ZINC000880797865 JF On-Demand Anodyne HCN1 41 31 O=C(NCCc1cnoc1)[C@@H]1CSCN1C(=O)c1ccccc1 ZINC000880797868 ED On-Demand Anodyne PREP 17 40 O=C(NCCc1cnoc1)[C@H]1CSCN1C(=O)c1ccccc1 ZINC000880797869 ED On-Demand Anodyne PREP 17 40 O=C(NCCc1cnoc1)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 ZINC000880797876 GE On-Demand Anodyne NAMPT 25 43 CCCCCCC(=O)NCCc1cnoc1 ZINC000880797880 BE On-Demand Anodyne NOD1 54 40 CCCCCCC(=O)NCCc1cnoc1 ZINC000880797880 BE On-Demand Anodyne CQSS 41 31 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne HTR1A 94 64 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne DRD2 67 43 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne DRD4 35 46 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne ADRA1D 78 46 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne HTR1D 23 64 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne HTR1B 29 64 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne HTR2A 23 51 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne ADRA1A 71 46 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne ADRA1B 62 46 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne DRD3 68 43 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne PDGFRB 59 45 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne HTR7 56 56 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne NPY2R 34 41 COc1ccccc1N1CCN(C(=O)Nc2ccc3c(c2)SCC(=O)N3)CC1 ZINC000880797901 GG On-Demand Anodyne RBP4 18 47 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne CTSB 24 45 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne CTSK 15 45 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne CAPNS1 43 37 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne CAPN2 73 37 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne TPSAB1 20 44 O=C(CNC(=O)OCc1ccccc1)NCCc1cnoc1 ZINC000880797904 DD On-Demand Anodyne NPR 63 41 C[S@@](=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880797921 ED On-Demand Anodyne MTNR1B 37 40 CCNC(=O)CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798027 ED On-Demand Anodyne MTNR1B 37 40 CN(C[C@H]1CCCN1C)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798092 FF On-Demand Anodyne ACKR3 60 29 CN(C[C@@H]1CCCN1C)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798093 FF On-Demand Anodyne ACKR3 60 29 C/C=C\CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798116 DG On-Demand Anodyne MTNR1B 37 40 C/C=C/CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798117 DG On-Demand Anodyne MTNR1B 37 40 CN(C)C1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880798141 GG On-Demand Anodyne MTNR1A 15 42 Cc1ccncc1CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798414 GG On-Demand Anodyne MTNR1A 31 40 Cc1ccncc1CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798414 GG On-Demand Anodyne MTNR1B 37 40 C=CCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798545 DG On-Demand Mild MTNR1B 37 40 C[C@@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)N(C)C ZINC000880798552 FF On-Demand Anodyne MTNR1B 38 42 C[C@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)N(C)C ZINC000880798553 FF On-Demand Anodyne MTNR1B 38 42 CC(=O)N[C@H]1CCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880798556 FE On-Demand Anodyne MTNR1A 24 54 CC(=O)N[C@@H]1CCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880798557 FE On-Demand Anodyne MTNR1A 24 54 O=C(Nc1c(Br)ccc2c1CCO2)N[C@H]1CCOC1=O ZINC000880798579 ED On-Demand Anodyne LUXR 74 40 O=C(Nc1c(Br)ccc2c1CCO2)N[C@H]1CCOC1=O ZINC000880798579 ED On-Demand Anodyne TRAR 89 45 O=C(Nc1c(Br)ccc2c1CCO2)N[C@H]1CCOC1=O ZINC000880798579 ED On-Demand Anodyne LASR 59 42 C=C(C)CN(C)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798589 EG On-Demand Mild MTNR1B 36 40 CC(=O)NCCN(C)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798626 FD On-Demand Anodyne MTNR1A 34 45 CC(=O)NCCN(C)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798626 FD On-Demand Anodyne MTNR1B 42 48 O=C(Nc1c(Br)ccc2c1CCO2)NC1CCC1 ZINC000880798734 DG On-Demand Anodyne MTNR1A 16 43 C[C@H](CCO)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798736 FF On-Demand Anodyne MTNR1B 37 40 C[C@@H](CCO)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798737 FF On-Demand Anodyne MTNR1B 37 40 CO[C@@H](C)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880798739 EF On-Demand Anodyne MTNR1B 38 40 O=C(NCCF)Nc1c(Br)ccc2c1CCO2 ZINC000880798743 DE On-Demand Anodyne MTNR1B 37 40 COC(=O)N1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880798746 GF On-Demand Anodyne MTNR1A 16 44 COC(=O)N1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880798746 GF On-Demand Anodyne MTNR1B 17 42 COC(=O)N1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880798746 GF On-Demand Anodyne EPHX2 33 40 Cc1nnc(CCNC(=O)Nc2c(Br)ccc3c2CCO3)s1 ZINC000880798798 GF On-Demand Anodyne MTNR1B 37 40 CCN1C[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)CC1=O ZINC000880798799 FE On-Demand Anodyne MTNR1A 24 42 CCN1C[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)CC1=O ZINC000880798799 FE On-Demand Anodyne MTNR1B 25 42 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1c(Br)ccc3c1CCO3)C2 ZINC000880798813 GG On-Demand Anodyne MTNR1A 19 42 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1c(Br)ccc3c1CCO3)C2 ZINC000880798813 GG On-Demand Anodyne MTNR1B 21 42 C=C(C)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799107 EG On-Demand Mild MTNR1B 40 44 CC(=O)NNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799227 DD On-Demand Reactive MTNR1B 37 42 CN(C)S(=O)(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799437 GD On-Demand Anodyne MTNR1B 37 41 Cn1nccc1CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799548 FE On-Demand Anodyne MTNR1B 41 45 O=C(NCCN1CCCOCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880799558 GE On-Demand Anodyne EPHX2 17 44 CCNC(=O)C(C)(C)NC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799635 FE On-Demand Anodyne MTNR1B 38 41 C[C@@H](O)CCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799776 EF On-Demand Anodyne MTNR1B 38 40 O=C(Nc1c(Br)ccc2c1CCO2)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880799834 GG On-Demand Anodyne CPT1A 45 35 O=C(Nc1c(Br)ccc2c1CCO2)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880799835 GG On-Demand Anodyne CPT1A 45 35 O=C(NCCc1cnccn1)Nc1c(Br)ccc2c1CCO2 ZINC000880799839 FF On-Demand Anodyne MTNR1A 30 40 O=C(NCCc1cnccn1)Nc1c(Br)ccc2c1CCO2 ZINC000880799839 FF On-Demand Anodyne MTNR1B 37 40 Cn1cnc(CCNC(=O)Nc2c(Br)ccc3c2CCO3)c1 ZINC000880799910 FE On-Demand Anodyne MTNR1A 34 40 Cn1cnc(CCNC(=O)Nc2c(Br)ccc3c2CCO3)c1 ZINC000880799910 FE On-Demand Anodyne MTNR1B 38 40 Cc1cnc(CCNC(=O)Nc2c(Br)ccc3c2CCO3)cn1 ZINC000880799912 GF On-Demand Anodyne MTNR1B 38 40 C[C@@H](F)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880799920 EG On-Demand Anodyne MTNR1B 38 41 CCNC(=O)C(C)(C)CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880800075 GF On-Demand Anodyne MTNR1B 37 40 O=C(CNC(=O)Nc1c(Br)ccc2c1CCO2)NCCO ZINC000880800157 FC On-Demand Anodyne MTNR1B 38 40 O=C(COc1ccccc1O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880800324 GF On-Demand Anodyne HTR1B 15 43 O=C(COc1ccccc1O)N1CCN(Cc2cccc3cccnc23)CC1 ZINC000880800324 GF On-Demand Anodyne CCR8 30 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880800326 GF On-Demand Anodyne MTNR1A 19 46 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880800326 GF On-Demand Anodyne MTNR1B 21 46 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880800327 GF On-Demand Anodyne MTNR1A 19 46 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880800327 GF On-Demand Anodyne MTNR1B 21 46 CCC(=O)NNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880800328 ED On-Demand Reactive MTNR1A 34 42 CCC(=O)NNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880800328 ED On-Demand Reactive MTNR1B 37 42 O=C(NCCc1ccc(CO)cc1)Nc1c(Br)ccc2c1CCO2 ZINC000880800348 GG On-Demand Anodyne MTNR1B 38 41 C=C(C)CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880800366 DG On-Demand Mild MTNR1B 37 41 O=C(NNC(=O)C1CC1)Nc1c(Br)ccc2c1CCO2 ZINC000880800480 ED On-Demand Reactive MTNR1A 16 42 Cc1ncc(CCNC(=O)Nc2c(Br)ccc3c2CCO3)s1 ZINC000880800512 GH On-Demand Anodyne MTNR1B 38 40 Cc1ccc2ccnc(NC(=O)C3CCC(S(C)(=O)=O)CC3)c2c1 ZINC000880800530 EG On-Demand Anodyne GSK3B 21 45 Cc1ccc2ccnc(NC(=O)C3CCC(S(C)(=O)=O)CC3)c2c1 ZINC000880800530 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1c(Br)ccc2c1CCO2)N[C@H]1CCCOCC1 ZINC000880800574 FG On-Demand Anodyne MTNR1A 15 40 O=C(Nc1c(Br)ccc2c1CCO2)N[C@@H]1CCCOCC1 ZINC000880800575 FG On-Demand Anodyne MTNR1A 15 40 O=C(NCCCNC(=O)C1CCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880800585 GF On-Demand Anodyne MTNR1A 26 42 O=C(NCCCNC(=O)C1CCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880800585 GF On-Demand Anodyne MTNR1B 26 42 O=C(NCCCNC(=O)C1CCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880800585 GF On-Demand Anodyne TBK1 57 36 O=C(Nc1c(Br)ccc2c1CCO2)N1CCN2CCCC[C@@H]2C1 ZINC000880800638 GG On-Demand Anodyne L3MBTL3 57 38 O=C(Nc1c(Br)ccc2c1CCO2)N1CCN2CCCC[C@H]2C1 ZINC000880800639 GG On-Demand Anodyne L3MBTL3 57 38 COc1ccc2c(c1)CC[C@H](C(=O)NNc1ncc(Cl)cn1)C2 ZINC000880800689 EE On-Demand Reactive FAAH 15 43 O=C(Nc1c(Br)ccc2c1CCO2)NC1CCCC1 ZINC000880800742 EG On-Demand Anodyne MTNR1A 15 43 Cc1cnc(Cl)c(C(=O)N2CCN(c3ccc(F)cc3C(N)=O)CC2)c1 ZINC000880800744 GE On-Demand Anodyne HCRTR1 44 45 Cc1cnc(Cl)c(C(=O)N2CCN(c3ccc(F)cc3C(N)=O)CC2)c1 ZINC000880800744 GE On-Demand Anodyne HCRTR2 29 45 COCCN1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880800762 GF On-Demand Anodyne HTR4 17 44 COCCN1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880800762 GF On-Demand Anodyne MTNR1B 15 41 O=C(Nc1ccc(Br)c(Br)c1)N1CCC(O)CC1 ZINC000880800769 GG On-Demand Anodyne EPHX2 28 41 O=C(NCCCN1CCOCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880800837 GE On-Demand Anodyne EPHX2 22 42 O=C(Nc1c(Br)ccc2c1CCO2)N1CCN(C2CCC2)CC1 ZINC000880800943 GG On-Demand Anodyne L3MBTL3 46 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC1(Cl)Cl ZINC000880800950 FF On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC1(Cl)Cl ZINC000880800952 FF On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC1(Cl)Cl ZINC000880800953 FF On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC1(Cl)Cl ZINC000880800954 FF On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)C[C@H]1Br ZINC000880801029 GE On-Demand Reactive PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)C[C@@H]1Br ZINC000880801033 GE On-Demand Reactive PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)C[C@H]1Br ZINC000880801034 GE On-Demand Reactive PAPA1_CARPA 39 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)C[C@@H]1Br ZINC000880801035 GE On-Demand Reactive PAPA1_CARPA 39 47 Cc1cnc(Cl)c(C(=O)NCC2CC(C)C2)c1 ZINC000880801051 CF On-Demand Anodyne CACNA1I 53 37 O=C(NCCC1CC1)Nc1c(Br)ccc2c1CCO2 ZINC000880801054 EG On-Demand Anodyne MTNR1A 32 43 O=C(NCCC1CC1)Nc1c(Br)ccc2c1CCO2 ZINC000880801054 EG On-Demand Anodyne MTNR1B 37 43 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@@H](O)C1 ZINC000880801107 GG On-Demand Anodyne EPHX2 24 43 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@H](O)C1 ZINC000880801109 GG On-Demand Anodyne EPHX2 24 43 O=C(NCCO)Nc1c(Br)ccc2c1CCO2 ZINC000880801128 DD On-Demand Anodyne MTNR1A 32 40 O=C(NCCO)Nc1c(Br)ccc2c1CCO2 ZINC000880801128 DD On-Demand Anodyne MTNR1B 39 43 O=C(NCCCn1ccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880801157 FF On-Demand Anodyne TBXAS1 33 45 O=C(NCCCn1ccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880801157 FF On-Demand Anodyne QPCT 47 47 Cc1ccc2ccnc(NC(=O)c3ccc(CN4CCOCC4)o3)c2c1 ZINC000880801159 FG On-Demand Anodyne EPHB4 47 37 O=C(Nc1c(Br)ccc2c1CCO2)NC1CC1 ZINC000880801192 CF On-Demand Anodyne MTNR1A 17 47 CCCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801231 DG On-Demand Anodyne MTNR1B 38 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MMP13 25 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MTNR1A 29 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MTNR1B 26 47 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MMP3 33 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MMP9 22 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne EPHX2 27 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MMP7 28 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)C2 ZINC000880801237 DD On-Demand Anodyne MMP1 28 42 CC[C@H](C)NC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801240 GF On-Demand Anodyne MTNR1A 33 43 CC[C@H](C)NC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801240 GF On-Demand Anodyne MTNR1B 39 43 O=C(Nc1c(Br)ccc2c1CCO2)NC1CCOCC1 ZINC000880801261 EF On-Demand Anodyne MTNR1A 17 43 C[C@H]1CCN(C(=O)c2ncccc2-c2ccccn2)C[C@H]1CO ZINC000880801296 DE On-Demand Anodyne MLNR 19 42 C[C@@H]1CCN(C(=O)c2ncccc2-c2ccccn2)C[C@H]1CO ZINC000880801297 DE On-Demand Anodyne MLNR 19 42 C[C@H]1CCN(C(=O)c2ncccc2-c2ccccn2)C[C@@H]1CO ZINC000880801298 DE On-Demand Anodyne MLNR 19 42 C[C@@H]1CCN(C(=O)c2ncccc2-c2ccccn2)C[C@@H]1CO ZINC000880801299 DE On-Demand Anodyne MLNR 19 42 Cc1nc(C(C)C)ncc1C(=O)N1CCN(c2ccc(F)cc2C(N)=O)CC1 ZINC000880801319 GE On-Demand Anodyne HCRTR1 18 43 NC(=O)c1cc(F)ccc1N1CCN(C(=O)COC2CC2)CC1 ZINC000880801320 DC On-Demand Anodyne LIPG 48 41 NC(=O)c1cc(F)ccc1N1CCN(C(=O)c2cnc(CC3CC3)s2)CC1 ZINC000880801322 GE On-Demand Anodyne SCD1 21 41 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C(C)=O)C2)c(O)n1 ZINC000880801325 FD On-Demand Anodyne DRD2 22 40 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C(C)=O)C2)c(O)n1 ZINC000880801325 FD On-Demand Anodyne HTR3A 23 43 C=CCCC[C@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)c1ccccc1 ZINC000880801330 DF On-Demand Mild C3AR1 30 40 C=CCCC[C@@H](C(=O)N[C@@H]1CCN(C(C)=O)C1)c1ccccc1 ZINC000880801331 DF On-Demand Mild C3AR1 30 40 CC(=O)NCC1CCN(C(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880801341 GF On-Demand Anodyne MTNR1B 37 42 O=C(Nc1ccc(Br)c(Br)c1)NC1CCOCC1 ZINC000880801355 GH On-Demand Anodyne EPHX2 55 46 O=C(Nc1ccc(Br)c(Br)c1)N1CCCC1 ZINC000880801400 EH On-Demand Anodyne EPHX2 26 49 O=C(Nc1ccc(Br)c(Br)c1)N1CCC(CO)CC1 ZINC000880801402 GG On-Demand Anodyne EPHX2 29 57 O=C(Nc1ccc(Br)c(Br)c1)N1CCOCC1 ZINC000880801403 FG On-Demand Anodyne EPHX2 40 46 CNC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801410 ED On-Demand Anodyne MTNR1B 40 45 CC(=O)NC[C@@H]1CN(C(=O)Nc2c(Br)ccc3c2CCO3)CCO1 ZINC000880801496 GD On-Demand Anodyne MTNR1B 36 42 CC(C)(C)C(=O)NCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801498 GF On-Demand Anodyne MTNR1B 38 40 CCNC(=O)CNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880801592 GE On-Demand Anodyne F7 25 41 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@@H](CO)C1 ZINC000880801596 GG On-Demand Anodyne CCR3 20 41 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@@H](CO)C1 ZINC000880801596 GG On-Demand Anodyne EPHX2 18 60 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@H](CO)C1 ZINC000880801597 GG On-Demand Anodyne CCR3 20 41 O=C(Nc1ccc(Br)c(Br)c1)N1CCC[C@H](CO)C1 ZINC000880801597 GG On-Demand Anodyne EPHX2 18 60 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@@H](N2CCCCC2)C1 ZINC000880801599 GG On-Demand Anodyne L3MBTL3 96 44 CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801600 CE On-Demand Anodyne MTNR1A 31 40 CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801600 CE On-Demand Anodyne MTNR1B 35 41 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@H](N2CCCCC2)C1 ZINC000880801604 GG On-Demand Anodyne L3MBTL3 96 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880801617 EC On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880801619 EC On-Demand Anodyne PAPA1_CARPA 33 41 O=C(NCCn1ccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880801641 FE On-Demand Anodyne QPCT 32 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC(CC2CC2)C1 ZINC000880801643 FH On-Demand Anodyne P2RX7 40 35 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC(CC2CC2)C1 ZINC000880801643 FH On-Demand Anodyne RBP4 56 31 CNC(=O)CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801651 ED On-Demand Anodyne MTNR1B 37 41 O=C(Nc1c(Br)ccc2c1CCO2)NC1CCN(CCO)CC1 ZINC000880801670 GD On-Demand Anodyne MTNR1B 15 44 CCn1cc(NC(=O)Nc2c(Br)ccc3c2CCO3)cn1 ZINC000880801696 FG On-Demand Anodyne PANC 45 34 COc1ccccc1-c1ccc(C(=O)NCC[C@@H]2CC2(Cl)Cl)c(O)n1 ZINC000880801710 GH On-Demand Anodyne KCNA3 40 35 COc1ccccc1-c1ccc(C(=O)NCC[C@H]2CC2(Cl)Cl)c(O)n1 ZINC000880801714 GH On-Demand Anodyne KCNA3 40 35 CC1CC(CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880801722 ED On-Demand Anodyne F2 26 40 COc1ccccc1-c1ccc(C(=O)NCC2CC(C)C2)c(O)n1 ZINC000880801731 EG On-Demand Anodyne DRD2 24 42 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@@H](N2CCCC2)C1 ZINC000880801747 GG On-Demand Anodyne L3MBTL3 92 44 O=C(Nc1c(Br)ccc2c1CCO2)N1CC[C@H](N2CCCC2)C1 ZINC000880801748 GG On-Demand Anodyne L3MBTL3 92 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801754 GF On-Demand Anodyne MTNR1B 29 41 O=C(NCCNC(=O)C1CC1)Nc1c(Br)ccc2c1CCO2 ZINC000880801764 FE On-Demand Anodyne MTNR1A 38 47 O=C(NCCNC(=O)C1CC1)Nc1c(Br)ccc2c1CCO2 ZINC000880801764 FE On-Demand Anodyne MTNR1B 37 47 CCN1CC[C@H](CNC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801765 FF On-Demand Anodyne CACNA1I 45 32 CN(C)C(=O)CCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801778 FE On-Demand Anodyne MTNR1B 37 41 CN1CCC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801827 FF On-Demand Anodyne MTNR1A 15 45 CN1CCC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801827 FF On-Demand Anodyne MTNR1B 15 45 CC[C@H]1CCC[C@]1(C)C(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880801837 CD On-Demand Anodyne EPHX2 16 49 CC[C@H]1CCC[C@@]1(C)C(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880801838 CD On-Demand Anodyne EPHX2 16 49 CC[C@@H]1CCC[C@@]1(C)C(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880801840 CD On-Demand Anodyne EPHX2 16 49 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC(CC2CC2)C1 ZINC000880801846 DH On-Demand Anodyne PDE4D 27 44 O=C(NCCN1CCOCC1)Nc1c(Br)ccc2c1CCO2 ZINC000880801857 FD On-Demand Anodyne EPHX2 20 47 O=C(C(=O)N1CC(CC2CC2)C1)c1c[nH]c2cc(F)ccc12 ZINC000880801859 DF On-Demand Anodyne GRIN2B 15 59 O=C(C(=O)N1CC(CC2CC2)C1)c1c[nH]c2cc(F)ccc12 ZINC000880801859 DF On-Demand Anodyne MPO 53 35 C=CC(C)(C)CC(=O)NCc1cc(OC)ccc1F ZINC000880801903 CG On-Demand Mild MTNR1A 75 36 C=CC(C)(C)CC(=O)NCc1cc(OC)ccc1F ZINC000880801903 CG On-Demand Mild MTNR1B 62 40 NC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801930 ED On-Demand Anodyne MTNR1B 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801933 FF On-Demand Anodyne GHRHR 47 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801933 FF On-Demand Anodyne P2RY12 89 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801933 FF On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801933 FF On-Demand Anodyne CTSK 23 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801933 FF On-Demand Anodyne FPR1 49 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801934 FF On-Demand Anodyne GHRHR 47 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801934 FF On-Demand Anodyne P2RY12 89 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801934 FF On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801934 FF On-Demand Anodyne CTSK 23 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(C)(c2ccccc2)C1 ZINC000880801934 FF On-Demand Anodyne FPR1 49 36 O=C(CN1CCCCS1(=O)=O)Nc1nc2cc(Cl)c(F)cc2[nH]1 ZINC000880801950 FD On-Demand Anodyne NR2E3 51 34 COCCn1cc(NC(=O)Nc2c(Br)ccc3c2CCO3)cn1 ZINC000880801968 GF On-Demand Anodyne PANC 50 35 C[C@@H]1C[C@H]1CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801986 EG On-Demand Anodyne MTNR1B 35 40 C[C@H]1C[C@H]1CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801988 EG On-Demand Anodyne MTNR1B 35 40 C[C@@H]1C[C@@H]1CNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880801989 EG On-Demand Anodyne MTNR1B 35 40 O=C(Nc1c(Br)ccc2c1CCO2)N1CCC[C@@H](N2CCCC2)C1 ZINC000880801990 GG On-Demand Anodyne L3MBTL3 64 39 O=C(Nc1c(Br)ccc2c1CCO2)N1CCC[C@H](N2CCCC2)C1 ZINC000880801991 GG On-Demand Anodyne L3MBTL3 64 39 CNC(=O)CCCNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880801995 GF On-Demand Anodyne HDAC10 19 48 CNC(=O)CCCNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880801995 GF On-Demand Anodyne HDAC1 16 48 CNC(=O)CCCNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880801995 GF On-Demand Anodyne HDAC3 23 43 CC(=O)N[C@@H]1CCCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801999 GF On-Demand Anodyne MTNR1A 21 40 CC(=O)N[C@@H]1CCCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880801999 GF On-Demand Anodyne MTNR1B 17 50 CC(=O)N[C@H]1CCCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880802000 GF On-Demand Anodyne MTNR1A 21 40 CC(=O)N[C@H]1CCCN(C(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880802000 GF On-Demand Anodyne MTNR1B 17 50 O=C(CNC(=O)Nc1ccc(Br)c(Br)c1)NC1CC1 ZINC000880802017 GF On-Demand Anodyne PRMT3 49 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccsc2)C1 ZINC000880802036 FF On-Demand Anodyne PAPA1_CARPA 36 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccsc2)C1 ZINC000880802036 FF On-Demand Anodyne FPR1 44 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccsc2)C1 ZINC000880802037 FF On-Demand Anodyne PAPA1_CARPA 36 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccsc2)C1 ZINC000880802037 FF On-Demand Anodyne FPR1 44 35 O=C(NCCCO)Nc1ccc(Br)c(Br)c1 ZINC000880802066 FF On-Demand Anodyne PRMT3 51 33 O=C(NCCc1cccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802076 FG On-Demand Anodyne MTNR1A 30 45 O=C(NCCc1cccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802076 FG On-Demand Anodyne MTNR1B 37 45 O=C(NCCc1cccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802076 FG On-Demand Anodyne NAMPT 35 43 O=C(NCCCCn1ccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802082 GG On-Demand Anodyne TBXAS1 33 44 O=C(NCCCCn1ccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802082 GG On-Demand Anodyne QPCT 44 45 CCN1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880802084 FF On-Demand Anodyne MTNR1A 23 46 CCN1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880802084 FF On-Demand Anodyne MTNR1B 25 46 CCN1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880802084 FF On-Demand Anodyne EPHX2 27 41 O=C(CNC(=O)Nc1c(Br)ccc2c1CCO2)NC1CC1 ZINC000880802096 FD On-Demand Anodyne MTNR1A 29 40 CNC(=O)CCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802102 FE On-Demand Anodyne MTNR1B 39 43 CC(=O)NCCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802122 FE On-Demand Anodyne MTNR1A 38 47 CC(=O)NCCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802122 FE On-Demand Anodyne MTNR1B 43 50 O=C(NCCOc1cccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802189 GF On-Demand Anodyne MTNR1A 25 40 O=C(NCCOc1cccnc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802189 GF On-Demand Anodyne MTNR1B 27 40 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1c(Br)ccc3c1CCO3)C2 ZINC000880802196 GH On-Demand Anodyne MTNR1A 18 40 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1c(Br)ccc3c1CCO3)C2 ZINC000880802196 GH On-Demand Anodyne MTNR1B 18 40 CC[C@@H](O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802215 EF On-Demand Anodyne MTNR1B 37 40 CC[C@H](O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802216 EF On-Demand Anodyne MTNR1B 37 40 C[C@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)[S@@](C)=O ZINC000880802217 GF On-Demand Anodyne MTNR1B 37 40 C[C@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)[S@](C)=O ZINC000880802218 GF On-Demand Anodyne MTNR1B 37 40 C[C@@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)[S@](C)=O ZINC000880802219 GF On-Demand Anodyne MTNR1B 37 40 C[C@@H](CCNC(=O)Nc1c(Br)ccc2c1CCO2)[S@@](C)=O ZINC000880802220 GF On-Demand Anodyne MTNR1B 37 40 CN1C[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)CCC1=O ZINC000880802230 FE On-Demand Anodyne MTNR1A 17 45 CN1C[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)CCC1=O ZINC000880802231 FE On-Demand Anodyne MTNR1A 17 45 C[S@@](=O)CCCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802246 FE On-Demand Anodyne MTNR1B 37 41 CC1CC(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880802256 CF On-Demand Anodyne GABRA1 19 51 CC1CC(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880802256 CF On-Demand Anodyne MPO 65 37 CC1CC(CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880802256 CF On-Demand Anodyne GABRA2 16 51 CN1CCC(CNC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880802259 FF On-Demand Anodyne CACNA1I 42 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(C)C1 ZINC000880802268 DE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(C)C1 ZINC000880802268 DE On-Demand Anodyne POLG_HCV1 21 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(C)C1 ZINC000880802269 DE On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(C)C1 ZINC000880802269 DE On-Demand Anodyne POLG_HCV1 21 40 O=C(NCC[C@@H]1CCCO1)Nc1c(Br)ccc2c1CCO2 ZINC000880802346 FG On-Demand Anodyne MTNR1A 27 44 O=C(NCC[C@@H]1CCCO1)Nc1c(Br)ccc2c1CCO2 ZINC000880802346 FG On-Demand Anodyne MTNR1B 31 44 O=C(NCC[C@H]1CCCO1)Nc1c(Br)ccc2c1CCO2 ZINC000880802347 FG On-Demand Anodyne MTNR1A 27 44 O=C(NCC[C@H]1CCCO1)Nc1c(Br)ccc2c1CCO2 ZINC000880802347 FG On-Demand Anodyne MTNR1B 31 44 CC(C)(C)NC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802370 GF On-Demand Anodyne MTNR1B 38 41 O=C(NCC[C@@H]1CC1(Cl)Cl)c1cc(C(F)F)[nH]n1 ZINC000880802403 CF On-Demand Anodyne ALPL 40 33 O=C(NCC[C@H]1CC1(Cl)Cl)c1cc(C(F)F)[nH]n1 ZINC000880802404 CF On-Demand Anodyne ALPL 40 33 O=C(NCCc1ccncc1)Nc1c(Br)ccc2c1CCO2 ZINC000880802422 FG On-Demand Anodyne MTNR1B 38 41 O=C(Nc1c(Br)ccc2c1CCO2)N[C@@H]1CC[C@H](CO)CC1 ZINC000880802454 FG On-Demand Anodyne MTNR1A 15 42 O=C(Nc1c(Br)ccc2c1CCO2)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880802457 FG On-Demand Anodyne MTNR1A 15 42 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@@H]1Br ZINC000880802465 DE On-Demand Reactive HCN1 70 32 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@@H]1Br ZINC000880802465 DE On-Demand Reactive HCN4 49 31 C[C@]1(CNC(=O)c2cccn3nccc23)C[C@H]1Br ZINC000880802466 DE On-Demand Reactive HCN1 70 32 C[C@]1(CNC(=O)c2cccn3nccc23)C[C@H]1Br ZINC000880802466 DE On-Demand Reactive HCN4 49 31 C[C@]1(CNC(=O)c2cccn3nccc23)C[C@@H]1Br ZINC000880802468 DE On-Demand Reactive HCN1 70 32 C[C@]1(CNC(=O)c2cccn3nccc23)C[C@@H]1Br ZINC000880802468 DE On-Demand Reactive HCN4 49 31 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@H]1Br ZINC000880802469 DE On-Demand Reactive HCN1 70 32 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@H]1Br ZINC000880802469 DE On-Demand Reactive HCN4 49 31 Cc1nc(C(C)C)ncc1C(=O)Nc1nc2cc(Cl)c(F)cc2[nH]1 ZINC000880802497 EH On-Demand Anodyne NR2E3 53 35 Cc1cnc(Cl)c(C(=O)NC[C@@]2(C)C[C@H]2Br)c1 ZINC000880802571 DF On-Demand Reactive P2RX7 18 43 Cc1cnc(Cl)c(C(=O)NC[C@@]2(C)C[C@@H]2Br)c1 ZINC000880802573 DF On-Demand Reactive P2RX7 18 43 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802648 GG On-Demand Reactive KCNA3 48 40 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802648 GG On-Demand Reactive HCN1 71 37 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802648 GG On-Demand Reactive HCN4 50 37 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802649 GG On-Demand Reactive KCNA3 48 40 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802649 GG On-Demand Reactive HCN1 71 37 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802649 GG On-Demand Reactive HCN4 50 37 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802650 GG On-Demand Reactive KCNA3 48 40 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802650 GG On-Demand Reactive HCN1 71 37 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@H]2Br)c(O)n1 ZINC000880802650 GG On-Demand Reactive HCN4 50 37 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802651 GG On-Demand Reactive KCNA3 48 40 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802651 GG On-Demand Reactive HCN1 71 37 COc1ccccc1-c1ccc(C(=O)NC[C@]2(C)C[C@@H]2Br)c(O)n1 ZINC000880802651 GG On-Demand Reactive HCN4 50 37 C[C@@]1(CNC(=O)c2ncsc2C2CC2)C[C@H]1Br ZINC000880802746 DF On-Demand Reactive MAP1 40 35 C[C@]1(CNC(=O)c2ncsc2C2CC2)C[C@H]1Br ZINC000880802747 DF On-Demand Reactive MAP1 40 35 C[C@]1(CNC(=O)c2ncsc2C2CC2)C[C@@H]1Br ZINC000880802748 DF On-Demand Reactive MAP1 40 35 C[C@@]1(CNC(=O)c2ncsc2C2CC2)C[C@@H]1Br ZINC000880802749 DF On-Demand Reactive MAP1 40 35 COC(=O)C1CCC(NC(=O)Nc2c(Br)ccc3c2CCO3)CC1 ZINC000880802764 GG On-Demand Anodyne MTNR1A 16 43 CC1CC(CNC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880802765 DF On-Demand Anodyne KCNQ2 44 35 O=C(NCC[C@@H]1CC1(Cl)Cl)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880802766 EG On-Demand Anodyne GABRA1 15 48 O=C(NCC[C@@H]1CC1(Cl)Cl)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880802766 EG On-Demand Anodyne MPO 40 34 O=C(NCC[C@H]1CC1(Cl)Cl)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880802767 EG On-Demand Anodyne GABRA1 15 48 O=C(NCC[C@H]1CC1(Cl)Cl)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880802767 EG On-Demand Anodyne MPO 40 34 Cc1noc(C)c1CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802774 GG On-Demand Anodyne MTNR1A 32 43 Cc1noc(C)c1CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802774 GG On-Demand Anodyne MTNR1B 38 40 O=C(NCC[C@@H]1CC1(Cl)Cl)c1cnc(CC2CC2)s1 ZINC000880802844 DG On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@@H]1CC1(Cl)Cl)c1cnc(CC2CC2)s1 ZINC000880802844 DG On-Demand Anodyne SIRT1 41 34 O=C(NCC[C@H]1CC1(Cl)Cl)c1cnc(CC2CC2)s1 ZINC000880802845 DG On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@H]1CC1(Cl)Cl)c1cnc(CC2CC2)s1 ZINC000880802845 DG On-Demand Anodyne SIRT1 41 34 O=C1CC[C@H](c2ccc(C(=O)NCC[C@@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802883 EF On-Demand Anodyne PLD1 40 34 O=C1CC[C@H](c2ccc(C(=O)NCC[C@@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802883 EF On-Demand Anodyne PLD2 42 34 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802884 EF On-Demand Anodyne PLD1 40 34 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802884 EF On-Demand Anodyne PLD2 42 34 O=C1CC[C@H](c2ccc(C(=O)NCC[C@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802885 EF On-Demand Anodyne PLD1 40 34 O=C1CC[C@H](c2ccc(C(=O)NCC[C@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802885 EF On-Demand Anodyne PLD2 42 34 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802886 EF On-Demand Anodyne PLD1 40 34 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@H]3CC3(Cl)Cl)cc2)N1 ZINC000880802886 EF On-Demand Anodyne PLD2 42 34 C[C@@H](Cn1cncn1)NC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880802896 FE On-Demand Anodyne HIS3 74 33 CN(CCN1CCOCC1)C(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880803082 GE On-Demand Anodyne CASR 50 38 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(Cl)Cl)C2 ZINC000880803086 EH On-Demand Anodyne NQO2 38 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(Cl)Cl)C2 ZINC000880803086 EH On-Demand Anodyne MTNR1A 57 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(Cl)Cl)C2 ZINC000880803086 EH On-Demand Anodyne MTNR1B 49 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(Cl)Cl)C2 ZINC000880803088 EH On-Demand Anodyne NQO2 38 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(Cl)Cl)C2 ZINC000880803088 EH On-Demand Anodyne MTNR1A 57 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(Cl)Cl)C2 ZINC000880803088 EH On-Demand Anodyne MTNR1B 49 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC1(F)F ZINC000880803126 EE On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC1(F)F ZINC000880803127 EE On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC1(F)F ZINC000880803128 EE On-Demand Anodyne PAPA1_CARPA 38 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC1(F)F ZINC000880803129 EE On-Demand Anodyne PAPA1_CARPA 38 46 COc1ccc2c(c1)CC[C@H](C(=O)NNc1nc3cccnc3s1)C2 ZINC000880803145 FF On-Demand Reactive FAAH 16 41 CCOC(=O)CCNC(=O)Nc1c(Br)ccc2c1CCO2 ZINC000880803164 FE On-Demand Anodyne MTNR1B 38 40 Cc1coc(C(=O)N[C@@H]2CCO[C@H]2c2cccnc2)c1 ZINC000880803165 CE On-Demand Anodyne CHRNA7 39 41 O=C(N[C@@H]1CCO[C@H]1c1cccnc1)c1ccc(CN2CCOCC2)o1 ZINC000880803170 FD On-Demand Anodyne CHRNA7 45 42 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@H](CCO)C1 ZINC000880803181 GG On-Demand Anodyne EPHX2 19 43 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@@H](CCO)C1 ZINC000880803182 GG On-Demand Anodyne EPHX2 19 43 O=C(COC1CC1)N[C@@H]1CCO[C@H]1c1cccnc1 ZINC000880803239 CD On-Demand Anodyne CHRNA7 44 35 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(F)F)C2 ZINC000880803282 DF On-Demand Anodyne NQO2 39 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(F)F)C2 ZINC000880803282 DF On-Demand Anodyne MTNR1A 63 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CC1(F)F)C2 ZINC000880803282 DF On-Demand Anodyne MTNR1B 54 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(F)F)C2 ZINC000880803284 DF On-Demand Anodyne NQO2 39 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(F)F)C2 ZINC000880803284 DF On-Demand Anodyne MTNR1A 63 47 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CC1(F)F)C2 ZINC000880803284 DF On-Demand Anodyne MTNR1B 54 47 CCC(=O)N1CC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803316 GF On-Demand Anodyne MTNR1A 20 48 CCC(=O)N1CC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803316 GF On-Demand Anodyne MTNR1B 22 47 CCC(=O)N1CC[C@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803316 GF On-Demand Anodyne EPHX2 25 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803317 GF On-Demand Anodyne MTNR1A 20 48 CCC(=O)N1CC[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803317 GF On-Demand Anodyne MTNR1B 22 47 CCC(=O)N1CC[C@@H](NC(=O)Nc2c(Br)ccc3c2CCO3)C1 ZINC000880803317 GF On-Demand Anodyne EPHX2 25 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803329 FE On-Demand Anodyne PAPA1_CARPA 41 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803329 FE On-Demand Anodyne CTSK 23 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803329 FE On-Demand Anodyne CTSL 31 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803329 FE On-Demand Anodyne CTSS 27 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803330 FE On-Demand Anodyne PAPA1_CARPA 41 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803330 FE On-Demand Anodyne CTSK 23 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803330 FE On-Demand Anodyne CTSL 31 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(OC)ccc1F ZINC000880803330 FE On-Demand Anodyne CTSS 27 49 O=C(NCC(F)(F)c1ccc(Br)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880803334 GF On-Demand Anodyne CACNA1G 35 40 O=C(NCC(F)(F)c1ccc(Br)cc1)[C@H]1CCc2nncn2CC1 ZINC000880803335 GF On-Demand Anodyne CACNA1G 35 40 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@@H](CO)C1 ZINC000880803382 GG On-Demand Anodyne EPHX2 23 50 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@H](CO)C1 ZINC000880803383 GG On-Demand Anodyne EPHX2 23 50 O=C(NOC1CCOCC1)Nc1ccc(Br)c(Br)c1 ZINC000880803398 GG On-Demand Anodyne P96878_MYCTU 40 35 CCn1cc([C@@H]2OCC[C@H]2NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cn1 ZINC000880803446 FE On-Demand Anodyne PANC 45 31 CCn1cc([C@@H]2OCC[C@H]2NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cn1 ZINC000880803447 FE On-Demand Anodyne PANC 45 31 CCn1cc([C@@H]2OCC[C@H]2NC(=O)c2ccc(OC(F)F)c(Cl)c2)cn1 ZINC000880803458 GG On-Demand Anodyne PDE4D 26 43 O=C(NC[C@]1(O)CCOC1)Nc1ccc(Br)c(Br)c1 ZINC000880803461 GE On-Demand Anodyne PRMT3 50 29 O=C(NC[C@@]1(O)CCOC1)Nc1ccc(Br)c(Br)c1 ZINC000880803462 GE On-Demand Anodyne PRMT3 50 29 CCn1cc([C@@H]2OCC[C@H]2NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)cn1 ZINC000880803466 FE On-Demand Anodyne GABRA1 17 42 CCn1cc([C@@H]2OCC[C@H]2NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)cn1 ZINC000880803466 FE On-Demand Anodyne GABRA2 15 42 O=C(NCC[C@@H]1CC1(F)F)c1ccc(OC(F)F)c(Cl)c1 ZINC000880803477 EH On-Demand Anodyne PDE4D 17 42 O=C(NCC[C@H]1CC1(F)F)c1ccc(OC(F)F)c(Cl)c1 ZINC000880803478 EH On-Demand Anodyne PDE4D 17 42 O=C1CC[C@H](c2ccc(C(=O)NCC[C@@H]3CC3(F)F)cc2)N1 ZINC000880803585 DE On-Demand Anodyne PLD1 43 33 O=C1CC[C@H](c2ccc(C(=O)NCC[C@@H]3CC3(F)F)cc2)N1 ZINC000880803585 DE On-Demand Anodyne PLD2 47 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@@H]3CC3(F)F)cc2)N1 ZINC000880803586 DE On-Demand Anodyne PLD1 43 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@@H]3CC3(F)F)cc2)N1 ZINC000880803586 DE On-Demand Anodyne PLD2 47 33 O=C1CC[C@H](c2ccc(C(=O)NCC[C@H]3CC3(F)F)cc2)N1 ZINC000880803587 DE On-Demand Anodyne PLD1 43 33 O=C1CC[C@H](c2ccc(C(=O)NCC[C@H]3CC3(F)F)cc2)N1 ZINC000880803587 DE On-Demand Anodyne PLD2 47 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@H]3CC3(F)F)cc2)N1 ZINC000880803588 DE On-Demand Anodyne PLD1 43 33 O=C1CC[C@@H](c2ccc(C(=O)NCC[C@H]3CC3(F)F)cc2)N1 ZINC000880803588 DE On-Demand Anodyne PLD2 47 33 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC[C@H](c3nc(C)no3)O1)C2 ZINC000880803623 FF On-Demand Anodyne MTNR1A 19 40 O=C(Nc1ccc(Br)c(Br)c1)N1CCCOCC1 ZINC000880803625 GG On-Demand Anodyne EPHX2 35 42 O=C(Nc1ccc(Br)c(Br)c1)N[C@@H]1CC[C@@H](O)CC1 ZINC000880803643 GH On-Demand Anodyne EPHX2 51 47 O=C(NCC1OCCCO1)Nc1ccc(Br)c(Br)c1 ZINC000880803657 GG On-Demand Anodyne EPHX2 16 40 O=C(NCC1OCCCO1)Nc1ccc(Br)c(Br)c1 ZINC000880803657 GG On-Demand Anodyne PRMT3 46 33 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCO[C@H]1c1cccnc1)C2 ZINC000880803661 FF On-Demand Anodyne FAAH 15 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccccc2N(C)C[C@@H]1C ZINC000880803713 GF On-Demand Anodyne FPR1 42 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccccc2N(C)C[C@@H]1C ZINC000880803715 GF On-Demand Anodyne FPR1 42 33 CCn1cc([C@@H]2OCC[C@H]2NC(=O)c2cc(-c3ccc(OC)cc3)on2)cn1 ZINC000880803742 GF On-Demand Anodyne PDK1 40 34 O=C(NNC(=O)C1CC1)Nc1ccc(Br)c(Br)c1 ZINC000880803744 GF On-Demand Reactive DHODH 18 42 O=C(NNC(=O)C1CC1)Nc1ccc(Br)c(Br)c1 ZINC000880803744 GF On-Demand Reactive TYK2 48 38 COC[C@@H](O)CCNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880803751 GF On-Demand Anodyne ADRB1 44 35 O=C(N[C@@H]1CCO[C@H]1c1cccnc1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880803775 FH On-Demand Anodyne PDE4D 18 43 O=C(NCC[C@@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803803 CF On-Demand Anodyne SIRT3 43 36 O=C(NCC[C@@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803803 CF On-Demand Anodyne SIRT2 47 36 O=C(NCC[C@@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803803 CF On-Demand Anodyne SIRT1 43 36 O=C(NCC[C@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803806 CF On-Demand Anodyne SIRT3 43 36 O=C(NCC[C@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803806 CF On-Demand Anodyne SIRT2 47 36 O=C(NCC[C@H]1CC1(F)F)c1cnc(CC2CC2)s1 ZINC000880803806 CF On-Demand Anodyne SIRT1 43 36 O=C(NCC[C@@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880803852 DF On-Demand Anodyne GABRA1 17 49 O=C(NCC[C@@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880803852 DF On-Demand Anodyne MPO 50 35 O=C(NCC[C@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880803855 DF On-Demand Anodyne GABRA1 17 49 O=C(NCC[C@H]1CC1(F)F)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880803855 DF On-Demand Anodyne MPO 50 35 C[C@H](CO)N(C)C(=O)Nc1ccc(Br)c(Br)c1 ZINC000880803867 FG On-Demand Anodyne NPY5R 36 41 C[C@@H](CO)N(C)C(=O)Nc1ccc(Br)c(Br)c1 ZINC000880803870 FG On-Demand Anodyne NPY5R 36 41 C[C@@H]1CN(C(=O)Nc2ccc(Br)c(Br)c2)CC[C@@H]1O ZINC000880803888 GG On-Demand Anodyne EPHX2 21 41 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803908 CH On-Demand Anodyne NQO2 21 45 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803908 CH On-Demand Anodyne MTNR1A 17 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803908 CH On-Demand Anodyne MTNR1B 17 40 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803909 CH On-Demand Anodyne NQO2 21 45 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803909 CH On-Demand Anodyne MTNR1A 17 40 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CC1(F)F ZINC000880803909 CH On-Demand Anodyne MTNR1B 17 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803910 CH On-Demand Anodyne NQO2 21 45 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803910 CH On-Demand Anodyne MTNR1A 17 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803910 CH On-Demand Anodyne MTNR1B 17 40 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803911 CH On-Demand Anodyne NQO2 21 45 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803911 CH On-Demand Anodyne MTNR1A 17 40 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CC1(F)F ZINC000880803911 CH On-Demand Anodyne MTNR1B 17 40 O=C(NCC[C@@H]1CC1(F)F)c1cc2ccccc2cc1F ZINC000880803927 CH On-Demand Anodyne POLR1A 45 31 O=C(NCC[C@H]1CC1(F)F)c1cc2ccccc2cc1F ZINC000880803928 CH On-Demand Anodyne POLR1A 45 31 O=C(NCC[C@@H]1CC1(F)F)c1ncsc1C1CC1 ZINC000880803941 CF On-Demand Anodyne MAP1 42 37 O=C(NCC[C@H]1CC1(F)F)c1ncsc1C1CC1 ZINC000880803942 CF On-Demand Anodyne MAP1 42 37 C[C@@H]1CN(C(=O)Nc2ccc(Br)c(Br)c2)CC[C@H]1O ZINC000880803949 GG On-Demand Anodyne EPHX2 21 41 C[C@H]1CN(C(=O)Nc2ccc(Br)c(Br)c2)CC[C@H]1O ZINC000880803950 GG On-Demand Anodyne EPHX2 21 41 C[C@H]1CN(C(=O)Nc2ccc(Br)c(Br)c2)CC[C@@H]1O ZINC000880803951 GG On-Demand Anodyne EPHX2 21 41 CN1CC[C@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1=O ZINC000880803966 GF On-Demand Anodyne CCKAR 36 41 CN1CC[C@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1=O ZINC000880803966 GF On-Demand Anodyne CCKBR 54 39 COc1ccccc1-c1ccc(C(=O)NCC[C@@H]2CC2(F)F)c(O)n1 ZINC000880804129 EG On-Demand Anodyne KCNA3 42 35 COc1ccccc1-c1ccc(C(=O)NCC[C@H]2CC2(F)F)c(O)n1 ZINC000880804130 EG On-Demand Anodyne KCNA3 42 35 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCO[C@H]1c1nccn1C)C2 ZINC000880804167 FE On-Demand Anodyne FAAH 15 41 COCCONC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880804203 FF On-Demand Anodyne P96878_MYCTU 45 37 CC(CO)(CO)NC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880804219 GE On-Demand Anodyne IMDH_CRYPV 59 38 CC[C@@H](NC(=O)Nc1ccc(Br)c(Br)c1)C(=O)NC ZINC000880804311 GF On-Demand Anodyne ANPEP 23 47 O=C(N[C@@H]1CCO[C@H]1c1cc[nH]n1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880804319 FF On-Demand Anodyne PDE4D 15 40 O=C(Nc1ccc(Br)c(Br)c1)N1CCC2(COC2)C1 ZINC000880804324 GG On-Demand Anodyne EPHX2 35 43 C#CCC1(O)CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880804338 DF On-Demand Mild RBP4 15 42 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1c(Cl)cccc1OC)C2 ZINC000880804360 FH On-Demand Anodyne RBP4 15 40 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1c(Cl)cccc1OC ZINC000880804379 EF On-Demand Anodyne SLC6A3 46 38 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1c(Cl)cccc1OC ZINC000880804380 EF On-Demand Anodyne SLC6A3 46 38 Cn1ccnc1[C@@H]1OCCC[C@H]1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880804411 GH On-Demand Anodyne PDE4D 24 41 Cn1ccnc1[C@@H]1OCCC[C@H]1CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880804411 GH On-Demand Anodyne CACNA1I 53 37 CCn1cc([C@@H]2OCC[C@H]2NC(=O)c2cccc3nsnc23)cn1 ZINC000880804413 EE On-Demand Anodyne HTR3A 22 41 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@](F)(CO)C1 ZINC000880804506 GG On-Demand Anodyne EPHX2 35 42 O=C(Nc1ccc(Br)c(Br)c1)N1CC[C@@](F)(CO)C1 ZINC000880804507 GG On-Demand Anodyne EPHX2 35 42 CC1CN(C(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804520 EH On-Demand Anodyne EPHX2 27 43 CONC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880804526 EE On-Demand Anodyne HTR4 42 38 CONC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880804526 EE On-Demand Anodyne SSTR1 44 36 CONC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880804526 EE On-Demand Anodyne RBP4 19 44 O=C(Nc1ccc(Br)c(Br)c1)N[C@@H]1CC[C@H](O)CC1 ZINC000880804528 GH On-Demand Anodyne EPHX2 51 47 COC[C@@H](NC(=O)Nc1ccc(Br)c(Br)c1)C(N)=O ZINC000880804608 GD On-Demand Anodyne ANPEP 18 45 COC[C@H](NC(=O)Nc1ccc(Br)c(Br)c1)C(N)=O ZINC000880804609 GD On-Demand Anodyne ANPEP 18 45 COC(=O)[C@H](CNC(=O)Nc1c(Cl)cccc1OC)OC ZINC000880804682 DD On-Demand Anodyne SOAT1 33 41 COCCN(CC1CCN(C)CC1)C(=O)Nc1c(Cl)cccc1OC ZINC000880804797 FG On-Demand Anodyne HTR4 47 36 COCCN(CC1CCN(C)CC1)C(=O)Nc1c(Cl)cccc1OC ZINC000880804797 FG On-Demand Anodyne ACKR3 60 31 CCn1ncc(NC(=O)Nc2c(Cl)cccc2OC)c1C ZINC000880804827 DH On-Demand Anodyne PDGFRA 18 40 O=C(Nc1ccc(Br)c(Br)c1)N[C@H]1CCOC1=O ZINC000880804840 GF On-Demand Anodyne LUXR 83 46 O=C(Nc1ccc(Br)c(Br)c1)N[C@H]1CCOC1=O ZINC000880804840 GF On-Demand Anodyne TRAR 100 51 O=C(Nc1ccc(Br)c(Br)c1)N[C@H]1CCOC1=O ZINC000880804840 GF On-Demand Anodyne LASR 66 47 C#CC1(F)CN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880804848 CF On-Demand Mild RBP4 15 43 COC[C@@H](O)CNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880804851 GE On-Demand Anodyne ADRB1 45 36 COC[C@@H](O)CNC(=O)Nc1ccc(Br)c(Br)c1 ZINC000880804851 GE On-Demand Anodyne PRMT3 52 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCO[C@H]1c1nccn1C)C2 ZINC000880804897 GF On-Demand Anodyne MTNR1A 26 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCO[C@H]1c1nccn1C)C2 ZINC000880804897 GF On-Demand Anodyne MTNR1B 24 43 Cn1ccnc1[C@@H]1OCCC[C@H]1CNC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880804901 FF On-Demand Anodyne CCR2 47 33 COc1ccccc1[C@@H]1CN(C(=O)Nc2c(Cl)cccc2OC)CCO1 ZINC000880804902 GH On-Demand Anodyne RBP4 27 42 COc1ccccc1[C@@H]1CN(C(=O)Nc2c(Cl)cccc2OC)CCO1 ZINC000880804902 GH On-Demand Anodyne SMO 16 40 COc1ccccc1[C@H]1CN(C(=O)Nc2c(Cl)cccc2OC)CCO1 ZINC000880804903 GH On-Demand Anodyne RBP4 27 42 COc1ccccc1[C@H]1CN(C(=O)Nc2c(Cl)cccc2OC)CCO1 ZINC000880804903 GH On-Demand Anodyne SMO 16 40 COc1ccc(CN(CCO)C(=O)Nc2c(Cl)cccc2OC)cc1 ZINC000880804986 FG On-Demand Anodyne BMP1 42 40 COc1ccc(CN(CCO)C(=O)Nc2c(Cl)cccc2OC)cc1 ZINC000880804986 FG On-Demand Anodyne ROCK2 15 43 NC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804989 GF On-Demand Anodyne EPHX2 39 40 NC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804989 GF On-Demand Anodyne MTCA1 23 43 NC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804989 GF On-Demand Anodyne P96878_MYCTU 24 43 NC(=O)C1CC(NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804990 GF On-Demand Anodyne EPHX2 39 40 NC(=O)C1CC(NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804990 GF On-Demand Anodyne MTCA1 23 43 NC(=O)C1CC(NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804990 GF On-Demand Anodyne P96878_MYCTU 24 43 NC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804991 GF On-Demand Anodyne EPHX2 39 40 NC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804991 GF On-Demand Anodyne MTCA1 23 43 NC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(Br)c(Br)c2)C1 ZINC000880804991 GF On-Demand Anodyne P96878_MYCTU 24 43 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805033 FG On-Demand Anodyne DRD4 18 40 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805033 FG On-Demand Anodyne HTR4 75 38 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805033 FG On-Demand Anodyne P2RY12 17 40 COCCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805076 GF On-Demand Anodyne CCR3 32 41 COCCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805076 GF On-Demand Anodyne EPHX2 38 40 COCCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805076 GF On-Demand Anodyne CXCR3 19 42 CCOC(=O)N1CCN(C(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805118 GF On-Demand Anodyne P2RY12 41 39 COC(=O)N1CCC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805146 EF On-Demand Anodyne HTR4 46 36 COC(=O)N1CCC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805146 EF On-Demand Anodyne EPHX2 28 43 COC(=O)N1CCC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805147 EF On-Demand Anodyne HTR4 46 36 COC(=O)N1CCC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880805147 EF On-Demand Anodyne EPHX2 28 43 COCCn1cc(NC(=O)Nc2cc(C(C)=O)ccc2Br)cn1 ZINC000880805178 GG On-Demand Anodyne PANC 44 34 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2c(Cl)cccc2OC)c1 ZINC000880805207 GG On-Demand Anodyne MTNR1A 39 48 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2c(Cl)cccc2OC)c1 ZINC000880805207 GG On-Demand Anodyne MTNR1B 42 38 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2c(Cl)cccc2OC)c1 ZINC000880805207 GG On-Demand Anodyne SOAT1 45 44 C#CCN(C(=O)Nc1c(Cl)cccc1OC)C1CC1 ZINC000880805309 CF On-Demand Mild MBTPS1 42 31 COC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805336 EF On-Demand Anodyne DRD2 15 51 COC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805336 EF On-Demand Anodyne DRD4 18 40 COC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805336 EF On-Demand Anodyne HTR4 42 39 COC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805336 EF On-Demand Anodyne EPHX2 57 45 CCS(=O)(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805434 FD On-Demand Anodyne RBP4 15 46 CCS(=O)(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805434 FD On-Demand Anodyne F13A1 41 35 C=CCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805471 GG On-Demand Mild EPHX2 34 41 C=CCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805471 GG On-Demand Mild CXCR3 19 43 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne HTR4 44 44 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne P2RY12 51 46 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne PDGFRB 26 40 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne TGM2 28 40 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne RBP4 15 47 CCOC(=O)N1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805482 EF On-Demand Anodyne F13A1 34 40 COC(=O)C1CCN(C(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805495 GG On-Demand Anodyne PTR1 46 34 CCn1c(S)nnc1C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880805637 GH On-Demand Anodyne RBP4 19 41 COC[C@@H](O)CNC(=O)Nc1c(Cl)cccc1OC ZINC000880805643 CD On-Demand Anodyne ADRB1 49 36 COC[C@@H](O)CNC(=O)Nc1c(Cl)cccc1OC ZINC000880805643 CD On-Demand Anodyne SOAT1 27 41 O=C(CN1CCCCS1(=O)=O)Nc1cc(Cl)c(O)c2ccccc12 ZINC000880805670 FF On-Demand Anodyne CDK1 15 41 CCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805692 FG On-Demand Anodyne SLC6A5 23 42 CCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805692 FG On-Demand Anodyne EPHX2 42 43 CCN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805692 FG On-Demand Anodyne CXCR3 20 45 CCN1CC[C@H](CNC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880805740 FG On-Demand Anodyne CCR3 57 40 CCN1CC[C@H](CNC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880805740 FG On-Demand Anodyne CACNA1I 67 37 C#CC(C)(C)NC(=O)Nc1c(Cl)cccc1OC ZINC000880805793 CF On-Demand Mild ECR 15 40 C#CC(C)(C)NC(=O)Nc1c(Cl)cccc1OC ZINC000880805793 CF On-Demand Mild IMDH_CRYPV 32 40 COc1ccc2c(c1)CN(C(=O)Nc1c(Cl)cccc1OC)CCO2 ZINC000880805808 FH On-Demand Anodyne DRD4 43 35 COc1ccc2c(c1)CN(C(=O)Nc1c(Cl)cccc1OC)CCO2 ZINC000880805808 FH On-Demand Anodyne RBP4 15 40 CC[C@@H](C)C(=O)NNC(=O)Nc1c(Cl)cccc1OC ZINC000880805853 CF On-Demand Reactive PYGL 15 40 COCCONC(=O)Nc1c(Cl)cccc1OC ZINC000880805882 CE On-Demand Anodyne PYGL 15 41 C=C(C)CN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805892 GH On-Demand Mild EPHX2 34 41 C=C(C)CN1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805892 GH On-Demand Mild CXCR3 19 43 CC(=O)NCC1CCN(C(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880805934 GG On-Demand Anodyne CACNA1I 58 34 CCONC(=O)Nc1c(Cl)cccc1OC ZINC000880806026 BE On-Demand Anodyne KCNK3 42 38 CCOC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806043 FG On-Demand Anodyne DRD4 21 40 CCOC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806043 FG On-Demand Anodyne HTR4 63 41 CCOC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806043 FG On-Demand Anodyne EPHX2 57 47 CCOC(=O)N1CCC(NC(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806043 FG On-Demand Anodyne CCR8 38 40 CCOC(=O)C1CCN(C(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880806111 GG On-Demand Anodyne PTR1 46 34 COC(=O)N1CCC(NC(=O)Nc2cc(C(C)=O)ccc2Br)CC1 ZINC000880806169 GG On-Demand Anodyne EPHX2 49 48 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880806172 GG On-Demand Anodyne CCR3 21 40 CCOC(=O)N1CCCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806178 FG On-Demand Anodyne HTR4 31 42 CCOC(=O)N1CCCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806178 FG On-Demand Anodyne P2RY12 38 44 CCOC(=O)N1CCCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806178 FG On-Demand Anodyne RBP4 15 44 COCCO[C@H](C)C(=O)NNC(=O)Nc1c(Cl)cccc1OC ZINC000880806307 ED On-Demand Reactive PYGL 18 42 COCCO[C@@H](C)C(=O)NNC(=O)Nc1c(Cl)cccc1OC ZINC000880806308 ED On-Demand Reactive PYGL 18 42 COC(=O)[C@H](F)CNC(=O)Nc1c(Cl)cccc1OC ZINC000880806315 DD On-Demand Anodyne SOAT1 31 41 C#CC[C@@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806579 DH On-Demand Mild HTR1A 21 41 C#CC[C@@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806579 DH On-Demand Mild RBP4 23 41 C#CC[C@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806580 DH On-Demand Mild HTR1A 21 41 C#CC[C@H]1CCCN(C(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806580 DH On-Demand Mild RBP4 23 41 CNc1nc(C(=O)N2CCN(CCOCCOC)CC2)cs1 ZINC000880806588 EC On-Demand Anodyne TRPC6 59 43 CNc1nc(C(=O)N2CCN(CCOCCOC)CC2)cs1 ZINC000880806588 EC On-Demand Anodyne TRPC3 52 43 CCc1nccn1C[C@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880806612 GH On-Demand Anodyne FKBP1A 50 44 CCc1nccn1C[C@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880806612 GH On-Demand Anodyne ACKR3 46 34 C=CCN(CCOC)C(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880806712 FG On-Demand Mild LSS 40 35 COC(=O)C1=NOC2(CCN(C(=O)Nc3c(Cl)cccc3OC)CC2)C1 ZINC000880806744 GF On-Demand Anodyne TRPM8 30 41 O=C(NCc1nnc2ccc(Cl)cn12)c1ccc(CN2CCOCC2)o1 ZINC000880806891 GD On-Demand Anodyne DPOL_VZVD 25 42 C#CCNC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806961 EE On-Demand Mild DRD2 15 40 C#CCNC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806961 EE On-Demand Mild EPHX2 24 43 C#CCNC(=O)C1CCN(C(=O)Nc2c(Cl)cccc2OC)CC1 ZINC000880806961 EE On-Demand Mild RBP4 19 42 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806981 EF On-Demand Anodyne DRD4 20 41 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806981 EF On-Demand Anodyne HTR4 76 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806981 EF On-Demand Anodyne EPHX2 40 43 CCOC(=O)N1CC[C@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806981 EF On-Demand Anodyne CCR8 48 39 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806982 EF On-Demand Anodyne DRD4 20 41 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806982 EF On-Demand Anodyne HTR4 76 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806982 EF On-Demand Anodyne EPHX2 40 43 CCOC(=O)N1CC[C@@H](NC(=O)Nc2c(Cl)cccc2OC)C1 ZINC000880806982 EF On-Demand Anodyne CCR8 48 39 CNC(=O)[C@@H](NC(=O)Nc1cc(C(C)=O)ccc1Br)C(C)C ZINC000880807146 FF On-Demand Anodyne PAPA1_CARPA 19 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880807206 GG On-Demand Anodyne CCR8 46 39 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880807207 GG On-Demand Anodyne CCR8 46 39 C#C[C@@](C)(CC)NC(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880807626 EH On-Demand Mild IMDH_CRYPV 43 34 C#C[C@](C)(CC)NC(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880807627 EH On-Demand Mild IMDH_CRYPV 43 34 C[C@H]1[C@H](C(=O)NCc2nnc3ccc(Cl)cn23)CCN1C ZINC000880808235 DD On-Demand Anodyne SLC6A3 17 40 C[C@H]1[C@H](C(=O)NCc2nnc3ccc(Cl)cn23)CCN1C ZINC000880808235 DD On-Demand Anodyne P2RX7 40 37 C[C@@H]1[C@@H](C(=O)NCc2nnc3ccc(Cl)cn23)CCN1C ZINC000880808236 DD On-Demand Anodyne SLC6A3 17 40 C[C@@H]1[C@@H](C(=O)NCc2nnc3ccc(Cl)cn23)CCN1C ZINC000880808236 DD On-Demand Anodyne P2RX7 40 37 CCNc1nc(C)c(C(=O)NCc2nnc3ccc(Cl)cn23)s1 ZINC000880808264 FF On-Demand Anodyne SCD1 29 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880808674 FE On-Demand Anodyne LGMN 51 34 C#CC(C)(C)NC(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880808895 DG On-Demand Mild IMDH_CRYPV 41 34 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880809128 GF On-Demand Anodyne EPHX2 36 53 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C(C)=O)ccc2Br)C1 ZINC000880809129 GF On-Demand Anodyne EPHX2 36 53 COC(=O)C[C@H]1CCCN1C(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880809344 GG On-Demand Anodyne ACKR3 61 32 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880809345 GG On-Demand Anodyne ACKR3 61 32 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne HTR1A 53 41 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne DRD2 39 41 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne DRD4 22 40 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne HTR1D 17 48 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne HTR1B 26 48 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne DRD3 48 40 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne PDGFRB 45 42 CCOc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809568 GE On-Demand Anodyne HTR7 39 42 COC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809585 EF On-Demand Anodyne RAF1 16 43 COC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809585 EF On-Demand Anodyne KCNK3 73 42 COC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809585 EF On-Demand Anodyne KCNK9 66 37 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809597 GI On-Demand Anodyne CCR3 47 51 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809597 GI On-Demand Anodyne FAAH 17 43 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809597 GI On-Demand Anodyne EPHX2 22 42 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne PDGFRB 37 47 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne CCR3 15 42 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne FAAH 29 55 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne S1PR2 28 47 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne EPHX2 35 42 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne P2RY14 47 34 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne LIMK2 26 46 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne KCNK3 77 42 CC(=O)N1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809614 FG On-Demand Anodyne KCNK9 64 40 Cc1ccccc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880809648 CD On-Demand Anodyne P2RX7 32 40 COCCN(CCO)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809698 EG On-Demand Anodyne KCNK3 78 43 COCCN(CCO)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809698 EG On-Demand Anodyne KCNK9 64 38 COC[C@@H](CCO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809706 EG On-Demand Anodyne KCNK3 72 40 COC[C@@H](CCO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809706 EG On-Demand Anodyne KCNK9 68 35 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne HRH2 36 41 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne CA1 26 41 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne CCR3 25 41 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne RAF1 20 41 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne MTNR1A 15 41 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne MTNR1B 17 45 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne EPHX2 19 44 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne KCNK3 66 39 CNC(=O)CCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809722 EG On-Demand Anodyne KCNK9 60 37 COc1cccc([C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)N2CCCC2)c1 ZINC000880809736 GE On-Demand Anodyne DRD4 41 31 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne CACNA1H 49 33 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne PDGFRB 41 41 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne FAAH 23 48 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne S1PR2 35 57 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne EPHX2 36 41 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne LIMK2 28 42 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne KCNK3 60 39 COCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809746 FH On-Demand Anodyne KCNK9 50 35 COc1ccc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880809761 FD On-Demand Clean HTR1B 16 45 COc1ccc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880809761 FD On-Demand Clean PDGFRB 41 36 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne PDGFRB 29 41 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne CCR3 44 46 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne FAAH 23 48 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne S1PR2 26 43 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne EPHX2 46 45 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne LIMK2 21 40 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne KCNK3 49 36 CC(=O)NCC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880809813 GI On-Demand Anodyne KCNK9 40 34 COc1ccc(C)cc1CN1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880809947 GD On-Demand Anodyne SLC9A1 45 31 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880809952 FE On-Demand Anodyne BMP1 47 35 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880809952 FE On-Demand Anodyne NOS2 63 34 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne HRH2 31 43 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne INHA 15 41 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne CA1 29 44 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne CCR3 32 43 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne RAF1 21 43 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne MTNR1A 58 44 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne MTNR1B 60 44 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne CCKBR 20 40 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne EPHX2 21 41 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne KCNK3 74 41 CC(=O)NCCCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880809976 EG On-Demand Anodyne KCNK9 63 39 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809992 GI On-Demand Anodyne CCKAR 23 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809992 GI On-Demand Anodyne CCR3 88 47 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809992 GI On-Demand Anodyne CCKBR 35 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809992 GI On-Demand Anodyne EPHX2 36 48 CC(=O)N1CCC[C@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809992 GI On-Demand Anodyne MCHR1 16 43 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809993 GI On-Demand Anodyne CCKAR 23 41 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809993 GI On-Demand Anodyne CCR3 88 47 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809993 GI On-Demand Anodyne CCKBR 35 41 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809993 GI On-Demand Anodyne EPHX2 36 48 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880809993 GI On-Demand Anodyne MCHR1 16 43 CCc1nnc2n1CCN(C(=O)Nc1cccc(Oc3cccc(C)c3)c1)C2 ZINC000880809996 GH On-Demand Anodyne P2RX7 19 44 CCc1nnc2n1CCN(C(=O)Nc1cccc(Oc3cccc(C)c3)c1)C2 ZINC000880809996 GH On-Demand Anodyne FAAH 20 44 CCc1nnc2n1CCN(C(=O)Nc1cccc(Oc3cccc(C)c3)c1)C2 ZINC000880809996 GH On-Demand Anodyne S1PR2 25 40 CCc1nnc2n1CCN(C(=O)Nc1cccc(Oc3cccc(C)c3)c1)C2 ZINC000880809996 GH On-Demand Anodyne P2RY14 50 37 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne ADRB2 18 48 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne ADRB1 47 44 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne RAF1 18 42 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne MTNR1B 17 45 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne KCNK3 70 41 COC[C@@H](O)CNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810002 EF On-Demand Anodyne KCNK9 61 37 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne CCKAR 19 40 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne CCR3 22 43 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne FAAH 26 46 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne S1PR2 25 42 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne EPHX2 48 51 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne MCHR1 19 40 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne CCR8 23 43 COCC(=O)NC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810047 GH On-Demand Anodyne KCNK3 49 37 C#CCN(C(=O)Nc1cccc(Oc2cccc(C)c2)c1)[C@@H]1CCS(=O)(=O)C1 ZINC000880810214 GG On-Demand Mild KCNK3 44 34 C#CCN(C(=O)Nc1cccc(Oc2cccc(C)c2)c1)[C@H]1CCS(=O)(=O)C1 ZINC000880810216 GG On-Demand Mild KCNK3 44 34 CNC(=O)[C@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880810230 FF On-Demand Anodyne KCNK3 44 35 CNC(=O)[C@@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880810232 FF On-Demand Anodyne KCNK3 44 35 CC(=O)Nc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880810253 ED On-Demand Anodyne ROCK2 18 47 C[C@@H](CCc1ccccc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880810313 EE On-Demand Anodyne ACE 42 38 C[C@H](CCc1ccccc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880810316 EE On-Demand Anodyne ACE 42 38 CCOc1ccccc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880810371 EE On-Demand Anodyne HCN1 61 39 CCOc1ccccc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880810371 EE On-Demand Anodyne HCN4 41 32 COc1ccc(OCCNC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880810412 ED On-Demand Anodyne HRH2 22 42 CC(=O)NC[C@@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880810433 GG On-Demand Anodyne FAAH 16 42 CCN1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880810440 DC On-Demand Anodyne CACNA1I 62 35 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@H]1CCc2ccccc21 ZINC000880810452 FF On-Demand Anodyne CA6 17 46 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@H]1CCc2ccccc21 ZINC000880810452 FF On-Demand Anodyne CA7 17 46 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@H]1CCc2ccccc21 ZINC000880810452 FF On-Demand Anodyne CA13 32 46 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@@H]1CCc2ccccc21 ZINC000880810454 FF On-Demand Anodyne CA6 17 46 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@@H]1CCc2ccccc21 ZINC000880810454 FF On-Demand Anodyne CA7 17 46 CN(C(=O)c1ccc(Cl)c(S(N)(=O)=O)c1)[C@@H]1CCc2ccccc21 ZINC000880810454 FF On-Demand Anodyne CA13 32 46 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne PDGFRB 35 42 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne FAAH 21 47 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne S1PR2 31 51 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne LIMK2 28 43 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne KCNK3 63 40 COC(=O)C1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810475 GG On-Demand Anodyne KCNK9 50 35 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne PDGFRB 28 40 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne CCR3 28 46 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne FAAH 22 47 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne S1PR2 26 42 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne EPHX2 34 44 CNC(=O)CC1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810479 GI On-Demand Anodyne KCNK3 49 35 COc1cc2c(cc1OC)CN(C(=O)Nc1cc3n(n1)CCN(C)C3)CC2 ZINC000880810546 FD On-Demand Anodyne ABCB1 15 41 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne PDGFRB 27 41 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne CCR3 15 41 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne FAAH 21 48 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne S1PR2 25 41 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne EPHX2 39 44 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne LIMK2 28 44 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne KCNK3 57 37 CC(=O)N(C)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810619 GI On-Demand Anodyne KCNK9 45 35 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880810674 EE On-Demand Anodyne ROCK2 19 40 COCC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810686 EG On-Demand Anodyne RAF1 20 42 COCC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810686 EG On-Demand Anodyne EPHX2 21 40 COCC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810686 EG On-Demand Anodyne KCNK3 85 44 COCC[C@@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810686 EG On-Demand Anodyne KCNK9 77 39 CCC(=O)Nc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880810687 FD On-Demand Anodyne ROCK2 17 41 COCC[C@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810689 EG On-Demand Anodyne RAF1 20 42 COCC[C@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810689 EG On-Demand Anodyne EPHX2 21 40 COCC[C@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810689 EG On-Demand Anodyne KCNK3 85 44 COCC[C@H](CO)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810689 EG On-Demand Anodyne KCNK9 77 39 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne PDGFRB 30 40 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne FAAH 17 44 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne S1PR2 24 40 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne EPHX2 33 42 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne LIMK2 26 44 CON(C)C(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880810699 GI On-Demand Anodyne KCNK3 47 37 COC[C@@H](O)CCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810732 EG On-Demand Anodyne ADRB1 44 41 COC[C@@H](O)CCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810732 EG On-Demand Anodyne HRH2 23 42 COC[C@@H](O)CCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810732 EG On-Demand Anodyne MTNR1B 15 43 COC[C@@H](O)CCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810732 EG On-Demand Anodyne KCNK3 66 40 COC[C@@H](O)CCNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810732 EG On-Demand Anodyne KCNK9 55 35 Cc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880810776 CD On-Demand Anodyne ROCK2 15 45 CCCNC(=O)c1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880810788 FD On-Demand Anodyne DRD4 40 31 CCCNC(=O)c1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880810788 FD On-Demand Anodyne ROCK2 17 42 CNC(=O)CCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810871 EG On-Demand Anodyne LTA4H 21 47 CNC(=O)CCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810871 EG On-Demand Anodyne MTNR1B 15 45 CNC(=O)CCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810871 EG On-Demand Anodyne KCNK3 82 41 CNC(=O)CCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880810871 EG On-Demand Anodyne KCNK9 67 39 COc1ccc(CN(C)C(=O)Nc2cc3n(n2)CCN(C)C3)cc1OC ZINC000880810916 FE On-Demand Anodyne MT-ND1 17 40 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne HTR1A 90 61 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne DRD2 65 48 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne DRD4 34 41 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne ADRA1D 65 40 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne HTR1D 22 61 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne HTR1B 30 61 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne HTR2A 22 49 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne ADRA1A 59 40 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne ADRA1B 52 41 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne DRD3 70 40 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne PDGFRB 55 42 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne HTR7 56 53 COc1ccccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810919 FD On-Demand Anodyne RBP4 19 48 Cc1ccccc1CN1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810958 GE On-Demand Anodyne DRD4 16 50 Cc1ccccc1CN1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880810958 GE On-Demand Anodyne SIGMAR1 15 43 COCCc1noc(CN(C)C(=O)Nc2cccc(Oc3cccc(C)c3)c2)n1 ZINC000880811028 GI On-Demand Anodyne KCNK3 61 36 COCCc1noc(CN(C)C(=O)Nc2cccc(Oc3cccc(C)c3)c2)n1 ZINC000880811028 GI On-Demand Anodyne KCNK9 53 34 CCCCCNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880811043 CD On-Demand Anodyne ASAH1 53 32 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild CCKAR 15 42 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild CCR3 16 41 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild FAAH 20 46 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild CCKBR 20 42 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild S1PR2 25 41 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild EPHX2 49 43 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild LIMK2 24 43 C#CCNC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811047 GH On-Demand Mild KCNK3 43 34 CC(C)c1ccc(CN2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880811055 GF On-Demand Anodyne FAAH 16 42 COCC1(O)CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811088 EG On-Demand Anodyne FAAH 19 45 COCC1(O)CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811088 EG On-Demand Anodyne S1PR2 28 46 COCC1(O)CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811088 EG On-Demand Anodyne EPHX2 26 40 COCC1(O)CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811088 EG On-Demand Anodyne KCNK3 65 40 COCC1(O)CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811088 EG On-Demand Anodyne KCNK9 54 35 COC[C@@H]1CCCN1C(=O)Nc1cc(C(C)=O)ccc1Br ZINC000880811105 FG On-Demand Anodyne ACKR3 61 32 COC(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cn1 ZINC000880811116 GE On-Demand Anodyne BDKRB1 20 43 COC(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cn1 ZINC000880811116 GE On-Demand Anodyne CCR8 41 40 CC(C)c1ccc(OC2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880811200 GH On-Demand Anodyne EPHX2 18 42 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880811218 GD On-Demand Anodyne EPHX2 29 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880811220 FC On-Demand Anodyne CCR8 44 34 CCOc1ccc([C@@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880811266 EF On-Demand Anodyne ACACB 19 42 Cc1nn(-c2ccccc2)c(C)c1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880811320 GE On-Demand Anodyne P2RX7 19 46 COc1ccc(CN(C(=O)Nc2cc3n(n2)CCN(C)C3)C2CC2)cc1 ZINC000880811335 FF On-Demand Anodyne BMP1 42 33 CNC(=O)C[C@H](C)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811371 EG On-Demand Anodyne KCNK3 69 39 CNC(=O)C[C@H](C)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811371 EG On-Demand Anodyne KCNK9 64 37 CNC(=O)C[C@@H](C)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811372 EG On-Demand Anodyne KCNK3 69 39 CNC(=O)C[C@@H](C)NC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811372 EG On-Demand Anodyne KCNK9 64 37 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne FAAH 18 43 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne S1PR2 29 47 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne EPHX2 35 40 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne LIMK2 25 40 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne KCNK3 54 38 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811377 FF On-Demand Anodyne KCNK9 44 34 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne PDGFRB 26 41 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne CCR3 20 43 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne FAAH 23 48 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne CCKBR 20 41 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne S1PR2 26 43 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne EPHX2 52 46 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne LIMK2 25 42 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne KCNK3 62 39 CC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811386 FJ On-Demand Anodyne KCNK9 47 37 C#CCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811439 FI On-Demand Mild PDGFRB 29 40 C#CCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811439 FI On-Demand Mild FAAH 21 46 C#CCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811439 FI On-Demand Mild S1PR2 34 55 C#CCC1(O)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880811439 FI On-Demand Mild KCNK3 44 35 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880811600 GE On-Demand Anodyne ROCK2 17 40 COc1ccc(OC2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880811604 GE On-Demand Anodyne PRSS2 55 32 COc1ccc(OC2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1 ZINC000880811604 GE On-Demand Anodyne EPHX2 19 46 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive KIT 18 40 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive CCKAR 21 40 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive RAF1 18 42 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive KDR 23 40 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive KCNK3 80 44 COCCOCC(=O)NNC(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880811829 FF On-Demand Reactive KCNK9 69 39 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811841 GG On-Demand Anodyne FAAH 15 42 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811841 GG On-Demand Anodyne S1PR2 28 45 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811841 GG On-Demand Anodyne EPHX2 30 41 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811842 GG On-Demand Anodyne FAAH 15 42 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811842 GG On-Demand Anodyne S1PR2 28 45 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880811842 GG On-Demand Anodyne EPHX2 30 41 CN(C)CCOc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880811951 FD On-Demand Anodyne ROCK2 31 46 CC(=O)NCCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880812176 EG On-Demand Anodyne MTNR1A 41 44 CC(=O)NCCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880812176 EG On-Demand Anodyne MTNR1B 40 44 CC(=O)NCCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880812176 EG On-Demand Anodyne KCNK3 66 39 CC(=O)NCCN(C)C(=O)Nc1cccc(Oc2cccc(C)c2)c1 ZINC000880812176 EG On-Demand Anodyne KCNK9 51 37 CO[C@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880812260 EH On-Demand Anodyne FAAH 15 43 CO[C@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880812260 EH On-Demand Anodyne LIMK2 31 40 CO[C@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880812260 EH On-Demand Anodyne KCNK3 59 38 CO[C@H]1CN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CCO1 ZINC000880812260 EH On-Demand Anodyne KCNK9 49 34 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne PDGFRB 28 41 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne FAAH 21 45 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne CCKBR 19 43 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne S1PR2 25 41 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne EPHX2 44 43 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne LIMK2 28 45 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne KCNK3 57 38 CONC(=O)C1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812306 GH On-Demand Anodyne KCNK9 44 34 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne CCR3 17 45 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne FAAH 19 44 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne CCKBR 18 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne EPHX2 49 44 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne LIMK2 27 42 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne KCNK3 57 37 CNC(=O)[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812372 FG On-Demand Anodyne KCNK9 44 35 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne CCKAR 18 40 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne CCR3 30 43 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne FAAH 20 45 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne S1PR2 24 40 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne EPHX2 42 49 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne KCNK3 63 37 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812394 FH On-Demand Anodyne KCNK9 51 35 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne CCKAR 18 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne CCR3 30 43 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne FAAH 20 45 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne S1PR2 24 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne EPHX2 42 49 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne KCNK3 63 37 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812395 FH On-Demand Anodyne KCNK9 51 35 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne PDGFRB 31 41 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne FAAH 26 52 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne NPY5R 18 41 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne S1PR2 30 52 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne EPHX2 33 40 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne LIMK2 29 42 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne KCNK3 59 38 COC1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)CC1 ZINC000880812416 FH On-Demand Anodyne KCNK9 49 34 COC[C@]1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812424 FH On-Demand Anodyne FAAH 21 45 COC[C@]1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812424 FH On-Demand Anodyne S1PR2 28 46 COC[C@]1(CO)CCN(C(=O)Nc2cccc(Oc3cccc(C)c3)c2)C1 ZINC000880812424 FH On-Demand Anodyne EPHX2 40 36 CSCC[C@H](NC(=O)Nc1cccc(Oc2cccc(C)c2)c1)C(N)=O ZINC000880812429 FH On-Demand Anodyne FPR1 39 41 CSCC[C@H](NC(=O)Nc1cccc(Oc2cccc(C)c2)c1)C(N)=O ZINC000880812429 FH On-Demand Anodyne KCNK3 50 36 CSCC[C@H](NC(=O)Nc1cccc(Oc2cccc(C)c2)c1)C(N)=O ZINC000880812429 FH On-Demand Anodyne KCNK9 40 34 CC[C@@H](NC(=O)Nc1cc2n(n1)CCN(C)C2)c1ccccc1 ZINC000880812534 DF On-Demand Anodyne TACR3 47 37 COc1cccc(C2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)c1 ZINC000880812555 FF On-Demand Anodyne MCHR1 20 40 COc1ccc(OCCCNC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812589 FD On-Demand Anodyne HRH2 26 45 COc1ccccc1C[C@@H]1CCCN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880812592 FF On-Demand Anodyne ACKR3 63 33 COc1ccccc1C[C@H]1CCCN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880812593 FF On-Demand Anodyne ACKR3 63 33 COc1ccc2c(c1)CN(C(=O)Nc1cc3n(n1)CCN(C)C3)CC2 ZINC000880812629 ED On-Demand Anodyne DRD5 17 40 CC(=O)NCC1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812671 EC On-Demand Anodyne CACNA1I 49 32 COc1ccc(CC[C@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812890 FE On-Demand Anodyne BMP1 49 34 COc1ccc(CC[C@@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812891 FE On-Demand Anodyne BMP1 49 34 CCCOc1ccc([C@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812912 FG On-Demand Anodyne ACACA 18 46 CCCOc1ccc([C@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812912 FG On-Demand Anodyne ACACB 19 46 CCCOc1ccc([C@@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812913 FG On-Demand Anodyne ACACA 18 46 CCCOc1ccc([C@@H](C)NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880812913 FG On-Demand Anodyne ACACB 19 46 COCCN(Cc1ccc(C#N)cc1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880812920 FD On-Demand Mild ITK 20 40 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne HTR1A 75 51 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne DRD2 61 47 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne DRD4 34 41 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne ADRA1D 66 47 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne HTR1D 15 51 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne HTR1B 20 51 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne ADRA1A 56 47 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne ADRA1B 53 47 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne DRD3 65 42 COc1ccccc1N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880812975 GE On-Demand Anodyne HTR7 47 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812979 GD On-Demand Anodyne HTR1A 63 45 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812979 GD On-Demand Anodyne DRD2 46 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812979 GD On-Demand Anodyne ADRA1D 40 35 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812979 GD On-Demand Anodyne DRD3 54 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812979 GD On-Demand Anodyne HTR7 42 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812980 GD On-Demand Anodyne HTR1A 63 45 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812980 GD On-Demand Anodyne DRD2 46 40 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812980 GD On-Demand Anodyne ADRA1D 40 35 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812980 GD On-Demand Anodyne DRD3 54 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880812980 GD On-Demand Anodyne HTR7 42 39 C[C@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813082 FE On-Demand Anodyne BMP1 60 37 C[C@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813082 FE On-Demand Anodyne NOS2 93 38 C[C@@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813083 FE On-Demand Anodyne BMP1 60 37 C[C@@H](CCc1ccc2c(c1)OCO2)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813083 FE On-Demand Anodyne NOS2 93 38 CCC1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880813094 DF On-Demand Anodyne CACNA1I 49 33 CCN(Cc1ccc(Cl)cc1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813161 EG On-Demand Anodyne FFAR2 37 40 C[C@@H](Nc1ccc(NC(=O)Nc2cc3n(n2)CCN(C)C3)cc1)c1ccccc1 ZINC000880813483 GI On-Demand Anodyne FPR2 41 33 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne HTR1A 17 53 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne HTR1D 73 42 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne HTR1B 61 53 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne NQO2 32 44 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne MTNR1A 74 61 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne MTNR1B 59 55 COc1ccc2[nH]cc(CCNC(=O)Nc3cc4n(n3)CCN(C)C4)c2c1 ZINC000880813601 FE On-Demand Anodyne ABCG2 25 40 COc1ccccc1[C@H](CC(C)C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813626 FG On-Demand Anodyne ABCC8 20 42 CSc1ccc(F)cc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813656 EF On-Demand Anodyne P2RX7 43 39 COCCN(Cc1cccnc1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813695 ED On-Demand Anodyne CHRNA7 43 35 Cc1ccccc1[C@H](CO)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813709 ED On-Demand Anodyne CTSA 53 34 Cc1ccccc1[C@@H](CO)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813711 ED On-Demand Anodyne CTSA 53 34 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813756 GD On-Demand Anodyne BMP1 57 36 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880813756 GD On-Demand Anodyne NOS2 47 33 Cc1cccc(C(C)(C)NC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880813810 EF On-Demand Anodyne IMDH_CRYPV 59 35 C[C@@H](Cn1cncn1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814056 DC On-Demand Anodyne HIS3 75 34 C[C@@H](C1CC1)N(Cc1ccccc1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814126 FG On-Demand Anodyne BRCA1 43 30 COc1cccc(OCCCNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880814128 FD On-Demand Anodyne DRD4 43 33 COc1cccc(OCCCNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880814128 FD On-Demand Anodyne HRH2 40 49 COc1cccc(OCCCNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880814128 FD On-Demand Anodyne MTNR1A 37 46 COc1cccc(OCCCNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880814128 FD On-Demand Anodyne MTNR1B 41 46 CCOc1ccccc1CCNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814141 EE On-Demand Anodyne HCN1 49 36 COCCN(Cc1ccc(F)cc1Cl)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814158 GF On-Demand Anodyne P2RX7 47 40 COCCC(=O)N1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880814266 FC On-Demand Anodyne EPHX2 27 40 COc1cccc(C=C2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)c1 ZINC000880814307 GG On-Demand Anodyne DRD4 40 30 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814341 GD On-Demand Anodyne P2RX3 27 44 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880814384 EF On-Demand Anodyne TRPM8 20 41 CCOc1cc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)ccc1OC ZINC000880814394 FE On-Demand Anodyne SSTR5 40 38 CCOc1cc(CCCNC(=O)Nc2cc3n(n2)CCN(C)C3)ccc1OC ZINC000880814733 GE On-Demand Anodyne SSTR5 43 36 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880814763 FE On-Demand Anodyne HTR1B 15 43 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880814763 FE On-Demand Anodyne RBP4 35 41 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880814764 FE On-Demand Anodyne HTR1B 15 43 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880814764 FE On-Demand Anodyne RBP4 35 41 Cc1ccccc1C1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880814838 FG On-Demand Anodyne HTR1F 59 37 CN1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)(N2CCCCC2)CC1 ZINC000880814892 GD On-Demand Anodyne HCN1 61 40 CN1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)(N2CCCCC2)CC1 ZINC000880814892 GD On-Demand Anodyne HCN4 49 31 COc1cccc([C@H](CO)NC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880815074 ED On-Demand Anodyne ROCK1 15 41 CCN(Cc1cccc(-c2ccncc2)c1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815152 GG On-Demand Anodyne FSHR 42 32 CCCCN1CCC(NC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880815238 ED On-Demand Anodyne HTR4 36 40 COc1ccnc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)n1 ZINC000880815330 FC On-Demand Anodyne FAAH 21 40 Cc1cccc2c1CCN(C(=O)Nc1cc3n(n1)CCN(C)C3)C2 ZINC000880815337 EE On-Demand Anodyne P2RY14 47 33 CN1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880815582 DC On-Demand Anodyne CACNA1I 63 37 COc1ccc(CN(C(=O)Nc2cc3n(n2)CCN(C)C3)[C@@H](C)C2CC2)cc1 ZINC000880815898 GG On-Demand Anodyne BMP1 44 33 COc1ccc(CN(C(=O)Nc2cc3n(n2)CCN(C)C3)[C@H](C)C2CC2)cc1 ZINC000880815901 GG On-Demand Anodyne BMP1 44 33 Cc1noc(C2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)n1 ZINC000880815910 ED On-Demand Anodyne SMO 36 40 Cc1noc(C2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)n1 ZINC000880815910 ED On-Demand Anodyne ETHR 52 34 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815931 EE On-Demand Anodyne OPRD1 45 32 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815931 EE On-Demand Anodyne CFTR 61 34 C[C@H]1Cc2ccccc2CN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815932 EE On-Demand Anodyne OPRD1 45 32 C[C@H]1Cc2ccccc2CN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815932 EE On-Demand Anodyne CFTR 61 34 C[C@@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815979 GE On-Demand Anodyne DRD4 29 47 C[C@@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815979 GE On-Demand Anodyne SIGMAR1 25 40 C[C@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815980 GE On-Demand Anodyne DRD4 29 47 C[C@H]1CN(Cc2ccccc2)CC[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815980 GE On-Demand Anodyne SIGMAR1 25 40 C[C@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815982 GE On-Demand Anodyne DRD4 29 47 C[C@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815982 GE On-Demand Anodyne SIGMAR1 25 40 C[C@@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815984 GE On-Demand Anodyne DRD4 29 47 C[C@@H]1CN(Cc2ccccc2)CC[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880815984 GE On-Demand Anodyne SIGMAR1 25 40 CN(CCNC(=O)Nc1cc2n(n1)CCN(C)C2)Cc1ccc(F)cc1 ZINC000880815986 FD On-Demand Anodyne CCR3 33 44 COc1cccc(O[C@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816171 FD On-Demand Anodyne DRD4 41 31 COc1cccc(O[C@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816171 FD On-Demand Anodyne MTNR1A 26 51 COc1cccc(O[C@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816171 FD On-Demand Anodyne MTNR1B 30 51 COc1cccc(O[C@@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816172 FD On-Demand Anodyne DRD4 41 31 COc1cccc(O[C@@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816172 FD On-Demand Anodyne MTNR1A 26 51 COc1cccc(O[C@@H](C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816172 FD On-Demand Anodyne MTNR1B 30 51 C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880816346 FE On-Demand Anodyne CCR3 47 37 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880816347 FE On-Demand Anodyne CCR3 47 37 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816547 DC On-Demand Anodyne EPHX2 26 46 CCC(=O)N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816548 DC On-Demand Anodyne EPHX2 26 46 COc1ccc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)cc1F ZINC000880816568 GD On-Demand Clean RBP4 17 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1=O ZINC000880816599 GD On-Demand Anodyne HTR1A 29 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1=O ZINC000880816600 GD On-Demand Anodyne HTR1A 29 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne HTR1A 55 47 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne DRD2 42 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne ADRA1D 43 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne ADRA1A 37 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne ADRA1B 32 42 COc1ccccc1N1CC[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816623 FD On-Demand Anodyne DRD3 50 38 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne HTR1A 55 47 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne DRD2 42 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne ADRA1D 43 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne ADRA1A 37 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne ADRA1B 32 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880816624 FD On-Demand Anodyne DRD3 50 38 COC(=O)c1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880816654 ED On-Demand Anodyne ROCK2 23 42 C[C@H]1C[C@H](NC(=O)Nc2cc3n(n2)CCN(C)C3)CCN1Cc1ccccc1 ZINC000880816729 GF On-Demand Anodyne SIGMAR1 17 41 CCOc1cc(Cl)ccc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880816986 FF On-Demand Anodyne P2RX7 48 39 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880817167 CD On-Demand Anodyne TRPC6 49 34 C[C@@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)[C@@H]1C ZINC000880817170 CD On-Demand Anodyne TRPC6 49 34 CCCOc1cccc(CCNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880817233 FE On-Demand Anodyne HRH2 37 43 Cc1cc(C)cc(C2=CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)c1 ZINC000880817368 FG On-Demand Anodyne ADAM10 20 40 Cc1cncc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880817379 DD On-Demand Anodyne NAMPT 18 46 COc1cccc(C(C)(C)CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880817515 FE On-Demand Anodyne DRD4 41 31 COCCCOc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880817789 FE On-Demand Anodyne HRH2 33 41 COCCCOc1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880817789 FE On-Demand Anodyne ROCK2 33 41 CCCCCCCCNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880817816 DF On-Demand Mild ASAH1 75 34 COc1cccc(C2=CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)C2)c1 ZINC000880817898 FE On-Demand Anodyne ADAM10 15 42 CC[C@@H](C(=O)NNC(=O)Nc1cc2n(n1)CCN(C)C2)c1ccccc1 ZINC000880817911 FD On-Demand Reactive KCNQ2 46 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818069 FD On-Demand Anodyne DRD4 18 46 C[C@H]1CN(Cc2ccccc2)C[C@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818070 FD On-Demand Anodyne DRD4 18 46 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818071 FD On-Demand Anodyne DRD4 18 46 C[C@H]1CN(Cc2ccccc2)C[C@@H]1NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818072 FD On-Demand Anodyne DRD4 18 46 COc1cc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)ncn1 ZINC000880818454 FC On-Demand Anodyne PDGFRB 45 38 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818669 FE On-Demand Anodyne NPY5R 15 40 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818670 FE On-Demand Anodyne NPY5R 15 40 COC(=O)[C@@H](Cc1ccccc1)[C@@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818746 GD On-Demand Anodyne BRCA1 42 29 COC(=O)[C@H](Cc1ccccc1)[C@@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818747 GD On-Demand Anodyne BRCA1 42 29 COC(=O)[C@H](Cc1ccccc1)[C@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818748 GD On-Demand Anodyne BRCA1 42 29 COC(=O)[C@@H](Cc1ccccc1)[C@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880818749 GD On-Demand Anodyne BRCA1 42 29 COc1cnccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880818800 FD On-Demand Anodyne HTR1A 15 48 COc1cnccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880818800 FD On-Demand Anodyne HTR1B 20 48 COc1cnccc1N1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880818800 FD On-Demand Anodyne PDGFRB 44 42 CCn1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1=O ZINC000880818860 EC On-Demand Anodyne P2RX7 42 36 CCCN(CCN1CCCC1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819165 ED On-Demand Anodyne CASR 45 38 CCSCCCNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819210 CD On-Demand Anodyne DOT1L 41 32 COc1cc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)ccc1F ZINC000880819235 GD On-Demand Anodyne RBP4 18 40 C[C@@H](c1ccccc1)N(C(=O)Nc1cc2n(n1)CCN(C)C2)C1CC1 ZINC000880819238 EG On-Demand Anodyne CCR5 30 41 CCCN(CCN1CCCCC1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819247 EE On-Demand Anodyne CASR 43 37 COCCC[C@@H](Cc1ccccc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819383 FE On-Demand Anodyne TACR2 47 33 COCCC[C@H](Cc1ccccc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819384 FE On-Demand Anodyne TACR2 47 33 Cc1ccccc1[C@H](CC(F)(F)F)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819467 GG On-Demand Anodyne CTSA 53 34 Cc1ccccc1[C@@H](CC(F)(F)F)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819469 GG On-Demand Anodyne CTSA 53 34 C[C@H](O)[C@](C)(CNC(=O)Nc1cc2n(n1)CCN(C)C2)Cc1ccccc1 ZINC000880819852 FE On-Demand Anodyne Q82323_9DELA 73 32 CCCN(CCN1CCCCCC1)C(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880819869 FE On-Demand Anodyne CASR 43 37 Cc1cc(F)ccc1C1CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880820095 FG On-Demand Anodyne HTR1F 64 37 O=C(/C=C\c1cccnc1)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880820406 FF On-Demand Anodyne CHRNA7 40 50 O=C(/C=C\c1cccnc1)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880820406 FF On-Demand Anodyne C3AR1 45 57 O=C(/C=C\c1cccnc1)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880820406 FF On-Demand Anodyne EPHX2 31 44 O=C(/C=C\c1cccnc1)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880820406 FF On-Demand Anodyne ACHP_LYMST 17 40 O=C(/C=C\c1cccnc1)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000880820406 FF On-Demand Anodyne NAMPT 27 51 COc1cccc(C2(CNC(=O)Nc3cc4n(n3)CCN(C)C4)CC2)c1 ZINC000880820655 FE On-Demand Anodyne DRD4 40 31 COc1cccc(C2(CNC(=O)Nc3cc4n(n3)CCN(C)C4)CC2)c1 ZINC000880820655 FE On-Demand Anodyne SOAT1 21 51 CC[C@@H](CN(CC)C(=O)Nc1cc2n(n1)CCN(C)C2)c1ccccc1 ZINC000880820808 FG On-Demand Anodyne CASR 43 38 CC[C@H](CN(CC)C(=O)Nc1cc2n(n1)CCN(C)C2)c1ccccc1 ZINC000880820809 FG On-Demand Anodyne CASR 43 38 C[C@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880820939 GE On-Demand Anodyne FAAH 18 43 C[C@@H]1CN(Cc2ccccc2)CCN(C(=O)Nc2cc3n(n2)CCN(C)C3)C1 ZINC000880820940 GE On-Demand Anodyne FAAH 18 43 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880821071 EE On-Demand Anodyne PTAFR 33 47 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880821071 EE On-Demand Anodyne CHRNA7 43 36 COc1ccc(CN(C)C(=O)Nc2cc3n(n2)CCN(C)C3)cc1Cl ZINC000880821172 FF On-Demand Anodyne PDE6A 41 31 CCn1ncc(C(=O)N(C)NC(=O)OCc2ccccc2)c1C1CC1 ZINC000880821344 EF On-Demand Reactive CAPN1 42 34 CCn1ncc(C(=O)N(C)NC(=O)OCc2ccccc2)c1C1CC1 ZINC000880821344 EF On-Demand Reactive CAPN2 84 34 CCn1ncc(C(=O)N(C)NC(=O)OCc2ccccc2)c1C1CC1 ZINC000880821344 EF On-Demand Reactive NPR 57 33 C[C@@H](Cc1cn(C)c2ccc(F)cc12)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880821374 GF On-Demand Anodyne CCR3 40 32 Cc1ccncc1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880821430 DD On-Demand Anodyne NAMPT 15 45 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive CYSP_TRYCR 47 34 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive CTSK 20 41 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive CAPNS1 48 34 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive CAPN1 52 35 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive CAPN2 88 34 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive NPR 58 32 Cc1ncc(CC(=O)N(C)NC(=O)OCc2ccccc2)o1 ZINC000880821439 DD On-Demand Reactive NAAA 32 40 COc1ccc(N2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)nc1 ZINC000880821739 FD On-Demand Anodyne PDGFRB 49 36 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive KLK3 44 32 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CTSB 45 37 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive PAPA1_CARPA 51 37 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CYSP_TRYCR 40 33 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CTSK 29 42 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CAPNS1 61 35 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CAPN1 66 37 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive CAPN2 111 36 Cc1nc(C(C)C)ncc1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880821928 EF On-Demand Reactive NPR 70 37 CC(=O)c1cccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c1 ZINC000880822128 ED On-Demand Anodyne ROCK2 20 41 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880822704 EE On-Demand Reactive NAAA 41 39 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880822705 EE On-Demand Reactive NAAA 41 39 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N(C)NC(=O)OCc1ccccc1 ZINC000880822707 EE On-Demand Reactive NAAA 41 39 Cc1cc(F)ccc1C[C@@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880822789 EF On-Demand Anodyne CCR3 45 34 Cc1cc(F)ccc1C[C@H](C)NC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880822790 EF On-Demand Anodyne CCR3 45 34 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@@H]1CCCN(C)[C@@H]1C)C2 ZINC000880822870 FD On-Demand Reactive DRD4 41 33 COC(=O)c1ccc(CNC(=O)Nc2cc3n(n2)CCN(C)C3)c(F)c1 ZINC000880822973 FD On-Demand Anodyne BDKRB1 25 40 COc1cccc([C@H](CNC(=O)CN2CCCCS2(=O)=O)OC)c1 ZINC000880823243 FC On-Demand Anodyne DRD4 41 32 COc1cccc([C@H](CNC(=O)CN2CCCCS2(=O)=O)OC)c1 ZINC000880823243 FC On-Demand Anodyne MTNR1A 40 38 COc1cccc([C@H](CNC(=O)CN2CCCCS2(=O)=O)OC)c1 ZINC000880823243 FC On-Demand Anodyne MTNR1B 45 38 COc1cccc([C@H](CNC(=O)COC2CC2)OC)c1 ZINC000880823328 CD On-Demand Anodyne MTNR1A 79 44 COc1cccc([C@H](CNC(=O)COC2CC2)OC)c1 ZINC000880823328 CD On-Demand Anodyne MTNR1B 71 44 CCn1nncc1CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880823390 EE On-Demand Anodyne ENPP1 65 32 C=CC(C)(C)CC(=O)NC[C@H](OC)c1cccc(OC)c1 ZINC000880823408 CG On-Demand Mild MTNR1A 42 41 C=CC(C)(C)CC(=O)NC[C@H](OC)c1cccc(OC)c1 ZINC000880823408 CG On-Demand Mild MTNR1B 44 41 C=CC(C)(C)CC(=O)NC[C@@H](OC)c1cccc(OC)c1 ZINC000880823409 CG On-Demand Mild MTNR1A 42 41 C=CC(C)(C)CC(=O)NC[C@@H](OC)c1cccc(OC)c1 ZINC000880823409 CG On-Demand Mild MTNR1B 44 41 COc1cccc([C@H](CNC(=O)c2nnn(C)n2)OC)c1 ZINC000880823491 CC On-Demand Anodyne DRD4 45 34 CCCCCCCNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880823517 DF On-Demand Mild EPHX2 15 43 CCCCCCCNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880823517 DF On-Demand Mild ASAH1 53 33 COc1cccc([C@H](CNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)OC)c1 ZINC000880823522 FD On-Demand Anodyne MTNR1A 38 51 COc1cccc([C@H](CNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)OC)c1 ZINC000880823522 FD On-Demand Anodyne MTNR1B 39 51 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CC[C@H](c3nc(C4CC4)no3)O1)C2 ZINC000880823528 GG On-Demand Anodyne MTNR1A 18 41 COc1cccc([C@H](CNC(=O)c2ncsc2C2CC2)OC)c1 ZINC000880823542 EG On-Demand Anodyne MAP1 38 42 COc1cccc([C@H](CNC(=O)[C@H]2CCc3nncn3CC2)OC)c1 ZINC000880823549 ED On-Demand Anodyne DRD4 44 35 COc1cccc([C@H](CNC(=O)[C@H]2CCc3nncn3CC2)OC)c1 ZINC000880823549 ED On-Demand Anodyne MTNR1A 24 46 COc1cccc([C@H](CNC(=O)[C@H]2CCc3nncn3CC2)OC)c1 ZINC000880823549 ED On-Demand Anodyne MTNR1B 29 46 COc1cccc([C@H](CNC(=O)[C@@H]2CCc3nncn3CC2)OC)c1 ZINC000880823550 ED On-Demand Anodyne DRD4 44 35 COc1cccc([C@H](CNC(=O)[C@@H]2CCc3nncn3CC2)OC)c1 ZINC000880823550 ED On-Demand Anodyne MTNR1A 24 46 COc1cccc([C@H](CNC(=O)[C@@H]2CCc3nncn3CC2)OC)c1 ZINC000880823550 ED On-Demand Anodyne MTNR1B 29 46 CCn1nncc1CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880823557 GD On-Demand Anodyne PREP 26 40 CCn1nncc1CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880823557 GD On-Demand Anodyne CAPN2 51 33 CCn1nncc1CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880823557 GD On-Demand Anodyne Q9NAW4_PLAFA 27 41 COc1cccc([C@H](CNC(=O)c2cc(C)cnc2Cl)OC)c1 ZINC000880823583 EG On-Demand Anodyne DRD4 44 33 COc1cccc([C@H](CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)OC)c1 ZINC000880823588 DE On-Demand Anodyne MTNR1A 28 43 COc1cccc([C@H](CNC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)OC)c1 ZINC000880823588 DE On-Demand Anodyne MTNR1B 28 43 COc1cccc([C@H](CNC(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)OC)c1 ZINC000880823621 EF On-Demand Anodyne MTNR1B 15 40 COc1cccc([C@H](CNC(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)OC)c1 ZINC000880823622 EF On-Demand Anodyne MTNR1B 15 40 COc1cccc([C@H](CNC(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)OC)c1 ZINC000880823623 EF On-Demand Anodyne MTNR1B 15 40 COc1cccc([C@H](CNC(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)OC)c1 ZINC000880823624 EF On-Demand Anodyne MTNR1B 15 40 CCCCCCCNC(=O)COC1CC1 ZINC000880823646 BE On-Demand Mild EPHX2 27 49 CCCCCCCNC(=O)COC1CC1 ZINC000880823646 BE On-Demand Mild ASAH1 87 38 CCCCCCCNC(=O)COC1CC1 ZINC000880823646 BE On-Demand Mild LASR 48 34 COc1cccc([C@H](CNC(=O)c2c3c(nn2C)CCSC3)OC)c1 ZINC000880823660 FE On-Demand Anodyne DRD4 44 33 COc1cccc([C@H](CNC(=O)Cc2ccccc2N2CCCC2=O)OC)c1 ZINC000880823736 GF On-Demand Anodyne DRD4 46 37 COc1cccc([C@H](CNC(=O)Cc2ccccc2N2CCCC2=O)OC)c1 ZINC000880823736 GF On-Demand Anodyne HTR7 15 40 COc1cccc([C@H](CNC(=O)Cc2ccccc2N2CCCC2=O)OC)c1 ZINC000880823736 GF On-Demand Anodyne KCNQ2 42 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCCOC1)C2 ZINC000880823749 DF On-Demand Anodyne NQO2 34 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCCOC1)C2 ZINC000880823749 DF On-Demand Anodyne MTNR1A 54 46 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCCOC1)C2 ZINC000880823749 DF On-Demand Anodyne MTNR1B 48 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCCOC1)C2 ZINC000880823752 DF On-Demand Anodyne NQO2 34 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCCOC1)C2 ZINC000880823752 DF On-Demand Anodyne MTNR1A 54 46 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCCOC1)C2 ZINC000880823752 DF On-Demand Anodyne MTNR1B 48 44 CCn1nncc1CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880823783 DD On-Demand Anodyne NQO2 28 40 CCn1nncc1CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880823783 DD On-Demand Anodyne MTNR1A 38 40 CCn1nncc1CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880823784 DD On-Demand Anodyne NQO2 28 40 CCn1nncc1CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880823784 DD On-Demand Anodyne MTNR1A 38 40 COc1cccc([C@H](CNC(=O)CC(C)(C)CC(F)(F)F)OC)c1 ZINC000880823815 EH On-Demand Anodyne MTNR1A 32 41 COc1cccc([C@H](CNC(=O)CC(C)(C)CC(F)(F)F)OC)c1 ZINC000880823815 EH On-Demand Anodyne MTNR1B 33 41 COc1cccc([C@H](CNC(=O)C[C@@H]2C[C@H]2C2CC2)OC)c1 ZINC000880823846 DF On-Demand Anodyne MTNR1A 29 41 COc1cccc([C@H](CNC(=O)C[C@@H]2C[C@H]2C2CC2)OC)c1 ZINC000880823846 DF On-Demand Anodyne MTNR1B 31 41 COc1cccc([C@H](CNC(=O)c2cnc(CC3CC3)s2)OC)c1 ZINC000880823859 EG On-Demand Anodyne MTNR1A 17 40 COc1cccc([C@H](CNC(=O)c2cnc(CC3CC3)s2)OC)c1 ZINC000880823859 EG On-Demand Anodyne MTNR1B 16 40 COc1cccc([C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)OC)c1 ZINC000880823864 FE On-Demand Anodyne DRD4 45 35 COc1cccc([C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)OC)c1 ZINC000880823864 FE On-Demand Anodyne CASR 41 45 CCn1ncc(CNC(=O)c2ccc(OC(F)F)c(Cl)c2)n1 ZINC000880823887 EE On-Demand Anodyne PDE4D 15 40 O=C(NCC[C@H]1CCCOC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880823893 DE On-Demand Anodyne GABRA1 16 44 O=C(NCC[C@@H]1CCCOC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880823894 DE On-Demand Anodyne GABRA1 16 44 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CC[C@H]3C[C@@H]3C2)N1Cc1ccccc1 ZINC000880823898 FE On-Demand Anodyne F2 16 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CC[C@@H]3C[C@H]3C2)N1Cc1ccccc1 ZINC000880823899 FE On-Demand Anodyne F2 16 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CC[C@H]3C[C@H]3C2)N1Cc1ccccc1 ZINC000880823900 FE On-Demand Anodyne F2 16 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CC[C@@H]3C[C@@H]3C2)N1Cc1ccccc1 ZINC000880823901 FE On-Demand Anodyne F2 16 41 O=C(NCc1ccc(-c2ccccc2)s1)[C@H]1CCc2nncn2CC1 ZINC000880823918 FG On-Demand Anodyne PDE8B 41 33 O=C(NCc1ccc(-c2ccccc2)s1)[C@@H]1CCc2nncn2CC1 ZINC000880823919 FG On-Demand Anodyne PDE8B 41 33 O=C(COC1CC1)NCc1ccc(-c2ccccc2)s1 ZINC000880823943 CG On-Demand Anodyne CYP2E1 18 40 COc1cccc([C@H](CNC(=O)CC(C)(C)CC(F)F)OC)c1 ZINC000880824006 EH On-Demand Anodyne MTNR1A 30 41 COc1cccc([C@H](CNC(=O)CC(C)(C)CC(F)F)OC)c1 ZINC000880824006 EH On-Demand Anodyne MTNR1B 32 41 CCn1nncc1CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880824008 CE On-Demand Anodyne NQO2 18 42 CCn1nncc1CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880824008 CE On-Demand Anodyne MTNR1B 15 42 CCn1nncc1CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880824009 CE On-Demand Anodyne NQO2 18 42 CCn1nncc1CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880824009 CE On-Demand Anodyne MTNR1B 15 42 O=C(NCc1ccc(-c2ccccc2)s1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880824074 GG On-Demand Anodyne CYP2E1 18 40 O=C(NCc1ccc(-c2ccccc2)s1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880824074 GG On-Demand Anodyne PDE8B 47 35 NC(=O)[C@@H]1CC[C@H](C(=O)NCC[C@H]2CCCOC2)N1Cc1ccccc1 ZINC000880824099 FD On-Demand Anodyne ACHE 15 40 NC(=O)[C@@H]1CC[C@H](C(=O)NCC[C@@H]2CCCOC2)N1Cc1ccccc1 ZINC000880824100 FD On-Demand Anodyne ACHE 15 40 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cc3n(n1)CCN(C)C3)CC2 ZINC000880824127 GE On-Demand Anodyne SLC18A2 46 35 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cc3n(n1)CCN(C)C3)CC2 ZINC000880824128 GE On-Demand Anodyne SLC18A2 46 35 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC[C@H]3C[C@H]3C2)c1 ZINC000880824129 CG On-Demand Anodyne CACNA1I 49 37 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC[C@@H]3C[C@H]3C2)c1 ZINC000880824130 CG On-Demand Anodyne CACNA1I 49 37 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC[C@@H]3C[C@@H]3C2)c1 ZINC000880824131 CG On-Demand Anodyne CACNA1I 49 37 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CC[C@H]3C[C@@H]3C2)c1 ZINC000880824132 CG On-Demand Anodyne CACNA1I 49 37 CCn1nncc1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880824261 ED On-Demand Anodyne KCNQ2 51 33 COc1cccc([C@H](CNC(=O)c2nccnc2SC)OC)c1 ZINC000880824264 EE On-Demand Anodyne MTNR1A 25 40 COc1cccc([C@H](CNC(=O)c2nccnc2SC)OC)c1 ZINC000880824264 EE On-Demand Anodyne MTNR1B 28 40 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880824291 GE On-Demand Anodyne DRD4 15 45 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880824292 GE On-Demand Anodyne DRD4 15 45 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880824293 GE On-Demand Anodyne DRD4 15 45 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)Nc1cc2n(n1)CCN(C)C2 ZINC000880824294 GE On-Demand Anodyne DRD4 15 45 CCCCCCCNC(=O)CN1CCCCS1(=O)=O ZINC000880824300 CD On-Demand Mild ASAH1 88 35 COc1cccc([C@H](CNC(=O)CC[C@H]2CC(C)(C)CO2)OC)c1 ZINC000880824313 EG On-Demand Anodyne MTNR1A 26 41 COc1cccc([C@H](CNC(=O)CC[C@H]2CC(C)(C)CO2)OC)c1 ZINC000880824313 EG On-Demand Anodyne MTNR1B 26 41 COc1cccc([C@H](CNC(=O)CC[C@@H]2CC(C)(C)CO2)OC)c1 ZINC000880824314 EG On-Demand Anodyne MTNR1A 26 41 COc1cccc([C@H](CNC(=O)CC[C@@H]2CC(C)(C)CO2)OC)c1 ZINC000880824314 EG On-Demand Anodyne MTNR1B 26 41 O=C(NCC[C@H]1CCCOC1)c1cnc(CC2CC2)s1 ZINC000880824443 CF On-Demand Anodyne SIRT3 42 34 O=C(NCC[C@H]1CCCOC1)c1cnc(CC2CC2)s1 ZINC000880824443 CF On-Demand Anodyne SIRT1 42 34 O=C(NCC[C@@H]1CCCOC1)c1cnc(CC2CC2)s1 ZINC000880824444 CF On-Demand Anodyne SIRT3 42 34 O=C(NCC[C@@H]1CCCOC1)c1cnc(CC2CC2)s1 ZINC000880824444 CF On-Demand Anodyne SIRT1 42 34 CCn1ncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)n1 ZINC000880824449 GD On-Demand Anodyne PREP 32 42 CCn1ncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)n1 ZINC000880824449 GD On-Demand Anodyne LGMN 43 33 CCn1ncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)n1 ZINC000880824449 GD On-Demand Anodyne Q9NAW4_PLAFA 26 41 CCn1ncc(CNC(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)n1 ZINC000880824449 GD On-Demand Anodyne VHL 51 34 CCCCCCCNC(=O)C[C@H]1CCNC1=O ZINC000880824455 BD On-Demand Mild ASAH1 95 38 CCCCCCCNC(=O)C[C@H]1CCNC1=O ZINC000880824455 BD On-Demand Mild LASR 49 35 CCCCCCCNC(=O)C[C@@H]1CCNC1=O ZINC000880824456 BD On-Demand Mild ASAH1 95 38 CCCCCCCNC(=O)C[C@@H]1CCNC1=O ZINC000880824456 BD On-Demand Mild LASR 49 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H]2C[C@H]2C1 ZINC000880824620 EE On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H]2C[C@@H]2C1 ZINC000880824621 EE On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@H]2C[C@@H]2C1 ZINC000880824622 EE On-Demand Anodyne PAPA1_CARPA 36 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CC[C@@H]2C[C@H]2C1 ZINC000880824623 EE On-Demand Anodyne PAPA1_CARPA 36 45 O=C(NCC[C@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824626 GF On-Demand Anodyne PREP 29 40 O=C(NCC[C@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824626 GF On-Demand Anodyne LGMN 52 37 O=C(NCC[C@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824626 GF On-Demand Anodyne KLK5 42 41 O=C(NCC[C@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824626 GF On-Demand Anodyne Q9NAW4_PLAFA 36 41 O=C(NCC[C@@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824627 GF On-Demand Anodyne PREP 29 40 O=C(NCC[C@@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824627 GF On-Demand Anodyne LGMN 52 37 O=C(NCC[C@@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824627 GF On-Demand Anodyne KLK5 42 41 O=C(NCC[C@@H]1CCCOC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880824627 GF On-Demand Anodyne Q9NAW4_PLAFA 36 41 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CCCOC1 ZINC000880824632 DG On-Demand Anodyne NQO2 19 45 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CCCOC1 ZINC000880824632 DG On-Demand Anodyne MTNR1A 15 40 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CCCOC1 ZINC000880824633 DG On-Demand Anodyne NQO2 19 45 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CCCOC1 ZINC000880824633 DG On-Demand Anodyne MTNR1A 15 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CCCOC1 ZINC000880824634 DG On-Demand Anodyne NQO2 19 45 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CCCOC1 ZINC000880824634 DG On-Demand Anodyne MTNR1A 15 40 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CCCOC1 ZINC000880824635 DG On-Demand Anodyne NQO2 19 45 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CCCOC1 ZINC000880824635 DG On-Demand Anodyne MTNR1A 15 40 O=C(NC[C@@H]1CC[C@H]2C[C@H]2C1)c1cnc2cc[nH]c2c1 ZINC000880824646 CF On-Demand Anodyne GRIN2B 15 40 O=C(NC[C@@H]1CC[C@@H]2C[C@H]2C1)c1cnc2cc[nH]c2c1 ZINC000880824647 CF On-Demand Anodyne GRIN2B 15 40 O=C(NC[C@@H]1CC[C@@H]2C[C@@H]2C1)c1cnc2cc[nH]c2c1 ZINC000880824648 CF On-Demand Anodyne GRIN2B 15 40 O=C(NC[C@@H]1CC[C@H]2C[C@@H]2C1)c1cnc2cc[nH]c2c1 ZINC000880824649 CF On-Demand Anodyne GRIN2B 15 40 COc1cccc([C@H](CNC(=O)C[C@@H]2CCNC2=O)OC)c1 ZINC000880824665 DD On-Demand Anodyne MTNR1A 29 40 COc1cccc([C@H](CNC(=O)C[C@@H]2CCNC2=O)OC)c1 ZINC000880824665 DD On-Demand Anodyne MTNR1B 31 40 COc1cccc([C@H](CNC(=O)C[C@H]2CCNC2=O)OC)c1 ZINC000880824666 DD On-Demand Anodyne MTNR1A 29 40 COc1cccc([C@H](CNC(=O)C[C@H]2CCNC2=O)OC)c1 ZINC000880824666 DD On-Demand Anodyne MTNR1B 31 40 COc1cccc([C@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)OC)c1 ZINC000880824673 FF On-Demand Anodyne DRD4 46 35 COc1cccc([C@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)OC)c1 ZINC000880824674 FF On-Demand Anodyne DRD4 46 35 COc1cccc([C@H](CNC(=O)c2cc(C)co2)OC)c1 ZINC000880824685 CF On-Demand Anodyne DRD4 41 34 COc1cccc([C@H](CNC(=O)c2cc(C)co2)OC)c1 ZINC000880824685 CF On-Demand Anodyne MTNR1A 42 40 COc1cccc([C@H](CNC(=O)c2cc(C)co2)OC)c1 ZINC000880824685 CF On-Demand Anodyne MTNR1B 42 40 COc1cccc([C@H](CNC(=O)Cc2c(Br)cnn2C)OC)c1 ZINC000880824699 GE On-Demand Anodyne DRD4 41 31 COc1cccc([C@H](CNC(=O)C2CCC(S(C)(=O)=O)CC2)OC)c1 ZINC000880824716 FE On-Demand Anodyne DRD4 40 30 COc1cccc([C@H](CNC(=O)C2CCC(S(C)(=O)=O)CC2)OC)c1 ZINC000880824716 FE On-Demand Anodyne MTNR1A 55 56 COc1cccc([C@H](CNC(=O)C2CCC(S(C)(=O)=O)CC2)OC)c1 ZINC000880824716 FE On-Demand Anodyne MTNR1B 46 56 COc1cccc([C@H](CNC(=O)Nc2cc3n(n2)CCN(C)C3)OC)c1 ZINC000880824729 FD On-Demand Anodyne DRD4 40 30 CS(=O)(=O)C1CCC(C(=O)NCc2ccc(-c3ccccc3)s2)CC1 ZINC000880824768 GH On-Demand Anodyne PDE8B 48 33 O=C(COC1CC1)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880824815 EF On-Demand Anodyne ETHR 28 44 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne HRH1 29 40 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne PRSS2 57 33 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne CCR3 46 43 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne MLNR 23 54 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne EPHX2 25 40 O=C(COC1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824832 CE On-Demand Anodyne SCD1 22 46 COc1ccccc1-c1ccc(C(=O)NCC[C@@H]2CCCOC2)c(O)n1 ZINC000880824851 FG On-Demand Anodyne DRD2 18 43 COc1ccccc1-c1ccc(C(=O)NCC[C@H]2CCCOC2)c(O)n1 ZINC000880824854 FG On-Demand Anodyne DRD2 18 43 O=C(c1cccn2nccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824855 EG On-Demand Anodyne HRH1 21 43 O=C(c1cccn2nccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880824855 EG On-Demand Anodyne CCR3 29 43 C[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C[C@@H](C)C1(F)F ZINC000880824860 GI On-Demand Anodyne RBP4 56 32 C[C@H]1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C[C@H](C)C1(F)F ZINC000880824863 GI On-Demand Anodyne RBP4 56 32 CN1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)(c2ccccc2)CC1 ZINC000880824887 GE On-Demand Anodyne KCNA3 44 37 CN1CCC(CNC(=O)Nc2cc3n(n2)CCN(C)C3)(c2ccccc2)CC1 ZINC000880824887 GE On-Demand Anodyne SOAT1 18 43 Cn1ncc(C(F)(F)F)c1CNC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880824893 FG On-Demand Anodyne P2RX7 20 44 Cn1ncc(C(F)(F)F)c1CNC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880824960 FG On-Demand Anodyne P2RX7 23 41 O=C(NCC[C@H]1CCCOC1)c1coc(-c2ccccn2)n1 ZINC000880824995 DE On-Demand Anodyne TBXA2R 32 44 O=C(NCC[C@@H]1CCCOC1)c1coc(-c2ccccn2)n1 ZINC000880824997 DE On-Demand Anodyne TBXA2R 32 44 Cn1ncc(C(F)(F)F)c1CNC(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880825007 EG On-Demand Anodyne P2RX7 39 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)N1 ZINC000880825031 GG On-Demand Anodyne CCR3 20 40 O=C1CC[C@@H](c2ccc(C(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)N1 ZINC000880825031 GG On-Demand Anodyne L3MBTL3 44 34 O=C1CC[C@H](c2ccc(C(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)N1 ZINC000880825034 GG On-Demand Anodyne CCR3 20 40 O=C1CC[C@H](c2ccc(C(=O)N3CCC(Oc4cccc(F)c4)CC3)cc2)N1 ZINC000880825034 GG On-Demand Anodyne L3MBTL3 44 34 CS(=O)(=O)C1CCC(C(=O)NCC2CCc3ccccc3CC2)CC1 ZINC000880825040 FF On-Demand Anodyne MTNR1A 30 42 CS(=O)(=O)C1CCC(C(=O)NCC2CCc3ccccc3CC2)CC1 ZINC000880825040 FF On-Demand Anodyne MTNR1B 28 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](n1cccn1)C(F)(F)F)C2 ZINC000880825051 FF On-Demand Anodyne MTNR1A 27 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](n1cccn1)C(F)(F)F)C2 ZINC000880825051 FF On-Demand Anodyne MTNR1B 27 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](n1cccn1)C(F)(F)F)C2 ZINC000880825053 FF On-Demand Anodyne MTNR1A 27 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](n1cccn1)C(F)(F)F)C2 ZINC000880825053 FF On-Demand Anodyne MTNR1B 27 42 Cn1ncc(Br)c1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825061 GF On-Demand Anodyne PRSS2 41 32 Cn1ncc(Br)c1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825061 GF On-Demand Anodyne CCR3 30 40 Cn1ncc(Br)c1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825061 GF On-Demand Anodyne MLNR 32 55 Cn1ncc(Br)c1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825061 GF On-Demand Anodyne SCD1 20 42 CN1CCN(C2CCN(C(=O)Nc3cc4n(n3)CCN(C)C4)CC2)CC1 ZINC000880825100 FC On-Demand Anodyne L3MBTL3 60 39 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne GRIN2B 18 43 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne PRSS2 46 32 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne HRH3 18 43 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne CCR3 37 40 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne MLNR 27 50 Cn1nnc(C(=O)N2CCC(Oc3cccc(F)c3)CC2)n1 ZINC000880825109 DD On-Demand Anodyne SCD1 23 45 C=CCCC[C@H](C(=O)NCC[C@@H]1CCCOC1)c1ccccc1 ZINC000880825113 DI On-Demand Mild PGA5 41 32 C=CCCC[C@@H](C(=O)NCC[C@H]1CCCOC1)c1ccccc1 ZINC000880825114 DI On-Demand Mild PGA5 41 32 C=CCCC[C@H](C(=O)NCC[C@H]1CCCOC1)c1ccccc1 ZINC000880825116 DI On-Demand Mild PGA5 41 32 C=CCCC[C@@H](C(=O)NCC[C@@H]1CCCOC1)c1ccccc1 ZINC000880825117 DI On-Demand Mild PGA5 41 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(C(F)(F)F)cnn1C ZINC000880825133 GD On-Demand Anodyne PAPA1_CARPA 35 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(C(F)(F)F)cnn1C ZINC000880825134 GD On-Demand Anodyne PAPA1_CARPA 35 40 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825154 GH On-Demand Anodyne OXTR 36 45 O=C(Cc1ccccc1N1CCCC1=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825154 GH On-Demand Anodyne MLNR 15 49 O=C(NCC[C@@H]1CCCOC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880825164 EG On-Demand Anodyne PDE4D 21 48 O=C(NCC[C@H]1CCCOC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880825165 EG On-Demand Anodyne PDE4D 21 48 CCn1ncc(CNC(=O)c2cc(-c3ccc(OC)cc3)on2)n1 ZINC000880825197 ED On-Demand Anodyne PDK1 44 37 COc1ccccc1[C@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825221 GG On-Demand Anodyne HTR1D 15 43 COc1ccccc1[C@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825221 GG On-Demand Anodyne HTR1B 16 43 COc1ccccc1[C@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825221 GG On-Demand Anodyne RBP4 34 43 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825222 GG On-Demand Anodyne HTR1D 15 43 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825222 GG On-Demand Anodyne HTR1B 16 43 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2cc3n(n2)CCN(C)C3)CC1 ZINC000880825222 GG On-Demand Anodyne RBP4 34 43 Cn1ncc(C(F)(F)F)c1CNC(=O)c1cnc(CC2CC2)s1 ZINC000880825227 EF On-Demand Anodyne P2RX7 25 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CCCOC1 ZINC000880825228 ED On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CCCOC1 ZINC000880825230 ED On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CCCOC1 ZINC000880825232 ED On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CCCOC1 ZINC000880825234 ED On-Demand Anodyne PAPA1_CARPA 35 42 CC(C)(C(=O)N1CCN(c2nccnn2)CC1)c1ccc(F)cc1F ZINC000880825284 ED On-Demand Anodyne FAAH 21 43 Cc1ccc(CN2CC[C@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825297 FE On-Demand Anodyne DRD4 25 45 Cc1ccc(CN2CC[C@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825297 FE On-Demand Anodyne SSTR5 42 36 Cc1ccc(CN2CC[C@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825297 FE On-Demand Anodyne CCR3 28 43 Cc1ccc(CN2CC[C@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825297 FE On-Demand Anodyne UTS2R 24 43 Cc1ccc(CN2CC[C@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825297 FE On-Demand Anodyne MCHR1 28 43 C=CC(C)(C)CC(=O)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880825317 EI On-Demand Mild ETHR 37 44 CCC[C@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)OCC ZINC000880825336 DF On-Demand Anodyne MPO 63 38 CCC[C@@H](CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)OCC ZINC000880825337 DF On-Demand Anodyne MPO 63 38 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825361 FE On-Demand Anodyne DRD4 25 45 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825361 FE On-Demand Anodyne SSTR5 42 36 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825361 FE On-Demand Anodyne CCR3 28 43 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825361 FE On-Demand Anodyne UTS2R 24 43 Cc1ccc(CN2CC[C@@H](NC(=O)Nc3cc4n(n3)CCN(C)C4)C2)cc1 ZINC000880825361 FE On-Demand Anodyne MCHR1 28 43 O=C(C[C@H]1CCNC1=O)NCc1ccc(-c2ccccc2)s1 ZINC000880825415 DF On-Demand Anodyne CYP2E1 19 42 O=C(C[C@@H]1CCNC1=O)NCc1ccc(-c2ccccc2)s1 ZINC000880825416 DF On-Demand Anodyne CYP2E1 19 42 Cn1ncc(C(F)(F)F)c1CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880825432 GE On-Demand Anodyne P2RX7 48 50 CC(C)(C)OC(=O)N1C[C@@H](C(=O)N2CCN(c3nccnn3)CC2)C(C)(C)C1 ZINC000880825437 GD On-Demand Anodyne GPR119 21 45 CC(C)(C)OC(=O)N1C[C@H](C(=O)N2CCN(c3nccnn3)CC2)C(C)(C)C1 ZINC000880825438 GD On-Demand Anodyne GPR119 21 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C(F)(F)F)cnn1C)C2 ZINC000880825491 FF On-Demand Anodyne NQO2 24 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C(F)(F)F)cnn1C)C2 ZINC000880825491 FF On-Demand Anodyne MTNR1A 26 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1c(C(F)(F)F)cnn1C)C2 ZINC000880825491 FF On-Demand Anodyne MTNR1B 25 42 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825500 DH On-Demand Anodyne MLNR 18 50 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825500 DH On-Demand Anodyne EPHX2 18 41 CC(C)n1nnnc1-c1cccc(NC(=O)COC2CC2)c1 ZINC000880825524 DE On-Demand Anodyne CCR3 54 38 CC(C)n1nnnc1-c1cccc(NC(=O)COC2CC2)c1 ZINC000880825524 DE On-Demand Anodyne HDAC10 37 40 CC(C)n1nnnc1-c1cccc(NC(=O)COC2CC2)c1 ZINC000880825524 DE On-Demand Anodyne HDAC2 18 40 CC(C)n1nnnc1-c1cccc(NC(=O)COC2CC2)c1 ZINC000880825524 DE On-Demand Anodyne HDAC3 38 40 CC(C)n1nnnc1-c1cccc(NC(=O)COC2CC2)c1 ZINC000880825524 DE On-Demand Anodyne HDAC6 29 40 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)c1cc(C)cs1)C2 ZINC000880825533 EF On-Demand Reactive MTNR1B 18 40 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@H]1CCc2nncn2CC1 ZINC000880825572 GF On-Demand Reactive TSHR 41 31 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@H]1CCc2nncn2CC1 ZINC000880825572 GF On-Demand Reactive LTA4H 41 44 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@H]1CCc2nncn2CC1 ZINC000880825572 GF On-Demand Reactive ADAM17 35 45 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880825573 GF On-Demand Reactive TSHR 41 31 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880825573 GF On-Demand Reactive LTA4H 41 44 O=C(NNc1ccc(OCc2ccccc2)cc1)[C@@H]1CCc2nncn2CC1 ZINC000880825573 GF On-Demand Reactive ADAM17 35 45 O=C(Nc1cccc(C2CCCCC2)c1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880825593 FI On-Demand Anodyne MCHR1 18 46 O=C(C(=O)N1[C@H]2CC[C@H]1CC(F)(F)C2)c1c[nH]c2cc(F)ccc12 ZINC000880825620 EG On-Demand Anodyne MPO 55 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825631 GE On-Demand Anodyne PAPA1_CARPA 42 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825631 GE On-Demand Anodyne CCKAR 40 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825631 GE On-Demand Anodyne REN 45 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825631 GE On-Demand Anodyne FPR1 46 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825632 GE On-Demand Anodyne PAPA1_CARPA 42 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825632 GE On-Demand Anodyne CCKAR 40 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825632 GE On-Demand Anodyne REN 45 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1Cc2ccccc2CO1 ZINC000880825632 GE On-Demand Anodyne FPR1 46 37 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne HRH1 34 45 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne HRH3 18 43 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne PRCP 44 32 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne CCR3 44 45 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne MLNR 23 45 Cc1cnc(Cl)c(C(=O)N2CCC(Oc3cccc(F)c3)CC2)c1 ZINC000880825685 EH On-Demand Anodyne EPHX2 15 40 CS(=O)(=O)C1CCC(C(=O)N2CCC(Oc3cccc(F)c3)CC2)CC1 ZINC000880825686 GF On-Demand Anodyne PRSS2 58 34 CS(=O)(=O)C1CCC(C(=O)N2CCC(Oc3cccc(F)c3)CC2)CC1 ZINC000880825686 GF On-Demand Anodyne HRH3 15 50 CS(=O)(=O)C1CCC(C(=O)N2CCC(Oc3cccc(F)c3)CC2)CC1 ZINC000880825686 GF On-Demand Anodyne MLNR 16 46 CS(=O)(=O)C1CCC(C(=O)N2CCC(Oc3cccc(F)c3)CC2)CC1 ZINC000880825686 GF On-Demand Anodyne EPHX2 15 40 CS(=O)(=O)C1CCC(C(=O)N2CCC(Oc3cccc(F)c3)CC2)CC1 ZINC000880825686 GF On-Demand Anodyne GPR119 48 43 O=C1NCC[C@H]1CC(=O)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880825687 FE On-Demand Anodyne ETHR 22 43 O=C1NCC[C@@H]1CC(=O)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880825688 FE On-Demand Anodyne ETHR 22 43 COc1ccc(CN(CCO)C(=O)Nc2cc3n(n2)CCN(C)C3)cc1 ZINC000880825694 FD On-Demand Anodyne ROCK2 17 41 O=C(c1ccc(CN2CCOCC2)o1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825703 GF On-Demand Anodyne HRH3 18 52 O=C(c1ccc(CN2CCOCC2)o1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825703 GF On-Demand Anodyne CCR3 48 41 O=C(c1ccc(CN2CCOCC2)o1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880825703 GF On-Demand Anodyne MLNR 31 49 Cc1coc(C(=O)Nc2cccc(-c3nnnn3C(C)C)c2)c1 ZINC000880825770 DG On-Demand Anodyne KCNK3 86 40 Cc1coc(C(=O)Nc2cccc(-c3nnnn3C(C)C)c2)c1 ZINC000880825770 DG On-Demand Anodyne KCNK9 60 37 CCC[C@@H](CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)OCC ZINC000880825823 FD On-Demand Anodyne TRY1_BOVIN 47 33 CCC[C@H](CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1)OCC ZINC000880825824 FD On-Demand Anodyne TRY1_BOVIN 47 33 Cn1nnc(C(=O)NCC2CCc3ccccc3CC2)n1 ZINC000880825859 CD On-Demand Anodyne HTR4 56 39 Cn1nnc(C(=O)NCC2CCc3ccccc3CC2)n1 ZINC000880825859 CD On-Demand Anodyne CACNA1I 63 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)COc2ccccc2O1 ZINC000880825874 GE On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)COc2ccccc2O1 ZINC000880825874 GE On-Demand Anodyne FPR1 43 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)COc2ccccc2O1 ZINC000880825875 GE On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@]1(C)COc2ccccc2O1 ZINC000880825875 GE On-Demand Anodyne FPR1 43 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)COc2ccccc2O1 ZINC000880825876 GE On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)COc2ccccc2O1 ZINC000880825876 GE On-Demand Anodyne FPR1 43 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)COc2ccccc2O1 ZINC000880825877 GE On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)COc2ccccc2O1 ZINC000880825877 GE On-Demand Anodyne FPR1 43 36 Cn1ncc(Br)c1CC(=O)NCc1c(C(F)(F)F)cnn1C ZINC000880825899 GD On-Demand Anodyne P2RX7 21 53 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880825900 FH On-Demand Anodyne ETHR 17 42 CCC[C@@H](CNC(=O)Cc1ccccc1N1CCCC1=O)OCC ZINC000880825908 EF On-Demand Anodyne KCNQ2 44 36 CCC[C@H](CNC(=O)Cc1ccccc1N1CCCC1=O)OCC ZINC000880825909 EF On-Demand Anodyne KCNQ2 44 36 O=C(CC[C@@H]1CCc2ccccc21)N1CCN(c2nccnn2)CC1 ZINC000880825927 EE On-Demand Anodyne SSTR1 42 41 Cn1nnc(C(=O)Nc2cccc(C3CCCCC3)c2)n1 ZINC000880825945 CF On-Demand Anodyne MCHR1 26 42 O=C1CC[C@H](C(=O)NNC(=O)c2ccc(OC(F)F)c(Cl)c2)N1 ZINC000880825952 EC On-Demand Reactive PDE4D 17 41 O=C1CC[C@@H](C(=O)NNC(=O)c2ccc(OC(F)F)c(Cl)c2)N1 ZINC000880825953 EC On-Demand Reactive PDE4D 17 41 O=C(COC1CC1)N1CCC(Cc2nc(C3CCCCC3)no2)CC1 ZINC000880825972 EG On-Demand Anodyne ETHR 23 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1cccc(F)c1Cl ZINC000880826008 GF On-Demand Reactive PAPA1_CARPA 38 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1cccc(F)c1Cl ZINC000880826009 GF On-Demand Reactive PAPA1_CARPA 38 47 O=C(CC[C@H]1CCc2ccccc21)N1CCN(c2nccnn2)CC1 ZINC000880826030 EE On-Demand Anodyne SSTR1 42 41 O=C(CN1CCCCS1(=O)=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826044 GE On-Demand Reactive LTA4H 34 46 O=C(CN1CCCCS1(=O)=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826044 GE On-Demand Reactive SLC12A5 43 35 Cn1ncc(C(F)(F)F)c1CNC(=O)COC1CC1 ZINC000880826055 CD On-Demand Anodyne P2RX7 26 43 O=C(CN1CCCCS1(=O)=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826058 FD On-Demand Anodyne MLNR 17 49 C=CCCC[C@@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826071 ED On-Demand Reactive HDAC10 33 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826071 ED On-Demand Reactive HDAC2 19 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826071 ED On-Demand Reactive HDAC3 15 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826071 ED On-Demand Reactive HDAC6 25 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826071 ED On-Demand Reactive HDAC11 45 43 C=CCCC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826073 ED On-Demand Reactive HDAC10 33 43 C=CCCC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826073 ED On-Demand Reactive HDAC2 19 43 C=CCCC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826073 ED On-Demand Reactive HDAC3 15 43 C=CCCC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826073 ED On-Demand Reactive HDAC6 25 43 C=CCCC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)c1ccccc1 ZINC000880826073 ED On-Demand Reactive HDAC11 45 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826075 ED On-Demand Reactive HDAC10 33 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826075 ED On-Demand Reactive HDAC2 19 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826075 ED On-Demand Reactive HDAC3 15 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826075 ED On-Demand Reactive HDAC6 25 43 C=CCCC[C@@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826075 ED On-Demand Reactive HDAC11 45 43 C=CCCC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826077 ED On-Demand Reactive HDAC10 33 43 C=CCCC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826077 ED On-Demand Reactive HDAC2 19 43 C=CCCC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826077 ED On-Demand Reactive HDAC3 15 43 C=CCCC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826077 ED On-Demand Reactive HDAC6 25 43 C=CCCC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)c1ccccc1 ZINC000880826077 ED On-Demand Reactive HDAC11 45 43 O=C(NCc1ccns1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880826100 FF On-Demand Anodyne GRIN2B 18 40 O=C(NCc1ccns1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880826100 FF On-Demand Anodyne PREP 27 42 O=C(NCc1ccns1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880826100 FF On-Demand Anodyne Q9NAW4_PLAFA 27 43 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826104 FG On-Demand Anodyne MLNR 19 45 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826105 FG On-Demand Anodyne MLNR 19 45 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826106 FG On-Demand Anodyne MLNR 19 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccns1)C2 ZINC000880826114 DF On-Demand Anodyne MTNR1A 38 40 O=C(c1ncsc1C1CC1)N1CCC(Cc2nc(C3CCCC3)no2)CC1 ZINC000880826126 GI On-Demand Anodyne ETHR 42 36 CC(C)n1nnnc1-c1cccc(NC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880826130 GF On-Demand Anodyne CASR 35 47 CC(C)n1nnnc1-c1cccc(NC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880826130 GF On-Demand Anodyne CCR3 46 37 Cn1ncc(C(F)(F)F)c1CNC(=O)C[C@H]1CCNC1=O ZINC000880826155 DC On-Demand Anodyne P2RX7 35 42 Cn1ncc(C(F)(F)F)c1CNC(=O)C[C@@H]1CCNC1=O ZINC000880826157 DC On-Demand Anodyne P2RX7 35 42 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCc4ccccc4CC3)cc2)N1 ZINC000880826190 FH On-Demand Anodyne GRIN2B 22 48 O=C1CC[C@@H](c2ccc(C(=O)NCC3CCc4ccccc4CC3)cc2)N1 ZINC000880826190 FH On-Demand Anodyne CACNA1I 47 32 O=C1CC[C@H](c2ccc(C(=O)NCC3CCc4ccccc4CC3)cc2)N1 ZINC000880826192 FH On-Demand Anodyne GRIN2B 22 48 O=C1CC[C@H](c2ccc(C(=O)NCC3CCc4ccccc4CC3)cc2)N1 ZINC000880826192 FH On-Demand Anodyne CACNA1I 47 32 O=C(C[C@@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826213 EE On-Demand Reactive TSHR 43 33 O=C(C[C@@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826213 EE On-Demand Reactive MAOB 18 40 O=C(C[C@@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826213 EE On-Demand Reactive LTA4H 35 47 O=C(C[C@@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826213 EE On-Demand Reactive ADAM17 28 45 O=C(C[C@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826214 EE On-Demand Reactive TSHR 43 33 O=C(C[C@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826214 EE On-Demand Reactive MAOB 18 40 O=C(C[C@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826214 EE On-Demand Reactive LTA4H 35 47 O=C(C[C@H]1CCNC1=O)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826214 EE On-Demand Reactive ADAM17 28 45 O=C(Nc1cccc(C2CCCCC2)c1)[C@H]1CCc2nncn2CC1 ZINC000880826256 EH On-Demand Anodyne MCHR1 25 50 O=C(Nc1cccc(C2CCCCC2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880826257 EH On-Demand Anodyne MCHR1 25 50 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive TSHR 49 34 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive MAOB 22 41 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive LTA4H 57 54 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive ADAM17 32 51 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive TIMP3 74 36 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive EPHX2 16 47 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive ADAMTS4 22 40 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive NAAA 16 43 O=C(COC1CC1)NNc1ccc(OCc2ccccc2)cc1 ZINC000880826291 DF On-Demand Reactive FFAR1 44 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccns1 ZINC000880826319 ED On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccns1 ZINC000880826321 ED On-Demand Anodyne PAPA1_CARPA 44 44 Cc1cnc(Cl)c(C(=O)NC[C@@]2(C)COc3ccccc3O2)c1 ZINC000880826371 EG On-Demand Anodyne G2YM83_BOTF4 51 32 C=CC(C)(C)CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826399 DH On-Demand Mild PRSS2 41 31 C=CC(C)(C)CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826399 DH On-Demand Mild MLNR 23 52 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2Cc3ccccc3CO2)CC1 ZINC000880826403 FD On-Demand Anodyne MTNR1A 18 40 CS(=O)(=O)C1CCC(C(=O)NC[C@@H]2Cc3ccccc3CO2)CC1 ZINC000880826403 FD On-Demand Anodyne MTNR1B 15 40 O=C1NCC[C@@H]1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826404 DD On-Demand Anodyne MLNR 28 53 O=C1NCC[C@H]1CC(=O)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826405 DD On-Demand Anodyne MLNR 28 53 O=C(c1cncc2[nH]ccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826413 EG On-Demand Anodyne HRH1 19 41 O=C(c1cncc2[nH]ccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826413 EG On-Demand Anodyne GRIN2B 17 40 O=C(c1cncc2[nH]ccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826413 EG On-Demand Anodyne CCR3 24 41 O=C(c1cncc2[nH]ccc12)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826413 EG On-Demand Anodyne SCD1 15 40 O=C(NCc1ccns1)c1ccc(CN2CCOCC2)o1 ZINC000880826415 DD On-Demand Anodyne DPOL_VZVD 23 40 O=C(NCc1ccns1)c1ccc(CN2CCOCC2)o1 ZINC000880826415 DD On-Demand Anodyne NAMPT 22 41 O=C(c1cnc2cc[nH]c2c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826429 EG On-Demand Anodyne HRH1 23 42 O=C(c1cnc2cc[nH]c2c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826429 EG On-Demand Anodyne GRIN2B 18 43 O=C(c1cnc2cc[nH]c2c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826429 EG On-Demand Anodyne HRH3 18 48 O=C(c1cnc2cc[nH]c2c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826429 EG On-Demand Anodyne CCR3 30 43 O=C(c1cnc2cc[nH]c2c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880826429 EG On-Demand Anodyne MLNR 27 44 CS(=O)(=O)C1CCC(C(=O)Nc2cccc(C3CCCCC3)c2)CC1 ZINC000880826480 FI On-Demand Anodyne EPHX2 22 40 CS(=O)(=O)C1CCC(C(=O)Nc2cccc(C3CCCCC3)c2)CC1 ZINC000880826480 FI On-Demand Anodyne MCHR1 22 47 CSc1nccnc1C(=O)Nc1cccc(-c2nnnn2C(C)C)c1 ZINC000880826513 FF On-Demand Anodyne KCNK3 51 34 CSc1nccnc1C(=O)Nc1cccc(-c2nnnn2C(C)C)c1 ZINC000880826513 FF On-Demand Anodyne KCNK9 46 32 CC[C@@H](C)c1cccc(NC(=O)COC2CC2)c1 ZINC000880826532 BG On-Demand Anodyne TIMP3 74 35 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)C2 ZINC000880826551 EC On-Demand Reactive MTNR1A 24 42 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@H]1CCC(=O)N1)C2 ZINC000880826551 EC On-Demand Reactive MTNR1B 23 42 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)C2 ZINC000880826552 EC On-Demand Reactive MTNR1A 24 42 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@@H]1CCC(=O)N1)C2 ZINC000880826552 EC On-Demand Reactive MTNR1B 23 42 CS(=O)(=O)c1ccc([C@@H]2CN(C(=O)COC3CC3)CCO2)cc1 ZINC000880826560 ED On-Demand Anodyne GPR119 27 45 CS(=O)(=O)c1ccc([C@H]2CN(C(=O)COC3CC3)CCO2)cc1 ZINC000880826561 ED On-Demand Anodyne GPR119 27 45 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c1 ZINC000880826615 EI On-Demand Anodyne TAAR1 43 39 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c1 ZINC000880826615 EI On-Demand Anodyne KCNK3 93 37 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c1 ZINC000880826615 EI On-Demand Anodyne KCNK9 52 34 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c1 ZINC000880826617 EI On-Demand Anodyne TAAR1 43 39 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c1 ZINC000880826617 EI On-Demand Anodyne KCNK3 93 37 CC[C@@H](C)c1cccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c1 ZINC000880826617 EI On-Demand Anodyne KCNK9 52 34 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)c1cn[nH]c1)C2 ZINC000880826706 DC On-Demand Reactive ROCK2 58 44 CC[C@@H](C)c1cccc(NC(=O)c2nnn(C)n2)c1 ZINC000880826721 CD On-Demand Anodyne KCNK3 57 34 CC[C@@H](C)c1cccc(NC(=O)c2nnn(C)n2)c1 ZINC000880826721 CD On-Demand Anodyne KCNK9 48 34 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@H](c2ccc(F)c(F)c2)C1 ZINC000880826728 FI On-Demand Anodyne MAP3K12 31 41 O=C(c1coc(-c2ccccn2)n1)N1CCC[C@@H](c2ccc(F)c(F)c2)C1 ZINC000880826729 FI On-Demand Anodyne MAP3K12 31 41 C=CC(C)(C)CC(=O)NNc1cccc(C)n1 ZINC000880826751 BE On-Demand Reactive GRM5 17 40 O=C(Nc1cccc2c1OCCCO2)N1CC(c2ccccc2)C1 ZINC000880826843 DG On-Demand Anodyne RBP4 53 35 O=C(COC1CC1)N1CC[C@@H](Oc2cccc(Cl)c2)C1 ZINC000880826878 CE On-Demand Anodyne HRH1 34 43 O=C(COC1CC1)N1CC[C@@H](Oc2cccc(Cl)c2)C1 ZINC000880826878 CE On-Demand Anodyne CCR3 39 43 O=C(COC1CC1)N1CC[C@@H](Oc2cccc(Cl)c2)C1 ZINC000880826878 CE On-Demand Anodyne EPHX2 17 49 CS(=O)(=O)C1CCC(C(=O)N2CC[C@@H](Oc3cccc(Cl)c3)C2)CC1 ZINC000880826994 GF On-Demand Anodyne HRH1 29 40 CS(=O)(=O)C1CCC(C(=O)N2CC[C@@H](Oc3cccc(Cl)c3)C2)CC1 ZINC000880826994 GF On-Demand Anodyne CCR3 32 40 CCN1CC[C@@H]1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880827029 DE On-Demand Anodyne DRD2 25 42 O=C(Nc1cccc2c1OCCCO2)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880827047 GF On-Demand Anodyne ETHR 53 37 O=C(Nc1cccc2c1OCCCO2)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880827048 GF On-Demand Anodyne ETHR 53 37 O=C(/C=C\c1cccnc1)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000880827155 GI On-Demand Anodyne HDAC8 35 40 O=C(/C=C\c1cccnc1)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000880827155 GI On-Demand Anodyne HDAC1 23 48 O=C(/C=C\c1cccnc1)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000880827155 GI On-Demand Anodyne HDAC6 23 40 COc1ccc(CN(C)C(=O)Nc2cccc3c2OCCCO3)cc1 ZINC000880827192 EH On-Demand Anodyne BMP1 42 32 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2cccc4c2OCCCO4)C3)c1 ZINC000880827217 GD On-Demand Anodyne P2RX7 22 40 COc1ccc(CN(CCO)C(=O)Nc2cccc3c2OCCCO3)cc1 ZINC000880827231 FF On-Demand Anodyne BMP1 51 37 COc1ccc(CN(CCO)C(=O)Nc2cccc3c2OCCCO3)cc1 ZINC000880827231 FF On-Demand Anodyne ROCK2 15 41 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880827238 FD On-Demand Anodyne P2RX7 43 36 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880827238 FD On-Demand Anodyne RBP4 46 34 O=C(NCc1ncccn1)Nc1cccc2c1OCCCO2 ZINC000880827266 DD On-Demand Anodyne G2YM83_BOTF4 40 34 O=C(Nc1cccc2c1OCCCO2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880827269 GH On-Demand Anodyne SMO 42 45 O=C(Nc1cccc2c1OCCCO2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880827269 GH On-Demand Anodyne ETHR 64 46 CN1CCN(C2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)CC1 ZINC000880827294 FE On-Demand Anodyne L3MBTL3 73 41 O=C(C(=O)N1C[C@@H](CO)[C@H](CO)C1)c1c[nH]c2cc(F)ccc12 ZINC000880827322 DC On-Demand Anodyne MPO 62 36 O=C(c1ccc(CN2CCOCC2)o1)N1CC[C@@H](Oc2cccc(Cl)c2)C1 ZINC000880827369 GG On-Demand Anodyne CCR3 32 40 O=C(c1ccc(CN2CCOCC2)o1)N1CC[C@@H](Oc2cccc(Cl)c2)C1 ZINC000880827369 GG On-Demand Anodyne MCHR1 15 41 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](c2nccs2)C1 ZINC000880827394 EG On-Demand Anodyne ETHR 41 32 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](c2nccs2)C1 ZINC000880827395 EG On-Demand Anodyne ETHR 41 32 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880827423 EH On-Demand Anodyne RBP4 45 34 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](C(F)(F)F)C1 ZINC000880827424 EH On-Demand Anodyne RBP4 45 34 CN1CCN(C(=O)Nc2cccc3c2OCCCO3)Cc2cccnc21 ZINC000880827497 FF On-Demand Anodyne G2YM83_BOTF4 42 37 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880827533 GC On-Demand Anodyne PREP 53 50 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880827533 GC On-Demand Anodyne Q9NAW4_PLAFA 37 44 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880827597 GF On-Demand Anodyne HTR4 30 40 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880827625 GG On-Demand Anodyne TRPM8 30 43 O=C(Nc1cccc2c1OCCCO2)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880827626 GG On-Demand Anodyne TRPM8 30 43 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880827627 GG On-Demand Anodyne TRPM8 30 43 O=C(Nc1cccc2c1OCCCO2)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880827628 GG On-Demand Anodyne TRPM8 30 43 O=C(NCc1cnc(C(F)(F)F)nc1)Nc1cccc2c1OCCCO2 ZINC000880827654 FF On-Demand Anodyne TRPV1 17 40 O=C(Nc1cccc2c1OCCCO2)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880827662 EE On-Demand Anodyne RBP4 52 35 O=C(Nc1cccc2c1OCCCO2)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880827664 EE On-Demand Anodyne RBP4 52 35 O=C(Nc1cccc2c1OCCCO2)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880827666 EE On-Demand Anodyne RBP4 52 35 O=C(Nc1cccc2c1OCCCO2)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880827668 EE On-Demand Anodyne RBP4 52 35 O=C(Nc1cccc2c1OCCCO2)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880827670 EE On-Demand Anodyne RBP4 52 35 COC[C@@H]1CCCN1NC(=O)c1cc(C)cnc1Cl ZINC000880827718 CD On-Demand Anodyne CASP7 49 36 COC[C@@H]1CCCN1NC(=O)CN(C(C)=O)c1ccccc1 ZINC000880827790 DD On-Demand Anodyne ACKR3 52 33 COC[C@@H]1CCCN1NC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880827948 DE On-Demand Anodyne CASP3 40 36 COC[C@@H]1CCCN1NC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880827948 DE On-Demand Anodyne CASP7 54 36 CN(C[C@H]1CCCN1C)C(=O)Nc1cccc2c1OCCCO2 ZINC000880827989 DE On-Demand Anodyne CHRNA10 46 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1cccc2c1OCCCO2 ZINC000880827990 DE On-Demand Anodyne CHRNA10 46 33 CN(C(=O)Nc1cccc2c1OCCCO2)[C@H](CO)Cc1ccccc1 ZINC000880828003 FF On-Demand Anodyne NPY5R 20 42 CN(C(=O)Nc1cccc2c1OCCCO2)[C@@H](CO)Cc1ccccc1 ZINC000880828004 FF On-Demand Anodyne NPY5R 20 42 COc1cccc([C@H](CO)NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880828114 FF On-Demand Anodyne KCNQ2 22 43 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1Cc2ccc(O)cc2C1 ZINC000880828134 GF On-Demand Anodyne CPT2 39 41 O=C([C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1)N1Cc2ccc(O)cc2C1 ZINC000880828134 GF On-Demand Anodyne PREP 54 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCC[C@@H]1COC ZINC000880828138 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCC[C@@H]1COC ZINC000880828139 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN1CCC[C@H]1COC ZINC000880828140 ED On-Demand Anodyne PAPA1_CARPA 33 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN1CCC[C@H]1COC ZINC000880828141 ED On-Demand Anodyne PAPA1_CARPA 33 40 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880828205 GG On-Demand Anodyne EPHX2 44 43 CC(=O)c1cccc(CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880828208 EG On-Demand Anodyne ROCK2 21 40 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880828228 FD On-Demand Anodyne EPHX2 27 43 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880828229 FD On-Demand Anodyne EPHX2 27 43 CN(C)C1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880828389 EF On-Demand Anodyne EPHX2 16 41 COC[C@@H]1CCCN1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880828407 DD On-Demand Anodyne GABRA1 15 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880828468 DD On-Demand Anodyne MTNR1A 15 50 CC(=O)N[C@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880828469 DD On-Demand Anodyne MTNR1A 15 50 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cccc2c1OCCCO2 ZINC000880828471 GF On-Demand Anodyne HTR4 17 41 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cccc2c1OCCCO2 ZINC000880828472 GF On-Demand Anodyne HTR4 17 41 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCOC1=O ZINC000880828526 CD On-Demand Anodyne LUXR 77 42 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCOC1=O ZINC000880828526 CD On-Demand Anodyne TRAR 90 41 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCOC1=O ZINC000880828526 CD On-Demand Anodyne LASR 60 41 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880828528 GF On-Demand Anodyne L3MBTL3 70 39 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880828529 GF On-Demand Anodyne L3MBTL3 70 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccc(O)cc2C1 ZINC000880828537 FE On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2ccc(O)cc2C1 ZINC000880828538 FE On-Demand Anodyne PAPA1_CARPA 35 41 COC[C@@H]1CCCN1NC(=O)c1cc(C(F)F)[nH]n1 ZINC000880828553 CD On-Demand Anodyne CASP7 43 36 Cn1nnc(C(=O)NCC2CC=CC2)n1 ZINC000880828569 BB On-Demand Anodyne CACNA1I 60 36 CS(=O)(=O)NCC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880828605 GD On-Demand Anodyne HTR4 22 45 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne FKBP1A 28 52 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne SCNN1A 47 40 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne SIGMAR1 17 42 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne SCN2A 17 42 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne MTNR1A 30 46 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne MTNR1B 31 46 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne FAAH 37 41 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne CES1 48 36 O=C(NCCCCCCc1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880828618 FG On-Demand Anodyne AMP1_PLAFQ 21 42 O=C(NC[C@@H]1CCN1C1CCCCC1)c1cccn2nccc12 ZINC000880828629 DE On-Demand Anodyne JAK3 15 40 O=C(NC[C@@H]1CCN1C1CCCCC1)c1cccn2nccc12 ZINC000880828629 DE On-Demand Anodyne TYK2 19 40 O=C(NC[C@H]1CCN1C1CCCCC1)c1cccn2nccc12 ZINC000880828630 DE On-Demand Anodyne JAK3 15 40 O=C(NC[C@H]1CCN1C1CCCCC1)c1cccn2nccc12 ZINC000880828630 DE On-Demand Anodyne TYK2 19 40 Cc1cnc(Cl)c(C(=O)NCC2CC=CC2)c1 ZINC000880828639 CF On-Demand Anodyne CACNA1I 66 40 O=C(Nc1cccc2c1OCCCO2)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880828718 EF On-Demand Anodyne PLM1_PLAFA 40 38 COC[C@@H]1CCCN1NC(=O)C[C@@H]1CCNC1=O ZINC000880828735 CB On-Demand Anodyne CASP7 43 36 COC[C@@H]1CCCN1NC(=O)C[C@H]1CCNC1=O ZINC000880828737 CB On-Demand Anodyne CASP7 43 36 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880828740 FG On-Demand Anodyne TRPV1 15 44 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880828740 FG On-Demand Anodyne SCN2A 17 42 O=C(NCc1cccnc1N1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880828740 FG On-Demand Anodyne SCN10A 19 42 CC(=O)NCCN(C)C(=O)Nc1cccc2c1OCCCO2 ZINC000880828749 DD On-Demand Anodyne MTNR1A 27 52 NC(=O)[C@@H]1CC[C@H](C(=O)N2Cc3ccc(O)cc3C2)N1Cc1ccccc1 ZINC000880828750 FD On-Demand Anodyne CPT2 35 41 O=C(NCCc1cc(C(F)(F)F)ccn1)Nc1cccc2c1OCCCO2 ZINC000880828799 GH On-Demand Anodyne TRPV1 15 45 O=C(Nc1cccc2c1OCCCO2)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880828819 FG On-Demand Anodyne EPHX2 48 45 O=C(Nc1cccc2c1OCCCO2)N(CCN1CCOCC1)CC1CC1 ZINC000880828827 GE On-Demand Anodyne CASR 57 41 O=C(NC[C@@H]1CCN1C1CCCCC1)c1cnc2cc[nH]c2c1 ZINC000880828829 DF On-Demand Anodyne JAK1 42 36 O=C(NC[C@H]1CCN1C1CCCCC1)c1cnc2cc[nH]c2c1 ZINC000880828831 DF On-Demand Anodyne JAK1 42 36 O=C(NCC1CC=CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880828832 CF On-Demand Anodyne GABRA1 19 52 O=C(NCC1CC=CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880828832 CF On-Demand Anodyne MPO 62 35 O=C(NCC1CC=CC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880828832 CF On-Demand Anodyne GABRA2 17 52 COC[C@@H]1CCCN1NC(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880828853 CE On-Demand Anodyne CASP7 45 36 O=C(NCC1CC=CC1)c1cccn2nccc12 ZINC000880828854 BE On-Demand Anodyne JAK3 17 41 O=C(NCC1CC=CC1)c1cccn2nccc12 ZINC000880828854 BE On-Demand Anodyne TYK2 20 41 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2C2CCCCC2)c1 ZINC000880828880 DG On-Demand Anodyne CACNA1I 53 35 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2C2CCCCC2)c1 ZINC000880828882 DG On-Demand Anodyne CACNA1I 53 35 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne DRD4 40 31 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne HRH2 16 40 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne MTNR1A 31 58 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne MTNR1B 41 58 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne GALR2 47 44 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne FPR2 15 41 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne TAAR1 38 41 COc1cccc(Nc2ccc(NC(=O)CN3CCCCS3(=O)=O)cc2)c1 ZINC000880828894 GF On-Demand Anodyne AKR1C3 25 42 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828904 GH On-Demand Anodyne DRD2 42 39 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828904 GH On-Demand Anodyne DRD3 28 50 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828904 GH On-Demand Anodyne HCN1 54 35 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828904 GH On-Demand Anodyne HCN4 52 35 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828905 GH On-Demand Anodyne DRD2 42 39 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828905 GH On-Demand Anodyne DRD3 28 50 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828905 GH On-Demand Anodyne HCN1 54 35 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCCC2)c(O)n1 ZINC000880828905 GH On-Demand Anodyne HCN4 52 35 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCc2ccc(O)cc21 ZINC000880828934 EG On-Demand Anodyne TRPV1 23 40 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCc2ccc(O)cc21 ZINC000880828937 EG On-Demand Anodyne TRPV1 23 40 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@H]1c1cc[nH]n1 ZINC000880828938 EG On-Demand Anodyne CPT1A 47 38 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@@H]1c1cc[nH]n1 ZINC000880828939 EG On-Demand Anodyne CPT1A 47 38 O=C(C[C@@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829096 DE On-Demand Anodyne FKBP1A 18 40 O=C(C[C@@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829096 DE On-Demand Anodyne SIGMAR1 15 43 O=C(C[C@@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829096 DE On-Demand Anodyne FAAH 43 40 O=C(C[C@@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829096 DE On-Demand Anodyne CES1 52 35 O=C(C[C@@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829096 DE On-Demand Anodyne AMP1_PLAFQ 20 40 O=C(C[C@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829097 DE On-Demand Anodyne FKBP1A 18 40 O=C(C[C@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829097 DE On-Demand Anodyne SIGMAR1 15 43 O=C(C[C@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829097 DE On-Demand Anodyne FAAH 43 40 O=C(C[C@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829097 DE On-Demand Anodyne CES1 52 35 O=C(C[C@H]1CCNC1=O)NCCCCCCc1ccccc1 ZINC000880829097 DE On-Demand Anodyne AMP1_PLAFQ 20 40 O=C(CC[C@@H]1CCc2ccccc21)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880829114 FE On-Demand Anodyne SSTR1 41 41 O=C(CC[C@H]1CCc2ccccc21)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880829115 FE On-Demand Anodyne SSTR1 41 41 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne FKBP1A 33 54 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne SCNN1A 47 40 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne SIGMAR1 16 41 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne SCN2A 21 42 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne MTNR1A 45 50 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne MTNR1B 44 50 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne FAAH 37 40 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne CES1 42 35 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne AMP1_PLAFQ 22 43 CS(=O)(=O)C1CCC(C(=O)NCCCCCCc2ccccc2)CC1 ZINC000880829116 FH On-Demand Anodyne CACNA1G 18 41 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)cc2)c1 ZINC000880829143 EF On-Demand Anodyne PDGFRB 15 41 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)cc2)c1 ZINC000880829143 EF On-Demand Anodyne MTNR1A 25 60 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)cc2)c1 ZINC000880829143 EF On-Demand Anodyne MTNR1B 32 60 COc1cccc(Nc2ccc(NC(=O)C[C@H]3CCNC3=O)cc2)c1 ZINC000880829143 EF On-Demand Anodyne AKR1C3 19 40 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)cc2)c1 ZINC000880829145 EF On-Demand Anodyne PDGFRB 15 41 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)cc2)c1 ZINC000880829145 EF On-Demand Anodyne MTNR1A 25 60 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)cc2)c1 ZINC000880829145 EF On-Demand Anodyne MTNR1B 32 60 COc1cccc(Nc2ccc(NC(=O)C[C@@H]3CCNC3=O)cc2)c1 ZINC000880829145 EF On-Demand Anodyne AKR1C3 19 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC=CC1 ZINC000880829165 DD On-Demand Anodyne PAPA1_CARPA 41 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC=CC1 ZINC000880829167 DD On-Demand Anodyne PAPA1_CARPA 41 48 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CC(F)(F)F)CC1 ZINC000880829191 FF On-Demand Anodyne EPHX2 36 42 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CC(F)(F)F)CC1 ZINC000880829191 FF On-Demand Anodyne HPGDS 38 41 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne S1PR3 17 40 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne MTNR1A 32 42 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne MTNR1B 35 42 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne FAAH 84 44 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne CES1 72 38 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne AMP1_PLAFQ 21 42 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne CRTM 42 42 Cc1nn(CC(=O)NCCCCCCc2ccccc2)c(=O)o1 ZINC000880829197 DE On-Demand Anodyne CES1D 58 34 O=C(Nc1cccc2c1OCCCO2)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880829199 FG On-Demand Anodyne EPHX2 18 44 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880829201 FG On-Demand Anodyne EPHX2 18 44 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880829238 GG On-Demand Anodyne EPHX2 18 50 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880829239 GG On-Demand Anodyne EPHX2 18 50 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829259 GH On-Demand Anodyne DRD4 42 33 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829259 GH On-Demand Anodyne MTNR1A 17 67 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829259 GH On-Demand Anodyne MTNR1B 25 67 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829259 GH On-Demand Anodyne GALR2 27 41 COc1cccc(Nc2ccc(NC(=O)[C@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829259 GH On-Demand Anodyne EPHX2 18 41 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829260 GH On-Demand Anodyne DRD4 42 33 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829260 GH On-Demand Anodyne MTNR1A 17 67 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829260 GH On-Demand Anodyne MTNR1B 25 67 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829260 GH On-Demand Anodyne GALR2 27 41 COc1cccc(Nc2ccc(NC(=O)[C@@H]3CCc4nncn4CC3)cc2)c1 ZINC000880829260 GH On-Demand Anodyne EPHX2 18 41 CCCN(CCN1CCCC1)C(=O)Nc1cccc2c1OCCCO2 ZINC000880829359 EG On-Demand Anodyne CASR 53 39 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880829372 GE On-Demand Anodyne L3MBTL3 45 34 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne FKBP1A 25 47 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne SCNN1A 75 41 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne SIGMAR1 18 43 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne MTNR1A 16 43 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne MTNR1B 19 43 O=C(NCCCCCCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880829485 EG On-Demand Anodyne CACNA1G 27 42 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne FKBP1A 25 47 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne SCNN1A 75 41 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne SIGMAR1 18 43 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne MTNR1A 16 43 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne MTNR1B 19 43 O=C(NCCCCCCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880829488 EG On-Demand Anodyne CACNA1G 27 42 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](N2CCOCC2)C1 ZINC000880829513 ED On-Demand Anodyne L3MBTL3 57 38 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](N2CCOCC2)C1 ZINC000880829527 ED On-Demand Anodyne L3MBTL3 57 38 O=C(NCC1CCN(CC2CC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880829548 FG On-Demand Anodyne HTR4 43 43 O=C(NCC1CCN(CC2CC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880829548 FG On-Demand Anodyne CCR3 41 35 O=C(NCCCCCN1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880829569 EG On-Demand Anodyne HTR1A 17 44 O=C(NCCCCCN1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880829569 EG On-Demand Anodyne DRD2 19 40 O=C(NCCCCCN1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880829569 EG On-Demand Anodyne CCR3 21 40 O=C(NCCCCCN1CCCC1)Nc1cccc2c1OCCCO2 ZINC000880829569 EG On-Demand Anodyne CHRNA7 17 49 COC[C@@H]1CCCN1NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880829581 EE On-Demand Anodyne CHRNA10 49 38 COC[C@@H]1CCCN1NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880829581 EE On-Demand Anodyne CASP7 46 37 COC[C@@H]1CCCN1NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880829581 EE On-Demand Anodyne PDK1 47 35 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](C2CCC2)C1 ZINC000880829592 EH On-Demand Anodyne RBP4 44 33 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](C2CCC2)C1 ZINC000880829593 EH On-Demand Anodyne RBP4 44 33 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H]2C[C@H]2C1 ZINC000880829615 CF On-Demand Anodyne RBP4 54 36 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H]2C[C@@H]2C1 ZINC000880829616 CF On-Demand Anodyne RBP4 54 36 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H]2C[C@H]2C1 ZINC000880829617 CF On-Demand Anodyne RBP4 54 36 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H]2C[C@@H]2C1 ZINC000880829618 CF On-Demand Anodyne RBP4 54 36 Cc1ccncc1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880829710 DF On-Demand Anodyne TRPV1 17 40 Cc1ccncc1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880829710 DF On-Demand Anodyne NAMPT 20 48 CC(C)(C)OC(=O)N1CCN(C(=O)N2CCN(C(=O)COC3CC3)CC2)CC1 ZINC000880829840 GC On-Demand Anodyne GPR119 38 44 O=C(NCc1cnccc1C(F)(F)F)Nc1cccc2c1OCCCO2 ZINC000880829847 FH On-Demand Anodyne TRPV1 26 55 O=C(Nc1cccc2c1OCCCO2)N1CC(C2CCCCC2)C1 ZINC000880829848 EH On-Demand Anodyne RBP4 44 33 O=C(Nc1cccc2c1OCCCO2)N1C[C@H]2CCCC[C@H]2C1 ZINC000880829851 DH On-Demand Anodyne RBP4 45 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C1CCCCC1 ZINC000880829870 GE On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C1CCCCC1 ZINC000880829874 GE On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C1CCCCC1 ZINC000880829878 GE On-Demand Anodyne PAPA1_CARPA 33 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C1CCCCC1 ZINC000880829882 GE On-Demand Anodyne PAPA1_CARPA 33 42 O=C1CC[C@@H](c2ccc(C(=O)N3CCN(S(=O)(=O)C4CC4)CC3)cc2)N1 ZINC000880829946 GC On-Demand Anodyne L3MBTL3 55 38 O=C1CC[C@H](c2ccc(C(=O)N3CCN(S(=O)(=O)C4CC4)CC3)cc2)N1 ZINC000880829948 GC On-Demand Anodyne L3MBTL3 55 38 O=C(NCC1CC=CC1)c1cnc2cc[nH]c2c1 ZINC000880830016 BE On-Demand Anodyne GRIN2B 17 41 O=C(NCC1CC=CC1)c1cnc2cc[nH]c2c1 ZINC000880830016 BE On-Demand Anodyne CACNA1I 52 34 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne S1PR3 18 41 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne MTNR1A 43 47 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne MTNR1B 48 47 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne FAAH 115 47 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne S1PR2 19 41 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne SLC6A5 22 41 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne CES1 81 44 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne AMP1_PLAFQ 24 43 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne CRTM 35 43 Cc1ncc(CC(=O)NCCCCCCc2ccccc2)o1 ZINC000880830038 DG On-Demand Anodyne CES1D 67 42 O=C(Nc1cccc2c1OCCCO2)N1CC(C(F)(F)F)C1 ZINC000880830066 DF On-Demand Anodyne RBP4 53 35 O=C(NCc1ccnc(C(F)(F)F)c1)Nc1cccc2c1OCCCO2 ZINC000880830106 FH On-Demand Anodyne CARM1 21 40 COC[C@@H]1CCCN1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880830172 FC On-Demand Anodyne CTRA_BOVIN 48 33 COC[C@@H]1CCCN1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880830172 FC On-Demand Anodyne SIGMAR1 23 40 COC[C@@H]1CCCN1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880830172 FC On-Demand Anodyne TRY1_BOVIN 48 33 COC[C@@H]1CCCN1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880830172 FC On-Demand Anodyne PREP 41 36 COC[C@@H]1CCCN1NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880830172 FC On-Demand Anodyne CELA2A 41 33 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cccc2c1OCCCO2 ZINC000880830183 EE On-Demand Anodyne MTNR1A 15 43 O=C(NCC1CC=CC1)c1ccc(CN2CCOCC2)o1 ZINC000880830209 CD On-Demand Anodyne CACNA1I 61 40 O=C(NCc1cccnc1O)Nc1cccc2c1OCCCO2 ZINC000880830235 DE On-Demand Anodyne G2YM83_BOTF4 40 34 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](C2CCC2)C1 ZINC000880830245 DH On-Demand Anodyne RBP4 44 33 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](C2CCC2)C1 ZINC000880830247 DH On-Demand Anodyne RBP4 44 33 COC[C@@H]1CCCN1NC(=O)c1cc(C)co1 ZINC000880830290 BD On-Demand Anodyne CASP7 50 36 COC[C@@H]1CCCN1NC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880830293 DD On-Demand Anodyne CASP3 31 40 COC[C@@H]1CCCN1NC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880830293 DD On-Demand Anodyne CCR2 59 38 COC[C@@H]1CCCN1NC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880830293 DD On-Demand Anodyne CHRNA10 57 44 COC[C@@H]1CCCN1NC(=O)c1cc(C(F)(F)F)ccn1 ZINC000880830293 DD On-Demand Anodyne CASP7 47 40 COC[C@@H]1CCCN1NC(=O)c1c[nH]cc1C1CC1 ZINC000880830312 CD On-Demand Anodyne CASP7 46 38 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne CASP3 42 41 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne MTNR1A 31 40 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne MTNR1B 31 42 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne MMP3 40 39 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne CASP7 55 41 COC[C@@H]1CCCN1NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880830313 DD On-Demand Anodyne MMP1 37 40 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne CASP3 42 41 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne MTNR1A 31 40 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne MTNR1B 31 42 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne MMP3 40 39 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne CASP7 55 41 COC[C@@H]1CCCN1NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880830314 DD On-Demand Anodyne MMP1 37 40 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne PDGFRB 15 42 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne TIMP3 57 36 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne MTNR1A 41 67 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne MTNR1B 44 67 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne ROCK2 22 40 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne GALR2 24 42 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne EPHX2 22 45 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne ACR 16 40 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne AKR1C3 27 45 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne AKR1C2 41 36 COc1cccc(Nc2ccc(NC(=O)COC3CC3)cc2)c1 ZINC000880830345 DH On-Demand Anodyne KCNK3 40 36 O=C1CC[C@@H](c2ccc(C(=O)NCC3CC=CC3)cc2)N1 ZINC000880830366 CE On-Demand Anodyne CACNA1I 40 32 O=C1CC[C@H](c2ccc(C(=O)NCC3CC=CC3)cc2)N1 ZINC000880830367 CE On-Demand Anodyne CACNA1I 40 32 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cccc2c1OCCCO2 ZINC000880830407 GG On-Demand Anodyne STAT6 40 35 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne HRH2 17 43 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne DRD3 45 38 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne SCNN1A 47 40 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne SIGMAR1 24 42 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne SCN2A 21 41 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne S1PR3 17 42 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne FAAH 83 67 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne S1PR2 24 42 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne SLC6A5 23 41 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne CES1 72 44 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne AMP1_PLAFQ 25 44 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne DAGLA 17 40 Cn1nnc(C(=O)NCCCCCCc2ccccc2)n1 ZINC000880830426 CD On-Demand Anodyne CES1D 57 34 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2c1OCCCO2 ZINC000880830495 GG On-Demand Anodyne ACHE 22 42 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2c1OCCCO2 ZINC000880830495 GG On-Demand Anodyne HTR4 43 49 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cccc2c1OCCCO2 ZINC000880830495 GG On-Demand Anodyne CCR3 50 42 O=C(NCc1cnc(Cl)s1)Nc1cccc2c1OCCCO2 ZINC000880830516 EG On-Demand Anodyne G2YM83_BOTF4 46 33 COC[C@@H]1CCCN1NC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880830556 DE On-Demand Anodyne CASP3 45 38 COC[C@@H]1CCCN1NC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880830556 DE On-Demand Anodyne CASP7 57 40 COC[C@@H]1CCCN1NC(=O)C(C)(C)c1ccc(F)cc1F ZINC000880830556 DE On-Demand Anodyne ACKR3 45 33 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCc2ccccc21 ZINC000880830590 DH On-Demand Anodyne TRPV1 17 43 COC[C@@H]1CCCN1NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880830619 DF On-Demand Anodyne EBP 29 43 COC[C@@H]1CCCN1NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880830620 DF On-Demand Anodyne EBP 29 43 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2CC=CC2)N1Cc1ccccc1 ZINC000880830688 ED On-Demand Anodyne F2 23 40 O=C(Nc1cccc2c1OCCCO2)N1CC(C2CC2)C1 ZINC000880830690 CF On-Demand Anodyne RBP4 45 34 COc1ccccc1-c1ccc(C(=O)NCC2CC=CC2)c(O)n1 ZINC000880830717 DG On-Demand Anodyne DRD2 23 42 COc1ccccc1-c1ccc(C(=O)NCC2CC=CC2)c(O)n1 ZINC000880830717 DG On-Demand Anodyne KCNA3 42 35 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880830729 FF On-Demand Anodyne P2RX7 24 40 COC[C@@H]1CCCN1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880830734 ED On-Demand Anodyne CASP3 48 38 COC[C@@H]1CCCN1NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880830734 ED On-Demand Anodyne CASP7 60 38 COCCn1ncc(C(=O)Nc2ccc(-c3cccc(C)c3)cn2)c1C ZINC000880830757 FG On-Demand Anodyne LUCI_LUCLA 44 40 COC[C@@H]1CCCN1NC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880830774 FF On-Demand Anodyne FKBP1A 56 45 COC[C@@H]1CCCN1NC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880830774 FF On-Demand Anodyne MTNR1B 17 40 COC[C@@H]1CCCN1NC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880830774 FF On-Demand Anodyne CASP7 46 36 COC[C@@H]1CCCN1NC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880830774 FF On-Demand Anodyne ACKR3 68 37 O=C(NCc1nccc(C(F)(F)F)n1)Nc1cccc2c1OCCCO2 ZINC000880830804 FF On-Demand Anodyne TRPV1 18 40 COc1ccc(N2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)nc1 ZINC000880830805 GF On-Demand Anodyne DGAT1 29 46 O=C(Nc1cccc2c1OCCCO2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880830856 GF On-Demand Anodyne CHRNA4 25 44 Cc1ncc(CC(=O)N2CCN(C(=O)OC(C)(C)C)C[C@H]2C(C)C)o1 ZINC000880830871 FF On-Demand Anodyne GPR119 34 41 Cc1ncc(CC(=O)N2CCN(C(=O)OC(C)(C)C)C[C@@H]2C(C)C)o1 ZINC000880830872 FF On-Demand Anodyne GPR119 34 41 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880830874 GD On-Demand Anodyne HCN1 56 37 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880830874 GD On-Demand Anodyne HCN4 47 30 O=C1C[C@@]2(CCN(C(=O)Nc3cccc4c3OCCCO4)C2)Oc2ccccc21 ZINC000880830883 GG On-Demand Anodyne EPHX2 20 51 O=C1C[C@@]2(CCN(C(=O)Nc3cccc4c3OCCCO4)C2)Oc2ccccc21 ZINC000880830883 GG On-Demand Anodyne TRPM8 29 44 O=C1C[C@]2(CCN(C(=O)Nc3cccc4c3OCCCO4)C2)Oc2ccccc21 ZINC000880830884 GG On-Demand Anodyne EPHX2 20 51 O=C1C[C@]2(CCN(C(=O)Nc3cccc4c3OCCCO4)C2)Oc2ccccc21 ZINC000880830884 GG On-Demand Anodyne TRPM8 29 44 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)C(=O)NCCc1ccccc1 ZINC000880830893 GF On-Demand Anodyne MTNR1A 18 45 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc3c1OCCCO3)C2 ZINC000880830991 EF On-Demand Anodyne HTR3A 35 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cccc3c2OCCCO3)cc1 ZINC000880831012 GG On-Demand Anodyne LPL 57 33 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880831039 EF On-Demand Anodyne CPT1A 72 37 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880831040 EF On-Demand Anodyne CPT1A 72 37 O=C(NCc1ccncc1OCC(F)(F)F)Nc1cccc2c1OCCCO2 ZINC000880831214 GH On-Demand Anodyne TRPV1 19 40 COC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831292 EE On-Demand Anodyne EPHX2 45 41 Nc1ccc(CNC(=O)Nc2cccc3c2OCCCO3)cn1 ZINC000880831303 DE On-Demand Anodyne NAMPT 25 47 O=C(Nc1cccc2c1OCCCO2)N1CC(C2CCCC2)C1 ZINC000880831433 DH On-Demand Anodyne RBP4 44 33 O=C(NCC1CCN(C2CC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880831464 EF On-Demand Anodyne HTR4 26 40 N#Cc1ccc(OC2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)cc1 ZINC000880831555 GH On-Demand Mild EPHX2 15 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831586 GI On-Demand Anodyne SLC18A3 24 40 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831586 GI On-Demand Anodyne WNT3A 49 34 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000880831711 DH On-Demand Anodyne EPHX2 21 42 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1C[C@H]1c1ccccc1 ZINC000880831712 DH On-Demand Anodyne EPHX2 21 42 O=C(Nc1cccc2c1OCCCO2)N[C@H]1C[C@H]1c1ccccc1 ZINC000880831713 DH On-Demand Anodyne EPHX2 21 42 O=C(Nc1cccc2c1OCCCO2)N[C@H]1C[C@@H]1c1ccccc1 ZINC000880831714 DH On-Demand Anodyne EPHX2 21 42 CNC(=O)NC[C@H]1CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880831763 FC On-Demand Anodyne MTNR1A 20 41 CNC(=O)NC[C@H]1CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880831763 FC On-Demand Anodyne MTNR1B 18 41 C[C@@H]1CN(CCCNC(=O)Nc2cccc3c2OCCCO3)CCCO1 ZINC000880831766 FE On-Demand Anodyne CCR3 30 40 O=C(NCc1ncccc1F)Nc1cccc2c1OCCCO2 ZINC000880831767 DF On-Demand Anodyne G2YM83_BOTF4 40 33 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880831840 FF On-Demand Anodyne EPHX2 15 45 COc1cnccc1N1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831861 GF On-Demand Anodyne HTR1A 17 41 COc1cnccc1N1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831861 GF On-Demand Anodyne PDGFRB 31 42 COc1cnccc1N1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880831861 GF On-Demand Anodyne RBP4 15 41 O=C(Nc1cccc2c1CCO2)Nc1cccc2c1OCCCO2 ZINC000880831972 EG On-Demand Anodyne MTNR1A 17 42 O=C(Nc1cccc2c1CCO2)Nc1cccc2c1OCCCO2 ZINC000880831972 EG On-Demand Anodyne MTNR1B 15 46 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880831997 EF On-Demand Anodyne PLM1_PLAFA 40 38 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880831998 EF On-Demand Anodyne PLM1_PLAFA 40 38 O=C(Nc1cccc2c1OCCCO2)N[C@H]1c2ccccc2C[C@H]1O ZINC000880831999 EF On-Demand Anodyne PLM1_PLAFA 40 38 O=C(Nc1cccc2c1OCCCO2)N(CCO)Cc1cccnc1Cl ZINC000880832013 GF On-Demand Anodyne G2YM83_BOTF4 68 35 O=C(NC[C@H](O)[C@@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832153 DD On-Demand Anodyne GABRA1 18 44 O=C(NC[C@H](O)[C@@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832153 DD On-Demand Anodyne GABRA2 15 44 O=C(NC[C@@H](O)[C@@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832154 DD On-Demand Anodyne GABRA1 18 44 O=C(NC[C@@H](O)[C@@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832154 DD On-Demand Anodyne GABRA2 15 44 O=C(NC[C@H](O)[C@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832155 DD On-Demand Anodyne GABRA1 18 44 O=C(NC[C@H](O)[C@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832155 DD On-Demand Anodyne GABRA2 15 44 O=C(NC[C@@H](O)[C@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832156 DD On-Demand Anodyne GABRA1 18 44 O=C(NC[C@@H](O)[C@H]1CCCO1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880832156 DD On-Demand Anodyne GABRA2 15 44 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne TRY1_BOVIN 43 30 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne PREP 26 42 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne LGMN 71 41 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne KLK5 41 40 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 O=C(NC[C@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832190 GD On-Demand Anodyne TMPRSS11D 41 35 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne TRY1_BOVIN 43 30 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne PREP 26 42 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne LGMN 71 41 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne KLK5 41 40 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 O=C(NC[C@@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832191 GD On-Demand Anodyne TMPRSS11D 41 35 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne TRY1_BOVIN 43 30 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne PREP 26 42 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne LGMN 71 41 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne KLK5 41 40 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 O=C(NC[C@@H](O)[C@@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832192 GD On-Demand Anodyne TMPRSS11D 41 35 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne TRY1_BOVIN 43 30 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne PREP 26 42 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne LGMN 71 41 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne KLK5 41 40 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 O=C(NC[C@H](O)[C@H]1CCCO1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880832193 GD On-Demand Anodyne TMPRSS11D 41 35 O=C(Nc1cc(C2CC2)[nH]n1)Nc1cccc2c1OCCCO2 ZINC000880832326 DG On-Demand Anodyne CDK2 15 47 O=C(Nc1cc(C2CC2)[nH]n1)Nc1cccc2c1OCCCO2 ZINC000880832326 DG On-Demand Anodyne PKNB 71 38 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cccn2nccc12 ZINC000880832330 DC On-Demand Anodyne JAK3 17 40 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cccn2nccc12 ZINC000880832330 DC On-Demand Anodyne TYK2 20 40 O=C(NCC1(N2CCOCC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880832434 ED On-Demand Anodyne HCN1 56 34 O=C(NCC1(N2CCOCC2)CC1)Nc1cccc2c1OCCCO2 ZINC000880832434 ED On-Demand Anodyne HCN4 47 30 O=C(NC[C@H]1CCCN1CC(F)F)c1cncc2[nH]ccc12 ZINC000880832515 DE On-Demand Anodyne DRD2 31 40 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2c1OCCCO2 ZINC000880832524 EE On-Demand Anodyne MTNR1A 23 44 O=C(NCCCNC(=O)C1CCC1)Nc1cccc2c1OCCCO2 ZINC000880832524 EE On-Demand Anodyne TBK1 62 35 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832563 EE On-Demand Anodyne MTNR1A 16 44 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832563 EE On-Demand Anodyne MTNR1B 15 44 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832563 EE On-Demand Anodyne EPHX2 31 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832563 EE On-Demand Anodyne CCR8 52 41 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832564 EE On-Demand Anodyne MTNR1A 16 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832564 EE On-Demand Anodyne MTNR1B 15 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832564 EE On-Demand Anodyne EPHX2 31 40 CCOC(=O)N1CC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832564 EE On-Demand Anodyne CCR8 52 41 O=C(Nc1cccc2c1OCC2)c1cnc(CC2CC2)s1 ZINC000880832702 DG On-Demand Anodyne G2YM83_BOTF4 41 36 O=C(NCCc1ccccc1O)Nc1cccc2c1OCCCO2 ZINC000880832734 EF On-Demand Anodyne MTNR1A 15 53 C[C@H]1c2ccccc2CCN1C(=O)Nc1cccc2c1OCCCO2 ZINC000880832743 EH On-Demand Anodyne TRPM8 25 41 CC[C@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832755 CD On-Demand Anodyne MME 49 38 CC[C@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832755 CD On-Demand Anodyne ANPEP 46 33 CC[C@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832755 CD On-Demand Anodyne MMP3 43 37 CC[C@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832755 CD On-Demand Anodyne BLA1_STEMA 40 31 CC[C@@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832756 CD On-Demand Anodyne MME 49 38 CC[C@@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832756 CD On-Demand Anodyne ANPEP 46 33 CC[C@@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832756 CD On-Demand Anodyne MMP3 43 37 CC[C@@H](CCc1ccccc1)NC(=O)c1nnn(C)n1 ZINC000880832756 CD On-Demand Anodyne BLA1_STEMA 40 31 CC[C@@H](CCc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880832764 FG On-Demand Anodyne ACE 43 36 CC[C@@H](CCc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880832764 FG On-Demand Anodyne CTSC 23 40 CC[C@H](CCc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880832765 FG On-Demand Anodyne ACE 43 36 CC[C@H](CCc1ccccc1)NC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880832765 FG On-Demand Anodyne CTSC 23 40 O=C(COC1CC1)NCCc1cccc2c1OC(F)(F)O2 ZINC000880832819 CD On-Demand Anodyne MTNR1A 22 40 O=C(NC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1)C1CC1 ZINC000880832843 FE On-Demand Anodyne EPHX2 26 41 O=C(NCCc1cccc2c1OC(F)(F)O2)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880832855 GE On-Demand Anodyne MTNR1A 17 40 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880832870 GE On-Demand Anodyne CACNA1I 41 36 CS(=O)(=O)C1CCC(C(=O)NCCc2cccc3c2OC(F)(F)O3)CC1 ZINC000880832871 GE On-Demand Anodyne MTNR1A 42 47 CS(=O)(=O)C1CCC(C(=O)NCCc2cccc3c2OC(F)(F)O3)CC1 ZINC000880832871 GE On-Demand Anodyne MTNR1B 24 44 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832910 GG On-Demand Anodyne HTR4 32 40 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832910 GG On-Demand Anodyne CACNA1I 42 33 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832910 GG On-Demand Anodyne GPR119 31 41 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832911 GG On-Demand Anodyne HTR4 32 40 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832911 GG On-Demand Anodyne CACNA1I 42 33 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880832911 GG On-Demand Anodyne GPR119 31 41 Cc1nc(C(C)C)ncc1C(=O)Nc1cccc2c1OCC2 ZINC000880832932 CG On-Demand Anodyne G2YM83_BOTF4 59 42 O=C(NC[C@H]1CCCN1CC(F)F)c1cc2c(cc1[N+](=O)[O-])OCCCO2 ZINC000880832947 GE On-Demand Bother DRD2 30 43 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@H]1CCCN(C2CCC2)C1 ZINC000880832953 FH On-Demand Anodyne XIAP 16 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@H]1CCCN(C2CCC2)C1 ZINC000880832953 FH On-Demand Anodyne BIRC3 43 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@H]1CCCN(C2CCC2)C1 ZINC000880832953 FH On-Demand Anodyne BIRC2 23 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@@H]1CCCN(C2CCC2)C1 ZINC000880832955 FH On-Demand Anodyne XIAP 16 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@@H]1CCCN(C2CCC2)C1 ZINC000880832955 FH On-Demand Anodyne BIRC3 43 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@@H]1CCCN(C2CCC2)C1 ZINC000880832955 FH On-Demand Anodyne BIRC2 23 42 CC[C@@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832962 ED On-Demand Anodyne ACE 51 37 CC[C@@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832962 ED On-Demand Anodyne MME 46 36 CC[C@@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832962 ED On-Demand Anodyne KCNQ2 47 33 CC[C@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832963 ED On-Demand Anodyne ACE 51 37 CC[C@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832963 ED On-Demand Anodyne MME 46 36 CC[C@H](CCc1ccccc1)NC(=O)CN1CCCCS1(=O)=O ZINC000880832963 ED On-Demand Anodyne KCNQ2 47 33 O=C(NC[C@H]1CCCN1CC(F)F)c1ncccc1-c1ccccn1 ZINC000880832964 EF On-Demand Anodyne HCRTR1 28 41 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)N1C[C@H](O)C[C@H]1C(N)=O ZINC000880833024 GE On-Demand Anodyne VHL 48 32 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)[C@H]1CCCO1)C2 ZINC000880833027 DD On-Demand Anodyne MTNR1A 34 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)[C@H]1CCCO1)C2 ZINC000880833027 DD On-Demand Anodyne MTNR1B 29 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)[C@@H]1CCCO1)C2 ZINC000880833028 DD On-Demand Anodyne MTNR1A 34 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)[C@@H]1CCCO1)C2 ZINC000880833028 DD On-Demand Anodyne MTNR1B 29 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)[C@H]1CCCO1)C2 ZINC000880833029 DD On-Demand Anodyne MTNR1A 34 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H](O)[C@H]1CCCO1)C2 ZINC000880833029 DD On-Demand Anodyne MTNR1B 29 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)[C@@H]1CCCO1)C2 ZINC000880833030 DD On-Demand Anodyne MTNR1A 34 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H](O)[C@@H]1CCCO1)C2 ZINC000880833030 DD On-Demand Anodyne MTNR1B 29 43 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cc2ccccc2cc1F ZINC000880833059 EE On-Demand Anodyne HTR1A 15 40 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cc2ccccc2cc1F ZINC000880833059 EE On-Demand Anodyne DRD2 20 42 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cc2ccccc2cc1F ZINC000880833059 EE On-Demand Anodyne POLR1A 47 35 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cccc2c1OCCCO2 ZINC000880833079 GG On-Demand Anodyne HTR4 35 42 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cccc2c1OCCCO2 ZINC000880833079 GG On-Demand Anodyne CACNA1I 43 34 O=C(NCCN1CCCOCC1)Nc1cccc2c1OCCCO2 ZINC000880833205 ED On-Demand Anodyne EPHX2 19 44 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cnc(CC2CC2)s1 ZINC000880833278 ED On-Demand Anodyne SIRT3 52 34 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cnc(CC2CC2)s1 ZINC000880833278 ED On-Demand Anodyne SIRT2 53 34 NC(=O)[C@@H]1CCCN1CCCNC(=O)c1cnc(CC2CC2)s1 ZINC000880833278 ED On-Demand Anodyne SIRT1 42 34 COC(=O)C1=CC[C@H](NC(=O)c2cc(-c3ccc(OC)cc3)on2)C1 ZINC000880833340 EE On-Demand Anodyne PDK1 46 35 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880833381 GF On-Demand Anodyne CCR3 48 37 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880833382 GF On-Demand Anodyne CCR3 48 37 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)c1 ZINC000880833456 II On-Demand Anodyne ROCK1 19 41 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)c1 ZINC000880833456 II On-Demand Anodyne ROCK2 15 41 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)c1 ZINC000880833456 II On-Demand Anodyne KCNK3 58 39 Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)c1 ZINC000880833456 II On-Demand Anodyne KCNK9 46 39 O=C(NC[C@H](O)[C@H]1CCCO1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880833466 EE On-Demand Anodyne PDE4D 17 42 O=C(NC[C@H](O)[C@@H]1CCCO1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880833467 EE On-Demand Anodyne PDE4D 17 42 O=C(NC[C@@H](O)[C@@H]1CCCO1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880833468 EE On-Demand Anodyne PDE4D 17 42 O=C(NC[C@@H](O)[C@H]1CCCO1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880833469 EE On-Demand Anodyne PDE4D 17 42 Cc1cc(NC(=O)Nc2cccc3c2OCCCO3)c(C)c(C)c1O ZINC000880833490 EI On-Demand Anodyne LPL 49 34 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1ccccc1 ZINC000880833495 EF On-Demand Anodyne MME 40 40 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1ccccc1 ZINC000880833495 EF On-Demand Anodyne ANPEP 51 31 O=C(Nc1cccc2c1OCCCO2)NC12CCC(CC1)C2 ZINC000880833562 DG On-Demand Anodyne EPHX2 34 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc2c1OCC2 ZINC000880833586 FE On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc2c1OCC2 ZINC000880833587 FE On-Demand Anodyne FPR1 45 36 O=C(CCOc1ccccc1)NNC(=O)Nc1cccc2c1OCCCO2 ZINC000880833611 FE On-Demand Reactive CYSLTR2 41 34 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCN2CC(F)F)c1 ZINC000880833624 DF On-Demand Anodyne DRD2 34 43 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCN2CC(F)F)c1 ZINC000880833624 DF On-Demand Anodyne CACNA1I 53 36 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCN2CC(F)F)c1 ZINC000880833625 DF On-Demand Anodyne DRD2 34 43 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCN2CC(F)F)c1 ZINC000880833625 DF On-Demand Anodyne CACNA1I 53 36 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne ACE 55 37 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne MME 48 37 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne TIMP3 44 33 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne MMP2 20 41 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne MMP3 31 41 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne CTSC 24 43 CC[C@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833677 EF On-Demand Anodyne XIAP 47 35 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne ACE 55 37 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne MME 48 37 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne TIMP3 44 33 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne MMP2 20 41 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne MMP3 31 41 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne CTSC 24 43 CC[C@@H](CCc1ccccc1)NC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880833678 EF On-Demand Anodyne XIAP 47 35 CCOC(=O)CCC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880833683 GG On-Demand Anodyne CCR8 39 40 Cc1coc(C(=O)NC[C@@H]2CCCN2CC(F)F)c1 ZINC000880833687 CE On-Demand Anodyne DRD2 33 40 Cc1coc(C(=O)NC[C@H]2CCCN2CC(F)F)c1 ZINC000880833688 CE On-Demand Anodyne DRD2 33 40 O=C(CCCc1ccccc1)NNC(=O)Nc1cccc2c1OCCCO2 ZINC000880833704 FG On-Demand Reactive MTNR1A 15 47 O=C(Cc1ccccc1N1CCCC1=O)Nc1cccc2c1OCC2 ZINC000880833724 EF On-Demand Anodyne KCNQ2 74 47 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833758 GF On-Demand Anodyne DRD2 55 47 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833758 GF On-Demand Anodyne DRD3 28 46 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833758 GF On-Demand Anodyne ACKR3 65 33 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833759 GF On-Demand Anodyne DRD2 55 47 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833759 GF On-Demand Anodyne DRD3 28 46 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCN2CC(F)F)c(O)n1 ZINC000880833759 GF On-Demand Anodyne ACKR3 65 33 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne ACE 69 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne MME 71 40 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CTSG 15 40 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CTSK 32 43 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne TIMP3 95 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CTRB1 25 40 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne MMP2 35 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne MMP3 63 40 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CTSS 18 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CAPN1 63 35 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne MMP9 18 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CAPN2 80 37 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne ACE2 48 37 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne CTSC 22 43 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne MMP1 28 41 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne NPR 46 36 CC[C@@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833778 CF On-Demand Anodyne PSMB5 40 39 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne ACE 69 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne MME 71 40 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CTSG 15 40 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CTSK 32 43 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne TIMP3 95 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CTRB1 25 40 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne MMP2 35 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne MMP3 63 40 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CTSS 18 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CAPN1 63 35 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne MMP9 18 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CAPN2 80 37 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne ACE2 48 37 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne CTSC 22 43 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne MMP1 28 41 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne NPR 46 36 CC[C@H](CCc1ccccc1)NC(=O)COC1CC1 ZINC000880833779 CF On-Demand Anodyne PSMB5 40 39 COc1cc(N2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)ncn1 ZINC000880833794 GE On-Demand Anodyne PDGFRB 54 41 CC[C@@H](CCc1ccccc1)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880833899 FH On-Demand Anodyne ACE 37 40 CC[C@@H](CCc1ccccc1)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880833899 FH On-Demand Anodyne PSMB5 25 44 CC[C@H](CCc1ccccc1)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880833900 FH On-Demand Anodyne ACE 37 40 CC[C@H](CCc1ccccc1)NC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880833900 FH On-Demand Anodyne PSMB5 25 44 CC[C@@H](CCc1ccccc1)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880833901 FH On-Demand Anodyne ACE 37 40 CC[C@@H](CCc1ccccc1)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880833901 FH On-Demand Anodyne PSMB5 25 44 CC[C@H](CCc1ccccc1)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880833902 FH On-Demand Anodyne ACE 37 40 CC[C@H](CCc1ccccc1)NC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880833902 FH On-Demand Anodyne PSMB5 25 44 O=C(NC[C@H]1CCCN1CC(F)F)c1ccc(CN2CCOCC2)o1 ZINC000880833964 FD On-Demand Anodyne DRD2 30 40 O=C(Nc1cccc2c1OCCCO2)N1CCOc2ncccc2C1 ZINC000880833975 EF On-Demand Anodyne G2YM83_BOTF4 40 34 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880834006 FD On-Demand Anodyne MTNR1A 15 50 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880834007 FD On-Demand Anodyne MTNR1A 15 50 CN1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880834018 DD On-Demand Anodyne HTR4 37 40 CN1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880834019 DD On-Demand Anodyne HTR4 37 40 Cn1nnc(C(=O)Nc2cccc3c2OCC3)n1 ZINC000880834054 BC On-Demand Anodyne G2YM83_BOTF4 42 38 O=C1CC[C@@H](c2ccc(C(=O)NC[C@H]3CCCN3CC(F)F)cc2)N1 ZINC000880834081 FE On-Demand Anodyne PLD1 41 33 O=C1CC[C@@H](c2ccc(C(=O)NC[C@@H]3CCCN3CC(F)F)cc2)N1 ZINC000880834082 FE On-Demand Anodyne PLD1 41 33 O=C1CC[C@H](c2ccc(C(=O)NC[C@H]3CCCN3CC(F)F)cc2)N1 ZINC000880834083 FE On-Demand Anodyne PLD1 41 33 O=C1CC[C@H](c2ccc(C(=O)NC[C@@H]3CCCN3CC(F)F)cc2)N1 ZINC000880834084 FE On-Demand Anodyne PLD1 41 33 CC[C@@H](CCc1ccccc1)NC(=O)c1nccnc1SC ZINC000880834100 DG On-Demand Anodyne CTSC 15 40 CC[C@H](CCc1ccccc1)NC(=O)c1nccnc1SC ZINC000880834101 DG On-Demand Anodyne CTSC 15 40 CC[C@@H](CCc1ccccc1)NC(=O)C[C@H]1CCNC1=O ZINC000880834124 CE On-Demand Anodyne GALR1 49 35 CC[C@@H](CCc1ccccc1)NC(=O)C[C@H]1CCNC1=O ZINC000880834124 CE On-Demand Anodyne CTSC 26 41 CC[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1CCNC1=O ZINC000880834125 CE On-Demand Anodyne GALR1 49 35 CC[C@@H](CCc1ccccc1)NC(=O)C[C@@H]1CCNC1=O ZINC000880834125 CE On-Demand Anodyne CTSC 26 41 CC[C@H](CCc1ccccc1)NC(=O)C[C@H]1CCNC1=O ZINC000880834126 CE On-Demand Anodyne GALR1 49 35 CC[C@H](CCc1ccccc1)NC(=O)C[C@H]1CCNC1=O ZINC000880834126 CE On-Demand Anodyne CTSC 26 41 CC[C@H](CCc1ccccc1)NC(=O)C[C@@H]1CCNC1=O ZINC000880834127 CE On-Demand Anodyne GALR1 49 35 CC[C@H](CCc1ccccc1)NC(=O)C[C@@H]1CCNC1=O ZINC000880834127 CE On-Demand Anodyne CTSC 26 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834164 GD On-Demand Anodyne F2 48 40 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834164 GD On-Demand Anodyne DRD2 32 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834164 GD On-Demand Anodyne CTRA_BOVIN 40 31 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834164 GD On-Demand Anodyne TRY1_BOVIN 52 34 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834164 GD On-Demand Anodyne TMPRSS11D 59 34 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834165 GD On-Demand Anodyne F2 48 40 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834165 GD On-Demand Anodyne DRD2 32 41 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834165 GD On-Demand Anodyne CTRA_BOVIN 40 31 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834165 GD On-Demand Anodyne TRY1_BOVIN 52 34 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCCN2CC(F)F)N1Cc1ccccc1 ZINC000880834165 GD On-Demand Anodyne TMPRSS11D 59 34 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1ccccc1 ZINC000880834166 EF On-Demand Anodyne MME 40 40 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1ccccc1 ZINC000880834166 EF On-Demand Anodyne ANPEP 51 31 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)[nH]n1 ZINC000880834213 CD On-Demand Anodyne JUN 18 43 COC(=O)c1cc(NC(=O)Nc2cccc3c2OCCCO3)cn1C ZINC000880834214 EF On-Demand Anodyne LPL 54 32 COCCC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880834232 GD On-Demand Anodyne EPHX2 36 42 COCCC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880834232 GD On-Demand Anodyne CCR8 57 37 O=C(CC[C@@H]1CCc2ccccc21)N1CCCC(F)(F)CC1 ZINC000880834233 DI On-Demand Anodyne EBP 18 42 O=C(CC[C@H]1CCc2ccccc21)N1CCCC(F)(F)CC1 ZINC000880834234 DI On-Demand Anodyne EBP 18 42 CN(CCOc1ccccc1C(=O)NN1CCOC1=O)C(=O)OC(C)(C)C ZINC000880834279 GE On-Demand Anodyne HCN1 57 33 CN(CCOc1ccccc1C(=O)NN1CCOC1=O)C(=O)OC(C)(C)C ZINC000880834279 GE On-Demand Anodyne HCN4 40 31 O=C(c1cnc2cc[nH]c2c1)N1CCCC(F)(F)CC1 ZINC000880834316 CF On-Demand Anodyne ACACA 23 55 O=C(Nc1cccc2c1OCCCO2)N1CCN(c2ccc(F)cn2)CC1 ZINC000880834337 FF On-Demand Anodyne DGAT1 28 46 O=C(Nc1cccc2c1OCCCO2)N1CCN(c2ccc(F)cn2)CC1 ZINC000880834337 FF On-Demand Anodyne SLC27A1 40 40 Cc1cncc(CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880834506 DF On-Demand Anodyne NAMPT 29 48 O=C(NN1CCOC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880834566 FD On-Demand Anodyne CTRA_BOVIN 53 30 O=C(NN1CCOC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880834566 FD On-Demand Anodyne PREP 28 41 O=C(NN1CCOC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880834566 FD On-Demand Anodyne LGMN 54 38 O=C(NN1CCOC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880834566 FD On-Demand Anodyne SLC12A5 51 35 O=C(NN1CCOC1=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880834566 FD On-Demand Anodyne Q9NAW4_PLAFA 38 44 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cccc2c1OCCCO2 ZINC000880834651 DD On-Demand Anodyne LGMN 44 31 O=C1CC[C@@H](c2ccc(C(=O)N3CCCC(F)(F)CC3)cc2)N1 ZINC000880834743 DF On-Demand Anodyne L3MBTL3 58 38 O=C1CC[C@H](c2ccc(C(=O)N3CCCC(F)(F)CC3)cc2)N1 ZINC000880834744 DF On-Demand Anodyne L3MBTL3 58 38 O=C(Nc1cccc2c1OCCCO2)N1CCC(Cc2cccnc2)CC1 ZINC000880834927 FH On-Demand Anodyne CCR3 21 41 O=C(Nc1cccc2c1OCCCO2)N1CCC(Cc2cccnc2)CC1 ZINC000880834927 FH On-Demand Anodyne CHRNA7 47 42 O=C(Nc1cccc2c1OCCCO2)N1CCC(Cc2cccnc2)CC1 ZINC000880834927 FH On-Demand Anodyne C3AR1 40 40 CCN(CCNC(=O)OC(C)(C)C)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880834943 GF On-Demand Anodyne MPO 43 35 CCn1nc2c(cc1=O)CN(C(=O)Nc1cccc3c1OCCCO3)CC2 ZINC000880835139 FE On-Demand Anodyne P2RY14 43 33 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880835150 GH On-Demand Anodyne ETHR 43 41 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880835151 GH On-Demand Anodyne ETHR 43 41 O=C(Nc1cccc2c1OCCCO2)N1CCn2c(nnc2-c2ccccc2)C1 ZINC000880835177 GG On-Demand Anodyne P2RX7 25 43 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCN(c2ncccc2Cl)C1 ZINC000880835206 GG On-Demand Anodyne G2YM83_BOTF4 44 32 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCN(c2ncccc2Cl)C1 ZINC000880835210 GG On-Demand Anodyne G2YM83_BOTF4 44 32 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCCC(F)(F)CC2)N1Cc1ccccc1 ZINC000880835219 FE On-Demand Anodyne PREP 72 42 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCOC1=O)C2 ZINC000880835229 CD On-Demand Anodyne MTNR1A 23 41 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCOC1=O)C2 ZINC000880835229 CD On-Demand Anodyne MTNR1B 21 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(OC)n[nH]1)C2 ZINC000880835254 DE On-Demand Anodyne GSK3A 17 40 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(OC)n[nH]1)C2 ZINC000880835254 DE On-Demand Anodyne ROCK2 22 41 COc1cc(NC(=O)c2ncsc2C2CC2)[nH]n1 ZINC000880835261 CE On-Demand Anodyne MAP1 62 36 O=C(Nc1cccc2c1OCCCO2)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880835282 GD On-Demand Anodyne EPHX2 29 48 O=C(NCc1ccccc1N1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880835314 GG On-Demand Anodyne KCNQ2 69 39 CC[C@@H](CN1CCCC1)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880835316 EF On-Demand Anodyne KCNQ2 44 34 CC[C@H](CN1CCCC1)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880835317 EF On-Demand Anodyne KCNQ2 44 34 O=C(Nc1cccc2c1OCCCO2)N1CCN(c2ccccc2O)CC1 ZINC000880835320 FF On-Demand Anodyne KCNQ2 65 34 C[C@@H]1CCCN(C(=O)Nc2cccc3c2OCCCO3)[C@@H]1C ZINC000880835343 DH On-Demand Anodyne TRPC6 50 36 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cccc2c1OCCCO2 ZINC000880835344 DH On-Demand Anodyne TRPC6 50 36 O=C(Nc1cccc2c1OCCCO2)NC1CCN(C2CCCC2)CC1 ZINC000880835354 FG On-Demand Anodyne EPHX2 27 40 O=C(Nc1cccc2c1OCCCO2)N1CCC(O)(C(F)(F)F)CC1 ZINC000880835385 FF On-Demand Anodyne TRPM8 30 41 CCN1CCC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835426 DE On-Demand Anodyne MTNR1A 15 42 CCN1CCC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835428 DE On-Demand Anodyne MTNR1A 15 42 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)[nH]n1 ZINC000880835432 DD On-Demand Anodyne AURKA 18 42 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@H](O)Cc1ccccc1 ZINC000880835467 FF On-Demand Anodyne MME 41 34 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)[C@@H](O)Cc1ccccc1 ZINC000880835468 FF On-Demand Anodyne MME 41 34 CSCC[C@H](NC(=O)[C@@H]1C[C@]1(C)c1ccccc1)C(N)=O ZINC000880835498 DD On-Demand Anodyne GAG-PRO 48 38 O=C(Nc1cccc2c1OCCCO2)N(CCO)CCN1CCOCC1 ZINC000880835524 FD On-Demand Anodyne CASR 63 45 O=C(Nc1cccc2c1OCCCO2)N1CCOC2(CCC2)C1 ZINC000880835625 DF On-Demand Anodyne EPHX2 16 42 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835627 FD On-Demand Anodyne HTR4 34 43 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835627 FD On-Demand Anodyne LPL 44 33 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835629 FD On-Demand Anodyne HTR4 34 43 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835629 FD On-Demand Anodyne LPL 44 33 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835710 FD On-Demand Anodyne CCR8 79 37 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880835711 FD On-Demand Anodyne CCR8 79 37 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cccc2c1OCCCO2 ZINC000880835720 FG On-Demand Anodyne TRPV1 18 40 C[S@@](=O)CCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880835733 DD On-Demand Anodyne MTNR1A 17 49 O=C(Nc1cccc2c1OCCCO2)N1CCC(N2CC=CC2)CC1 ZINC000880835852 EF On-Demand Anodyne L3MBTL3 54 35 O=C(Nc1cccc2c1OCCCO2)N1CCOC2(CCCC2)C1 ZINC000880835861 EG On-Demand Anodyne EPHX2 16 42 CSCC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(N)=O ZINC000880835864 ED On-Demand Anodyne KCNQ2 49 33 CSCC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(N)=O ZINC000880835864 ED On-Demand Anodyne FURIN 53 43 CSCC[C@H](NC(=O)Cc1ccccc1N1CCCC1=O)C(N)=O ZINC000880835864 ED On-Demand Anodyne POLG_WNV 41 30 O=C(Nc1cccc2c1OCCCO2)N1CC(CC(F)(F)F)C1 ZINC000880835910 EG On-Demand Anodyne RBP4 45 33 Cc1c(NC(=O)OC(C)(C)C)cccc1NC(=O)c1cccn2nccc12 ZINC000880835934 FI On-Demand Anodyne PIM1 49 32 Cc1c(NC(=O)OC(C)(C)C)cccc1NC(=O)c1cccn2nccc12 ZINC000880835934 FI On-Demand Anodyne EPHB3 37 43 Cc1c(NC(=O)OC(C)(C)C)cccc1NC(=O)c1cccn2nccc12 ZINC000880835934 FI On-Demand Anodyne PIM3 41 32 Cc1c(NC(=O)OC(C)(C)C)cccc1NC(=O)c1cccn2nccc12 ZINC000880835934 FI On-Demand Anodyne G2YM83_BOTF4 44 32 C[C@@H](CNc1ccccc1)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880835938 EG On-Demand Anodyne LPL 42 32 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1cccc2c1OCCCO2 ZINC000880835981 FH On-Demand Anodyne NPY5R 17 41 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)cnc1OC ZINC000880836008 ED On-Demand Anodyne SSTR5 42 36 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)cnc1OC ZINC000880836008 ED On-Demand Anodyne MET 16 40 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)cnc1OC ZINC000880836008 ED On-Demand Anodyne EPHX2 17 40 COc1cc(NC(=O)c2ccc(CN3CCOCC3)o2)cnc1OC ZINC000880836008 ED On-Demand Anodyne AURKA 19 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CC[C@H]2CC[C@@H](C1)S2 ZINC000880836012 GI On-Demand Anodyne RBP4 41 39 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cccc2c1OCCCO2 ZINC000880836067 GF On-Demand Anodyne NPFFR2 40 40 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cccc2c1OCCCO2 ZINC000880836067 GF On-Demand Anodyne NPFFR1 50 40 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cccc2c1OCCCO2 ZINC000880836068 GF On-Demand Anodyne NPFFR2 40 40 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cccc2c1OCCCO2 ZINC000880836068 GF On-Demand Anodyne NPFFR1 50 40 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)cnc1OC ZINC000880836096 DF On-Demand Anodyne KCNK3 44 40 COc1cc(NC(=O)c2cnc(C(C)C)nc2C)cnc1OC ZINC000880836096 DF On-Demand Anodyne KCNK9 38 40 COc1ccccc1[C@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880836124 FH On-Demand Anodyne RBP4 54 42 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880836125 FH On-Demand Anodyne RBP4 54 42 O=C(Nc1cccc2c1OCCCO2)N1CCCN(C2CCCC2)CC1 ZINC000880836161 FG On-Demand Anodyne HRH3 25 44 O=C(Nc1cccc2c1OCCCO2)N1CCCN(C2CCCC2)CC1 ZINC000880836161 FG On-Demand Anodyne L3MBTL3 55 36 COC(=O)c1cnc(C2CCN(C(=O)CC[C@H]3CC(C)(C)CO3)CC2)s1 ZINC000880836175 GG On-Demand Anodyne ETHR 51 35 COC(=O)c1cnc(C2CCN(C(=O)CC[C@@H]3CC(C)(C)CO3)CC2)s1 ZINC000880836176 GG On-Demand Anodyne ETHR 51 35 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne TACR1 24 43 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne CCKAR 76 44 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne CTSL 23 42 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne NMBR 74 33 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne GRPR 47 34 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne ECE1 52 40 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne MMP11 62 33 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne CCKBR 55 44 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836199 GG On-Demand Anodyne GHSR 47 43 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne TACR1 24 43 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne CCKAR 76 44 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne CTSL 23 42 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne NMBR 74 33 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne GRPR 47 34 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne ECE1 52 40 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne MMP11 62 33 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne CCKBR 55 44 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000880836200 GG On-Demand Anodyne GHSR 47 43 O=C(NC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1)c1ccccc1 ZINC000880836203 GG On-Demand Anodyne CCR8 45 37 O=C(Nc1cccc2c1OCCCO2)N1CCN(C2CC2)CC1 ZINC000880836278 DE On-Demand Anodyne L3MBTL3 45 35 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H]4CC[C@@H](C3)S4)cc2)N1 ZINC000880836289 EF On-Demand Anodyne L3MBTL3 53 38 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@H]4CC[C@@H](C3)S4)cc2)N1 ZINC000880836290 EF On-Demand Anodyne L3MBTL3 53 38 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cccc3c1OCCCO3)C2 ZINC000880836305 EF On-Demand Anodyne HTR3A 36 44 CCCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836336 EG On-Demand Anodyne HTR4 48 40 CCCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836336 EG On-Demand Anodyne CHRM3 15 43 CCCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836336 EG On-Demand Anodyne MTNR1A 15 40 CCCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836336 EG On-Demand Anodyne EPHX2 30 42 COC(=O)c1cnc(C2CCN(C(=O)c3cnc(CC4CC4)s3)CC2)s1 ZINC000880836339 GG On-Demand Anodyne PTR1 46 33 O=C(Nc1cccc2c1OCCCO2)N1CCO[C@@H](C(F)(F)F)C1 ZINC000880836370 EF On-Demand Anodyne RBP4 45 34 O=C(Nc1cccc2c1OCCCO2)N1CCO[C@H](C(F)(F)F)C1 ZINC000880836371 EF On-Demand Anodyne RBP4 45 34 COc1cc(NC(=O)c2ncsc2C2CC2)cnc1OC ZINC000880836390 DF On-Demand Anodyne MAP1 76 36 N#CCCN(CCN1CCOCC1)C(=O)Nc1cccc2c1OCCCO2 ZINC000880836418 FD On-Demand Mild CASR 59 45 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC[C@H]1CCCN1C ZINC000880836419 CD On-Demand Anodyne CHRNA10 52 34 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC[C@H]1CCCN1C ZINC000880836420 CD On-Demand Anodyne CHRNA10 52 34 C=CC(C)(C)CC(=O)Nc1cnc(OC)c(OC)c1 ZINC000880836442 CF On-Demand Mild ENPP1 70 34 O=C(Nc1cccc2c1OCCCO2)N[C@@H](CO)c1cccc(F)c1 ZINC000880836489 EF On-Demand Anodyne KCNQ2 21 40 O=C(Nc1cccc2c1OCCCO2)N[C@H](CO)c1cccc(F)c1 ZINC000880836490 EF On-Demand Anodyne KCNQ2 21 40 O=C(NCCCc1ccc(O)cc1)Nc1cccc2c1OCCCO2 ZINC000880836555 EG On-Demand Anodyne MTNR1A 20 48 O=C(Nc1cccc2c1OCCCO2)N1CCN(CC2CCOCC2)CC1 ZINC000880836579 GE On-Demand Anodyne TACR2 21 41 CS(=O)(=O)C1CCC(C(=O)Nc2nccc3cc[nH]c23)CC1 ZINC000880836588 DE On-Demand Anodyne GSK3B 19 40 CS(=O)(=O)C1CCC(C(=O)Nc2nccc3cc[nH]c23)CC1 ZINC000880836588 DE On-Demand Anodyne GSK3A 36 40 O=C(Nc1cccc2c1OCCCO2)N1CCC(C(F)(F)F)CC1 ZINC000880836590 EH On-Demand Anodyne RBP4 39 40 COC(=O)c1cnc(C2CCN(C(=O)CC(C)(C)CC(F)(F)F)CC2)s1 ZINC000880836594 GI On-Demand Anodyne ETHR 42 34 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2CC[C@@H](C1)S2 ZINC000880836611 CF On-Demand Anodyne JAK1 22 41 O=C(NC[C@H](O)c1cccc(Cl)c1)Nc1cccc2c1OCCCO2 ZINC000880836685 FG On-Demand Anodyne ADRB3 39 40 O=C(NC[C@H](O)c1cccc(Cl)c1)Nc1cccc2c1OCCCO2 ZINC000880836685 FG On-Demand Anodyne CYP3A4 40 32 O=C(NC[C@@H](O)c1cccc(Cl)c1)Nc1cccc2c1OCCCO2 ZINC000880836686 FG On-Demand Anodyne ADRB3 39 40 O=C(NC[C@@H](O)c1cccc(Cl)c1)Nc1cccc2c1OCCCO2 ZINC000880836686 FG On-Demand Anodyne CYP3A4 40 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(Cl)oc2ccccc12 ZINC000880836710 GH On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(Cl)oc2ccccc12 ZINC000880836710 GH On-Demand Anodyne FPR1 44 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(Cl)oc2ccccc12 ZINC000880836714 GH On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1c(Cl)oc2ccccc12 ZINC000880836714 GH On-Demand Anodyne FPR1 44 36 CN1CCC(CNC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836722 DE On-Demand Anodyne HTR4 42 42 CN1CCC(CNC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880836722 DE On-Demand Anodyne CACNA1I 41 33 CC1(C)CC[C@@H](CC(=O)N[C@@H](c2ccccn2)C2CCC2)OC1 ZINC000880836741 DH On-Demand Anodyne TTK 27 43 CC1(C)CC[C@@H](CC(=O)N[C@H](c2ccccn2)C2CCC2)OC1 ZINC000880836744 DH On-Demand Anodyne TTK 27 43 O=C(Nn1cccn1)c1c[nH]cc1C1CC1 ZINC000880836751 BD On-Demand Anodyne HTR1F 65 35 O=C(COC1CC1)N[C@H](c1ccccn1)C1CCC1 ZINC000880836753 CE On-Demand Anodyne TTK 34 46 O=C(COC1CC1)N[C@@H](c1ccccn1)C1CCC1 ZINC000880836755 CE On-Demand Anodyne TTK 34 46 Cn1nnc(C(=O)N[C@@H](c2ccccn2)C2CCC2)n1 ZINC000880836768 CC On-Demand Anodyne TTK 41 47 Cn1nnc(C(=O)N[C@H](c2ccccn2)C2CCC2)n1 ZINC000880836769 CC On-Demand Anodyne TTK 41 47 Cc1coc(C(=O)N[C@H](c2ccccn2)C2CCC2)c1 ZINC000880836778 CG On-Demand Anodyne TTK 35 45 Cc1coc(C(=O)N[C@@H](c2ccccn2)C2CCC2)c1 ZINC000880836781 CG On-Demand Anodyne TTK 35 45 O=C(N[C@H](c1ccccn1)C1CCC1)c1cccc2nsnc12 ZINC000880836786 DG On-Demand Anodyne TTK 25 41 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cccc2nsnc12 ZINC000880836790 DG On-Demand Anodyne TTK 25 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836809 ED On-Demand Reactive PGC 43 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836809 ED On-Demand Reactive PAPA1_CARPA 38 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836809 ED On-Demand Reactive REN 53 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836809 ED On-Demand Reactive FPR1 46 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836811 ED On-Demand Reactive PGC 43 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836811 ED On-Demand Reactive PAPA1_CARPA 38 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836811 ED On-Demand Reactive REN 53 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NN(C)c1ccccn1 ZINC000880836811 ED On-Demand Reactive FPR1 46 37 O=C(CC[C@H]1CCc2ccccc21)Nn1cccn1 ZINC000880836814 CE On-Demand Anodyne NQO2 19 40 O=C(CC[C@@H]1CCc2ccccc21)Nn1cccn1 ZINC000880836817 CE On-Demand Anodyne NQO2 19 40 O=C(Nn1cccn1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880836833 ED On-Demand Anodyne GRIN2B 20 43 O=C(Nn1cccn1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880836833 ED On-Demand Anodyne PREP 27 41 O=C(Nn1cccn1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880836833 ED On-Demand Anodyne LGMN 52 38 O=C(Nn1cccn1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880836833 ED On-Demand Anodyne SLC12A5 51 35 O=C(Nn1cccn1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880836833 ED On-Demand Anodyne Q9NAW4_PLAFA 39 46 COc1ccccc1-c1ccc(C(=O)N[C@H](c2ccccn2)C2CCC2)c(O)n1 ZINC000880836841 GI On-Demand Anodyne TTK 21 41 COc1ccccc1-c1ccc(C(=O)N[C@@H](c2ccccn2)C2CCC2)c(O)n1 ZINC000880836842 GI On-Demand Anodyne TTK 21 41 Cc1nc(C(C)C)ncc1C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880836916 DH On-Demand Anodyne TTK 22 40 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880836917 DH On-Demand Anodyne TTK 22 40 COc1ccccc1[C@@H](O)CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880836941 FF On-Demand Anodyne SOAT1 28 43 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)C(=O)Nc1ccccc1 ZINC000880836957 FF On-Demand Anodyne LPL 43 33 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837014 GG On-Demand Anodyne EPHX2 44 40 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837014 GG On-Demand Anodyne CCR8 32 42 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](N2CCCC2)C1 ZINC000880837040 EF On-Demand Anodyne L3MBTL3 93 43 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](N2CCCC2)C1 ZINC000880837041 EF On-Demand Anodyne L3MBTL3 93 43 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880837045 GI On-Demand Anodyne PRCP 43 37 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880837046 GI On-Demand Anodyne PRCP 43 37 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne HTR1A 70 45 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne DRD2 52 53 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne ADRA1D 63 53 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne HTR1B 15 40 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne ADRA1A 53 53 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne ADRA1B 50 53 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne DRD3 50 40 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne HTR7 40 38 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne KCNQ2 61 34 COc1ccccc1N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837055 GH On-Demand Anodyne MTNR1A 16 45 N#Cc1ccccc1N1CCCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837076 GG On-Demand Mild KCNQ2 56 33 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCCc2nc(O)ccc21 ZINC000880837089 FG On-Demand Anodyne TRPV1 16 41 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCCc2nc(O)ccc21 ZINC000880837090 FG On-Demand Anodyne TRPV1 16 41 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CC(F)F)CC1 ZINC000880837091 FF On-Demand Anodyne EPHX2 36 40 COC(=O)[C@@]1(OC)CCN(C(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880837137 DC On-Demand Anodyne ACACA 22 49 O=C(NN1CCS(=O)(=O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880837142 GC On-Demand Anodyne PREP 27 41 O=C(NN1CCS(=O)(=O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880837142 GC On-Demand Anodyne LGMN 62 39 O=C(NN1CCS(=O)(=O)CC1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880837142 GC On-Demand Anodyne Q9NAW4_PLAFA 38 45 O=C(NCc1ccc(Cl)nc1)Nc1cccc2c1OCCCO2 ZINC000880837151 EG On-Demand Anodyne NAMPT 24 47 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](N2CCCCC2)C1 ZINC000880837154 EF On-Demand Anodyne L3MBTL3 89 43 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](N2CCCCC2)C1 ZINC000880837155 EF On-Demand Anodyne L3MBTL3 89 43 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H](c3ccccn3)C3CCC3)cc2)N1 ZINC000880837169 EG On-Demand Anodyne TTK 46 46 O=C1CC[C@@H](c2ccc(C(=O)N[C@H](c3ccccn3)C3CCC3)cc2)N1 ZINC000880837170 EG On-Demand Anodyne TTK 46 46 O=C1CC[C@H](c2ccc(C(=O)N[C@H](c3ccccn3)C3CCC3)cc2)N1 ZINC000880837171 EG On-Demand Anodyne TTK 46 46 O=C1CC[C@H](c2ccc(C(=O)N[C@@H](c3ccccn3)C3CCC3)cc2)N1 ZINC000880837172 EG On-Demand Anodyne TTK 46 46 O=C(N[C@H](c1ccccn1)C1CCC1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880837182 EE On-Demand Anodyne TTK 24 40 O=C(N[C@@H](c1ccccn1)C1CCC1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880837183 EE On-Demand Anodyne TTK 24 40 O=C(N[C@@H](c1ccccn1)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880837185 FH On-Demand Anodyne TTK 24 40 O=C(N[C@H](c1ccccn1)C1CCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880837186 FH On-Demand Anodyne TTK 24 40 COc1ccc2c(c1)CC[C@H](C(=O)NN(C)c1ccccn1)C2 ZINC000880837187 DE On-Demand Reactive FAAH 19 45 O=C(Nc1cccc2c1OCCCO2)N1CCN(C2CCC2)CC1 ZINC000880837191 EF On-Demand Anodyne HRH3 24 44 O=C(Nc1cccc2c1OCCCO2)N1CCN(C2CCC2)CC1 ZINC000880837191 EF On-Demand Anodyne L3MBTL3 45 35 O=C(Nn1cccn1)c1ncsc1C1CC1 ZINC000880837205 BD On-Demand Anodyne MAP1 48 36 CN(CC1(C)COC1)C(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880837260 FE On-Demand Anodyne SLC12A5 45 34 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](c2ccccc2)C1 ZINC000880837289 EH On-Demand Anodyne RBP4 53 40 O=C(Nc1cccc2c1OCCCO2)N1CC[C@H](c2ccccc2)C1 ZINC000880837289 EH On-Demand Anodyne ADAM10 19 40 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](c2ccccc2)C1 ZINC000880837290 EH On-Demand Anodyne RBP4 53 40 O=C(Nc1cccc2c1OCCCO2)N1CC[C@@H](c2ccccc2)C1 ZINC000880837290 EH On-Demand Anodyne ADAM10 19 40 Cc1noc(C2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)n1 ZINC000880837292 FF On-Demand Anodyne SMO 43 49 Cc1noc(C2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)n1 ZINC000880837292 FF On-Demand Anodyne ETHR 61 36 COc1ccc(O)c(CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880837295 EF On-Demand Clean MTNR1A 47 39 N#CCCCOc1cccc(NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880837305 FI On-Demand Mild EPHX2 21 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837309 GF On-Demand Anodyne PGC 54 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837309 GF On-Demand Anodyne ECE1 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837309 GF On-Demand Anodyne REN 79 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837309 GF On-Demand Anodyne FPR1 48 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837310 GF On-Demand Anodyne PGC 54 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837310 GF On-Demand Anodyne ECE1 18 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837310 GF On-Demand Anodyne REN 79 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837310 GF On-Demand Anodyne FPR1 48 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837311 GF On-Demand Anodyne PGC 54 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837311 GF On-Demand Anodyne ECE1 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837311 GF On-Demand Anodyne REN 79 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837311 GF On-Demand Anodyne FPR1 48 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837312 GF On-Demand Anodyne PGC 54 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837312 GF On-Demand Anodyne ECE1 18 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837312 GF On-Demand Anodyne REN 79 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837312 GF On-Demand Anodyne FPR1 48 41 C=CC(C)(C)CC(=O)NC[C@@H]1CCN1Cc1ccc(OC)cc1 ZINC000880837322 DF On-Demand Mild PROKR1 59 32 C=CC(C)(C)CC(=O)NC[C@H]1CCN1Cc1ccc(OC)cc1 ZINC000880837323 DF On-Demand Mild PROKR1 59 32 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837351 GE On-Demand Anodyne CCR8 46 37 COC(=O)[C@@]1(OC)CCN(C(=O)C(C)(C)c2ccc(C(F)(F)F)cc2)C1 ZINC000880837356 FF On-Demand Anodyne EPHX2 25 41 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)C(=O)N1CCCC[C@@H]1C ZINC000880837370 FF On-Demand Anodyne ACE 21 40 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)C(=O)N1CCCC[C@H]1C ZINC000880837371 FF On-Demand Anodyne ACE 21 40 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880837372 FF On-Demand Anodyne ACE 21 40 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)c1cccnc1 ZINC000880837387 DG On-Demand Anodyne KCNA5 18 42 O=C(N[C@H](c1ccccn1)C1CCC1)c1cncc2[nH]ccc12 ZINC000880837392 DG On-Demand Anodyne TTK 33 43 C[C@@H](Cn1cncn1)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880837397 DD On-Demand Anodyne HIS3 77 37 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880837400 GG On-Demand Anodyne HTR4 32 40 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880837401 GG On-Demand Anodyne HTR4 32 40 O=C(Nc1cccc2c1OCCCO2)N1CCN2CCCC[C@H]2C1 ZINC000880837409 EF On-Demand Anodyne L3MBTL3 51 37 O=C(Nc1cccc2c1OCCCO2)N1CCN2CCCC[C@@H]2C1 ZINC000880837410 EF On-Demand Anodyne L3MBTL3 51 37 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880837440 EE On-Demand Anodyne MTNR1A 17 43 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cncc2[nH]ccc12 ZINC000880837478 DG On-Demand Anodyne TTK 33 43 CN(CC1(C)COC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880837481 DD On-Demand Anodyne MPO 45 34 CCCCNC(=O)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837487 GG On-Demand Anodyne MTNR1A 17 41 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CCO)CC1 ZINC000880837496 ED On-Demand Anodyne EPHX2 24 40 O=C(N[C@H](c1ccccn1)C1CCC1)c1cnc2cc[nH]c2c1 ZINC000880837515 DG On-Demand Anodyne TTK 48 47 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cnc2cc[nH]c2c1 ZINC000880837516 DG On-Demand Anodyne TTK 48 47 O=C(N[C@H](c1ccccn1)C1CCC1)c1ccc(CN2CCOCC2)o1 ZINC000880837522 FF On-Demand Anodyne TTK 20 41 O=C(N[C@@H](c1ccccn1)C1CCC1)c1ccc(CN2CCOCC2)o1 ZINC000880837523 FF On-Demand Anodyne TTK 20 41 O=C(C[C@H]1CCNC1=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837542 CD On-Demand Anodyne TTK 22 40 O=C(C[C@H]1CCNC1=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837543 CD On-Demand Anodyne TTK 22 40 O=C(C[C@@H]1CCNC1=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837544 CD On-Demand Anodyne TTK 22 40 O=C(C[C@@H]1CCNC1=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837545 CD On-Demand Anodyne TTK 22 40 Cn1ncc(Br)c1CC(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837547 FF On-Demand Anodyne TTK 22 43 Cn1ncc(Br)c1CC(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837548 FF On-Demand Anodyne TTK 22 43 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880837571 GF On-Demand Anodyne HCN1 56 37 O=C(NCC1(N2CCCC2)CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880837571 GF On-Demand Anodyne HCN4 47 30 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837577 DG On-Demand Anodyne TTK 22 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837578 DG On-Demand Anodyne TTK 22 40 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837579 DG On-Demand Anodyne TTK 22 40 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837580 DG On-Demand Anodyne TTK 22 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837602 FE On-Demand Clean PAPA1_CARPA 41 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837602 FE On-Demand Clean CTSL 20 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837602 FE On-Demand Clean CTSS 15 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837602 FE On-Demand Clean FPR1 43 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837603 FE On-Demand Clean PAPA1_CARPA 41 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837603 FE On-Demand Clean CTSL 20 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837603 FE On-Demand Clean CTSS 15 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cc(C)ccc1O ZINC000880837603 FE On-Demand Clean FPR1 43 35 O=C(NCCCc1nc2ccccc2[nH]1)Nc1cccc2c1OCCCO2 ZINC000880837622 FG On-Demand Anodyne MTNR1A 21 42 CN(CCN1CCOCC1)C(=O)Nc1cccc2c1OCCCO2 ZINC000880837623 ED On-Demand Anodyne CASR 54 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837666 FG On-Demand Anodyne TTK 20 40 O=C(Cc1ccccc1N1CCCC1=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837668 FG On-Demand Anodyne TTK 20 40 O=C(N[C@H](c1ccccn1)C1CCC1)c1coc(-c2ccccn2)n1 ZINC000880837670 EG On-Demand Anodyne TTK 25 43 O=C(N[C@@H](c1ccccn1)C1CCC1)c1coc(-c2ccccn2)n1 ZINC000880837672 EG On-Demand Anodyne TTK 25 43 Cn1nc2c(c1C(=O)N[C@H](c1ccccn1)C1CCC1)CSCC2 ZINC000880837674 EF On-Demand Anodyne TTK 25 42 Cn1nc2c(c1C(=O)N[C@@H](c1ccccn1)C1CCC1)CSCC2 ZINC000880837676 EF On-Demand Anodyne TTK 25 42 N#Cc1cccc(OC2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)c1 ZINC000880837712 GH On-Demand Mild EPHX2 15 51 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@H](N2CCCC2)C1 ZINC000880837716 FG On-Demand Anodyne L3MBTL3 57 38 O=C(Nc1cccc2c1OCCCO2)N1CCCC[C@@H](N2CCCC2)C1 ZINC000880837718 FG On-Demand Anodyne L3MBTL3 57 38 COc1ccc(N2CCC(NC(=O)Nc3cccc4c3OCCCO4)CC2)cc1 ZINC000880837722 GH On-Demand Clean MTNR1A 15 41 CC(=O)Nc1ccc(NC(=O)Nc2cccc3c2OCCCO3)cc1C ZINC000880837724 FH On-Demand Anodyne LPL 48 32 COC(=O)[C@@]1(OC)CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880837735 ED On-Demand Anodyne MTNR1A 18 44 COC(=O)[C@@]1(OC)CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880837735 ED On-Demand Anodyne MTNR1B 19 44 COC(=O)[C@@]1(OC)CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880837737 ED On-Demand Anodyne MTNR1A 18 44 COC(=O)[C@@]1(OC)CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C1 ZINC000880837737 ED On-Demand Anodyne MTNR1B 19 44 CC(=O)Nc1ccc(CCNC(=O)Nc2cccc3c2OCCCO3)cc1 ZINC000880837744 FG On-Demand Anodyne MTNR1A 21 52 O=C(N[C@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837753 DG On-Demand Anodyne JAK3 15 40 O=C(N[C@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837753 DG On-Demand Anodyne CTSS 15 40 O=C(N[C@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837753 DG On-Demand Anodyne TYK2 19 40 O=C(N[C@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837753 DG On-Demand Anodyne TTK 33 45 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837754 DG On-Demand Anodyne JAK3 15 40 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837754 DG On-Demand Anodyne CTSS 15 40 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837754 DG On-Demand Anodyne TYK2 19 40 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cccn2nccc12 ZINC000880837754 DG On-Demand Anodyne TTK 33 45 COC(=O)[C@@]1(OC)CCN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880837773 EE On-Demand Anodyne EBP 18 44 COC(=O)[C@@]1(OC)CCN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880837774 EE On-Demand Anodyne EBP 18 44 O=C(CN1CCCCS1(=O)=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837779 ED On-Demand Anodyne TTK 34 46 O=C(CN1CCCCS1(=O)=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837780 ED On-Demand Anodyne TTK 34 46 O=C(NN1CCS(=O)(=O)CC1)c1c[nH]cc1C1CC1 ZINC000880837783 CC On-Demand Anodyne HTR1F 57 33 O=C(Cc1cccc(F)c1)NCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880837801 GE On-Demand Anodyne KCNQ2 17 44 COc1cc(Br)ccc1[C@@H]1CCCN1C(=O)COC1CC1 ZINC000880837826 FG On-Demand Anodyne CPT1A 76 35 COc1cc(Br)ccc1[C@H]1CCCN1C(=O)COC1CC1 ZINC000880837828 FG On-Demand Anodyne CPT1A 76 35 O=C(N[C@H](c1ccccn1)C1CCC1)c1cnc(CC2CC2)s1 ZINC000880837831 EH On-Demand Anodyne TTK 27 40 O=C(N[C@@H](c1ccccn1)C1CCC1)c1cnc(CC2CC2)s1 ZINC000880837833 EH On-Demand Anodyne TTK 27 40 O=C(NCC1(OCCO)CCC(F)(F)CC1)c1cccn2nccc12 ZINC000880837845 FE On-Demand Anodyne HCN1 47 31 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc4c3OCCCO4)ccc21 ZINC000880837870 FF On-Demand Anodyne LPL 41 30 COC(=O)N1CCC[C@@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880837890 EE On-Demand Anodyne BIRC2 17 41 COC(=O)N1CCC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880837892 EE On-Demand Anodyne BIRC2 17 41 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne MTNR1A 51 41 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne MTNR1B 45 41 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne MMP3 48 40 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne MMP8 27 40 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne EBP 15 41 COc1ccc2c(c1)CC[C@H](C(=O)Nn1cccn1)C2 ZINC000880837908 CD On-Demand Anodyne MMP1 41 38 C=CC(C)(C)CC(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880837918 CH On-Demand Mild TTK 22 41 C=CC(C)(C)CC(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880837919 CH On-Demand Mild TTK 22 41 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880837921 GG On-Demand Anodyne GPR119 28 41 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne DRD5 15 40 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne MMP13 30 41 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne MTNR1A 25 42 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne MTNR1B 26 42 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne MMP3 41 41 COc1ccc2c(c1)CC[C@H](C(=O)NN1CCS(=O)(=O)CC1)C2 ZINC000880837943 EC On-Demand Anodyne MMP1 35 43 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)Nn3cccn3)ccn2)CC1 ZINC000880837948 FD On-Demand Anodyne GPR119 42 48 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cccc2c1OCCCO2 ZINC000880837956 GE On-Demand Anodyne MAPK10 17 49 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cccc2c1OCCCO2 ZINC000880837956 GE On-Demand Anodyne EPHX2 22 41 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)c1ccccc1 ZINC000880837973 DH On-Demand Anodyne KCNQ2 43 37 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cccc2c1OCCCO2 ZINC000880837993 GF On-Demand Anodyne ADRB2 15 44 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cccc2c1OCCCO2 ZINC000880837993 GF On-Demand Anodyne ADRB1 42 44 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cccc2c1OCCCO2 ZINC000880837994 GF On-Demand Anodyne ADRB2 15 44 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cccc2c1OCCCO2 ZINC000880837994 GF On-Demand Anodyne ADRB1 42 44 COc1ccc(OC2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)cc1 ZINC000880838024 GH On-Demand Anodyne PRSS2 65 31 COc1ccc(OC2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)cc1 ZINC000880838024 GH On-Demand Anodyne EPHX2 19 49 Cc1coc(C(=O)N[C@@H]2CCN(c3ccc4nncn4n3)C2)c1 ZINC000880838044 DD On-Demand Anodyne MAPK13 44 33 Cc1coc(C(=O)N[C@H]2CCN(c3ccc4nncn4n3)C2)c1 ZINC000880838045 DD On-Demand Anodyne MAPK13 44 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838100 CC On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838100 CC On-Demand Anodyne FPR1 46 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838100 CC On-Demand Anodyne AMP1_PLAFQ 19 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838101 CC On-Demand Anodyne PAPA1_CARPA 39 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838101 CC On-Demand Anodyne FPR1 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nn1cccn1 ZINC000880838101 CC On-Demand Anodyne AMP1_PLAFQ 19 43 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838102 GG On-Demand Anodyne HRH2 28 44 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838102 GG On-Demand Anodyne MTNR1A 31 49 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838102 GG On-Demand Anodyne MTNR1B 24 42 CC(=O)Nc1cccc(OCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838102 GG On-Demand Anodyne EPHX2 18 40 O=C(NC[C@@H](O)COc1ccc(F)c(F)c1)Nc1cccc2c1OCCCO2 ZINC000880838117 GF On-Demand Anodyne ADRB1 37 45 O=C(NC[C@H](O)COc1ccc(F)c(F)c1)Nc1cccc2c1OCCCO2 ZINC000880838118 GF On-Demand Anodyne ADRB1 37 45 N#Cc1ccccc1N1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838199 GG On-Demand Mild KCNQ2 42 32 CSc1nccnc1C(=O)N[C@@H](c1ccccn1)C1CCC1 ZINC000880838211 DF On-Demand Anodyne TTK 23 42 CSc1nccnc1C(=O)N[C@H](c1ccccn1)C1CCC1 ZINC000880838212 DF On-Demand Anodyne TTK 23 42 O=C(COC1CC1)NC[C@H]1c2ccccc2C(=O)N1Cc1ccccc1 ZINC000880838222 FF On-Demand Anodyne TSHR 43 35 O=C(COC1CC1)NC[C@@H]1c2ccccc2C(=O)N1Cc1ccccc1 ZINC000880838223 FF On-Demand Anodyne TSHR 43 35 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(C)ccc1O)C2 ZINC000880838226 EG On-Demand Clean MTNR1A 38 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cc(C)ccc1O)C2 ZINC000880838226 EG On-Demand Clean MTNR1B 31 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880838230 FD On-Demand Anodyne LPL 42 32 COCCOc1ncccc1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880838236 FF On-Demand Anodyne G2YM83_BOTF4 69 36 CC(=O)Nc1cc(NC(=O)Nc2cccc3c2OCCCO3)ccc1C ZINC000880838269 FH On-Demand Anodyne LPL 48 32 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838279 GG On-Demand Anodyne LPL 42 31 O=C(N[C@H](c1ccccn1)C1CCC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880838280 DF On-Demand Anodyne TTK 20 42 O=C(N[C@@H](c1ccccn1)C1CCC1)[C@@H]1OC[C@@H]2CCC[C@@H]21 ZINC000880838281 DF On-Demand Anodyne TTK 20 42 COc1cccc(C(=O)NCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838324 GE On-Demand Anodyne DRD4 55 42 COc1cccc(C(=O)NCCNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838324 GE On-Demand Anodyne MTNR1A 40 39 N#Cc1ccc(CN2CCN(C(=O)Nc3cccc4c3OCCCO4)CC2)cc1 ZINC000880838336 GG On-Demand Mild FAAH 15 42 O=C(Nc1cccc2c1OCCCO2)NC1CCN(c2ccccc2)CC1 ZINC000880838337 FH On-Demand Anodyne MTNR1A 15 45 O=C(Nc1cccc2c1OCCCO2)NC1CCN(c2ccccc2)CC1 ZINC000880838337 FH On-Demand Anodyne EPHX2 25 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)c1ccc(C)cn1 ZINC000880838382 GF On-Demand Anodyne PAPA1_CARPA 40 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)c1ccc(C)cn1 ZINC000880838382 GF On-Demand Anodyne FPR1 41 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)c1ccc(C)cn1 ZINC000880838384 GF On-Demand Anodyne PAPA1_CARPA 40 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)c1ccc(C)cn1 ZINC000880838384 GF On-Demand Anodyne FPR1 41 36 COc1cccc([C@@H](C)NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838391 EH On-Demand Anodyne MTNR1A 19 41 COc1cccc([C@@H](C)NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838391 EH On-Demand Anodyne MTNR1B 21 41 COc1cccc([C@H](C)NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838392 EH On-Demand Anodyne MTNR1A 19 41 COc1cccc([C@H](C)NC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838392 EH On-Demand Anodyne MTNR1B 21 41 O=C(NCCCCn1ccnc1)Nc1cccc2c1OCCCO2 ZINC000880838403 EF On-Demand Anodyne TBXAS1 39 43 O=C(NCCCCn1ccnc1)Nc1cccc2c1OCCCO2 ZINC000880838403 EF On-Demand Anodyne QPCT 51 45 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1cccc2c1OCCCO2 ZINC000880838433 EF On-Demand Anodyne TRPV1 16 41 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1cccc2c1OCCCO2 ZINC000880838434 EF On-Demand Anodyne TRPV1 16 41 O=C1C[C@]2(CCCN(C(=O)c3cnc(CC4CC4)s3)C2)Oc2ccccc21 ZINC000880838446 GH On-Demand Anodyne ACACA 55 35 O=C1C[C@@]2(CCCN(C(=O)c3cnc(CC4CC4)s3)C2)Oc2ccccc21 ZINC000880838447 GH On-Demand Anodyne ACACA 55 35 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838451 GG On-Demand Anodyne EPHX2 39 44 COCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838456 EE On-Demand Anodyne HTR4 41 45 COCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838456 EE On-Demand Anodyne CCR3 28 41 COCCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838456 EE On-Demand Anodyne EPHX2 32 42 C[C@@H](Cc1ccc(O)cc1)NC(=O)Nc1cccc2c1OCCCO2 ZINC000880838468 EG On-Demand Anodyne YARS 72 32 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1cccc2c1OCCCO2 ZINC000880838484 FF On-Demand Anodyne PANC 49 33 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1cccc2c1OCCCO2 ZINC000880838485 FF On-Demand Anodyne PANC 49 33 Cn1nc2c(c1C(=O)N1CCC[C@]3(CC(=O)c4ccccc4O3)C1)CSCC2 ZINC000880838492 GF On-Demand Anodyne ACACA 40 35 Cn1nc2c(c1C(=O)N1CCC[C@@]3(CC(=O)c4ccccc4O3)C1)CSCC2 ZINC000880838493 GF On-Demand Anodyne ACACA 40 35 COc1cccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)c1C ZINC000880838505 DG On-Demand Anodyne KCNK3 48 38 COc1cccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)c1C ZINC000880838506 DG On-Demand Anodyne KCNK3 48 38 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](N2CCCC2)C1 ZINC000880838520 EF On-Demand Anodyne L3MBTL3 58 38 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](N2CCCC2)C1 ZINC000880838521 EF On-Demand Anodyne L3MBTL3 58 38 O=C1C[C@@]2(CCCN(C(=O)c3coc(-c4ccccn4)n3)C2)Oc2ccccc21 ZINC000880838524 GG On-Demand Anodyne ACACA 36 42 O=C1C[C@]2(CCCN(C(=O)c3coc(-c4ccccn4)n3)C2)Oc2ccccc21 ZINC000880838525 GG On-Demand Anodyne ACACA 36 42 O=C(Nc1cccc2c1OCCCO2)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880838529 GG On-Demand Anodyne EPHX2 41 48 O=C(Nc1cccc2c1OCCCO2)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880838529 GG On-Demand Anodyne L3MBTL3 56 36 Cc1cnc(Cl)c(C(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880838531 FH On-Demand Anodyne ACACA 61 45 Cc1cnc(Cl)c(C(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)c1 ZINC000880838532 FH On-Demand Anodyne ACACA 61 45 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cccc2c1OCCCO2 ZINC000880838554 GG On-Demand Clean STAT6 53 35 CCCCCNC(=O)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838557 GG On-Demand Anodyne MTNR1A 16 42 C=CC(C)(C)CC(=O)Nc1cccc(OC)c1C ZINC000880838567 BH On-Demand Mild KCNK3 42 36 O=C(Nc1cccc2c1OCCCO2)N1CCC(N2CCCCC2)CC1 ZINC000880838569 FG On-Demand Anodyne L3MBTL3 110 43 C=CC(C)(C)CC(=O)Nc1ccc2c(c1)COC(=O)N2 ZINC000880838573 CG On-Demand Mild PTPRF 41 32 O=C(COC1CC1)Nc1ccc2c(c1)COC(=O)N2 ZINC000880838588 CD On-Demand Anodyne PTPRF 40 31 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cccc2c1OCCCO2 ZINC000880838595 GF On-Demand Anodyne ADRB2 29 43 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cccc2c1OCCCO2 ZINC000880838595 GF On-Demand Anodyne ADRB1 64 40 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cccc2c1OCCCO2 ZINC000880838596 GF On-Demand Anodyne ADRB2 29 43 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cccc2c1OCCCO2 ZINC000880838596 GF On-Demand Anodyne ADRB1 64 40 CC1(C)CC[C@@H](CC(=O)Nc2ccc3c(c2)COC(=O)N3)OC1 ZINC000880838607 DG On-Demand Anodyne PTPRF 42 32 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@@H](OCC(F)(F)F)C1 ZINC000880838619 FG On-Demand Anodyne RBP4 44 33 O=C(Nc1cccc2c1OCCCO2)N1CCC[C@H](OCC(F)(F)F)C1 ZINC000880838620 FG On-Demand Anodyne RBP4 44 33 CC(=O)NCC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838624 EE On-Demand Anodyne HTR4 39 41 CC(=O)NCC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838624 EE On-Demand Anodyne MTNR1A 18 45 O=C(CC[C@@H]1CCc2ccccc21)Nc1ccc2c(c1)COC(=O)N2 ZINC000880838637 EI On-Demand Anodyne PTPRF 43 33 O=C(CC[C@H]1CCc2ccccc21)Nc1ccc2c(c1)COC(=O)N2 ZINC000880838638 EI On-Demand Anodyne PTPRF 43 33 O=C(Nc1cccc2c1OCCCO2)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880838642 GG On-Demand Anodyne DGAT1 23 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](CO)CCC(C)C)C2 ZINC000880838645 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](CO)CCC(C)C)C2 ZINC000880838645 DF On-Demand Anodyne MTNR1A 42 39 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H](CO)CCC(C)C)C2 ZINC000880838645 DF On-Demand Anodyne MTNR1B 40 39 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](CO)CCC(C)C)C2 ZINC000880838647 DF On-Demand Anodyne NQO2 27 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](CO)CCC(C)C)C2 ZINC000880838647 DF On-Demand Anodyne MTNR1A 42 39 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H](CO)CCC(C)C)C2 ZINC000880838647 DF On-Demand Anodyne MTNR1B 40 39 C[C@H](NC(=O)Nc1cccc2c1OCCCO2)c1ccc(N2CCOCC2)cc1 ZINC000880838653 GH On-Demand Clean KCNQ2 37 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1ccc3c(c1)COC(=O)N3)C2 ZINC000880838655 FH On-Demand Anodyne ROCK2 25 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838672 FF On-Demand Anodyne PAPA1_CARPA 39 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838672 FF On-Demand Anodyne CTSL 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838672 FF On-Demand Anodyne FPR1 46 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838673 FF On-Demand Anodyne PAPA1_CARPA 39 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838673 FF On-Demand Anodyne CTSL 18 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(OC)c1C ZINC000880838673 FF On-Demand Anodyne FPR1 46 36 Cc1cc(NC(=O)NC[C@H]2CCCN2C)cc(S(C)(=O)=O)c1 ZINC000880838728 ED On-Demand Anodyne CCR3 30 40 Cc1cc(NC(=O)NC[C@@H]2CCCN2C)cc(S(C)(=O)=O)c1 ZINC000880838729 ED On-Demand Anodyne CCR3 30 40 Cc1cc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)cc(S(C)(=O)=O)c1 ZINC000880838736 FD On-Demand Anodyne CXCR3 18 41 Cc1cc(NC(=O)NCCCCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880838744 DG On-Demand Anodyne CCR3 34 46 CC(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880838793 EE On-Demand Anodyne EPHX2 28 43 Cc1nc(C(C)C)ncc1C(=O)N1CCC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880838799 GH On-Demand Anodyne ACACA 57 42 Cc1nc(C(C)C)ncc1C(=O)N1CCC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880838800 GH On-Demand Anodyne ACACA 57 42 CCS(=O)(=O)NC1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880838801 GD On-Demand Anodyne CCR8 91 43 CC(=O)Nc1cccc(CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880838819 FG On-Demand Anodyne ROCK2 18 45 O=C(Nc1cccc2c1OCCCO2)N1CCN(Cc2cscn2)CC1 ZINC000880838831 FF On-Demand Anodyne SCN5A 40 33 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne DRD4 20 46 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne SIGMAR1 21 53 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne SSTR5 40 33 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne EPHX2 21 40 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne CXCR3 19 41 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccncc2)CC1 ZINC000880838858 GG On-Demand Anodyne MCHR1 39 41 CCN1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880838865 DE On-Demand Anodyne HTR4 45 42 CCN1CC[C@H](CNC(=O)Nc2cccc3c2OCCCO3)C1 ZINC000880838865 DE On-Demand Anodyne CCR3 41 33 O=C1C[C@]2(CCCN(C(=O)c3cncc4[nH]ccc34)C2)Oc2ccccc21 ZINC000880838869 FG On-Demand Anodyne ACACA 43 39 O=C1C[C@@]2(CCCN(C(=O)c3cncc4[nH]ccc34)C2)Oc2ccccc21 ZINC000880838870 FG On-Demand Anodyne ACACA 43 39 O=C(Nc1cccc2c1OCCCO2)NC1CCN(Cc2ccccn2)CC1 ZINC000880838873 GG On-Demand Anodyne MCHR1 21 41 O=C1C[C@]2(CCCN(C(=O)c3csc(-c4ncc[nH]4)n3)C2)Oc2ccccc21 ZINC000880838880 GG On-Demand Anodyne ACACA 40 36 O=C1C[C@@]2(CCCN(C(=O)c3csc(-c4ncc[nH]4)n3)C2)Oc2ccccc21 ZINC000880838881 GG On-Demand Anodyne ACACA 40 36 NC(=O)[C@@H]1C[C@@H](NC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880838903 DC On-Demand Anodyne KCNQ2 44 39 CC(=O)N(C)c1ccc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880838919 GF On-Demand Anodyne PRMT3 18 44 O=C(NC[C@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838998 FE On-Demand Anodyne ADRB2 35 45 O=C(NC[C@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838998 FE On-Demand Anodyne ADRB1 66 46 O=C(NC[C@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838998 FE On-Demand Anodyne ADRB3 36 43 O=C(NC[C@@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838999 FE On-Demand Anodyne ADRB2 35 45 O=C(NC[C@@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838999 FE On-Demand Anodyne ADRB1 66 46 O=C(NC[C@@H](O)COc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880838999 FE On-Demand Anodyne ADRB3 36 43 Cn1nnc(C(=O)N2CCC[C@]3(CC(=O)c4ccccc4O3)C2)n1 ZINC000880839011 EC On-Demand Anodyne ACACA 60 38 Cn1nnc(C(=O)N2CCC[C@@]3(CC(=O)c4ccccc4O3)C2)n1 ZINC000880839012 EC On-Demand Anodyne ACACA 60 38 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CC2CC2)CC1 ZINC000880839034 EF On-Demand Anodyne SIGMAR1 16 45 O=C(Nc1cccc2c1OCCCO2)NC1CCN(CC2CC2)CC1 ZINC000880839034 EF On-Demand Anodyne CXCR3 15 42 C[C@@H]1C[C@@H]1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839047 CF On-Demand Anodyne MTNR1A 16 42 C[C@@H]1C[C@H]1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839048 CF On-Demand Anodyne MTNR1A 16 42 C[C@H]1C[C@H]1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839049 CF On-Demand Anodyne MTNR1A 16 42 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cccc2c1OCCCO2 ZINC000880839066 FG On-Demand Anodyne BMP1 56 35 O=C1CC[C@@H](c2ccc(C(=O)Nc3cnn(CCF)c3)cc2)N1 ZINC000880839072 DE On-Demand Anodyne PANC 60 40 O=C1CC[C@H](c2ccc(C(=O)Nc3cnn(CCF)c3)cc2)N1 ZINC000880839073 DE On-Demand Anodyne PANC 60 40 CN1CCN(c2ncccc2CNC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880839087 GE On-Demand Anodyne G2YM83_BOTF4 52 34 CC[C@@H]1CCC[C@@]1(C)C(=O)Nc1cnn(CCF)c1 ZINC000880839115 CG On-Demand Anodyne PANC 49 33 CC[C@H]1CCC[C@]1(C)C(=O)Nc1cnn(CCF)c1 ZINC000880839117 CG On-Demand Anodyne PANC 49 33 CC[C@H]1CCC[C@@]1(C)C(=O)Nc1cnn(CCF)c1 ZINC000880839121 CG On-Demand Anodyne PANC 49 33 Cc1cc(NC(=O)NCc2ccc(C)nc2Cl)cc(S(C)(=O)=O)c1 ZINC000880839126 FG On-Demand Anodyne NAMPT 22 40 CCOC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880839131 FF On-Demand Anodyne EPHX2 44 43 CCOC(=O)N1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880839131 FF On-Demand Anodyne CCR8 59 44 CCn1ncc(C(=O)N2CCC[C@@](O)(c3ccccc3)C2)c1C1CC1 ZINC000880839133 EF On-Demand Anodyne CCR5 18 44 CCn1ncc(C(=O)N2CCC[C@](O)(c3ccccc3)C2)c1C1CC1 ZINC000880839134 EF On-Demand Anodyne CCR5 18 44 CC(C)(C(=O)Nc1cnn(CCF)c1)c1ccc(C(F)(F)F)cc1 ZINC000880839135 EH On-Demand Anodyne PANC 40 31 Cc1nc(C(C)C)ncc1C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839142 DE On-Demand Anodyne CACNA1I 52 33 Cc1nc(C(C)C)ncc1C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839143 DE On-Demand Anodyne CACNA1I 52 33 CSc1nccnc1C(=O)Nc1cnn(CCF)c1 ZINC000880839149 CD On-Demand Anodyne PANC 46 34 O=C(Nc1cccc2c1OCCCO2)N[C@H]1CCOc2ccccc21 ZINC000880839153 EG On-Demand Anodyne TRPV1 16 51 O=C(Nc1cccc2c1OCCCO2)N[C@@H]1CCOc2ccccc21 ZINC000880839154 EG On-Demand Anodyne TRPV1 16 51 O=C(Nc1cnn(CCF)c1)c1ncsc1C1CC1 ZINC000880839159 CE On-Demand Anodyne PANC 56 37 CN1CCCC[C@H](CNC(=O)c2cc3c(cc2[N+](=O)[O-])OCCCO3)C1 ZINC000880839182 FE On-Demand Bother CACNA1I 44 31 O=C(Nc1cnn(CCF)c1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880839187 DF On-Demand Anodyne PANC 50 33 O=C(NCCCN1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880839188 ED On-Demand Anodyne CCR3 25 42 O=C(NCCCN1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880839188 ED On-Demand Anodyne EPHX2 23 42 Cc1cc(NC(=O)NC[C@@H](O)[C@@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839203 GF On-Demand Anodyne LPL 43 34 Cc1cc(NC(=O)NC[C@H](O)[C@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839204 GF On-Demand Anodyne LPL 43 34 Cc1cc(NC(=O)NC[C@H](O)[C@@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839205 GF On-Demand Anodyne LPL 43 34 Cc1cc(NC(=O)NC[C@@H](O)[C@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839206 GF On-Demand Anodyne LPL 43 34 CCC(CC)C(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880839207 GF On-Demand Anodyne S1PR2 26 42 Cc1cc(NC(=O)N[C@H](C)CC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880839225 DG On-Demand Anodyne CCR3 46 37 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880839262 GG On-Demand Anodyne ACACA 41 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880839263 GG On-Demand Anodyne ACACA 41 36 Cc1cc(NC(=O)N[C@H]2Cc3ccc(C#N)cc3C2)cc(S(C)(=O)=O)c1 ZINC000880839277 FF On-Demand Mild MTTP 23 40 COc1ccccc1[C@H](C)NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880839293 FG On-Demand Anodyne CA1 18 40 COc1ccccc1[C@H](C)NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880839293 FG On-Demand Anodyne KCNK3 37 40 COc1ccccc1[C@H](C)NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880839293 FG On-Demand Anodyne KCNK9 33 40 Cc1cc(NC(=O)NCCC[C@H]2C=CCC2)cc(S(C)(=O)=O)c1 ZINC000880839303 EG On-Demand Anodyne CCR3 20 41 Cc1cc(NC(=O)NCCC[C@@H]2C=CCC2)cc(S(C)(=O)=O)c1 ZINC000880839305 EG On-Demand Anodyne CCR3 20 41 Cc1cc(NC(=O)NCCC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880839306 DF On-Demand Anodyne CCR3 29 43 Cc1cc(NC(=O)NCCC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880839306 DF On-Demand Anodyne PRMT3 18 43 Cc1cc(-c2nc(C)c(C(=O)N[C@@H]3C[C@@H](C(N)=O)C3)s2)ccc1F ZINC000880839328 EF On-Demand Anodyne MAPK13 42 30 Cc1coc(C(=O)N[C@H](CCc2ccccc2)C(F)F)c1 ZINC000880839342 CH On-Demand Anodyne ANPEP 40 35 Cc1coc(C(=O)N[C@H](CCc2ccccc2)C(F)F)c1 ZINC000880839342 CH On-Demand Anodyne LAP3 43 35 Cc1coc(C(=O)N[C@@H](CCc2ccccc2)C(F)F)c1 ZINC000880839343 CH On-Demand Anodyne ANPEP 40 35 Cc1coc(C(=O)N[C@@H](CCc2ccccc2)C(F)F)c1 ZINC000880839343 CH On-Demand Anodyne LAP3 43 35 CN1CCCC[C@H](CNC(=O)Cc2ccccc2N2CCCC2=O)C1 ZINC000880839355 EE On-Demand Anodyne CACNA1I 41 36 CN1CCCC[C@H](CNC(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880839372 GG On-Demand Anodyne CACNA1I 62 37 O=C(Nc1cccc2c1OCCCO2)N1CCC(c2nc3ccccc3[nH]2)CC1 ZINC000880839378 GI On-Demand Anodyne SMO 41 45 O=C(NCCOc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880839403 EG On-Demand Anodyne ADRB1 21 41 O=C(NCCOc1ccccc1)Nc1cccc2c1OCCCO2 ZINC000880839403 EG On-Demand Anodyne HRH2 24 41 Cc1cc(NC(=O)NC[C@@H](O)Cc2cccc(Cl)c2)cc(S(C)(=O)=O)c1 ZINC000880839441 GF On-Demand Anodyne CTSV 27 40 Cc1cc(NC(=O)NC[C@H](O)Cc2cccc(Cl)c2)cc(S(C)(=O)=O)c1 ZINC000880839442 GF On-Demand Anodyne CTSV 27 40 Cc1cc(NC(=O)Nc2cnn(C)c2C2CC2)cc(S(C)(=O)=O)c1 ZINC000880839450 EF On-Demand Anodyne LPL 41 32 CN1CCCC[C@H](CNC(=O)c2cccc3nsnc23)C1 ZINC000880839540 DE On-Demand Anodyne HTR4 54 38 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCCN(C)C2)c1 ZINC000880839544 CF On-Demand Anodyne HTR4 27 40 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCCN(C)C2)c1 ZINC000880839544 CF On-Demand Anodyne CCR3 15 41 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCCCN(C)C2)c1 ZINC000880839544 CF On-Demand Anodyne CACNA1I 72 41 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCCN(C)C2)c1 ZINC000880839545 CF On-Demand Anodyne HTR4 27 40 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCCN(C)C2)c1 ZINC000880839545 CF On-Demand Anodyne CCR3 15 41 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCCCN(C)C2)c1 ZINC000880839545 CF On-Demand Anodyne CACNA1I 72 41 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne BMP1 76 46 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP13 29 44 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP3 21 40 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP8 19 40 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne ROCK2 16 46 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP9 30 40 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP12 23 40 COc1ccc(CN(CCO)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880839546 GE On-Demand Anodyne MMP1 31 44 O=C(Nc1cccc2c1OCCCO2)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880839557 GF On-Demand Anodyne EPHX2 28 41 NC(=O)[C@@H]1CC[C@H](C(=O)Nc2cnn(CCF)c2)N1Cc1ccccc1 ZINC000880839558 FD On-Demand Anodyne ITK 15 42 NC(=O)[C@@H]1CC[C@H](C(=O)Nc2cnn(CCF)c2)N1Cc1ccccc1 ZINC000880839558 FD On-Demand Anodyne PANC 54 40 CN1CCCC[C@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880839571 DF On-Demand Anodyne HTR4 38 41 CN1CCCC[C@H](CNC(=O)c2ncccc2-c2ccccn2)C1 ZINC000880839571 DF On-Demand Anodyne HCRTR1 20 41 CN1CCCC[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880839573 ED On-Demand Anodyne HTR4 45 41 CN1CCCC[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880839573 ED On-Demand Anodyne CCR3 15 40 CN1CCCC[C@H](CNC(=O)c2ccc(CN3CCOCC3)o2)C1 ZINC000880839573 ED On-Demand Anodyne CACNA1I 63 40 CN1CCCC[C@H](CNC(=O)c2nnn(C)n2)C1 ZINC000880839574 CB On-Demand Anodyne CACNA1I 65 34 O=C(Nc1cnn(CCF)c1)c1ccc(CN2CCOCC2)o1 ZINC000880839580 DD On-Demand Anodyne PANC 51 35 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cnn(CCF)c1)C2 ZINC000880839602 DF On-Demand Anodyne MTNR1A 45 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cnn(CCF)c1)C2 ZINC000880839602 DF On-Demand Anodyne MTNR1B 40 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cnn(CCF)c1)C2 ZINC000880839602 DF On-Demand Anodyne PANC 51 34 O=C(Nc1cccc2c1OCCCO2)N1CCN(C2CCCC2)CC1 ZINC000880839606 EF On-Demand Anodyne HRH3 23 45 O=C(Nc1cccc2c1OCCCO2)N1CCN(C2CCCC2)CC1 ZINC000880839606 EF On-Demand Anodyne L3MBTL3 41 34 CN1CCCC[C@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880839608 CE On-Demand Anodyne CCR3 15 44 CN1CCCC[C@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880839608 CE On-Demand Anodyne CXCR3 20 41 CN1CCCC[C@H](CNC(=O)c2cnc3cc[nH]c3c2)C1 ZINC000880839608 CE On-Demand Anodyne CACNA1I 73 37 O=C(Cc1ccccc1N1CCCC1=O)Nc1cnn(CCF)c1 ZINC000880839620 EE On-Demand Anodyne PANC 43 34 CC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880839638 EE On-Demand Anodyne EPHX2 22 41 CC(=O)[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880839639 EE On-Demand Anodyne EPHX2 22 41 Cc1cc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839643 GF On-Demand Anodyne ACHE 15 40 Cc1cc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839643 GF On-Demand Anodyne LPL 44 35 Cc1cc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839643 GF On-Demand Anodyne SIGMAR1 17 42 Cc1cc(NC(=O)NC[C@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839643 GF On-Demand Anodyne CCR3 49 42 Cc1cc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839644 GF On-Demand Anodyne ACHE 15 40 Cc1cc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839644 GF On-Demand Anodyne LPL 44 35 Cc1cc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839644 GF On-Demand Anodyne SIGMAR1 17 42 Cc1cc(NC(=O)NC[C@@H]2CCN2Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880839644 GF On-Demand Anodyne CCR3 49 42 NC(=O)c1cn(C2CCN(C(=O)c3cc4ccccc4cc3F)CC2)nn1 ZINC000880839646 FE On-Demand Anodyne L3MBTL3 48 38 Cc1cc(NC(=O)NCCN2CC[C@@H](O)C2)cc(S(C)(=O)=O)c1 ZINC000880839670 EC On-Demand Anodyne CCR3 44 47 Cc1cc(NC(=O)NCCN2CC[C@H](O)C2)cc(S(C)(=O)=O)c1 ZINC000880839671 EC On-Demand Anodyne CCR3 44 47 Cc1cc(NC(=O)NCCC2CCN(C(C)C)CC2)cc(S(C)(=O)=O)c1 ZINC000880839703 GG On-Demand Anodyne CCR3 35 43 O=C(c1cc(C(F)(F)F)ccn1)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880839741 FG On-Demand Anodyne MAP3K12 20 40 O=C(c1cc(C(F)(F)F)ccn1)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880839742 FG On-Demand Anodyne MAP3K12 20 40 Cc1coc(C(=O)Nc2cnn(CCF)c2)c1 ZINC000880839747 BE On-Demand Anodyne PANC 50 33 O=C(CC[C@@H]1CCc2ccccc21)Nc1cnn(CCF)c1 ZINC000880839754 DG On-Demand Anodyne PANC 41 32 O=C(CC[C@H]1CCc2ccccc21)Nc1cnn(CCF)c1 ZINC000880839755 DG On-Demand Anodyne PANC 41 32 CC(C)(C(=O)Nc1cnn(CCF)c1)c1ccc(F)cc1F ZINC000880839764 DG On-Demand Anodyne PANC 51 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839769 FD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839769 FD On-Demand Anodyne CACNA1B 17 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839769 FD On-Demand Anodyne REN 46 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839770 FD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839770 FD On-Demand Anodyne CACNA1B 17 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839770 FD On-Demand Anodyne REN 46 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839771 FD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839771 FD On-Demand Anodyne CACNA1B 17 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839771 FD On-Demand Anodyne REN 46 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839772 FD On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839772 FD On-Demand Anodyne CACNA1B 17 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839772 FD On-Demand Anodyne REN 46 39 CN1CCCC[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880839774 DG On-Demand Anodyne MTNR1A 19 44 CN1CCCC[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880839774 DG On-Demand Anodyne MTNR1B 22 44 CN1CCCC[C@H](CNC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880839774 DG On-Demand Anodyne EBP 16 44 CN1CCCC[C@H](CNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880839776 DG On-Demand Anodyne MTNR1A 19 44 CN1CCCC[C@H](CNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880839776 DG On-Demand Anodyne MTNR1B 22 44 CN1CCCC[C@H](CNC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880839776 DG On-Demand Anodyne EBP 16 44 CN1CCCC[C@H](CNC(=O)c2cnc(CC3CC3)s2)C1 ZINC000880839778 DF On-Demand Anodyne CACNA1I 57 35 COCCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839791 CE On-Demand Anodyne HRH2 22 40 CCOC(=O)C1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880839802 EF On-Demand Anodyne CCR8 22 42 C#CCC1(O)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880839809 FD On-Demand Mild S1PR2 29 46 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne DRD2 21 46 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne CNR1 15 45 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne DRD4 19 46 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne SLC6A1 46 33 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne HTR4 56 40 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne CNR2 18 40 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne CCR3 48 41 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne CACNA1I 70 36 CN1CCCC[C@H](CNC(=O)c2cc3ccccc3cc2F)C1 ZINC000880839818 DG On-Demand Anodyne POLR1A 70 37 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880839822 GE On-Demand Anodyne MTOR 38 41 O=C(NCc1cccnc1N1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880839822 GE On-Demand Anodyne SCN10A 20 45 CCn1ncc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1C ZINC000880839834 EF On-Demand Anodyne LPL 47 31 C=CC[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880839843 DF On-Demand Mild F13A1 42 35 C=CC[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880839844 DF On-Demand Mild F13A1 42 35 NC(=O)[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880839848 DD On-Demand Anodyne PDE4D 18 44 NC(=O)[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880839848 DD On-Demand Anodyne EZH2 42 40 COC[C@@H]1CCCN1NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880839860 ED On-Demand Anodyne CASP7 54 38 Cc1cc(NC(=O)Nc2cnn3c2CCCC3)cc(S(C)(=O)=O)c1 ZINC000880839881 EF On-Demand Anodyne LPL 45 36 COc1cccc([C@H](CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)OC)c1 ZINC000880839903 GF On-Demand Anodyne MTNR1B 25 40 NC(=O)[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880839913 CC On-Demand Anodyne JAK3 18 44 NC(=O)[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880839913 CC On-Demand Anodyne JAK1 15 44 NC(=O)[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880839913 CC On-Demand Anodyne TYK2 22 44 NC(=O)[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880839913 CC On-Demand Anodyne EPHB3 37 41 CCC1(N2CCCC2)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880839918 GG On-Demand Anodyne S1PR2 26 42 C=CC(C)(C)CC(=O)NC[C@H]1CCCCN(C)C1 ZINC000880839921 CE On-Demand Mild CACNA1I 42 33 C=CC(C)(C)CC(=O)NC[C@@H]1CCCCN(C)C1 ZINC000880839922 CE On-Demand Mild CACNA1I 42 33 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](C(N)=O)C1)C2 ZINC000880839932 DD On-Demand Anodyne NQO2 23 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](C(N)=O)C1)C2 ZINC000880839932 DD On-Demand Anodyne MTNR1A 33 42 COc1ccc(CN(C)C(=O)Nc2cccc3c2OCCCO3)cc1OC ZINC000880839937 FH On-Demand Anodyne MT-ND1 17 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnn(CCF)c1 ZINC000880839953 ED On-Demand Anodyne PANC 47 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cnn(CCF)c1 ZINC000880839954 ED On-Demand Anodyne PANC 47 33 CCCCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839966 CG On-Demand Anodyne MTNR1A 23 51 CC(=O)NCCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880839984 DD On-Demand Anodyne MTNR1A 48 61 Cn1nnc(C(=O)N[C@@H](CCc2ccccc2)C(F)F)n1 ZINC000880839985 CD On-Demand Anodyne BLA1_STEMA 40 31 Cn1nnc(C(=O)N[C@H](CCc2ccccc2)C(F)F)n1 ZINC000880839986 CD On-Demand Anodyne BLA1_STEMA 40 31 O=C(NCCN1CCOCC1)Nc1cccc2c1OCCCO2 ZINC000880839987 DD On-Demand Anodyne EPHX2 22 46 CN1CCCC[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880839996 EE On-Demand Anodyne GABRA1 17 47 CN1CCCC[C@H](CNC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880839996 EE On-Demand Anodyne HTR1F 40 37 CN(CCOc1ccccc1)C(=O)Nc1cccc2c1OCCCO2 ZINC000880839998 EG On-Demand Anodyne LTA4H 17 40 Cc1coc(C(=O)NC[C@H]2CCCCN(C)C2)c1 ZINC000880840010 CE On-Demand Anodyne CACNA1I 73 40 Cc1coc(C(=O)NC[C@@H]2CCCCN(C)C2)c1 ZINC000880840011 CE On-Demand Anodyne CACNA1I 73 40 CN1CCCC[C@H](CNC(=O)c2ncsc2C2CC2)C1 ZINC000880840026 CE On-Demand Anodyne CACNA1I 52 32 O=C(COC1CC1)Nc1cnn(CCF)c1 ZINC000880840032 BC On-Demand Anodyne PANC 45 32 CCN1CCC(NC(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880840034 DE On-Demand Anodyne MTNR1A 15 42 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne BMP1 71 41 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne MMP13 36 42 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne ROCK2 15 42 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne MMP9 40 39 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne CA9 19 40 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880840047 FG On-Demand Anodyne MMP1 39 42 CN1CCCC[C@H](CNC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)C1 ZINC000880840082 EE On-Demand Anodyne CACNA1I 71 35 CN1CCCC[C@H](CNC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)C1 ZINC000880840084 EE On-Demand Anodyne CACNA1I 71 35 O=C(NCCc1cccnc1)Nc1cccc2c1OCCCO2 ZINC000880840095 DF On-Demand Anodyne NAMPT 40 47 CC(C)(C)OC(=O)CC[C@@H]1C[C@H](C(=O)Nc2cnn(CCF)c2)CO1 ZINC000880840097 FE On-Demand Anodyne PANC 50 33 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)Nc2cnn(CCF)c2)CO1 ZINC000880840098 FE On-Demand Anodyne PANC 50 33 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)Nc2cnn(CCF)c2)CO1 ZINC000880840099 FE On-Demand Anodyne PANC 50 33 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)Nc2cnn(CCF)c2)CO1 ZINC000880840100 FE On-Demand Anodyne PANC 50 33 Cc1cc(NC(=O)N[C@H]2C(=O)N(C)Cc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880840129 GE On-Demand Anodyne CCKBR 44 38 CN1CCCC[C@H](CNC(=O)c2cncc3[nH]ccc23)C1 ZINC000880840149 CE On-Demand Anodyne HTR4 49 40 O=C(Nc1cccc2c1OCCCO2)N1CCN(Cc2cccnc2)CC1 ZINC000880840153 FF On-Demand Anodyne FAAH 25 46 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCCN(C)C1)C2 ZINC000880840160 EF On-Demand Anodyne DRD4 43 34 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCCN(C)C1)C2 ZINC000880840160 EF On-Demand Anodyne DRD5 16 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCCN(C)C1)C2 ZINC000880840160 EF On-Demand Anodyne MTNR1A 44 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCCCN(C)C1)C2 ZINC000880840160 EF On-Demand Anodyne MTNR1B 44 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCCN(C)C1)C2 ZINC000880840161 EF On-Demand Anodyne DRD4 43 34 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCCN(C)C1)C2 ZINC000880840161 EF On-Demand Anodyne DRD5 16 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCCN(C)C1)C2 ZINC000880840161 EF On-Demand Anodyne MTNR1A 44 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCCN(C)C1)C2 ZINC000880840161 EF On-Demand Anodyne MTNR1B 44 43 O=C(NCCn1ccnc1)Nc1cccc2c1OCCCO2 ZINC000880840162 DD On-Demand Anodyne QPCT 34 40 O=C(Nc1cccc2c1OCCCO2)N1CCN(Cc2ccncc2)CC1 ZINC000880840165 FF On-Demand Anodyne FAAH 25 45 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne HTR1A 40 41 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne DRD2 52 42 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne DRD4 29 42 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne DRD3 57 40 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne HTR4 53 40 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne HCN1 52 37 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCCN(C)C2)c(O)n1 ZINC000880840174 FF On-Demand Anodyne HCN4 40 34 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne HTR1A 40 41 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne DRD2 52 42 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne DRD4 29 42 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne DRD3 57 40 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne HTR4 53 40 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne HCN1 52 37 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCCN(C)C2)c(O)n1 ZINC000880840176 FF On-Demand Anodyne HCN4 40 34 O=C1C[C@]2(CCCN(C(=O)c3cnc4cc[nH]c4c3)C2)Oc2ccccc21 ZINC000880840186 FG On-Demand Anodyne ACACA 75 47 O=C1C[C@]2(CCCN(C(=O)c3cnc4cc[nH]c4c3)C2)Oc2ccccc21 ZINC000880840186 FG On-Demand Anodyne ACACB 49 47 CC(C)(C)OC(=O)NC1(CNC(=O)c2cccn3nccc23)CCOCC1 ZINC000880840188 FE On-Demand Anodyne HCN1 60 36 CC(C)(C)OC(=O)NC1(CNC(=O)c2cccn3nccc23)CCOCC1 ZINC000880840188 FE On-Demand Anodyne HCN4 46 29 O=C1C[C@@]2(CCCN(C(=O)c3cnc4cc[nH]c4c3)C2)Oc2ccccc21 ZINC000880840189 FG On-Demand Anodyne ACACA 75 47 O=C1C[C@@]2(CCCN(C(=O)c3cnc4cc[nH]c4c3)C2)Oc2ccccc21 ZINC000880840189 FG On-Demand Anodyne ACACB 49 47 Cn1nc2c(c1C(=O)Nc1cnn(CCF)c1)CSCC2 ZINC000880840192 DD On-Demand Anodyne PANC 40 31 CN1CCCC[C@H](CNC(=O)CC(C)(C)CC(F)(F)F)C1 ZINC000880840210 DG On-Demand Anodyne CACNA1I 47 33 Cc1cc(NC(=O)NC[C@@H]2CCO[C@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880840211 GG On-Demand Anodyne LPL 51 36 O=C(Nc1cccc2c1OCCCO2)NC1CCN(C(=O)C2CC2)CC1 ZINC000880840215 FE On-Demand Anodyne EPHX2 42 48 COC[C@@H]1CCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840255 EE On-Demand Anodyne CASP3 40 38 COC[C@@H]1CCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840255 EE On-Demand Anodyne CASP7 54 38 Cc1cc(NC(=O)NCC2CCN(CC3CC3)CC2)cc(S(C)(=O)=O)c1 ZINC000880840262 GF On-Demand Anodyne CCR3 44 44 Cc1cc(NC(=O)NCC2CCN(CC3CC3)CC2)cc(S(C)(=O)=O)c1 ZINC000880840262 GF On-Demand Anodyne CACNA1I 61 37 Cc1cc(NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)cc(S(C)(=O)=O)c1 ZINC000880840280 GF On-Demand Anodyne CCR3 78 43 Cc1cc(NC(=O)NC[C@H]2CCCN(CC3CC3)C2)cc(S(C)(=O)=O)c1 ZINC000880840281 GF On-Demand Anodyne CCR3 78 43 CCC1(N(C)C)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880840291 FF On-Demand Anodyne S1PR2 27 43 O=C1C[C@]2(CCCN(C(=O)c3ncccc3-c3ccccn3)C2)Oc2ccccc21 ZINC000880840319 GH On-Demand Anodyne ACACA 39 43 O=C1C[C@]2(CCCN(C(=O)c3ncccc3-c3ccccn3)C2)Oc2ccccc21 ZINC000880840319 GH On-Demand Anodyne ACACB 21 43 O=C1C[C@@]2(CCCN(C(=O)c3ncccc3-c3ccccn3)C2)Oc2ccccc21 ZINC000880840320 GH On-Demand Anodyne ACACA 39 43 O=C1C[C@@]2(CCCN(C(=O)c3ncccc3-c3ccccn3)C2)Oc2ccccc21 ZINC000880840320 GH On-Demand Anodyne ACACB 21 43 CN1CCCC[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880840329 EG On-Demand Anodyne CCR3 15 40 CN1CCCC[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880840329 EG On-Demand Anodyne PDE4D 24 47 CN1CCCC[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880840329 EG On-Demand Anodyne UTS2R 23 42 CN1CCCC[C@H](CNC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880840329 EG On-Demand Anodyne CACNA1I 91 48 O=C(Nc1cnn(CCF)c1)c1cc(Br)ccc1C1CC1 ZINC000880840342 FH On-Demand Anodyne PANC 46 33 O=C(NCCCn1ccnc1)Nc1cccc2c1OCCCO2 ZINC000880840354 DE On-Demand Anodyne TBXAS1 39 44 O=C(NCCCn1ccnc1)Nc1cccc2c1OCCCO2 ZINC000880840354 DE On-Demand Anodyne QPCT 54 48 CN(C)C(=O)c1cccc(CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880840357 FF On-Demand Anodyne ROCK2 19 40 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840365 EE On-Demand Anodyne HPGD 43 40 O=C(c1ccc2c(O)ncnc2c1)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840366 EE On-Demand Anodyne HPGD 43 40 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc3c1OCCCO3)CC2 ZINC000880840377 GG On-Demand Anodyne ABCB1B 54 38 COc1cc2c(cc1OC)CN(C(=O)Nc1cccc3c1OCCCO3)CC2 ZINC000880840377 GG On-Demand Anodyne ABCB1 18 41 CN1CCCC[C@H](CNC(=O)[C@@]2(c3ccccc3)C[C@H](F)C2)C1 ZINC000880840404 DF On-Demand Anodyne CACNA1I 22 45 CC(C)(C)OC(=O)N1C[C@H](C(=O)Nc2cnn(CCF)c2)C(C)(C)C1 ZINC000880840405 FF On-Demand Anodyne PANC 51 34 CC(C)(C)OC(=O)N1C[C@@H](C(=O)Nc2cnn(CCF)c2)C(C)(C)C1 ZINC000880840406 FF On-Demand Anodyne PANC 51 34 CN1CCCC[C@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)C1 ZINC000880840415 GH On-Demand Anodyne DRD4 44 34 CN1CCCC[C@H](CNC(=O)c2cccc(N(C)C(=O)OC(C)(C)C)c2)C1 ZINC000880840415 GH On-Demand Anodyne CACNA1I 79 47 CN1CCCC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880840426 FD On-Demand Anodyne F2 55 41 CN1CCCC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880840426 FD On-Demand Anodyne SIGMAR1 18 41 CN1CCCC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880840426 FD On-Demand Anodyne TRY1_BOVIN 51 33 CN1CCCC[C@H](CNC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880840426 FD On-Demand Anodyne TMPRSS11D 61 35 CN1CCCC[C@H](CNC(=O)CC(C)(C)CC(F)F)C1 ZINC000880840429 CF On-Demand Anodyne CACNA1I 45 32 O=C(NCc1cccnc1)Nc1cccc2c1OCCCO2 ZINC000880840436 CF On-Demand Anodyne NAMPT 69 48 O=C(Nc1cnn(CCF)c1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880840438 GF On-Demand Anodyne Q9NAW4_PLAFA 27 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840442 GE On-Demand Anodyne GHRHR 52 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840442 GE On-Demand Anodyne P2RY12 90 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840442 GE On-Demand Anodyne PGC 46 31 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840442 GE On-Demand Anodyne CCR1 17 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840442 GE On-Demand Anodyne FPR1 46 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840443 GE On-Demand Anodyne GHRHR 52 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840443 GE On-Demand Anodyne P2RY12 90 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840443 GE On-Demand Anodyne PGC 46 31 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840443 GE On-Demand Anodyne CCR1 17 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880840443 GE On-Demand Anodyne FPR1 46 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840444 GE On-Demand Anodyne GHRHR 52 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840444 GE On-Demand Anodyne P2RY12 90 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840444 GE On-Demand Anodyne PGC 46 31 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840444 GE On-Demand Anodyne CCR1 17 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840444 GE On-Demand Anodyne FPR1 46 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840445 GE On-Demand Anodyne GHRHR 52 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840445 GE On-Demand Anodyne P2RY12 90 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840445 GE On-Demand Anodyne PGC 46 31 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840445 GE On-Demand Anodyne CCR1 17 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880840445 GE On-Demand Anodyne FPR1 46 34 O=C(N[C@H](CCc1ccccc1)C(F)F)c1ncsc1C1CC1 ZINC000880840450 EI On-Demand Anodyne MAP1 28 40 O=C(N[C@@H](CCc1ccccc1)C(F)F)c1ncsc1C1CC1 ZINC000880840451 EI On-Demand Anodyne MAP1 28 40 CN1CCCC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880840457 CD On-Demand Anodyne HTR4 59 41 CN1CCCC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880840457 CD On-Demand Anodyne JAK3 17 40 CN1CCCC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880840457 CD On-Demand Anodyne TYK2 20 40 CN1CCCC[C@H](CNC(=O)c2cccn3nccc23)C1 ZINC000880840457 CD On-Demand Anodyne CACNA1I 48 35 O=C(COC1CC1)N[C@H](CCc1ccccc1)C(F)F ZINC000880840463 CF On-Demand Anodyne ACE 47 38 O=C(COC1CC1)N[C@H](CCc1ccccc1)C(F)F ZINC000880840463 CF On-Demand Anodyne TIMP3 83 37 O=C(COC1CC1)N[C@@H](CCc1ccccc1)C(F)F ZINC000880840464 CF On-Demand Anodyne ACE 47 38 O=C(COC1CC1)N[C@@H](CCc1ccccc1)C(F)F ZINC000880840464 CF On-Demand Anodyne TIMP3 83 37 CN1CCCC[C@H](CNC(=O)C(C)(C)c2ccc(F)cc2F)C1 ZINC000880840466 DG On-Demand Anodyne CACNA1I 58 39 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cccc3c2OCCCO3)c1 ZINC000880840483 GF On-Demand Anodyne MTNR1A 29 43 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cccc3c2OCCCO3)CC1 ZINC000880840492 GF On-Demand Anodyne GPR119 30 42 CCCCNC(=O)Nc1cccc2c1OCCCO2 ZINC000880840497 CF On-Demand Anodyne MTNR1A 25 50 O=C(NCCCN1CCCCC1)Nc1cccc2c1OCCCO2 ZINC000880840509 EF On-Demand Anodyne HRH2 26 41 O=C(NCCCN1CCCCC1)Nc1cccc2c1OCCCO2 ZINC000880840509 EF On-Demand Anodyne CCR3 28 43 O=C(NCCCN1CCCCC1)Nc1cccc2c1OCCCO2 ZINC000880840509 EF On-Demand Anodyne CHRNA7 21 49 O=C(NCCCN1CCCCC1)Nc1cccc2c1OCCCO2 ZINC000880840509 EF On-Demand Anodyne HNMT 49 33 COc1ncccc1CNC(=O)Nc1cccc2c1OCCCO2 ZINC000880840515 EF On-Demand Anodyne G2YM83_BOTF4 47 34 COC(=O)[C@@H](C)Oc1ccc(NC(=O)c2cnc(C(C)C)nc2C)cc1F ZINC000880840558 GG On-Demand Anodyne MET 47 39 Cc1cc(NC(=O)NC[C@@H]2CC[C@@H](c3ccccc3)O2)cc(S(C)(=O)=O)c1 ZINC000880840599 GG On-Demand Anodyne LPL 43 33 Cc1cc(NC(=O)NC[C@H]2CC[C@H](c3ccccc3)O2)cc(S(C)(=O)=O)c1 ZINC000880840600 GG On-Demand Anodyne LPL 43 33 Cc1cc(NC(=O)NC[C@H]2CC[C@@H](c3ccccc3)O2)cc(S(C)(=O)=O)c1 ZINC000880840601 GG On-Demand Anodyne LPL 43 33 Cc1cc(NC(=O)NC[C@@H]2CC[C@H](c3ccccc3)O2)cc(S(C)(=O)=O)c1 ZINC000880840602 GG On-Demand Anodyne LPL 43 33 Cc1cc(NC(=O)NC[C@H]2CC(=O)N(C)C2)cc(S(C)(=O)=O)c1 ZINC000880840658 EC On-Demand Anodyne CCR3 17 40 Cc1cc(NC(=O)NC[C@@H]2CC(=O)N(C)C2)cc(S(C)(=O)=O)c1 ZINC000880840659 EC On-Demand Anodyne CCR3 17 40 C#CC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880840703 DE On-Demand Mild EPHX2 20 42 CO[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880840709 EE On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)NCCN2C[C@@H]3CCCCN3C2=O)cc(S(C)(=O)=O)c1 ZINC000880840749 GD On-Demand Anodyne CCR3 19 40 Cc1cc(NC(=O)NCCN2C[C@H]3CCCCN3C2=O)cc(S(C)(=O)=O)c1 ZINC000880840750 GD On-Demand Anodyne CCR3 19 40 CC(C)(C(=O)N1CC2(CCCO2)C1)c1ccc(C(F)(F)F)cc1 ZINC000880840773 EG On-Demand Anodyne EPHX2 16 50 Cc1cc(NC(=O)N[C@H](c2ccccc2)C(C)(C)CO)cc(S(C)(=O)=O)c1 ZINC000880840803 GG On-Demand Anodyne CTSF 43 32 Cc1cc(NC(=O)NC[C@@H]2CCN(C(C)(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880840812 FF On-Demand Anodyne CACNA1I 49 33 Cc1cc(NC(=O)NC[C@H]2CCN(C(C)(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880840813 FF On-Demand Anodyne CACNA1I 49 33 C=C[C@H](C)ONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840878 CE On-Demand Mild MTCA1 15 44 C=C[C@H](C)ONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840878 CE On-Demand Mild P96878_MYCTU 18 44 C=C[C@@H](C)ONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840879 CE On-Demand Mild MTCA1 15 44 C=C[C@@H](C)ONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880840879 CE On-Demand Mild P96878_MYCTU 18 44 Cc1cc(NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)cc(S(C)(=O)=O)c1 ZINC000880840905 FE On-Demand Anodyne PLM1_PLAFA 43 39 Cc1cc(NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)cc(S(C)(=O)=O)c1 ZINC000880840905 FE On-Demand Anodyne PLM2_PLAFA 68 38 Cc1cc(NC(=O)NCCCC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880840967 DG On-Demand Anodyne CCR3 37 46 Cc1cc(NC(=O)N[C@H]2C[C@@H](O)c3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880840982 FF On-Demand Anodyne CCKAR 21 40 Cc1cc(NC(=O)N[C@H]2C[C@@H](O)c3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880840982 FF On-Demand Anodyne CCKBR 27 40 Cc1cc(NC(=O)N[C@H]2C[C@H](O)c3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880840986 FF On-Demand Anodyne CCKAR 21 40 Cc1cc(NC(=O)N[C@H]2C[C@H](O)c3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880840986 FF On-Demand Anodyne CCKBR 27 40 Cc1cc(NC(=O)NCCOCC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880841002 EE On-Demand Anodyne CCR3 15 40 Cc1cc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc(S(C)(=O)=O)c1 ZINC000880841018 GE On-Demand Anodyne CCKAR 56 48 Cc1cc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc(S(C)(=O)=O)c1 ZINC000880841018 GE On-Demand Anodyne PYGL 34 49 Cc1cc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc(S(C)(=O)=O)c1 ZINC000880841018 GE On-Demand Anodyne PYGM 30 49 Cc1cc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc(S(C)(=O)=O)c1 ZINC000880841018 GE On-Demand Anodyne CCKBR 82 48 CC(=O)N(C)c1ccc(CNC(=O)c2ncsc2C2CC2)cc1 ZINC000880841038 EF On-Demand Anodyne VHL 40 31 CNC(=O)[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880841044 EC On-Demand Anodyne EPHX2 32 44 COC(=O)[C@@H](C)Oc1ccc(NC(=O)c2ncsc2C2CC2)cc1F ZINC000880841051 FG On-Demand Anodyne MAP1 55 34 COC(=O)[C@@H](C)Oc1ccc(NC(=O)c2ncsc2C2CC2)cc1F ZINC000880841051 FG On-Demand Anodyne MET 62 37 Cc1cc(NC(=O)NC[C@@H](C)c2ccccn2)cc(S(C)(=O)=O)c1 ZINC000880841053 EF On-Demand Anodyne NAMPT 21 41 Cc1cc(NC(=O)NC[C@H](C)c2ccccn2)cc(S(C)(=O)=O)c1 ZINC000880841054 EF On-Demand Anodyne NAMPT 21 41 COC[C@]1(CO)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880841057 FD On-Demand Anodyne S1PR2 20 40 C[Si](C)(C)c1ccc(CCNC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)cc1 ZINC000880841071 GE On-Demand Anodyne GPBAR1 26 40 Cc1cc(NC(=O)NCCC[C@@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880841072 EE On-Demand Anodyne CCR3 25 42 Cc1cc(NC(=O)NCCC[C@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880841073 EE On-Demand Anodyne CCR3 25 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)N(C)c2ccccc2C1 ZINC000880841083 GD On-Demand Anodyne P2RY12 45 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)N(C)c2ccccc2C1 ZINC000880841083 GD On-Demand Anodyne FPR1 41 32 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)N(C)c2ccccc2C1 ZINC000880841085 GD On-Demand Anodyne P2RY12 45 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(=O)N(C)c2ccccc2C1 ZINC000880841085 GD On-Demand Anodyne FPR1 41 32 CCN1CC[C@H](N(CC)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880841110 FE On-Demand Anodyne CCR5 26 46 CCN1CC[C@@H](N(CC)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880841120 FE On-Demand Anodyne CCR5 26 46 COC1(CO)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880841137 FD On-Demand Anodyne S1PR2 27 44 Cc1cc(NC(=O)NCCCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880841157 DF On-Demand Anodyne CCR3 36 47 Cc1cc(NC(=O)N[C@H](C)[C@@](C)(O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880841241 GF On-Demand Anodyne MTCA1 15 41 Cc1cc(NC(=O)N[C@H](C)[C@@](C)(O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880841241 GF On-Demand Anodyne P96878_MYCTU 20 41 Cc1cc(NC(=O)N[C@H](C)[C@](C)(O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880841249 GF On-Demand Anodyne MTCA1 15 41 Cc1cc(NC(=O)N[C@H](C)[C@](C)(O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880841249 GF On-Demand Anodyne P96878_MYCTU 20 41 Cc1ccc(CC2CN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880841257 FG On-Demand Anodyne CCR3 26 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)C2 ZINC000880841313 FF On-Demand Anodyne MMP13 17 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)C2 ZINC000880841313 FF On-Demand Anodyne MMP3 22 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)C2 ZINC000880841313 FF On-Demand Anodyne MMP9 17 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)C2 ZINC000880841313 FF On-Demand Anodyne MMP1 19 41 COC(=O)[C@@H](C)Oc1ccc(NC(=O)c2c3c(nn2C)CCSC3)cc1F ZINC000880841316 GF On-Demand Anodyne MET 51 33 COC(=O)[C@@H](C)Oc1ccc(NC(=O)c2nccnc2SC)cc1F ZINC000880841330 FF On-Demand Anodyne MET 75 39 COC(=O)[C@@H](C)Oc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1F ZINC000880841389 ED On-Demand Anodyne MET 40 38 COC(=O)[C@@H](C)Oc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1F ZINC000880841389 ED On-Demand Anodyne ENPP1 55 31 COC(=O)[C@@H](C)Oc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1F ZINC000880841392 ED On-Demand Anodyne MET 40 38 COC(=O)[C@@H](C)Oc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1F ZINC000880841392 ED On-Demand Anodyne ENPP1 55 31 COC(=O)[C@H]1CC[C@H](C(=O)OC)N(C(=O)c2cnc(CC3CC3)s2)C1 ZINC000880841411 FD On-Demand Anodyne PTR1 47 34 COC(=O)[C@H]1CC[C@@H](C(=O)OC)N(C(=O)c2cnc(CC3CC3)s2)C1 ZINC000880841412 FD On-Demand Anodyne PTR1 47 34 Cc1cc(NC(=O)NCCc2cnccc2C)cc(S(C)(=O)=O)c1 ZINC000880841423 EE On-Demand Anodyne NAMPT 35 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(N(C)C(C)=O)cc1 ZINC000880841554 GE On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(N(C)C(C)=O)cc1 ZINC000880841554 GE On-Demand Anodyne FPR1 44 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(N(C)C(C)=O)cc1 ZINC000880841555 GE On-Demand Anodyne PAPA1_CARPA 44 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccc(N(C)C(C)=O)cc1 ZINC000880841555 GE On-Demand Anodyne FPR1 44 36 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(N(C)C(C)=O)cc1)C2 ZINC000880841577 FG On-Demand Anodyne NQO2 28 40 COc1ccc2c(c1)CC[C@H](C(=O)NCc1ccc(N(C)C(C)=O)cc1)C2 ZINC000880841577 FG On-Demand Anodyne MTNR1A 42 41 Cc1cc(NC(=O)NCCc2ncccc2C)cc(S(C)(=O)=O)c1 ZINC000880841579 EE On-Demand Anodyne NAMPT 30 41 Cc1cc(NC(=O)NC[C@@H]2CCCN2CCCO)cc(S(C)(=O)=O)c1 ZINC000880841737 FD On-Demand Anodyne CCR3 35 41 C[Si](C)(C)c1ccc(CCNC(=O)C2CCC(S(C)(=O)=O)CC2)cc1 ZINC000880841738 GE On-Demand Anodyne MTNR1A 20 43 Cc1cc(NC(=O)NC[C@H]2CCCN2CCCO)cc(S(C)(=O)=O)c1 ZINC000880841739 FD On-Demand Anodyne CCR3 35 41 Cc1cc(NC(=O)NCc2cc(C)cs2)cc(S(C)(=O)=O)c1 ZINC000880841770 EG On-Demand Anodyne LPL 42 31 COC[C@@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880841787 EE On-Demand Anodyne EPHX2 15 42 COC[C@@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880841787 EE On-Demand Anodyne CASP7 47 36 Cc1cc(NC(=O)NC[C@H](O)C2CCC2)cc(S(C)(=O)=O)c1 ZINC000880841814 ED On-Demand Anodyne PRMT3 18 44 Cc1cc(NC(=O)NC[C@@H](O)C2CCC2)cc(S(C)(=O)=O)c1 ZINC000880841815 ED On-Demand Anodyne PRMT3 18 44 Cc1cc(NC(=O)N[C@H]2CCO[C@@H](c3cccnc3)C2)cc(S(C)(=O)=O)c1 ZINC000880841816 GF On-Demand Anodyne NAMPT 46 42 NC(=O)[C@@H]1CCCN1C(=O)COC1CC1 ZINC000880841838 BB On-Demand Anodyne TRHR 54 33 NC(=O)[C@@H]1CCCN1C(=O)COC1CC1 ZINC000880841838 BB On-Demand Anodyne PREP 47 45 NC(=O)[C@@H]1CCCN1C(=O)COC1CC1 ZINC000880841838 BB On-Demand Anodyne TPP2 24 48 NC(=O)[C@@H]1CCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880841862 FE On-Demand Anodyne SFRP1 44 34 NC(=O)[C@@H]1CCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880841862 FE On-Demand Anodyne WNT3 48 34 NC(=O)[C@@H]1CCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880841891 DC On-Demand Anodyne TRHR 54 35 Cc1cc(NC(=O)NC[C@H]2CCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880841973 ED On-Demand Anodyne CCR3 41 43 Cc1cc(NC(=O)NC[C@@H]2CCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880841975 ED On-Demand Anodyne CCR3 41 43 Cc1cc(NC(=O)N[C@H]2CCO[C@H](c3cccnc3)C2)cc(S(C)(=O)=O)c1 ZINC000880842070 GF On-Demand Anodyne NAMPT 46 42 Cc1cc(NC(=O)NCCOCC2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880842104 FF On-Demand Anodyne CCR3 15 40 CS(=O)(=O)NC1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880842109 GD On-Demand Anodyne RBP4 66 36 CS(=O)(=O)NC1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880842109 GD On-Demand Anodyne SFRP1 96 35 CS(=O)(=O)NC1CN(C(=O)c2cc3cccc(C(F)(F)F)c3nc2O)C1 ZINC000880842109 GD On-Demand Anodyne WNT3 52 31 Cc1cc(NC(=O)N[C@](C)(CO)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880842129 FE On-Demand Anodyne IMDH_CRYPV 56 36 CCC1(c2ccccc2)CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880842131 FH On-Demand Anodyne S1PR2 17 43 CCC1(c2ccccc2)CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880842131 FH On-Demand Anodyne EPHX2 17 41 NC(=O)[C@@H]1CCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880842141 DC On-Demand Anodyne TRHR 60 39 NC(=O)[C@@H]1CCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880842141 DC On-Demand Anodyne PREP 67 38 Cc1cc(NC(=O)NCCN2CCCOCC2)cc(S(C)(=O)=O)c1 ZINC000880842192 FD On-Demand Anodyne CCR3 22 42 Cc1cc(NC(=O)NCCN2CCCOCC2)cc(S(C)(=O)=O)c1 ZINC000880842192 FD On-Demand Anodyne EPHX2 19 43 Cc1cc(NC(=O)NCCN2CCCOCC2)cc(S(C)(=O)=O)c1 ZINC000880842192 FD On-Demand Anodyne NAMPT 18 43 CC[C@@H](NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000880842203 EH On-Demand Anodyne LPL 43 33 CC[C@@H](NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000880842203 EH On-Demand Anodyne TACR3 50 43 NC(=O)[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880842209 CE On-Demand Anodyne HCRTR1 19 40 NC(=O)[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880842209 CE On-Demand Anodyne DPP4 15 48 NC(=O)[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880842209 CE On-Demand Anodyne PREP 64 41 CC(C)(C)OC(=O)CC[C@H]1C[C@@H](C(=O)N2CCC[C@H]2C(N)=O)CO1 ZINC000880842236 EC On-Demand Anodyne PREP 18 41 CC(C)(C)OC(=O)CC[C@H]1C[C@H](C(=O)N2CCC[C@H]2C(N)=O)CO1 ZINC000880842237 EC On-Demand Anodyne PREP 18 41 CC(C)(C)OC(=O)CC[C@@H]1C[C@@H](C(=O)N2CCC[C@H]2C(N)=O)CO1 ZINC000880842239 EC On-Demand Anodyne PREP 18 41 CC(C)(C)OC(=O)CC[C@@H]1C[C@H](C(=O)N2CCC[C@H]2C(N)=O)CO1 ZINC000880842240 EC On-Demand Anodyne PREP 18 41 Cc1nc(C(C)C)ncc1C(=O)N1CCC[C@H]1C(N)=O ZINC000880842249 CC On-Demand Anodyne TRHR 69 35 Cc1cc(NC(=O)NCc2cc(C)nc(C)c2)cc(S(C)(=O)=O)c1 ZINC000880842252 EF On-Demand Anodyne PRMT3 17 43 Cc1cc(NC(=O)NCc2cc(C)nc(C)c2)cc(S(C)(=O)=O)c1 ZINC000880842252 EF On-Demand Anodyne NAMPT 42 42 Cc1cc(-c2nc(C)c(C(=O)N3CCC[C@H]3C(N)=O)s2)ccc1F ZINC000880842257 EF On-Demand Anodyne LGMN 54 35 Cc1cc(-c2nc(C)c(C(=O)N3CCC[C@H]3C(N)=O)s2)ccc1F ZINC000880842257 EF On-Demand Anodyne TRPC6 47 35 COC[C@@H]1CCCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880842264 FF On-Demand Anodyne EPHX2 20 42 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N1CCC[C@H]1C(N)=O ZINC000880842271 CC On-Demand Anodyne TRHR 72 36 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC[C@H]1C(N)=O ZINC000880842272 CC On-Demand Anodyne TRHR 72 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N1CCC[C@H]1C(N)=O ZINC000880842273 CC On-Demand Anodyne TRHR 72 36 Cc1cc(NC(=O)NCC2OCCCO2)cc(S(C)(=O)=O)c1 ZINC000880842330 ED On-Demand Anodyne LPL 41 31 Cc1cc(NC(=O)NCCC[C@@H]2CCCCO2)cc(S(C)(=O)=O)c1 ZINC000880842351 FF On-Demand Anodyne CCR3 24 40 Cc1cc(NC(=O)NCCC[C@H]2CCCCO2)cc(S(C)(=O)=O)c1 ZINC000880842352 FF On-Demand Anodyne CCR3 24 40 Cc1cc(NC(=O)NC[C@@H]2Cc3ccccc3O2)cc(S(C)(=O)=O)c1 ZINC000880842423 FF On-Demand Anodyne LPL 43 32 Cc1cc(NC(=O)NC[C@H]2Cc3ccccc3O2)cc(S(C)(=O)=O)c1 ZINC000880842424 FF On-Demand Anodyne LPL 43 32 CN1C(=O)CN(C(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)Cc2ccccc21 ZINC000880842425 FE On-Demand Anodyne AVPR1A 17 41 CN1C(=O)CN(C(=O)c2ccc([C@H]3CCC(=O)N3)cc2)Cc2ccccc21 ZINC000880842426 FE On-Demand Anodyne AVPR1A 17 41 Cc1cc(NC(=O)NCCCCN(C)C2CC2)cc(S(C)(=O)=O)c1 ZINC000880842457 FE On-Demand Anodyne CCR3 29 44 CC(=O)N(C)c1ccc(CNC(=O)CC[C@@H]2CCc3ccccc32)cc1 ZINC000880842458 FH On-Demand Anodyne MTNR1B 25 44 CC(=O)N(C)c1ccc(CNC(=O)CC[C@H]2CCc3ccccc32)cc1 ZINC000880842459 FH On-Demand Anodyne MTNR1B 25 44 NC(=O)[C@@H]1CCCN1C(=O)c1cccn2nccc12 ZINC000880842492 CC On-Demand Anodyne JAK3 17 40 NC(=O)[C@@H]1CCCN1C(=O)c1cccn2nccc12 ZINC000880842492 CC On-Demand Anodyne PREP 58 37 NC(=O)[C@@H]1CCCN1C(=O)c1cccn2nccc12 ZINC000880842492 CC On-Demand Anodyne TYK2 20 40 NC(=O)[C@@H]1CCCN1C(=O)c1ccc(OC(F)F)c(Br)c1 ZINC000880842501 FE On-Demand Anodyne PREP 31 42 CCC[C@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880842505 EH On-Demand Anodyne EPHX2 15 41 CCC[C@@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880842506 EH On-Demand Anodyne EPHX2 15 41 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880842510 GE On-Demand Anodyne S1PR2 25 40 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880842511 GE On-Demand Anodyne S1PR2 25 40 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880842512 GE On-Demand Anodyne S1PR2 25 40 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880842513 GE On-Demand Anodyne S1PR2 25 40 CC(=O)N1CCc2c(NC(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)cccc21 ZINC000880842515 GF On-Demand Anodyne LPL 53 35 NC(=O)[C@@H]1CCCN1C(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880842562 BC On-Demand Anodyne TRHR 47 32 NC(=O)[C@@H]1CCCN1C(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880842562 BC On-Demand Anodyne PREP 32 40 NC(=O)[C@@H]1CCCN1C(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880842562 BC On-Demand Anodyne TPP2 18 45 CCOC(=O)CCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880842564 GF On-Demand Anodyne GPR119 28 41 CC[C@H](C)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880842593 FE On-Demand Anodyne S1PR2 26 41 NC(=O)c1cc(-c2csc(NC(=O)[C@@H]3Cc4ccccc4CN3C(=O)c3ccccc3)n2)c[nH]1 ZINC000880842635 JG On-Demand Anodyne OPRM1 20 40 NC(=O)c1cc(-c2csc(NC(=O)[C@@H]3Cc4ccccc4CN3C(=O)c3ccccc3)n2)c[nH]1 ZINC000880842635 JG On-Demand Anodyne OPRD1 73 38 NC(=O)c1cc(-c2csc(NC(=O)[C@@H]3Cc4ccccc4CN3C(=O)c3ccccc3)n2)c[nH]1 ZINC000880842635 JG On-Demand Anodyne CFTR 79 48 Cc1cc(NC(=O)NC[C@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880842746 EG On-Demand Anodyne LPL 43 36 Cc1cc(NC(=O)NC[C@@H](C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880842747 EG On-Demand Anodyne LPL 43 36 Cc1cc(NC(=O)N[C@H](C)CCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880842755 DG On-Demand Anodyne CCR3 42 36 NC(=O)[C@@H]1CCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880842759 CD On-Demand Anodyne TRHR 65 34 NC(=O)[C@@H]1CCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880842759 CD On-Demand Anodyne PREP 85 37 Cc1cc(NC(=O)Nc2cc(C)c(O)c(C)c2C)cc(S(C)(=O)=O)c1 ZINC000880842764 FH On-Demand Anodyne LPL 54 36 Cc1cc(NC(=O)Nc2cc(C)c(O)c(C)c2C)cc(S(C)(=O)=O)c1 ZINC000880842764 FH On-Demand Anodyne P96878_MYCTU 16 45 Cc1cnc(Cl)c(C(=O)N2CCC[C@H]2C(N)=O)c1 ZINC000880842785 CD On-Demand Anodyne TRHR 56 34 NC(=O)[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880842799 CD On-Demand Anodyne ACE 29 41 NC(=O)[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880842799 CD On-Demand Anodyne TRHR 57 38 NC(=O)[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880842799 CD On-Demand Anodyne HTR7 18 45 NC(=O)[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880842799 CD On-Demand Anodyne CPT2 40 38 NC(=O)[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880842799 CD On-Demand Anodyne PREP 103 45 NC(=O)[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880842800 CD On-Demand Anodyne ACE 29 41 NC(=O)[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880842800 CD On-Demand Anodyne TRHR 57 38 NC(=O)[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880842800 CD On-Demand Anodyne HTR7 18 45 NC(=O)[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880842800 CD On-Demand Anodyne CPT2 40 38 NC(=O)[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880842800 CD On-Demand Anodyne PREP 103 45 CCN(Cc1c[nH]c2ccccc12)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880842822 GH On-Demand Anodyne EDNRB 52 34 CCN(Cc1c[nH]c2ccccc12)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880842822 GH On-Demand Anodyne CFTR 32 41 Cc1cc(NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)cc(S(C)(=O)=O)c1 ZINC000880842831 FD On-Demand Anodyne CCR3 27 44 NC(=O)[C@@H]1CCCN1C(=O)c1cccc2nsnc12 ZINC000880842846 CC On-Demand Anodyne PREP 57 39 CC(=O)N[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880842856 ED On-Demand Anodyne EPHX2 24 41 CC(=O)N[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880842857 ED On-Demand Anodyne EPHX2 24 41 Cc1cc(NC(=O)N[C@H]2C[C@H]3CCCCN3C2=O)cc(S(C)(=O)=O)c1 ZINC000880842862 FD On-Demand Anodyne CCKAR 15 41 Cc1cc(NC(=O)N[C@H]2C[C@@H]3CCCCN3C2=O)cc(S(C)(=O)=O)c1 ZINC000880842865 FD On-Demand Anodyne CCKAR 15 41 NC(=O)[C@@H]1CCCN1C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880842871 DE On-Demand Anodyne PREP 32 42 COC1(C(F)(F)F)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880842911 GF On-Demand Anodyne S1PR2 26 41 COC[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880842914 FF On-Demand Anodyne CASP7 40 34 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CCO2 ZINC000880842926 GF On-Demand Anodyne MMP13 16 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CCO2 ZINC000880842926 GF On-Demand Anodyne MMP3 20 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CCO2 ZINC000880842926 GF On-Demand Anodyne MMP9 15 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CCO2 ZINC000880842926 GF On-Demand Anodyne MMP1 15 41 CS(=O)(=O)NC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880842932 GC On-Demand Anodyne PREP 42 47 CS(=O)(=O)NC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880842932 GC On-Demand Anodyne TGM2 28 40 CS(=O)(=O)NC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880842932 GC On-Demand Anodyne F13A1 37 40 CS(=O)(=O)NC1CN(C(=O)[C@H]2C[C@@H](F)CN2C(=O)OCc2ccccc2)C1 ZINC000880842932 GC On-Demand Anodyne Q9NAW4_PLAFA 26 40 NC(=O)[C@@H]1CCCN1C(=O)c1cncc2[nH]ccc12 ZINC000880842934 CC On-Demand Anodyne TRHR 61 32 C=CC(C)(C)CC(=O)N1CCC[C@H]1C(N)=O ZINC000880843047 BD On-Demand Mild TRHR 54 34 C=CC(C)(C)CC(=O)N1CCC[C@H]1C(N)=O ZINC000880843047 BD On-Demand Mild PREP 34 41 C=CC(C)(C)CC(=O)N1CCC[C@H]1C(N)=O ZINC000880843047 BD On-Demand Mild TPP2 27 48 Cn1ncc(Br)c1CC(=O)N1CCC[C@H]1C(N)=O ZINC000880843090 DC On-Demand Anodyne TRHR 69 34 Cn1ncc(Br)c1CC(=O)N1CCC[C@H]1C(N)=O ZINC000880843090 DC On-Demand Anodyne PREP 50 35 Cc1cc(NC(=O)N[C@H](CO)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843094 FE On-Demand Anodyne LPL 41 33 Cc1cc(NC(=O)N[C@H](CO)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843094 FE On-Demand Anodyne MME 44 39 Cc1cc(NC(=O)N[C@H](CO)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843094 FE On-Demand Anodyne ANPEP 55 34 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1Cl ZINC000880843118 GH On-Demand Anodyne PDE6A 43 33 Cc1cc(NC(=O)NCC(C)(C)c2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880843137 FF On-Demand Anodyne NAMPT 65 39 CC(=O)N(C)c1ccc(CNC(=O)c2ccc(CN3CCOCC3)o2)cc1 ZINC000880843141 FE On-Demand Anodyne DPOL_VZVD 25 43 Cc1cc(NC(=O)N[C@H]2CCCc3cc(C#N)ccc32)cc(S(C)(=O)=O)c1 ZINC000880843173 GG On-Demand Mild BDKRB1 40 37 CS(=O)(=O)NC1CN(C(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880843194 DD On-Demand Anodyne CCR8 43 38 CS(=O)(=O)NC1CN(C(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880843195 DD On-Demand Anodyne CCR8 43 38 Cc1cc(NC(=O)NCC[C@@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880843196 FE On-Demand Anodyne CCR3 53 44 Cc1cc(NC(=O)NCC[C@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880843197 FE On-Demand Anodyne CCR3 53 44 Cc1cc(NC(=O)N[C@H](C)CCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880843204 GG On-Demand Anodyne TBXAS1 38 46 Cc1cc(NC(=O)N[C@H](C)CCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880843204 GG On-Demand Anodyne PTAFR 35 48 Cc1cc(NC(=O)N[C@H](C)CCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880843204 GG On-Demand Anodyne NAMPT 51 40 CCOC(=O)C1=CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880843226 EE On-Demand Anodyne GABRA1 18 44 CCOC(=O)C1=CC[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880843226 EE On-Demand Anodyne GABRA2 15 44 NC(=O)[C@@H]1CCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880843231 CC On-Demand Anodyne TRHR 62 34 NC(=O)[C@@H]1CCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880843231 CC On-Demand Anodyne PREP 65 45 Cc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843234 GF On-Demand Anodyne TRPV1 26 47 Cc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843234 GF On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)NCc2ccc(C(C)(C)O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843234 GF On-Demand Anodyne NAMPT 41 40 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)N1CCC[C@H]1C(N)=O ZINC000880843241 GG On-Demand Anodyne TRPC6 41 37 Cc1cc(NC(=O)NCC2=CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880843404 DD On-Demand Anodyne NAMPT 15 41 Cc1cc(NC(=O)NC[C@@H]2COc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880843441 FF On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)NC[C@H]2COc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880843442 FF On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)N[C@H](C)CCN2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880843502 GD On-Demand Anodyne CCR3 51 41 Cc1cc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843649 EG On-Demand Anodyne EPHX2 28 52 Cc1cc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843651 EG On-Demand Anodyne EPHX2 28 52 COCCONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880843658 DD On-Demand Anodyne P96878_MYCTU 16 44 CCn1cccc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1=O ZINC000880843691 FD On-Demand Anodyne NAMPT 28 42 Cc1cc(NC(=O)NCC(C)(C)c2ccccn2)cc(S(C)(=O)=O)c1 ZINC000880843698 FF On-Demand Anodyne NAMPT 23 44 Cc1cc(NC(=O)NCCCn2ccnc2C)cc(S(C)(=O)=O)c1 ZINC000880843715 FE On-Demand Anodyne CCR3 21 42 Cc1cc(NC(=O)NCCCn2ccnc2C)cc(S(C)(=O)=O)c1 ZINC000880843715 FE On-Demand Anodyne QPCT 40 40 Cc1cc(NC(=O)NCCCc2cccc(C)n2)cc(S(C)(=O)=O)c1 ZINC000880843729 FF On-Demand Anodyne CCR3 15 41 COC1(C)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880843778 EE On-Demand Anodyne S1PR2 26 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)c1ccc(OC)c(F)c1 ZINC000880843815 GG On-Demand Anodyne PAPA1_CARPA 37 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC(C)(C)c1ccc(OC)c(F)c1 ZINC000880843816 GG On-Demand Anodyne PAPA1_CARPA 37 40 Cc1cc(NC(=O)NCCCCCN2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880843835 FF On-Demand Anodyne HRH2 29 41 Cc1cc(NC(=O)NCCCCCN2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880843835 FF On-Demand Anodyne HTR2A 17 41 Cc1cc(NC(=O)NCCCCCN2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880843835 FF On-Demand Anodyne CCR3 42 52 Cc1cc(NC(=O)NCCCCCN2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880843835 FF On-Demand Anodyne CHRNA7 18 50 Cc1cc(NC(=O)NCc2ccc(C[S@@](C)=O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843845 GF On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)NCc2ccc(C[S@@](C)=O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843845 GF On-Demand Anodyne NAMPT 38 42 Cc1cc(NC(=O)NCc2ccc(C[S@](C)=O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843846 GF On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)NCc2ccc(C[S@](C)=O)cc2)cc(S(C)(=O)=O)c1 ZINC000880843846 GF On-Demand Anodyne NAMPT 38 42 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC[C@H]1NS(C)(=O)=O)C2 ZINC000880843847 GD On-Demand Anodyne MMP13 23 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC[C@H]1NS(C)(=O)=O)C2 ZINC000880843847 GD On-Demand Anodyne MMP3 32 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC[C@H]1NS(C)(=O)=O)C2 ZINC000880843847 GD On-Demand Anodyne MMP7 26 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC[C@H]1NS(C)(=O)=O)C2 ZINC000880843847 GD On-Demand Anodyne MMP1 26 40 Cc1cc(NC(=O)N[C@H](CCO)c2ccc(Cl)cc2)cc(S(C)(=O)=O)c1 ZINC000880843857 GG On-Demand Anodyne UTS2 47 38 Cc1cc(NC(=O)NCCC2CC(O)C2)cc(S(C)(=O)=O)c1 ZINC000880843882 ED On-Demand Anodyne CCR3 15 40 Cc1cc(NC(=O)N[C@H]2CCN(C)[C@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843895 GF On-Demand Anodyne CCKBR 48 35 Cc1cc(NC(=O)N[C@H]2CCN(C)[C@@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880843896 GF On-Demand Anodyne CCKBR 48 35 Cc1cc(NC(=O)NCC2=CCCOC2)cc(S(C)(=O)=O)c1 ZINC000880843983 DD On-Demand Anodyne NAMPT 18 41 CS(=O)(=O)N[C@@H]1CCCC[C@H]1NC(=O)c1cc2ccccc2cc1F ZINC000880843993 FF On-Demand Anodyne SSTR3 29 40 C=CCOC(=O)[C@H](CC(=O)N1CCO[C@@H]2CCC[C@@H]21)NC(=O)OC(C)(C)C ZINC000880843994 GD On-Demand Mild REN 41 37 CCC[C@]1(CO)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880844020 FE On-Demand Anodyne S1PR2 21 40 NC(=O)c1cc(-c2csc(NC(=O)C(O)(c3ccccc3)c3ccccc3)n2)c[nH]1 ZINC000880844190 HG On-Demand Anodyne ROCK1 20 41 NC(=O)c1cc(-c2csc(NC(=O)C(O)(c3ccccc3)c3ccccc3)n2)c[nH]1 ZINC000880844190 HG On-Demand Anodyne ROCK2 17 41 Cc1cc(NC(=O)Nc2ccc([C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880844209 FH On-Demand Anodyne LPL 49 34 Cc1cc(NC(=O)Nc2ccc([C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880844209 FH On-Demand Anodyne P96878_MYCTU 36 45 Cc1cc(NC(=O)Nc2ccc([C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880844210 FH On-Demand Anodyne LPL 49 34 Cc1cc(NC(=O)Nc2ccc([C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880844210 FH On-Demand Anodyne P96878_MYCTU 36 45 Cc1cc(NC(=O)NC[C@@H]2CSc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880844219 GG On-Demand Anodyne LPL 42 33 Cc1cc(NC(=O)NC[C@H]2CSc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880844220 GG On-Demand Anodyne LPL 42 33 Cc1cc(NC(=O)NCCCC2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880844223 FF On-Demand Anodyne CCR3 30 44 CCCN(CCN1CCCC1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880844232 FF On-Demand Anodyne CASR 38 48 Cc1cc(NC(=O)NC[C@@]2(CO)C[C@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880844239 GF On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)NC[C@]2(CO)C[C@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880844240 GF On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)NC[C@]2(CO)C[C@@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880844241 GF On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)NC[C@@]2(CO)C[C@@H]2c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880844242 GF On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccc3F)C2)cc(S(C)(=O)=O)c1 ZINC000880844274 GF On-Demand Anodyne EPHX2 37 40 Cc1cc(NC(=O)NCC2(c3ccccn3)CCC2)cc(S(C)(=O)=O)c1 ZINC000880844280 FG On-Demand Anodyne NMBR 45 40 Cc1cc(NC(=O)NCC2(c3ccccn3)CCC2)cc(S(C)(=O)=O)c1 ZINC000880844280 FG On-Demand Anodyne GRPR 24 40 Cc1cc(NC(=O)NCC2(c3ccccn3)CCC2)cc(S(C)(=O)=O)c1 ZINC000880844280 FG On-Demand Anodyne NAMPT 35 42 Cc1cc(NC(=O)N[C@H]2CCCN(CCCO)C2)cc(S(C)(=O)=O)c1 ZINC000880844348 FD On-Demand Anodyne CCR3 48 43 Cc1cc(NC(=O)Nc2cn(C)nc2C2CC2)cc(S(C)(=O)=O)c1 ZINC000880844381 EF On-Demand Anodyne LPL 41 32 Cc1cc(NC(=O)NCC2CCN(C3CC3)CC2)cc(S(C)(=O)=O)c1 ZINC000880844453 FE On-Demand Anodyne CCR3 33 41 Cc1cc(NC(=O)NCC2CCN(C3CC3)CC2)cc(S(C)(=O)=O)c1 ZINC000880844453 FE On-Demand Anodyne CACNA1I 49 33 CCOC(=O)[C@@]1(C(C)C)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880844458 GF On-Demand Anodyne S1PR2 26 41 CCOC(=O)[C@]1(C(C)C)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880844459 GF On-Demand Anodyne S1PR2 26 41 Cc1cc(NC(=O)NCCCN2CCCO[C@@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880844495 GE On-Demand Anodyne CCR3 45 45 Cc1cc(NC(=O)NCCCN2CCCO[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880844496 GE On-Demand Anodyne CCR3 45 45 Cc1cc(NC(=O)Nc2cnn(C3CCCC3)c2C)cc(S(C)(=O)=O)c1 ZINC000880844541 GH On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)N[C@H]2c3ccccc3C[C@H]2O)cc(S(C)(=O)=O)c1 ZINC000880844603 FE On-Demand Anodyne PLM1_PLAFA 43 39 Cc1cc(NC(=O)N[C@H]2c3ccccc3C[C@H]2O)cc(S(C)(=O)=O)c1 ZINC000880844603 FE On-Demand Anodyne PLM2_PLAFA 68 38 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880844611 GG On-Demand Anodyne NPY5R 33 48 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880844612 GG On-Demand Anodyne NPY5R 33 48 Cc1cc(NC(=O)NCC2(N3CCOCC3)CC2)cc(S(C)(=O)=O)c1 ZINC000880844688 FD On-Demand Anodyne NAMPT 15 44 C#CCNC(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880844738 GD On-Demand Mild EPHX2 32 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccco2)C1 ZINC000880844739 FE On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2ccco2)C1 ZINC000880844740 FE On-Demand Anodyne FPR1 45 36 CCO[C@@]1(C)C[C@H]1NC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880844760 ED On-Demand Anodyne PAPA1_CARPA 33 42 CCO[C@@]1(C)C[C@H]1NC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880844761 ED On-Demand Anodyne PAPA1_CARPA 33 42 CCO[C@@]1(C)C[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880844784 DE On-Demand Anodyne GABRA1 18 41 CCO[C@@]1(C)C[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880844784 DE On-Demand Anodyne MPO 46 34 CCO[C@@]1(C)C[C@H]1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880844784 DE On-Demand Anodyne GABRA2 16 41 CCC1(O)CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880844830 DD On-Demand Anodyne S1PR2 26 41 CCO[C@@]1(C)C[C@H]1NC(=O)c1cccn2nccc12 ZINC000880844847 CD On-Demand Anodyne JAK3 20 42 CCO[C@@]1(C)C[C@H]1NC(=O)c1cccn2nccc12 ZINC000880844847 CD On-Demand Anodyne JAK1 16 42 CCO[C@@]1(C)C[C@H]1NC(=O)c1cccn2nccc12 ZINC000880844847 CD On-Demand Anodyne TYK2 23 42 Cc1cc(NC(=O)NCc2ccc(CCN(C)C)cc2)cc(S(C)(=O)=O)c1 ZINC000880844899 GF On-Demand Anodyne PRMT3 19 47 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc(S(C)(=O)=O)c1 ZINC000880844912 FG On-Demand Anodyne IDO1 19 40 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc(S(C)(=O)=O)c1 ZINC000880844912 FG On-Demand Anodyne MTCA1 20 44 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc(S(C)(=O)=O)c1 ZINC000880844912 FG On-Demand Anodyne P96878_MYCTU 23 44 Cc1cc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc(S(C)(=O)=O)c1 ZINC000880844912 FG On-Demand Anodyne IMDH_CRYPV 59 35 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845004 FD On-Demand Anodyne CCR3 42 41 CC(=O)N1CCC[C@H](CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845005 FD On-Demand Anodyne CCR3 42 41 Cc1cc(NC(=O)NCCN2CC=CCC2)cc(S(C)(=O)=O)c1 ZINC000880845012 ED On-Demand Anodyne CCR3 16 42 Cc1cc(NC(=O)NCc2cc(C)c(O)c(C)c2)cc(S(C)(=O)=O)c1 ZINC000880845021 FG On-Demand Anodyne NAMPT 40 42 Cc1cc(NC(=O)NC[C@@H]2CCCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880845072 GF On-Demand Anodyne CCR3 71 38 Cc1cc(NC(=O)NC[C@H]2CCCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880845073 GF On-Demand Anodyne CCR3 71 38 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccn3)C2)cc(S(C)(=O)=O)c1 ZINC000880845112 FE On-Demand Anodyne EPHX2 40 39 Cc1cc(NC(=O)N[C@]2(C)CCOC2)cc(S(C)(=O)=O)c1 ZINC000880845150 DD On-Demand Anodyne LPL 49 35 COC[C@H](NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000880845161 FF On-Demand Anodyne LPL 42 35 COC[C@@H](NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000880845162 FF On-Demand Anodyne LPL 42 35 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845194 FD On-Demand Anodyne EPHX2 41 58 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845195 FD On-Demand Anodyne EPHX2 41 58 CCC1(O)CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880845216 FF On-Demand Anodyne EPHX2 24 40 Cc1cc(NC(=O)NCC2([C@H](O)c3ccccc3)CC2)cc(S(C)(=O)=O)c1 ZINC000880845238 GG On-Demand Anodyne LPL 44 36 Cc1cc(NC(=O)NCC2([C@@H](O)c3ccccc3)CC2)cc(S(C)(=O)=O)c1 ZINC000880845239 GG On-Demand Anodyne LPL 44 36 CSc1cc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)ccn1 ZINC000880845257 FF On-Demand Anodyne NAMPT 41 39 NC(=O)[C@@H]1CCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880845344 DC On-Demand Anodyne TRHR 42 33 NC(=O)[C@@H]1CCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880845344 DC On-Demand Anodyne MPO 42 38 Cc1cc(NC(=O)NCCc2ccncc2C)cc(S(C)(=O)=O)c1 ZINC000880845345 EE On-Demand Anodyne NAMPT 36 42 Cc1cc(NC(=O)N[C@H](c2cccnc2)C2CC2)cc(S(C)(=O)=O)c1 ZINC000880845412 FG On-Demand Anodyne NAMPT 43 45 Cc1cc(NC(=O)N[C@]2(C)CCCOC2)cc(S(C)(=O)=O)c1 ZINC000880845419 EE On-Demand Anodyne LPL 42 33 Cc1cc(NC(=O)NCCc2ccc(CO)cc2)cc(S(C)(=O)=O)c1 ZINC000880845475 FE On-Demand Anodyne CA2 17 47 Cc1cc(NC(=O)NCCc2ccc(CO)cc2)cc(S(C)(=O)=O)c1 ZINC000880845475 FE On-Demand Anodyne CA1 19 46 Cc1cc(NC(=O)NCCc2ccc(CO)cc2)cc(S(C)(=O)=O)c1 ZINC000880845475 FE On-Demand Anodyne CA12 18 43 Cc1cc(NC(=O)NCCc2ccc(CO)cc2)cc(S(C)(=O)=O)c1 ZINC000880845475 FE On-Demand Anodyne CA9 17 43 COCCNc1ccccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880845493 GF On-Demand Anodyne LPL 42 36 Cc1cc(NC(=O)NCCc2ccccc2C)cc(S(C)(=O)=O)c1 ZINC000880845498 EG On-Demand Anodyne NQO2 26 43 Cc1cc(NC(=O)NCCc2ccccc2C)cc(S(C)(=O)=O)c1 ZINC000880845498 EG On-Demand Anodyne MTNR1A 17 43 Cc1cc(NC(=O)NCCc2ccccc2C)cc(S(C)(=O)=O)c1 ZINC000880845498 EG On-Demand Anodyne P96878_MYCTU 15 40 Cc1cncc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880845509 EE On-Demand Anodyne NAMPT 52 62 Cc1cc(NC(=O)NCC2(CO)CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880845551 FE On-Demand Anodyne LPL 48 35 COC(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880845569 FD On-Demand Anodyne EPHX2 26 42 Cc1cc(NC(=O)N[C@H]2CC(=O)N(C3CCCCC3)C2)cc(S(C)(=O)=O)c1 ZINC000880845712 GE On-Demand Anodyne INHA 17 43 CCN1CCC[C@@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845720 EE On-Demand Anodyne CCR3 39 42 CCN1CCC[C@@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845720 EE On-Demand Anodyne EPHX2 32 41 CCN1CCC[C@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845721 EE On-Demand Anodyne CCR3 39 42 CCN1CCC[C@H](NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845721 EE On-Demand Anodyne EPHX2 32 41 Cc1cc(NC(=O)Nc2cc(C)n(C)n2)cc(S(C)(=O)=O)c1 ZINC000880845730 DE On-Demand Anodyne P96878_MYCTU 21 45 NC(=O)c1cc(-c2csc(NC(=O)c3ccc(Cl)c(S(=O)(=O)N4CCCCC4)c3)n2)c[nH]1 ZINC000880845745 JG On-Demand Anodyne MPL 44 41 Cc1cc(NC(=O)N[C@H](C)C[C@H](O)c2ccc(F)cc2)cc(S(C)(=O)=O)c1 ZINC000880845746 GG On-Demand Anodyne CCR3 49 38 Cc1cc(NC(=O)N[C@H](C)C[C@@H](O)c2ccc(F)cc2)cc(S(C)(=O)=O)c1 ZINC000880845747 GG On-Demand Anodyne CCR3 49 38 Cc1cc(NC(=O)NC[C@@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845796 GG On-Demand Anodyne ADRB3 27 40 Cc1cc(NC(=O)NC[C@@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845796 GG On-Demand Anodyne KCNA5 22 44 Cc1cc(NC(=O)NC[C@@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845796 GG On-Demand Anodyne NAMPT 58 38 Cc1cc(NC(=O)NC[C@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845797 GG On-Demand Anodyne ADRB3 27 40 Cc1cc(NC(=O)NC[C@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845797 GG On-Demand Anodyne KCNA5 22 44 Cc1cc(NC(=O)NC[C@H](c2cccnc2)C(C)C)cc(S(C)(=O)=O)c1 ZINC000880845797 GG On-Demand Anodyne NAMPT 58 38 CC[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880845823 DF On-Demand Anodyne EPHX2 20 40 COc1ccccc1C[C@H](C)N(C)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880845885 GH On-Demand Anodyne NPY5R 33 43 COc1ccccc1C[C@@H](C)N(C)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880845887 GH On-Demand Anodyne NPY5R 33 43 CCC(F)(F)C(C)(C)CNC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880845914 GF On-Demand Anodyne CACNA1G 33 42 Cc1cc(NC(=O)NCCCn2cccn2)cc(S(C)(=O)=O)c1 ZINC000880845921 ED On-Demand Anodyne CCR3 19 42 CCN(CC)C(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880845931 GF On-Demand Anodyne EPHX2 23 41 Cc1cc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880845941 GE On-Demand Anodyne CCR3 20 41 Cc1cc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880845941 GE On-Demand Anodyne EPHX2 40 43 Cc1cc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880845941 GE On-Demand Anodyne CXCR3 19 45 Cc1cc(NC(=O)NCCc2ccc3c(c2)OCO3)cc(S(C)(=O)=O)c1 ZINC000880845956 GE On-Demand Anodyne BMP1 57 39 Cc1cc(NC(=O)NCCN2CCc3ccccc3C2)cc(S(C)(=O)=O)c1 ZINC000880845998 GF On-Demand Anodyne HTR7 15 46 Cc1cc(NC(=O)NCCN2CCc3ccccc3C2)cc(S(C)(=O)=O)c1 ZINC000880845998 GF On-Demand Anodyne CCR3 26 44 Cc1cc(NC(=O)NCCN2CCc3ccccc3C2)cc(S(C)(=O)=O)c1 ZINC000880845998 GF On-Demand Anodyne AKR1C3 40 42 Cc1cc(NC(=O)NCCN2CCc3ccccc3C2)cc(S(C)(=O)=O)c1 ZINC000880845998 GF On-Demand Anodyne NOD2 43 37 C=CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846012 GH On-Demand Mild BMP1 44 41 Cc1cc(NC(=O)NC[C@H]2COc3ccccc3O2)cc(S(C)(=O)=O)c1 ZINC000880846027 GE On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)NC[C@@H]2COc3ccccc3O2)cc(S(C)(=O)=O)c1 ZINC000880846029 GE On-Demand Anodyne LPL 42 32 CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846051 BD On-Demand Anodyne SMG1 50 33 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c(OC)c1 ZINC000880846065 GG On-Demand Anodyne PDGFRB 23 45 Cc1cc(NC(=O)NCCC2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880846077 DG On-Demand Anodyne CCR3 30 43 Cc1cc(NC(=O)NCCC2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880846077 DG On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)Nc2ccccc2O[C@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880846128 GG On-Demand Anodyne LPL 58 37 Cc1cc(NC(=O)Nc2ccccc2O[C@@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880846129 GG On-Demand Anodyne LPL 58 37 Cc1cc(NC(=O)N[C@H]2CCN(C)[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880846138 EE On-Demand Anodyne EPHX2 29 40 Cc1cc(NC(=O)N[C@H]2CCN(C)[C@@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880846140 EE On-Demand Anodyne EPHX2 29 40 Cc1cc(NC(=O)NCCCCn2ccnc2C)cc(S(C)(=O)=O)c1 ZINC000880846145 FF On-Demand Anodyne CCR3 19 42 Cc1cc(NC(=O)NCC[C@H](O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846154 FF On-Demand Anodyne LPL 41 32 Cc1cc(NC(=O)NCC[C@@H](O)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846155 FF On-Demand Anodyne LPL 41 32 Cc1cc(NC(=O)N[C@H](C)COCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846203 GG On-Demand Anodyne CTSB 39 41 Cc1cc(NC(=O)N[C@H](C)COCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846203 GG On-Demand Anodyne CAPN2 51 39 COC[C@H](Cc1ccccc1)NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846209 GF On-Demand Anodyne CAPN2 45 33 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846210 GF On-Demand Anodyne CAPN2 45 33 C=CCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846213 FE On-Demand Mild EPHX2 33 43 C=CCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846213 FE On-Demand Mild CXCR3 20 42 Cc1cc(NC(=O)N[C@H]2CCCOc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880846233 FG On-Demand Anodyne BDKRB1 16 40 CC[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846251 EG On-Demand Anodyne EPHX2 16 41 CC[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846252 EG On-Demand Anodyne EPHX2 16 41 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c(C)c1 ZINC000880846260 GG On-Demand Anodyne LPL 57 38 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c(C)c1 ZINC000880846260 GG On-Demand Anodyne CA1 27 42 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c(C)c1 ZINC000880846260 GG On-Demand Anodyne CA12 15 50 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c(C)c1 ZINC000880846260 GG On-Demand Anodyne CA9 15 47 Cc1cc(NC(=O)NC[C@H]2CN(C)CCN2C)cc(S(C)(=O)=O)c1 ZINC000880846269 FC On-Demand Anodyne CCR3 25 40 Cc1cc(NC(=O)NC[C@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880846272 GE On-Demand Anodyne CCR3 37 43 Cc1cc(NC(=O)NC[C@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880846272 GE On-Demand Anodyne CACNA1I 61 38 Cc1cc(NC(=O)NC[C@@H]2CN(C)CCN2C)cc(S(C)(=O)=O)c1 ZINC000880846273 FC On-Demand Anodyne CCR3 25 40 Cc1cc(NC(=O)NC[C@@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880846276 GE On-Demand Anodyne CCR3 37 43 Cc1cc(NC(=O)NC[C@@H]2CCN(CC(F)(F)F)C2)cc(S(C)(=O)=O)c1 ZINC000880846276 GE On-Demand Anodyne CACNA1I 61 38 Cc1cc(NC(=O)NCCCc2ccc(O)cc2)cc(S(C)(=O)=O)c1 ZINC000880846302 FF On-Demand Anodyne CCR3 24 43 Cc1cc(NC(=O)NCCn2c(C)nc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880846307 GF On-Demand Anodyne ALDH3A1 40 38 COc1ccc(OC)c([C@H](C)NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880846314 GG On-Demand Anodyne CA1 16 40 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846316 GG On-Demand Anodyne BMP1 59 43 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846316 GG On-Demand Anodyne MMP13 31 41 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846316 GG On-Demand Anodyne ROCK2 19 44 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846316 GG On-Demand Anodyne MMP9 33 40 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846316 GG On-Demand Anodyne MMP1 34 41 Cc1cc(NC(=O)NCCC[S@](C)=O)cc(S(C)(=O)=O)c1 ZINC000880846322 ED On-Demand Anodyne CCR3 18 41 Cc1cc(NC(=O)NCCC[S@@](C)=O)cc(S(C)(=O)=O)c1 ZINC000880846324 ED On-Demand Anodyne CCR3 18 41 CC(=O)OC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846325 FD On-Demand Anodyne EPHX2 15 41 Cc1cc(NC(=O)NC[C@@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846353 GG On-Demand Anodyne LPL 44 36 Cc1cc(NC(=O)NC[C@@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846353 GG On-Demand Anodyne CCR3 38 41 Cc1cc(NC(=O)NC[C@@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846353 GG On-Demand Anodyne NAMPT 30 41 Cc1cc(NC(=O)NC[C@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846355 GG On-Demand Anodyne LPL 44 36 Cc1cc(NC(=O)NC[C@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846355 GG On-Demand Anodyne CCR3 38 41 Cc1cc(NC(=O)NC[C@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880846355 GG On-Demand Anodyne NAMPT 30 41 Cc1cc(NC(=O)N[C@H]2CCN(C(=O)C3CCCC3)C2)cc(S(C)(=O)=O)c1 ZINC000880846364 GE On-Demand Anodyne EPHX2 46 43 Cc1cc(NC(=O)NCCN(C)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846369 GF On-Demand Anodyne LIMK2 27 42 Cc1cc(NC(=O)N[C@H]2CCCOCC2)cc(S(C)(=O)=O)c1 ZINC000880846388 EE On-Demand Anodyne EPHX2 26 40 CCONC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846403 CD On-Demand Anodyne MTCA1 15 46 COCCOc1ccc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880846404 GF On-Demand Anodyne CA1 19 48 COCCOc1ccc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880846404 GF On-Demand Anodyne CA12 15 48 COCCOc1ccc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880846404 GF On-Demand Anodyne PRMT3 18 45 CCC1(CO)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846439 FE On-Demand Anodyne S1PR2 27 45 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846444 GI On-Demand Anodyne TRPM8 15 56 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846447 GI On-Demand Anodyne TRPM8 15 56 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846464 GE On-Demand Anodyne EPHX2 24 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846466 GE On-Demand Anodyne EPHX2 24 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846468 GE On-Demand Anodyne EPHX2 24 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846470 GE On-Demand Anodyne EPHX2 24 40 Cc1cc(NC(=O)N[C@H](C)CN2CCC[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880846488 FF On-Demand Anodyne CCR3 70 40 Cc1cc(NC(=O)NCCc2ccncc2)cc(S(C)(=O)=O)c1 ZINC000880846491 EE On-Demand Anodyne CA5B 17 44 Cc1cc(NC(=O)NCCc2ccncc2)cc(S(C)(=O)=O)c1 ZINC000880846491 EE On-Demand Anodyne CA5A 15 44 Cc1cc(NC(=O)NCCc2ccncc2)cc(S(C)(=O)=O)c1 ZINC000880846491 EE On-Demand Anodyne CA9 15 41 Cc1cc(NC(=O)NCCc2ccncc2)cc(S(C)(=O)=O)c1 ZINC000880846491 EE On-Demand Anodyne PRMT3 17 41 Cc1cc(NC(=O)NCCc2ccncc2)cc(S(C)(=O)=O)c1 ZINC000880846491 EE On-Demand Anodyne NAMPT 43 42 Cc1cc(NC(=O)N[C@H](C)CN2CCC[C@@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880846492 FF On-Demand Anodyne CCR3 70 40 COCC1(O)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846506 FD On-Demand Anodyne S1PR2 31 49 Cc1cc(NC(=O)NCc2c(C)cccc2C)cc(S(C)(=O)=O)c1 ZINC000880846508 EG On-Demand Anodyne NAMPT 34 40 Cc1cc(NC(=O)N[C@H]2CN(C)Cc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880846510 FF On-Demand Anodyne CCKAR 24 42 Cc1cc(NC(=O)N[C@H]2CN(C)Cc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880846510 FF On-Demand Anodyne CCKBR 34 42 CCC1(O)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846540 EE On-Demand Anodyne S1PR2 32 51 Cc1cc(NC(=O)NCCC(=O)N2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880846615 FD On-Demand Anodyne LPL 44 35 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846675 GC On-Demand Anodyne ACOX1 48 33 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846675 GC On-Demand Anodyne ABCB1 16 44 Cc1cc(NC(=O)NCCCNc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846699 FG On-Demand Anodyne CCR3 32 46 Cc1cc(NC(=O)NCCCNc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846699 FG On-Demand Anodyne FBP1 15 42 Cc1cc(NC(=O)NCCCCN2CCC[C@H]2CO)cc(S(C)(=O)=O)c1 ZINC000880846704 GD On-Demand Anodyne CCR3 37 45 Cc1cc(NC(=O)NCCCCN2CCC[C@@H]2CO)cc(S(C)(=O)=O)c1 ZINC000880846705 GD On-Demand Anodyne CCR3 37 45 Cc1cc(NC(=O)NCC2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880846708 DF On-Demand Anodyne CCR3 19 40 CCC(F)(F)C(C)(C)CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880846714 FH On-Demand Anodyne KCNQ2 59 36 CCC(F)(F)C(C)(C)CNC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880846716 EH On-Demand Anodyne MPO 53 38 Cc1cc(NC(=O)N[C@H](CN(C)C)c2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880846725 GF On-Demand Anodyne LPL 42 33 Cc1cc(NC(=O)NC[C@H](O)C2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880846731 FE On-Demand Anodyne PRMT3 33 48 Cc1cc(NC(=O)NC[C@@H](O)C2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880846732 FE On-Demand Anodyne PRMT3 33 48 COC(=O)c1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880846750 GF On-Demand Anodyne LIMK2 22 40 Cc1cc(NC(=O)NCc2ccc(C)cc2C)cc(S(C)(=O)=O)c1 ZINC000880846769 EG On-Demand Anodyne NAMPT 23 41 CC(=O)N(C)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846774 FD On-Demand Anodyne EPHX2 15 43 Cc1cc(NC(=O)NCCCOC2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880846779 FF On-Demand Anodyne CCR3 24 42 COCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846783 FD On-Demand Anodyne HTR4 34 40 COCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846783 FD On-Demand Anodyne CCR3 28 41 COCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846783 FD On-Demand Anodyne EPHX2 38 42 COCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880846783 FD On-Demand Anodyne CXCR3 20 41 COc1ncccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880846852 EE On-Demand Anodyne NAMPT 47 39 CCC(F)(F)C(C)(C)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880846861 EH On-Demand Anodyne NQO2 33 45 CCC(F)(F)C(C)(C)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880846861 EH On-Demand Anodyne MTNR1A 47 43 CCC(F)(F)C(C)(C)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880846861 EH On-Demand Anodyne MTNR1B 41 43 CCC(F)(F)C(C)(C)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880846862 EH On-Demand Anodyne NQO2 33 45 CCC(F)(F)C(C)(C)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880846862 EH On-Demand Anodyne MTNR1A 47 43 CCC(F)(F)C(C)(C)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880846862 EH On-Demand Anodyne MTNR1B 41 43 CC[C@]1(C)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880846875 DG On-Demand Anodyne S1PR2 26 41 Cc1cc(NC(=O)NCc2ccc(N3CC=CC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880846895 GG On-Demand Clean PRMT3 18 44 Cc1cc(NC(=O)NCc2ccc(N3CC=CC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880846895 GG On-Demand Clean NAMPT 59 43 Cc1cc(NC(=O)NCCN2CCC(N(C)C)CC2)cc(S(C)(=O)=O)c1 ZINC000880846898 GD On-Demand Anodyne CCR3 41 49 Cc1cc(NC(=O)NCCc2ccc(Cl)nc2)cc(S(C)(=O)=O)c1 ZINC000880846909 FF On-Demand Anodyne RAF1 17 40 Cc1cc(NC(=O)NCCc2ccc(Cl)nc2)cc(S(C)(=O)=O)c1 ZINC000880846909 FF On-Demand Anodyne NAMPT 18 47 Cc1cc(NC(=O)NCCCOCC2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880846931 GE On-Demand Anodyne CCR3 20 41 O=C(NC[C@@H]1CCO[C@H]1c1cn[nH]c1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880846948 FG On-Demand Anodyne PDE4D 15 43 Cc1cc(NC(=O)NCC2CCC2)cc(S(C)(=O)=O)c1 ZINC000880847017 CE On-Demand Anodyne CCR3 17 40 Cc1cc(NC(=O)NCc2ccc(C(=O)N(C)C)cc2)cc(S(C)(=O)=O)c1 ZINC000880847031 GE On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)NCc2ccc(C(=O)N(C)C)cc2)cc(S(C)(=O)=O)c1 ZINC000880847031 GE On-Demand Anodyne NAMPT 42 40 Cc1cc(NC(=O)NCCCCN2CCC(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880847042 GG On-Demand Anodyne CCR3 49 56 Cc1cc(NC(=O)NCc2ccc(N3CCCC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847046 GG On-Demand Clean PRMT3 17 43 Cc1cc(NC(=O)NCc2ccc(N3CCCC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847046 GG On-Demand Clean NAMPT 72 47 Cc1cc(NC(=O)N[C@H](C)COc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880847050 FF On-Demand Anodyne LPL 41 32 CCN1CC[C@H](CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847051 ED On-Demand Anodyne CCR3 40 44 CCN1CC[C@H](CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847051 ED On-Demand Anodyne CACNA1I 47 34 Cc1cc(NC(=O)NCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847068 EE On-Demand Anodyne HRH2 24 40 Cc1cc(NC(=O)NCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847068 EE On-Demand Anodyne CCR3 34 46 Cc1cc(NC(=O)NCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847068 EE On-Demand Anodyne EPHX2 16 40 COCc1ccccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880847084 FF On-Demand Anodyne NAMPT 26 45 Cc1cc(NC(=O)N[C@H](C)CNc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880847122 FG On-Demand Anodyne LPL 47 37 CC[C@H]1CCCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880847135 EH On-Demand Anodyne EPHX2 21 41 CC[C@@H]1CCCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880847136 EH On-Demand Anodyne EPHX2 21 41 CCCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847142 FF On-Demand Anodyne CCR3 30 45 CCCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847142 FF On-Demand Anodyne EPHX2 39 45 CCCCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847142 FF On-Demand Anodyne CXCR3 20 42 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847146 GG On-Demand Anodyne EPHX2 21 46 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847146 GG On-Demand Anodyne RBP4 39 42 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847147 GG On-Demand Anodyne EPHX2 21 46 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847147 GG On-Demand Anodyne RBP4 39 42 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne LPL 44 38 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne CA1 22 40 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne EPHX2 23 43 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne CA9 15 40 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne KCNK3 54 37 COCCCOc1cccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)c1 ZINC000880847149 GG On-Demand Anodyne KCNK9 57 33 Cc1cc(NC(=O)NC[C@@H](CO)Cc2ccc(F)cc2)cc(S(C)(=O)=O)c1 ZINC000880847173 GF On-Demand Anodyne CCR3 27 42 Cc1cc(NC(=O)NC[C@H](CO)Cc2ccc(F)cc2)cc(S(C)(=O)=O)c1 ZINC000880847174 GF On-Demand Anodyne CCR3 27 42 Cc1cc(NC(=O)N[C@H](CO)c2ccccc2C)cc(S(C)(=O)=O)c1 ZINC000880847189 FF On-Demand Anodyne CTSA 43 33 COC(=O)CCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847210 GF On-Demand Anodyne ST14 22 40 COC(=O)CCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847210 GF On-Demand Anodyne GPR119 26 40 CCOC(=O)N1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847227 GE On-Demand Anodyne S1PR2 25 40 CCOC(=O)N1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847227 GE On-Demand Anodyne TGM2 42 46 CCOC(=O)N1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847227 GE On-Demand Anodyne F13A1 57 46 Cc1cc(NC(=O)NCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880847235 EE On-Demand Anodyne ADRB3 22 44 Cc1cc(NC(=O)NCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880847235 EE On-Demand Anodyne TBXAS1 52 43 Cc1cc(NC(=O)NCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880847235 EE On-Demand Anodyne PTAFR 20 42 Cc1cc(NC(=O)NCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880847235 EE On-Demand Anodyne CYP2C9 16 47 Cc1cc(NC(=O)NCCc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880847235 EE On-Demand Anodyne NAMPT 78 57 Cc1cc(NC(=O)N[C@H]2CCN3CCC[C@@H]3C2)cc(S(C)(=O)=O)c1 ZINC000880847245 FE On-Demand Anodyne EPHX2 25 40 Cc1cc(NC(=O)N[C@H]2CCN3CCC[C@H]3C2)cc(S(C)(=O)=O)c1 ZINC000880847248 FE On-Demand Anodyne EPHX2 25 40 Cc1cc(NC(=O)NCc2ccc(N(C)C)nc2)cc(S(C)(=O)=O)c1 ZINC000880847249 FE On-Demand Anodyne PRMT3 18 45 Cc1cc(NC(=O)NCc2ccc(N(C)C)nc2)cc(S(C)(=O)=O)c1 ZINC000880847249 FE On-Demand Anodyne NAMPT 51 47 Cc1cc(NC(=O)NCCCCN2CCCC[C@@H]2C)cc(S(C)(=O)=O)c1 ZINC000880847255 GG On-Demand Anodyne CCR3 35 45 Cc1cc(NC(=O)NCCCCN2CCCC[C@H]2C)cc(S(C)(=O)=O)c1 ZINC000880847256 GG On-Demand Anodyne CCR3 35 45 Cc1cc(NC(=O)NCCCN2C[C@H](C)O[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880847267 GE On-Demand Anodyne CCR3 34 48 Cc1cc(NC(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880847268 GE On-Demand Anodyne CCR3 34 48 Cc1cc(NC(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880847269 GE On-Demand Anodyne CCR3 34 48 Cc1cc(NC(=O)NCCCCN2CCC[C@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880847306 GG On-Demand Anodyne CCR3 56 49 Cc1cc(NC(=O)NCCCCN2CCC[C@@H](C)C2)cc(S(C)(=O)=O)c1 ZINC000880847307 GG On-Demand Anodyne CCR3 56 49 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne HRH2 16 43 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne CA1 22 41 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne MTNR1A 33 40 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne MTNR1B 23 40 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne CA12 17 41 COc1ccc(OCCNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880847311 GF On-Demand Anodyne CA9 21 40 Cc1cc(NC(=O)N[C@H](C)CCc2cccn2C)cc(S(C)(=O)=O)c1 ZINC000880847360 FF On-Demand Anodyne CCR3 45 36 Cc1cc(NC(=O)NCCCOC[C@@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880847368 FD On-Demand Anodyne CCR3 17 40 Cc1cc(NC(=O)NCCCOC[C@H]2CCOC2)cc(S(C)(=O)=O)c1 ZINC000880847369 FD On-Demand Anodyne CCR3 17 40 Cc1cc(NC(=O)N[C@H]2CCCC[C@@H]2CO)cc(S(C)(=O)=O)c1 ZINC000880847375 EE On-Demand Anodyne CCR3 26 41 Cc1cc(NC(=O)N[C@H]2CCCC[C@H]2CO)cc(S(C)(=O)=O)c1 ZINC000880847378 EE On-Demand Anodyne CCR3 26 41 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847412 ED On-Demand Anodyne EPHX2 27 41 COC(=O)[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847413 ED On-Demand Anodyne EPHX2 27 41 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847414 FD On-Demand Anodyne EPHX2 18 41 CC(=O)N[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847415 FD On-Demand Anodyne EPHX2 18 41 Cc1cc(NC(=O)NCCN2CCCC[C@@H]2C)cc(S(C)(=O)=O)c1 ZINC000880847476 FE On-Demand Anodyne HRH3 23 40 Cc1cc(NC(=O)NCCN2CCCC[C@@H]2C)cc(S(C)(=O)=O)c1 ZINC000880847476 FE On-Demand Anodyne CCR3 29 42 CC(=O)NCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847505 FD On-Demand Anodyne EPHX2 21 41 CC(=O)NCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847505 FD On-Demand Anodyne CACNA1I 48 33 Cc1cc(NC(=O)N[C@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880847511 ED On-Demand Anodyne EPHX2 34 40 Cc1cc(NC(=O)NCCN2CCC(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880847512 FE On-Demand Anodyne CCR3 46 51 Cc1cc(NC(=O)NCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880847513 EE On-Demand Anodyne MAPK9 20 40 Cc1cc(NC(=O)NCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880847513 EE On-Demand Anodyne PRMT3 19 48 Cc1cc(NC(=O)NCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880847513 EE On-Demand Anodyne NAMPT 68 61 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880847517 FF On-Demand Anodyne MMP13 19 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880847517 FF On-Demand Anodyne MMP3 25 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880847517 FF On-Demand Anodyne MMP9 21 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880847517 FF On-Demand Anodyne MMP1 23 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1)CC2 ZINC000880847517 FF On-Demand Anodyne AKR1C3 26 45 Cc1cc(NC(=O)NCCCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880847530 FE On-Demand Anodyne TBXAS1 42 51 Cc1cc(NC(=O)NCCCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880847530 FE On-Demand Anodyne QPCT 82 58 CCCOc1ncccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880847536 GF On-Demand Anodyne NAMPT 37 49 Cc1cc(NC(=O)NCCN2CCc3sccc3C2)cc(S(C)(=O)=O)c1 ZINC000880847537 GF On-Demand Anodyne CCR3 16 40 Cc1cc(NC(=O)NCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880847540 CD On-Demand Anodyne CCR3 15 41 Cc1cc(NC(=O)NCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880847540 CD On-Demand Anodyne CACNA1I 45 33 Cc1cc(NC(=O)NCCC(=O)N2CCCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847557 GE On-Demand Anodyne LPL 44 35 Cc1cc(NC(=O)NCc2ccc(N3CCCC3)nc2)cc(S(C)(=O)=O)c1 ZINC000880847575 GF On-Demand Anodyne PRMT3 24 42 Cc1cc(NC(=O)NCc2ccc(N3CCCC3)nc2)cc(S(C)(=O)=O)c1 ZINC000880847575 GF On-Demand Anodyne NAMPT 81 46 Cc1cc(NC(=O)NCCN2CCCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847602 FE On-Demand Anodyne HRH2 24 40 Cc1cc(NC(=O)NCCN2CCCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847602 FE On-Demand Anodyne CCR3 34 46 Cc1cc(NC(=O)NCCN2CCCCCC2)cc(S(C)(=O)=O)c1 ZINC000880847602 FE On-Demand Anodyne EPHX2 16 40 COc1ccc2c(c1)CC[C@H](C(=O)NNC(=O)[C@@H]1CCCN(C(C)=O)[C@@H]1C)C2 ZINC000880847624 GD On-Demand Reactive MTNR1B 26 41 CCOC[C@H]1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847646 EE On-Demand Anodyne GPR119 21 40 Cc1cc(NC(=O)NC[C@@H]2CCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880847745 FE On-Demand Anodyne CCR3 40 42 Cc1cc(NC(=O)NC[C@@H]2CCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880847745 FE On-Demand Anodyne CACNA1I 50 37 Cc1cc(NC(=O)NC[C@H]2CCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880847746 FE On-Demand Anodyne CCR3 40 42 Cc1cc(NC(=O)NC[C@H]2CCN(CC(C)C)C2)cc(S(C)(=O)=O)c1 ZINC000880847746 FE On-Demand Anodyne CACNA1I 50 37 Cc1cc(NC(=O)NCCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880847756 CE On-Demand Anodyne CCR3 26 44 Cc1cc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847761 GG On-Demand Anodyne CA1 34 48 Cc1cc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847761 GG On-Demand Anodyne CA12 22 48 Cc1cc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847761 GG On-Demand Anodyne CA9 21 48 Cc1cc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847761 GG On-Demand Anodyne MTCA1 27 45 Cc1cc(NC(=O)Nc2ccc(O[C@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847761 GG On-Demand Anodyne P96878_MYCTU 32 45 Cc1cc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847762 GG On-Demand Anodyne CA1 34 48 Cc1cc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847762 GG On-Demand Anodyne CA12 22 48 Cc1cc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847762 GG On-Demand Anodyne CA9 21 48 Cc1cc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847762 GG On-Demand Anodyne MTCA1 27 45 Cc1cc(NC(=O)Nc2ccc(O[C@@H]3CCOC3)cc2)cc(S(C)(=O)=O)c1 ZINC000880847762 GG On-Demand Anodyne P96878_MYCTU 32 45 Cc1cc(NC(=O)NCC2(CO)CC2)cc(S(C)(=O)=O)c1 ZINC000880847787 DD On-Demand Anodyne NAMPT 27 40 CCC1(CC)CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847798 EG On-Demand Anodyne S1PR2 26 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCO[C@H]1c1cn[nH]c1)C2 ZINC000880847884 FE On-Demand Anodyne ROCK2 51 40 Cc1cc(NC(=O)NCCOc2ncccc2Cl)cc(S(C)(=O)=O)c1 ZINC000880847890 GF On-Demand Anodyne NAMPT 28 41 Cc1cc(NC(=O)Nc2cnn(C)c2C)cc(S(C)(=O)=O)c1 ZINC000880847907 DE On-Demand Anodyne LPL 49 33 CC[C@H](O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847908 FD On-Demand Anodyne S1PR2 26 42 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847909 FD On-Demand Anodyne S1PR2 26 42 Cc1cc(NC(=O)NCCCc2cnn(C)c2)cc(S(C)(=O)=O)c1 ZINC000880847937 FD On-Demand Anodyne CCR3 27 43 COC[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880847943 EE On-Demand Anodyne CASP7 43 34 COCC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847952 EE On-Demand Anodyne EPHX2 17 41 C=C(C)CN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847954 FF On-Demand Mild EPHX2 34 43 C=C(C)CN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880847954 FF On-Demand Mild CXCR3 21 44 Cc1cc(NC(=O)NC[C@@H](O)C2CC2)cc(S(C)(=O)=O)c1 ZINC000880847955 DD On-Demand Anodyne PRMT3 18 41 Cc1cc(NC(=O)NC[C@H](O)C2CC2)cc(S(C)(=O)=O)c1 ZINC000880847956 DD On-Demand Anodyne PRMT3 18 41 Cc1cc(NC(=O)NCC[S@@](=O)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880847994 GE On-Demand Anodyne NAMPT 20 40 Cc1cc(NC(=O)NCC[S@](=O)Cc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880847995 GE On-Demand Anodyne NAMPT 20 40 Cc1cc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc(S(C)(=O)=O)c1 ZINC000880848042 FE On-Demand Anodyne CCR3 33 40 Cc1cc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc(S(C)(=O)=O)c1 ZINC000880848042 FE On-Demand Anodyne EPHX2 31 41 Cc1cc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc(S(C)(=O)=O)c1 ZINC000880848042 FE On-Demand Anodyne CXCR3 17 48 C=CCNC(=O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848044 GC On-Demand Mild TGM2 42 39 C=CCNC(=O)CN1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848044 GC On-Demand Mild F13A1 59 39 Cc1cc(NC(=O)NCCCn2cnc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848080 GF On-Demand Anodyne CCR3 15 41 Cc1cc(NC(=O)NCCCn2cnc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848080 GF On-Demand Anodyne NR1I2 50 40 Cc1cc(NC(=O)NCCCn2cnc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848080 GF On-Demand Anodyne QPCT 50 38 Cc1cc(NC(=O)NCC2(N3CCCC3)CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880848081 GE On-Demand Anodyne NAMPT 17 41 CCOc1cc(CNC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)ccc1OC ZINC000880848089 GG On-Demand Anodyne ROCK2 19 48 Cc1cc(NC(=O)NC[C@@H]2CCOc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848111 FG On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)NC[C@H]2CCOc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848112 FG On-Demand Anodyne LPL 42 32 Cc1cc(NC(=O)N[C@H]2CCOc3ccccc32)cc(S(C)(=O)=O)c1 ZINC000880848121 FG On-Demand Anodyne BDKRB1 24 45 CC[C@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848131 DG On-Demand Anodyne EPHX2 19 42 CC[C@@H]1CCCCN1C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848132 DG On-Demand Anodyne EPHX2 19 42 CCOC(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848140 FE On-Demand Anodyne EPHX2 26 40 Cc1cc(NC(=O)NCCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880848165 FD On-Demand Anodyne CASR 17 42 Cc1cc(NC(=O)NCCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880848165 FD On-Demand Anodyne CCR3 38 51 Cc1cc(NC(=O)NCCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880848165 FD On-Demand Anodyne EPHX2 28 48 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne BMP1 86 39 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP13 51 41 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP2 26 41 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP3 50 41 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP9 46 38 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP7 33 41 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne MMP1 51 41 COc1ccc(CN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C2CC2)cc1 ZINC000880848166 GH On-Demand Anodyne GIPR 38 42 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne CA1 24 46 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne CCR3 30 44 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne FBP1 15 42 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne CA12 16 46 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne CA9 15 46 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne AMP1_PLAFQ 21 40 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne P96878_MYCTU 15 40 Cc1cc(NC(=O)NCCCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848175 EG On-Demand Anodyne NAMPT 33 40 COC(=O)c1cc(NC(=O)N[C@@H]2CCN(C(C)=O)C2)cc2ccccc12 ZINC000880848179 FE On-Demand Anodyne EPHX2 44 48 COC(=O)c1cc(NC(=O)N[C@@H]2CCN(C(C)=O)C2)cc2ccccc12 ZINC000880848179 FE On-Demand Anodyne CCR8 75 38 COc1ccc([C@@H]2CCCN2C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848184 GH On-Demand Anodyne MMP1 35 41 COC(=O)c1cc(NC(=O)N2CC[C@H](O)C(F)(F)C2)cc2ccccc12 ZINC000880848190 FF On-Demand Anodyne CCR8 48 34 COC(=O)c1cc(NC(=O)N2CC[C@@H](O)C(F)(F)C2)cc2ccccc12 ZINC000880848191 FF On-Demand Anodyne CCR8 48 34 Cc1cc(NC(=O)NCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848201 FE On-Demand Anodyne HRH2 34 44 Cc1cc(NC(=O)NCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848201 FE On-Demand Anodyne HTR2A 17 41 Cc1cc(NC(=O)NCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848201 FE On-Demand Anodyne CCR3 44 52 Cc1cc(NC(=O)NCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848201 FE On-Demand Anodyne CHRNA7 21 51 COC(=O)c1cc(NC(=O)N2CCC(C(C)(C)O)CC2)cc2ccccc12 ZINC000880848202 FH On-Demand Anodyne RBP4 20 42 COC(=O)c1cc(NC(=O)N2CCC(C(C)(C)O)CC2)cc2ccccc12 ZINC000880848202 FH On-Demand Anodyne CCR8 51 33 CCN(Cc1ccccc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848207 EG On-Demand Anodyne LIMK2 27 46 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne CA2 23 52 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne LPL 50 37 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne CA1 55 52 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne EPHX2 15 47 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne CA12 39 52 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne CA9 40 52 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne NCE103 20 47 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne MTCA1 42 50 COCCOc1ccc(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1 ZINC000880848219 GG On-Demand Anodyne P96878_MYCTU 51 50 Cc1cc(NC(=O)NCCCCOCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848233 GH On-Demand Anodyne CA1 19 40 Cc1cc(NC(=O)NCCCCOCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848233 GH On-Demand Anodyne CCR3 25 42 Cc1cc(NC(=O)NCCCCOCc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848233 GH On-Demand Anodyne FBP1 15 40 Cc1cc(NC(=O)NCCOc2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880848242 ED On-Demand Anodyne NAMPT 58 43 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880848255 FF On-Demand Anodyne EPHX2 43 42 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccc3)C2=O)cc(S(C)(=O)=O)c1 ZINC000880848258 GE On-Demand Anodyne CCKAR 43 43 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccc3)C2=O)cc(S(C)(=O)=O)c1 ZINC000880848258 GE On-Demand Anodyne CCKBR 63 39 Cc1cc(NC(=O)N[C@H]2CCN(c3ccccc3)C2=O)cc(S(C)(=O)=O)c1 ZINC000880848258 GE On-Demand Anodyne EPHX2 24 40 Cc1cc(NC(=O)NCCCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848266 GG On-Demand Anodyne HRH2 32 43 Cc1cc(NC(=O)NCCCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848266 GG On-Demand Anodyne HTR2A 15 40 Cc1cc(NC(=O)NCCCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848266 GG On-Demand Anodyne CCR3 41 51 Cc1cc(NC(=O)NCCCCCN2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848266 GG On-Demand Anodyne CHRNA7 20 52 COCCN(Cc1cccnc1)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848271 GE On-Demand Anodyne NAMPT 40 36 Cc1cc(NC(=O)NCCCNC2CCCCC2)cc(S(C)(=O)=O)c1 ZINC000880848272 FF On-Demand Anodyne CCR3 25 42 Cc1cc(NC(=O)NCCCCN2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848303 GD On-Demand Anodyne HTR2A 20 41 Cc1cc(NC(=O)NCCCCN2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848303 GD On-Demand Anodyne DRD3 29 42 Cc1cc(NC(=O)NCCCCN2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848303 GD On-Demand Anodyne CCR3 39 52 Cc1cc(NC(=O)NCCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880848312 EE On-Demand Anodyne RAF1 17 41 Cc1cc(NC(=O)NCCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880848312 EE On-Demand Anodyne PRMT3 17 42 Cc1cc(NC(=O)NCCc2ccc(C)nc2)cc(S(C)(=O)=O)c1 ZINC000880848312 EE On-Demand Anodyne NAMPT 33 48 COC(=O)c1cc(NC(=O)N2CCC(c3ccon3)CC2)cc2ccccc12 ZINC000880848333 GI On-Demand Anodyne RBP4 15 41 COC(=O)c1cc(NC(=O)N2CCC(c3ccon3)CC2)cc2ccccc12 ZINC000880848333 GI On-Demand Anodyne SMO 39 45 Cc1cc(NC(=O)NCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880848344 DD On-Demand Anodyne TBXAS1 36 43 Cc1cc(NC(=O)NCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880848344 DD On-Demand Anodyne QPCT 40 52 COC(=O)c1cc(NC(=O)N2CCOC3(CCN(C)CC3)C2)cc2ccccc12 ZINC000880848355 GF On-Demand Anodyne EPHX2 27 46 Cc1cc(NC(=O)NCCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880848356 ED On-Demand Anodyne TBXAS1 43 49 Cc1cc(NC(=O)NCCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880848356 ED On-Demand Anodyne HMOX2 44 33 Cc1cc(NC(=O)NCCCn2ccnc2)cc(S(C)(=O)=O)c1 ZINC000880848356 ED On-Demand Anodyne QPCT 87 59 COC(=O)c1cc(NC(=O)N2CCC(O)(CO)CC2)cc2ccccc12 ZINC000880848371 FD On-Demand Anodyne S1PR2 29 45 Cc1cc(NC(=O)NC[C@H](c2ccccc2)N(C)C)cc(S(C)(=O)=O)c1 ZINC000880848375 GF On-Demand Anodyne LPL 43 34 Cc1cc(NC(=O)NC[C@@H](c2ccccc2)N(C)C)cc(S(C)(=O)=O)c1 ZINC000880848376 GF On-Demand Anodyne LPL 43 34 COC(=O)c1cc(NC(=O)N2CCC[C@H](CF)C2)cc2ccccc12 ZINC000880848392 EH On-Demand Anodyne CCR3 27 43 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CF)C2)cc2ccccc12 ZINC000880848393 EH On-Demand Anodyne CCR3 27 43 COC(=O)c1cc(NC(=O)N(C)[C@H](C)CCO)cc2ccccc12 ZINC000880848401 EF On-Demand Anodyne NPY5R 34 43 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)CCO)cc2ccccc12 ZINC000880848402 EF On-Demand Anodyne NPY5R 34 43 COC(=O)[C@@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848417 EE On-Demand Anodyne JAK3 17 44 COC(=O)[C@@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848417 EE On-Demand Anodyne TYK2 20 44 COC(=O)[C@@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848417 EE On-Demand Anodyne HCN1 40 31 COC(=O)[C@@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848417 EE On-Demand Anodyne HCN4 40 31 COC(=O)[C@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848419 EE On-Demand Anodyne JAK3 17 44 COC(=O)[C@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848419 EE On-Demand Anodyne TYK2 20 44 COC(=O)[C@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848419 EE On-Demand Anodyne HCN1 40 31 COC(=O)[C@H](CNC(=O)c1cccn2nccc12)C1CCCCC1 ZINC000880848419 EE On-Demand Anodyne HCN4 40 31 COC(=O)c1cc(NC(=O)N2CC[C@@H](O)[C@@H](O)C2)cc2ccccc12 ZINC000880848421 ED On-Demand Anodyne CCR8 58 32 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880848452 GG On-Demand Anodyne MMP13 45 44 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880848452 GG On-Demand Anodyne MMP3 43 44 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880848452 GG On-Demand Anodyne MMP9 32 44 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880848452 GG On-Demand Anodyne EPHX2 21 42 COc1ccc([C@@H]2CCN(C(=O)Nc3cc(C)cc(S(C)(=O)=O)c3)C2)cc1 ZINC000880848452 GG On-Demand Anodyne MMP1 43 44 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880848474 GE On-Demand Anodyne EPHX2 23 42 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880848475 GE On-Demand Anodyne EPHX2 23 42 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848534 GG On-Demand Anodyne BMP1 65 40 COC(=O)c1cc(NC(=O)N2CCC[C@](CO)(OC)C2)cc2ccccc12 ZINC000880848584 FF On-Demand Anodyne EPHX2 24 42 COC(=O)c1cc(NC(=O)N2CCC[C@@](CO)(OC)C2)cc2ccccc12 ZINC000880848586 FF On-Demand Anodyne EPHX2 24 42 COC(=O)c1cc(NC(=O)N2CCC[C@H]2C(=O)N(C)C)cc2ccccc12 ZINC000880848593 FF On-Demand Anodyne AVPR2 17 43 COC(=O)c1cc(NC(=O)N2CCC[C@H]2C(=O)N(C)C)cc2ccccc12 ZINC000880848593 FF On-Demand Anodyne UL80 40 38 COC(=O)c1cc(NC(=O)N2CCC([C@@H](C)O)CC2)cc2ccccc12 ZINC000880848611 FG On-Demand Anodyne RBP4 15 40 COC(=O)c1cc(NC(=O)N2CCC([C@H](C)O)CC2)cc2ccccc12 ZINC000880848613 FG On-Demand Anodyne RBP4 15 40 CCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848624 EE On-Demand Anodyne EPHX2 45 48 CCN1CCC(NC(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848624 EE On-Demand Anodyne CXCR3 22 44 CCCO[C@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848658 FG On-Demand Anodyne GPR119 40 39 CCCO[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848659 FG On-Demand Anodyne GPR119 40 39 Cc1cc(NC(=O)NCCN2Cc3ccccc3C2)cc(S(C)(=O)=O)c1 ZINC000880848668 FF On-Demand Anodyne CCR3 25 45 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)C1 ZINC000880848675 FD On-Demand Anodyne EPHX2 27 42 Cc1cc(NC(=O)NC[C@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880848689 ED On-Demand Anodyne CCR3 52 42 Cc1cc(NC(=O)NC[C@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880848689 ED On-Demand Anodyne CACNA1I 49 33 Cc1cc(NC(=O)NC[C@@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880848690 ED On-Demand Anodyne CCR3 52 42 Cc1cc(NC(=O)NC[C@@H]2CCCN(C)C2)cc(S(C)(=O)=O)c1 ZINC000880848690 ED On-Demand Anodyne CACNA1I 49 33 Cc1cc(NC(=O)NCC2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848701 ED On-Demand Anodyne CCR3 39 44 Cc1cc(NC(=O)NCC2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848701 ED On-Demand Anodyne EPHX2 26 40 Cc1cc(NC(=O)NCC2CCN(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880848701 ED On-Demand Anodyne CACNA1I 56 36 CCOc1ccccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848705 FG On-Demand Anodyne CA1 15 41 CCOc1ccccc1CNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848705 FG On-Demand Anodyne NAMPT 24 46 Cc1cc(NC(=O)NCCN2CCSCC2)cc(S(C)(=O)=O)c1 ZINC000880848708 FD On-Demand Anodyne CCR3 28 46 Cc1cc(NC(=O)NCCCN2CCCCC2=O)cc(S(C)(=O)=O)c1 ZINC000880848715 FD On-Demand Anodyne CCR3 31 45 C#CCNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848736 CD On-Demand Mild MTCA1 21 46 C#CCNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880848736 CD On-Demand Mild P96878_MYCTU 27 46 CCCCNC(=O)C1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848737 GF On-Demand Anodyne EPHX2 31 46 Cc1cc(NC(=O)NC[C@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848750 FF On-Demand Anodyne CA1 37 40 Cc1cc(NC(=O)NC[C@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848750 FF On-Demand Anodyne CA12 16 40 Cc1cc(NC(=O)NC[C@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848750 FF On-Demand Anodyne CA9 16 40 Cc1cc(NC(=O)NC[C@@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848751 FF On-Demand Anodyne CA1 37 40 Cc1cc(NC(=O)NC[C@@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848751 FF On-Demand Anodyne CA12 16 40 Cc1cc(NC(=O)NC[C@@H](C)Oc2ccccc2)cc(S(C)(=O)=O)c1 ZINC000880848751 FF On-Demand Anodyne CA9 16 40 C=CC1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848763 DF On-Demand Mild F13A1 44 34 CCOC(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848777 FD On-Demand Anodyne P2RY12 39 40 CCOC(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848777 FD On-Demand Anodyne S1PR2 26 42 CCOC(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848777 FD On-Demand Anodyne TGM2 40 48 CCOC(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848777 FD On-Demand Anodyne F13A1 58 48 CCOC(=O)N1CCN(C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)CC1 ZINC000880848777 FD On-Demand Anodyne GPR119 23 41 COC(=O)c1cc(NC(=O)N2CC[C@H](CF)C2)cc2ccccc12 ZINC000880848793 EG On-Demand Anodyne CCR3 17 42 COC(=O)c1cc(NC(=O)N2CC[C@@H](CF)C2)cc2ccccc12 ZINC000880848794 EG On-Demand Anodyne CCR3 17 42 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1C)C2 ZINC000880848811 DF On-Demand Anodyne NQO2 34 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1C)C2 ZINC000880848811 DF On-Demand Anodyne MTNR1A 53 45 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1C)C2 ZINC000880848811 DF On-Demand Anodyne MTNR1B 42 39 COC(=O)c1cc(NC(=O)N2CCCc3n[nH]cc3C2)cc2ccccc12 ZINC000880848825 FG On-Demand Anodyne P2RY14 46 33 COC(=O)c1cc(NC(=O)N2CCCNC(=O)C2)cc2ccccc12 ZINC000880848841 ED On-Demand Anodyne P2RY14 45 32 COC(=O)c1cc(NC(=O)N2CCC3(COC3)C2)cc2ccccc12 ZINC000880848846 EF On-Demand Anodyne EPHX2 33 42 COC(=O)c1cc(NC(=O)N2CCC(F)(F)CC2)cc2ccccc12 ZINC000880848862 EH On-Demand Anodyne CACNA1H 52 37 COC(=O)c1cc(NC(=O)N2CCC(F)(F)CC2)cc2ccccc12 ZINC000880848862 EH On-Demand Anodyne NPY5R 29 40 COC(=O)c1cc(NC(=O)N2CCC3(CC2)COCCO3)cc2ccccc12 ZINC000880848863 GG On-Demand Anodyne NPY5R 19 40 Cc1cc(NC(=O)NCc2ccc(N(C)C)cc2)cc(S(C)(=O)=O)c1 ZINC000880848967 FF On-Demand Clean PRMT3 19 46 Cc1cc(NC(=O)NCc2ccc(N(C)C)cc2)cc(S(C)(=O)=O)c1 ZINC000880848967 FF On-Demand Clean NAMPT 42 40 COC(=O)c1cc(NC(=O)N2CCC3(CCNC3=O)CC2)cc2ccccc12 ZINC000880848970 GF On-Demand Anodyne CACNA1H 56 38 COC(=O)c1cc(NC(=O)N2CC[C@H]3CC[C@@H](C2)[S@@]3=O)cc2ccccc12 ZINC000880848976 GG On-Demand Anodyne CCR8 43 30 COC(=O)c1cc(NC(=O)N2CC[C@H]3CC[C@@H](C2)[S@]3=O)cc2ccccc12 ZINC000880848977 GG On-Demand Anodyne CCR8 43 30 COC(=O)c1cc(NC(=O)N2CCO[C@@]3(CCSC3)C2)cc2ccccc12 ZINC000880848978 GG On-Demand Anodyne EPHX2 22 41 COC(=O)c1cc(NC(=O)N2CCO[C@]3(CCSC3)C2)cc2ccccc12 ZINC000880848979 GG On-Demand Anodyne EPHX2 22 41 Cc1cc(NC(=O)NCCCOCC2CC2)cc(S(C)(=O)=O)c1 ZINC000880848984 EE On-Demand Anodyne CCR3 32 44 COC(=O)c1cc(NC(=O)N(C)CCNC(C)=O)cc2ccccc12 ZINC000880848988 EE On-Demand Anodyne NQO2 30 41 COC(=O)c1cc(NC(=O)N(C)CCNC(C)=O)cc2ccccc12 ZINC000880848988 EE On-Demand Anodyne MTNR1A 53 41 COC(=O)c1cc(NC(=O)N(C)CCNC(C)=O)cc2ccccc12 ZINC000880848988 EE On-Demand Anodyne MTNR1B 43 41 COC(=O)c1cc(NC(=O)N2CCN(c3nncn3C)CC2)cc2ccccc12 ZINC000880848997 GE On-Demand Anodyne PDGFRB 49 38 COC(=O)c1cc(NC(=O)N2CC[C@H]3C[C@@H]3C2)cc2ccccc12 ZINC000880848998 DH On-Demand Anodyne RBP4 47 33 COC(=O)c1cc(NC(=O)N2CC[C@H]3C[C@@H]3C2)cc2ccccc12 ZINC000880848998 DH On-Demand Anodyne CCR8 59 32 COC(=O)c1cc(NC(=O)N2CC[C@H]3C[C@H]3C2)cc2ccccc12 ZINC000880848999 DH On-Demand Anodyne RBP4 47 33 COC(=O)c1cc(NC(=O)N2CC[C@H]3C[C@H]3C2)cc2ccccc12 ZINC000880848999 DH On-Demand Anodyne CCR8 59 32 COC(=O)c1cc(NC(=O)N2CC[C@@H]3C[C@H]3C2)cc2ccccc12 ZINC000880849000 DH On-Demand Anodyne RBP4 47 33 COC(=O)c1cc(NC(=O)N2CC[C@@H]3C[C@H]3C2)cc2ccccc12 ZINC000880849000 DH On-Demand Anodyne CCR8 59 32 COC(=O)c1cc(NC(=O)N2CC[C@@H]3C[C@@H]3C2)cc2ccccc12 ZINC000880849001 DH On-Demand Anodyne RBP4 47 33 COC(=O)c1cc(NC(=O)N2CC[C@@H]3C[C@@H]3C2)cc2ccccc12 ZINC000880849001 DH On-Demand Anodyne CCR8 59 32 COC(=O)c1cc(NC(=O)NC2CCN([C@@H]3CCOC3)CC2)cc2ccccc12 ZINC000880849003 GG On-Demand Anodyne EPHX2 33 42 COC(=O)c1cc(NC(=O)NC2CCN([C@@H]3CCOC3)CC2)cc2ccccc12 ZINC000880849003 GG On-Demand Anodyne CXCR3 17 40 COC(=O)c1cc(NC(=O)NC2CCN([C@H]3CCOC3)CC2)cc2ccccc12 ZINC000880849004 GG On-Demand Anodyne EPHX2 33 42 COC(=O)c1cc(NC(=O)NC2CCN([C@H]3CCOC3)CC2)cc2ccccc12 ZINC000880849004 GG On-Demand Anodyne CXCR3 17 40 Cc1cc(NC(=O)N[C@H](C)c2ccc(C)o2)cc(S(C)(=O)=O)c1 ZINC000880849011 EG On-Demand Anodyne LPL 41 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849016 ED On-Demand Anodyne PAPA1_CARPA 44 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849016 ED On-Demand Anodyne REN 40 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849016 ED On-Demand Anodyne SCN10A 29 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849016 ED On-Demand Anodyne FPR1 46 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849017 ED On-Demand Anodyne PAPA1_CARPA 44 46 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849017 ED On-Demand Anodyne REN 40 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849017 ED On-Demand Anodyne SCN10A 29 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1cccnc1C ZINC000880849017 ED On-Demand Anodyne FPR1 46 37 COC(=O)c1cc(NC(=O)N[C@@H]2C[C@H](CO)C2)cc2ccccc12 ZINC000880849021 EF On-Demand Anodyne EPHX2 20 40 COC(=O)c1cc(NC(=O)NC2CC(CO)C2)cc2ccccc12 ZINC000880849022 EF On-Demand Anodyne EPHX2 20 40 Cc1cc(NC(=O)N[C@H](C)c2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880849062 EF On-Demand Anodyne KCNA5 19 42 Cc1cc(NC(=O)N[C@H](C)c2cccnc2)cc(S(C)(=O)=O)c1 ZINC000880849062 EF On-Demand Anodyne NAMPT 43 62 COC(=O)c1cc(NC(=O)N2CCC(C(C)=O)CC2)cc2ccccc12 ZINC000880849066 FG On-Demand Anodyne CCR8 41 32 Cc1cc(NC(=O)NCCCN2CCC(C)CC2)cc(S(C)(=O)=O)c1 ZINC000880849070 FF On-Demand Anodyne CCR3 52 57 COc1ccc(CN(C)C(=O)Nc2cc(C)cc(S(C)(=O)=O)c2)cc1OC ZINC000880849112 GG On-Demand Anodyne MT-ND1 18 43 Cc1cc(NC(=O)NCCc2ccccn2)cc(S(C)(=O)=O)c1 ZINC000880849116 EE On-Demand Anodyne NAMPT 23 42 CCCCCNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880849117 CF On-Demand Anodyne TBXA2R 15 43 CCCCCNC(=O)Nc1cc(C)cc(S(C)(=O)=O)c1 ZINC000880849117 CF On-Demand Anodyne ASAH1 49 31 COCC1CC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880849131 EG On-Demand Anodyne EPHX2 20 40 COC(=O)c1cc(NC(=O)N2CC[C@H]3[C@H](CCN3C)C2)cc2ccccc12 ZINC000880849163 FG On-Demand Anodyne CCR8 57 32 COC(=O)c1cc(NC(=O)N2CC[C@@H]3[C@H](CCN3C)C2)cc2ccccc12 ZINC000880849164 FG On-Demand Anodyne CCR8 57 32 COC(=O)c1cc(NC(=O)N2CC[C@@H]3[C@@H](CCN3C)C2)cc2ccccc12 ZINC000880849165 FG On-Demand Anodyne CCR8 57 32 COC(=O)c1cc(NC(=O)N2CC[C@H]3[C@@H](CCN3C)C2)cc2ccccc12 ZINC000880849166 FG On-Demand Anodyne CCR8 57 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC=CCC1 ZINC000880849184 EF On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC=CCC1 ZINC000880849185 EF On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CC=CCC1 ZINC000880849186 EF On-Demand Anodyne PAPA1_CARPA 37 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CC=CCC1 ZINC000880849187 EF On-Demand Anodyne PAPA1_CARPA 37 43 COC(=O)c1cc(NC(=O)N2CCC(F)CC2)cc2ccccc12 ZINC000880849208 EH On-Demand Anodyne RBP4 25 44 COC(=O)c1cc(NC(=O)N2CCC(F)CC2)cc2ccccc12 ZINC000880849208 EH On-Demand Anodyne CCR8 46 33 COC(=O)c1cc(NC(=O)N2CCC(O)CC2)cc2ccccc12 ZINC000880849214 EF On-Demand Anodyne RBP4 18 42 COC(=O)c1cc(NC(=O)N2CCC(O)CC2)cc2ccccc12 ZINC000880849214 EF On-Demand Anodyne CCR8 46 33 Cc1cc(NC(=O)NCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880849215 EC On-Demand Anodyne CASR 17 43 Cc1cc(NC(=O)NCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880849215 EC On-Demand Anodyne CCR3 25 45 Cc1cc(NC(=O)NCCN2CCOCC2)cc(S(C)(=O)=O)c1 ZINC000880849215 EC On-Demand Anodyne EPHX2 27 46 COC(=O)c1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)cc2ccccc12 ZINC000880849219 FG On-Demand Anodyne RBP4 15 40 COC(=O)c1cc(NC(=O)N2CC[C@H](C(C)(C)O)C2)cc2ccccc12 ZINC000880849219 FG On-Demand Anodyne CCR8 51 31 COC(=O)c1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)cc2ccccc12 ZINC000880849220 FG On-Demand Anodyne RBP4 15 40 COC(=O)c1cc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)cc2ccccc12 ZINC000880849220 FG On-Demand Anodyne CCR8 51 31 COC(=O)[C@H](CNC(=O)c1ncsc1C1CC1)C1CCCCC1 ZINC000880849233 EG On-Demand Anodyne MAP1 59 45 COC(=O)[C@@H](CNC(=O)c1ncsc1C1CC1)C1CCCCC1 ZINC000880849234 EG On-Demand Anodyne MAP1 59 45 COC(=O)c1cc(NC(=O)NCCN2CC[C@H](O)C2)cc2ccccc12 ZINC000880849240 FD On-Demand Anodyne DRD3 20 41 COC(=O)c1cc(NC(=O)NCCN2CC[C@H](O)C2)cc2ccccc12 ZINC000880849240 FD On-Demand Anodyne CCR3 58 41 COC(=O)c1cc(NC(=O)NCCN2CC[C@H](O)C2)cc2ccccc12 ZINC000880849240 FD On-Demand Anodyne PLD2 42 33 COC(=O)c1cc(NC(=O)NCCN2CC[C@H](O)C2)cc2ccccc12 ZINC000880849240 FD On-Demand Anodyne MCHR1 24 43 COC(=O)c1cc(NC(=O)NCCN2CC[C@@H](O)C2)cc2ccccc12 ZINC000880849241 FD On-Demand Anodyne DRD3 20 41 COC(=O)c1cc(NC(=O)NCCN2CC[C@@H](O)C2)cc2ccccc12 ZINC000880849241 FD On-Demand Anodyne CCR3 58 41 COC(=O)c1cc(NC(=O)NCCN2CC[C@@H](O)C2)cc2ccccc12 ZINC000880849241 FD On-Demand Anodyne PLD2 42 33 COC(=O)c1cc(NC(=O)NCCN2CC[C@@H](O)C2)cc2ccccc12 ZINC000880849241 FD On-Demand Anodyne MCHR1 24 43 O=C(NCc1ccc(Br)c(F)c1F)[C@@H]1CCc2nncn2CC1 ZINC000880849251 GF On-Demand Anodyne P2RX7 42 39 O=C(NCc1ccc(Br)c(F)c1F)[C@H]1CCc2nncn2CC1 ZINC000880849252 GF On-Demand Anodyne P2RX7 42 39 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CC#N)C2)cc2ccccc12 ZINC000880849269 FH On-Demand Mild CCR3 18 43 COC(=O)c1cc(NC(=O)N2CCC[C@H](CC#N)C2)cc2ccccc12 ZINC000880849270 FH On-Demand Mild CCR3 18 43 Cc1cc(NC(=O)NCCCN2CCCC2=O)cc(S(C)(=O)=O)c1 ZINC000880849276 FD On-Demand Anodyne CCR3 29 44 Cc1cc(NC(=O)NCCCN2CCCCCC2=O)cc(S(C)(=O)=O)c1 ZINC000880849277 GE On-Demand Anodyne CCR3 30 44 Cc1cc(NC(=O)NC[C@@H](c2ccco2)N2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880849281 GF On-Demand Anodyne LPL 42 33 Cc1cc(NC(=O)NC[C@H](c2ccco2)N2CCCC2)cc(S(C)(=O)=O)c1 ZINC000880849282 GF On-Demand Anodyne LPL 42 33 C#CCC1(O)CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880849286 FG On-Demand Mild S1PR2 28 41 COC(=O)c1cc(NC(=O)N2CCC(Cn3cnnc3)CC2)cc2ccccc12 ZINC000880849304 GG On-Demand Anodyne CCR8 44 35 COC(=O)c1cc(NC(=O)N[C@@H]2CC[C@H](O)CC2)cc2ccccc12 ZINC000880849314 EG On-Demand Anodyne EPHX2 44 36 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne CHRM2 15 45 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne DRD2 19 57 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne DRD4 50 57 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne ACHE 40 44 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne DRD3 15 57 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne CHRM3 21 45 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne SIGMAR1 41 52 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne SSTR5 30 40 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne CCR3 77 54 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne UTS2R 18 40 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne MLNR 41 36 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne CCR2 20 44 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne EPHX2 43 42 Cc1cc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc(S(C)(=O)=O)c1 ZINC000880849316 GF On-Demand Anodyne MCHR1 30 48 COC(=O)c1cc(NC(=O)N(C)[C@H](C)CO)cc2ccccc12 ZINC000880849396 DE On-Demand Anodyne NPY5R 35 44 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)CO)cc2ccccc12 ZINC000880849397 DE On-Demand Anodyne NPY5R 35 44 COC(=O)c1cc(NC(=O)N2CC[C@H](S(C)(=O)=O)C2)cc2ccccc12 ZINC000880849421 GE On-Demand Anodyne CCR8 72 32 COC(=O)c1cc(NC(=O)N2CC[C@@H](S(C)(=O)=O)C2)cc2ccccc12 ZINC000880849422 GE On-Demand Anodyne CCR8 72 32 COC(=O)c1cc(NC(=O)N2CCC[C@H]2c2nc(C)no2)cc2ccccc12 ZINC000880849427 GH On-Demand Anodyne CPT1A 72 41 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2c2nc(C)no2)cc2ccccc12 ZINC000880849428 GH On-Demand Anodyne CPT1A 72 41 COC(=O)c1cc(NC(=O)N2CCC[C@H]2c2cc(C)on2)cc2ccccc12 ZINC000880849438 GI On-Demand Anodyne CPT1A 67 41 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2c2cc(C)on2)cc2ccccc12 ZINC000880849439 GI On-Demand Anodyne CPT1A 67 41 COCCO[C@H]1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880849450 FF On-Demand Anodyne CCR8 61 35 COCCO[C@@H]1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880849451 FF On-Demand Anodyne CCR8 61 35 COC(=O)c1cc(NC(=O)N2CCCC[C@@H]2c2nc(C)no2)cc2ccccc12 ZINC000880849487 GI On-Demand Anodyne CPT1A 102 44 COC(=O)c1cc(NC(=O)N2CCCC[C@H]2c2nc(C)no2)cc2ccccc12 ZINC000880849488 GI On-Demand Anodyne CPT1A 102 44 COC(=O)c1cc(NC(=O)N2CCC3(CC2)OCCO3)cc2ccccc12 ZINC000880849489 FF On-Demand Anodyne NPY5R 26 40 COC(=O)c1cc(NC(=O)NC2CCN(OC)CC2)cc2ccccc12 ZINC000880849493 FF On-Demand Anodyne EPHX2 45 48 COC(=O)c1cc(NC(=O)NC2CCN(OC)CC2)cc2ccccc12 ZINC000880849493 FF On-Demand Anodyne CXCR3 18 41 COC(=O)c1cc(NC(=O)NC2C[C@@H]3CC[C@H](C2)N3C)cc2ccccc12 ZINC000880849542 FG On-Demand Anodyne HTR3A 36 40 COC(=O)c1cc(NC(=O)NC2C[C@@H]3CC[C@H](C2)N3C)cc2ccccc12 ZINC000880849542 FG On-Demand Anodyne HTR4 41 41 COC(=O)c1cc(NC(=O)NC2C[C@@H]3CC[C@H](C2)N3C)cc2ccccc12 ZINC000880849542 FG On-Demand Anodyne EPHX2 28 40 COC(=O)c1cc(NC(=O)NC2C[C@@H]3CC[C@H](C2)N3C)cc2ccccc12 ZINC000880849542 FG On-Demand Anodyne GLRA1 56 40 COC(=O)c1cc(NC(=O)N2CCCc3c(cnn3C)C2)cc2ccccc12 ZINC000880849579 GG On-Demand Anodyne P2RY14 47 33 Cn1nnc(C(=O)N[C@@H]2CCN(c3ccc(Cl)cc3F)C2=O)n1 ZINC000880849590 EC On-Demand Anodyne F10 20 43 Cn1nnc(C(=O)N[C@H]2CCN(c3ccc(Cl)cc3F)C2=O)n1 ZINC000880849591 EC On-Demand Anodyne F10 20 43 COC(=O)c1cc(NC(=O)NC2CCN(C(=O)C(C)C)CC2)cc2ccccc12 ZINC000880849597 GG On-Demand Anodyne EPHX2 47 55 COC(=O)c1cc(NC(=O)NC2CCN(C(=O)C(C)C)CC2)cc2ccccc12 ZINC000880849597 GG On-Demand Anodyne CCR8 67 33 COC(=O)c1cc(NC(=O)N(C)C2C[C@@H]3CC[C@H](C2)N3C)cc2ccccc12 ZINC000880849612 GH On-Demand Anodyne GLRA1 54 39 COC(=O)c1cc(NC(=O)N2CCC3(CCO3)CC2)cc2ccccc12 ZINC000880849667 FG On-Demand Anodyne NPY5R 26 40 COC(=O)c1cc(NC(=O)N2CCC3(CCO3)CC2)cc2ccccc12 ZINC000880849667 FG On-Demand Anodyne EPHX2 26 40 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849702 FD On-Demand Anodyne F10 19 42 O=C(C[C@@H]1CCNC1=O)N[C@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849703 FD On-Demand Anodyne F10 19 42 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849704 FD On-Demand Anodyne F10 19 42 O=C(C[C@H]1CCNC1=O)N[C@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849705 FD On-Demand Anodyne F10 19 42 COC(=O)c1cc(NC(=O)NCCCCO)cc2ccccc12 ZINC000880849796 DF On-Demand Anodyne CA1 17 40 Cc1nc(C(C)C)ncc1C(=O)N1CCC(C)(N2CCOCC2)CC1 ZINC000880849797 EE On-Demand Anodyne CCR5 42 41 COC(=O)c1cc(NC(=O)NC[C@@H]2CCCN(C(C)=O)C2)cc2ccccc12 ZINC000880849827 GG On-Demand Anodyne CCR3 60 42 COC(=O)c1cc(NC(=O)NC[C@H]2CCCN(C(C)=O)C2)cc2ccccc12 ZINC000880849828 GG On-Demand Anodyne CCR3 60 42 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCc2c(cccc2C(F)(F)F)C1 ZINC000880849830 EG On-Demand Anodyne RBP4 41 33 COC(=O)c1cc(NC(=O)N2CC(C(F)(F)F)C2)cc2ccccc12 ZINC000880849872 FH On-Demand Anodyne RBP4 51 31 COC(=O)c1cc(NC(=O)N2CCC3(CCN(C)C3=O)CC2)cc2ccccc12 ZINC000880849931 GG On-Demand Anodyne CACNA1H 43 36 COC(=O)c1cc(NC(=O)N2CC(c3nc(C)no3)C2)cc2ccccc12 ZINC000880849936 FF On-Demand Anodyne SMO 30 40 COC(=O)c1cc(NC(=O)N2CCN(C[C@H](C)O)CC2)cc2ccccc12 ZINC000880849945 FE On-Demand Anodyne PDGFRB 41 34 COC(=O)c1cc(NC(=O)N2CCN(C[C@H](C)O)CC2)cc2ccccc12 ZINC000880849945 FE On-Demand Anodyne ABCB1 20 41 CSc1nccnc1C(=O)N[C@@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849991 GF On-Demand Anodyne F10 19 44 CSc1nccnc1C(=O)N[C@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880849992 GF On-Demand Anodyne F10 19 44 COC(=O)c1cc(NC(=O)N2CC[C@H](C)[S@@](=O)CC2)cc2ccccc12 ZINC000880849996 FG On-Demand Anodyne RBP4 17 41 COC(=O)c1cc(NC(=O)N2CC[C@@H](C)[S@@](=O)CC2)cc2ccccc12 ZINC000880849997 FG On-Demand Anodyne RBP4 17 41 COC(=O)c1cc(NC(=O)N2CC[C@H](C)[S@](=O)CC2)cc2ccccc12 ZINC000880849998 FG On-Demand Anodyne RBP4 17 41 COC(=O)c1cc(NC(=O)N2CC[C@@H](C)[S@](=O)CC2)cc2ccccc12 ZINC000880849999 FG On-Demand Anodyne RBP4 17 41 COC(=O)c1cc(NC(=O)N2CC[C@]3(CCN(C)C3)C2)cc2ccccc12 ZINC000880850001 FG On-Demand Anodyne EPHX2 31 42 COC(=O)c1cc(NC(=O)N2CC[C@@]3(CCN(C)C3)C2)cc2ccccc12 ZINC000880850002 FG On-Demand Anodyne EPHX2 31 42 COC(=O)c1cc(NC(=O)N2CCC[C@H](N(C)C)CC2)cc2ccccc12 ZINC000880850011 FH On-Demand Anodyne RBP4 19 41 COC(=O)c1cc(NC(=O)N2CCC[C@@H](N(C)C)CC2)cc2ccccc12 ZINC000880850012 FH On-Demand Anodyne RBP4 19 41 NC(=O)c1cc(-c2csc(NC(=O)c3ccc(NC4=NS(=O)(=O)c5ccccc54)cc3)n2)c[nH]1 ZINC000880850019 JG On-Demand Anodyne MPL 62 41 Cc1cnc(Cl)c(C(=O)N2CCC(C)(N3CCOCC3)CC2)c1 ZINC000880850025 EE On-Demand Anodyne CCR5 42 39 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CCNC(C)=O)C2)cc2ccccc12 ZINC000880850031 GG On-Demand Anodyne CCR3 15 41 COC(=O)c1cc(NC(=O)N2CCC[C@H](CCNC(C)=O)C2)cc2ccccc12 ZINC000880850032 GG On-Demand Anodyne CCR3 15 41 COC(=O)c1cc(NC(=O)N2CC[C@H](NC(C)=O)C2)cc2ccccc12 ZINC000880850034 FE On-Demand Anodyne CCR8 79 39 COC(=O)c1cc(NC(=O)N2CC[C@@H](NC(C)=O)C2)cc2ccccc12 ZINC000880850035 FE On-Demand Anodyne CCR8 79 39 COC[C@@H](O)CNC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880850076 ED On-Demand Anodyne ADRB1 42 32 COC(=O)c1cc(NC(=O)N2CC[C@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880850084 GG On-Demand Anodyne SMO 41 46 COC(=O)c1cc(NC(=O)N2CC[C@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880850084 GG On-Demand Anodyne ETHR 43 35 COC(=O)c1cc(NC(=O)N2CC[C@@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880850085 GG On-Demand Anodyne SMO 41 46 COC(=O)c1cc(NC(=O)N2CC[C@@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880850085 GG On-Demand Anodyne ETHR 43 35 COC(=O)c1cc(NC(=O)N2CC[C@@H](F)C2)cc2ccccc12 ZINC000880850115 DG On-Demand Anodyne RBP4 24 42 COC(=O)c1cc(NC(=O)N2CC[C@@H](F)C2)cc2ccccc12 ZINC000880850115 DG On-Demand Anodyne CCR8 70 32 COC(=O)c1cc(NC(=O)N2CC[C@H](F)C2)cc2ccccc12 ZINC000880850116 DG On-Demand Anodyne RBP4 24 42 COC(=O)c1cc(NC(=O)N2CC[C@H](F)C2)cc2ccccc12 ZINC000880850116 DG On-Demand Anodyne CCR8 70 32 COC(=O)c1cc(NC(=O)N2CCO[C@@]3(CCCOC3)C2)cc2ccccc12 ZINC000880850162 GG On-Demand Anodyne EPHX2 25 42 COC(=O)c1cc(NC(=O)N2CCO[C@]3(CCCOC3)C2)cc2ccccc12 ZINC000880850163 GG On-Demand Anodyne EPHX2 25 42 COC(=O)c1cc(NC(=O)NC2CCC(NC(C)=O)CC2)cc2ccccc12 ZINC000880850178 GG On-Demand Anodyne EPHX2 45 36 COC(=O)c1cc(NC(=O)N2CC[C@@H](CS(C)(=O)=O)C2)cc2ccccc12 ZINC000880850187 GF On-Demand Anodyne CCR8 75 33 COC(=O)c1cc(NC(=O)N2CC[C@H](CS(C)(=O)=O)C2)cc2ccccc12 ZINC000880850188 GF On-Demand Anodyne CCR8 75 33 O=C(COC1CC1)N[C@@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880850201 ED On-Demand Anodyne F10 27 44 O=C(COC1CC1)N[C@H]1CCN(c2ccc(Cl)cc2F)C1=O ZINC000880850202 ED On-Demand Anodyne F10 27 44 COC(=O)c1cc(NC(=O)N2CCC[C@H]2CCO)cc2ccccc12 ZINC000880850210 EG On-Demand Anodyne HCRTR1 19 41 COC(=O)c1cc(NC(=O)N2CCC[C@H]2CCO)cc2ccccc12 ZINC000880850210 EG On-Demand Anodyne ACKR3 51 32 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2CCO)cc2ccccc12 ZINC000880850211 EG On-Demand Anodyne HCRTR1 19 41 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2CCO)cc2ccccc12 ZINC000880850211 EG On-Demand Anodyne ACKR3 51 32 Cc1coc(C(=O)N[C@@H]2CCN(c3ccc(Cl)cc3F)C2=O)c1 ZINC000880850212 EF On-Demand Anodyne F10 22 44 Cc1coc(C(=O)N[C@H]2CCN(c3ccc(Cl)cc3F)C2=O)c1 ZINC000880850214 EF On-Demand Anodyne F10 22 44 COC(=O)c1cc(NC(=O)N2CC[C@@](O)(C(F)(F)F)C2)cc2ccccc12 ZINC000880850222 GG On-Demand Anodyne EPHX2 34 42 COC(=O)c1cc(NC(=O)N2CC[C@](O)(C(F)(F)F)C2)cc2ccccc12 ZINC000880850223 GG On-Demand Anodyne EPHX2 34 42 COC(=O)c1cc(NC(=O)N2CCC(c3ccncn3)CC2)cc2ccccc12 ZINC000880850237 GH On-Demand Anodyne RBP4 18 40 COC(=O)c1cc(NC(=O)N2CC[C@H](SC)C2)cc2ccccc12 ZINC000880850257 EH On-Demand Anodyne CCR8 46 31 COC(=O)c1cc(NC(=O)N2CC[C@@H](SC)C2)cc2ccccc12 ZINC000880850258 EH On-Demand Anodyne CCR8 46 31 CC[C@@H](NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1)C(=O)NC ZINC000880850281 EE On-Demand Anodyne ANPEP 15 40 COC(=O)c1cc(NC(=O)N[C@@H]2CC[C@@H](O)CC2)cc2ccccc12 ZINC000880850294 EG On-Demand Anodyne EPHX2 44 36 CS(=O)(=O)C1CCC(C(=O)Nc2cccc(C3CCOCC3)c2)CC1 ZINC000880850303 FG On-Demand Anodyne MCHR1 22 41 COC(=O)c1cc(NC(=O)NCC(=O)NC(C)C)cc2ccccc12 ZINC000880850320 EE On-Demand Anodyne F7 26 42 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CNC(C)=O)C2)cc2ccccc12 ZINC000880850326 GG On-Demand Anodyne CCR3 26 43 COC(=O)c1cc(NC(=O)N2CCC[C@H](CNC(C)=O)C2)cc2ccccc12 ZINC000880850328 GG On-Demand Anodyne CCR3 26 43 Cc1nc(C(C)C)ncc1C(=O)Nc1cccc(C2CCOCC2)c1 ZINC000880850330 EI On-Demand Anodyne KCNK3 49 34 Cc1nc(C(C)C)ncc1C(=O)Nc1cccc(C2CCOCC2)c1 ZINC000880850330 EI On-Demand Anodyne KCNK9 43 34 COC(=O)c1cc(NC(=O)N2CC[C@H](CCCO)C2)cc2ccccc12 ZINC000880850331 FG On-Demand Anodyne CCR8 45 34 COC(=O)c1cc(NC(=O)N2CC[C@@H](CCCO)C2)cc2ccccc12 ZINC000880850332 FG On-Demand Anodyne CCR8 45 34 CS(=O)(=O)C1CCC(C(=O)N2CCc3c(cccc3C(F)(F)F)C2)CC1 ZINC000880850333 GG On-Demand Anodyne RBP4 41 33 CS(=O)(=O)C1CCC(C(=O)N2CCc3c(cccc3C(F)(F)F)C2)CC1 ZINC000880850333 GG On-Demand Anodyne SFRP1 85 33 CS(=O)(=O)C1CCC(C(=O)N2CCc3c(cccc3C(F)(F)F)C2)CC1 ZINC000880850333 GG On-Demand Anodyne WNT3 58 32 COC(=O)c1cc(NC(=O)N2CC(C3CC3)C2)cc2ccccc12 ZINC000880850335 DH On-Demand Anodyne RBP4 44 30 COC(=O)c1cc(NC(=O)NC2CCN(CC#N)CC2)cc2ccccc12 ZINC000880850365 FF On-Demand Mild DRD4 18 44 COC(=O)c1cc(NC(=O)NC2CCN(CC#N)CC2)cc2ccccc12 ZINC000880850365 FF On-Demand Mild EPHX2 38 45 COC(=O)c1cc(NC(=O)NC2CCN(CC#N)CC2)cc2ccccc12 ZINC000880850365 FF On-Demand Mild CXCR3 21 43 COC(=O)c1cc(NC(=O)NC2CCN(CC#N)CC2)cc2ccccc12 ZINC000880850365 FF On-Demand Mild MCHR1 16 40 COCC1(O)CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880850379 FF On-Demand Anodyne S1PR2 29 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(O)ccc1C ZINC000880850404 EF On-Demand Anodyne PAPA1_CARPA 39 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(O)ccc1C ZINC000880850407 EF On-Demand Anodyne PAPA1_CARPA 39 44 O=C(Nc1cccc(C2CCOCC2)c1)c1coc(-c2ccccn2)n1 ZINC000880850414 EH On-Demand Anodyne GRM4 57 41 O=C(Nc1cccc(C2CCOCC2)c1)c1coc(-c2ccccn2)n1 ZINC000880850414 EH On-Demand Anodyne KCNK3 27 42 COC(=O)c1cc(NC(=O)N2CCC[C@H](S(C)(=O)=O)C2)cc2ccccc12 ZINC000880850425 GF On-Demand Anodyne CCR8 44 32 COC(=O)c1cc(NC(=O)N2CCC(NC(C)C)CC2)cc2ccccc12 ZINC000880850426 FH On-Demand Anodyne CCR8 77 35 COC(=O)c1cc(NC(=O)N2CCC[C@@H](S(C)(=O)=O)C2)cc2ccccc12 ZINC000880850429 GF On-Demand Anodyne CCR8 44 32 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne HTR1A 59 44 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne DRD2 58 45 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne DRD4 40 31 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne HTR2A 47 44 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne HTR2C 31 42 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne ADRA1A 49 39 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne DRD3 92 48 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne HTR7 65 41 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne NPY1R 22 42 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne CCR3 46 44 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne CHRNA7 15 46 COC(=O)c1cc(NC(=O)NCCCCN2CCN(C)CC2)cc2ccccc12 ZINC000880850432 GF On-Demand Anodyne MCHR1 17 41 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(O)ccc1C)C2 ZINC000880850433 DG On-Demand Anodyne ROCK2 17 40 Nc1ncnc2c1ncn2CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880850447 FE On-Demand Anodyne AHCY 49 39 Nc1ncnc2c1ncn2CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880850447 FE On-Demand Anodyne OXGR1 96 35 Nc1ncnc2c1ncn2CCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880850447 FE On-Demand Anodyne DOT1L 50 34 Nc1ncnc2c1ncn2CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880850451 FE On-Demand Anodyne AHCY 49 39 Nc1ncnc2c1ncn2CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880850451 FE On-Demand Anodyne OXGR1 96 35 Nc1ncnc2c1ncn2CCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880850451 FE On-Demand Anodyne DOT1L 50 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1COC ZINC000880850468 ED On-Demand Anodyne CELA1 24 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@@H]1COC ZINC000880850469 ED On-Demand Anodyne CELA1 24 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]1COC ZINC000880850470 ED On-Demand Anodyne CELA1 24 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]1COC ZINC000880850471 ED On-Demand Anodyne CELA1 24 40 COC(=O)c1cc(NC(=O)N2CCC(CC#N)CC2)cc2ccccc12 ZINC000880850481 FH On-Demand Mild P2RY12 15 41 COC(=O)c1cc(NC(=O)N2CCC(CC#N)CC2)cc2ccccc12 ZINC000880850481 FH On-Demand Mild CCR8 41 31 COC(=O)c1cc(NC(=O)N2CCC(c3cn[nH]c3)CC2)cc2ccccc12 ZINC000880850489 GH On-Demand Anodyne RBP4 19 40 CCc1nc([C@H]2CCCN2C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)no1 ZINC000880850520 GH On-Demand Anodyne CPT1A 56 40 O=C(Nc1cccc(C2CCOCC2)c1)c1cnc2cc[nH]c2c1 ZINC000880850552 DH On-Demand Anodyne KCNK3 48 35 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1Cc3ccccc3NC1=O)C2 ZINC000880850562 FE On-Demand Anodyne PYGM 18 43 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1Cc3ccccc3NC1=O)C2 ZINC000880850563 FE On-Demand Anodyne PYGM 18 43 O=C1Nc2ccccc2C[C@@H]1NC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880850572 EF On-Demand Anodyne PYGM 15 44 O=C1Nc2ccccc2C[C@H]1NC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880850573 EF On-Demand Anodyne PYGM 15 44 COC(=O)c1cc(NC(=O)N2CCC3(CC2)C[C@@H]3C(=O)OC)cc2ccccc12 ZINC000880850577 GG On-Demand Anodyne CACNA1H 41 38 COC(=O)c1cc(NC(=O)N2CCC3(CC2)C[C@H]3C(=O)OC)cc2ccccc12 ZINC000880850578 GG On-Demand Anodyne CACNA1H 41 38 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880850580 GE On-Demand Anodyne P2RY12 85 36 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880850580 GE On-Demand Anodyne PSMB8 45 36 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880850583 GE On-Demand Anodyne P2RY12 85 36 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880850583 GE On-Demand Anodyne PSMB8 45 36 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CCO)C2)cc2ccccc12 ZINC000880850590 FG On-Demand Anodyne CCR3 15 43 COC(=O)c1cc(NC(=O)N2CCC[C@H](CCO)C2)cc2ccccc12 ZINC000880850591 FG On-Demand Anodyne CCR3 15 43 COCC(=O)NC1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880850595 GE On-Demand Anodyne EPHX2 25 42 COCC(=O)NC1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880850595 GE On-Demand Anodyne CCR8 78 38 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880850623 FE On-Demand Anodyne PYGL 15 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880850623 FE On-Demand Anodyne PYGM 27 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880850625 FE On-Demand Anodyne PYGL 15 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880850625 FE On-Demand Anodyne PYGM 27 41 COC(=O)c1cc(NC(=O)N2CCC(c3nc(C)no3)CC2)cc2ccccc12 ZINC000880850635 GH On-Demand Anodyne SMO 45 50 COC(=O)c1cc(NC(=O)N2CCC(c3nc(C)no3)CC2)cc2ccccc12 ZINC000880850635 GH On-Demand Anodyne ETHR 49 35 NC(=O)c1cc(-c2csc(NC(=O)Cn3cnc4sc(-c5ccccc5)cc4c3=O)n2)c[nH]1 ZINC000880850639 JG On-Demand Anodyne TRPA1 16 49 COC(=O)c1cc(NC(=O)N(C)CCCn2ccnc2)cc2ccccc12 ZINC000880850670 FG On-Demand Anodyne TBXAS1 47 41 COC(=O)c1cc(NC(=O)N(C)CCCn2ccnc2)cc2ccccc12 ZINC000880850670 FG On-Demand Anodyne QPCT 39 43 COC(=O)c1cc(NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850688 GF On-Demand Anodyne DRD4 19 41 COC(=O)c1cc(NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850688 GF On-Demand Anodyne EPHX2 41 45 COC(=O)c1cc(NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850688 GF On-Demand Anodyne CCR8 67 33 COC(=O)c1cc(NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850689 GF On-Demand Anodyne DRD4 19 41 COC(=O)c1cc(NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850689 GF On-Demand Anodyne EPHX2 41 45 COC(=O)c1cc(NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)cc2ccccc12 ZINC000880850689 GF On-Demand Anodyne CCR8 67 33 COC(=O)c1cc(NC(=O)N2CC[C@@H](CN3CCOCC3)C2)cc2ccccc12 ZINC000880850690 GF On-Demand Anodyne CCR3 15 46 COC(=O)c1cc(NC(=O)N2CC[C@@H](CN3CCOCC3)C2)cc2ccccc12 ZINC000880850690 GF On-Demand Anodyne PTGDS 42 37 COC(=O)c1cc(NC(=O)N2CC[C@H](CN3CCOCC3)C2)cc2ccccc12 ZINC000880850691 GF On-Demand Anodyne CCR3 15 46 COC(=O)c1cc(NC(=O)N2CC[C@H](CN3CCOCC3)C2)cc2ccccc12 ZINC000880850691 GF On-Demand Anodyne PTGDS 42 37 COC[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880850704 CG On-Demand Anodyne PREP 45 38 COC[C@@H]1CCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880850704 CG On-Demand Anodyne EBP 30 43 COC[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880850705 CG On-Demand Anodyne PREP 45 38 COC[C@@H]1CCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880850705 CG On-Demand Anodyne EBP 30 43 COC(=O)c1cc(NC(=O)N2CCC(C(=O)OC)CC2)cc2ccccc12 ZINC000880850714 FG On-Demand Anodyne CCR8 41 32 Nc1ncnc2c1ncn2CCNC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880850715 FD On-Demand Anodyne AHCY 64 41 Nc1ncnc2c1ncn2CCNC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880850715 FD On-Demand Anodyne OXGR1 101 38 Nc1ncnc2c1ncn2CCNC(=O)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880850715 FD On-Demand Anodyne DOT1L 53 37 COC[C@@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880850716 EG On-Demand Anodyne FKBP1A 75 48 COC[C@@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880850716 EG On-Demand Anodyne INHA 43 34 COC[C@@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880850716 EG On-Demand Anodyne PREP 44 40 COC[C@@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880850716 EG On-Demand Anodyne CASP7 47 36 COC[C@@H]1CCCN1C(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880850716 EG On-Demand Anodyne ACKR3 67 37 O=C(COC1CC1)N[C@@H]1Cc2ccccc2NC1=O ZINC000880850848 CC On-Demand Anodyne PYGL 15 51 O=C(COC1CC1)N[C@@H]1Cc2ccccc2NC1=O ZINC000880850848 CC On-Demand Anodyne PYGM 19 51 O=C(COC1CC1)N[C@H]1Cc2ccccc2NC1=O ZINC000880850849 CC On-Demand Anodyne PYGL 15 51 O=C(COC1CC1)N[C@H]1Cc2ccccc2NC1=O ZINC000880850849 CC On-Demand Anodyne PYGM 19 51 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880850860 FF On-Demand Anodyne EPHX2 42 60 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880850860 FF On-Demand Anodyne CCR8 84 39 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880850861 FF On-Demand Anodyne EPHX2 42 60 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880850861 FF On-Demand Anodyne CCR8 84 39 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1ccc(Oc2cc(C)ccn2)cc1 ZINC000880850862 GG On-Demand Anodyne CTSS 18 40 Cc1cnc(Cl)c(C(=O)NC[C@H]2COCCN2C)c1 ZINC000880850863 CD On-Demand Anodyne CACNA1I 52 33 Cc1cnc(Cl)c(C(=O)NC[C@@H]2COCCN2C)c1 ZINC000880850864 CD On-Demand Anodyne CACNA1I 52 33 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1ccc(Oc2cc(C)ccn2)cc1 ZINC000880850866 GG On-Demand Anodyne CTSS 18 40 COC(=O)c1cc(NC(=O)NCC2CCOCC2)cc2ccccc12 ZINC000880850871 EG On-Demand Anodyne CNR2 15 48 COC(=O)c1cc(NC(=O)N2CCC(N3CC=CC3)CC2)cc2ccccc12 ZINC000880850873 GG On-Demand Anodyne CCR8 60 34 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880850880 FE On-Demand Anodyne UL80 43 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880850880 FE On-Demand Anodyne BRCA1 42 29 COC(=O)c1cc(NC(=O)N[C@@H]2CCN(C(C)=O)C[C@H]2C)cc2ccccc12 ZINC000880850885 GG On-Demand Anodyne EPHX2 18 40 COC(=O)c1cc(NC(=O)N[C@H]2CCN(C(C)=O)C[C@@H]2C)cc2ccccc12 ZINC000880850886 GG On-Demand Anodyne EPHX2 18 40 COC(=O)c1cc(NC(=O)N2CCC(N3CCNC3=O)CC2)cc2ccccc12 ZINC000880850887 GF On-Demand Anodyne CCR8 46 33 COC(=O)c1cc(NC(=O)N[C@@H]2CCN(C(C)=O)C[C@@H]2C)cc2ccccc12 ZINC000880850888 GG On-Demand Anodyne EPHX2 18 40 COC(=O)c1cc(NC(=O)N[C@H]2CCN(C(C)=O)C[C@H]2C)cc2ccccc12 ZINC000880850889 GG On-Demand Anodyne EPHX2 18 40 COC(=O)c1cc(NC(=O)N2CCC(N(C)C)CC2)cc2ccccc12 ZINC000880850906 FG On-Demand Anodyne RBP4 23 43 COC(=O)c1cc(NC(=O)NCC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880850907 GG On-Demand Anodyne CCR3 59 38 COC(=O)c1cc(NC(=O)NCC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880850907 GG On-Demand Anodyne EPHX2 25 46 COC(=O)c1cc(NC(=O)NCC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880850907 GG On-Demand Anodyne CCR8 71 36 CC(C)(C(=O)N[C@H]1Cc2ccccc2NC1=O)c1ccc(F)cc1F ZINC000880850920 EF On-Demand Anodyne PYGM 32 45 COC[C@@H]1CCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880850921 DD On-Demand Anodyne CASP3 44 39 COC[C@@H]1CCCN1C(=O)Cc1ccccc1N1CCCC1=O ZINC000880850921 DD On-Demand Anodyne CASP7 60 39 CC(C)(C(=O)N[C@@H]1Cc2ccccc2NC1=O)c1ccc(F)cc1F ZINC000880850925 EF On-Demand Anodyne PYGM 32 45 O=C(Nc1cccc(C2CCOCC2)c1)c1ncsc1C1CC1 ZINC000880850928 EI On-Demand Anodyne MAP1 54 33 COc1cccc(/C=C(\C(=O)NC2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)n2nnnc2C)c1 ZINC000880850931 JE On-Demand Anodyne EPHX2 20 43 COC(=O)c1cc(NC(=O)NCCCNC(C)=O)cc2ccccc12 ZINC000880850932 EE On-Demand Anodyne NQO2 35 41 COC(=O)c1cc(NC(=O)NCCCNC(C)=O)cc2ccccc12 ZINC000880850932 EE On-Demand Anodyne CA1 17 40 COC(=O)c1cc(NC(=O)NCCCNC(C)=O)cc2ccccc12 ZINC000880850932 EE On-Demand Anodyne MTNR1A 71 41 COC(=O)c1cc(NC(=O)NCCCNC(C)=O)cc2ccccc12 ZINC000880850932 EE On-Demand Anodyne MTNR1B 63 41 COC(=O)c1cc(NC(=O)NC2CCSCC2)cc2ccccc12 ZINC000880850949 EH On-Demand Anodyne EPHX2 43 36 Cn1nc(C2CCOCC2)cc1NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880850957 FF On-Demand Anodyne HTR1F 42 36 CC1(C)CC[C@@H](CC(=O)N[C@@H]2Cc3ccccc3NC2=O)OC1 ZINC000880850958 DE On-Demand Anodyne PYGM 17 43 COC(=O)c1cc(NC(=O)N2CCCC[C@@H]2c2ncc[nH]2)cc2ccccc12 ZINC000880850959 GI On-Demand Anodyne CPT1A 73 38 COC(=O)c1cc(NC(=O)N2CCCC[C@H]2c2ncc[nH]2)cc2ccccc12 ZINC000880850960 GI On-Demand Anodyne CPT1A 73 38 CC1(C)CC[C@@H](CC(=O)N[C@H]2Cc3ccccc3NC2=O)OC1 ZINC000880850964 DE On-Demand Anodyne PYGM 17 43 COC(=O)c1cc(NC(=O)N2CCC(Cn3cncn3)CC2)cc2ccccc12 ZINC000880850977 GG On-Demand Anodyne PDGFRB 41 36 COC(=O)c1cc(NC(=O)N2CC[C@@H](Cc3cnn(C)c3)C2)cc2ccccc12 ZINC000880850979 GG On-Demand Anodyne CCR3 52 41 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2COCCN2C)c(O)n1 ZINC000880850980 FD On-Demand Anodyne DRD2 40 40 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2COCCN2C)c(O)n1 ZINC000880850980 FD On-Demand Anodyne HTR3A 15 40 COc1ccccc1-c1ccc(C(=O)NC[C@H]2COCCN2C)c(O)n1 ZINC000880850981 FD On-Demand Anodyne DRD2 40 40 COc1ccccc1-c1ccc(C(=O)NC[C@H]2COCCN2C)c(O)n1 ZINC000880850981 FD On-Demand Anodyne HTR3A 15 40 COC(=O)c1cc(NC(=O)N2CC[C@H](Cc3cnn(C)c3)C2)cc2ccccc12 ZINC000880850984 GG On-Demand Anodyne CCR3 52 41 COC(=O)c1cc(NC(=O)N2CCC(NC(C)=O)CC2)cc2ccccc12 ZINC000880850993 FF On-Demand Anodyne EPHX2 29 42 COC(=O)c1cc(NC(=O)N2CCC(NC(C)=O)CC2)cc2ccccc12 ZINC000880850993 FF On-Demand Anodyne CCR8 82 41 O=C(N[C@@H]1Cc2ccccc2NC1=O)c1cnc(CC2CC2)s1 ZINC000880850998 EE On-Demand Anodyne PYGL 26 48 O=C(N[C@@H]1Cc2ccccc2NC1=O)c1cnc(CC2CC2)s1 ZINC000880850998 EE On-Demand Anodyne PYGM 28 45 O=C(N[C@H]1Cc2ccccc2NC1=O)c1cnc(CC2CC2)s1 ZINC000880850999 EE On-Demand Anodyne PYGL 26 48 O=C(N[C@H]1Cc2ccccc2NC1=O)c1cnc(CC2CC2)s1 ZINC000880850999 EE On-Demand Anodyne PYGM 28 45 COC[C@@H]1CCCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)C1 ZINC000880851029 FH On-Demand Anodyne CCR3 21 44 COC(=O)c1cc(NC(=O)N2CCC(N(C)CCO)CC2)cc2ccccc12 ZINC000880851053 GF On-Demand Anodyne RBP4 17 41 COC(=O)c1cc(NC(=O)N2CCC(N(C)CCO)CC2)cc2ccccc12 ZINC000880851053 GF On-Demand Anodyne CCR8 49 33 COC(=O)c1cc(NC(=O)NCC(=O)N2CCOCC2)cc2ccccc12 ZINC000880851054 FD On-Demand Anodyne EPHX2 17 42 COC(=O)c1cc(NC(=O)NCCN2CCNC(=O)C2)cc2ccccc12 ZINC000880851061 FD On-Demand Anodyne PLD2 51 36 COC[C@@H]1CCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880851070 DE On-Demand Anodyne MPO 60 35 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(C(F)(F)F)cc1 ZINC000880851071 GF On-Demand Anodyne AHCY 63 42 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(C(F)(F)F)cc1 ZINC000880851071 GF On-Demand Anodyne OXGR1 100 36 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(C(F)(F)F)cc1 ZINC000880851071 GF On-Demand Anodyne DOT1L 70 44 COC(=O)c1cc(NC(=O)N[C@@H](C)CCN2CCN(C)CC2)cc2ccccc12 ZINC000880851078 GF On-Demand Anodyne CCR3 54 43 COC(=O)c1cc(NC(=O)N[C@H](C)CCN2CCN(C)CC2)cc2ccccc12 ZINC000880851079 GF On-Demand Anodyne CCR3 54 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1COCCN1C ZINC000880851080 EC On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1COCCN1C ZINC000880851081 EC On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1COCCN1C ZINC000880851082 EC On-Demand Anodyne PAPA1_CARPA 35 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1COCCN1C ZINC000880851083 EC On-Demand Anodyne PAPA1_CARPA 35 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851118 GG On-Demand Anodyne EPHX2 21 43 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851119 GG On-Demand Anodyne EPHX2 21 43 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851120 GG On-Demand Anodyne EPHX2 21 43 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851121 GG On-Demand Anodyne EPHX2 21 43 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(F)cc1F ZINC000880851262 FD On-Demand Anodyne AHCY 61 41 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(F)cc1F ZINC000880851262 FD On-Demand Anodyne OXGR1 100 36 CC(C)(C(=O)NCCn1cnc2c(N)ncnc21)c1ccc(F)cc1F ZINC000880851262 FD On-Demand Anodyne DOT1L 59 41 CC[C@@H](CC#N)NC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851264 EG On-Demand Mild DHODH 16 40 COC(=O)c1cc(NC(=O)N[C@H]2CCn3ccnc3C2)cc2ccccc12 ZINC000880851265 FF On-Demand Anodyne EPHX2 28 40 COC(=O)c1cc(NC(=O)N[C@@H]2CCn3ccnc3C2)cc2ccccc12 ZINC000880851266 FF On-Demand Anodyne EPHX2 28 40 COC[C@@H]1CCCN1C(=O)c1cc(C)cnc1Cl ZINC000880851274 CE On-Demand Anodyne CASP7 40 34 CC[C@H](O)CCNC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851300 EF On-Demand Anodyne ADRB1 40 32 CC[C@@H](O)CCNC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851301 EF On-Demand Anodyne ADRB1 40 32 COC(=O)c1cc(NC(=O)N(C)C(C)C)cc2ccccc12 ZINC000880851304 DG On-Demand Anodyne NPY5R 33 40 COC(=O)c1cc(NC(=O)N2CCC(S(C)(=O)=O)CC2)cc2ccccc12 ZINC000880851318 GF On-Demand Anodyne RBP4 24 40 COC(=O)c1cc(NC(=O)N2CCC(S(C)(=O)=O)CC2)cc2ccccc12 ZINC000880851318 GF On-Demand Anodyne CCR8 76 35 COC[C@@H]1CCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880851339 CD On-Demand Anodyne CPT1A 69 40 COC(=O)c1cc(NC(=O)N2CCC(c3cnc[nH]3)CC2)cc2ccccc12 ZINC000880851340 GH On-Demand Anodyne RBP4 21 40 COC(=O)c1cc(NC(=O)NOCCC(F)(F)F)cc2ccccc12 ZINC000880851343 FH On-Demand Anodyne KCNJ11 41 34 COC[C@@H]1CCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880851348 CD On-Demand Anodyne CASP7 40 35 COC(=O)c1cc(NC(=O)N2CCOC3(CCOCC3)CC2)cc2ccccc12 ZINC000880851349 GG On-Demand Anodyne NPY5R 15 43 COC(=O)c1cc(NC(=O)N2CCOC3(CCOCC3)CC2)cc2ccccc12 ZINC000880851349 GG On-Demand Anodyne EPHX2 21 41 COC(=O)c1cc(NC(=O)N2CCCN(C)CC2)cc2ccccc12 ZINC000880851359 EF On-Demand Anodyne HTR1B 15 46 COC(=O)c1cc(NC(=O)NCCCF)cc2ccccc12 ZINC000880851360 DG On-Demand Anodyne CA1 17 40 COC(=O)c1cc(NC(=O)N2CCC[C@](C)(O)C2)cc2ccccc12 ZINC000880851363 EG On-Demand Anodyne EPHX2 31 43 COC(=O)c1cc(NC(=O)N2CCC[C@@](C)(O)C2)cc2ccccc12 ZINC000880851364 EG On-Demand Anodyne EPHX2 31 43 COC[C@@H](O)CCNC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880851375 EE On-Demand Anodyne ADRB1 41 31 Nc1ncnc2c1ncn2CCNC(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880851384 DC On-Demand Anodyne AHCY 84 41 Nc1ncnc2c1ncn2CCNC(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880851384 DC On-Demand Anodyne ADCY5 30 47 Nc1ncnc2c1ncn2CCNC(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880851384 DC On-Demand Anodyne OXGR1 117 41 Nc1ncnc2c1ncn2CCNC(=O)C[C@@H]1C[C@H]1C1CC1 ZINC000880851384 DC On-Demand Anodyne DOT1L 60 34 COC(=O)c1cc(NC(=O)NC(C)(C)[C@@H](C)O)cc2ccccc12 ZINC000880851386 EF On-Demand Anodyne IMDH_CRYPV 46 38 COC(=O)c1cc(NC(=O)NC(C)(C)[C@H](C)O)cc2ccccc12 ZINC000880851387 EF On-Demand Anodyne IMDH_CRYPV 46 38 COC(=O)c1cc(NC(=O)N2CCO[C@@]3(CCOC3)C2)cc2ccccc12 ZINC000880851399 FF On-Demand Anodyne EPHX2 25 43 COC(=O)c1cc(NC(=O)N2CCO[C@]3(CCOC3)C2)cc2ccccc12 ZINC000880851400 FF On-Demand Anodyne EPHX2 25 43 COC(=O)c1cc(NC(=O)N2CCOC3(CCOCC3)C2)cc2ccccc12 ZINC000880851404 GG On-Demand Anodyne EPHX2 26 44 C=CCCC[C@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851406 FF On-Demand Mild AHCY 42 41 C=CCCC[C@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851406 FF On-Demand Mild PRKACA 40 31 C=CCCC[C@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851406 FF On-Demand Mild OXGR1 69 35 C=CCCC[C@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851406 FF On-Demand Mild DOT1L 59 36 C=CCCC[C@@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851407 FF On-Demand Mild AHCY 42 41 C=CCCC[C@@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851407 FF On-Demand Mild PRKACA 40 31 C=CCCC[C@@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851407 FF On-Demand Mild OXGR1 69 35 C=CCCC[C@@H](C(=O)NCCn1cnc2c(N)ncnc21)c1ccccc1 ZINC000880851407 FF On-Demand Mild DOT1L 59 36 COC(=O)c1cc(NC(=O)N2CC[C@]3(CCOC3)C2)cc2ccccc12 ZINC000880851441 FG On-Demand Anodyne EPHX2 34 41 COC(=O)c1cc(NC(=O)N2CC[C@@]3(CCOC3)C2)cc2ccccc12 ZINC000880851442 FG On-Demand Anodyne EPHX2 34 41 CC[C@@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851443 DD On-Demand Anodyne AHCY 67 40 CC[C@@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851443 DD On-Demand Anodyne OXGR1 110 38 CC[C@@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851443 DD On-Demand Anodyne DOT1L 56 33 CC[C@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851445 DD On-Demand Anodyne AHCY 67 40 CC[C@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851445 DD On-Demand Anodyne OXGR1 110 38 CC[C@H]1CCC[C@@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851445 DD On-Demand Anodyne DOT1L 56 33 CC[C@H]1CCC[C@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851446 DD On-Demand Anodyne AHCY 67 40 CC[C@H]1CCC[C@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851446 DD On-Demand Anodyne OXGR1 110 38 CC[C@H]1CCC[C@]1(C)C(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851446 DD On-Demand Anodyne DOT1L 56 33 O=C1NCC[C@H]1CC(=O)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880851462 ED On-Demand Anodyne ETHR 22 41 O=C1NCC[C@@H]1CC(=O)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880851463 ED On-Demand Anodyne ETHR 22 41 C/C=C\CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851464 CD On-Demand Anodyne PAPA1_CARPA 41 51 C/C=C\CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851464 CD On-Demand Anodyne CTSK 19 52 C/C=C\CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851464 CD On-Demand Anodyne POLG_HCV1 17 40 C/C=C/CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851465 CD On-Demand Anodyne PAPA1_CARPA 41 51 C/C=C/CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851465 CD On-Demand Anodyne CTSK 19 52 C/C=C/CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851465 CD On-Demand Anodyne POLG_HCV1 17 40 C/C=C/CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851466 CD On-Demand Anodyne PAPA1_CARPA 41 51 C/C=C/CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851466 CD On-Demand Anodyne CTSK 19 52 C/C=C/CNC(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851466 CD On-Demand Anodyne POLG_HCV1 17 40 C/C=C\CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851467 CD On-Demand Anodyne PAPA1_CARPA 41 51 C/C=C\CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851467 CD On-Demand Anodyne CTSK 19 52 C/C=C\CNC(=O)[C@H](CCOC)NC(=O)OC(C)(C)C ZINC000880851467 CD On-Demand Anodyne POLG_HCV1 17 40 COc1cc(NC(=O)c2ccco2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880851486 IH On-Demand Anodyne GRM4 17 43 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne HCRTR1 38 48 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne CPT1A 48 34 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne CHRNA10 60 38 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne CASP7 51 35 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne HCRTR2 22 43 COC[C@@H]1CCCN1C(=O)c1cc2ccccc2cc1F ZINC000880851519 CG On-Demand Anodyne ACKR3 61 32 COC(=O)c1cc(NC(=O)NC(C)(C)CO)cc2ccccc12 ZINC000880851533 DF On-Demand Anodyne DHODH 15 40 COC(=O)c1cc(NC(=O)N2CCC[C@H](Cn3ccnn3)C2)cc2ccccc12 ZINC000880851537 GG On-Demand Anodyne CCR3 17 43 COC(=O)c1cc(NC(=O)N2CCC[C@@H](Cn3ccnn3)C2)cc2ccccc12 ZINC000880851539 GG On-Demand Anodyne CCR3 17 43 C=CC(C)(C)CC(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851564 CD On-Demand Mild AHCY 81 47 C=CC(C)(C)CC(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851564 CD On-Demand Mild OXGR1 106 38 C=CC(C)(C)CC(=O)NCCn1cnc2c(N)ncnc21 ZINC000880851564 CD On-Demand Mild DOT1L 56 35 COC[C@@H]1CCCN1C(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880851603 CF On-Demand Anodyne PREP 72 38 COC(=O)c1cc(NC(=O)N2CCC(F)(F)C2)cc2ccccc12 ZINC000880851605 EG On-Demand Anodyne CACNA1H 40 36 COC(=O)c1cc(NC(=O)N2CCC(F)(F)C2)cc2ccccc12 ZINC000880851605 EG On-Demand Anodyne EPHX2 33 40 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)C[S@@](C)=O)cc2ccccc12 ZINC000880851607 FF On-Demand Anodyne NPY5R 34 44 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)C[S@](C)=O)cc2ccccc12 ZINC000880851609 FF On-Demand Anodyne NPY5R 34 44 COC(=O)c1cc(NC(=O)N(C)[C@H](C)C[S@@](C)=O)cc2ccccc12 ZINC000880851611 FF On-Demand Anodyne NPY5R 34 44 COC(=O)c1cc(NC(=O)N(C)[C@H](C)C[S@](C)=O)cc2ccccc12 ZINC000880851613 FF On-Demand Anodyne NPY5R 34 44 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2CC[C@@H](C1)[S@@]2=O ZINC000880851622 FG On-Demand Anodyne L3MBTL3 53 36 COC(=O)c1cc(NC(=O)N2CCN(CCO)CC2)cc2ccccc12 ZINC000880851633 FD On-Demand Anodyne DRD3 22 40 COC(=O)c1cc(NC(=O)N2CCN(CCO)CC2)cc2ccccc12 ZINC000880851633 FD On-Demand Anodyne PDGFRB 44 37 COC(=O)c1cc(NC(=O)N2CCN(CCO)CC2)cc2ccccc12 ZINC000880851633 FD On-Demand Anodyne FAAH 15 45 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2CC[C@@H](C1)[S@]2=O ZINC000880851635 FG On-Demand Anodyne L3MBTL3 53 36 COC[C@@H]1CCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880851646 DE On-Demand Anodyne CASP3 37 40 COC[C@@H]1CCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880851646 DE On-Demand Anodyne MTNR1A 22 41 COC[C@@H]1CCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880851646 DE On-Demand Anodyne MTNR1B 24 42 COC[C@@H]1CCCN1C(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880851646 DE On-Demand Anodyne CASP7 48 40 COC[C@@H]1CCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880851648 DE On-Demand Anodyne CASP3 37 40 COC[C@@H]1CCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880851648 DE On-Demand Anodyne MTNR1A 22 41 COC[C@@H]1CCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880851648 DE On-Demand Anodyne MTNR1B 24 42 COC[C@@H]1CCCN1C(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880851648 DE On-Demand Anodyne CASP7 48 40 COC(=O)c1cc(NC(=O)N2CCC(O)(C(F)F)CC2)cc2ccccc12 ZINC000880851654 GG On-Demand Anodyne CACNA1H 41 35 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2CC[C@@H](C1)S2(=O)=O ZINC000880851665 DD On-Demand Anodyne L3MBTL3 43 35 CS(=O)(=O)C1CCC(C(=O)N2CCc3cccc(C(F)(F)F)c3C2)CC1 ZINC000880851681 GG On-Demand Anodyne SFRP1 83 33 CS(=O)(=O)C1CCC(C(=O)N2CCc3cccc(C(F)(F)F)c3C2)CC1 ZINC000880851681 GG On-Demand Anodyne WNT3 58 30 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne ACE 17 41 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne CELA1 20 43 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne PREP 32 43 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne LGMN 61 38 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne SLC12A5 45 35 C/C=C\CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851700 DE On-Demand Anodyne Q9NAW4_PLAFA 39 46 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne ACE 17 41 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne CELA1 20 43 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne PREP 32 43 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne LGMN 61 38 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne SLC12A5 45 35 C/C=C/CNC(=O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880851701 DE On-Demand Anodyne Q9NAW4_PLAFA 39 46 O=C(c1ccc(OC(F)F)c(Cl)c1)N1CC[C@H]2CC[C@@H](C1)S2(=O)=O ZINC000880851715 GF On-Demand Anodyne L3MBTL3 54 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne DRD4 43 33 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne MTNR1A 44 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne MTNR1B 42 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne MMP3 22 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne SSTR1 40 33 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1COCCN1C)C2 ZINC000880851718 DD On-Demand Anodyne MMP1 19 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne DRD4 43 33 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne MTNR1A 44 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne MTNR1B 42 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne MMP3 22 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne SSTR1 40 33 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1COCCN1C)C2 ZINC000880851720 DD On-Demand Anodyne MMP1 19 40 O=C(N[C@@H]1CCO[C@H]1c1ccc(O)nc1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880851742 GG On-Demand Anodyne PDE4D 18 42 COC(=O)c1cc(NC(=O)N(C)CCNC(=O)C(C)C)cc2ccccc12 ZINC000880851794 FF On-Demand Anodyne NQO2 27 42 COC(=O)c1cc(NC(=O)N(C)CCNC(=O)C(C)C)cc2ccccc12 ZINC000880851794 FF On-Demand Anodyne MTNR1A 20 42 COC[C@@H]1CCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880851829 DD On-Demand Anodyne HCRTR1 24 41 COC[C@@H]1CCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880851829 DD On-Demand Anodyne CASP7 45 38 COC(=O)c1cc(NC(=O)NC[C@H]2CCN(C)C2)cc2ccccc12 ZINC000880851837 EF On-Demand Anodyne HTR4 43 34 COC(=O)c1cc(NC(=O)NC[C@H]2CCN(C)C2)cc2ccccc12 ZINC000880851837 EF On-Demand Anodyne CCR3 58 41 COC(=O)c1cc(NC(=O)NC[C@H]2CCN(C)C2)cc2ccccc12 ZINC000880851837 EF On-Demand Anodyne CACNA1I 42 34 COC(=O)c1cc(NC(=O)NC[C@@H]2CCN(C)C2)cc2ccccc12 ZINC000880851838 EF On-Demand Anodyne HTR4 43 34 COC(=O)c1cc(NC(=O)NC[C@@H]2CCN(C)C2)cc2ccccc12 ZINC000880851838 EF On-Demand Anodyne CCR3 58 41 COC(=O)c1cc(NC(=O)NC[C@@H]2CCN(C)C2)cc2ccccc12 ZINC000880851838 EF On-Demand Anodyne CACNA1I 42 34 COC[C@@H]1CCCN1C(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880851840 EF On-Demand Anodyne HCRTR1 25 43 COC[C@@H]1CCCN1C(=O)c1ccc(-c2ccccc2OC)nc1O ZINC000880851840 EF On-Demand Anodyne HCRTR2 17 43 COC(=O)c1cc(NC(=O)NCCCC(=O)NC2CC2)cc2ccccc12 ZINC000880851846 FF On-Demand Anodyne TNKS 57 34 COC(=O)c1cc(NC(=O)N(C)[C@H](C)CC#N)cc2ccccc12 ZINC000880851849 EG On-Demand Mild DHODH 17 40 COC(=O)c1cc(NC(=O)N(C)[C@H](C)CC#N)cc2ccccc12 ZINC000880851849 EG On-Demand Mild NPY5R 32 41 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)CC#N)cc2ccccc12 ZINC000880851850 EG On-Demand Mild DHODH 17 40 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)CC#N)cc2ccccc12 ZINC000880851850 EG On-Demand Mild NPY5R 32 41 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne HTR1A 19 40 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne DRD4 42 32 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne DRD3 31 44 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne HTR4 63 36 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne NPY1R 24 40 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne CCR3 68 43 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne PLD1 56 37 COC(=O)c1cc(NC(=O)NCCN2CCC(OC)CC2)cc2ccccc12 ZINC000880851851 GF On-Demand Anodyne PLD2 76 37 COC(=O)c1cc(NC(=O)N2CCC(NC(=O)C3CC3)CC2)cc2ccccc12 ZINC000880851861 GG On-Demand Anodyne EPHX2 43 43 COC(=O)c1cc(NC(=O)N2CCC(NC(=O)C3CC3)CC2)cc2ccccc12 ZINC000880851861 GG On-Demand Anodyne CCR8 71 34 COC(=O)c1cc(NC(=O)N2CCC[C@H]2c2noc(C)n2)cc2ccccc12 ZINC000880851872 GH On-Demand Anodyne CPT1A 51 40 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2c2noc(C)n2)cc2ccccc12 ZINC000880851873 GH On-Demand Anodyne CPT1A 51 40 COC(=O)c1cc(NC(=O)N2CC[C@@H](O)C2)cc2ccccc12 ZINC000880851876 DE On-Demand Anodyne CCR8 43 31 COC(=O)c1cc(NC(=O)N2CC[C@H](O)C2)cc2ccccc12 ZINC000880851877 DE On-Demand Anodyne CCR8 43 31 COC(=O)c1cc(NC(=O)N2CCc3c(ncn3C)C2)cc2ccccc12 ZINC000880851880 FF On-Demand Anodyne P2RY14 47 34 COC[C@@H]1CCCN1C(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880851881 EG On-Demand Anodyne HRH3 19 43 COC[C@@H]1CCCN1C(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880851892 DF On-Demand Anodyne CPT1A 74 42 COC[C@@H]1CCCN1C(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880851892 DF On-Demand Anodyne CHRNA10 44 37 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2C(=O)N(C)C)cc2ccccc12 ZINC000880851895 FF On-Demand Anodyne AVPR2 17 43 COC(=O)c1cc(NC(=O)N2CCC[C@@H]2C(=O)N(C)C)cc2ccccc12 ZINC000880851895 FF On-Demand Anodyne UL80 40 38 CNC(=O)CN1CCC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880851903 GD On-Demand Anodyne DRD4 30 46 CNC(=O)CN1CCC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880851903 GD On-Demand Anodyne EPHX2 38 45 CNC(=O)CN1CCC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880851903 GD On-Demand Anodyne CXCR3 21 44 CNC(=O)CN1CCC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880851903 GD On-Demand Anodyne MCHR1 21 42 CNC(=O)CN1CCC(NC(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880851903 GD On-Demand Anodyne CCR8 47 34 Cn1nnc(C(=O)Nc2cccc(C3CCOCC3)c2)n1 ZINC000880851907 CD On-Demand Anodyne MCHR1 26 41 O=C(Nc1cccc(C2CCOCC2)c1)c1ccc(CN2CCOCC2)o1 ZINC000880851908 FG On-Demand Anodyne EPHX2 23 44 O=C(Nc1cccc(C2CCOCC2)c1)c1ccc(CN2CCOCC2)o1 ZINC000880851908 FG On-Demand Anodyne MCHR1 36 46 COC(=O)c1cc(NC(=O)N2CC[C@H](N3CC=CC3)C2)cc2ccccc12 ZINC000880851914 FG On-Demand Anodyne CCR8 55 32 COC(=O)c1cc(NC(=O)N2CC[C@@H](N3CC=CC3)C2)cc2ccccc12 ZINC000880851915 FG On-Demand Anodyne CCR8 55 32 C=CC(C)(C)CC(=O)Nc1n[nH]c(C)c1-c1ccccc1F ZINC000880851930 DI On-Demand Mild GSK3A 18 43 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3Cc4ccccc4NC3=O)cc2)N1 ZINC000880851931 ED On-Demand Anodyne PYGM 33 48 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3Cc4ccccc4NC3=O)cc2)N1 ZINC000880851932 ED On-Demand Anodyne PYGM 33 48 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3Cc4ccccc4NC3=O)cc2)N1 ZINC000880851933 ED On-Demand Anodyne PYGM 33 48 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3Cc4ccccc4NC3=O)cc2)N1 ZINC000880851934 ED On-Demand Anodyne PYGM 33 48 O=C(C[C@@H]1C[C@H]1C1CC1)Nc1cccc(C2CCOCC2)c1 ZINC000880851940 CH On-Demand Anodyne MCHR1 18 40 C=CC(C)(C)CC(=O)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880851954 EH On-Demand Mild ETHR 37 42 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@H]2Cc3c(Cl)cccc3[C@H]21 ZINC000880851961 GG On-Demand Anodyne KCNQ2 42 43 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1[C@@H]2c3cccc(Cl)c3C[C@H]21 ZINC000880851962 GG On-Demand Anodyne KCNQ2 42 43 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@@H]2Cc3c(Cl)cccc3[C@@H]21 ZINC000880851963 GG On-Demand Anodyne KCNQ2 42 43 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1[C@H]2Cc3c(Cl)cccc3[C@@H]21 ZINC000880851965 GG On-Demand Anodyne KCNQ2 42 43 COc1ccc2c(c1)CC[C@H](C(=O)NNCC(F)(F)C(F)(F)F)C2 ZINC000880851968 FF On-Demand Reactive NQO2 25 44 COc1ccc2c(c1)CC[C@H](C(=O)NNCC(F)(F)C(F)(F)F)C2 ZINC000880851968 FF On-Demand Reactive MTNR1B 29 41 Cc1nc(C(C)C)ncc1C(=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880851996 DE On-Demand Anodyne PYGL 24 48 Cc1nc(C(C)C)ncc1C(=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880851996 DE On-Demand Anodyne PYGM 31 46 NC(=O)c1cc(-c2csc(NC(=O)Cn3c(S)nc4ccccc4c3=O)n2)c[nH]1 ZINC000880852001 ID On-Demand Anodyne TRPA1 15 45 Cc1nc(C(C)C)ncc1C(=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880852005 DE On-Demand Anodyne PYGL 24 48 Cc1nc(C(C)C)ncc1C(=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880852005 DE On-Demand Anodyne PYGM 31 46 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2CC[C@@H](C1)[S@]2=O ZINC000880852008 DD On-Demand Anodyne L3MBTL3 44 36 O=C(c1cnc2cc[nH]c2c1)N1CC[C@H]2CC[C@@H](C1)[S@@]2=O ZINC000880852009 DD On-Demand Anodyne L3MBTL3 44 36 Cn1nc(C2CCOCC2)cc1NC(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880852047 FF On-Demand Anodyne HTR1F 40 33 Cn1nc(C2CCOCC2)cc1NC(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880852047 FF On-Demand Anodyne WNT3A 40 33 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCO[C@H]1c1ccc(O)nc1)C2 ZINC000880852073 FF On-Demand Anodyne FAAH 15 42 O=C(c1ncsc1C1CC1)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880852097 FH On-Demand Anodyne ETHR 42 34 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852191 EG On-Demand Anodyne CCR2 29 41 COC(=O)c1cc(NC(=O)N2CCC[C@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880852247 GH On-Demand Anodyne SMO 36 41 COC(=O)c1cc(NC(=O)N2CCC[C@@H](c3nc(C)no3)C2)cc2ccccc12 ZINC000880852248 GH On-Demand Anodyne SMO 36 41 COC(=O)c1cc(NC(=O)N2CCN(c3cnn(C)c3)CC2)cc2ccccc12 ZINC000880852257 GF On-Demand Anodyne PDGFRB 51 39 COC(=O)c1cc(NC(=O)N2CCC(C3OCCO3)CC2)cc2ccccc12 ZINC000880852260 GG On-Demand Anodyne RBP4 15 41 COC(=O)c1cc(NC(=O)N2CCN(C[C@@H](C)O)CC2)cc2ccccc12 ZINC000880852262 FE On-Demand Anodyne PDGFRB 41 34 COC(=O)c1cc(NC(=O)N2CCN(C[C@@H](C)O)CC2)cc2ccccc12 ZINC000880852262 FE On-Demand Anodyne ABCB1 20 41 O=C(N[C@@H]1Cc2ccccc2NC1=O)c1ncsc1C1CC1 ZINC000880852265 DE On-Demand Anodyne PYGM 31 47 O=C(N[C@H]1Cc2ccccc2NC1=O)c1ncsc1C1CC1 ZINC000880852266 DE On-Demand Anodyne PYGM 31 47 Cn1nc2c(c1C(=O)N[C@H]1Cc3ccccc3NC1=O)CSCC2 ZINC000880852270 ED On-Demand Anodyne PYGL 27 45 Cn1nc2c(c1C(=O)N[C@H]1Cc3ccccc3NC1=O)CSCC2 ZINC000880852270 ED On-Demand Anodyne PYGM 32 42 Cn1nc2c(c1C(=O)N[C@@H]1Cc3ccccc3NC1=O)CSCC2 ZINC000880852271 ED On-Demand Anodyne PYGL 27 45 Cn1nc2c(c1C(=O)N[C@@H]1Cc3ccccc3NC1=O)CSCC2 ZINC000880852271 ED On-Demand Anodyne PYGM 32 42 O=C1CC[C@@H](c2ccc(C(=O)Nc3cccc(C4CCOCC4)c3)cc2)N1 ZINC000880852304 FH On-Demand Anodyne KCNK3 73 39 O=C1CC[C@H](c2ccc(C(=O)Nc3cccc(C4CCOCC4)c3)cc2)N1 ZINC000880852309 FH On-Demand Anodyne KCNK3 73 39 Cc1ncc(CC(=O)Nc2cccc3c2OC(C)(C)CC3)o1 ZINC000880852315 DG On-Demand Anodyne G2YM83_BOTF4 47 52 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852336 DI On-Demand Anodyne CCR2 19 41 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852336 DI On-Demand Anodyne LIPG 46 32 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne DRD2 15 45 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne DRD4 23 45 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne DRD3 21 45 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne HTR4 49 42 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne CCR3 46 39 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne EPHX2 41 47 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne CXCR3 22 49 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne MCHR1 30 42 COC(=O)c1cc(NC(=O)NC2CCN(CCO)CC2)cc2ccccc12 ZINC000880852337 FE On-Demand Anodyne SHH 18 40 O=C(c1cc2ccccc2cc1F)N1CC[C@H]2CC[C@@H](C1)[S@@]2=O ZINC000880852340 EG On-Demand Anodyne L3MBTL3 43 38 O=C(c1cc2ccccc2cc1F)N1CC[C@H]2CC[C@@H](C1)[S@]2=O ZINC000880852341 EG On-Demand Anodyne L3MBTL3 43 38 CS(=O)(=O)C1CCC(C(=O)NNc2ccnc(C(F)(F)F)c2)CC1 ZINC000880852390 FE On-Demand Reactive TYK2 49 35 CS(=O)(=O)C1CCC(C(=O)NNc2ccnc(C(F)(F)F)c2)CC1 ZINC000880852390 FE On-Demand Reactive SFRP1 84 33 CS(=O)(=O)C1CCC(C(=O)NNc2ccnc(C(F)(F)F)c2)CC1 ZINC000880852390 FE On-Demand Reactive WNT3 40 31 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(F)c(Cl)c1 ZINC000880852441 GF On-Demand Reactive PAPA1_CARPA 37 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNc1ccc(F)c(Cl)c1 ZINC000880852442 GF On-Demand Reactive PAPA1_CARPA 37 42 CSc1nccnc1C(=O)Nc1cccc2c1OC(C)(C)CC2 ZINC000880852494 EH On-Demand Anodyne G2YM83_BOTF4 80 60 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCO[C@H](CCF)C1 ZINC000880852515 FG On-Demand Anodyne PIK3CB 39 40 O=C(c1cc2cccc(C(F)(F)F)c2nc1O)N1CCO[C@@H](CCF)C1 ZINC000880852517 FG On-Demand Anodyne PIK3CB 39 40 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCc2cccc(C(F)(F)F)c2C1 ZINC000880852524 EG On-Demand Anodyne RBP4 41 33 Cn1nc(C2CCOCC2)cc1NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880852563 GH On-Demand Anodyne PDE4D 24 45 O=C(Nc1cccc(C2CCOCC2)c1)[C@H]1CCc2nncn2CC1 ZINC000880852564 EF On-Demand Anodyne EPHX2 16 41 O=C(Nc1cccc(C2CCOCC2)c1)[C@H]1CCc2nncn2CC1 ZINC000880852564 EF On-Demand Anodyne MCHR1 24 43 O=C(Nc1cccc(C2CCOCC2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880852565 EF On-Demand Anodyne EPHX2 16 41 O=C(Nc1cccc(C2CCOCC2)c1)[C@@H]1CCc2nncn2CC1 ZINC000880852565 EF On-Demand Anodyne MCHR1 24 43 COC(=O)c1cc(NC(=O)N2CCC3(CCOCC3)C2)cc2ccccc12 ZINC000880852574 FH On-Demand Anodyne EPHX2 36 44 COC(=O)c1cc(NC(=O)N2CCC(CNC(C)=O)CC2)cc2ccccc12 ZINC000880852594 GG On-Demand Anodyne HTR4 50 35 COC(=O)c1cc(NC(=O)N2CCC(CNC(C)=O)CC2)cc2ccccc12 ZINC000880852594 GG On-Demand Anodyne EPHX2 16 41 COC(=O)c1cc(NC(=O)NCCNC(=O)C2CC2)cc2ccccc12 ZINC000880852612 FE On-Demand Anodyne MTNR1A 30 44 CC1(C)[C@@H](c2cccc(F)c2)CCN1C(=O)c1ccc(CN2CCOCC2)o1 ZINC000880852671 GH On-Demand Anodyne CCR5 51 31 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852685 GF On-Demand Anodyne CCR2 23 40 COC(=O)c1cc(NC(=O)N2CCC(N(C)C(C)=O)CC2)cc2ccccc12 ZINC000880852757 GG On-Demand Anodyne RBP4 18 41 COC(=O)c1cc(NC(=O)N(C)[C@H](C)CS(C)(=O)=O)cc2ccccc12 ZINC000880852774 GF On-Demand Anodyne NPY5R 32 41 COC(=O)c1cc(NC(=O)N(C)[C@@H](C)CS(C)(=O)=O)cc2ccccc12 ZINC000880852779 GF On-Demand Anodyne NPY5R 32 41 COC(=O)c1cc(NC(=O)N2CC[C@H](N(C)C)C2)cc2ccccc12 ZINC000880852784 EF On-Demand Anodyne RBP4 17 40 COC(=O)c1cc(NC(=O)N2CC[C@@H](N(C)C)C2)cc2ccccc12 ZINC000880852789 EF On-Demand Anodyne RBP4 17 40 CS(=O)(=O)C1CCC(C(=O)N[C@@H]2Cc3ccccc3NC2=O)CC1 ZINC000880852791 FD On-Demand Anodyne PYGM 18 44 CS(=O)(=O)C1CCC(C(=O)N[C@H]2Cc3ccccc3NC2=O)CC1 ZINC000880852795 FD On-Demand Anodyne PYGM 18 44 COC(=O)c1cc(NC(=O)NCCNC(=O)C(C)C)cc2ccccc12 ZINC000880852816 FF On-Demand Anodyne NQO2 30 43 COC(=O)c1cc(NC(=O)NCCNC(=O)C(C)C)cc2ccccc12 ZINC000880852816 FF On-Demand Anodyne CA1 15 43 COC(=O)c1cc(NC(=O)NCCNC(=O)C(C)C)cc2ccccc12 ZINC000880852816 FF On-Demand Anodyne MTNR1A 25 43 O=C(COC1CC1)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880852819 DE On-Demand Anodyne ETHR 27 42 O=C(COC1CC1)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852820 CF On-Demand Anodyne CCR2 24 40 O=C(COC1CC1)N1CCc2cc(C(F)(F)F)ccc2C1 ZINC000880852820 CF On-Demand Anodyne LIPG 56 42 CCc1nnc2n1CCN(C(=O)Nc1cc(C(=O)OC)c3ccccc3c1)C2 ZINC000880852830 GF On-Demand Anodyne P2RY14 43 33 CS(=O)(=O)C1CCC(C(=O)N2CCc3cc(C(F)(F)F)ccc3C2)CC1 ZINC000880852831 GG On-Demand Anodyne CACNA1B 47 37 CS(=O)(=O)C1CCC(C(=O)N2CCc3cc(C(F)(F)F)ccc3C2)CC1 ZINC000880852831 GG On-Demand Anodyne CCR2 26 41 Cc1coc(C(=O)Nc2cccc(C3CCOCC3)c2)c1 ZINC000880852856 CH On-Demand Anodyne MCHR1 23 40 Cc1coc(C(=O)Nc2cccc(C3CCOCC3)c2)c1 ZINC000880852856 CH On-Demand Anodyne KCNK3 91 41 Cc1coc(C(=O)Nc2cccc(C3CCOCC3)c2)c1 ZINC000880852856 CH On-Demand Anodyne KCNK9 47 38 O=C(CN1CCCCS1(=O)=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880852869 EC On-Demand Anodyne PYGL 16 48 O=C(CN1CCCCS1(=O)=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880852869 EC On-Demand Anodyne PYGM 24 48 O=C(CN1CCCCS1(=O)=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880852870 EC On-Demand Anodyne PYGL 16 48 O=C(CN1CCCCS1(=O)=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880852870 EC On-Demand Anodyne PYGM 24 48 COC(=O)c1cc(NC(=O)N2CCC(N(C)CCCO)CC2)cc2ccccc12 ZINC000880852884 GF On-Demand Anodyne CCR8 42 33 Cn1ncc(Br)c1CC(=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880852893 FD On-Demand Anodyne PYGM 27 41 Cn1ncc(Br)c1CC(=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880852894 FD On-Demand Anodyne PYGM 27 41 COC(=O)c1cc(NC(=O)N2CCn3c(C)nnc3C2)cc2ccccc12 ZINC000880852895 FF On-Demand Anodyne P2RX7 19 40 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880852909 GD On-Demand Anodyne MMP2 48 37 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880852910 GD On-Demand Anodyne MMP2 48 37 COC(=O)c1cc(NC(=O)N2CCC(c3ncc[nH]3)CC2)cc2ccccc12 ZINC000880852913 GH On-Demand Anodyne RBP4 18 40 COC(=O)c1cc(NC(=O)N2CC[C@@H](C(=O)OC)C2)cc2ccccc12 ZINC000880852919 FF On-Demand Anodyne CCR8 60 33 COC(=O)c1cc(NC(=O)N2CC[C@H](C(=O)OC)C2)cc2ccccc12 ZINC000880852920 FF On-Demand Anodyne CCR8 60 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(C2CCOCC2)c1 ZINC000880852921 GG On-Demand Anodyne HDAC11 44 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(C2CCOCC2)c1 ZINC000880852922 GG On-Demand Anodyne HDAC11 44 38 Cn1nnc(C(=O)Nc2cccc3c2OC(C)(C)CC3)n1 ZINC000880852950 CD On-Demand Anodyne G2YM83_BOTF4 56 56 O=C(NNc1ccc(F)c(Cl)c1)c1ccc(CN2CCOCC2)o1 ZINC000880852951 FF On-Demand Reactive EGFR 19 44 O=C(NNc1ccc(F)c(Cl)c1)c1ccc(CN2CCOCC2)o1 ZINC000880852951 FF On-Demand Reactive EPHX2 15 41 O=C(NNc1ccc(F)c(Cl)c1)c1ccc(CN2CCOCC2)o1 ZINC000880852951 FF On-Demand Reactive DPOL_VZVD 23 40 CS(=O)(=O)C1CCC(C(=O)NNc2ccc(F)c(Cl)c2)CC1 ZINC000880852975 EF On-Demand Reactive EPHX2 31 40 O=C(NNc1ccc(F)c(Cl)c1)c1cnc(CC2CC2)s1 ZINC000880852985 EH On-Demand Reactive ERBB4 51 35 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCC(Cc2nc(C3CCC3)no2)CC1 ZINC000880853005 EH On-Demand Anodyne ETHR 17 40 O=C(N[C@@H]1CCO[C@H]1c1ccncc1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880853015 FH On-Demand Anodyne PDE4D 24 43 COC(=O)c1cc(NC(=O)N2CCC(CO)CC2)cc2ccccc12 ZINC000880853110 EF On-Demand Anodyne CCR8 42 36 Cc1coc(C(=O)NC[C@@H]2COCCN2C(=O)OC(C)(C)C)c1 ZINC000880853118 DD On-Demand Anodyne CACNA1I 40 32 Cc1coc(C(=O)NC[C@H]2COCCN2C(=O)OC(C)(C)C)c1 ZINC000880853119 DD On-Demand Anodyne CACNA1I 40 32 Cc1cnc(Cl)c(C(=O)NC[C@@H]2COCCN2C(=O)OC(C)(C)C)c1 ZINC000880853125 FE On-Demand Anodyne CACNA1I 57 34 Cc1cnc(Cl)c(C(=O)NC[C@H]2COCCN2C(=O)OC(C)(C)C)c1 ZINC000880853126 FE On-Demand Anodyne CACNA1I 57 34 CCC1(O)CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880853140 FG On-Demand Anodyne S1PR2 31 45 COC(=O)c1cc(NC(=O)N2CCC(N3CCCC3=O)CC2)cc2ccccc12 ZINC000880853148 GG On-Demand Anodyne SCD1 16 41 O=C(N[C@H]1Cc2ccccc2NC1=O)c1ccc(CN2CCOCC2)o1 ZINC000880853157 FD On-Demand Anodyne PYGM 20 43 O=C(N[C@@H]1Cc2ccccc2NC1=O)c1ccc(CN2CCOCC2)o1 ZINC000880853158 FD On-Demand Anodyne PYGM 20 43 COC(=O)c1cc(NC(=O)N2CCC(NC(=O)C(C)C)CC2)cc2ccccc12 ZINC000880853166 GG On-Demand Anodyne EPHX2 29 41 COC(=O)c1cc(NC(=O)N2CCC(NC(=O)C(C)C)CC2)cc2ccccc12 ZINC000880853166 GG On-Demand Anodyne RBP4 18 41 COC(=O)c1cc(NC(=O)N2CCC(NC(=O)C(C)C)CC2)cc2ccccc12 ZINC000880853166 GG On-Demand Anodyne CCR8 70 34 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880853174 GG On-Demand Anodyne PDE4D 25 44 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880853176 GG On-Demand Anodyne PDE4D 25 44 COC(=O)c1cc(NC(=O)N2CC[C@H](CCO)C2)cc2ccccc12 ZINC000880853179 EF On-Demand Anodyne CCR8 58 32 COC(=O)c1cc(NC(=O)N2CC[C@@H](CCO)C2)cc2ccccc12 ZINC000880853180 EF On-Demand Anodyne CCR8 58 32 O=C(Nc1cccc(C2CCOCC2)c1)c1cccn2nccc12 ZINC000880853186 DG On-Demand Anodyne KCNK3 66 33 O=C(Nc1cccc(C2CCOCC2)c1)c1cccn2nccc12 ZINC000880853186 DG On-Demand Anodyne KCNK9 47 33 O=C(Cc1ccccc1N1CCCC1=O)Nc1cccc(C2CCOCC2)c1 ZINC000880853191 GH On-Demand Anodyne MCHR1 28 44 COC(=O)c1cc(NC(=O)N2CCC(c3cc[nH]n3)CC2)cc2ccccc12 ZINC000880853248 GH On-Demand Anodyne RBP4 19 41 COC(=O)c1cc(NC(=O)N2CCC(c3cc[nH]n3)CC2)cc2ccccc12 ZINC000880853248 GH On-Demand Anodyne SMO 20 40 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1cc2ccccc2cc1F ZINC000880853251 FG On-Demand Anodyne CTSL 15 41 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1cc2ccccc2cc1F ZINC000880853251 FG On-Demand Anodyne CTSS 36 41 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1cc2ccccc2cc1F ZINC000880853252 FG On-Demand Anodyne CTSL 15 41 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1cc2ccccc2cc1F ZINC000880853252 FG On-Demand Anodyne CTSS 36 41 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880853254 GF On-Demand Anodyne NPY5R 32 42 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880853255 GF On-Demand Anodyne NPY5R 32 42 COC(=O)c1cc(NC(=O)NC2CCOCC2)cc2ccccc12 ZINC000880853260 EF On-Demand Anodyne EPHX2 37 42 COC(=O)c1cc(NC(=O)N2CCC(CCO)CC2)cc2ccccc12 ZINC000880853271 FG On-Demand Anodyne EPHX2 15 44 COC(=O)c1cc(NC(=O)N2CCC(CCO)CC2)cc2ccccc12 ZINC000880853271 FG On-Demand Anodyne RBP4 18 41 COC(=O)c1cc(NC(=O)N2CCC(CCO)CC2)cc2ccccc12 ZINC000880853271 FG On-Demand Anodyne CCR8 66 37 COC(=O)[C@@H](C[C@@H]1CCCOC1)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880853280 GG On-Demand Anodyne CTSS 15 40 COC(=O)[C@@H](C[C@H]1CCCOC1)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880853281 GG On-Demand Anodyne CTSS 15 40 COC(=O)c1cc(NC(=O)NC2CCN(C(=O)C3CC3)CC2)cc2ccccc12 ZINC000880853282 GG On-Demand Anodyne EPHX2 53 53 COC(=O)c1cc(NC(=O)NC2CCN(C(=O)C3CC3)CC2)cc2ccccc12 ZINC000880853282 GG On-Demand Anodyne CCR8 74 41 COC(=O)c1cc(NC(=O)NC2CC2)cc2ccccc12 ZINC000880853298 CF On-Demand Anodyne EPHX2 51 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880853303 FF On-Demand Anodyne PAPA1_CARPA 36 46 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880853304 FF On-Demand Anodyne PAPA1_CARPA 36 46 COC(=O)c1cc(NC(=O)NCC(=O)NC2CC2)cc2ccccc12 ZINC000880853317 EE On-Demand Anodyne EPHX2 20 41 COC(=O)c1cc(NC(=O)NCC(=O)NC2CC2)cc2ccccc12 ZINC000880853317 EE On-Demand Anodyne TNKS 44 30 C[C@@]1(CO)CN(C(=O)C(=O)c2c[nH]c3cc(F)ccc23)C[C@]1(C)CO ZINC000880853328 ED On-Demand Anodyne MPO 74 36 CC(C)(C)OC(=O)N1CCN(C(=O)Cc2csc(COc3ccc(Cl)cc3)n2)CC1 ZINC000880853371 JH On-Demand Anodyne GPR119 38 42 C[C@@H]1O[C@H](C)[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@H]1C ZINC000880853377 DE On-Demand Anodyne GABRA1 18 42 C[C@@H]1O[C@H](C)[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@H]1C ZINC000880853377 DE On-Demand Anodyne GABRA2 16 42 C[C@@H]1O[C@H](C)[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@@H]1C ZINC000880853378 DE On-Demand Anodyne GABRA1 18 42 C[C@@H]1O[C@H](C)[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@@H]1C ZINC000880853378 DE On-Demand Anodyne GABRA2 16 42 C[C@@H]1O[C@H](C)[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@H]1C ZINC000880853379 DE On-Demand Anodyne GABRA1 18 42 C[C@@H]1O[C@H](C)[C@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@H]1C ZINC000880853379 DE On-Demand Anodyne GABRA2 16 42 C[C@@H]1O[C@H](C)[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@@H]1C ZINC000880853380 DE On-Demand Anodyne GABRA1 18 42 C[C@@H]1O[C@H](C)[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)[C@@H]1C ZINC000880853380 DE On-Demand Anodyne GABRA2 16 42 CCOC(=O)C1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880853395 GG On-Demand Anodyne P2RY12 21 41 CCOC(=O)C1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880853395 GG On-Demand Anodyne CCR8 64 36 CCOC(=O)C1CCN(C(=O)Nc2cc(C(=O)OC)c3ccccc3c2)CC1 ZINC000880853395 GG On-Demand Anodyne P2RY14 42 31 CS(=O)(=O)C1CCC(C(=O)N2CCN(c3cccc4[nH]ccc34)CC2)CC1 ZINC000880853396 GE On-Demand Anodyne SSTR1 46 33 CS(=O)(=O)C1CCC(C(=O)N2CCN(c3cccc4[nH]ccc34)CC2)CC1 ZINC000880853396 GE On-Demand Anodyne MAPK9 19 50 CS(=O)(=O)C1CCC(C(=O)N2CCN(c3cccc4[nH]ccc34)CC2)CC1 ZINC000880853396 GE On-Demand Anodyne MAPK8 22 50 COC(=O)c1cc(NC(=O)NCCCO)cc2ccccc12 ZINC000880853448 DE On-Demand Anodyne CA1 18 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@H]1c1ccsc1)C2 ZINC000880853478 EH On-Demand Anodyne NPBWR1 84 36 Cc1cnc(Cl)c(C(=O)NC[C@H]2CCN2C2CCCC2)c1 ZINC000880853480 DF On-Demand Anodyne CACNA1I 54 35 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CCN2C2CCCC2)c1 ZINC000880853481 DF On-Demand Anodyne CACNA1I 54 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN1C1CCCC1)C2 ZINC000880853483 EF On-Demand Anodyne MTNR1A 38 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCN1C1CCCC1)C2 ZINC000880853483 EF On-Demand Anodyne MTNR1B 37 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN1C1CCCC1)C2 ZINC000880853486 EF On-Demand Anodyne MTNR1A 38 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CCN1C1CCCC1)C2 ZINC000880853486 EF On-Demand Anodyne MTNR1B 37 40 COC(=O)C[C@@H](O)CNC(=O)c1ncsc1C1CC1 ZINC000880853522 CC On-Demand Anodyne MAP1 48 37 COC(=O)C[C@H](O)CNC(=O)c1ncsc1C1CC1 ZINC000880853523 CC On-Demand Anodyne MAP1 48 37 Cc1nc(C(C)C)ncc1C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880853531 DG On-Demand Anodyne NPBWR1 64 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C1CCCC1 ZINC000880853557 FE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C1CCCC1 ZINC000880853558 FE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCN1C1CCCC1 ZINC000880853559 FE On-Demand Anodyne PAPA1_CARPA 35 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCN1C1CCCC1 ZINC000880853560 FE On-Demand Anodyne PAPA1_CARPA 35 43 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853571 GG On-Demand Anodyne DRD2 42 40 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853571 GG On-Demand Anodyne DRD3 32 49 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853571 GG On-Demand Anodyne HTR3A 16 44 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853571 GG On-Demand Anodyne HCN1 51 34 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853571 GG On-Demand Anodyne HCN4 50 34 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853572 GG On-Demand Anodyne DRD2 42 40 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853572 GG On-Demand Anodyne DRD3 32 49 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853572 GG On-Demand Anodyne HTR3A 16 44 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853572 GG On-Demand Anodyne HCN1 51 34 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCN2C2CCCC2)c(O)n1 ZINC000880853572 GG On-Demand Anodyne HCN4 50 34 CC1(C)CC[C@@H](CC(=O)N[C@@H]2C[C@H]2c2ccsc2)OC1 ZINC000880853582 CG On-Demand Anodyne NPBWR1 44 31 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@H]2CCN2C2CCCC2)N1Cc1ccccc1 ZINC000880853587 GD On-Demand Anodyne TMPRSS11D 50 32 NC(=O)[C@@H]1CC[C@H](C(=O)NC[C@@H]2CCN2C2CCCC2)N1Cc1ccccc1 ZINC000880853588 GD On-Demand Anodyne TMPRSS11D 50 32 COC(=O)c1cc(NC(=O)NC2CCN(C)CC2)cc2ccccc12 ZINC000880853612 EF On-Demand Anodyne EPHX2 48 48 COC(=O)c1cc(NC(=O)NC2CCN(C)CC2)cc2ccccc12 ZINC000880853612 EF On-Demand Anodyne CXCR3 19 44 C[C@@]1(CO)CN(C(=O)CC[C@H]2CCc3ccccc32)C[C@]1(C)CO ZINC000880853613 EE On-Demand Anodyne EBP 18 42 C[C@@]1(CO)CN(C(=O)CC[C@@H]2CCc3ccccc32)C[C@]1(C)CO ZINC000880853614 EE On-Demand Anodyne EBP 18 42 COC(=O)c1cc(NC(=O)NC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880853655 FF On-Demand Anodyne EPHX2 59 53 COC(=O)c1cc(NC(=O)NC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880853655 FF On-Demand Anodyne CXCR3 19 45 COC(=O)c1cc(NC(=O)NC2CCN(C(C)=O)CC2)cc2ccccc12 ZINC000880853655 FF On-Demand Anodyne CCR8 79 39 COC(=O)C[C@@H](O)CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880853737 EC On-Demand Anodyne KCNQ2 44 33 COC(=O)C[C@H](O)CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880853738 EC On-Demand Anodyne KCNQ2 44 33 COC(=O)C[C@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853739 DD On-Demand Anodyne NQO2 21 43 COC(=O)C[C@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853739 DD On-Demand Anodyne MTNR1A 21 40 COC(=O)C[C@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853739 DD On-Demand Anodyne MTNR1B 22 40 COC(=O)C[C@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853740 DD On-Demand Anodyne NQO2 21 43 COC(=O)C[C@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853740 DD On-Demand Anodyne MTNR1A 21 40 COC(=O)C[C@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853740 DD On-Demand Anodyne MTNR1B 22 40 COC(=O)C[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853741 DD On-Demand Anodyne NQO2 21 43 COC(=O)C[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853741 DD On-Demand Anodyne MTNR1A 21 40 COC(=O)C[C@@H](O)CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880853741 DD On-Demand Anodyne MTNR1B 22 40 COC(=O)C[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853742 DD On-Demand Anodyne NQO2 21 43 COC(=O)C[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853742 DD On-Demand Anodyne MTNR1A 21 40 COC(=O)C[C@@H](O)CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880853742 DD On-Demand Anodyne MTNR1B 22 40 O=C(COC1CC1)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880853831 CD On-Demand Anodyne HTR1A 20 46 O=C(COC1CC1)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880853831 CD On-Demand Anodyne HTR1D 17 43 O=C(COC1CC1)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880853831 CD On-Demand Anodyne HTR1B 21 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H](C)O[C@H](C)[C@H]1C ZINC000880853884 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H](C)O[C@H](C)[C@@H]1C ZINC000880853885 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H](C)O[C@@H](C)[C@@H]1C ZINC000880853886 ED On-Demand Anodyne PAPA1_CARPA 34 42 Cc1cnc(Cl)c(C(=O)NCC2(C)C[C@H]3C[C@@H]3C2)c1 ZINC000880853899 CG On-Demand Anodyne P2RX7 19 40 Cc1cnc(Cl)c(C(=O)NC[C@@]2(C)C[C@@H]3C[C@@H]3C2)c1 ZINC000880853900 CG On-Demand Anodyne P2RX7 19 40 Cc1cnc(Cl)c(C(=O)NCC2(C)C[C@@H]3C[C@H]3C2)c1 ZINC000880853901 CG On-Demand Anodyne P2RX7 19 40 CCN(CC)C(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853914 DF On-Demand Anodyne MTNR1A 54 38 CCN(CC)C(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853914 DF On-Demand Anodyne MTNR1B 45 41 CNS(=O)(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853926 ED On-Demand Anodyne BMP1 19 40 CNS(=O)(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853926 ED On-Demand Anodyne NQO2 27 40 CNS(=O)(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853926 ED On-Demand Anodyne CCR3 44 48 CNS(=O)(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880853926 ED On-Demand Anodyne MTNR1A 49 41 C/C=C\CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853932 CE On-Demand Anodyne NQO2 35 43 C/C=C\CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853932 CE On-Demand Anodyne MTNR1A 70 44 C/C=C\CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853932 CE On-Demand Anodyne MTNR1B 62 42 C/C=C\CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853932 CE On-Demand Anodyne MMP3 21 40 C/C=C/CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853933 CE On-Demand Anodyne NQO2 35 43 C/C=C/CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853933 CE On-Demand Anodyne MTNR1A 70 44 C/C=C/CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853933 CE On-Demand Anodyne MTNR1B 62 42 C/C=C/CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853933 CE On-Demand Anodyne MMP3 21 40 C/C=C\CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853934 CE On-Demand Anodyne NQO2 35 43 C/C=C\CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853934 CE On-Demand Anodyne MTNR1A 70 44 C/C=C\CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853934 CE On-Demand Anodyne MTNR1B 62 42 C/C=C\CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880853934 CE On-Demand Anodyne MMP3 21 40 C/C=C/CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853935 CE On-Demand Anodyne NQO2 35 43 C/C=C/CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853935 CE On-Demand Anodyne MTNR1A 70 44 C/C=C/CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853935 CE On-Demand Anodyne MTNR1B 62 42 C/C=C/CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880853935 CE On-Demand Anodyne MMP3 21 40 Cn1c(=O)oc2ccc(CNC(=O)c3ccc(CN4CCOCC4)o3)cc21 ZINC000880853936 FD On-Demand Anodyne DPOL_VZVD 35 46 CNC(=O)N(C)c1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880853984 FH On-Demand Anodyne CA1 26 42 CNC(=O)N(C)c1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880853984 FH On-Demand Anodyne RAF1 22 42 CNC(=O)N(C)c1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880853984 FH On-Demand Anodyne MTNR1A 17 44 CNC(=O)N(C)c1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880853984 FH On-Demand Anodyne MTNR1B 18 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1[C@H](C)O[C@@H](C)[C@H]1C ZINC000880853987 ED On-Demand Anodyne PAPA1_CARPA 34 42 COCC1CC(NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880853993 DG On-Demand Anodyne MTNR1A 45 40 COCC1CC(NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880853993 DG On-Demand Anodyne MTNR1B 39 40 COC(=O)c1cc(NC(=O)N2CCN(C)CC2)cc2ccccc12 ZINC000880854041 EE On-Demand Anodyne HTR1B 19 49 COC(=O)c1cc(NC(=O)N2CCN(C)CC2)cc2ccccc12 ZINC000880854041 EE On-Demand Anodyne PDGFRB 41 38 C/C=C/CNC(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880854130 BF On-Demand Anodyne DPEP1 54 39 C/C=C\CNC(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880854132 BF On-Demand Anodyne DPEP1 54 39 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1c3ccccc3C(=O)N1C)C2 ZINC000880854139 FF On-Demand Anodyne MTNR1A 51 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1c3ccccc3C(=O)N1C)C2 ZINC000880854139 FF On-Demand Anodyne MTNR1B 49 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1c3ccccc3C(=O)N1C)C2 ZINC000880854141 FF On-Demand Anodyne MTNR1A 51 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1c3ccccc3C(=O)N1C)C2 ZINC000880854141 FF On-Demand Anodyne MTNR1B 49 41 O=C(NC[C@@H]1CCN1C1CCCC1)c1cccn2nccc12 ZINC000880854173 CE On-Demand Anodyne JAK3 16 41 O=C(NC[C@@H]1CCN1C1CCCC1)c1cccn2nccc12 ZINC000880854173 CE On-Demand Anodyne TYK2 19 41 O=C(NC[C@H]1CCN1C1CCCC1)c1cccn2nccc12 ZINC000880854174 CE On-Demand Anodyne JAK3 16 41 O=C(NC[C@H]1CCN1C1CCCC1)c1cccn2nccc12 ZINC000880854174 CE On-Demand Anodyne TYK2 19 41 O=C(N[C@@H]1C[C@H]1c1ccsc1)c1cnc(CC2CC2)s1 ZINC000880854177 DG On-Demand Anodyne NPBWR1 40 32 COC[C@@H]1CCCN1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854188 DF On-Demand Anodyne MTNR1A 24 41 COC[C@@H]1CCCN1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854188 DF On-Demand Anodyne MTNR1B 22 41 C#CC1(F)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880854289 CF On-Demand Mild RBP4 31 40 C/C=C\CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854347 CG On-Demand Anodyne INHA 56 39 C/C=C\CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854347 CG On-Demand Anodyne MTNR1A 18 48 C/C=C\CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854347 CG On-Demand Anodyne MTNR1B 27 48 C/C=C\CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854347 CG On-Demand Anodyne ENPP1 55 32 C/C=C/CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854348 CG On-Demand Anodyne INHA 56 39 C/C=C/CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854348 CG On-Demand Anodyne MTNR1A 18 48 C/C=C/CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854348 CG On-Demand Anodyne MTNR1B 27 48 C/C=C/CNC(=O)CCCCc1ccc(OC)c(OC)c1 ZINC000880854348 CG On-Demand Anodyne ENPP1 55 32 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]3C[C@@H]3C2)c(O)n1 ZINC000880854364 FH On-Demand Anodyne KCNA3 46 39 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]3C[C@@H]3C2)c(O)n1 ZINC000880854364 FH On-Demand Anodyne HCN1 71 38 COc1ccccc1-c1ccc(C(=O)NC[C@@]2(C)C[C@@H]3C[C@@H]3C2)c(O)n1 ZINC000880854364 FH On-Demand Anodyne HCN4 49 38 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@@H]3C[C@H]3C2)c(O)n1 ZINC000880854365 FH On-Demand Anodyne KCNA3 46 39 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@@H]3C[C@H]3C2)c(O)n1 ZINC000880854365 FH On-Demand Anodyne HCN1 71 38 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@@H]3C[C@H]3C2)c(O)n1 ZINC000880854365 FH On-Demand Anodyne HCN4 49 38 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@H]3C[C@@H]3C2)c(O)n1 ZINC000880854366 FH On-Demand Anodyne KCNA3 46 39 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@H]3C[C@@H]3C2)c(O)n1 ZINC000880854366 FH On-Demand Anodyne HCN1 71 38 COc1ccccc1-c1ccc(C(=O)NCC2(C)C[C@H]3C[C@@H]3C2)c(O)n1 ZINC000880854366 FH On-Demand Anodyne HCN4 49 38 Cn1ncc(Br)c1CC(=O)NCc1cn(C(F)F)c2ccccc12 ZINC000880854375 GG On-Demand Anodyne P2RX7 15 43 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854376 EG On-Demand Anodyne SLC6A4 19 40 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854376 EG On-Demand Anodyne SLC6A3 34 40 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854377 EG On-Demand Anodyne SLC6A4 19 40 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854377 EG On-Demand Anodyne SLC6A3 34 40 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880854404 DF On-Demand Anodyne NPBWR1 84 31 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880854405 DF On-Demand Anodyne NPBWR1 84 31 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880854406 DF On-Demand Anodyne NPBWR1 84 31 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H]1C[C@H]1c1ccsc1 ZINC000880854407 DF On-Demand Anodyne NPBWR1 84 31 O=C(NC[C@@H]1CCN1C1CCCC1)c1ncccc1-c1ccccn1 ZINC000880854436 EF On-Demand Anodyne HCRTR1 20 44 O=C(NC[C@H]1CCN1C1CCCC1)c1ncccc1-c1ccccn1 ZINC000880854438 EF On-Demand Anodyne HCRTR1 20 44 COCCCNC(=O)Nc1cc(C(=O)OC)c2ccccc2c1 ZINC000880854444 DF On-Demand Anodyne CA1 17 40 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](O)C1)C2 ZINC000880854522 CD On-Demand Anodyne NQO2 32 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](O)C1)C2 ZINC000880854522 CD On-Demand Anodyne MTNR1A 52 46 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](O)C1)C2 ZINC000880854522 CD On-Demand Anodyne MTNR1B 46 41 C/C=C\CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854528 CG On-Demand Anodyne MTNR1A 57 39 C/C=C\CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854528 CG On-Demand Anodyne MTNR1B 51 40 C/C=C/CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854530 CG On-Demand Anodyne MTNR1A 57 39 C/C=C/CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854530 CG On-Demand Anodyne MTNR1B 51 40 CONC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880854610 EE On-Demand Anodyne MTNR1A 21 41 CONC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880854610 EE On-Demand Anodyne MTNR1B 22 41 CONC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880854610 EE On-Demand Anodyne RBP4 26 40 COCC(C)(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854619 DH On-Demand Anodyne MTNR1A 41 38 C/C=C\CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880854676 CG On-Demand Anodyne PDE4D 16 41 C/C=C/CNC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880854677 CG On-Demand Anodyne PDE4D 16 41 O=C(NCC1CC(O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854691 CD On-Demand Anodyne GABRA1 18 51 O=C(NCC1CC(O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854691 CD On-Demand Anodyne MPO 55 35 O=C(NCC1CC(O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854691 CD On-Demand Anodyne GABRA2 16 51 O=C(NC[C@@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854692 CD On-Demand Anodyne GABRA1 18 51 O=C(NC[C@@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854692 CD On-Demand Anodyne MPO 55 35 O=C(NC[C@@H]1C[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880854692 CD On-Demand Anodyne GABRA2 16 51 COC[C@@H]1CCCN1C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854732 DG On-Demand Anodyne CHRNA10 42 40 C#CC[C@H](COC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854776 DF On-Demand Mild MTNR1B 21 40 C#CC[C@@H](COC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880854777 DF On-Demand Mild MTNR1B 21 40 Cc1cc(CNC(=O)[C@H]2CCc3nncn3CC2)c(C)n1-c1ccccc1 ZINC000880854783 FF On-Demand Clean EPHX2 17 41 Cc1cc(CNC(=O)[C@@H]2CCc3nncn3CC2)c(C)n1-c1ccccc1 ZINC000880854784 FF On-Demand Clean EPHX2 17 41 O=C(N[C@@H]1CCO[C@H]1c1ccncc1)c1ccc(CN2CCOCC2)o1 ZINC000880854790 FD On-Demand Anodyne NAMPT 25 40 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880854825 GE On-Demand Anodyne SSTR1 45 33 O=C(NC[C@H]1CCN1C1CCCC1)c1cccc2nsnc12 ZINC000880854862 DE On-Demand Anodyne HCRTR1 29 40 O=C(NC[C@@H]1CCN1C1CCCC1)c1cccc2nsnc12 ZINC000880854863 DE On-Demand Anodyne HCRTR1 29 40 COC(=O)C[C@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854880 DC On-Demand Anodyne NQO2 29 40 COC(=O)C[C@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854880 DC On-Demand Anodyne MTNR1A 43 47 COC(=O)C[C@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854880 DC On-Demand Anodyne MTNR1B 38 47 COC(=O)C[C@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854881 DC On-Demand Anodyne NQO2 29 40 COC(=O)C[C@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854881 DC On-Demand Anodyne MTNR1A 43 47 COC(=O)C[C@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854881 DC On-Demand Anodyne MTNR1B 38 47 COC(=O)C[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854882 DC On-Demand Anodyne NQO2 29 40 COC(=O)C[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854882 DC On-Demand Anodyne MTNR1A 43 47 COC(=O)C[C@@H](O)CNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880854882 DC On-Demand Anodyne MTNR1B 38 47 COC(=O)C[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854883 DC On-Demand Anodyne NQO2 29 40 COC(=O)C[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854883 DC On-Demand Anodyne MTNR1A 43 47 COC(=O)C[C@@H](O)CNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880854883 DC On-Demand Anodyne MTNR1B 38 47 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@@H]2C[C@@H]2C1 ZINC000880854975 CF On-Demand Anodyne HCN1 70 33 C[C@@]1(CNC(=O)c2cccn3nccc23)C[C@@H]2C[C@@H]2C1 ZINC000880854975 CF On-Demand Anodyne HCN4 48 31 Cc1cc(-c2nc(C)c(C(=O)NC[C@@H]3C[C@H](O)C3)s2)ccc1F ZINC000880855065 EG On-Demand Anodyne SCD1 19 41 Cc1cc(-c2nc(C)c(C(=O)NCC3CC(O)C3)s2)ccc1F ZINC000880855066 EG On-Demand Anodyne SCD1 19 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(F)c1O ZINC000880855092 EE On-Demand Anodyne PAPA1_CARPA 40 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(F)c1O ZINC000880855092 EE On-Demand Anodyne FPR1 44 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(F)c1O ZINC000880855093 EE On-Demand Anodyne PAPA1_CARPA 40 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc(F)c1O ZINC000880855093 EE On-Demand Anodyne FPR1 44 38 O=C(NC[C@@H]1CCN1C1CCCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880855102 EF On-Demand Anodyne GABRA1 15 45 O=C(NC[C@H]1CCN1C1CCCC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880855103 EF On-Demand Anodyne GABRA1 15 45 COC(=O)c1cc(NC(=O)N2CCC[C@@H](CO)C2)cc2ccccc12 ZINC000880855115 EF On-Demand Anodyne CCR3 21 44 COC(=O)c1cc(NC(=O)N2CCC[C@H](CO)C2)cc2ccccc12 ZINC000880855116 EF On-Demand Anodyne CCR3 21 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855202 GD On-Demand Anodyne PGC 51 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855202 GD On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855202 GD On-Demand Anodyne REN 42 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855202 GD On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855203 GD On-Demand Anodyne PGC 51 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855203 GD On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855203 GD On-Demand Anodyne REN 42 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1c2ccccc2C(=O)N1C ZINC000880855203 GD On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855204 GD On-Demand Anodyne PGC 51 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855204 GD On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855204 GD On-Demand Anodyne REN 42 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855204 GD On-Demand Anodyne FPR1 45 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855222 GD On-Demand Anodyne PGC 51 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855222 GD On-Demand Anodyne PAPA1_CARPA 42 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855222 GD On-Demand Anodyne REN 42 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1c2ccccc2C(=O)N1C ZINC000880855222 GD On-Demand Anodyne FPR1 45 36 COC(=O)c1cc(NC(=O)NCCCN2CCCC2=O)cc2ccccc12 ZINC000880855228 FF On-Demand Anodyne TYRO3 20 42 COC(=O)[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)Oc1ccccc1 ZINC000880855231 GG On-Demand Anodyne MTNR1A 46 44 COC(=O)[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)Oc1ccccc1 ZINC000880855231 GG On-Demand Anodyne MTNR1B 42 44 Cn1c(=O)oc2ccc(CNC(=O)C[C@@H]3CCNC3=O)cc21 ZINC000880855232 DC On-Demand Anodyne NOS2 44 31 Cn1c(=O)oc2ccc(CNC(=O)C[C@H]3CCNC3=O)cc21 ZINC000880855233 DC On-Demand Anodyne NOS2 44 31 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)C(=O)N1CCCC1 ZINC000880855255 GD On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)C(=O)N1CCCC1 ZINC000880855256 GD On-Demand Anodyne PAPA1_CARPA 37 45 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880855265 IH On-Demand Anodyne MPL 49 38 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880855265 IH On-Demand Anodyne ROCK1 21 40 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880855265 IH On-Demand Anodyne ROCK2 22 40 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880855265 IH On-Demand Anodyne HDAC1 23 41 CC(C)(C)OC(=O)NCc1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880855265 IH On-Demand Anodyne HDAC2 19 41 C/C=C\CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880855289 CE On-Demand Anodyne KCNQ2 41 37 C/C=C/CNC(=O)Cc1ccccc1N1CCCC1=O ZINC000880855290 CE On-Demand Anodyne KCNQ2 41 37 C#CC[C@@H](CCOC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855306 DG On-Demand Mild MTNR1B 17 40 C#CC[C@H](CCOC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855307 DG On-Demand Mild MTNR1B 17 40 CCn1ncc(CNC(=O)Nc2cc(OC)ccc2C2CC2)n1 ZINC000880855308 DF On-Demand Anodyne ROCK2 35 42 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NC[C@@H]1C[C@H](O)C1 ZINC000880855331 FH On-Demand Anodyne PPARD 25 42 Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1C(=O)NCC1CC(O)C1 ZINC000880855332 FH On-Demand Anodyne PPARD 25 42 CCC(CC)C(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880855351 FH On-Demand Anodyne MTNR1A 25 43 CCC(CC)C(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880855351 FH On-Demand Anodyne MTNR1B 28 43 O=C(NC[C@@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880855354 DE On-Demand Anodyne PDE4D 20 48 O=C(NC[C@@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880855354 DE On-Demand Anodyne CACNA1I 68 42 O=C(NCC1CC(O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880855355 DE On-Demand Anodyne PDE4D 20 48 O=C(NCC1CC(O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880855355 DE On-Demand Anodyne CACNA1I 68 42 C/C=C/CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855443 BG On-Demand Anodyne NQO2 20 43 C/C=C/CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855443 BG On-Demand Anodyne MTNR1A 19 45 C/C=C/CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855443 BG On-Demand Anodyne MTNR1B 22 45 C/C=C/CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855444 BG On-Demand Anodyne NQO2 20 43 C/C=C/CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855444 BG On-Demand Anodyne MTNR1A 19 45 C/C=C/CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855444 BG On-Demand Anodyne MTNR1B 22 45 C/C=C\CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855445 BG On-Demand Anodyne NQO2 20 43 C/C=C\CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855445 BG On-Demand Anodyne MTNR1A 19 45 C/C=C\CNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880855445 BG On-Demand Anodyne MTNR1B 22 45 C/C=C\CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855446 BG On-Demand Anodyne NQO2 20 43 C/C=C\CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855446 BG On-Demand Anodyne MTNR1A 19 45 C/C=C\CNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880855446 BG On-Demand Anodyne MTNR1B 22 45 COC[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855456 CF On-Demand Anodyne MTNR1A 41 43 COC[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855456 CF On-Demand Anodyne MTNR1B 36 43 COc1ccc(CN(CCO)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880855476 FH On-Demand Anodyne BMP1 41 37 COc1ccc(CN(CCO)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880855476 FH On-Demand Anodyne ROCK2 28 45 C#Cc1cccc(N(C)C(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880855492 DI On-Demand Mild MTNR1A 19 41 C#Cc1cccc(N(C)C(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880855492 DI On-Demand Mild MTNR1B 21 41 CCNC(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855559 CD On-Demand Anodyne MTNR1A 72 41 CCNC(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855559 CD On-Demand Anodyne MTNR1B 60 45 CCON(C)C(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855567 DE On-Demand Anodyne MTNR1A 42 37 Cn1c(=O)oc2ccc(CNC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)cc21 ZINC000880855708 FE On-Demand Anodyne PLD1 42 33 Cn1c(=O)oc2ccc(CNC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)cc21 ZINC000880855710 FE On-Demand Anodyne PLD1 42 33 CCO[C@@H]1C[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880855758 DG On-Demand Anodyne EPHX2 34 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)C[C@@H]2C[C@@H]2C1 ZINC000880855813 EE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(C)C[C@@H]2C[C@H]2C1 ZINC000880855814 EE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@]1(C)C[C@@H]2C[C@@H]2C1 ZINC000880855815 EE On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(C)C[C@H]2C[C@@H]2C1 ZINC000880855816 EE On-Demand Anodyne PAPA1_CARPA 37 45 NC(=O)c1cc(-c2csc(NC(=O)CCCCCn3c(S)nc4ccccc4c3=O)n2)c[nH]1 ZINC000880855839 JG On-Demand Anodyne HDAC10 15 42 NC(=O)c1cc(-c2csc(NC(=O)CCCCCn3c(S)nc4ccccc4c3=O)n2)c[nH]1 ZINC000880855839 JG On-Demand Anodyne HDAC9 17 49 COC(=O)C[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855840 DD On-Demand Anodyne MTNR1A 36 40 COC(=O)C[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855840 DD On-Demand Anodyne MTNR1B 29 40 COC(=O)C[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855841 DD On-Demand Anodyne MTNR1A 36 40 COC(=O)C[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855841 DD On-Demand Anodyne MTNR1B 29 40 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC[C@@H]3C[C@H](O)C3)ccn2)CC1 ZINC000880855859 GD On-Demand Anodyne CACNA1I 70 43 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NC[C@@H]3C[C@H](O)C3)ccn2)CC1 ZINC000880855859 GD On-Demand Anodyne GPR119 51 45 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NCC3CC(O)C3)ccn2)CC1 ZINC000880855860 GD On-Demand Anodyne CACNA1I 70 43 CC(C)(C)OC(=O)N1CCN(c2cc(C(=O)NCC3CC(O)C3)ccn2)CC1 ZINC000880855860 GD On-Demand Anodyne GPR119 51 45 CN(CCOc1ccccc1C(=O)NC[C@@H]1C[C@H](O)C1)C(=O)OC(C)(C)C ZINC000880855872 GE On-Demand Anodyne HCN1 52 31 CN(CCOc1ccccc1C(=O)NC[C@@H]1C[C@H](O)C1)C(=O)OC(C)(C)C ZINC000880855872 GE On-Demand Anodyne HCN4 40 31 CN(CCOc1ccccc1C(=O)NCC1CC(O)C1)C(=O)OC(C)(C)C ZINC000880855873 GE On-Demand Anodyne HCN1 52 31 CN(CCOc1ccccc1C(=O)NCC1CC(O)C1)C(=O)OC(C)(C)C ZINC000880855873 GE On-Demand Anodyne HCN4 40 31 Cc1cnc(Cl)c(C(=O)NC[C@@H]2C[C@H](O)C2)c1 ZINC000880855874 CD On-Demand Anodyne CACNA1I 49 37 Cc1cnc(Cl)c(C(=O)NCC2CC(O)C2)c1 ZINC000880855875 CD On-Demand Anodyne CACNA1I 49 37 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne CELA1 19 41 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne GRIN2B 21 43 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne PREP 28 43 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne LGMN 52 38 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne SLC12A5 45 35 O=C(NCC1CC(O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855889 FD On-Demand Anodyne Q9NAW4_PLAFA 43 51 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne CELA1 19 41 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne GRIN2B 21 43 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne PREP 28 43 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne LGMN 52 38 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne SLC12A5 45 35 O=C(NC[C@@H]1C[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880855890 FD On-Demand Anodyne Q9NAW4_PLAFA 43 51 O=C(CC[C@@H]1CCc2ccccc21)NC[C@@H]1C[C@H](O)C1 ZINC000880855902 CE On-Demand Anodyne MTNR1A 23 46 O=C(CC[C@@H]1CCc2ccccc21)NC[C@@H]1C[C@H](O)C1 ZINC000880855902 CE On-Demand Anodyne MTNR1B 26 46 O=C(CC[C@@H]1CCc2ccccc21)NCC1CC(O)C1 ZINC000880855903 CE On-Demand Anodyne MTNR1A 23 46 O=C(CC[C@@H]1CCc2ccccc21)NCC1CC(O)C1 ZINC000880855903 CE On-Demand Anodyne MTNR1B 26 46 O=C(CC[C@H]1CCc2ccccc21)NCC1CC(O)C1 ZINC000880855904 CE On-Demand Anodyne MTNR1A 23 46 O=C(CC[C@H]1CCc2ccccc21)NCC1CC(O)C1 ZINC000880855904 CE On-Demand Anodyne MTNR1B 26 46 O=C(CC[C@H]1CCc2ccccc21)NC[C@@H]1C[C@H](O)C1 ZINC000880855905 CE On-Demand Anodyne MTNR1A 23 46 O=C(CC[C@H]1CCc2ccccc21)NC[C@@H]1C[C@H](O)C1 ZINC000880855905 CE On-Demand Anodyne MTNR1B 26 46 O=C(C[C@@H]1CCNC1=O)N[C@H]1CCCc2ccc(Cl)cc21 ZINC000880855930 DE On-Demand Anodyne BDKRB1 44 46 O=C(C[C@H]1CCNC1=O)N[C@H]1CCCc2ccc(Cl)cc21 ZINC000880855931 DE On-Demand Anodyne BDKRB1 44 46 COC(=O)N(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855933 DE On-Demand Anodyne MTNR1A 53 40 CC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)C(=O)OC ZINC000880855936 DF On-Demand Anodyne MTNR1A 47 40 CC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)C(=O)OC ZINC000880855936 DF On-Demand Anodyne MTNR1B 39 40 CCSC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880855937 DH On-Demand Anodyne MTNR1A 49 35 CCSC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880855937 DH On-Demand Anodyne MTNR1B 43 38 COC(=O)Cc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855950 FH On-Demand Anodyne MTNR1A 68 40 COC(=O)Cc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855950 FH On-Demand Anodyne MTNR1B 56 38 C=CCOCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855955 CF On-Demand Mild MTNR1A 47 37 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@@H]1C ZINC000880855984 EG On-Demand Anodyne RBP4 25 40 C#CC[C@H](CO)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855997 CE On-Demand Mild MTNR1B 23 41 C#CC[C@@H](CO)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880855998 CE On-Demand Mild MTNR1B 23 41 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)C1CC1 ZINC000880856006 CH On-Demand Anodyne MTNR1A 43 37 NC(=O)c1cc(-c2csc(NC(=O)c3ccc4c(c3)-c3ccccc3C4)n2)c[nH]1 ZINC000880856045 HI On-Demand Anodyne MPL 69 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](O)C1 ZINC000880856056 DC On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(O)C1 ZINC000880856057 DC On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1CC(O)C1 ZINC000880856058 DC On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](O)C1 ZINC000880856059 DC On-Demand Anodyne PAPA1_CARPA 39 48 COc1ccc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880856063 EI On-Demand Anodyne BMP1 40 33 COc1ccc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880856063 EI On-Demand Anodyne ROCK1 15 43 COc1ccc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880856063 EI On-Demand Anodyne MTNR1A 44 39 COc1ccc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880856063 EI On-Demand Anodyne MTNR1B 41 39 COc1ccc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880856063 EI On-Demand Anodyne ROCK2 31 42 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856070 EH On-Demand Anodyne MTNR1A 27 42 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856070 EH On-Demand Anodyne MTNR1B 29 42 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856070 EH On-Demand Anodyne RBP4 33 41 Cc1ncc(CC(=O)NCc2cc(C)n(-c3ccccc3)c2C)o1 ZINC000880856072 DG On-Demand Clean P2RX7 33 41 O=C(NC[C@@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880856087 FF On-Demand Anodyne PDE4D 18 42 O=C(NC[C@@H]1C[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880856087 FF On-Demand Anodyne CACNA1I 56 36 O=C(NCC1CC(O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880856088 FF On-Demand Anodyne PDE4D 18 42 O=C(NCC1CC(O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880856088 FF On-Demand Anodyne CACNA1I 56 36 O=C(NC[C@@H]1C[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880856098 CD On-Demand Anodyne PLD2 40 38 O=C(NCC1CC(O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880856099 CD On-Demand Anodyne PLD2 40 38 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856143 GG On-Demand Anodyne EPHX2 28 41 O=C(COC1CC1)N[C@H]1CCCc2ccc(Cl)cc21 ZINC000880856154 CG On-Demand Anodyne BDKRB1 49 37 O=C(COC1CC1)N[C@H]1CCCc2ccc(Cl)cc21 ZINC000880856154 CG On-Demand Anodyne KCNN3 15 46 C#CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856165 CG On-Demand Mild RBP4 36 43 C=CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856178 DG On-Demand Mild HRH2 22 44 C=CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856178 DG On-Demand Mild CCR3 18 43 C=CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856178 DG On-Demand Mild MTNR1A 49 38 C=CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856179 DI On-Demand Mild MTNR1A 17 40 C=CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856179 DI On-Demand Mild MTNR1B 20 40 C=CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856180 DI On-Demand Mild MTNR1A 17 40 C=CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856180 DI On-Demand Mild MTNR1B 20 40 C#CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856181 DH On-Demand Mild MTNR1A 24 42 C#CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856181 DH On-Demand Mild MTNR1B 24 42 C#CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856181 DH On-Demand Mild RBP4 33 41 C#CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856182 DH On-Demand Mild MTNR1A 24 42 C#CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856182 DH On-Demand Mild MTNR1B 24 42 C#CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856182 DH On-Demand Mild RBP4 33 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)C2 ZINC000880856185 EI On-Demand Anodyne MTNR1A 26 40 COc1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)C2 ZINC000880856185 EI On-Demand Anodyne MTNR1B 30 40 Cc1cc(Br)ccc1[C@@H]1CCCN1C(=O)COC1CC1 ZINC000880856189 EH On-Demand Anodyne CPT1A 90 36 Cc1cc(Br)ccc1[C@H]1CCCN1C(=O)COC1CC1 ZINC000880856190 EH On-Demand Anodyne CPT1A 90 36 COC[C@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1cccc(OC)c1 ZINC000880856289 FI On-Demand Anodyne MTNR1A 40 39 COC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1cccc(OC)c1 ZINC000880856290 FI On-Demand Anodyne MTNR1A 40 39 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@H]1c1ccccc1 ZINC000880856306 GH On-Demand Anodyne SLC6A3 24 42 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@H]1c1ccccc1 ZINC000880856306 GH On-Demand Anodyne RBP4 45 32 O=C(N[C@H]1CCCc2ccc(Cl)cc21)[C@H]1CCc2nncn2CC1 ZINC000880856307 EG On-Demand Anodyne CNR1 49 30 O=C(N[C@H]1CCCc2ccc(Cl)cc21)[C@@H]1CCc2nncn2CC1 ZINC000880856308 EG On-Demand Anodyne CNR1 49 30 C=CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856315 CG On-Demand Mild MTNR1A 65 39 C=CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856315 CG On-Demand Mild MTNR1B 51 37 CCN1CC[C@H](N(CC)C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856347 EH On-Demand Anodyne CCR5 19 46 CCN1CC[C@@H](N(CC)C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856348 EH On-Demand Anodyne CCR5 19 46 C#C[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856351 CG On-Demand Mild MTNR1A 16 43 C#C[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856351 CG On-Demand Mild MTNR1B 18 43 C#C[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856352 CG On-Demand Mild MTNR1A 16 43 C#C[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856352 CG On-Demand Mild MTNR1B 18 43 CCCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856386 CG On-Demand Anodyne MTNR1A 57 40 CCCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856386 CG On-Demand Anodyne MTNR1B 49 37 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@H]1C ZINC000880856387 EF On-Demand Anodyne RBP4 15 40 Cn1nnc(C(=O)N[C@H]2CCCc3ccc(Cl)cc32)n1 ZINC000880856398 CD On-Demand Anodyne KCNN3 15 44 CCn1c(O)nnc1C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856579 GG On-Demand Anodyne RBP4 27 41 COc1cccc([C@H](CO)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880856618 FG On-Demand Anodyne MTNR1A 42 40 COc1cccc([C@H](CO)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880856618 FG On-Demand Anodyne MTNR1B 39 40 CC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856656 CE On-Demand Anodyne MTNR1A 59 41 CC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856656 CE On-Demand Anodyne MTNR1B 49 41 C=C(C)CONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856675 CG On-Demand Mild MTNR1A 45 38 C=C(C)CONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856675 CG On-Demand Mild MTNR1B 40 36 O=C1CC[C@H](c2ccc(C(=O)N[C@H]3CCCc4ccc(Cl)cc43)cc2)N1 ZINC000880856690 FI On-Demand Anodyne BDKRB1 20 41 O=C1CC[C@@H](c2ccc(C(=O)N[C@H]3CCCc4ccc(Cl)cc43)cc2)N1 ZINC000880856691 FI On-Demand Anodyne BDKRB1 20 41 C=C(CC)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856794 CH On-Demand Mild MTNR1A 63 39 C=C(CC)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856794 CH On-Demand Mild MTNR1B 53 40 COCC(C)(C)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856803 FG On-Demand Anodyne MTNR1A 19 40 COCC(C)(C)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880856803 FG On-Demand Anodyne MTNR1B 19 40 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@@H](CC)O1 ZINC000880856828 EH On-Demand Anodyne MTNR1A 42 37 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@@H](CC)O1 ZINC000880856828 EH On-Demand Anodyne RBP4 15 40 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@H](CC)O1 ZINC000880856829 EH On-Demand Anodyne MTNR1A 42 37 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@H](CC)O1 ZINC000880856829 EH On-Demand Anodyne RBP4 15 40 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)C(=O)NC ZINC000880856842 DE On-Demand Anodyne MTNR1A 47 39 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)C(=O)NC ZINC000880856842 DE On-Demand Anodyne MTNR1B 42 39 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)C(OC)OC ZINC000880856875 DG On-Demand Anodyne MTNR1A 45 38 CCC(C)(C)OCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880856878 DH On-Demand Anodyne MTNR1A 43 38 CCO[C@H]1C[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856883 DG On-Demand Anodyne EPHX2 34 40 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856885 FE On-Demand Anodyne RBP4 22 40 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880856886 FE On-Demand Anodyne RBP4 22 40 O=C(c1cc(C(F)(F)F)ccn1)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880856976 EH On-Demand Anodyne RBP4 49 31 Cn1nnc(C(=O)N2C[C@H](C(C)(C)C)Cc3ccccc32)n1 ZINC000880857002 CE On-Demand Anodyne TPP2 42 30 Cn1nnc(C(=O)N2C[C@@H](C(C)(C)C)Cc3ccccc32)n1 ZINC000880857003 CE On-Demand Anodyne TPP2 42 30 COCC(COC)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880857077 GE On-Demand Anodyne MTNR1A 22 40 COCC(COC)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880857077 GE On-Demand Anodyne MTNR1B 23 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne CA2 19 47 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne LPL 49 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne CA1 52 47 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne KCNA5 16 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne CCR3 41 45 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne RAF1 15 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne MTNR1A 37 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne MTNR1B 33 42 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne EPHX2 17 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne CA12 31 47 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne CA9 32 47 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne LIPG 17 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne MTCA1 15 45 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857111 GI On-Demand Anodyne P96878_MYCTU 21 45 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@@H]1c1ccccc1 ZINC000880857116 GH On-Demand Anodyne SLC6A3 24 42 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C[C@@H]1c1ccccc1 ZINC000880857116 GH On-Demand Anodyne RBP4 45 32 CCNC(=O)C(C)(C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857207 DF On-Demand Anodyne NQO2 31 42 CCNC(=O)C(C)(C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857207 DF On-Demand Anodyne MTNR1A 53 40 CCNC(=O)C(C)(C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857207 DF On-Demand Anodyne MTNR1B 43 41 CCC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857260 DF On-Demand Anodyne MTNR1A 38 42 CCC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857260 DF On-Demand Anodyne MTNR1B 39 48 Cc1nn(CC(=O)N2C[C@@H](C(C)(C)C)Cc3ccccc32)c(=O)o1 ZINC000880857285 EE On-Demand Anodyne TPP2 44 32 Cc1nn(CC(=O)N2C[C@H](C(C)(C)C)Cc3ccccc32)c(=O)o1 ZINC000880857286 EE On-Demand Anodyne TPP2 44 32 O=C(Nc1nc(C2CCOCC2)ns1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880857376 GH On-Demand Anodyne PDE4D 17 47 COc1ccc([C@H](CO)CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857393 FG On-Demand Anodyne MTNR1A 41 44 COc1ccc([C@@H](CO)CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857394 FG On-Demand Anodyne MTNR1A 41 44 COCC[C@@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857497 DG On-Demand Anodyne MTNR1A 35 42 COCC[C@@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857497 DG On-Demand Anodyne MTNR1B 28 42 COCC[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857498 DG On-Demand Anodyne MTNR1A 35 42 COCC[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857498 DG On-Demand Anodyne MTNR1B 28 42 O=C(Nc1nc(C2CCOCC2)ns1)c1ncsc1C1CC1 ZINC000880857500 EG On-Demand Anodyne MAP1 60 38 COCC1(O)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857507 DD On-Demand Anodyne MTNR1A 43 36 COCC1(O)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857507 DD On-Demand Anodyne MTNR1B 43 37 CNC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857508 DE On-Demand Anodyne MMP13 15 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857508 DE On-Demand Anodyne MMP3 17 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857508 DE On-Demand Anodyne MMP1 17 40 COC(=O)[C@H](F)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857524 DE On-Demand Anodyne MTNR1A 43 41 COC(=O)[C@H](F)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857524 DE On-Demand Anodyne MTNR1B 37 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880857583 GG On-Demand Anodyne P2RY12 57 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880857583 GG On-Demand Anodyne FPR1 47 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880857584 GG On-Demand Anodyne P2RY12 57 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880857584 GG On-Demand Anodyne FPR1 47 35 COCCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857599 CE On-Demand Anodyne MTNR1A 50 38 COCCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857599 CE On-Demand Anodyne MTNR1B 42 38 COc1ccccc1-c1ccc(C(=O)N[C@H]2CO[C@H](C3CC3)C2)c(O)n1 ZINC000880857711 FF On-Demand Anodyne HTR3A 17 45 COc1ccccc1-c1ccc(C(=O)N[C@H]2CO[C@@H](C3CC3)C2)c(O)n1 ZINC000880857712 FF On-Demand Anodyne HTR3A 17 45 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CO[C@@H](C3CC3)C2)c(O)n1 ZINC000880857713 FF On-Demand Anodyne HTR3A 17 45 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CO[C@H](C3CC3)C2)c(O)n1 ZINC000880857714 FF On-Demand Anodyne HTR3A 17 45 COCC(COC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857728 DE On-Demand Anodyne MTNR1A 44 38 COCC(COC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857728 DE On-Demand Anodyne MTNR1B 40 38 CCC1(CC)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857737 DI On-Demand Anodyne MTNR1A 50 39 CCC1(CC)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880857737 DI On-Demand Anodyne MTNR1B 48 39 C#Cc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880857743 DH On-Demand Mild CCR3 19 40 C#Cc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880857743 DH On-Demand Mild MTNR1A 40 38 C#Cc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880857743 DH On-Demand Mild ROCK2 38 46 C=CC(C)(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880857763 CH On-Demand Mild MTNR1A 41 36 CC(C)(C(=O)N[C@@H]1CCOC[C@H]1O)c1ccc(C(F)(F)F)cc1 ZINC000880857785 EE On-Demand Anodyne CCR2 22 40 CC(C)(C(=O)N[C@@H]1CCOC[C@@H]1O)c1ccc(C(F)(F)F)cc1 ZINC000880857786 EE On-Demand Anodyne CCR2 22 40 CC(C)(C(=O)N[C@H]1CCOC[C@H]1O)c1ccc(C(F)(F)F)cc1 ZINC000880857787 EE On-Demand Anodyne CCR2 22 40 CC(C)(C(=O)N[C@H]1CCOC[C@@H]1O)c1ccc(C(F)(F)F)cc1 ZINC000880857788 EE On-Demand Anodyne CCR2 22 40 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCCO1 ZINC000880857799 DH On-Demand Anodyne CCR3 15 45 CC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCCO1 ZINC000880857799 DH On-Demand Anodyne RBP4 29 40 C#Cc1ccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880857887 DH On-Demand Mild ROCK2 18 41 CC[C@H]1CCC[C@@]1(C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880857961 CH On-Demand Anodyne SSTR1 51 37 CC[C@@H]1CCC[C@]1(C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880857962 CH On-Demand Anodyne SSTR1 51 37 CC[C@H]1CCC[C@]1(C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880857963 CH On-Demand Anodyne SSTR1 51 37 CC[C@@H]1CCC[C@@]1(C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880857964 CH On-Demand Anodyne SSTR1 51 37 O=C(N[C@@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857988 FD On-Demand Anodyne PREP 25 42 O=C(N[C@@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857988 FD On-Demand Anodyne LGMN 45 37 O=C(N[C@@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857988 FD On-Demand Anodyne KLK5 42 42 O=C(N[C@@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857988 FD On-Demand Anodyne Q9NAW4_PLAFA 40 45 O=C(N[C@@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857989 FD On-Demand Anodyne PREP 25 42 O=C(N[C@@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857989 FD On-Demand Anodyne LGMN 45 37 O=C(N[C@@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857989 FD On-Demand Anodyne KLK5 42 42 O=C(N[C@@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857989 FD On-Demand Anodyne Q9NAW4_PLAFA 40 45 O=C(N[C@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857990 FD On-Demand Anodyne PREP 25 42 O=C(N[C@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857990 FD On-Demand Anodyne LGMN 45 37 O=C(N[C@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857990 FD On-Demand Anodyne KLK5 42 42 O=C(N[C@H]1CCOC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857990 FD On-Demand Anodyne Q9NAW4_PLAFA 40 45 O=C(N[C@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857991 FD On-Demand Anodyne PREP 25 42 O=C(N[C@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857991 FD On-Demand Anodyne LGMN 45 37 O=C(N[C@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857991 FD On-Demand Anodyne KLK5 42 42 O=C(N[C@H]1CCOC[C@@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880857991 FD On-Demand Anodyne Q9NAW4_PLAFA 40 45 COC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858028 EF On-Demand Anodyne MTNR1A 28 40 COC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858028 EF On-Demand Anodyne MTNR1B 27 40 COC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858028 EF On-Demand Anodyne EPHX2 55 52 O=C(N[C@@H]1CCOC[C@H]1O)c1ccc(OC(F)F)c(Br)c1 ZINC000880858034 FD On-Demand Anodyne PDE4D 19 48 O=C(N[C@H]1CCOC[C@@H]1O)c1ccc(OC(F)F)c(Br)c1 ZINC000880858035 FD On-Demand Anodyne PDE4D 19 48 O=C(N[C@H]1CCOC[C@H]1O)c1ccc(OC(F)F)c(Br)c1 ZINC000880858036 FD On-Demand Anodyne PDE4D 19 48 O=C(N[C@@H]1CCOC[C@@H]1O)c1ccc(OC(F)F)c(Br)c1 ZINC000880858037 FD On-Demand Anodyne PDE4D 19 48 C#C[C@@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858081 CG On-Demand Mild MTNR1A 24 40 C#C[C@@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858081 CG On-Demand Mild MTNR1B 25 40 C#C[C@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858082 CG On-Demand Mild MTNR1A 24 40 C#C[C@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858082 CG On-Demand Mild MTNR1B 25 40 C=C(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858136 CH On-Demand Mild NQO2 36 40 C=C(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858136 CH On-Demand Mild CCR3 15 41 C=C(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858136 CH On-Demand Mild MTNR1A 85 41 C=C(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858136 CH On-Demand Mild MTNR1B 75 37 CC[C@@H](C)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858139 DH On-Demand Anodyne MTNR1A 51 44 CC[C@@H](C)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858139 DH On-Demand Anodyne MTNR1B 44 44 CC[C@H](C)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858140 DH On-Demand Anodyne MTNR1A 51 44 CC[C@H](C)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858140 DH On-Demand Anodyne MTNR1B 44 44 C=CC(C)(C)CC(=O)N1Cc2cccc(OC)c2C1 ZINC000880858181 CG On-Demand Mild SSTR1 49 34 CC[C@@H](NC(=O)c1nnn(C)n1)c1cc(C)ccc1C ZINC000880858188 CD On-Demand Anodyne CTSA 60 34 CCC(CC)(CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858215 DH On-Demand Anodyne MTNR1A 62 38 CCC(CC)(CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858215 DH On-Demand Anodyne MTNR1B 52 39 C#CCn1ccc(CN(CC)C(=O)Nc2cc(OC)ccc2C2CC2)n1 ZINC000880858257 FG On-Demand Mild ROCK2 32 43 CCC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)COC1 ZINC000880858346 DG On-Demand Anodyne MTNR1A 63 37 CCC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)COC1 ZINC000880858346 DG On-Demand Anodyne MTNR1B 51 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880858427 FE On-Demand Anodyne P2RY12 45 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880858427 FE On-Demand Anodyne SSTR1 55 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880858429 FE On-Demand Anodyne P2RY12 45 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cccc(OC)c2C1 ZINC000880858429 FE On-Demand Anodyne SSTR1 55 38 CC[C@H](C)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858446 EH On-Demand Anodyne MTNR1A 29 42 CC[C@H](C)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858446 EH On-Demand Anodyne MTNR1B 31 42 O=C(N[C@H]1CCOC[C@@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858571 DC On-Demand Anodyne GABRA1 17 45 O=C(N[C@H]1CCOC[C@@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858571 DC On-Demand Anodyne GABRA2 17 45 O=C(N[C@@H]1CCOC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858572 DC On-Demand Anodyne GABRA1 17 45 O=C(N[C@@H]1CCOC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858572 DC On-Demand Anodyne GABRA2 17 45 O=C(N[C@H]1CCOC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858573 DC On-Demand Anodyne GABRA1 17 45 O=C(N[C@H]1CCOC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858573 DC On-Demand Anodyne GABRA2 17 45 O=C(N[C@@H]1CCOC[C@@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858574 DC On-Demand Anodyne GABRA1 17 45 O=C(N[C@@H]1CCOC[C@@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880858574 DC On-Demand Anodyne GABRA2 17 45 CCN(C)C(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858586 DE On-Demand Anodyne MTNR1A 43 36 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858603 EF On-Demand Anodyne MTNR1A 30 44 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858603 EF On-Demand Anodyne MTNR1B 31 44 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858603 EF On-Demand Anodyne EPHX2 36 48 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858604 EF On-Demand Anodyne MTNR1A 30 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858604 EF On-Demand Anodyne MTNR1B 31 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880858604 EF On-Demand Anodyne EPHX2 36 48 CC[C@@H](C)C(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858625 DF On-Demand Reactive MTNR1A 46 40 CC[C@@H](C)C(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858625 DF On-Demand Reactive MTNR1B 40 40 CCC1(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858740 CH On-Demand Anodyne MTNR1A 46 36 CCC1(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858740 CH On-Demand Anodyne MTNR1B 40 36 NC(=O)c1cc(-c2csc(NC(=O)c3ccc(Cl)c(S(N)(=O)=O)c3)n2)c[nH]1 ZINC000880858753 ID On-Demand Anodyne MPL 44 43 C#CCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858818 CF On-Demand Mild MTNR1A 33 40 C#CCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858818 CF On-Demand Mild MTNR1B 32 44 Cn1ncc(Br)c1CC(=O)N[C@@H]1C[C@H]1c1ccc(F)cc1F ZINC000880858854 FF On-Demand Anodyne PRCP 45 32 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccc(F)cc1F ZINC000880858856 GF On-Demand Anodyne PAPA1_CARPA 34 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@H]1c1ccc(F)cc1F ZINC000880858857 GF On-Demand Anodyne PAPA1_CARPA 34 42 C=C(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858876 CG On-Demand Mild MTNR1A 72 40 C=C(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880858876 CG On-Demand Mild MTNR1B 65 39 COC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858906 DF On-Demand Anodyne MTNR1A 53 39 COC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880858906 DF On-Demand Anodyne MTNR1B 43 37 CC[C@@](C)(CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880858967 DH On-Demand Anodyne MTNR1A 44 38 CCC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CCOCC1 ZINC000880858985 EH On-Demand Anodyne MTNR1A 42 36 CCNC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CCC1 ZINC000880859026 EG On-Demand Anodyne MTNR1A 40 38 CCNC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CCC1 ZINC000880859026 EG On-Demand Anodyne MTNR1B 33 41 O=C(N[C@@H]1CCOC[C@H]1O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880859037 DD On-Demand Anodyne PDE4D 22 48 O=C(N[C@H]1CCOC[C@@H]1O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880859039 DD On-Demand Anodyne PDE4D 22 48 O=C(N[C@H]1CCOC[C@H]1O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880859041 DD On-Demand Anodyne PDE4D 22 48 O=C(N[C@@H]1CCOC[C@@H]1O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880859042 DD On-Demand Anodyne PDE4D 22 48 C#CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859044 CG On-Demand Mild HRH2 18 44 C#CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859044 CG On-Demand Mild CCR3 23 44 C#CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859044 CG On-Demand Mild MTNR1A 61 40 C#CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859044 CG On-Demand Mild MTNR1B 50 40 CCn1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1=O ZINC000880859065 EG On-Demand Anodyne MTNR1A 43 36 CCC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880859085 DH On-Demand Anodyne MTNR1A 46 39 CCC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880859085 DH On-Demand Anodyne MTNR1B 38 40 CCC[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880859087 DH On-Demand Anodyne MTNR1A 46 39 CCC[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880859087 DH On-Demand Anodyne MTNR1B 38 40 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880859115 GH On-Demand Anodyne NPY1R 17 46 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880859115 GH On-Demand Anodyne RBP4 46 35 O=C(N[C@H]1CO[C@H](C2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880859295 DE On-Demand Anodyne GABRA1 16 42 O=C(N[C@H]1CO[C@H](C2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880859295 DE On-Demand Anodyne GABRA2 15 42 O=C(N[C@H]1CO[C@@H](C2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880859297 DE On-Demand Anodyne GABRA1 16 42 O=C(N[C@H]1CO[C@@H](C2CC2)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880859297 DE On-Demand Anodyne GABRA2 15 42 C#C[C@@](C)(CC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859303 CG On-Demand Mild MTNR1B 31 40 C#C[C@](C)(CC)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859305 CG On-Demand Mild MTNR1B 31 40 C#CCC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859344 DE On-Demand Mild MTNR1A 31 40 C#CCC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859344 DE On-Demand Mild MTNR1B 25 40 C#CCC[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859346 DE On-Demand Mild MTNR1A 31 40 C#CCC[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859346 DE On-Demand Mild MTNR1B 25 40 C#CCN(C(=O)Nc1cc(OC)ccc1C1CC1)C1CC1 ZINC000880859391 CG On-Demand Mild MTNR1A 41 41 C#CCN(C(=O)Nc1cc(OC)ccc1C1CC1)C1CC1 ZINC000880859391 CG On-Demand Mild MTNR1B 40 43 C#CCN(C(=O)Nc1cc(OC)ccc1C1CC1)C1CC1 ZINC000880859391 CG On-Demand Mild ROCK2 22 40 CCN1C[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)CC1=O ZINC000880859395 DE On-Demand Anodyne EPHX2 15 40 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)[C@H](C)O ZINC000880859403 CF On-Demand Anodyne MTNR1A 45 38 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)[C@@H](C)O ZINC000880859404 CF On-Demand Anodyne MTNR1A 45 38 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CCCO[C@H]1c1cn[nH]c1)C2 ZINC000880859509 FF On-Demand Anodyne ROCK2 49 39 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859518 DC On-Demand Anodyne DRD4 44 33 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859518 DC On-Demand Anodyne PLD1 93 43 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859518 DC On-Demand Anodyne PLD2 111 43 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859520 DC On-Demand Anodyne DRD4 44 33 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859520 DC On-Demand Anodyne PLD1 93 43 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@@H](O)C3)cc2)N1 ZINC000880859520 DC On-Demand Anodyne PLD2 111 43 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne HTR1A 18 47 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne DRD2 23 40 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne DRD4 44 35 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne SLC6A1 61 36 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne DRD3 40 43 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne CCR3 57 40 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne PLD1 96 42 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne PLD2 117 42 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne MCHR1 26 44 O=C(NCCN1CC[C@@H](O)C1)c1cc2ccccc2cc1F ZINC000880859528 DD On-Demand Anodyne POLR1A 62 42 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1C[C@H]1c1ccc(F)cc1F ZINC000880859537 FG On-Demand Anodyne KCNQ2 35 42 O=C(NCCN1CC[C@@H](O)C1)c1cccn2nccc12 ZINC000880859546 CC On-Demand Anodyne DRD4 43 33 O=C(NCCN1CC[C@@H](O)C1)c1cccn2nccc12 ZINC000880859546 CC On-Demand Anodyne DRD3 16 52 O=C(NCCN1CC[C@@H](O)C1)c1cccn2nccc12 ZINC000880859546 CC On-Demand Anodyne PLD1 67 38 O=C(NCCN1CC[C@@H](O)C1)c1cccn2nccc12 ZINC000880859546 CC On-Demand Anodyne PLD2 77 37 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)C(N)=O ZINC000880859557 CD On-Demand Anodyne MTNR1A 41 36 COc1ccc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)nc1 ZINC000880859561 GG On-Demand Anodyne PDGFRB 57 42 COc1ccc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)nc1 ZINC000880859561 GG On-Demand Anodyne MTNR1A 21 40 COc1ccc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)nc1 ZINC000880859561 GG On-Demand Anodyne MTNR1B 25 42 COc1ccc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)nc1 ZINC000880859561 GG On-Demand Anodyne DGAT1 37 47 COc1ccc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)nc1 ZINC000880859561 GG On-Demand Anodyne NPBWR1 67 40 O=C(NCCN1CC[C@@H](O)C1)c1cccc2nsnc12 ZINC000880859603 CC On-Demand Anodyne PLD2 46 36 Cc1cc(-c2nc(C)c(C(=O)NCCN3CC[C@@H](O)C3)s2)ccc1F ZINC000880859658 FE On-Demand Anodyne PLD1 48 35 Cc1cc(-c2nc(C)c(C(=O)NCCN3CC[C@@H](O)C3)s2)ccc1F ZINC000880859658 FE On-Demand Anodyne PLD2 54 35 Cc1coc(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880859665 BC On-Demand Anodyne DRD4 41 35 Cc1coc(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880859665 BC On-Demand Anodyne PLD1 53 39 Cc1coc(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880859665 BC On-Demand Anodyne PLD2 45 39 O=C(NCCN1CC[C@@H](O)C1)c1csc(-c2ncc[nH]2)n1 ZINC000880859711 DC On-Demand Anodyne PLD1 47 33 O=C(NCCN1CC[C@@H](O)C1)c1csc(-c2ncc[nH]2)n1 ZINC000880859711 DC On-Demand Anodyne PLD2 49 33 O=C(NCCN1CC[C@@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880859719 CC On-Demand Anodyne PLD1 45 35 O=C(NCCN1CC[C@@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880859719 CC On-Demand Anodyne PLD2 50 35 O=C(NCCN1CC[C@@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880859719 CC On-Demand Anodyne SIRT2 40 37 O=C(NCCN1CC[C@@H](O)C1)c1ncccc1-c1ccccn1 ZINC000880859735 DC On-Demand Anodyne PLD1 49 39 O=C(NCCN1CC[C@@H](O)C1)c1ncccc1-c1ccccn1 ZINC000880859735 DC On-Demand Anodyne PLD2 63 39 C=CC(C)(C)CC(=O)N1CCc2c(O)cccc2C1 ZINC000880859754 CF On-Demand Mild AKR1C3 17 41 CNC(=O)COc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880859772 GG On-Demand Anodyne HRH2 24 43 CNC(=O)COc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880859772 GG On-Demand Anodyne ROCK1 37 44 CNC(=O)COc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880859772 GG On-Demand Anodyne MTNR1A 44 37 CNC(=O)COc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880859772 GG On-Demand Anodyne MTNR1B 40 37 CNC(=O)COc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880859772 GG On-Demand Anodyne ROCK2 48 49 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne CELA1 19 41 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne PREP 28 41 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne LGMN 65 39 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne SLC12A5 58 36 O=C(NCCN1CC[C@@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880859774 GC On-Demand Anodyne Q9NAW4_PLAFA 40 46 CC/C=C\CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859822 CH On-Demand Anodyne MTNR1A 56 39 CC/C=C\CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859822 CH On-Demand Anodyne MTNR1B 48 42 CC/C=C/CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859824 CH On-Demand Anodyne MTNR1A 56 39 CC/C=C/CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880859824 CH On-Demand Anodyne MTNR1B 48 42 CCOC(=O)c1csc(CCNC(=O)Nc2cc(OC)ccc2C2CC2)n1 ZINC000880859857 GH On-Demand Anodyne MTNR1A 48 38 O=C(COC1CC1)N1CCc2c(O)cccc2C1 ZINC000880860002 BD On-Demand Anodyne CPT2 27 42 C=CCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860032 CF On-Demand Mild MTNR1A 43 36 CCc1nc(CNC(=O)Nc2cc(OC)ccc2C2CC2)n[nH]1 ZINC000880860035 DF On-Demand Anodyne ROCK2 29 40 COCCCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860036 CF On-Demand Anodyne MTNR1A 42 36 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880860071 GD On-Demand Anodyne DRD4 44 35 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880860071 GD On-Demand Anodyne PLD1 60 40 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880860071 GD On-Demand Anodyne UTS2R 25 41 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880860071 GD On-Demand Anodyne PLD2 80 39 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880860071 GD On-Demand Anodyne CACNA1I 58 34 C#CCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880860076 FF On-Demand Mild MTNR1A 29 42 C#CCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880860076 FF On-Demand Mild MTNR1B 28 42 C#CCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880860076 FF On-Demand Mild RBP4 28 40 CS(=O)(=O)C1CCC(C(=O)N2CCc3c(O)cccc3C2)CC1 ZINC000880860085 ED On-Demand Anodyne AKR1C3 25 42 O=C(N[C@@H]1C[C@H]1c1ccc(F)cc1F)[C@@H]1CCc2nncn2CC1 ZINC000880860122 EE On-Demand Anodyne PRCP 46 32 O=C(N[C@@H]1C[C@H]1c1ccc(F)cc1F)[C@H]1CCc2nncn2CC1 ZINC000880860123 EE On-Demand Anodyne PRCP 46 32 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3C[C@H]3c3ccc(F)cc3F)cc2)N1 ZINC000880860131 FG On-Demand Anodyne SSTR3 26 42 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3C[C@H]3c3ccc(F)cc3F)cc2)N1 ZINC000880860132 FG On-Demand Anodyne SSTR3 26 42 Cn1nnc(C(=O)N[C@@H]2C[C@H]2c2ccc(F)cc2F)n1 ZINC000880860145 CC On-Demand Anodyne PRCP 44 33 CCC1(O)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860224 CF On-Demand Anodyne MTNR1A 44 38 CCC1(O)CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860224 CF On-Demand Anodyne MTNR1B 43 38 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880860254 CC On-Demand Anodyne CACNA1H 20 40 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880860254 CC On-Demand Anodyne DRD4 44 35 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880860254 CC On-Demand Anodyne PLD1 48 38 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880860254 CC On-Demand Anodyne PLD2 55 38 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@@H](O)C2)c1 ZINC000880860254 CC On-Demand Anodyne CACNA1I 56 35 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne DRD2 15 41 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne DRD4 49 38 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne PDE4D 17 41 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne PLD1 67 42 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne UTS2R 26 45 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne PLD2 84 42 O=C(NCCN1CC[C@@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880860263 ED On-Demand Anodyne CACNA1I 68 42 O=C(NCCN1CC[C@@H](O)C1)c1coc(-c2ccccn2)n1 ZINC000880860284 DC On-Demand Anodyne PLD1 45 37 O=C(NCCN1CC[C@@H](O)C1)c1coc(-c2ccccn2)n1 ZINC000880860284 DC On-Demand Anodyne PLD2 56 37 O=C(NCCN1CC[C@@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880860299 DC On-Demand Anodyne CCR3 50 40 O=C(NCCN1CC[C@@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880860299 DC On-Demand Anodyne PYGL 27 40 O=C(NCCN1CC[C@@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880860299 DC On-Demand Anodyne PLD1 113 51 O=C(NCCN1CC[C@@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880860299 DC On-Demand Anodyne PLD2 119 51 O=C(NCCN1CC[C@@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880860299 DC On-Demand Anodyne WNT3A 46 34 C=CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860381 CI On-Demand Mild CCR3 20 43 C=CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860381 CI On-Demand Mild MTNR1A 49 39 C=CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860381 CI On-Demand Mild MTNR1B 40 35 COC[C@@H]1CCCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860450 EH On-Demand Anodyne CCR3 15 46 COC[C@@H]1CCCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860450 EH On-Demand Anodyne RBP4 24 40 C=CCCC[C@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860455 DE On-Demand Mild SLC6A1 49 34 C=CCCC[C@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860455 DE On-Demand Mild OPRK1 22 42 C=CCCC[C@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860455 DE On-Demand Mild CCR5 27 40 C=CCCC[C@@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860456 DE On-Demand Mild SLC6A1 49 34 C=CCCC[C@@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860456 DE On-Demand Mild OPRK1 22 42 C=CCCC[C@@H](C(=O)NCCN1CC[C@@H](O)C1)c1ccccc1 ZINC000880860456 DE On-Demand Mild CCR5 27 40 COCC(C)(C)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860486 EI On-Demand Anodyne NQO2 25 40 COCC(C)(C)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860486 EI On-Demand Anodyne CCR3 17 42 O=C(CC[C@H]1CCc2ccccc21)NCCN1CC[C@@H](O)C1 ZINC000880860487 DD On-Demand Anodyne OPRK1 16 40 O=C(CC[C@H]1CCc2ccccc21)NCCN1CC[C@@H](O)C1 ZINC000880860487 DD On-Demand Anodyne NQO2 17 41 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CC[C@@H](O)C1 ZINC000880860489 DD On-Demand Anodyne OPRK1 16 40 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CC[C@@H](O)C1 ZINC000880860489 DD On-Demand Anodyne NQO2 17 41 Cn1nnc(C(=O)N[C@@H]2CCN(c3ccc(Cl)cc3F)C2)n1 ZINC000880860502 DD On-Demand Anodyne MAPK13 43 32 Cn1nnc(C(=O)N[C@H]2CCN(c3ccc(Cl)cc3F)C2)n1 ZINC000880860503 DD On-Demand Anodyne MAPK13 43 32 CC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880860508 CG On-Demand Anodyne MTNR1A 51 41 CC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880860508 CG On-Demand Anodyne MTNR1B 42 41 O=C1CC[C@@H](c2ccc(C(=O)N3CCc4c(O)cccc4C3)cc2)N1 ZINC000880860510 EF On-Demand Anodyne FABI 43 35 O=C1CC[C@H](c2ccc(C(=O)N3CCc4c(O)cccc4C3)cc2)N1 ZINC000880860511 EF On-Demand Anodyne FABI 43 35 COCC(=O)NC1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860534 ED On-Demand Anodyne MTNR1A 21 40 COCC(=O)NC1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860534 ED On-Demand Anodyne MTNR1B 22 40 O=C(COC1CC1)N[C@@H]1CCN(c2ccc(Cl)cc2F)C1 ZINC000880860542 DE On-Demand Anodyne LIPG 49 36 O=C(COC1CC1)N[C@H]1CCN(c2ccc(Cl)cc2F)C1 ZINC000880860544 DE On-Demand Anodyne LIPG 49 36 CC#CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860651 CF On-Demand Mild MTNR1A 61 39 CC#CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860651 CF On-Demand Mild MTNR1B 51 39 C#C[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860659 CF On-Demand Mild MTNR1A 36 40 C#C[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860659 CF On-Demand Mild MTNR1B 31 40 C#C[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860660 CF On-Demand Mild MTNR1A 36 40 C#C[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860660 CF On-Demand Mild MTNR1B 31 40 Cc1coc(C(=O)N[C@@H]2C[C@H]2c2ccc(F)cc2F)c1 ZINC000880860667 CG On-Demand Anodyne PRCP 40 31 COCCO[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860834 EG On-Demand Anodyne MTNR1A 15 42 COCCO[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860834 EG On-Demand Anodyne MTNR1B 18 42 COCCO[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860835 EG On-Demand Anodyne MTNR1A 15 42 COCCO[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860835 EG On-Demand Anodyne MTNR1B 18 42 C#CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860858 EI On-Demand Mild ROCK1 20 40 C#CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860858 EI On-Demand Mild MTNR1B 27 41 C#CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860858 EI On-Demand Mild ROCK2 33 40 C#CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860858 EI On-Demand Mild PTGES 23 45 O=C(NCCN1CC[C@@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880860885 FD On-Demand Anodyne DRD4 40 31 O=C(NCCN1CC[C@@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880860885 FD On-Demand Anodyne PLD1 53 34 O=C(NCCN1CC[C@@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880860885 FD On-Demand Anodyne PLD2 64 34 O=C(NCCN1CC[C@@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880860899 DC On-Demand Anodyne GABRA1 16 45 O=C(NCCN1CC[C@@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880860899 DC On-Demand Anodyne HTR1D 26 42 O=C(NCCN1CC[C@@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880860899 DC On-Demand Anodyne HTR1B 23 42 O=C(NCCN1CC[C@@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880860899 DC On-Demand Anodyne PLD1 50 40 O=C(NCCN1CC[C@@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880860899 DC On-Demand Anodyne PLD2 58 38 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860923 GH On-Demand Anodyne EPHX2 31 42 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880860923 GH On-Demand Anodyne RBP4 43 39 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860950 GH On-Demand Anodyne CCR3 22 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860950 GH On-Demand Anodyne MTNR1B 15 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860951 GH On-Demand Anodyne CCR3 22 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860951 GH On-Demand Anodyne MTNR1B 15 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860977 GH On-Demand Anodyne CCR3 26 41 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860977 GH On-Demand Anodyne MTNR1B 22 41 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860979 GH On-Demand Anodyne CCR3 26 41 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860979 GH On-Demand Anodyne MTNR1B 22 41 CC#CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860986 CG On-Demand Mild MTNR1A 54 38 CC#CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880860986 CG On-Demand Mild MTNR1B 43 37 CCC1(O)CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880860989 EH On-Demand Anodyne EPHX2 28 42 O=C(NCCN1CC[C@@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880861030 CC On-Demand Anodyne DRD4 44 34 O=C(NCCN1CC[C@@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880861030 CC On-Demand Anodyne PLD1 87 50 O=C(NCCN1CC[C@@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880861030 CC On-Demand Anodyne PLD2 116 50 O=C(NCCN1CC[C@@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880861030 CC On-Demand Anodyne HPGDS 47 35 O=C(C[C@H]1CCNC1=O)N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861034 EF On-Demand Anodyne SIRT1 15 50 O=C(C[C@@H]1CCNC1=O)N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861035 EF On-Demand Anodyne SIRT1 15 50 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861036 EF On-Demand Anodyne SIRT1 15 50 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861037 EF On-Demand Anodyne SIRT1 15 50 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne NQO2 28 42 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne CCR3 40 46 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne ROCK1 22 42 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne MTNR1A 47 37 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne MTNR1B 42 39 COC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880861049 FI On-Demand Anodyne ROCK2 41 48 CCCC[C@@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861052 DJ On-Demand Anodyne MTNR1A 40 39 CCCC[C@@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861052 DJ On-Demand Anodyne MTNR1B 40 39 CCCC[C@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861053 DJ On-Demand Anodyne MTNR1A 40 39 CCCC[C@H](C)N(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861053 DJ On-Demand Anodyne MTNR1B 40 39 COC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861092 CD On-Demand Anodyne ADRB1 27 44 COC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861092 CD On-Demand Anodyne MTNR1A 43 41 COC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861092 CD On-Demand Anodyne MTNR1B 36 41 O=C(N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21)[C@@H]1CCc2nncn2CC1 ZINC000880861094 GH On-Demand Anodyne SIRT1 15 48 O=C(N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21)[C@H]1CCc2nncn2CC1 ZINC000880861095 GH On-Demand Anodyne SIRT1 15 48 O=C(N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21)[C@@H]1CCc2nncn2CC1 ZINC000880861096 GH On-Demand Anodyne SIRT1 15 48 O=C(N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21)[C@H]1CCc2nncn2CC1 ZINC000880861097 GH On-Demand Anodyne SIRT1 15 48 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne HTR1A 48 43 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne DRD2 52 47 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne DRD4 44 47 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne ADRA1D 25 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne ADRA1A 24 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne ADRA1B 15 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne DRD3 69 44 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne OPRK1 20 49 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne HTR4 40 37 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne HCN1 51 33 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@@H](O)C2)c(O)n1 ZINC000880861104 FD On-Demand Anodyne HCN4 47 32 O=C(c1ccc(CN2CCOCC2)o1)N1CCc2c(O)cccc2C1 ZINC000880861110 EE On-Demand Anodyne FABI 49 34 Cc1cnc(Cl)c(C(=O)N2CCc3c(O)cccc3C2)c1 ZINC000880861119 DF On-Demand Anodyne FABI 49 39 Cc1cnc(Cl)c(C(=O)N2CCc3c(O)cccc3C2)c1 ZINC000880861119 DF On-Demand Anodyne P2RX7 41 39 O=C(NCCN1CC[C@@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880861226 FE On-Demand Anodyne DRD4 42 33 O=C(NCCN1CC[C@@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880861226 FE On-Demand Anodyne DRD3 16 44 O=C(NCCN1CC[C@@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880861226 FE On-Demand Anodyne PLD1 56 41 O=C(NCCN1CC[C@@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880861226 FE On-Demand Anodyne PLD2 63 41 O=C(COC1CC1)N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861249 DG On-Demand Anodyne PYGL 52 40 O=C(COC1CC1)N[C@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861249 DG On-Demand Anodyne SIRT1 17 55 O=C(COC1CC1)N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861250 DG On-Demand Anodyne PYGL 52 40 O=C(COC1CC1)N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21 ZINC000880861250 DG On-Demand Anodyne SIRT1 17 55 CC(C)(C(=O)NCCN1CC[C@@H](O)C1)c1ccc(F)cc1F ZINC000880861256 DD On-Demand Anodyne CCR3 40 36 CCSCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861266 DH On-Demand Anodyne HRH2 15 41 CCSCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861266 DH On-Demand Anodyne CCR3 32 46 CCSCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861266 DH On-Demand Anodyne MTNR1A 52 41 CCSCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861266 DH On-Demand Anodyne MTNR1B 44 40 O=C(NCCN1CC[C@@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880861274 EE On-Demand Anodyne DRD4 44 36 O=C(NCCN1CC[C@@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880861274 EE On-Demand Anodyne PLD1 54 35 O=C(NCCN1CC[C@@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880861274 EE On-Demand Anodyne PLD2 67 35 O=C(Cc1ccccc1N1CCCC1=O)NCCN1CC[C@@H](O)C1 ZINC000880861278 EC On-Demand Anodyne PLD1 66 36 O=C(Cc1ccccc1N1CCCC1=O)NCCN1CC[C@@H](O)C1 ZINC000880861278 EC On-Demand Anodyne PLD2 54 35 O=C(NCCN1CC[C@@H](O)C1)c1cncc2[nH]ccc12 ZINC000880861283 CC On-Demand Anodyne PLD1 57 37 O=C(NCCN1CC[C@@H](O)C1)c1cncc2[nH]ccc12 ZINC000880861283 CC On-Demand Anodyne PLD2 66 37 O=C(NCCN1CC[C@@H](O)C1)c1cncc2[nH]ccc12 ZINC000880861283 CC On-Demand Anodyne PRKCQ 18 42 COC[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861285 CF On-Demand Anodyne MTNR1A 41 43 COC[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861285 CF On-Demand Anodyne MTNR1B 36 43 O=C(NCCN1CC[C@@H](O)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880861310 DD On-Demand Anodyne SIGMAR1 15 40 O=C(NCCN1CC[C@@H](O)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880861310 DD On-Demand Anodyne PLD2 41 32 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CC[C@@H](O)C2)N1Cc1ccccc1 ZINC000880861339 FB On-Demand Anodyne SIGMAR1 29 44 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCc3c(O)cccc3C2)N1Cc1ccccc1 ZINC000880861345 GD On-Demand Anodyne FABI 40 33 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCc3c(O)cccc3C2)N1Cc1ccccc1 ZINC000880861345 GD On-Demand Anodyne CPT2 21 45 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCc3c(O)cccc3C2)N1Cc1ccccc1 ZINC000880861345 GD On-Demand Anodyne PREP 47 36 Cn1nnc(C(=O)N[C@@H]2CCCc3c2[nH]c2ccc(Cl)cc32)n1 ZINC000880861346 EE On-Demand Anodyne SIRT1 17 53 Cn1nnc(C(=O)N[C@H]2CCCc3c2[nH]c2ccc(Cl)cc32)n1 ZINC000880861347 EE On-Demand Anodyne SIRT1 17 53 CC(C)(C(=O)NCCN1CC[C@@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880861363 EE On-Demand Anodyne OPRK1 15 46 CC(C)(C(=O)NCCN1CC[C@@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880861363 EE On-Demand Anodyne EPHX2 15 42 CC(C)(C(=O)NCCN1CC[C@@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880861363 EE On-Demand Anodyne MCHR1 36 42 CC(C)(C(=O)NCCN1CC[C@@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880861363 EE On-Demand Anodyne CACNA1I 43 38 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne DRD4 44 34 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne HTR4 16 42 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne CASR 43 44 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne HRH3 21 40 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne SIGMAR1 18 41 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne ROCK2 24 41 CCCN(CCN1CCCC1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861364 EH On-Demand Anodyne EBP 42 41 COc1cccc(C2=CCN(C(=O)Nc3cc(OC)ccc3C3CC3)C2)c1 ZINC000880861419 FJ On-Demand Anodyne ADAM10 16 42 CNC(=O)CCCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861420 DF On-Demand Anodyne MTNR1A 28 40 CNC(=O)CCCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861420 DF On-Demand Anodyne MTNR1B 28 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861428 FG On-Demand Anodyne CCR3 34 43 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861428 FG On-Demand Anodyne MTNR1A 22 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861428 FG On-Demand Anodyne MTNR1B 21 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861428 FG On-Demand Anodyne EPHX2 18 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861429 FG On-Demand Anodyne CCR3 34 43 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861429 FG On-Demand Anodyne MTNR1A 22 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861429 FG On-Demand Anodyne MTNR1B 21 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861429 FG On-Demand Anodyne EPHX2 18 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861430 FG On-Demand Anodyne CCR3 34 43 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861430 FG On-Demand Anodyne MTNR1A 22 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861430 FG On-Demand Anodyne MTNR1B 21 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861430 FG On-Demand Anodyne EPHX2 18 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861431 FG On-Demand Anodyne CCR3 34 43 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861431 FG On-Demand Anodyne MTNR1A 22 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861431 FG On-Demand Anodyne MTNR1B 21 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861431 FG On-Demand Anodyne EPHX2 18 42 CCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861436 CF On-Demand Anodyne MTNR1A 61 39 CCONC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861436 CF On-Demand Anodyne MTNR1B 53 38 CCC1(CO)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880861480 EH On-Demand Anodyne MTNR1A 24 40 CCC1(CO)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880861480 EH On-Demand Anodyne MTNR1B 28 40 CCC(CC)(CNC(=O)Nc1cc(OC)ccc1C1CC1)C(=O)OC ZINC000880861495 EH On-Demand Anodyne MTNR1A 41 35 C#CCOCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861504 CE On-Demand Mild MTNR1A 46 38 C=CCCOCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861515 DG On-Demand Mild MTNR1A 51 37 CCOC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861674 CE On-Demand Reactive MTNR1A 41 41 CCOC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861674 CE On-Demand Reactive MTNR1B 34 43 CNC(C)(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861679 CF On-Demand Anodyne MTNR1A 51 37 CNC(C)(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861679 CF On-Demand Anodyne MTNR1B 43 38 CCC(CC)(CO)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861807 DG On-Demand Anodyne MTNR1A 40 35 COC(=O)c1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)CC2 ZINC000880861863 GH On-Demand Anodyne HDAC6 35 42 CCC[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCO1 ZINC000880861899 DH On-Demand Anodyne RBP4 22 41 CCC[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCO1 ZINC000880861900 DH On-Demand Anodyne RBP4 22 41 COC[C@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861910 EI On-Demand Anodyne MTNR1B 39 41 COC[C@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861910 EI On-Demand Anodyne SOAT1 29 40 COC[C@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861910 EI On-Demand Anodyne PSMB8 44 32 COC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861911 EI On-Demand Anodyne MTNR1B 39 41 COC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861911 EI On-Demand Anodyne SOAT1 29 40 COC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880861911 EI On-Demand Anodyne PSMB8 44 32 COC(=O)c1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1C ZINC000880861928 EG On-Demand Anodyne CCR3 15 41 C=CCS(=O)(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861937 EE On-Demand Mild MTNR1A 55 40 C=CCS(=O)(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861937 EE On-Demand Mild MTNR1B 42 37 C=CCNC(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880861960 DD On-Demand Mild MTNR1A 44 35 COC[C@@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862115 DE On-Demand Anodyne ADRB1 16 43 COC[C@@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862115 DE On-Demand Anodyne MTNR1A 45 37 CCC(CO)(CO)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862141 DD On-Demand Anodyne MTNR1A 42 37 COCC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862180 CD On-Demand Reactive MTNR1A 48 45 COCC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862180 CD On-Demand Reactive MTNR1B 40 45 COC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CCOCC1 ZINC000880862189 FF On-Demand Anodyne MTNR1A 40 36 COC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880862199 DE On-Demand Anodyne MTNR1A 36 40 COC[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)OC ZINC000880862199 DE On-Demand Anodyne MTNR1B 30 40 CCC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862230 CE On-Demand Reactive NQO2 31 43 CCC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862230 CE On-Demand Reactive MTNR1A 74 43 CCC(=O)NNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862230 CE On-Demand Reactive MTNR1B 62 43 C=CCSCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862264 DH On-Demand Mild MTNR1A 40 36 COCCOC1CN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862269 DE On-Demand Anodyne RBP4 15 40 C#CC[C@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880862286 EI On-Demand Mild MTNR1B 29 40 C#CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccccc1 ZINC000880862287 EI On-Demand Mild MTNR1B 29 40 CCc1nc([C@H]2CCCN2C(=O)Nc2cc(OC)ccc2C2CC2)no1 ZINC000880862352 FH On-Demand Anodyne CPT1A 49 41 COCC1(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862367 CF On-Demand Anodyne EPHX2 17 41 CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862405 DI On-Demand Anodyne CCR3 15 49 CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862405 DI On-Demand Anodyne MTNR1A 37 42 CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862405 DI On-Demand Anodyne MTNR1B 38 42 CC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862405 DI On-Demand Anodyne RBP4 25 40 CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862406 DI On-Demand Anodyne CCR3 15 49 CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862406 DI On-Demand Anodyne MTNR1A 37 42 CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862406 DI On-Demand Anodyne MTNR1B 38 42 CC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862406 DI On-Demand Anodyne RBP4 25 40 CCC1(NC(=O)Nc2cc(OC)ccc2C2CC2)CCC1 ZINC000880862420 CI On-Demand Anodyne MTNR1A 41 35 C#CCN(CC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862438 CG On-Demand Mild MTNR1B 29 42 CCOC[C@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862539 DG On-Demand Anodyne RBP4 22 40 CC[C@H](CCO)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862544 DG On-Demand Anodyne MTNR1A 41 39 CC[C@@H](CCO)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862545 DG On-Demand Anodyne MTNR1A 41 39 CCC(CC)(CO)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862550 DG On-Demand Anodyne MTNR1A 42 37 CCC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862610 CH On-Demand Anodyne MTNR1A 58 37 CCC1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862610 CH On-Demand Anodyne MTNR1B 49 40 COC(=O)C[C@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCO1 ZINC000880862612 EE On-Demand Anodyne RBP4 24 40 COC(=O)C[C@@H]1CN(C(=O)Nc2cc(OC)ccc2C2CC2)CCO1 ZINC000880862613 EE On-Demand Anodyne RBP4 24 40 CCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862666 BG On-Demand Anodyne MTNR1A 56 40 CCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862666 BG On-Demand Anodyne MTNR1B 49 40 CC[C@@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862709 CF On-Demand Anodyne CCR3 18 41 CC[C@@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862709 CF On-Demand Anodyne MTNR1A 63 39 CC[C@@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862709 CF On-Demand Anodyne MTNR1B 51 38 CC[C@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862710 CF On-Demand Anodyne CCR3 18 41 CC[C@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862710 CF On-Demand Anodyne MTNR1A 63 39 CC[C@H](O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862710 CF On-Demand Anodyne MTNR1B 51 38 COC(=O)C1(CNC(=O)Nc2cc(OC)ccc2C2CC2)CCCC1 ZINC000880862783 EG On-Demand Anodyne MTNR1A 47 38 CC[C@]1(C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862801 DI On-Demand Anodyne MTNR1A 27 40 CC[C@]1(C)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862801 DI On-Demand Anodyne MTNR1B 29 40 CCc1cnc(CN(C)C(=O)Nc2cc(OC)ccc2C2CC2)s1 ZINC000880862823 EI On-Demand Anodyne ROCK2 26 40 COCCC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862826 GF On-Demand Anodyne C3AR1 35 40 COCCC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862826 GF On-Demand Anodyne EPHX2 46 53 COCCC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862826 GF On-Demand Anodyne PDK1 44 31 COCCC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862826 GF On-Demand Anodyne CCR8 45 34 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne DRD2 19 44 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne CCR3 40 43 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne MTNR1A 26 40 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne MTNR1B 26 40 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne EPHX2 27 42 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne MCHR1 19 45 CCN1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862853 DG On-Demand Anodyne BIRC2 30 43 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne DRD2 19 44 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne CCR3 40 43 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne MTNR1A 26 40 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne MTNR1B 26 40 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne EPHX2 27 42 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne MCHR1 19 45 CCN1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880862854 DG On-Demand Anodyne BIRC2 30 43 CCN(Cc1ccccn1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862888 EI On-Demand Anodyne ROCK2 30 42 CC[C@@H](CN1CCCC1)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862927 EH On-Demand Anodyne KCNQ2 22 40 CC[C@@H](CN1CCCC1)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862927 EH On-Demand Anodyne CCR3 19 41 CC[C@H](CN1CCCC1)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862928 EH On-Demand Anodyne KCNQ2 22 40 CC[C@H](CN1CCCC1)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862928 EH On-Demand Anodyne CCR3 19 41 CNc1nc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cs1 ZINC000880862935 EG On-Demand Anodyne AVPR1B 17 43 CNc1nc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cs1 ZINC000880862935 EG On-Demand Anodyne ROCK2 16 43 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862963 DE On-Demand Anodyne LGMN 65 39 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880862963 DE On-Demand Anodyne MMP1 15 43 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862973 ED On-Demand Anodyne DRD4 41 32 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862973 ED On-Demand Anodyne MTNR1A 24 43 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880862973 ED On-Demand Anodyne MTNR1B 27 43 C=C(C)COCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863036 DG On-Demand Mild MTNR1A 64 39 C=C(C)COCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863036 DG On-Demand Mild MTNR1B 53 39 COc1cccc([C@H]2CN(C(=O)Nc3cc(OC)ccc3C3CC3)CCO2)c1 ZINC000880863044 GI On-Demand Anodyne RBP4 43 39 COCCNc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863086 FH On-Demand Anodyne MTNR1A 58 39 COCCNc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863086 FH On-Demand Anodyne MTNR1B 47 36 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863091 EE On-Demand Anodyne ACOX1 44 32 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863091 EE On-Demand Anodyne CCR3 20 40 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863091 EE On-Demand Anodyne MTNR1A 23 41 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863091 EE On-Demand Anodyne MTNR1B 25 42 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863092 EE On-Demand Anodyne ACOX1 44 32 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863092 EE On-Demand Anodyne CCR3 20 40 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863092 EE On-Demand Anodyne MTNR1A 23 41 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863092 EE On-Demand Anodyne MTNR1B 25 42 CCNC(=O)C(C)(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863105 EF On-Demand Anodyne MTNR1A 45 39 CCNC(=O)C(C)(C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863105 EF On-Demand Anodyne MTNR1B 38 42 C#CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863127 CG On-Demand Mild HRH2 17 43 C#CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863127 CG On-Demand Mild CCR3 22 43 C#CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863127 CG On-Demand Mild MTNR1A 55 39 C#CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863127 CG On-Demand Mild MTNR1B 46 39 CCOC(=O)[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863133 DF On-Demand Anodyne MTNR1A 49 42 CCOC(=O)[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863133 DF On-Demand Anodyne MTNR1B 41 42 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863160 GF On-Demand Anodyne CCR3 22 42 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863161 GF On-Demand Anodyne CCR3 22 42 COC(=O)CCC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863178 FH On-Demand Anodyne RBP4 37 42 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863216 EF On-Demand Anodyne MTNR1A 30 42 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863216 EF On-Demand Anodyne MTNR1B 29 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863216 EF On-Demand Anodyne EPHX2 41 60 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863217 EF On-Demand Anodyne MTNR1A 30 42 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863217 EF On-Demand Anodyne MTNR1B 29 43 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863217 EF On-Demand Anodyne EPHX2 41 60 CNC(=O)[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863229 CD On-Demand Anodyne MTNR1B 31 40 COC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863232 EF On-Demand Anodyne RBP4 33 42 CC[C@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863240 CH On-Demand Anodyne CCR3 16 47 CC[C@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863240 CH On-Demand Anodyne MTNR1A 38 41 CC[C@H]1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863240 CH On-Demand Anodyne MTNR1B 37 41 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863342 GI On-Demand Anodyne EPHX2 48 51 CNC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863350 CD On-Demand Anodyne NQO2 39 40 CNC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863350 CD On-Demand Anodyne CCR3 15 42 CNC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863350 CD On-Demand Anodyne MTNR1A 89 45 CNC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863350 CD On-Demand Anodyne MTNR1B 73 38 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863357 FG On-Demand Anodyne NQO2 23 42 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863357 FG On-Demand Anodyne MTNR1A 44 41 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863357 FG On-Demand Anodyne MTNR1B 41 40 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863357 FG On-Demand Anodyne TBK1 58 32 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863358 FG On-Demand Anodyne NQO2 23 42 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863358 FG On-Demand Anodyne MTNR1A 44 41 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863358 FG On-Demand Anodyne MTNR1B 41 40 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863358 FG On-Demand Anodyne TBK1 58 32 COCCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863370 EG On-Demand Anodyne CCR3 19 41 COCCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863370 EG On-Demand Anodyne PANC 46 32 CCC(=O)N1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863388 EG On-Demand Anodyne MTNR1A 38 43 CCC(=O)N1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863388 EG On-Demand Anodyne MTNR1B 41 50 CCCN(CC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863421 CH On-Demand Anodyne MTNR1A 44 38 CCCN(CC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863421 CH On-Demand Anodyne ROCK2 25 40 CCCCCN(C(=O)c1coc(-c2ccccn2)n1)C(C)C ZINC000880863424 DH On-Demand Anodyne FAAH 15 41 CCCN(CC)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863515 DG On-Demand Anodyne MTNR1A 58 42 CCCN(CC)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863515 DG On-Demand Anodyne MTNR1B 44 37 CCO[C@@H](CCNC(=O)Nc1cc(OC)ccc1C1CC1)C(C)C ZINC000880863546 EI On-Demand Anodyne MTNR1A 40 38 CC[C@@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863606 DG On-Demand Anodyne BMP1 18 40 CC[C@@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863606 DG On-Demand Anodyne CCR3 34 44 CC[C@@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863606 DG On-Demand Anodyne MTNR1A 53 41 CC[C@@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863606 DG On-Demand Anodyne MTNR1B 44 37 CC[C@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863607 DG On-Demand Anodyne BMP1 18 40 CC[C@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863607 DG On-Demand Anodyne CCR3 34 44 CC[C@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863607 DG On-Demand Anodyne MTNR1A 53 41 CC[C@H](O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863607 DG On-Demand Anodyne MTNR1B 44 37 CNC(=O)CCN(C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863652 DE On-Demand Anodyne MTNR1A 30 41 CCOC(=O)N1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863678 FG On-Demand Anodyne P2RY12 28 40 CCOC(=O)N1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863678 FG On-Demand Anodyne MTNR1A 38 42 CCOC(=O)N1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863678 FG On-Demand Anodyne MTNR1B 39 43 COc1ccc(N2CCCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)cc1 ZINC000880863703 GI On-Demand Clean PDGFRB 42 39 C=CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863713 DI On-Demand Mild MTNR1A 17 40 C=CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863713 DI On-Demand Mild MTNR1B 20 40 C=CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863713 DI On-Demand Mild RBP4 31 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(F)cc1)C(C)C ZINC000880863714 GG On-Demand Anodyne PAPA1_CARPA 38 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(F)cc1)C(C)C ZINC000880863714 GG On-Demand Anodyne FPR1 47 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(F)cc1)C(C)C ZINC000880863715 GG On-Demand Anodyne PAPA1_CARPA 38 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(F)cc1)C(C)C ZINC000880863715 GG On-Demand Anodyne FPR1 47 35 CCN(CCNC(=O)Nc1cc(OC)ccc1C1CC1)C1CC1 ZINC000880863721 DG On-Demand Anodyne MTNR1A 51 40 CCO[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863738 DH On-Demand Anodyne MTNR1A 24 42 CCO[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880863738 DH On-Demand Anodyne MTNR1B 27 42 CNS(=O)(=O)CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880863742 DD On-Demand Anodyne NQO2 21 44 CNS(=O)(=O)CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880863742 DD On-Demand Anodyne MTNR1A 20 41 CNS(=O)(=O)CCCNC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880863742 DD On-Demand Anodyne MTNR1B 19 41 CNS(=O)(=O)CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880863746 DD On-Demand Anodyne NQO2 21 44 CNS(=O)(=O)CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880863746 DD On-Demand Anodyne MTNR1A 20 41 CNS(=O)(=O)CCCNC(=O)CC[C@H]1CCc2ccccc21 ZINC000880863746 DD On-Demand Anodyne MTNR1B 19 41 CCC(CC)[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863765 DG On-Demand Anodyne MTNR1A 52 40 CCC(CC)[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863765 DG On-Demand Anodyne MTNR1B 43 40 COC[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863768 CF On-Demand Anodyne MTNR1A 42 43 COC[C@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863768 CF On-Demand Anodyne MTNR1B 35 43 COC[C@@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863769 CF On-Demand Anodyne MTNR1A 42 43 COC[C@@H](C)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863769 CF On-Demand Anodyne MTNR1B 35 43 CCC(CC)[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863770 DG On-Demand Anodyne MTNR1A 52 40 CCC(CC)[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863770 DG On-Demand Anodyne MTNR1B 43 40 CCCCCN(C(=O)Cc1ccccc1N1CCCC1=O)C(C)C ZINC000880863776 EH On-Demand Anodyne KCNQ2 45 34 C=C(Br)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863782 EH On-Demand Mild MTNR1A 49 37 COCCCOC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863862 FH On-Demand Anodyne MTNR1A 15 40 COCCCOC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863862 FH On-Demand Anodyne MTNR1B 18 40 CC(=O)N1CCC[C@@H]1C(=O)N1CC[C@@H](Oc2ccc(C)cn2)C1 ZINC000880863892 DD On-Demand Anodyne PREP 49 38 CC(=O)N1CCC[C@@H]1C(=O)N1CC[C@H](Oc2ccc(C)cn2)C1 ZINC000880863893 DD On-Demand Anodyne PREP 49 38 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne PDGFRB 31 45 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne CCR3 21 40 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne MTNR1A 43 34 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne MTNR1B 40 39 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne FLT4 22 42 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne FLT3 16 42 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne TBK1 28 41 CCn1cc(NC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880863929 DG On-Demand Anodyne PANC 45 31 COc1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)CC2 ZINC000880863957 FI On-Demand Anodyne MTNR1A 17 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)CC2 ZINC000880863957 FI On-Demand Anodyne MTNR1B 23 42 COc1ccc2c(c1)CN(C(=O)Nc1cc(OC)ccc1C1CC1)CC2 ZINC000880863957 FI On-Demand Anodyne AKR1C3 15 43 C=CCN(Cc1cccc(C#N)c1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863961 FJ On-Demand Mild PTGES 27 44 CC[C@H](C)N(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880863980 DG On-Demand Anodyne MTNR1A 50 39 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne DRD4 43 33 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne HRH1 16 46 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne PDGFRB 40 38 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne SIGMAR1 15 41 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne MTNR1A 18 41 CCOCCN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880863998 EF On-Demand Anodyne MTNR1B 22 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864029 GG On-Demand Anodyne PAPA1_CARPA 38 52 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864029 GG On-Demand Anodyne CTSL 17 52 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864029 GG On-Demand Anodyne FPR1 45 37 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864031 GG On-Demand Anodyne PAPA1_CARPA 38 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864031 GG On-Demand Anodyne CTSL 17 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1cccc(F)c1)C(C)C ZINC000880864031 GG On-Demand Anodyne FPR1 45 37 COc1ccnc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)c1 ZINC000880864032 GG On-Demand Anodyne PDGFRB 51 42 COc1ccnc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)c1 ZINC000880864032 GG On-Demand Anodyne EBP 22 40 COCCN(Cc1cccnc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864039 FH On-Demand Anodyne PTAFR 23 40 COCCN(Cc1cccnc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864039 FH On-Demand Anodyne CHRNA7 42 44 COCCN(Cc1cccnc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864039 FH On-Demand Anodyne ROCK1 28 42 COCCN(Cc1cccnc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864039 FH On-Demand Anodyne ROCK2 46 43 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864040 EF On-Demand Anodyne MTNR1A 19 41 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864040 EF On-Demand Anodyne MTNR1B 19 41 CCOCCCN1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)[C@@H](C)C1 ZINC000880864093 GH On-Demand Anodyne HRH2 21 40 CCOCCCN1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)[C@@H](C)C1 ZINC000880864094 GH On-Demand Anodyne HRH2 21 40 CCOCCCN1CC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)[C@H](C)C1 ZINC000880864095 GH On-Demand Anodyne HRH2 21 40 CCOCCCN1CC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)[C@H](C)C1 ZINC000880864096 GH On-Demand Anodyne HRH2 21 40 CCOc1ccnc(N2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)n1 ZINC000880864100 GG On-Demand Anodyne PDGFRB 48 38 CCCCCN(CCO)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864103 DH On-Demand Anodyne SOAT1 29 40 CCOC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864163 DF On-Demand Anodyne MTNR1A 62 39 CCOC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864163 DF On-Demand Anodyne MTNR1B 48 38 COc1cccc([C@@H](C)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864267 EI On-Demand Anodyne MTNR1A 40 41 COc1cccc([C@@H](C)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864267 EI On-Demand Anodyne MTNR1B 36 41 COc1cccc([C@H](C)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864268 EI On-Demand Anodyne MTNR1A 40 41 COc1cccc([C@H](C)NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864268 EI On-Demand Anodyne MTNR1B 36 41 COC(=O)C1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864293 EG On-Demand Anodyne MTNR1A 32 40 COC(=O)C1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864293 EG On-Demand Anodyne MTNR1B 27 40 COC(=O)C1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864293 EG On-Demand Anodyne EPHX2 40 37 CCN(Cc1ccc(C(=O)N(C)C)cc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864298 GI On-Demand Anodyne ROCK2 23 41 CCN(CC)C(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864317 FH On-Demand Anodyne MTNR1A 24 40 CCN(CC)C(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864317 FH On-Demand Anodyne MTNR1B 25 40 COCC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864363 DG On-Demand Anodyne MTNR1A 28 41 COCC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864363 DG On-Demand Anodyne MTNR1B 27 41 COCC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864363 DG On-Demand Anodyne RBP4 31 41 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild DRD4 18 40 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild CCR3 27 42 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild EPHX2 38 42 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild PDK1 46 33 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild CXCR3 17 43 C=C(C)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864367 EH On-Demand Mild MCHR1 21 45 CCNS(=O)(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864378 ED On-Demand Anodyne MTNR1A 53 42 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnc(OC)nc1)C2 ZINC000880864380 ED On-Demand Anodyne NQO2 40 44 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnc(OC)nc1)C2 ZINC000880864380 ED On-Demand Anodyne MTNR1A 91 47 COc1ccc2c(c1)CC[C@H](C(=O)NCCc1cnc(OC)nc1)C2 ZINC000880864380 ED On-Demand Anodyne MTNR1B 77 41 CCN(CC)C(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864410 EG On-Demand Anodyne CCR3 16 42 CCN(CC)C(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864410 EG On-Demand Anodyne MTNR1A 48 41 CCN(CC)C(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864410 EG On-Demand Anodyne MTNR1B 37 41 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne LPL 44 37 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne CA1 34 44 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne TRPV1 16 54 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne P2RY1 42 39 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne CCR3 47 54 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne RAF1 25 55 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne KDR 29 45 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne MTNR1A 50 49 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne MTNR1B 47 49 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne EPHX2 39 53 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne CA12 15 44 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne PDGFRA 39 45 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne CA9 16 44 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne MCHR1 15 40 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne TAAR1 36 44 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne AKR1C3 22 49 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne AKR1C2 44 41 COc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864413 DI On-Demand Anodyne KCNK3 35 44 CC[C@@H](NC(=O)Nc1cc(OC)ccc1C1CC1)c1ccncc1 ZINC000880864464 EI On-Demand Anodyne PDE4A 18 41 COC(=O)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)CC(C)C ZINC000880864481 EH On-Demand Anodyne MTNR1A 33 41 COC(=O)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)CC(C)C ZINC000880864481 EH On-Demand Anodyne MTNR1B 26 41 COC(=O)[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)CC(C)C ZINC000880864482 EH On-Demand Anodyne MTNR1A 33 41 COC(=O)[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)CC(C)C ZINC000880864482 EH On-Demand Anodyne MTNR1B 26 41 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne DRD4 60 45 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne NQO2 31 45 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne CTSL 26 42 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne CCR3 28 48 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne RAF1 19 40 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne MTNR1A 69 40 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne MTNR1B 60 41 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne CTSS 19 44 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne MCHR1 18 42 COc1cccc(C(=O)NCCNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880864485 GG On-Demand Anodyne KCNK3 17 44 CCN(Cc1ccoc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864488 DI On-Demand Anodyne ROCK2 21 43 CNC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864489 DE On-Demand Anodyne NQO2 33 42 CNC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864489 DE On-Demand Anodyne CCR3 20 44 CNC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864489 DE On-Demand Anodyne MTNR1A 69 43 CNC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864489 DE On-Demand Anodyne MTNR1B 56 37 COc1ccc(OC2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)cc1 ZINC000880864508 GJ On-Demand Anodyne PRSS2 67 32 COc1ccc(OC2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)cc1 ZINC000880864508 GJ On-Demand Anodyne EPHX2 26 52 COc1ccc(OC2CCN(C(=O)Nc3cc(OC)ccc3C3CC3)CC2)cc1 ZINC000880864508 GJ On-Demand Anodyne RBP4 30 41 COC(=O)CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864553 EG On-Demand Anodyne CCR3 21 44 COC(=O)CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864553 EG On-Demand Anodyne MTNR1A 66 40 COC(=O)CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864553 EG On-Demand Anodyne MTNR1B 55 36 COC(=O)CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864553 EG On-Demand Anodyne EPHX2 21 45 CC[C@@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864617 CF On-Demand Anodyne MTNR1A 48 36 O=C(c1cc(C(F)(F)F)ccn1)N1CC[C@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880864724 GH On-Demand Anodyne CCR2 30 42 O=C(c1cc(C(F)(F)F)ccn1)N1CC[C@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880864724 GH On-Demand Anodyne LIPG 47 49 COCCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864725 DH On-Demand Anodyne HRH2 20 44 COCCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864725 DH On-Demand Anodyne CCR3 24 45 COCCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864725 DH On-Demand Anodyne MTNR1A 73 40 COCCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864725 DH On-Demand Anodyne MTNR1B 62 37 O=C(c1cc(C(F)(F)F)ccn1)N1CC[C@@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880864727 GH On-Demand Anodyne CCR2 30 42 O=C(c1cc(C(F)(F)F)ccn1)N1CC[C@@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880864727 GH On-Demand Anodyne LIPG 47 49 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864758 EF On-Demand Anodyne CCR3 21 41 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864758 EF On-Demand Anodyne MTNR1A 20 45 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864758 EF On-Demand Anodyne MTNR1B 22 45 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864758 EF On-Demand Anodyne EPHX2 27 41 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864760 EF On-Demand Anodyne CCR3 21 41 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864760 EF On-Demand Anodyne MTNR1A 20 45 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864760 EF On-Demand Anodyne MTNR1B 22 45 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864760 EF On-Demand Anodyne EPHX2 27 41 COc1cnc(C(=O)N2CC[C@@H](Oc3ccc(C)cn3)C2)c(F)c1 ZINC000880864823 EE On-Demand Anodyne HCRTR1 15 44 COc1cnc(C(=O)N2CC[C@H](Oc3ccc(C)cn3)C2)c(F)c1 ZINC000880864824 EE On-Demand Anodyne HCRTR1 15 44 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne DRD2 22 40 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne DRD4 41 31 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne HTR4 65 43 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne SIGMAR1 27 53 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne CCR3 47 46 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne MTNR1A 31 40 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne MTNR1B 31 40 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne EBP 44 40 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne EPHX2 49 47 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne PDK1 46 33 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne CXCR3 17 43 CCCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864851 EH On-Demand Anodyne MCHR1 36 45 CCN(CCNC(=O)Nc1cc(OC)ccc1C1CC1)C(C)C ZINC000880864852 DG On-Demand Anodyne MTNR1A 53 39 CCN(CCNC(=O)Nc1cc(OC)ccc1C1CC1)C(C)C ZINC000880864852 DG On-Demand Anodyne MTNR1B 40 38 CC[C@H](C)NC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864861 EF On-Demand Anodyne NQO2 29 42 CC[C@H](C)NC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864861 EF On-Demand Anodyne CCR3 15 40 CC[C@H](C)NC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864861 EF On-Demand Anodyne MTNR1A 73 39 CC[C@H](C)NC(=O)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864861 EF On-Demand Anodyne MTNR1B 59 39 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne DRD2 19 42 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne DRD4 44 33 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne DRD3 19 42 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne HTR4 50 39 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne CCR3 47 44 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne EBP 41 37 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne EPHX2 48 45 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne PDK1 48 35 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne CXCR3 18 44 COCCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864883 EF On-Demand Anodyne MCHR1 37 47 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864905 GF On-Demand Anodyne MTNR1A 23 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864905 GF On-Demand Anodyne MTNR1B 21 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864905 GF On-Demand Anodyne EPHX2 15 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864905 GF On-Demand Anodyne CCR8 83 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864909 GG On-Demand Anodyne PAPA1_CARPA 39 52 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864909 GG On-Demand Anodyne CTSK 18 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864909 GG On-Demand Anodyne TACR3 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864909 GG On-Demand Anodyne FPR1 50 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864910 GG On-Demand Anodyne PAPA1_CARPA 39 52 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864910 GG On-Demand Anodyne CTSK 18 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864910 GG On-Demand Anodyne TACR3 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccc1F)C(C)C ZINC000880864910 GG On-Demand Anodyne FPR1 50 38 CNC(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864928 CD On-Demand Anodyne MTNR1A 67 41 CNC(=O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880864928 CD On-Demand Anodyne MTNR1B 57 39 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864957 FG On-Demand Anodyne CCR3 16 41 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864957 FG On-Demand Anodyne MTNR1A 16 41 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880864957 FG On-Demand Anodyne MTNR1B 19 41 COCC(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864962 FE On-Demand Anodyne MTNR1A 21 41 COCC(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864962 FE On-Demand Anodyne MTNR1B 23 41 COCC(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864962 FE On-Demand Anodyne EPHX2 23 43 COCC(=O)NC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880864962 FE On-Demand Anodyne RBP4 28 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccc(C)cn2)C1 ZINC000880865046 GE On-Demand Anodyne P2RY12 43 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](Oc2ccc(C)cn2)C1 ZINC000880865047 GE On-Demand Anodyne P2RY12 43 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](Oc2ccc(C)cn2)C1 ZINC000880865049 GE On-Demand Anodyne P2RY12 43 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](Oc2ccc(C)cn2)C1 ZINC000880865051 GE On-Demand Anodyne P2RY12 43 34 COCCCN(C)CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865068 EF On-Demand Anodyne MTNR1A 45 37 CCC[C@H](CCO)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865077 DG On-Demand Anodyne MTNR1A 41 39 CCC[C@@H](CCO)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865078 DG On-Demand Anodyne MTNR1A 41 39 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865083 GE On-Demand Anodyne ACOX1 50 34 COC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865109 EF On-Demand Anodyne MTNR1A 20 42 COC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865109 EF On-Demand Anodyne MTNR1B 22 42 COC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865109 EF On-Demand Anodyne RBP4 22 40 COCCOc1ccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cn1 ZINC000880865119 FG On-Demand Anodyne ROCK2 32 41 CCN(Cc1cccs1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865173 EJ On-Demand Anodyne ROCK2 21 41 COCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865193 CG On-Demand Anodyne HRH2 22 45 COCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865193 CG On-Demand Anodyne CCR3 28 45 COCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865193 CG On-Demand Anodyne MTNR1A 74 41 COCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865193 CG On-Demand Anodyne MTNR1B 63 37 CCOC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H](Oc3ccc(C)cn3)C2)C1 ZINC000880865239 EE On-Demand Anodyne PTR1 43 32 CCOC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H](Oc3ccc(C)cn3)C2)C1 ZINC000880865240 EE On-Demand Anodyne PTR1 43 32 O=C(c1ccc2c(O)ncnc2c1)N1CC[C@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880865253 GF On-Demand Anodyne PDE3B 41 34 O=C(c1ccc2c(O)ncnc2c1)N1CC[C@@H](Oc2ccc(C3CC3)cn2)C1 ZINC000880865254 GF On-Demand Anodyne PDE3B 41 34 CCC1(O)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865307 DG On-Demand Anodyne MTNR1A 29 41 CCC1(O)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865307 DG On-Demand Anodyne MTNR1B 31 41 CCC1(O)CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865307 DG On-Demand Anodyne S1PR2 29 41 CCNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865314 FD On-Demand Anodyne DRD4 41 33 CCNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865314 FD On-Demand Anodyne MTNR1A 40 50 CCNC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865314 FD On-Demand Anodyne MTNR1B 40 50 COCc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865317 EI On-Demand Anodyne MTNR1A 64 40 COCc1ccccc1CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865317 EI On-Demand Anodyne MTNR1B 54 38 CCOC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865335 DG On-Demand Anodyne CCR3 20 43 CCOC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865335 DG On-Demand Anodyne MTNR1A 58 41 CCOC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865335 DG On-Demand Anodyne MTNR1B 49 38 CCOC(=O)CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865335 DG On-Demand Anodyne EPHX2 15 42 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865336 GI On-Demand Anodyne NQO2 21 40 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865336 GI On-Demand Anodyne MTNR1A 48 42 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865336 GI On-Demand Anodyne MTNR1B 44 40 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865336 GI On-Demand Anodyne TBK1 66 34 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne PDGFRB 15 41 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne CCR3 38 45 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne ROCK1 19 43 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne MTNR1A 64 46 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne MTNR1B 58 46 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne ROCK2 38 47 CCC(=O)Nc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865344 FI On-Demand Anodyne FLT4 18 41 COCC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865372 ED On-Demand Anodyne MTNR1A 28 42 COCC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865372 ED On-Demand Anodyne MTNR1B 29 42 C#CCNS(=O)(=O)c1ccc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)cc1 ZINC000880865373 ID On-Demand Mild MPL 44 38 CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865380 BE On-Demand Anodyne MTNR1A 49 42 CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865380 BE On-Demand Anodyne MTNR1B 41 41 CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865380 BE On-Demand Anodyne AKR1C2 42 38 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865395 GF On-Demand Anodyne MTNR1A 24 42 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865395 GF On-Demand Anodyne MTNR1B 29 42 COc1ccc([C@@H](O)CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880865402 FG On-Demand Anodyne MTNR1A 51 42 COc1ccc([C@@H](O)CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880865402 FG On-Demand Anodyne MTNR1B 40 41 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne DRD4 28 43 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne CCR3 30 42 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne EPHX2 44 41 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne PDK1 48 35 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne CXCR3 18 44 CNC(=O)CN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865410 FD On-Demand Anodyne MCHR1 27 45 CCOC(=O)CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865413 FH On-Demand Anodyne MTNR1A 20 40 CCOC(=O)CC1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865413 FH On-Demand Anodyne MTNR1B 22 40 CCn1ncc(C(=O)N2CC[C@H](Oc3ccc(C)cn3)C2)c1C ZINC000880865474 DE On-Demand Anodyne HCRTR2 15 46 CCn1ncc(C(=O)N2CC[C@@H](Oc3ccc(C)cn3)C2)c1C ZINC000880865475 DE On-Demand Anodyne HCRTR2 15 46 CNS(=O)(=O)CCCNC(=O)c1cc2ccccc2cc1F ZINC000880865699 DD On-Demand Anodyne POLR1A 40 34 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865712 GJ On-Demand Mild HRH2 16 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865712 GJ On-Demand Mild CCR3 21 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865712 GJ On-Demand Mild ROCK1 27 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865712 GJ On-Demand Mild ROCK2 36 45 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865713 GJ On-Demand Mild HRH2 16 40 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865713 GJ On-Demand Mild CCR3 21 40 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865713 GJ On-Demand Mild ROCK1 27 40 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865713 GJ On-Demand Mild ROCK2 36 45 CCOCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865738 CF On-Demand Anodyne MTNR1A 74 40 CCOCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865738 CF On-Demand Anodyne MTNR1B 61 40 COCCOc1ccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880865763 FH On-Demand Anodyne MTNR1A 40 36 COCCOc1ccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880865763 FH On-Demand Anodyne ROCK2 22 40 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865779 GF On-Demand Anodyne MTNR1A 29 40 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865779 GF On-Demand Anodyne MTNR1B 26 40 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880865779 GF On-Demand Anodyne RBP4 38 40 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865797 GH On-Demand Anodyne EDNRB 74 41 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865797 GH On-Demand Anodyne EDNRA 72 41 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865797 GH On-Demand Anodyne BMP1 70 41 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865797 GH On-Demand Anodyne MCHR1 17 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865803 GG On-Demand Mild PAPA1_CARPA 48 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865803 GG On-Demand Mild FPR1 41 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865803 GG On-Demand Mild CTRB_BOVIN 57 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865804 GG On-Demand Mild PAPA1_CARPA 48 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865804 GG On-Demand Mild FPR1 41 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccc(C#N)cc1)C(C)C ZINC000880865804 GG On-Demand Mild CTRB_BOVIN 57 35 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne DRD4 49 37 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne NQO2 22 40 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne CCR3 19 40 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne MTNR1A 49 41 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne MTNR1B 43 35 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880865808 GI On-Demand Anodyne ROCK2 34 46 CCN1CC[C@H](CNC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865826 DG On-Demand Anodyne HTR4 41 32 CCN1CC[C@H](CNC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865826 DG On-Demand Anodyne CCR3 48 44 CCN1CC[C@H](CNC(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880865826 DG On-Demand Anodyne CACNA1I 59 36 C=CCN(C(=O)C(=O)c1c[nH]c2cc(F)ccc12)C(C)C ZINC000880865883 CF On-Demand Mild MPO 61 35 CCOCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865885 DH On-Demand Anodyne HRH2 20 44 CCOCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865885 DH On-Demand Anodyne CCR3 22 44 CCOCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865885 DH On-Demand Anodyne MTNR1A 68 42 CCOCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880865885 DH On-Demand Anodyne MTNR1B 57 39 C=CCN(C(=O)[C@@H](CCOC)NC(=O)OC(C)(C)C)C(C)C ZINC000880865911 DE On-Demand Mild CTSK 15 49 C=CCN(C(=O)[C@H](CCOC)NC(=O)OC(C)(C)C)C(C)C ZINC000880865912 DE On-Demand Mild CTSK 15 49 COc1ccc(O)c(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866039 EH On-Demand Clean MTNR1A 61 44 COc1ccc(O)c(CNC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866039 EH On-Demand Clean MTNR1B 50 44 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild DRD4 15 40 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild CCR3 30 42 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild EPHX2 41 36 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild PDK1 46 33 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild CXCR3 17 43 C=CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866053 EG On-Demand Mild MCHR1 23 45 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne LPL 42 35 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne CA1 23 41 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne CCR3 32 47 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne MTNR1A 35 41 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne MTNR1B 32 41 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne EPHX2 20 45 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne AKR1C3 18 41 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne AKR1C2 42 39 COC(=O)Nc1cccc(NC(=O)Nc2cc(OC)ccc2C2CC2)c1 ZINC000880866056 FI On-Demand Anodyne KCNK3 34 42 CNS(=O)(=O)CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880866061 EC On-Demand Anodyne NQO2 39 47 CNS(=O)(=O)CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880866061 EC On-Demand Anodyne MTNR1A 70 45 CNS(=O)(=O)CCCNC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880866061 EC On-Demand Anodyne MTNR1B 61 41 CNS(=O)(=O)CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880866062 EC On-Demand Anodyne NQO2 39 47 CNS(=O)(=O)CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880866062 EC On-Demand Anodyne MTNR1A 70 45 CNS(=O)(=O)CCCNC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880866062 EC On-Demand Anodyne MTNR1B 61 41 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne CA1 34 43 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne CCR3 32 43 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne RAF1 19 40 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne MTNR1A 36 40 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne MTNR1B 35 42 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne ROCK2 24 43 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne CA12 16 43 COC(=O)NCc1ccc(NC(=O)Nc2cc(OC)ccc2C2CC2)cc1 ZINC000880866070 FI On-Demand Anodyne CA9 17 43 CCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866089 FH On-Demand Anodyne NQO2 23 41 CCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866089 FH On-Demand Anodyne MTNR1A 52 42 CCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866089 FH On-Demand Anodyne MTNR1B 47 41 CCCCNC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866089 FH On-Demand Anodyne TBK1 67 34 CCS(=O)(=O)C[C@@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866091 EF On-Demand Anodyne MTNR1A 43 38 CCS(=O)(=O)C[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866092 EF On-Demand Anodyne MTNR1A 43 38 C#CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866106 CF On-Demand Mild CCR3 15 41 C#CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866106 CF On-Demand Mild MTNR1A 71 41 C#CCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866106 CF On-Demand Mild MTNR1B 59 41 CCN(CC)C(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866110 GF On-Demand Anodyne MTNR1A 15 43 CCN(CC)C(=O)CN1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866110 GF On-Demand Anodyne MTNR1B 19 43 CCC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866147 CF On-Demand Anodyne MTNR1A 51 40 CCC[C@@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866147 CF On-Demand Anodyne MTNR1B 42 40 CCC[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866148 CF On-Demand Anodyne MTNR1A 51 40 CCC[C@H](O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866148 CF On-Demand Anodyne MTNR1B 42 40 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866176 DG On-Demand Anodyne CCR3 16 49 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866176 DG On-Demand Anodyne MTNR1A 25 42 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866176 DG On-Demand Anodyne MTNR1B 27 42 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866176 DG On-Demand Anodyne RBP4 25 40 CC[C@H](C)[C@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866233 DG On-Demand Anodyne MTNR1A 40 38 CC[C@@H](C)[C@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866234 DG On-Demand Anodyne MTNR1A 40 38 CC[C@H](C)[C@@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866235 DG On-Demand Anodyne MTNR1A 40 38 CC[C@@H](C)[C@@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866236 DG On-Demand Anodyne MTNR1A 40 38 CCCO[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866238 EI On-Demand Anodyne MTNR1B 19 41 CCCO[C@@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866239 EI On-Demand Anodyne MTNR1B 19 41 COC(=O)[C@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)Cc1ccc(O)cc1 ZINC000880866242 GG On-Demand Anodyne YARS 41 32 COC(=O)[C@@H](CNC(=O)Nc1cc(OC)ccc1C1CC1)Cc1ccc(O)cc1 ZINC000880866243 GG On-Demand Anodyne YARS 41 32 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MMP13 26 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MTNR1A 34 44 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MTNR1B 31 44 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MMP3 26 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MMP9 17 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne MMP1 21 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866268 FE On-Demand Anodyne RBP4 39 42 C#CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866289 BE On-Demand Mild MTNR1A 73 42 C#CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866289 BE On-Demand Mild MTNR1B 61 47 CCC[C@](C)(O)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866296 DG On-Demand Anodyne MTNR1A 43 36 CCOC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866300 EH On-Demand Anodyne MTNR1A 21 40 CCOC[C@H]1CCCN(C(=O)Nc2cc(OC)ccc2C2CC2)C1 ZINC000880866300 EH On-Demand Anodyne MTNR1B 24 40 C=C(Cl)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866321 CG On-Demand Mild MTNR1A 53 38 C=C(Cl)CNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866321 CG On-Demand Mild MTNR1B 45 39 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866322 GI On-Demand Anodyne TSPO 18 41 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866322 GI On-Demand Anodyne ROCK2 22 40 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866322 GI On-Demand Anodyne TNKS 57 32 CC[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866339 CG On-Demand Anodyne MTNR1A 54 40 CC[C@H](C)NC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866339 CG On-Demand Anodyne MTNR1B 48 40 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne HRH2 17 43 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne NQO2 40 44 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne CCR3 32 46 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne MTNR1A 96 47 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne MTNR1B 82 40 CCCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866343 CH On-Demand Anodyne EPHX2 17 44 CCOC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866457 EF On-Demand Anodyne P2RY12 41 42 CCOC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866457 EF On-Demand Anodyne MTNR1A 47 44 CCOC(=O)N1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866457 EF On-Demand Anodyne MTNR1B 44 44 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne HTR4 24 42 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne CCR3 35 44 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne MTNR1A 41 41 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne MTNR1B 38 41 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne EPHX2 48 50 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne PDK1 48 35 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne CXCR3 20 46 CCN1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866540 DG On-Demand Anodyne MCHR1 29 47 CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866618 CG On-Demand Anodyne HRH2 18 44 CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866618 CG On-Demand Anodyne NQO2 41 44 CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866618 CG On-Demand Anodyne CCR3 33 47 CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866618 CG On-Demand Anodyne MTNR1A 100 47 CCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866618 CG On-Demand Anodyne MTNR1B 88 41 C=CCN(CC=C)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866632 CH On-Demand Mild MTNR1A 41 39 CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866656 CG On-Demand Anodyne HRH2 25 46 CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866656 CG On-Demand Anodyne NQO2 36 40 CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866656 CG On-Demand Anodyne CCR3 25 45 CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866656 CG On-Demand Anodyne MTNR1A 78 43 CCOCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866656 CG On-Demand Anodyne MTNR1B 65 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccn1)C(C)C ZINC000880866665 FF On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(Cc1ccccn1)C(C)C ZINC000880866666 FF On-Demand Anodyne FPR1 45 36 CCN(Cc1ccncc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866668 EI On-Demand Anodyne ROCK1 16 44 CCN(Cc1ccncc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866668 EI On-Demand Anodyne ROCK2 24 44 CCOC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866674 FG On-Demand Anodyne GRIN2B 19 41 CCOC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866674 FG On-Demand Anodyne MTNR1A 35 41 CCOC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866674 FG On-Demand Anodyne MTNR1B 33 41 CCOC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866674 FG On-Demand Anodyne EPHX2 54 53 CCOC(=O)N1CCC(NC(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866674 FG On-Demand Anodyne MCHR1 17 41 C=CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866677 BF On-Demand Mild MTNR1A 59 39 C=CCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866677 BF On-Demand Mild MTNR1B 51 41 CCCCN(CC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866780 CI On-Demand Anodyne MTNR1A 37 40 CCCCN(CC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866780 CI On-Demand Anodyne MTNR1B 34 40 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne DRD4 40 30 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne HRH2 24 48 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne NQO2 38 41 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne CCR3 30 46 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne MTNR1A 80 42 COCCCNC(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866798 CF On-Demand Anodyne MTNR1B 69 39 CCOC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866819 EG On-Demand Anodyne MTNR1A 26 40 CCOC(=O)C1CCN(C(=O)Nc2cc(OC)ccc2C2CC2)CC1 ZINC000880866819 EG On-Demand Anodyne MTNR1B 27 40 CCCN(CCC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866905 CI On-Demand Anodyne MTNR1A 53 39 CCCN(CCC)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866905 CI On-Demand Anodyne MTNR1B 47 39 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne OPRD1 19 41 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne ROCK1 18 47 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne MTNR1A 43 38 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne MTNR1B 44 38 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne ROCK2 36 47 CCN(Cc1ccccc1)C(=O)Nc1cc(OC)ccc1C1CC1 ZINC000880866909 DJ On-Demand Anodyne PTGES 23 45 C=CC(C)(C)CC(=O)N(Cc1ccc([N+](=O)[O-])cc1)C(C)C ZINC000880866999 DH On-Demand Mild COLA 24 42 C=CC(C)(C)CC(=O)N(Cc1ccc([N+](=O)[O-])cc1)C(C)C ZINC000880866999 DH On-Demand Mild MMP2 18 42 C=CC(C)(C)CC(=O)N(Cc1ccc([N+](=O)[O-])cc1)C(C)C ZINC000880866999 DH On-Demand Mild MMP8 36 42 C=CC(C)(C)CC(=O)N(Cc1ccc([N+](=O)[O-])cc1)C(C)C ZINC000880866999 DH On-Demand Mild MMP9 19 42 C=CC(C)(C)CC(=O)N(Cc1ccc([N+](=O)[O-])cc1)C(C)C ZINC000880866999 DH On-Demand Mild MMP1 27 42 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1Cc2ccccc2NC1=O ZINC000880867033 FF On-Demand Anodyne PYGM 17 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1Cc2ccccc2NC1=O ZINC000880867034 FF On-Demand Anodyne PYGM 17 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880867091 GF On-Demand Anodyne PYGL 34 46 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880867091 GF On-Demand Anodyne PYGM 30 46 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880867092 GF On-Demand Anodyne PYGL 34 46 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880867092 GF On-Demand Anodyne PYGM 30 46 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](O)c1ccccc1OC ZINC000880867120 GG On-Demand Anodyne SOAT1 33 42 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)c1cccc(O)c1 ZINC000880867165 EH On-Demand Anodyne HSD17B2 49 42 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1CCN(C(C)=O)C1 ZINC000880867169 ED On-Demand Anodyne EPHX2 29 42 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880867295 FF On-Demand Anodyne PLM1_PLAFA 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880867295 FF On-Demand Anodyne PLM2_PLAFA 70 41 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccnc1N1CCCC1 ZINC000880867361 GG On-Demand Anodyne SCN10A 16 41 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(=O)C(C)(C)C)CC1 ZINC000880867494 GG On-Demand Anodyne EPHX2 41 40 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)[C@H](CO)Cc1ccccc1 ZINC000880867759 GG On-Demand Anodyne NPY5R 28 45 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)[C@@H](CO)Cc1ccccc1 ZINC000880867760 GG On-Demand Anodyne NPY5R 28 45 COC(=O)c1c(C)sc(C)c1NC(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880867812 GF On-Demand Anodyne CASR 56 43 Cc1coc(C(=O)NC[C@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880867846 DD On-Demand Anodyne DRD4 17 42 Cc1coc(C(=O)NC[C@@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880867847 DD On-Demand Anodyne DRD4 17 42 O=C(C[C@@H]1C[C@H]1C1CC1)NCc1ccnc(-c2ccccc2)c1 ZINC000880867853 DH On-Demand Anodyne NOS2 71 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1csc(C(F)(F)F)c1 ZINC000880867865 GG On-Demand Anodyne PAPA1_CARPA 40 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1csc(C(F)(F)F)c1 ZINC000880867866 GG On-Demand Anodyne PAPA1_CARPA 40 44 CCC1(N2CCOCC2)CCN(C(=O)c2cncc3[nH]ccc23)CC1 ZINC000880867908 EE On-Demand Anodyne ATR 41 32 CCC1(N2CCOCC2)CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880867922 EE On-Demand Anodyne ACACA 51 52 CCC1(N2CCOCC2)CCN(C(=O)c2cnc3cc[nH]c3c2)CC1 ZINC000880867922 EE On-Demand Anodyne ACACB 33 52 O=C(COC1CC1)NCc1ccnc(-c2ccccc2)c1 ZINC000880867932 CF On-Demand Anodyne NOS2 70 33 O=C(COC1CC1)NCc1ccnc(-c2ccccc2)c1 ZINC000880867932 CF On-Demand Anodyne VCP 56 36 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880868088 DD On-Demand Anodyne LUXR 69 39 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880868088 DD On-Demand Anodyne TRAR 84 39 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880868088 DD On-Demand Anodyne LASR 62 39 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H](CCO)c1ccc(OC)cc1 ZINC000880868133 GG On-Demand Anodyne UTS2 22 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H](CCO)c1ccc(OC)cc1 ZINC000880868134 GG On-Demand Anodyne UTS2 22 41 O=C(NCc1ccnc(-c2ccccc2)c1)c1ccc(CN2CCOCC2)o1 ZINC000880868247 GG On-Demand Anodyne HDAC1 18 45 O=C(NCc1ccnc(-c2ccccc2)c1)c1ccc(CN2CCOCC2)o1 ZINC000880868247 GG On-Demand Anodyne HPGDS 31 41 O=C(NCc1ccnc(-c2ccccc2)c1)c1ccc(CN2CCOCC2)o1 ZINC000880868247 GG On-Demand Anodyne NAMPT 37 41 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)c1ncccc1-c1ccccn1 ZINC000880868271 GE On-Demand Anodyne DRD4 17 40 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)c1ncccc1-c1ccccn1 ZINC000880868272 GE On-Demand Anodyne DRD4 17 40 CS(=O)(=O)C1CCC(C(=O)NCc2ccnc(-c3ccccc3)c2)CC1 ZINC000880868294 FF On-Demand Anodyne F11 31 44 CS(=O)(=O)C1CCC(C(=O)NCc2ccnc(-c3ccccc3)c2)CC1 ZINC000880868294 FF On-Demand Anodyne VCP 56 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne PGC 47 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne PAPA1_CARPA 52 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne CCKAR 44 35 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne CTSK 27 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne CTSL 39 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne TACR3 26 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne REN 62 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne CTSS 26 48 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne CAPN1 18 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne SCN10A 21 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868329 GG On-Demand Anodyne FPR1 50 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne PGC 47 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne PAPA1_CARPA 52 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne CCKAR 44 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne CTSK 27 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne CTSL 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne TACR3 26 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne REN 62 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne CTSS 26 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne CAPN1 18 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne SCN10A 21 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868330 GG On-Demand Anodyne FPR1 50 42 Cn1nc2c(c1C(=O)NCC(=O)Nc1ccc3c(c1)OCCO3)CSCC2 ZINC000880868332 GD On-Demand Anodyne QPCT 16 40 Cc1cnc(Cl)c(C(=O)NC[C@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880868368 FE On-Demand Anodyne DRD4 20 47 Cc1cnc(Cl)c(C(=O)NC[C@@H]2CN(Cc3ccncc3)CCO2)c1 ZINC000880868369 FE On-Demand Anodyne DRD4 20 47 O=C(C[C@@H]1CCNC1=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868400 DD On-Demand Anodyne NOS2 64 33 O=C(C[C@H]1CCNC1=O)NCc1ccnc(-c2ccccc2)c1 ZINC000880868401 DD On-Demand Anodyne NOS2 64 33 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](NC(=O)NC2CC2)C1 ZINC000880868404 GE On-Demand Anodyne EPHX2 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@H](NC(=O)NC2CC2)C1 ZINC000880868405 GE On-Demand Anodyne EPHX2 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ccc(F)cn2)CC1 ZINC000880868429 GG On-Demand Anodyne DGAT1 28 44 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ccc(F)cn2)CC1 ZINC000880868429 GG On-Demand Anodyne SLC27A1 57 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880868449 GI On-Demand Anodyne GRIN2B 48 39 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880868449 GI On-Demand Anodyne CHRNA7 51 42 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880868449 GI On-Demand Anodyne C3AR1 41 41 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)c1cc2ccccc2cc1F ZINC000880868530 GG On-Demand Anodyne DRD4 30 42 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)c1cc2ccccc2cc1F ZINC000880868530 GG On-Demand Anodyne CCR3 29 45 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)c1cc2ccccc2cc1F ZINC000880868531 GG On-Demand Anodyne DRD4 30 42 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)c1cc2ccccc2cc1F ZINC000880868531 GG On-Demand Anodyne CCR3 29 45 C[C@H]1CCc2n[nH]cc2[C@@H]1C(=O)NC[C@@H]1CCCN1C ZINC000880868609 CD On-Demand Anodyne CHRNA10 52 34 C[C@H]1CCc2n[nH]cc2[C@H]1C(=O)NC[C@@H]1CCCN1C ZINC000880868610 CD On-Demand Anodyne CHRNA10 52 34 O=C(NC[C@H]1CN(Cc2ccncc2)CCO1)c1cccn2nccc12 ZINC000880868676 FD On-Demand Anodyne DRD4 16 40 O=C(NC[C@@H]1CN(Cc2ccncc2)CCO1)c1cccn2nccc12 ZINC000880868677 FD On-Demand Anodyne DRD4 16 40 CCCOc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1C ZINC000880868695 CE On-Demand Anodyne ENPP1 63 36 CCCOc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1C ZINC000880868696 CE On-Demand Anodyne ENPP1 63 36 CCCOc1ccc(NC(=O)Cc2csc(S[C@@H](C)C(N)=O)n2)cc1F ZINC000880868698 GG On-Demand Anodyne ENPP1 54 30 CCCOc1ccc(NC(=O)Cc2csc(S[C@H](C)C(N)=O)n2)cc1F ZINC000880868699 GG On-Demand Anodyne ENPP1 54 30 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne HTR2A 24 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne MST1R 17 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne MET 63 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne EPHX2 21 44 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne MAPK12 18 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne STK10 20 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne EPHA8 15 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne EPHA5 17 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne EPHA4 16 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne EPHA6 22 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne RET 16 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne TIE1 18 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne DDR2 16 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1F ZINC000880868720 FG On-Demand Anodyne CDK8 20 40 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCc2cnc(C(C)C)nc2C1 ZINC000880868739 GH On-Demand Anodyne MAPK1 52 38 CCCOc1ccc(NC(=O)CN2CCCCS2(=O)=O)cc1F ZINC000880868760 ED On-Demand Anodyne MET 55 37 CCCOc1ccc(NC(=O)CN2CCCCS2(=O)=O)cc1F ZINC000880868760 ED On-Demand Anodyne ENPP1 49 32 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880868885 GG On-Demand Anodyne TRPV1 15 47 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880868885 GG On-Demand Anodyne RBP4 17 43 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880868890 FH On-Demand Anodyne CCR3 58 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@H](Cc2ccncc2)C1 ZINC000880868891 FH On-Demand Anodyne CCR3 58 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CN(Cc3ccncc3)CCO1)C2 ZINC000880868909 GE On-Demand Anodyne DRD4 22 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1CN(Cc3ccncc3)CCO1)C2 ZINC000880868909 GE On-Demand Anodyne PDK1 41 41 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CN(Cc3ccncc3)CCO1)C2 ZINC000880868910 GE On-Demand Anodyne DRD4 22 42 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@H]1CN(Cc3ccncc3)CCO1)C2 ZINC000880868910 GE On-Demand Anodyne PDK1 41 41 Cc1coc(C(=O)NCC(=O)Nc2ccc3c(c2)OCCO3)c1 ZINC000880868937 DD On-Demand Anodyne QPCT 15 40 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880868963 FF On-Demand Anodyne TBK1 49 34 O=C(NCc1csc(C(F)(F)F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880868976 FG On-Demand Anodyne NAMPT 19 40 CCCOc1ccc(NC(=O)c2c3c(nn2C)CCSC3)cc1F ZINC000880868977 EG On-Demand Anodyne KDR 15 40 CCCOc1ccc(NC(=O)c2c3c(nn2C)CCSC3)cc1F ZINC000880868977 EG On-Demand Anodyne MET 76 34 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](CO)c1ccccc1 ZINC000880868996 FG On-Demand Anodyne SOAT1 25 42 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](CO)c1ccccc1 ZINC000880868998 FG On-Demand Anodyne SOAT1 25 42 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1C ZINC000880869004 CD On-Demand Anodyne PDE5A 18 44 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1C ZINC000880869004 CD On-Demand Anodyne ENPP1 74 38 CCCOc1ccc(NC(=O)CN2CCCCS2(=O)=O)cc1C ZINC000880869016 EE On-Demand Anodyne ENPP1 61 34 NC(=O)[C@@H]1CC[C@H](C(=O)NCC2(C(F)(F)F)CCCC2)N1Cc1ccccc1 ZINC000880869017 GF On-Demand Anodyne CACNA1G 18 42 CCCOc1ccc(NC(=O)Cc2cnc(C)o2)cc1C ZINC000880869030 CG On-Demand Anodyne ENPP1 61 34 CCC(=O)N1CC[C@@H](NC(=O)Nc2c(C)sc(C)c2C(=O)OC)C1 ZINC000880869070 FE On-Demand Anodyne EPHX2 31 47 CCC(=O)N1CC[C@H](NC(=O)Nc2c(C)sc(C)c2C(=O)OC)C1 ZINC000880869071 FE On-Demand Anodyne EPHX2 31 47 O=C(NCc1cccnc1O)c1ncsc1C1CC1 ZINC000880869085 CE On-Demand Anodyne MAP1 63 33 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1O)C2 ZINC000880869093 DE On-Demand Anodyne NQO2 32 41 COc1ccc2c(c1)CC[C@H](C(=O)NCc1cccnc1O)C2 ZINC000880869093 DE On-Demand Anodyne MTNR1A 44 43 O=C(NCc1cccnc1O)c1ccc(CN2CCOCC2)o1 ZINC000880869146 DD On-Demand Anodyne SCN10A 19 42 CCCOc1ccc(NC(=O)Cc2csc(S[C@H](C)C(N)=O)n2)cc1C ZINC000880869206 GG On-Demand Anodyne ENPP1 62 34 CCCOc1ccc(NC(=O)Cc2csc(S[C@@H](C)C(N)=O)n2)cc1C ZINC000880869207 GG On-Demand Anodyne ENPP1 62 34 CCCOc1ccc(NC(=O)c2ncsc2C2CC2)cc1F ZINC000880869208 DI On-Demand Anodyne MAP1 77 34 CCCOc1ccc(NC(=O)c2ncsc2C2CC2)cc1F ZINC000880869208 DI On-Demand Anodyne KDR 15 40 CCCOc1ccc(NC(=O)c2ncsc2C2CC2)cc1F ZINC000880869208 DI On-Demand Anodyne MET 78 34 O=C(NCC1(C(F)(F)F)CCCC1)c1cccn2nccc12 ZINC000880869214 DG On-Demand Anodyne HCN1 60 35 O=C(NCC1(C(F)(F)F)CCCC1)c1cccn2nccc12 ZINC000880869214 DG On-Demand Anodyne HCN4 52 33 CCCOc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1F ZINC000880869239 CE On-Demand Anodyne MET 56 39 CCCOc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1F ZINC000880869239 CE On-Demand Anodyne ENPP1 55 32 CCCOc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1F ZINC000880869240 CE On-Demand Anodyne MET 56 39 CCCOc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1F ZINC000880869240 CE On-Demand Anodyne ENPP1 55 32 CCCOc1ccc(NC(=O)[C@@H]2CCc3nncn3CC2)cc1F ZINC000880869241 EF On-Demand Anodyne MET 62 36 CCCOc1ccc(NC(=O)[C@H]2CCc3nncn3CC2)cc1F ZINC000880869242 EF On-Demand Anodyne MET 62 36 CCCOc1ccc(NC(=O)Cn2ccc(C(=O)OC)n2)cc1C ZINC000880869258 EE On-Demand Anodyne ENPP1 68 36 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1c2ccccc2C[C@H]1O ZINC000880869368 FF On-Demand Anodyne PLM1_PLAFA 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H]1c2ccccc2C[C@H]1O ZINC000880869368 FF On-Demand Anodyne PLM2_PLAFA 70 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880869369 FF On-Demand Anodyne PLM1_PLAFA 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880869369 FF On-Demand Anodyne PLM2_PLAFA 70 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880869370 FF On-Demand Anodyne PLM1_PLAFA 41 41 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880869370 FF On-Demand Anodyne PLM2_PLAFA 70 41 Cn1nnc(C(=O)N2CCN(Cc3cc4ccccc4[nH]3)CC2)n1 ZINC000880869416 EC On-Demand Anodyne HRH4 25 52 Cn1nnc(C(=O)N2CCN(Cc3cc4ccccc4[nH]3)CC2)n1 ZINC000880869416 EC On-Demand Anodyne AKR1C3 16 40 Cn1ncc(Br)c1CC(=O)NCc1cccnc1O ZINC000880869419 ED On-Demand Anodyne P2RX7 23 46 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1F ZINC000880869463 DG On-Demand Anodyne KDR 16 43 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1F ZINC000880869463 DG On-Demand Anodyne MET 89 36 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1F ZINC000880869463 DG On-Demand Anodyne ENPP1 55 35 CCCOc1ccc(NC(=O)c2c[nH]cc2C2CC2)cc1C ZINC000880869502 CI On-Demand Anodyne HTR1F 53 34 CCC1(N2CCOCC2)CCN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880869613 GF On-Demand Anodyne MTNR1B 16 43 CCC1(N2CCOCC2)CCN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)CC1 ZINC000880869623 GF On-Demand Anodyne MTNR1B 16 43 CC(C)(C)OC(=O)N1C[C@]2(C)CN(C(=O)COC3CC3)C[C@]2(C)C1 ZINC000880869784 EE On-Demand Anodyne GPR119 25 41 COCCC(=O)N1CCC(NC(=O)Nc2c(C)sc(C)c2C(=O)OC)CC1 ZINC000880869830 GE On-Demand Anodyne EPHX2 35 44 CCCOc1ccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cc1F ZINC000880869835 FH On-Demand Anodyne MET 70 36 CCCOc1ccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cc1F ZINC000880869836 FH On-Demand Anodyne MET 70 36 CC(C)(C(=O)NCc1cccnc1O)c1ccc(C(F)(F)F)cc1 ZINC000880869914 EG On-Demand Anodyne SUCNR1 20 43 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880869921 GG On-Demand Anodyne EPHX2 20 45 CCn1nc2c(cc1=O)CN(C(=O)Nc1c(C)sc(C)c1C(=O)OC)CC2 ZINC000880869982 GE On-Demand Anodyne P2RY14 44 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC1(C(F)(F)F)CCCC1 ZINC000880870004 GG On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC1(C(F)(F)F)CCCC1 ZINC000880870006 GG On-Demand Anodyne PAPA1_CARPA 37 45 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne ATF1 53 32 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne KDR 19 49 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne MST1R 43 37 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne MET 65 40 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne NFKB1 49 32 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne KCNK3 41 35 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1F ZINC000880870013 DI On-Demand Anodyne KCNK9 48 35 CCCOc1ccc(NC(=O)COC2CC2)cc1F ZINC000880870035 CF On-Demand Anodyne MET 51 38 CCCOc1ccc(NC(=O)COC2CC2)cc1C ZINC000880870050 CF On-Demand Anodyne ENPP1 56 34 COC(=O)c1c(C)sc(C)c1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880870262 GD On-Demand Anodyne CASR 60 46 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1C ZINC000880870276 DH On-Demand Anodyne ENPP1 62 36 C=CC(C)(C)CC(=O)Nc1ccc(COC)c(OC)c1 ZINC000880870278 CG On-Demand Mild ENPP1 72 35 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1F ZINC000880870324 CD On-Demand Anodyne HTR2A 30 40 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1F ZINC000880870324 CD On-Demand Anodyne KDR 21 45 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1F ZINC000880870324 CD On-Demand Anodyne MET 99 38 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1F ZINC000880870324 CD On-Demand Anodyne ENPP1 70 34 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(=O)OC)CC1 ZINC000880870366 FF On-Demand Anodyne EPHX2 40 41 COc1ccccc1-c1ccc(C(=O)NCC2(C(F)(F)F)CCCC2)c(O)n1 ZINC000880870399 GI On-Demand Anodyne KCNA3 47 40 COc1ccccc1-c1ccc(C(=O)NCC2(C(F)(F)F)CCCC2)c(O)n1 ZINC000880870399 GI On-Demand Anodyne HCN1 72 41 COc1ccccc1-c1ccc(C(=O)NCC2(C(F)(F)F)CCCC2)c(O)n1 ZINC000880870399 GI On-Demand Anodyne HCN4 55 41 COC(=O)c1c(C)sc(C)c1NC(=O)Nc1cc(C2CC2)[nH]n1 ZINC000880870443 EG On-Demand Anodyne PKNB 50 33 CCCOc1ccc(NC(=O)Cn2nc(C)oc2=O)cc1C ZINC000880870450 DD On-Demand Anodyne ENPP1 61 35 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCC(OC)CC1 ZINC000880870475 EG On-Demand Anodyne EPHX2 30 48 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](c2nc(C)no2)C1 ZINC000880870504 FF On-Demand Anodyne ETHR 47 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@H](c2nc(C)no2)C1 ZINC000880870505 FF On-Demand Anodyne ETHR 47 35 Cn1nnc(C(=O)N2CCN(Cc3ccc(C(F)(F)F)cc3)C(=O)C2)n1 ZINC000880870625 FC On-Demand Anodyne P2RX7 19 50 O=C(NCc1cccnc1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880870639 FE On-Demand Anodyne GRIN2B 21 43 O=C(NCc1cccnc1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880870639 FE On-Demand Anodyne PREP 26 40 O=C(NCc1cccnc1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880870639 FE On-Demand Anodyne LGMN 41 37 O=C(NCc1cccnc1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880870639 FE On-Demand Anodyne Q9NAW4_PLAFA 38 44 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(Cc2ccccn2)CC1 ZINC000880870653 GF On-Demand Anodyne FAAH 16 40 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccccc1Cn1ccnc1 ZINC000880870876 GH On-Demand Anodyne CYP19A1 25 41 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccccc1Cn1ccnc1 ZINC000880870876 GH On-Demand Anodyne CYP11B1 35 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccccc1Cn1ccnc1 ZINC000880870876 GH On-Demand Anodyne TBXAS1 38 42 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccccc1Cn1ccnc1 ZINC000880870876 GH On-Demand Anodyne CYP11B2 22 44 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000880870891 GF On-Demand Anodyne EPHX2 39 51 COc1ccccc1-c1ccc(CN(C(=O)C[C@@H]2CCNC2=O)C(C)C)cc1 ZINC000880871022 GH On-Demand Anodyne MBTPS1 49 35 COc1ccccc1-c1ccc(CN(C(=O)C[C@H]2CCNC2=O)C(C)C)cc1 ZINC000880871023 GH On-Demand Anodyne MBTPS1 49 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880871054 GG On-Demand Anodyne EPHX2 21 46 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880871055 GG On-Demand Anodyne EPHX2 21 46 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCCC[C@@H]1c1nc(C)no1 ZINC000880871296 GH On-Demand Anodyne CPT1A 46 38 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCCC[C@H]1c1nc(C)no1 ZINC000880871297 GH On-Demand Anodyne CPT1A 46 38 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](O)c1ccccc1OC ZINC000880871706 GG On-Demand Anodyne SOAT1 33 42 COC(=O)c1c(C)sc(C)c1NC(=O)NCC1(N2CCCC2)CCOCC1 ZINC000880871713 GF On-Demand Anodyne HCN1 42 36 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)[C@@H](C)c1cccnc1 ZINC000880871739 EH On-Demand Anodyne KCNA5 19 41 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)[C@H](C)c1cccnc1 ZINC000880871740 EH On-Demand Anodyne KCNA5 19 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880871751 GI On-Demand Anodyne PRCP 50 39 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880871752 GI On-Demand Anodyne PRCP 50 39 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@H](N2CCCCC2)C1 ZINC000880871784 FG On-Demand Anodyne L3MBTL3 79 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](N2CCCCC2)C1 ZINC000880871785 FG On-Demand Anodyne L3MBTL3 79 41 COC(=O)c1c(C)sc(C)c1NC(=O)N(CCC#N)CCN1CCOCC1 ZINC000880871834 GE On-Demand Mild CASR 57 44 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@H](C)Cn1cncn1 ZINC000880871877 ED On-Demand Anodyne HIS3 79 35 COC(=O)c1c(C)sc(C)c1NC(=O)N[C@@H](C)Cn1cncn1 ZINC000880871878 ED On-Demand Anodyne HIS3 79 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@@H](N2CCCC2)C1 ZINC000880871915 FF On-Demand Anodyne L3MBTL3 82 42 COC(=O)c1c(C)sc(C)c1NC(=O)N1CC[C@H](N2CCCC2)C1 ZINC000880871916 FF On-Demand Anodyne L3MBTL3 82 42 Cc1cc(O)cc(NC(=O)[C@@H]2CCc3nncn3CC2)c1 ZINC000880872059 CD On-Demand Anodyne EPHX2 16 41 Cc1cc(O)cc(NC(=O)[C@H]2CCc3nncn3CC2)c1 ZINC000880872060 CD On-Demand Anodyne EPHX2 16 41 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC(N2CCCCC2)CC1 ZINC000880872065 GH On-Demand Anodyne L3MBTL3 90 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)cc(O)c1 ZINC000880872071 EF On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)cc(O)c1 ZINC000880872071 EF On-Demand Anodyne FPR1 40 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)cc(O)c1 ZINC000880872072 EF On-Demand Anodyne PAPA1_CARPA 38 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cc(C)cc(O)c1 ZINC000880872072 EF On-Demand Anodyne FPR1 40 33 CS(=O)(=O)C1CCC(C(=O)Nc2cccc(SC(F)(F)F)c2)CC1 ZINC000880872085 GH On-Demand Anodyne ITGAL 40 32 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(CC2CC2)CC1 ZINC000880872094 FG On-Demand Anodyne CXCR3 15 42 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(=O)CC(C)C)CC1 ZINC000880872100 GG On-Demand Anodyne EPHX2 36 51 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(C)cc(O)c1)C2 ZINC000880872101 DG On-Demand Anodyne MTNR1A 20 43 COc1ccc2c(c1)CC[C@H](C(=O)Nc1cc(C)cc(O)c1)C2 ZINC000880872101 DG On-Demand Anodyne MTNR1B 20 43 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCCn1ccnc1 ZINC000880872129 FF On-Demand Anodyne TBXAS1 44 46 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCCn1ccnc1 ZINC000880872129 FF On-Demand Anodyne QPCT 46 52 Cc1coc(C(=O)N[C@H](CCO)c2cc(Cl)cc(Cl)c2)c1 ZINC000880872185 EH On-Demand Anodyne UTS2 48 36 Cc1coc(C(=O)N[C@@H](CCO)c2cc(Cl)cc(Cl)c2)c1 ZINC000880872186 EH On-Demand Anodyne UTS2 48 36 O=C(/C=C\c1cccnc1)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880872195 EF On-Demand Anodyne C3AR1 27 40 O=C(/C=C\c1cccnc1)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880872195 EF On-Demand Anodyne NAMPT 84 58 O=C(Nc1cccc(SC(F)(F)F)c1)c1c[nH]cc1C1CC1 ZINC000880872264 EJ On-Demand Anodyne HTR1F 41 34 O=C(Nc1cccc(SC(F)(F)F)c1)c1c[nH]cc1C1CC1 ZINC000880872264 EJ On-Demand Anodyne KCNK3 61 36 O=C(Nc1cccc(SC(F)(F)F)c1)c1c[nH]cc1C1CC1 ZINC000880872264 EJ On-Demand Anodyne KCNK9 50 36 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(O)c1 ZINC000880872273 EG On-Demand Anodyne ROCK2 22 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(O)c1 ZINC000880872273 EG On-Demand Anodyne PKN1 15 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(O)c1 ZINC000880872273 EG On-Demand Anodyne IKBKE 15 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(O)c1 ZINC000880872273 EG On-Demand Anodyne PAK1 15 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(O)c1 ZINC000880872273 EG On-Demand Anodyne DMPK 15 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccc(C)nc1 ZINC000880872279 EG On-Demand Anodyne NAMPT 21 47 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@H](N2CCCC2)C1 ZINC000880872316 FG On-Demand Anodyne L3MBTL3 41 37 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@@H](N2CCCC2)C1 ZINC000880872317 FG On-Demand Anodyne L3MBTL3 41 37 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(CCN(C)C)CC1 ZINC000880872334 GE On-Demand Anodyne SLC6A5 16 41 CN(C)S(=O)(=O)N1CC(NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880872369 GD On-Demand Anodyne UTS2R 24 41 C[C@H]1CC(=O)N(C)c2ccc(NC(=O)Cc3ccccc3N3CCCC3=O)cc21 ZINC000880872389 GG On-Demand Anodyne KCNQ2 62 36 Cn1nnc(C(=O)N[C@@H](CCO)c2cc(Cl)cc(Cl)c2)n1 ZINC000880872391 ED On-Demand Anodyne UTS2 40 32 Cn1nnc(C(=O)N[C@H](CCO)c2cc(Cl)cc(Cl)c2)n1 ZINC000880872392 ED On-Demand Anodyne UTS2 40 32 C[C@H]1CC(=O)N(C)c2ccc(NC(=O)c3ccc([C@H]4CCC(=O)N4)cc3)cc21 ZINC000880872412 GG On-Demand Anodyne HTR1F 21 41 C[C@H]1CC(=O)N(C)c2ccc(NC(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)cc21 ZINC000880872413 GG On-Demand Anodyne HTR1F 21 41 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)CCN1CCOCC1 ZINC000880872430 FD On-Demand Anodyne CASR 47 40 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880872524 GF On-Demand Anodyne CHRNA7 41 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880872524 GF On-Demand Anodyne FAAH 30 46 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000880872542 GF On-Demand Anodyne EPHX2 43 49 Cc1cc(O)cc(NC(=O)c2cnc(C(C)C)nc2C)c1 ZINC000880872561 CG On-Demand Anodyne JUN 21 48 CCN1CC[C@H](CNC(=O)Nc2c(C)sc(C)c2C(=O)OC)C1 ZINC000880872570 EF On-Demand Anodyne CACNA1I 44 32 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1nccs1 ZINC000880872591 EF On-Demand Anodyne MAP1 43 33 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)Cc1cccc(O)c1 ZINC000880872598 EH On-Demand Anodyne HSD17B2 32 46 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880872726 FD On-Demand Mild PDGFRB 45 40 CCCCN(CCO)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880872799 CE On-Demand Mild INHA 46 36 CCNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880872810 EC On-Demand Mild PDGFRB 45 42 CCNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880872810 EC On-Demand Mild ENPP1 55 33 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC(c2nc(C)no2)CC1 ZINC000880872819 GG On-Demand Anodyne ETHR 42 34 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880872823 FH On-Demand Mild ROCK2 15 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880872823 FH On-Demand Mild MT-ND1 19 41 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880872823 FH On-Demand Mild ENPP1 66 32 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](CCO)c1ccccc1 ZINC000880872862 GG On-Demand Anodyne SOAT1 24 41 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](CCO)c1ccccc1 ZINC000880872863 GG On-Demand Anodyne SOAT1 24 41 C[C@@H](NC(=O)c1ncsc1C1CC1)c1ccns1 ZINC000880872875 CF On-Demand Anodyne MAP1 57 36 C[C@H](NC(=O)c1ncsc1C1CC1)c1ccns1 ZINC000880872876 CF On-Demand Anodyne MAP1 57 36 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)Cc1cccc(C#N)c1 ZINC000880872882 FH On-Demand Mild HSD17B2 21 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2cccs2)C1 ZINC000880872948 FF On-Demand Anodyne PAPA1_CARPA 35 49 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2cccs2)C1 ZINC000880872948 FF On-Demand Anodyne FPR1 43 35 CO[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880872949 BD On-Demand Anodyne JAK3 17 40 CO[C@@H]1C[C@@H](NC(=O)c2cccn3nccc23)C1 ZINC000880872949 BD On-Demand Anodyne TYK2 20 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2cccs2)C1 ZINC000880872950 FF On-Demand Anodyne PAPA1_CARPA 35 49 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(Cc2cccs2)C1 ZINC000880872950 FF On-Demand Anodyne FPR1 43 35 CO[C@@H]1C[C@@H](NC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880872966 CF On-Demand Anodyne NQO2 20 41 CO[C@@H]1C[C@@H](NC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880872966 CF On-Demand Anodyne MTNR1A 22 40 CO[C@@H]1C[C@@H](NC(=O)CC[C@@H]2CCc3ccccc32)C1 ZINC000880872966 CF On-Demand Anodyne MTNR1B 26 40 CO[C@@H]1C[C@@H](NC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880872968 CF On-Demand Anodyne NQO2 20 41 CO[C@@H]1C[C@@H](NC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880872968 CF On-Demand Anodyne MTNR1A 22 40 CO[C@@H]1C[C@@H](NC(=O)CC[C@H]2CCc3ccccc32)C1 ZINC000880872968 CF On-Demand Anodyne MTNR1B 26 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1ccns1 ZINC000880872983 EE On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](C)c1ccns1 ZINC000880872985 EE On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1ccns1 ZINC000880872987 EE On-Demand Anodyne FPR1 48 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)c1ccns1 ZINC000880872989 EE On-Demand Anodyne FPR1 48 38 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccc(OC)cc1 ZINC000880873015 EG On-Demand Anodyne CA9 15 40 COc1ccccc1-c1ccc(C(=O)N[C@@H]2C[C@@H](OC)C2)c(O)n1 ZINC000880873053 EE On-Demand Anodyne HTR3A 19 45 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@H](c4ccc(O)cc4)C3)cc2)N1 ZINC000880873082 FF On-Demand Anodyne L3MBTL3 60 40 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@@H](c4ccc(O)cc4)C3)cc2)N1 ZINC000880873085 FF On-Demand Anodyne L3MBTL3 60 40 O=C1CC[C@@H](c2ccc(C(=O)N3CC[C@@H](c4ccc(O)cc4)C3)cc2)N1 ZINC000880873087 FF On-Demand Anodyne L3MBTL3 60 40 O=C1CC[C@H](c2ccc(C(=O)N3CC[C@H](c4ccc(O)cc4)C3)cc2)N1 ZINC000880873088 FF On-Demand Anodyne L3MBTL3 60 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2c(CC#N)cccc2C1 ZINC000880873097 GF On-Demand Mild PAPA1_CARPA 41 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2c(CC#N)cccc2C1 ZINC000880873097 GF On-Demand Mild CTSL 16 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2c(CC#N)cccc2C1 ZINC000880873099 GF On-Demand Mild PAPA1_CARPA 41 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2c(CC#N)cccc2C1 ZINC000880873099 GF On-Demand Mild CTSL 16 41 O=C(C[C@@H]1CCNC1=O)N[C@H]1CCc2ccc(Cl)cc21 ZINC000880873102 CD On-Demand Anodyne BDKRB1 37 40 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCc2ccc(Cl)cc21 ZINC000880873104 CD On-Demand Anodyne BDKRB1 37 40 O=C(C[C@H]1CCNC1=O)N[C@H]1CCc2ccc(Cl)cc21 ZINC000880873105 CD On-Demand Anodyne BDKRB1 37 40 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880873111 GF On-Demand Mild HTR1B 15 46 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880873111 GF On-Demand Mild PDGFRB 60 46 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880873111 GF On-Demand Mild NPY2R 29 41 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880873111 GF On-Demand Mild EPHX2 19 40 COc1ccc(C(=O)N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880873111 GF On-Demand Mild PDGFRA 20 41 CN(C(=O)COC1CC1)[C@@H](CCc1ccccc1)C(F)F ZINC000880873120 CF On-Demand Anodyne TIMP3 76 36 CN(C(=O)COC1CC1)[C@H](CCc1ccccc1)C(F)F ZINC000880873121 CF On-Demand Anodyne TIMP3 76 36 COC[C@@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873138 CD On-Demand Mild ADRB1 44 33 COC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873139 CD On-Demand Mild ADRB1 44 33 CCOC(=O)CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873140 EF On-Demand Mild P2RY12 20 44 CCOC(=O)CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873140 EF On-Demand Mild PDGFRB 41 43 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild DRD4 16 42 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild HTR4 32 45 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild SSTR5 55 39 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild EPHX2 52 45 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild CXCR3 22 44 CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873146 DE On-Demand Mild MCHR1 26 45 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild HTR1B 16 46 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild P2RY12 52 51 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild PDGFRB 51 48 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild NPY2R 16 43 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild F13A1 25 40 CCOC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873147 ED On-Demand Mild ENPP1 70 34 CC[C@H]1c2ccsc2CCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873313 EI On-Demand Mild TRPM8 17 54 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873315 EI On-Demand Mild TRPM8 17 54 CN(C(=O)c1ccc([C@H]2CCC(=O)N2)cc1)[C@@H](CCc1ccccc1)C(F)F ZINC000880873339 GH On-Demand Anodyne MBTPS1 58 34 CN(C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)[C@@H](CCc1ccccc1)C(F)F ZINC000880873342 GH On-Demand Anodyne MBTPS1 58 34 CN(C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1)[C@H](CCc1ccccc1)C(F)F ZINC000880873343 GH On-Demand Anodyne MBTPS1 58 34 CN(C(=O)c1ccc([C@H]2CCC(=O)N2)cc1)[C@H](CCc1ccccc1)C(F)F ZINC000880873346 GH On-Demand Anodyne MBTPS1 58 34 CCCCNC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873357 FF On-Demand Mild PDGFRB 38 40 Cc1cc(O)cc(NC(=O)c2ncsc2C2CC2)c1 ZINC000880873365 CG On-Demand Anodyne MAP1 51 36 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCc2ccc(Cl)cc21 ZINC000880873383 CD On-Demand Anodyne BDKRB1 37 40 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCn1ccnc1 ZINC000880873439 EF On-Demand Anodyne TBXAS1 44 46 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCn1ccnc1 ZINC000880873439 EF On-Demand Anodyne QPCT 49 55 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCn1ccnc1 ZINC000880873439 EF On-Demand Anodyne NAMPT 22 41 COC(=O)c1c(C)sc(C)c1NC(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000880873454 GG On-Demand Anodyne PANC 46 36 CCOC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873458 EE On-Demand Mild P2RY12 26 45 CCOC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873458 EE On-Demand Mild PDGFRB 37 42 CCOC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873458 EE On-Demand Mild ENPP1 44 30 CCOC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873458 EE On-Demand Mild PTR1 46 33 COC(=O)c1c(C)sc(C)c1NC(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000880873460 GG On-Demand Anodyne PANC 46 36 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@H]1c1cccnc1 ZINC000880873463 FH On-Demand Anodyne CHRNA7 16 44 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCC[C@@H]1c1cccnc1 ZINC000880873466 FH On-Demand Anodyne CHRNA7 16 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cc(OC)ccc1O ZINC000880873471 FG On-Demand Clean MTNR1A 20 42 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cc(OC)ccc1O ZINC000880873471 FG On-Demand Clean MTNR1B 16 42 CO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880873488 CD On-Demand Anodyne GABRA1 19 43 CO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880873488 CD On-Demand Anodyne MPO 42 34 CO[C@@H]1C[C@@H](NC(=O)C(=O)c2c[nH]c3cc(F)ccc23)C1 ZINC000880873488 CD On-Demand Anodyne GABRA2 17 43 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873504 FF On-Demand Mild XDH 18 40 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873504 FF On-Demand Mild P2RY12 17 43 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873504 FF On-Demand Mild PDGFRB 49 43 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880873504 FF On-Demand Mild NPY2R 28 41 CO[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880873515 DF On-Demand Anodyne PDE4D 20 42 CO[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880873515 DF On-Demand Anodyne UTS2R 22 41 CO[C@@H]1C[C@@H](NC(=O)c2ccc(OC(F)F)c(Cl)c2)C1 ZINC000880873515 DF On-Demand Anodyne EZH2 43 40 NC(=O)[C@@H]1CC[C@H](C(=O)N2CCCC3(CC2)CC3)N1Cc1ccccc1 ZINC000880873533 FE On-Demand Anodyne PREP 77 42 O=C(c1cnc2cc[nH]c2c1)N1CCCC2(CC1)CC2 ZINC000880873542 CF On-Demand Anodyne ACACA 33 58 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](c2ccc(O)cc2)C1 ZINC000880873563 GF On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](c2ccc(O)cc2)C1 ZINC000880873563 GF On-Demand Anodyne CCR1 32 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](c2ccc(O)cc2)C1 ZINC000880873565 GF On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](c2ccc(O)cc2)C1 ZINC000880873565 GF On-Demand Anodyne CCR1 32 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](c2ccc(O)cc2)C1 ZINC000880873568 GF On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@H](c2ccc(O)cc2)C1 ZINC000880873568 GF On-Demand Anodyne CCR1 32 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](c2ccc(O)cc2)C1 ZINC000880873571 GF On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC[C@@H](c2ccc(O)cc2)C1 ZINC000880873571 GF On-Demand Anodyne CCR1 32 44 CO[C@@H]1C[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880873598 EC On-Demand Anodyne DRD2 22 42 CO[C@@H]1C[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880873598 EC On-Demand Anodyne DRD3 15 42 CO[C@@H]1C[C@@H](NC(=O)[C@@H]2CC[C@H](C(N)=O)N2Cc2ccccc2)C1 ZINC000880873598 EC On-Demand Anodyne SIGMAR1 20 42 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880873604 GF On-Demand Mild P2RY12 23 47 CCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873611 CF On-Demand Mild ADRB1 48 37 CCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873611 CF On-Demand Mild QPCT 22 47 COC(=O)c1c(C)sc(C)c1NC(=O)N(C)Cc1ccc(Cl)nc1 ZINC000880873637 FH On-Demand Anodyne NACHRBETA2 23 40 CC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873652 BE On-Demand Mild ADRB1 41 32 CC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873652 BE On-Demand Mild XDH 20 40 CC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873652 BE On-Demand Mild ENPP1 54 30 COCCOc1ccc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873663 FF On-Demand Mild ADRB1 45 39 COCCOc1ccc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873663 FF On-Demand Mild TSHR 44 33 COCCOc1ccc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873663 FF On-Demand Mild PDGFRB 16 43 COCCOc1ccc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873663 FF On-Demand Mild ROCK2 24 44 COc1ccc([C@@H]2CCCN2C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873666 FH On-Demand Mild TSHR 47 31 COc1ccc([C@@H]2CCCN2C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880873666 FH On-Demand Mild PFKFB3 49 33 CN(C(=O)c1nnn(C)n1)[C@H](CCc1ccccc1)C(F)F ZINC000880873731 DD On-Demand Anodyne DAGLA 19 40 CN(C(=O)c1nnn(C)n1)[C@@H](CCc1ccccc1)C(F)F ZINC000880873732 DD On-Demand Anodyne DAGLA 19 40 Cc1cnc(Cl)c(C(=O)N2CC[C@@H](c3ccc(O)cc3)C2)c1 ZINC000880873771 DG On-Demand Anodyne FASN 41 35 Cc1cnc(Cl)c(C(=O)N2CC[C@H](c3ccc(O)cc3)C2)c1 ZINC000880873772 DG On-Demand Anodyne FASN 41 35 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ccccn2)CC1 ZINC000880873813 FF On-Demand Anodyne DRD4 22 40 CCOC(=O)N1CCC(NC(=O)Nc2c(C)sc(C)c2C(=O)OC)CC1 ZINC000880873851 GF On-Demand Anodyne EPHX2 44 42 O=C(CN1CCCCS1(=O)=O)NCCc1c[nH]c2cc(F)c(Cl)cc12 ZINC000880873872 GE On-Demand Anodyne MPO 50 36 COCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873907 CD On-Demand Mild ADRB1 49 37 COCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873907 CD On-Demand Mild QPCT 22 47 COCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873911 CE On-Demand Mild ADRB1 48 37 COCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880873911 CE On-Demand Mild QPCT 21 47 NC(=O)c1cc(-c2csc(NC(=O)c3ccccc3NC(=O)c3ccccc3)n2)c[nH]1 ZINC000880873956 IH On-Demand Anodyne MPL 59 39 NC(=O)c1cc(-c2csc(NC(=O)c3ccccc3NC(=O)c3ccccc3)n2)c[nH]1 ZINC000880873956 IH On-Demand Anodyne ROCK1 20 40 NC(=O)c1cc(-c2csc(NC(=O)c3ccccc3NC(=O)c3ccccc3)n2)c[nH]1 ZINC000880873956 IH On-Demand Anodyne ROCK2 17 40 O=C(Cc1csc([C@@H]2CCS(=O)(=O)C2)n1)N1CC(Cc2cccs2)C1 ZINC000880873970 GE On-Demand Anodyne ETHR 34 41 O=C(Cc1csc([C@H]2CCS(=O)(=O)C2)n1)N1CC(Cc2cccs2)C1 ZINC000880873971 GE On-Demand Anodyne ETHR 34 41 CCN(CC)C(=O)CN1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880874035 GD On-Demand Mild PDGFRB 40 40 CC[C@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874098 CG On-Demand Mild QRFPR 43 37 CC[C@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874098 CG On-Demand Mild ACKR3 46 31 CC[C@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874098 CG On-Demand Mild PFKFB3 59 33 CC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874100 CG On-Demand Mild QRFPR 43 37 CC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874100 CG On-Demand Mild ACKR3 46 31 CC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874100 CG On-Demand Mild PFKFB3 59 33 CC(C)(C)OC(=O)N1C[C@@H](C(=O)N2CC[C@@H]3CC[C@@H](O)[C@@H]32)C(C)(C)C1 ZINC000880874110 FE On-Demand Anodyne GPR119 21 41 Cn1nccc1C(NC(=O)COC1CC1)c1ccnn1C ZINC000880874111 CC On-Demand Anodyne TIMP3 57 32 CC(C)(C)OC(=O)N1C[C@H](C(=O)N2CC[C@@H]3CC[C@@H](O)[C@@H]32)C(C)(C)C1 ZINC000880874112 FE On-Demand Anodyne GPR119 21 41 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880874153 EE On-Demand Mild P2RY12 22 41 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880874153 EE On-Demand Mild FDFT1 15 41 CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880874170 CG On-Demand Mild PDGFRB 48 42 CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880874171 CG On-Demand Mild PDGFRB 48 42 O=C(N[C@H]1CCc2ccc(Cl)cc21)c1ccc(CN2CCOCC2)o1 ZINC000880874175 FG On-Demand Anodyne HTR2A 21 40 O=C(N[C@@H]1CCc2ccc(Cl)cc21)c1ccc(CN2CCOCC2)o1 ZINC000880874178 FG On-Demand Anodyne HTR2A 21 40 O=C(N1CC[C@@H](c2ccc(O)cc2)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880874180 EH On-Demand Anodyne ADAM10 16 40 O=C(N1CC[C@H](c2ccc(O)cc2)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880874181 EH On-Demand Anodyne ADAM10 16 40 CCCN(CCC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874242 CG On-Demand Mild ENPP1 59 31 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(NC(C)=O)c1 ZINC000880874302 GG On-Demand Anodyne ROCK2 24 48 Cc1noc(C)c1COc1ccc(CC(=O)Nc2ccc(CS(N)(=O)=O)cc2)cc1 ZINC000880874331 IF On-Demand Anodyne CA2 17 47 Cc1noc(C)c1COc1ccc(CC(=O)Nc2ccc(CS(N)(=O)=O)cc2)cc1 ZINC000880874331 IF On-Demand Anodyne CA12 22 47 Cc1noc(C)c1COc1ccc(CC(=O)Nc2ccc(CS(N)(=O)=O)cc2)cc1 ZINC000880874331 IF On-Demand Anodyne CA9 25 47 Cc1noc(C)c1COc1ccc(CC(=O)Nc2ccc(CS(N)(=O)=O)cc2)cc1 ZINC000880874331 IF On-Demand Anodyne RORC 25 49 COC(=O)c1c(C)sc(C)c1NC(=O)NCCc1cccnc1 ZINC000880874345 EF On-Demand Anodyne NAMPT 35 43 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880874405 GF On-Demand Anodyne ADRB2 43 45 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880874405 GF On-Demand Anodyne ADRB1 66 46 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880874405 GF On-Demand Anodyne ADRB3 38 46 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880874406 GF On-Demand Anodyne ADRB2 43 45 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880874406 GF On-Demand Anodyne ADRB1 66 46 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880874406 GF On-Demand Anodyne ADRB3 38 46 O=C(c1csc(-c2ncc[nH]2)n1)N1CC[C@@H]2CC[C@@H](O)[C@@H]21 ZINC000880874408 DD On-Demand Anodyne TRPC3 42 34 O=C(COC1CC1)NCCc1c[nH]c2cc(F)c(Cl)cc12 ZINC000880874423 DF On-Demand Anodyne MPO 45 36 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(c2ccc(C#N)cn2)CC1 ZINC000880874424 GF On-Demand Mild PDGFRB 20 42 Cc1cc(O)cc(NC(=O)Cc2ccccc2N2CCCC2=O)c1 ZINC000880874430 DG On-Demand Anodyne KCNQ2 58 38 CCCCN(CC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874470 CG On-Demand Mild INHA 47 37 CCOCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874471 CE On-Demand Mild ADRB1 47 36 O=C(COC1CC1)N[C@@H]1CCc2ccc(Cl)cc21 ZINC000880874501 CF On-Demand Anodyne PYGL 40 36 O=C(COC1CC1)N[C@H]1CCc2ccc(Cl)cc21 ZINC000880874502 CF On-Demand Anodyne PYGL 40 36 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccnc1 ZINC000880874569 DF On-Demand Anodyne ROCK2 18 40 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccnc1 ZINC000880874569 DF On-Demand Anodyne NAMPT 67 50 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000880874574 GG On-Demand Anodyne ROCK2 24 40 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1ccc(O)c(OC)c1 ZINC000880874624 FG On-Demand Anodyne TRPV1 16 47 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@H]1CCN(CC(F)(F)F)C1 ZINC000880874644 GG On-Demand Anodyne CACNA1I 48 34 COC(=O)c1c(C)sc(C)c1NC(=O)NC[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880874645 GG On-Demand Anodyne CACNA1I 48 34 Cc1cc(O)cc(NC(=O)C2CCC(S(C)(=O)=O)CC2)c1 ZINC000880874659 DE On-Demand Anodyne EPHX2 18 42 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880874778 GF On-Demand Anodyne FAAH 22 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCCCN1CCOCC1 ZINC000880874779 FD On-Demand Anodyne EPHX2 21 46 COC(=O)c1c(C)sc(C)c1NC(=O)N1CCc2ccccc2C1 ZINC000880874784 EH On-Demand Anodyne NOD2 40 35 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(OC)c1 ZINC000880874793 EG On-Demand Anodyne DRD4 41 33 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(OC)c1 ZINC000880874793 EG On-Demand Anodyne ROCK1 40 49 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(OC)c1 ZINC000880874793 EG On-Demand Anodyne MTNR1A 33 41 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(OC)c1 ZINC000880874793 EG On-Demand Anodyne MTNR1B 35 41 COC(=O)c1c(C)sc(C)c1NC(=O)NCc1cccc(OC)c1 ZINC000880874793 EG On-Demand Anodyne ROCK2 52 52 O=C1CC[C@@H](c2ccc(C(=O)N3CCCC4(CC3)CC4)cc2)N1 ZINC000880874815 DG On-Demand Anodyne L3MBTL3 60 43 O=C1CC[C@H](c2ccc(C(=O)N3CCCC4(CC3)CC4)cc2)N1 ZINC000880874816 DG On-Demand Anodyne L3MBTL3 60 43 C[C@@H](CN(C)C(=O)COC1CC1)NC(=O)OC(C)(C)C ZINC000880874839 CD On-Demand Anodyne ECE1 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](OC)C1)C2 ZINC000880874853 CE On-Demand Anodyne NQO2 25 41 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1C[C@@H](OC)C1)C2 ZINC000880874853 CE On-Demand Anodyne MTNR1A 36 45 CCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874857 BE On-Demand Mild ADRB1 48 38 CCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874857 BE On-Demand Mild QPCT 22 48 CCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880874857 BE On-Demand Mild ENPP1 54 30 C[C@@H](CN(C)C(=O)Cc1ccccc1N1CCCC1=O)NC(=O)OC(C)(C)C ZINC000880874859 GF On-Demand Anodyne CCKAR 22 40 C[C@@H](CN(C)C(=O)Cc1ccccc1N1CCCC1=O)NC(=O)OC(C)(C)C ZINC000880874859 GF On-Demand Anodyne FPR1 44 34 Cn1ncc(Br)c1CC(=O)N[C@@H]1CCc2ccc(Cl)cc21 ZINC000880874876 FG On-Demand Anodyne P2RX7 20 42 Cn1ncc(Br)c1CC(=O)N[C@H]1CCc2ccc(Cl)cc21 ZINC000880874877 FG On-Demand Anodyne P2RX7 20 42 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCCC1 ZINC000880874914 CG On-Demand Anodyne EPHX2 24 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](OC)C1 ZINC000880874943 DD On-Demand Anodyne PAPA1_CARPA 36 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1C[C@@H](OC)C1 ZINC000880874944 DD On-Demand Anodyne PAPA1_CARPA 36 44 COC(=O)c1c(C)sc(C)c1NC(=O)NCCN1CCOCC1 ZINC000880874962 ED On-Demand Anodyne EPHX2 16 41 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@@H](c3ccc(O)cc3)C2)N1Cc1ccccc1 ZINC000880874963 GE On-Demand Anodyne PREP 54 39 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC[C@H](c3ccc(O)cc3)C2)N1Cc1ccccc1 ZINC000880874964 GE On-Demand Anodyne PREP 54 39 COC(=O)c1c(C)sc(C)c1NC(=O)NCCn1ccnc1 ZINC000880874969 DE On-Demand Anodyne QPCT 36 48 Cc1nc(C(C)C)ncc1C(=O)N1CC[C@H](c2ccc(O)cc2)C1 ZINC000880874975 EG On-Demand Anodyne FASN 40 35 Cc1nc(C(C)C)ncc1C(=O)N1CC[C@@H](c2ccc(O)cc2)C1 ZINC000880874976 EG On-Demand Anodyne FASN 40 35 C=CC(C)(C)CC(=O)N(C)C[C@@H](C)NC(=O)OC(C)(C)C ZINC000880874982 CF On-Demand Mild CTSK 15 43 C=CC(C)(C)CC(=O)N(C)C[C@H](C)NC(=O)OC(C)(C)C ZINC000880874983 CF On-Demand Mild CTSK 15 43 COc1ccc([C@@H]2CCN(C(=O)c3ccc([C@H]4CCC(=O)N4)cc3)C2)cc1F ZINC000880874985 GG On-Demand Anodyne L3MBTL3 42 34 COc1ccc([C@@H]2CCN(C(=O)c3ccc([C@@H]4CCC(=O)N4)cc3)C2)cc1F ZINC000880874986 GG On-Demand Anodyne L3MBTL3 42 34 COC(=O)c1c(C)sc(C)c1NC(=O)NC1CCN(C(C)=O)CC1 ZINC000880875012 FE On-Demand Anodyne EPHX2 43 47 CC(=O)N(CC(=O)N(C)C[C@H](C)NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880875020 FE On-Demand Anodyne FPR1 46 36 CC(=O)N(CC(=O)N(C)C[C@@H](C)NC(=O)OC(C)(C)C)c1ccccc1 ZINC000880875021 FE On-Demand Anodyne FPR1 46 36 COc1ccc(N2CCC(NC(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875027 GG On-Demand Mild EPHX2 50 41 COc1ccc(N2CCC(NC(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875027 GG On-Demand Mild PDGFRA 20 40 COc1ccc(N2CCC(NC(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875027 GG On-Demand Mild MCHR1 18 41 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875032 FG On-Demand Mild NPY2R 15 40 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875032 FG On-Demand Mild EPHX2 54 49 CCOCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875033 CD On-Demand Mild ADRB1 48 37 O=C(/C=C\c1cccnc1)NCc1ccc(C(=O)N2CCOCC2)cc1 ZINC000880875078 FD On-Demand Anodyne NAMPT 69 55 CCOCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875099 CF On-Demand Mild ADRB1 46 35 COc1cccc([C@H](O)C2CCN(C(=O)[C@@H]3C[C@]3(C)c3ccccc3)CC2)c1 ZINC000880875101 GH On-Demand Anodyne NPY1R 17 49 CCN(Cc1ccc(OC)cc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875113 EH On-Demand Mild ROCK2 17 44 CCN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875122 BE On-Demand Mild ENPP1 60 31 CCN(CC)C(=O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875127 DD On-Demand Mild ADRB1 42 32 CCN(CC)C(=O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875127 DD On-Demand Mild ENPP1 61 33 CC(C)(C)OC(=O)N1CC[C@H](OCC2CCN(C(=O)COC3CC3)CC2)C1 ZINC000880875132 GE On-Demand Anodyne GPR119 39 54 CC(C)(C)OC(=O)N1CC[C@@H](OCC2CCN(C(=O)COC3CC3)CC2)C1 ZINC000880875133 GE On-Demand Anodyne GPR119 39 54 O=C1OC[C@H]2CN(C(=O)[C@H]3C[C@@H](F)CN3C(=O)OCc3ccccc3)C[C@@H]12 ZINC000880875151 GD On-Demand Anodyne PREP 36 44 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild DRD2 22 40 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild HTR2A 39 41 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild DRD3 20 40 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild HTR4 57 40 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild SSTR5 41 37 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild CCR3 44 38 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild EPHX2 53 44 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild CXCR3 21 43 COCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875152 ED On-Demand Mild MCHR1 28 43 COCCN(Cc1ccccn1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875173 EF On-Demand Mild GRM4 27 42 CCO[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875180 DF On-Demand Mild P2RY12 15 40 COc1cccc([C@H](O)C2CCN(C(=O)c3cnc4cc[nH]c4c3)CC2)c1 ZINC000880875202 FG On-Demand Anodyne HPGD 21 40 CC[C@@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875205 CD On-Demand Mild ADRB1 41 32 COc1cccc([C@H](O)C2CCN(C(=O)[C@H]3CCc4nncn4CC3)CC2)c1 ZINC000880875234 GE On-Demand Anodyne DRD4 40 30 COc1cccc([C@H](O)C2CCN(C(=O)[C@@H]3CCc4nncn4CC3)CC2)c1 ZINC000880875235 GE On-Demand Anodyne DRD4 40 30 COc1ccc(N2CCCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875243 GG On-Demand Mild HTR1D 15 52 COc1ccc(N2CCCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875243 GG On-Demand Mild HTR1B 21 52 COc1ccc(N2CCCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875243 GG On-Demand Mild P2RY12 15 47 COc1ccc(N2CCCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875243 GG On-Demand Mild PDGFRB 61 45 COc1cccc([C@H](O)C2CCN(C(=O)CN(C(C)=O)c3ccccc3)CC2)c1 ZINC000880875253 GG On-Demand Anodyne OPRD1 18 42 COc1cccc([C@H](O)C2CCN(C(=O)CN(C(C)=O)c3ccccc3)CC2)c1 ZINC000880875253 GG On-Demand Anodyne MTNR1A 17 40 COc1cccc([C@H](O)C2CCN(C(=O)CN(C(C)=O)c3ccccc3)CC2)c1 ZINC000880875253 GG On-Demand Anodyne MTNR1B 30 40 COCC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875265 EC On-Demand Mild HTR1B 16 46 COCC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875265 EC On-Demand Mild PDGFRB 50 45 COCC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875265 EC On-Demand Mild ENPP1 50 32 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875275 FF On-Demand Mild P2RY12 19 44 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875275 FF On-Demand Mild PDGFRB 31 41 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875293 EE On-Demand Mild P2RY12 41 49 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875293 EE On-Demand Mild PDGFRB 48 46 CCOC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875293 EE On-Demand Mild ENPP1 67 32 COc1cccc([C@H](O)C2CCN(C(=O)c3ccc4c(O)ncnc4c3)CC2)c1 ZINC000880875312 GF On-Demand Anodyne HPGD 47 46 COc1cccc([C@H](O)C2CCN(C(=O)[C@@]3(c4ccccc4)C[C@H](F)C3)CC2)c1 ZINC000880875315 GI On-Demand Anodyne NPY1R 15 49 CCC(=O)N1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875317 EE On-Demand Mild PDGFRB 49 43 COCCN(Cc1ccccc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875344 EG On-Demand Mild ROCK2 16 47 COc1cccc([C@H](O)C2CCN(C(=O)C[C@H]3CCNC3=O)CC2)c1 ZINC000880875373 ED On-Demand Anodyne C3AR1 36 40 COc1cccc([C@H](O)C2CCN(C(=O)C[C@@H]3CCNC3=O)CC2)c1 ZINC000880875374 ED On-Demand Anodyne C3AR1 36 40 COc1ccc([C@@H]2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)C2)cc1 ZINC000880875390 FH On-Demand Mild MCHR1 17 50 COc1ccc([C@@H]2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)C2)cc1 ZINC000880875390 FH On-Demand Mild PFKFB3 41 31 COC[C@@H](C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875408 CD On-Demand Mild ADRB1 50 38 COC[C@H](C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875409 CD On-Demand Mild ADRB1 50 38 COc1cccc([C@H](O)C2CCN(C(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880875438 GG On-Demand Anodyne TRPC6 31 40 COc1cccc([C@H](O)C2CCN(C(=O)c3csc(-c4ncc[nH]4)n3)CC2)c1 ZINC000880875438 GG On-Demand Anodyne TRPC3 22 40 COc1ccc2c(c1)CN(C(=O)Nc1ccc(OC)c(C#N)c1)CC2 ZINC000880875459 EG On-Demand Mild HDAC6 28 43 COc1ccc2c(c1)CN(C(=O)Nc1ccc(OC)c(C#N)c1)CC2 ZINC000880875459 EG On-Demand Mild ABCB1 17 42 COc1ccc2c(c1)CN(C(=O)Nc1ccc(OC)c(C#N)c1)CC2 ZINC000880875459 EG On-Demand Mild AKR1C3 19 41 COC(=O)[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875460 DD On-Demand Mild PDGFRB 29 40 COC(=O)[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875461 DD On-Demand Mild PDGFRB 29 40 CCN1CCC[C@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875521 DE On-Demand Mild CCR3 41 38 CCN1CCC[C@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875521 DE On-Demand Mild EPHX2 40 40 CCN1CCC[C@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875521 DE On-Demand Mild MCHR1 17 41 CCN1CCC[C@@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875522 DE On-Demand Mild CCR3 41 38 CCN1CCC[C@@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875522 DE On-Demand Mild EPHX2 40 40 CCN1CCC[C@@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875522 DE On-Demand Mild MCHR1 17 41 COc1cccc([C@H](O)C2CCN(C(=O)c3cc(C(F)F)[nH]n3)CC2)c1 ZINC000880875546 FF On-Demand Anodyne GRIN2B 15 46 COCCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875567 CF On-Demand Mild ADRB1 47 36 COCCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875567 CF On-Demand Mild QPCT 16 46 COc1ccc(OC2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875575 GH On-Demand Mild PDGFRB 46 40 COc1ccc(OC2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875575 GH On-Demand Mild PRSS2 56 32 COc1ccc(OC2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875575 GH On-Demand Mild EPHX2 32 48 COc1ccc(OC2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880875575 GH On-Demand Mild PFKFB3 54 33 CCN1CC[C@H](CNC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875587 DE On-Demand Mild CCR3 63 40 CCN1CC[C@H](CNC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875587 DE On-Demand Mild MCHR1 17 40 CCN1CC[C@H](CNC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880875587 DE On-Demand Mild CACNA1I 66 35 CCc1nc(CN2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cs1 ZINC000880875591 GF On-Demand Mild PDGFRB 53 43 C=CCSCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875595 CF On-Demand Mild ADRB1 44 34 C=CC(C)(C)CC(=O)N1CCC(CO[C@@H]2CCN(C(=O)OC(C)(C)C)C2)CC1 ZINC000880875602 GH On-Demand Mild GPR119 34 48 C=CC(C)(C)CC(=O)N1CCC(CO[C@H]2CCN(C(=O)OC(C)(C)C)C2)CC1 ZINC000880875603 GH On-Demand Mild GPR119 34 48 COCC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875617 CE On-Demand Mild ADRB1 41 31 COCC[C@@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875618 CE On-Demand Mild ADRB1 41 31 CCCOc1ncccc1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875633 EG On-Demand Mild ADRB1 43 33 CCCOc1ncccc1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875633 EG On-Demand Mild ENPP1 40 35 COc1cccc([C@H](O)C2CCN(C(=O)c3cc(C)cnc3Cl)CC2)c1 ZINC000880875642 FH On-Demand Anodyne DRD4 42 32 CCN(CC)C(=O)CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875651 EE On-Demand Mild ADRB1 45 34 CCN(CC)C(=O)CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875651 EE On-Demand Mild QPCT 19 45 COCCN(CCOC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875670 DD On-Demand Mild ENPP1 49 30 CC[C@H](C)N(C)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875698 DE On-Demand Mild ADRB1 47 37 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCC12CC2 ZINC000880875699 EF On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCC12CC2 ZINC000880875700 EF On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1CCCC12CC2 ZINC000880875701 EF On-Demand Anodyne PAPA1_CARPA 37 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@H]1CCCC12CC2 ZINC000880875702 EF On-Demand Anodyne PAPA1_CARPA 37 45 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2C[C@H](OC)C2)c(O)n1 ZINC000880875703 EF On-Demand Anodyne KCNA3 40 35 COC(=O)c1cc(-c2csc(NC(=O)C/N=C3/NS(=O)(=O)c4ccccc43)n2)c[nH]1 ZINC000880875725 ID On-Demand Mild GABRA1 20 40 CCc1nc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cs1 ZINC000880875752 DF On-Demand Mild ADRB1 44 33 CCc1nc(CNC(=O)Nc2ccc(OC)c(C#N)c2)cs1 ZINC000880875752 DF On-Demand Mild ENPP1 64 32 CNC(=O)CCN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875758 CD On-Demand Mild ENPP1 59 32 C#CC[C@@H](CCOC)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880875802 ED On-Demand Mild KCNQ2 50 33 C#CC[C@H](CCOC)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880875803 ED On-Demand Mild KCNQ2 50 33 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCC23CC3)c(O)n1 ZINC000880875834 FH On-Demand Anodyne KCNA3 46 38 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCC23CC3)c(O)n1 ZINC000880875834 FH On-Demand Anodyne HCN1 57 37 COc1ccccc1-c1ccc(C(=O)NC[C@@H]2CCCC23CC3)c(O)n1 ZINC000880875834 FH On-Demand Anodyne HCN4 50 37 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCC23CC3)c(O)n1 ZINC000880875835 FH On-Demand Anodyne KCNA3 46 38 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCC23CC3)c(O)n1 ZINC000880875835 FH On-Demand Anodyne HCN1 57 37 COc1ccccc1-c1ccc(C(=O)NC[C@H]2CCCC23CC3)c(O)n1 ZINC000880875835 FH On-Demand Anodyne HCN4 50 37 O=C(NCC[C@@H](O)COCc1ccccc1)c1coc(-c2ccccn2)n1 ZINC000880875838 FE On-Demand Anodyne TBXA2R 16 42 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](O)COCc1ccccc1)C2 ZINC000880875860 GF On-Demand Anodyne MTNR1A 45 42 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](O)COCc1ccccc1)C2 ZINC000880875860 GF On-Demand Anodyne MTNR1B 44 42 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H](O)COCc1ccccc1)C2 ZINC000880875860 GF On-Demand Anodyne GHSR 18 40 CS(=O)(=O)C1CCC(C(=O)NCC[C@@H](O)COCc2ccccc2)CC1 ZINC000880875888 GD On-Demand Anodyne CAPN2 40 37 O=C(NCc1ccccc1CC(F)(F)F)[C@@H]1CCc2nncn2CC1 ZINC000880875897 FF On-Demand Anodyne P2RX7 41 38 O=C(NCc1ccccc1CC(F)(F)F)[C@@H]1CCc2nncn2CC1 ZINC000880875897 FF On-Demand Anodyne EPHX2 17 45 O=C(NCc1ccccc1CC(F)(F)F)[C@H]1CCc2nncn2CC1 ZINC000880875898 FF On-Demand Anodyne P2RX7 41 38 O=C(NCc1ccccc1CC(F)(F)F)[C@H]1CCc2nncn2CC1 ZINC000880875898 FF On-Demand Anodyne EPHX2 17 45 CCC(CC)[C@@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875901 DE On-Demand Mild ADRB1 49 38 CCC(CC)[C@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875902 DE On-Demand Mild ADRB1 49 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](OC)C1 ZINC000880875908 ED On-Demand Anodyne PAPA1_CARPA 39 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC[C@@H]1C[C@H](OC)C1 ZINC000880875909 ED On-Demand Anodyne PAPA1_CARPA 39 48 CCC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875931 CD On-Demand Mild ADRB1 51 40 CCC[C@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875932 CD On-Demand Mild ADRB1 51 40 CCC[C@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880875945 CE On-Demand Mild ADRB1 40 32 COCCOc1ccc(NC(=O)Nc2ccc(OC)c(C#N)c2)c(C)c1 ZINC000880875947 FH On-Demand Mild KDR 24 45 COCCOc1ccc(NC(=O)Nc2ccc(OC)c(C#N)c2)c(C)c1 ZINC000880875947 FH On-Demand Mild PDGFRA 46 39 CS(=O)(=O)C1CCC(C(=O)NCc2ccccc2CC(F)(F)F)CC1 ZINC000880875976 GG On-Demand Anodyne EPHX2 17 42 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875995 DD On-Demand Mild XDH 15 41 COC(=O)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880875995 DD On-Demand Mild PDGFRB 38 43 CCN(CCNC(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880876002 DE On-Demand Mild ADRB1 43 33 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild HTR1A 20 45 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild DRD2 19 40 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild HTR1D 15 45 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild HTR1B 17 45 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild DRD3 25 40 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild P2RY12 15 43 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild PDGFRB 57 47 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876025 ED On-Demand Mild SLC9A1 56 31 CC[C@@H](C)[C@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876030 DE On-Demand Mild ADRB1 42 32 CC[C@@H](C)[C@@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876031 DE On-Demand Mild ADRB1 42 32 CC[C@H](C)[C@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876032 DE On-Demand Mild ADRB1 42 32 CC[C@H](C)[C@@](C)(O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876033 DE On-Demand Mild ADRB1 42 32 COCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876038 DE On-Demand Mild AR 17 40 COCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876038 DE On-Demand Mild PDGFRB 48 44 COCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876038 DE On-Demand Mild EPHX2 15 41 C#CC[C@H](COC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876059 DD On-Demand Mild MPO 60 35 C#CC[C@@H](COC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876060 DD On-Demand Mild MPO 60 35 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](OC)C1)C2 ZINC000880876065 DE On-Demand Anodyne NQO2 36 43 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](OC)C1)C2 ZINC000880876065 DE On-Demand Anodyne MTNR1A 60 48 COc1ccc2c(c1)CC[C@H](C(=O)NC[C@@H]1C[C@H](OC)C1)C2 ZINC000880876065 DE On-Demand Anodyne MTNR1B 52 42 C#CC[C@H](CCOC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876083 DE On-Demand Mild GABRA1 15 40 C#CC[C@H](CCOC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876083 DE On-Demand Mild MPO 56 34 C#CC[C@@H](CCOC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876084 DE On-Demand Mild GABRA1 15 40 C#CC[C@@H](CCOC)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880876084 DE On-Demand Mild MPO 56 34 C=CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876085 CF On-Demand Mild PDGFRB 33 41 C=CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876088 DE On-Demand Mild EPHX2 45 40 C=CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876088 DE On-Demand Mild CXCR3 20 42 C=CCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876088 DE On-Demand Mild MCHR1 16 43 O=C(NC[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880876113 CF On-Demand Anodyne JAK3 19 40 O=C(NC[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880876113 CF On-Demand Anodyne JAK1 15 40 O=C(NC[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880876113 CF On-Demand Anodyne TYK2 22 40 O=C(NC[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880876113 CF On-Demand Anodyne HCN4 40 30 C=C(C)CN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876137 EF On-Demand Mild DRD4 15 40 C=C(C)CN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876137 EF On-Demand Mild EPHX2 45 41 C=C(C)CN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876137 EF On-Demand Mild CXCR3 20 42 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(OC)c(C#N)c1)CC2 ZINC000880876140 EE On-Demand Mild PDGFRB 30 40 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876167 GF On-Demand Mild BMP1 57 38 CCCCN(CCOC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876213 DF On-Demand Mild INHA 40 36 CCC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccccn1 ZINC000880876256 DH On-Demand Mild ADRB1 42 32 CCC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccccn1 ZINC000880876256 DH On-Demand Mild GRM4 15 43 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880876267 DE On-Demand Mild PDGFRB 49 43 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880876267 DE On-Demand Mild CCR3 18 46 CCOC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880876270 DF On-Demand Mild PDGFRB 45 41 COc1ccnc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880876271 FE On-Demand Mild HTR1B 16 49 COc1ccnc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880876271 FE On-Demand Mild P2RY12 16 46 COc1ccnc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880876271 FE On-Demand Mild PDGFRB 68 49 COc1ccnc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880876271 FE On-Demand Mild PDGFRA 29 42 CCCC[C@@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876287 DF On-Demand Mild ADRB1 41 32 CCCC[C@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876288 DF On-Demand Mild ADRB1 41 32 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)CCN1CCOC ZINC000880876291 EE On-Demand Mild PDGFRB 42 41 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cccc2nsnc12 ZINC000880876314 DD On-Demand Anodyne HCRTR1 42 47 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cccc2nsnc12 ZINC000880876314 DD On-Demand Anodyne HCRTR2 21 47 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880876324 ED On-Demand Anodyne HCRTR1 29 48 C=CCNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876327 FD On-Demand Mild PDGFRB 45 41 CC(=O)NC[C@@H]1CCCCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880876346 ED On-Demand Anodyne TRPC6 20 40 CC(=O)NC[C@@H]1CCCCN1C(=O)c1csc(-c2ncc[nH]2)n1 ZINC000880876346 ED On-Demand Anodyne TRPC3 22 40 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild DRD2 26 40 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild DRD4 25 40 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild DRD3 26 40 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild HTR4 67 46 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild SSTR5 40 37 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild CCR3 48 39 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild EPHX2 58 45 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild CXCR3 20 42 CCCCN1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876357 EF On-Demand Mild MCHR1 29 42 C#CC[C@@H](COC)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880876375 CF On-Demand Mild NQO2 20 40 C#CC[C@@H](COC)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880876376 CF On-Demand Mild NQO2 20 40 COCCN(Cc1cccnc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876380 EF On-Demand Mild PTAFR 21 41 COCCN(Cc1cccnc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876380 EF On-Demand Mild ROCK2 20 40 C#CC[C@H](CCOC)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880876422 EG On-Demand Mild PDE4D 15 40 C#CC[C@@H](CCOC)NC(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880876423 EG On-Demand Mild PDE4D 15 40 CCN1CCC[C@H]1CN(Cc1ccncc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876432 GG On-Demand Mild PDE4A 20 44 CCN1CCC[C@H]1CN(Cc1ccncc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876432 GG On-Demand Mild ACKR3 55 31 CCN1CCC[C@@H]1CN(Cc1ccncc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876433 GG On-Demand Mild PDE4A 20 44 CCN1CCC[C@@H]1CN(Cc1ccncc1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876433 GG On-Demand Mild ACKR3 55 31 Cn1ncc(Br)c1CC(=O)NCc1ccccc1CC(F)(F)F ZINC000880876443 GG On-Demand Anodyne P2RX7 34 54 C#CC[C@@H](CCOC)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880876446 EF On-Demand Mild PDK1 42 31 C#CC[C@H](CCOC)NC(=O)c1cc(-c2ccc(OC)cc2)on1 ZINC000880876447 EF On-Demand Mild PDK1 42 31 C#CC[C@@H](COC)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880876455 DD On-Demand Mild NQO2 26 40 C#CC[C@@H](COC)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880876456 DD On-Demand Mild NQO2 26 40 C#CC[C@H](COC)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880876457 DD On-Demand Mild NQO2 26 40 C#CC[C@H](COC)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880876458 DD On-Demand Mild NQO2 26 40 C#CC[C@H](COC)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880876477 CF On-Demand Mild NQO2 20 40 C#CC[C@H](COC)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880876478 CF On-Demand Mild NQO2 20 40 CC[C@@H](O)CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876479 CE On-Demand Mild ADRB1 54 43 CC[C@H](O)CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876480 CE On-Demand Mild ADRB1 54 43 CN(CCNC(=O)C(=O)c1c[nH]c2cc(F)ccc12)CC(F)F ZINC000880876491 ED On-Demand Anodyne MPO 57 36 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc(C)cnc1Cl ZINC000880876500 DE On-Demand Anodyne HCRTR1 35 44 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc(C)cnc1Cl ZINC000880876500 DE On-Demand Anodyne HCRTR2 18 44 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880876574 FG On-Demand Anodyne HRH3 16 42 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880876574 FG On-Demand Anodyne ACACB 19 42 O=C(C[C@H]1CCNC1=O)N[C@@H]1CCCc2ccc(Cl)cc21 ZINC000880876579 DE On-Demand Anodyne BDKRB1 44 46 O=C(C[C@@H]1CCNC1=O)N[C@@H]1CCCc2ccc(Cl)cc21 ZINC000880876581 DE On-Demand Anodyne BDKRB1 44 46 O=C(COC1CC1)NCC[C@@H](O)COCc1ccccc1 ZINC000880876591 CD On-Demand Anodyne CTSK 15 40 O=C(COC1CC1)NCC[C@@H](O)COCc1ccccc1 ZINC000880876591 CD On-Demand Anodyne TIMP3 51 34 CCc1nnc2n1CCN(C(=O)Nc1ccc(OC)c(C#N)c1)C2 ZINC000880876604 ED On-Demand Mild ENPP1 64 32 CCCCCN(CCO)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876605 DF On-Demand Mild INHA 58 38 CC[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876683 CF On-Demand Mild DPP4 23 40 CC[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876683 CF On-Demand Mild QRFPR 42 35 CC[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876683 CF On-Demand Mild ACKR3 64 33 CC[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876683 CF On-Demand Mild PFKFB3 60 34 CC[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876684 CF On-Demand Mild DPP4 23 40 CC[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876684 CF On-Demand Mild QRFPR 42 35 CC[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876684 CF On-Demand Mild ACKR3 64 33 CC[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876684 CF On-Demand Mild PFKFB3 60 34 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876735 FD On-Demand Mild PDGFRB 43 39 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876735 FD On-Demand Mild ABCB1 34 46 CCSCC[C@@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876791 DG On-Demand Mild ENPP1 66 32 CCSCC[C@H](C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880876792 DG On-Demand Mild ENPP1 66 32 COCCCOC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880876801 EF On-Demand Mild PDGFRB 44 43 O=C(COC1CC1)N[C@@H]1CCCc2ccc(Cl)cc21 ZINC000880876838 CG On-Demand Anodyne BDKRB1 49 37 O=C(COC1CC1)N[C@@H]1CCCc2ccc(Cl)cc21 ZINC000880876838 CG On-Demand Anodyne KCNN3 15 46 CN(CCNC(=O)c1cccn2nccc12)CC(F)F ZINC000880876840 CD On-Demand Anodyne POLR1A 43 37 CCc1cnc(CNC(=O)Nc2ccc(OC)c(C#N)c2)s1 ZINC000880876856 DF On-Demand Mild ADRB1 44 35 CCN(CCNC(=O)Nc1ccc(OC)c(C#N)c1)C(C)C ZINC000880876861 DE On-Demand Mild ADRB1 47 38 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@@H]1C ZINC000880876897 EE On-Demand Mild PDGFRB 40 41 CCOCCN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@H]1C ZINC000880876940 EE On-Demand Mild PDGFRB 40 41 CN(CCNC(=O)CC[C@@H]1CCc2ccccc21)CC(F)F ZINC000880876942 DF On-Demand Anodyne NQO2 20 42 CN(CCNC(=O)CC[C@@H]1CCc2ccccc21)CC(F)F ZINC000880876942 DF On-Demand Anodyne MTNR1A 17 40 CN(CCNC(=O)CC[C@H]1CCc2ccccc21)CC(F)F ZINC000880876943 DF On-Demand Anodyne NQO2 20 42 CN(CCNC(=O)CC[C@H]1CCc2ccccc21)CC(F)F ZINC000880876943 DF On-Demand Anodyne MTNR1A 17 40 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cnc2cc[nH]c2c1 ZINC000880877021 DD On-Demand Anodyne HCRTR1 23 42 O=C(N[C@@H]1CCCc2ccc(Cl)cc21)[C@@H]1CCc2nncn2CC1 ZINC000880877043 EG On-Demand Anodyne CNR1 49 30 O=C(N[C@@H]1CCCc2ccc(Cl)cc21)[C@H]1CCc2nncn2CC1 ZINC000880877044 EG On-Demand Anodyne CNR1 49 30 CCN(CC)C(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877068 FD On-Demand Mild P2RY12 15 42 CCN(CC)C(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877068 FD On-Demand Mild PDGFRB 44 41 COCCCN(C)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877071 DD On-Demand Mild ADRB1 44 34 CCOC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880877088 DE On-Demand Mild PDGFRB 41 40 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C(C)C ZINC000880877126 CE On-Demand Mild ADRB1 45 34 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C(C)C ZINC000880877128 CE On-Demand Mild ADRB1 45 34 COc1ccc([C@H](CO)N(C)C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880877131 FF On-Demand Mild ENPP1 68 33 COc1ccc([C@@H](CO)N(C)C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880877135 FF On-Demand Mild ENPP1 68 33 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccco1 ZINC000880877136 DF On-Demand Mild ADRB1 44 33 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccco1 ZINC000880877137 DF On-Demand Mild ADRB1 44 33 COC[C@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877168 EF On-Demand Mild ADRB1 44 34 COC[C@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877168 EF On-Demand Mild PAPA1_CARPA 43 37 COC[C@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877168 EF On-Demand Mild CTRB_BOVIN 44 30 COC[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877170 EF On-Demand Mild ADRB1 44 34 COC[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877170 EF On-Demand Mild PAPA1_CARPA 43 37 COC[C@@H](Cc1ccccc1)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877170 EF On-Demand Mild CTRB_BOVIN 44 30 CCO[C@@H](CCNC(=O)Nc1ccc(OC)c(C#N)c1)C(C)C ZINC000880877178 DG On-Demand Mild ADRB1 47 36 COCC1(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877188 CD On-Demand Mild ENPP1 61 31 Cn1ncc(Br)c1CC(=O)NCCc1c[nH]c2c(Cl)cccc12 ZINC000880877189 GG On-Demand Anodyne P2RX7 17 42 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880877225 ED On-Demand Anodyne HCRTR1 18 42 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880877227 ED On-Demand Anodyne HCRTR1 18 42 CCc1cnc(CN(C)C(=O)Nc2ccc(OC)c(C#N)c2)s1 ZINC000880877236 EG On-Demand Mild ENPP1 55 30 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880877237 DD On-Demand Mild PDGFRB 26 41 C#CC[C@@H](COC)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880877244 DD On-Demand Mild KCNQ2 50 34 C#CC[C@H](COC)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880877245 DD On-Demand Mild KCNQ2 50 34 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc2ccccc2cc1F ZINC000880877246 EG On-Demand Anodyne HCRTR1 54 50 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc2ccccc2cc1F ZINC000880877246 EG On-Demand Anodyne HCRTR2 28 50 Cn1nnc(C(=O)N[C@@H]2CCCc3ccc(Cl)cc32)n1 ZINC000880877252 CD On-Demand Anodyne KCNN3 15 44 CCC[C@H](CCO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877255 DE On-Demand Mild ADRB1 45 34 CCC[C@@H](CCO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877256 DE On-Demand Mild ADRB1 45 34 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877264 DE On-Demand Mild PDGFRB 48 43 CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877264 DE On-Demand Mild S1PR2 31 46 CC(=O)NC[C@@H]1CCCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880877282 EE On-Demand Anodyne HCRTR1 18 42 CC(=O)NC[C@@H]1CCCCN1C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880877282 EE On-Demand Anodyne MPO 52 36 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cncc2[nH]ccc12 ZINC000880877309 DD On-Demand Anodyne HCRTR1 24 45 CC[C@@H]1CN2CCCC[C@@H]2CN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877341 EG On-Demand Mild QRFPR 40 33 CC[C@@H]1CN2CCCC[C@H]2CN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877345 EG On-Demand Mild QRFPR 40 33 CCSCC[C@@H](C)N(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877351 DH On-Demand Mild ENPP1 60 31 CCSCC[C@H](C)N(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877357 DH On-Demand Mild ENPP1 60 31 C#CCSCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877386 CE On-Demand Mild ADRB1 47 37 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880877411 EG On-Demand Anodyne HCRTR1 19 40 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880877411 EG On-Demand Anodyne NQO2 18 41 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880877411 EG On-Demand Anodyne MTNR1A 24 46 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880877411 EG On-Demand Anodyne MTNR1B 30 46 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@H]1CCc2ccccc21 ZINC000880877411 EG On-Demand Anodyne EBP 16 41 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880877414 EG On-Demand Anodyne HCRTR1 19 40 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880877414 EG On-Demand Anodyne NQO2 18 41 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880877414 EG On-Demand Anodyne MTNR1A 24 46 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880877414 EG On-Demand Anodyne MTNR1B 30 46 CC(=O)NC[C@@H]1CCCCN1C(=O)CC[C@@H]1CCc2ccccc21 ZINC000880877414 EG On-Demand Anodyne EBP 16 41 CC[C@H](CCO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877439 CD On-Demand Mild ADRB1 40 30 CC[C@@H](CCO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877440 CD On-Demand Mild ADRB1 40 30 CNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877450 EC On-Demand Mild HTR1B 15 44 CNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877450 EC On-Demand Mild XDH 17 40 CNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877450 EC On-Demand Mild PDGFRB 47 43 CNC(=O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877450 EC On-Demand Mild ENPP1 66 33 CC(=O)NC[C@@H]1CCCCN1C(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880877490 DE On-Demand Anodyne FKBP1A 18 40 CC(=O)NC[C@@H]1CCCCN1C(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880877490 DE On-Demand Anodyne HCRTR1 23 47 CC(=O)NC[C@@H]1CCCCN1C(=O)[C@@H]1C[C@]1(C)c1ccccc1 ZINC000880877490 DE On-Demand Anodyne PREP 41 37 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880877501 GG On-Demand Anodyne HCRTR1 35 47 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880877501 GG On-Demand Anodyne HCRTR2 19 47 C#CCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877517 CE On-Demand Mild ADRB1 46 36 C#CCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877517 CE On-Demand Mild QPCT 16 46 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cnc(C(C)C)nc1C ZINC000880877532 DE On-Demand Anodyne HCRTR1 24 41 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cnc(CC2CC2)s1 ZINC000880877547 DE On-Demand Anodyne HCRTR1 23 40 CCC1(NC(=O)Nc2ccc(OC)c(C#N)c2)CCC1 ZINC000880877554 CG On-Demand Mild ADRB1 41 32 CCCn1cc(CN2CCCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cn1 ZINC000880877559 GF On-Demand Mild PDGFRB 48 42 CCCN(CC)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877575 DE On-Demand Mild ADRB1 45 35 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)CCS1 ZINC000880877595 DF On-Demand Mild ENPP1 54 32 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCCc4ccc(Cl)cc43)cc2)N1 ZINC000880877643 FI On-Demand Anodyne BDKRB1 20 41 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCCc4ccc(Cl)cc43)cc2)N1 ZINC000880877644 FI On-Demand Anodyne BDKRB1 20 41 CC(=O)NC[C@@H]1CCCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880877646 ED On-Demand Anodyne HCRTR1 31 45 CC(=O)NC[C@@H]1CCCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880877646 ED On-Demand Anodyne CPT1A 59 38 CC(=O)NC[C@@H]1CCCCN1C(=O)c1coc(-c2ccccn2)n1 ZINC000880877646 ED On-Demand Anodyne HCRTR2 15 45 CN(CCNC(=O)c1cc2ccccc2cc1F)CC(F)F ZINC000880877671 DF On-Demand Anodyne POLR1A 46 39 C/C=C/C[C@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880877695 DH On-Demand Anodyne MAP3K12 29 40 C/C=C\C[C@@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880877696 DH On-Demand Anodyne MAP3K12 29 40 C/C=C/C[C@@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880877697 DH On-Demand Anodyne MAP3K12 29 40 C/C=C\C[C@H]1CCCN(C(=O)c2ncccc2-c2ccccn2)C1 ZINC000880877698 DH On-Demand Anodyne MAP3K12 29 40 COCCCOC1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880877723 DD On-Demand Mild PDGFRB 34 40 CCC1(CNC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877735 CF On-Demand Mild ADRB1 42 32 CC[C@@H](C)CN(CC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877736 CG On-Demand Mild ENPP1 54 31 CC[C@H](C)CN(CC)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877737 CG On-Demand Mild ENPP1 54 31 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880877747 FG On-Demand Anodyne HCRTR1 19 40 CC(=O)NC[C@@H]1CCCCN1C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880877747 FG On-Demand Anodyne PDE4D 17 41 CNC(=O)CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877778 ED On-Demand Mild PDGFRB 42 42 CNC(=O)CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877778 ED On-Demand Mild ENPP1 65 32 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccc(C)o1 ZINC000880877811 EF On-Demand Mild ADRB1 42 33 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1ccc(C)o1 ZINC000880877812 EF On-Demand Mild ADRB1 42 33 CC[C@@H](O)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877816 CD On-Demand Mild ADRB1 55 44 CC[C@H](O)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877817 CD On-Demand Mild ADRB1 55 44 COC(=O)CCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877837 EF On-Demand Mild PDGFRB 44 42 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877854 DD On-Demand Mild LGMN 70 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877854 DD On-Demand Mild PFKFB3 54 32 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)[C@H](CC)CN1C(C)=O ZINC000880877868 FF On-Demand Mild AR 15 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)[C@@H](CC)CN1C(C)=O ZINC000880877870 FF On-Demand Mild AR 15 40 CC[C@H]1CN(C(C)=O)[C@H](CC)CN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880877871 FF On-Demand Mild AR 15 40 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877903 DC On-Demand Anodyne DRD4 44 33 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877903 DC On-Demand Anodyne PLD1 93 43 O=C1CC[C@@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877903 DC On-Demand Anodyne PLD2 111 43 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877904 DC On-Demand Anodyne DRD4 44 33 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877904 DC On-Demand Anodyne PLD1 93 43 O=C1CC[C@H](c2ccc(C(=O)NCCN3CC[C@H](O)C3)cc2)N1 ZINC000880877904 DC On-Demand Anodyne PLD2 111 43 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne HTR1A 18 47 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne DRD2 23 40 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne DRD4 44 35 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne SLC6A1 61 36 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne DRD3 40 43 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne CCR3 57 40 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne PLD1 96 42 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne PLD2 117 42 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne MCHR1 26 44 O=C(NCCN1CC[C@H](O)C1)c1cc2ccccc2cc1F ZINC000880877915 DD On-Demand Anodyne POLR1A 62 42 O=C(NCCN1CC[C@H](O)C1)c1cccn2nccc12 ZINC000880877925 CC On-Demand Anodyne DRD4 43 33 O=C(NCCN1CC[C@H](O)C1)c1cccn2nccc12 ZINC000880877925 CC On-Demand Anodyne DRD3 16 52 O=C(NCCN1CC[C@H](O)C1)c1cccn2nccc12 ZINC000880877925 CC On-Demand Anodyne PLD1 67 38 O=C(NCCN1CC[C@H](O)C1)c1cccn2nccc12 ZINC000880877925 CC On-Demand Anodyne PLD2 77 37 O=C(NCCN1CC[C@H](O)C1)c1cccc2nsnc12 ZINC000880877949 CC On-Demand Anodyne PLD2 46 36 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880877973 GG On-Demand Mild NPY2R 17 47 Cc1cc(-c2nc(C)c(C(=O)NCCN3CC[C@H](O)C3)s2)ccc1F ZINC000880877978 FE On-Demand Anodyne PLD1 48 35 Cc1cc(-c2nc(C)c(C(=O)NCCN3CC[C@H](O)C3)s2)ccc1F ZINC000880877978 FE On-Demand Anodyne PLD2 54 35 Cc1coc(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880877983 BC On-Demand Anodyne DRD4 41 35 Cc1coc(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880877983 BC On-Demand Anodyne PLD1 53 39 Cc1coc(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880877983 BC On-Demand Anodyne PLD2 45 39 O=C(NCCN1CC[C@H](O)C1)c1csc(-c2ncc[nH]2)n1 ZINC000880878007 DC On-Demand Anodyne PLD1 47 33 O=C(NCCN1CC[C@H](O)C1)c1csc(-c2ncc[nH]2)n1 ZINC000880878007 DC On-Demand Anodyne PLD2 49 33 O=C(NCCN1CC[C@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880878012 CC On-Demand Anodyne PLD1 45 35 O=C(NCCN1CC[C@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880878012 CC On-Demand Anodyne PLD2 50 35 O=C(NCCN1CC[C@H](O)C1)c1cnc(CC2CC2)s1 ZINC000880878012 CC On-Demand Anodyne SIRT2 40 37 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878069 ED On-Demand Mild ADRB1 40 32 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878069 ED On-Demand Mild PDGFRB 45 42 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878069 ED On-Demand Mild ABCB1 22 44 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878070 ED On-Demand Mild ADRB1 40 32 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878070 ED On-Demand Mild PDGFRB 45 42 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878070 ED On-Demand Mild ABCB1 22 44 CC[C@@](C)(CO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878073 CD On-Demand Mild ENPP1 60 31 CS(=O)(=O)C1CCC(C(=O)NCCc2c[nH]c3c(Cl)cccc23)CC1 ZINC000880878081 GG On-Demand Anodyne MTNR1A 42 47 CS(=O)(=O)C1CCC(C(=O)NCCc2c[nH]c3c(Cl)cccc23)CC1 ZINC000880878081 GG On-Demand Anodyne MTNR1B 28 44 COC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880878096 CD On-Demand Mild ADRB1 49 38 O=C(NCCN1CC[C@H](O)C1)c1ncccc1-c1ccccn1 ZINC000880878108 DC On-Demand Anodyne PLD1 49 39 O=C(NCCN1CC[C@H](O)C1)c1ncccc1-c1ccccn1 ZINC000880878108 DC On-Demand Anodyne PLD2 63 39 O=C(CC[C@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878127 EF On-Demand Anodyne ACE 22 41 O=C(CC[C@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878127 EF On-Demand Anodyne MME 19 41 O=C(CC[C@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878127 EF On-Demand Anodyne XIAP 29 40 O=C(CC[C@@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878128 EF On-Demand Anodyne ACE 22 41 O=C(CC[C@@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878128 EF On-Demand Anodyne MME 19 41 O=C(CC[C@@H]1CCc2ccccc21)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880878128 EF On-Demand Anodyne XIAP 29 40 O=C(CC[C@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878129 EF On-Demand Anodyne ACE 22 41 O=C(CC[C@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878129 EF On-Demand Anodyne MME 19 41 O=C(CC[C@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878129 EF On-Demand Anodyne XIAP 29 40 O=C(CC[C@@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878130 EF On-Demand Anodyne ACE 22 41 O=C(CC[C@@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878130 EF On-Demand Anodyne MME 19 41 O=C(CC[C@@H]1CCc2ccccc21)N[C@H]1CCN(C2CCC2)C1=O ZINC000880878130 EF On-Demand Anodyne XIAP 29 40 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne CELA1 19 41 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne CTRA_BOVIN 40 30 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne PREP 28 41 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne LGMN 65 39 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne SLC12A5 58 36 O=C(NCCN1CC[C@H](O)C1)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880878140 GC On-Demand Anodyne Q9NAW4_PLAFA 40 46 COC(=O)c1ccc2c(c1)CN(C(=O)Nc1ccc(OC)c(C#N)c1)CC2 ZINC000880878143 FF On-Demand Mild PDGFRB 26 40 CCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878144 BD On-Demand Mild ENPP1 68 33 C=CC[C@H](CO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878160 CD On-Demand Mild ADRB1 43 34 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878228 DF On-Demand Mild DRD2 31 40 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878228 DF On-Demand Mild ACKR3 64 33 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878229 DF On-Demand Mild DRD2 31 40 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878229 DF On-Demand Mild ACKR3 64 33 CC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878268 CF On-Demand Mild AR 17 40 CC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878268 CF On-Demand Mild PDGFRB 41 41 CC[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878268 CF On-Demand Mild CCR3 16 43 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cc(C)co1 ZINC000880878271 CD On-Demand Anodyne HCRTR1 19 42 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878286 DD On-Demand Mild PDGFRB 22 40 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(C3CCC3)C2=O)c(O)n1 ZINC000880878335 GE On-Demand Anodyne HTR3A 23 44 COc1ccccc1-c1ccc(C(=O)N[C@@H]2CCN(C3CCC3)C2=O)c(O)n1 ZINC000880878336 GE On-Demand Anodyne HTR3A 23 44 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880878337 GD On-Demand Anodyne DRD4 44 35 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880878337 GD On-Demand Anodyne PLD1 60 40 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880878337 GD On-Demand Anodyne UTS2R 25 41 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880878337 GD On-Demand Anodyne PLD2 80 39 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Br)c1 ZINC000880878337 GD On-Demand Anodyne CACNA1I 58 34 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880878338 CE On-Demand Mild ADRB1 41 31 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880878338 CE On-Demand Mild ENPP1 45 31 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880878339 CE On-Demand Mild ADRB1 41 31 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880878339 CE On-Demand Mild ENPP1 45 31 C=CCOCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878342 CD On-Demand Mild ADRB1 46 35 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878353 FF On-Demand Mild EPHX2 24 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878354 FF On-Demand Mild EPHX2 24 40 CCOC(=O)CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878375 FG On-Demand Mild P2RY12 18 42 CCOC(=O)CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878375 FG On-Demand Mild PDGFRB 35 41 CCOC(=O)CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878376 FG On-Demand Mild P2RY12 18 42 CCOC(=O)CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878376 FG On-Demand Mild PDGFRB 35 41 CC[C@H](CCO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878437 CE On-Demand Mild ADRB1 47 36 CC[C@@H](CCO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878438 CE On-Demand Mild ADRB1 47 36 O=C(COC1CC1)NCCc1c[nH]c2c(Cl)cccc12 ZINC000880878441 CF On-Demand Anodyne MTNR1A 23 41 C=C(C)COCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878444 CE On-Demand Mild ADRB1 46 35 COc1cccc(C2(NC(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880878456 EG On-Demand Mild TAAR1 29 44 C#CCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878474 CE On-Demand Mild ADRB1 46 36 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880878513 CC On-Demand Anodyne CACNA1H 20 40 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880878513 CC On-Demand Anodyne DRD4 44 35 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880878513 CC On-Demand Anodyne PLD1 48 38 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880878513 CC On-Demand Anodyne PLD2 55 38 Cc1cnc(Cl)c(C(=O)NCCN2CC[C@H](O)C2)c1 ZINC000880878513 CC On-Demand Anodyne CACNA1I 56 35 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne DRD2 15 41 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne DRD4 49 38 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne PDE4D 17 41 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne PLD1 67 42 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne UTS2R 26 45 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne PLD2 84 42 O=C(NCCN1CC[C@H](O)C1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880878522 ED On-Demand Anodyne CACNA1I 68 42 CNC(=O)CCCN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878524 DD On-Demand Mild ENPP1 66 33 O=C(NCCN1CC[C@H](O)C1)c1coc(-c2ccccn2)n1 ZINC000880878530 DC On-Demand Anodyne PLD1 45 37 O=C(NCCN1CC[C@H](O)C1)c1coc(-c2ccccn2)n1 ZINC000880878530 DC On-Demand Anodyne PLD2 56 37 O=C(NCCN1CC[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880878540 DC On-Demand Anodyne CCR3 50 40 O=C(NCCN1CC[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880878540 DC On-Demand Anodyne PYGL 27 40 O=C(NCCN1CC[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880878540 DC On-Demand Anodyne PLD1 113 51 O=C(NCCN1CC[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880878540 DC On-Demand Anodyne PLD2 119 51 O=C(NCCN1CC[C@H](O)C1)c1cc2cc(F)ccc2[nH]c1=O ZINC000880878540 DC On-Demand Anodyne WNT3A 46 34 C=CCCC[C@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878571 DE On-Demand Mild SLC6A1 49 34 C=CCCC[C@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878571 DE On-Demand Mild OPRK1 22 42 C=CCCC[C@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878571 DE On-Demand Mild CCR5 27 40 C=CCCC[C@@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878572 DE On-Demand Mild SLC6A1 49 34 C=CCCC[C@@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878572 DE On-Demand Mild OPRK1 22 42 C=CCCC[C@@H](C(=O)NCCN1CC[C@H](O)C1)c1ccccc1 ZINC000880878572 DE On-Demand Mild CCR5 27 40 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878610 DD On-Demand Mild EPHX2 47 58 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878611 DD On-Demand Mild EPHX2 47 58 C#CC(C)(C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878617 CE On-Demand Mild IMDH_CRYPV 58 40 CCO[C@@H](CCN(C)C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878624 EE On-Demand Mild ADRB1 42 32 CCC1(CO)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878702 DF On-Demand Mild PDGFRB 39 40 O=C(CC[C@H]1CCc2ccccc21)NCCN1CC[C@H](O)C1 ZINC000880878707 DD On-Demand Anodyne OPRK1 16 40 O=C(CC[C@H]1CCc2ccccc21)NCCN1CC[C@H](O)C1 ZINC000880878707 DD On-Demand Anodyne NQO2 17 41 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CC[C@H](O)C1 ZINC000880878708 DD On-Demand Anodyne OPRK1 16 40 O=C(CC[C@@H]1CCc2ccccc21)NCCN1CC[C@H](O)C1 ZINC000880878708 DD On-Demand Anodyne NQO2 17 41 CC#CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878720 CE On-Demand Mild ADRB1 47 37 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@@H]1O ZINC000880878723 CD On-Demand Mild ENPP1 60 32 CC[C@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@H]1O ZINC000880878724 CD On-Demand Mild ENPP1 60 32 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCN(C3CCC3)C1=O)C2 ZINC000880878730 EE On-Demand Anodyne FKBP1A 44 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(C3CCC3)C1=O)C2 ZINC000880878732 EE On-Demand Anodyne FKBP1A 44 40 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878739 DD On-Demand Mild PDGFRB 48 43 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878739 DD On-Demand Mild S1PR2 30 44 COCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878739 DD On-Demand Mild ENPP1 61 33 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](O)C(F)(F)F ZINC000880878776 EE On-Demand Mild ADRB1 43 34 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](O)C(F)(F)F ZINC000880878777 EE On-Demand Mild ADRB1 43 34 CCC1(O)CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878783 DF On-Demand Mild EPHX2 44 38 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cccn2nccc12 ZINC000880878786 DD On-Demand Anodyne HCRTR1 40 48 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cccn2nccc12 ZINC000880878786 DD On-Demand Anodyne TYK2 15 40 CC(=O)NC[C@@H]1CCCCN1C(=O)c1cccn2nccc12 ZINC000880878786 DD On-Demand Anodyne HCRTR2 25 48 COCCNc1ccccc1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878833 FF On-Demand Mild ADRB1 45 34 COCCNc1ccccc1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878833 FF On-Demand Mild ROCK2 15 41 CC[C@]1(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878844 CG On-Demand Mild PDGFRB 30 42 CC[C@]1(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880878844 CG On-Demand Mild S1PR2 25 41 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878851 FD On-Demand Mild PDGFRB 46 42 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880878851 FD On-Demand Mild ENPP1 55 32 COCC(C)(C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878856 CE On-Demand Mild AR 17 40 COCC(C)(C)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878856 CE On-Demand Mild IMDH_CRYPV 54 38 O=C(NCCc1c[nH]c2c(Cl)cccc12)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880878919 GF On-Demand Anodyne MTNR1A 17 40 CCC(CC)(CCO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878926 DF On-Demand Mild ADRB1 41 31 O=C(NCCN1CC[C@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880878957 FD On-Demand Anodyne DRD4 40 31 O=C(NCCN1CC[C@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880878957 FD On-Demand Anodyne PLD1 53 34 O=C(NCCN1CC[C@H](O)C1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880878957 FD On-Demand Anodyne PLD2 64 34 C=CCCOCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880878964 CE On-Demand Mild ADRB1 45 34 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne ACE 35 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne MME 20 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne XIAP 75 42 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne BIRC3 63 37 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne BIRC2 69 39 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878966 GC On-Demand Anodyne BIRC8 56 35 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne ACE 35 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne MME 20 41 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne XIAP 75 42 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne BIRC3 63 37 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne BIRC2 69 39 NC(=O)[C@@H]1CC[C@H](C(=O)N[C@H]2CCN(C3CCC3)C2=O)N1Cc1ccccc1 ZINC000880878967 GC On-Demand Anodyne BIRC8 56 35 O=C(NCCN1CC[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880878969 DC On-Demand Anodyne GABRA1 16 45 O=C(NCCN1CC[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880878969 DC On-Demand Anodyne HTR1D 26 42 O=C(NCCN1CC[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880878969 DC On-Demand Anodyne HTR1B 23 42 O=C(NCCN1CC[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880878969 DC On-Demand Anodyne PLD1 50 40 O=C(NCCN1CC[C@H](O)C1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880878969 DC On-Demand Anodyne PLD2 58 38 O=C(NCCN1CC[C@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880879011 CC On-Demand Anodyne DRD4 44 34 O=C(NCCN1CC[C@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880879011 CC On-Demand Anodyne PLD1 87 50 O=C(NCCN1CC[C@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880879011 CC On-Demand Anodyne PLD2 116 50 O=C(NCCN1CC[C@H](O)C1)c1cnc2cc[nH]c2c1 ZINC000880879011 CC On-Demand Anodyne HPGDS 47 35 CCCCN(CCCO)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879108 DF On-Demand Mild INHA 46 36 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne HTR1A 48 43 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne DRD2 52 47 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne DRD4 44 47 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne ADRA1D 25 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne ADRA1A 24 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne ADRA1B 15 40 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne DRD3 69 44 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne OPRK1 20 49 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne HTR4 40 37 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne HCN1 51 33 COc1ccccc1-c1ccc(C(=O)NCCN2CC[C@H](O)C2)c(O)n1 ZINC000880879115 FD On-Demand Anodyne HCN4 47 32 CC(C)(C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccc(C(F)(F)F)cc1 ZINC000880879127 FG On-Demand Anodyne BIRC2 27 41 CC(C)(C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccc(C(F)(F)F)cc1 ZINC000880879128 FG On-Demand Anodyne BIRC2 27 41 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879138 DE On-Demand Mild DPP4 25 41 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879138 DE On-Demand Mild QRFPR 40 34 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879138 DE On-Demand Mild ACKR3 62 32 COC(=O)C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879138 DE On-Demand Mild PFKFB3 55 33 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879139 DE On-Demand Mild DPP4 25 41 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879139 DE On-Demand Mild QRFPR 40 34 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879139 DE On-Demand Mild ACKR3 62 32 COC(=O)C[C@@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879139 DE On-Demand Mild PFKFB3 55 33 CCC(CC)(CO)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879150 DE On-Demand Mild ADRB1 41 32 O=C(NCCN1CC[C@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880879152 FE On-Demand Anodyne DRD4 42 33 O=C(NCCN1CC[C@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880879152 FE On-Demand Anodyne DRD3 16 44 O=C(NCCN1CC[C@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880879152 FE On-Demand Anodyne PLD1 56 41 O=C(NCCN1CC[C@H](O)C1)c1cc(Br)ccc1C1CC1 ZINC000880879152 FE On-Demand Anodyne PLD2 63 41 O=C(N[C@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879157 ED On-Demand Anodyne PYGL 16 44 O=C(N[C@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879157 ED On-Demand Anodyne PYGM 25 44 O=C(N[C@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879157 ED On-Demand Anodyne PLD2 42 39 O=C(N[C@@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879158 ED On-Demand Anodyne PYGL 16 44 O=C(N[C@@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879158 ED On-Demand Anodyne PYGM 25 44 O=C(N[C@@H]1CCN(C2CCC2)C1=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880879158 ED On-Demand Anodyne PLD2 42 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879174 GG On-Demand Anodyne PAPA1_CARPA 38 45 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879174 GG On-Demand Anodyne CTSK 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879174 GG On-Demand Anodyne FPR1 45 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879175 GG On-Demand Anodyne PAPA1_CARPA 38 45 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879175 GG On-Demand Anodyne CTSK 15 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NC1(c2c(F)cccc2F)CCC1 ZINC000880879175 GG On-Demand Anodyne FPR1 45 36 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1CCN(C2CCC2)C1=O ZINC000880879203 FD On-Demand Anodyne BIRC2 48 35 O=C(Cc1ccccc1N1CCCC1=O)N[C@@H]1CCN(C2CCC2)C1=O ZINC000880879204 FD On-Demand Anodyne BIRC2 48 35 CC(C)(C(=O)NCCN1CC[C@H](O)C1)c1ccc(F)cc1F ZINC000880879237 DD On-Demand Anodyne CCR3 40 36 O=C(NCCN1CC[C@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880879252 EE On-Demand Anodyne DRD4 44 36 O=C(NCCN1CC[C@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880879252 EE On-Demand Anodyne PLD1 54 35 O=C(NCCN1CC[C@H](O)C1)c1sc2cccc(F)c2c1Cl ZINC000880879252 EE On-Demand Anodyne PLD2 67 35 O=C(Cc1ccccc1N1CCCC1=O)NCCN1CC[C@H](O)C1 ZINC000880879256 EC On-Demand Anodyne PLD1 66 36 O=C(Cc1ccccc1N1CCCC1=O)NCCN1CC[C@H](O)C1 ZINC000880879256 EC On-Demand Anodyne PLD2 54 35 O=C(NCCN1CC[C@H](O)C1)c1cncc2[nH]ccc12 ZINC000880879259 CC On-Demand Anodyne PLD1 57 37 O=C(NCCN1CC[C@H](O)C1)c1cncc2[nH]ccc12 ZINC000880879259 CC On-Demand Anodyne PLD2 66 37 O=C(NCCN1CC[C@H](O)C1)c1cncc2[nH]ccc12 ZINC000880879259 CC On-Demand Anodyne PRKCQ 18 42 COCCOC1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879267 DD On-Demand Mild PDGFRB 35 41 CNC(C)(C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879270 CD On-Demand Mild ADRB1 42 33 COC[C@]1(C)CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880879300 EE On-Demand Anodyne MTNR1B 15 42 COC[C@]1(C)CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880879301 EE On-Demand Anodyne MTNR1B 15 42 COC[C@@]1(C)CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880879302 EE On-Demand Anodyne MTNR1B 15 42 COC[C@@]1(C)CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)CCO1 ZINC000880879303 EE On-Demand Anodyne MTNR1B 15 42 O=C(NCCN1CC[C@H](O)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880879304 DD On-Demand Anodyne SIGMAR1 15 40 O=C(NCCN1CC[C@H](O)C1)[C@@]1(c2ccccc2)C[C@H](F)C1 ZINC000880879304 DD On-Demand Anodyne PLD2 41 32 NC(=O)[C@@H]1CC[C@H](C(=O)NCCN2CC[C@H](O)C2)N1Cc1ccccc1 ZINC000880879336 FB On-Demand Anodyne SIGMAR1 29 44 CC[C@@H](C)n1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C1CC1 ZINC000880879353 FI On-Demand Mild HTR2A 33 40 C=CCCC[C@@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879357 EG On-Demand Mild XIAP 50 41 C=CCCC[C@@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879357 EG On-Demand Mild BIRC3 54 38 C=CCCC[C@@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879357 EG On-Demand Mild BIRC2 74 41 C=CCCC[C@@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879357 EG On-Demand Mild BIRC8 51 38 C=CCCC[C@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879358 EG On-Demand Mild XIAP 50 41 C=CCCC[C@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879358 EG On-Demand Mild BIRC3 54 38 C=CCCC[C@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879358 EG On-Demand Mild BIRC2 74 41 C=CCCC[C@H](C(=O)N[C@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879358 EG On-Demand Mild BIRC8 51 38 C=CCCC[C@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879359 EG On-Demand Mild XIAP 50 41 C=CCCC[C@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879359 EG On-Demand Mild BIRC3 54 38 C=CCCC[C@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879359 EG On-Demand Mild BIRC2 74 41 C=CCCC[C@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879359 EG On-Demand Mild BIRC8 51 38 C=CCCC[C@@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879360 EG On-Demand Mild XIAP 50 41 C=CCCC[C@@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879360 EG On-Demand Mild BIRC3 54 38 C=CCCC[C@@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879360 EG On-Demand Mild BIRC2 74 41 C=CCCC[C@@H](C(=O)N[C@@H]1CCN(C2CCC2)C1=O)c1ccccc1 ZINC000880879360 EG On-Demand Mild BIRC8 51 38 CC(C)(C(=O)NCCN1CC[C@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880879374 EE On-Demand Anodyne OPRK1 15 46 CC(C)(C(=O)NCCN1CC[C@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880879374 EE On-Demand Anodyne EPHX2 15 42 CC(C)(C(=O)NCCN1CC[C@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880879374 EE On-Demand Anodyne MCHR1 36 42 CC(C)(C(=O)NCCN1CC[C@H](O)C1)c1ccc(C(F)(F)F)cc1 ZINC000880879374 EE On-Demand Anodyne CACNA1I 43 38 O=C(N[C@@H]1CCN(C2CCC2)C1=O)c1cccc2nsnc12 ZINC000880879404 DD On-Demand Anodyne HTR3A 29 40 O=C(N[C@H]1CCN(C2CCC2)C1=O)c1cccc2nsnc12 ZINC000880879405 DD On-Demand Anodyne HTR3A 29 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879422 EE On-Demand Mild EPHX2 28 40 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879423 EE On-Demand Mild EPHX2 28 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879424 EE On-Demand Mild EPHX2 28 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879425 EE On-Demand Mild EPHX2 28 40 CCC1(CC)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879484 CG On-Demand Mild XDH 15 40 CCC1(CC)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879484 CG On-Demand Mild PDGFRB 40 39 CCC1(CC)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879484 CG On-Demand Mild ENPP1 62 33 CSc1nccnc1C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880879492 DG On-Demand Anodyne GRIA4 17 42 O=C(c1cc2ccccc2cc1F)N1CCC[C@@H]1Cn1ccnc1 ZINC000880879503 DG On-Demand Anodyne HCRTR1 27 42 O=C(c1cc2ccccc2cc1F)N1CCC[C@@H]1Cn1ccnc1 ZINC000880879503 DG On-Demand Anodyne HCRTR2 15 42 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880879660 GH On-Demand Mild PDGFRB 42 38 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)cc1 ZINC000880879660 GH On-Demand Mild ENPP1 60 32 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1OC ZINC000880879677 EI On-Demand Anodyne GRM4 24 42 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1OC ZINC000880879677 EI On-Demand Anodyne ENPP1 78 41 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1OC ZINC000880879677 EI On-Demand Anodyne KCNK3 52 40 CCCOc1ccc(NC(=O)c2cc(C)cnc2Cl)cc1OC ZINC000880879677 EI On-Demand Anodyne KCNK9 47 40 CCCOc1ccc(NC(=O)CC(C)(C)CC(F)F)cc1OC ZINC000880879690 EI On-Demand Anodyne ENPP1 77 38 COCCCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879716 CD On-Demand Mild ENPP1 50 31 CCCOc1ccc(NC(=O)Cc2c(Br)cnn2C)cc1OC ZINC000880879717 GG On-Demand Anodyne HTR2A 47 46 CCCOc1ccc(NC(=O)Cc2c(Br)cnn2C)cc1OC ZINC000880879717 GG On-Demand Anodyne HTR2C 16 46 CCCOc1ccc(NC(=O)Cc2c(Br)cnn2C)cc1OC ZINC000880879717 GG On-Demand Anodyne ENPP1 84 42 O=C(COC1CC1)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880879827 CF On-Demand Anodyne GRIA4 15 44 O=C(COC1CC1)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880879827 CF On-Demand Anodyne EPHX2 18 41 CC[C@H](C)CONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879836 CF On-Demand Mild ADRB1 41 32 CC[C@H](C)CONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879836 CF On-Demand Mild ENPP1 44 29 CC[C@@H](C)CONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879837 CF On-Demand Mild ADRB1 41 32 CC[C@@H](C)CONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879837 CF On-Demand Mild ENPP1 44 29 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCC[C@@H]3c3ccccc3)cc2)N1 ZINC000880879843 EH On-Demand Anodyne SSTR3 32 43 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCC[C@@H]3c3ccccc3)cc2)N1 ZINC000880879843 EH On-Demand Anodyne PRKACA 41 36 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCC[C@@H]3c3ccccc3)cc2)N1 ZINC000880879844 EH On-Demand Anodyne SSTR3 32 43 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCC[C@@H]3c3ccccc3)cc2)N1 ZINC000880879844 EH On-Demand Anodyne PRKACA 41 36 C[C@H](Sc1nc(CC(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)cs1)C(N)=O ZINC000880879865 GG On-Demand Anodyne GRIA4 15 41 C[C@@H](Sc1nc(CC(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)cs1)C(N)=O ZINC000880879866 GG On-Demand Anodyne GRIA4 15 41 CCn1c(S)nnc1C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880879875 GF On-Demand Mild PDGFRB 38 40 C#CCOCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879879 CD On-Demand Mild ADRB1 46 35 COC[C@@H]1CCCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879883 DF On-Demand Mild PDGFRB 49 42 COC[C@@H]1CCCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880879883 DF On-Demand Mild QRFPR 41 35 COCC1(NC(=O)Nc2ccc(OC)c(C#N)c2)CCC1 ZINC000880879911 CE On-Demand Mild ADRB1 41 32 COCC1(NC(=O)Nc2ccc(OC)c(C#N)c2)CCC1 ZINC000880879911 CE On-Demand Mild ENPP1 50 32 C=CCCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880879951 CG On-Demand Mild ADRB1 45 35 CCc1nnc(CNC(=O)Nc2ccc(OC)c(C#N)c2)s1 ZINC000880880026 DE On-Demand Mild ADRB1 43 32 CCc1nnc(CNC(=O)Nc2ccc(OC)c(C#N)c2)s1 ZINC000880880026 DE On-Demand Mild ENPP1 65 31 CCCN(CCN1CCCC1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880042 EF On-Demand Mild DRD4 41 32 CCCN(CCN1CCCC1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880042 EF On-Demand Mild CASR 39 42 CCCN(CCN1CCCC1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880042 EF On-Demand Mild MCHR1 29 45 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880063 FF On-Demand Mild AR 22 40 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880063 FF On-Demand Mild EPHX2 33 42 Cn1nnc(C(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)n1 ZINC000880880076 CD On-Demand Anodyne GRIA4 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne PGC 51 34 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne PAPA1_CARPA 41 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne CCKAR 34 47 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne CTSK 19 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne CTSL 20 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne REN 61 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880081 GG On-Demand Anodyne FPR1 49 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne PGC 51 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne PAPA1_CARPA 41 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne CCKAR 34 47 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne CTSK 19 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne CTSL 20 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne REN 61 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCC[C@@H]1c1ccccc1 ZINC000880880082 GG On-Demand Anodyne FPR1 49 41 C=C(C)[C@H]1OCC[C@H]1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880085 DF On-Demand Mild ADRB1 41 32 C=C(C)[C@@H]1OCC[C@H]1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880086 DF On-Demand Mild ADRB1 41 32 C=C(C)[C@H]1OCC[C@@H]1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880087 DF On-Demand Mild ADRB1 41 32 C=C(C)[C@@H]1OCC[C@@H]1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880089 DF On-Demand Mild ADRB1 41 32 CC[C@@H](C)n1nc(NC(=O)Nc2ccc(OC)c(C#N)c2)cc1C ZINC000880880092 EH On-Demand Mild HTR2A 28 42 CC[C@@H](C)n1nc(NC(=O)Nc2ccc(OC)c(C#N)c2)cc1C ZINC000880880092 EH On-Demand Mild ENPP1 60 31 COCC[C@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880131 DD On-Demand Mild ADRB1 42 32 COCC[C@@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880132 DD On-Demand Mild ADRB1 42 32 C=C[C@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880145 CG On-Demand Mild QRFPR 40 34 C=C[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880146 CG On-Demand Mild QRFPR 40 34 CCCOc1ccc(NC(=O)[C@H]2c3c[nH]nc3CC[C@@H]2C)cc1OC ZINC000880880148 EH On-Demand Anodyne ENPP1 76 36 CCCOc1ccc(NC(=O)[C@H]2c3c[nH]nc3CC[C@H]2C)cc1OC ZINC000880880149 EH On-Demand Anodyne ENPP1 76 36 CCCOc1ccc(NC(=O)[C@@H]2c3c[nH]nc3CC[C@@H]2C)cc1OC ZINC000880880150 EH On-Demand Anodyne ENPP1 76 36 CCCOc1ccc(NC(=O)[C@@H]2c3c[nH]nc3CC[C@H]2C)cc1OC ZINC000880880151 EH On-Demand Anodyne ENPP1 76 36 CCCOc1ccc(NC(=O)COC2CC2)cc1OC ZINC000880880154 CF On-Demand Anodyne ENPP1 83 39 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880224 GF On-Demand Mild PDGFRB 31 40 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880224 GF On-Demand Mild EPHX2 31 40 CS(=O)(=O)C1CCC(C(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)CC1 ZINC000880880276 EG On-Demand Anodyne GRIA4 20 50 CCC1(O)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880281 CD On-Demand Mild PDGFRB 39 41 CCC1(O)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880880281 CD On-Demand Mild ENPP1 62 34 COCC(C)(C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880294 CE On-Demand Mild ADRB1 42 32 CCCOc1ccc(NC(=O)CN2CCCCS2(=O)=O)cc1OC ZINC000880880295 FD On-Demand Anodyne ENPP1 82 41 O=C(N[C@@H]1CCC[C@@H]1c1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880880299 EF On-Demand Anodyne GRIA4 15 43 O=C(N[C@@H]1CCC[C@@H]1c1ccccc1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880880299 EF On-Demand Anodyne EPHX2 15 40 CCC(CC)(CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880880346 DF On-Demand Mild ADRB1 44 34 O=C(c1cnc(CC2CC2)s1)N1CCC[C@@H]1Cn1ccnc1 ZINC000880880469 DF On-Demand Anodyne TBXAS1 18 42 CCCOc1ccc(NC(=O)C[C@H]2CCNC2=O)cc1OC ZINC000880880558 DD On-Demand Anodyne ENPP1 85 41 CCCOc1ccc(NC(=O)C[C@@H]2CCNC2=O)cc1OC ZINC000880880559 DD On-Demand Anodyne ENPP1 85 41 CCOC(=O)CCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880880568 FG On-Demand Mild P2RY12 20 44 CCOC(=O)CCC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880880568 FG On-Demand Mild PDGFRB 40 43 CCCOc1ccc(NC(=O)[C@@H]2OC[C@@H]3CCC[C@@H]32)cc1OC ZINC000880880604 DG On-Demand Anodyne ENPP1 68 32 CCOC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C(C)C ZINC000880880605 DF On-Demand Mild ADRB1 43 33 COCCN(CCOC)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880880617 GE On-Demand Mild HTR1B 15 40 COCCN(CCOC)C1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880880617 GE On-Demand Mild PDGFRB 43 43 CCCOc1ccc(NC(=O)c2cc(C)co2)cc1OC ZINC000880880630 CH On-Demand Anodyne GRM4 17 43 CCCOc1ccc(NC(=O)c2cc(C)co2)cc1OC ZINC000880880630 CH On-Demand Anodyne ENPP1 77 37 CCCOc1ccc(NC(=O)c2cc(C)co2)cc1OC ZINC000880880630 CH On-Demand Anodyne KCNK3 44 38 CCCOc1ccc(NC(=O)c2cc(C)co2)cc1OC ZINC000880880630 CH On-Demand Anodyne KCNK9 42 38 COCC(C)(C)CCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880640 DG On-Demand Mild ADRB1 44 34 CC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880880671 CE On-Demand Mild ADRB1 46 36 CC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880880671 CE On-Demand Mild ENPP1 60 31 CCSCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880788 CF On-Demand Mild ADRB1 46 36 CCSCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880788 CF On-Demand Mild ENPP1 59 31 CCCOc1ccc(NC(=O)[C@@H]2CCc3nncn3CC2)cc1OC ZINC000880880850 EF On-Demand Anodyne STK17B 40 37 CCCOc1ccc(NC(=O)[C@@H]2CCc3nncn3CC2)cc1OC ZINC000880880850 EF On-Demand Anodyne ENPP1 71 34 CCCOc1ccc(NC(=O)[C@H]2CCc3nncn3CC2)cc1OC ZINC000880880851 EF On-Demand Anodyne STK17B 40 37 CCCOc1ccc(NC(=O)[C@H]2CCc3nncn3CC2)cc1OC ZINC000880880851 EF On-Demand Anodyne ENPP1 71 34 CCC1(CC)CN(C(=O)Nc2ccc(OC)c(C#N)c2)CC[S@@]1=O ZINC000880880861 EF On-Demand Mild ENPP1 61 32 C#CCC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880864 CD On-Demand Mild ADRB1 49 39 CCC1(CC)CN(C(=O)Nc2ccc(OC)c(C#N)c2)CC[S@]1=O ZINC000880880865 EF On-Demand Mild ENPP1 61 32 C#CCC[C@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880866 CD On-Demand Mild ADRB1 49 39 COCCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880948 CD On-Demand Mild ADRB1 41 31 COCCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880880948 CD On-Demand Mild ENPP1 67 33 CCN(CCNC(=O)Nc1ccc(OC)c(C#N)c1)CCC(F)(F)F ZINC000880880986 FF On-Demand Mild ADRB1 43 34 CCCOc1ccc(NC(=O)C2CCC(S(C)(=O)=O)CC2)cc1OC ZINC000880881013 FG On-Demand Anodyne MTNR1B 19 40 CCCOc1ccc(NC(=O)C2CCC(S(C)(=O)=O)CC2)cc1OC ZINC000880881013 FG On-Demand Anodyne ENPP1 68 32 CC[C@@H](C)n1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C ZINC000880881070 EH On-Demand Mild HTR2A 35 42 CC[C@@H](C)n1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C ZINC000880881070 EH On-Demand Mild ENPP1 45 31 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](O)c1ccccc1 ZINC000880881074 EG On-Demand Mild ADRB1 46 36 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](O)c1ccccc1 ZINC000880881076 EG On-Demand Mild ADRB1 46 36 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1OC ZINC000880881081 FG On-Demand Anodyne SSTR5 20 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1OC ZINC000880881081 FG On-Demand Anodyne EPHX2 19 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1OC ZINC000880881081 FG On-Demand Anodyne AURKA 21 40 CCCOc1ccc(NC(=O)c2ccc(CN3CCOCC3)o2)cc1OC ZINC000880881081 FG On-Demand Anodyne ENPP1 70 35 CCN(C)C(=O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881113 CD On-Demand Mild ADRB1 41 32 CCN(C)C(=O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881113 CD On-Demand Mild ENPP1 59 32 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1OC ZINC000880881131 EG On-Demand Anodyne GRM4 18 42 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1OC ZINC000880881131 EG On-Demand Anodyne MET 49 34 CCCOc1ccc(NC(=O)c2nccnc2SC)cc1OC ZINC000880881131 EG On-Demand Anodyne ENPP1 84 45 CCCOc1ccc(NC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)cc1OC ZINC000880881141 FF On-Demand Anodyne ENPP1 68 32 CCCOc1ccc(NC(=O)c2cnc(C(C)C)nc2C)cc1OC ZINC000880881165 EH On-Demand Anodyne ENPP1 79 38 CCCOc1ccc(NC(=O)c2cnc(C(C)C)nc2C)cc1OC ZINC000880881165 EH On-Demand Anodyne KCNK3 50 39 CCCOc1ccc(NC(=O)c2cnc(C(C)C)nc2C)cc1OC ZINC000880881165 EH On-Demand Anodyne KCNK9 42 39 CCCOc1ccc(NC(=O)c2ncsc2C2CC2)cc1OC ZINC000880881225 EI On-Demand Anodyne MAP1 74 38 CCCOc1ccc(NC(=O)c2ncsc2C2CC2)cc1OC ZINC000880881225 EI On-Demand Anodyne ENPP1 74 37 CCCOc1ccc(NC(=O)c2c3c(nn2C)CCSC3)cc1OC ZINC000880881257 FG On-Demand Anodyne ENPP1 72 34 CCCn1ccnc1CCCN(C)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881289 FG On-Demand Mild ENPP1 49 31 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1OC ZINC000880881292 CD On-Demand Anodyne KDR 16 48 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1OC ZINC000880881292 CD On-Demand Anodyne MET 50 36 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1OC ZINC000880881292 CD On-Demand Anodyne QPCT 23 45 CCCOc1ccc(NC(=O)c2nnn(C)n2)cc1OC ZINC000880881292 CD On-Demand Anodyne ENPP1 92 44 CCCOc1ccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cc1OC ZINC000880881298 FH On-Demand Anodyne TSHR 41 33 CCCOc1ccc(NC(=O)c2ccc([C@@H]3CCC(=O)N3)cc2)cc1OC ZINC000880881298 FH On-Demand Anodyne ENPP1 72 35 CCCOc1ccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cc1OC ZINC000880881299 FH On-Demand Anodyne TSHR 41 33 CCCOc1ccc(NC(=O)c2ccc([C@H]3CCC(=O)N3)cc2)cc1OC ZINC000880881299 FH On-Demand Anodyne ENPP1 72 35 CC[C@]1(C)CN(C(=O)Nc2ccc(OC)c(C#N)c2)CCO1 ZINC000880881334 DF On-Demand Mild EPHX2 18 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881343 DD On-Demand Mild PDGFRB 37 42 COCCO[C@@H]1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881344 DD On-Demand Mild PDGFRB 37 42 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)C(OC)OC ZINC000880881362 DE On-Demand Mild ADRB1 41 32 C#CCN(C(=O)Nc1ccc(OC)c(C#N)c1)C1CC1 ZINC000880881385 CE On-Demand Mild QRFPR 41 34 COCC(C)(C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881398 EE On-Demand Mild PDGFRB 47 42 COCC(COC)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881422 FD On-Demand Mild PDGFRB 50 45 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881441 CC On-Demand Mild PDGFRB 37 40 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881441 CC On-Demand Mild TRPV4 42 32 COCC1(O)CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881441 CC On-Demand Mild ENPP1 64 34 COCC(COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881444 CD On-Demand Mild ADRB1 44 34 COCC(COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881444 CD On-Demand Mild ENPP1 59 30 CCn1cc([C@H](C)NC(=O)Nc2ccc(OC)c(C#N)c2)cn1 ZINC000880881492 DF On-Demand Mild HTR2A 24 41 CCn1cc([C@H](C)NC(=O)Nc2ccc(OC)c(C#N)c2)cn1 ZINC000880881492 DF On-Demand Mild ENPP1 66 32 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild HTR1B 17 46 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild P2RY12 21 48 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild PDGFRB 80 49 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild SSTR1 22 40 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild PDGFRA 18 49 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild GPR119 15 43 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild ENPP1 61 32 COc1ccc(N2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)nc1 ZINC000880881511 FE On-Demand Mild DGAT1 34 44 COCC1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881512 DF On-Demand Mild EPHX2 46 39 COCC1CCC(NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881512 DF On-Demand Mild PDGFRA 19 41 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](C)O ZINC000880881571 CD On-Demand Mild ADRB1 44 36 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](C)O ZINC000880881571 CD On-Demand Mild ENPP1 61 31 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](C)O ZINC000880881573 CD On-Demand Mild ADRB1 44 36 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](C)O ZINC000880881573 CD On-Demand Mild ENPP1 61 31 COCC[C@@H](C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881575 CE On-Demand Mild ADRB1 46 35 COCC[C@H](C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881576 CE On-Demand Mild ADRB1 46 35 CCC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881579 DD On-Demand Mild HTR1B 15 43 CCC(=O)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881579 DD On-Demand Mild PDGFRB 43 42 CCCn1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C1CC1 ZINC000880881609 EH On-Demand Mild HTR2A 40 40 CCC(C)(C)OCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881627 DF On-Demand Mild ADRB1 46 35 C=C(C)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881643 CF On-Demand Mild ADRB1 49 37 CC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)CC(F)(F)F ZINC000880881649 EH On-Demand Mild ADRB1 45 36 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881686 DF On-Demand Mild PDGFRB 49 44 COC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881686 DF On-Demand Mild CCR3 15 42 CC/C=C\CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881715 CF On-Demand Mild ADRB1 45 37 CC/C=C\CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881715 CF On-Demand Mild ENPP1 61 31 CC/C=C/CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881716 CF On-Demand Mild ADRB1 45 37 CC/C=C/CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881716 CF On-Demand Mild ENPP1 61 31 C=CC(C)(C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881750 CF On-Demand Mild ADRB1 41 32 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881766 EE On-Demand Mild PDGFRB 23 40 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881766 EE On-Demand Mild EPHX2 23 40 C=C(CC)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881777 CF On-Demand Mild ADRB1 42 33 C=C(CC)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881777 CF On-Demand Mild ENPP1 61 33 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881823 ED On-Demand Mild HTR1B 15 48 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881823 ED On-Demand Mild PDGFRB 44 42 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881824 ED On-Demand Mild HTR1B 15 48 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881824 ED On-Demand Mild PDGFRB 44 42 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880881825 FE On-Demand Mild EPHX2 31 41 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](O)C(F)F ZINC000880881832 DE On-Demand Mild ADRB1 44 35 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](O)C(F)F ZINC000880881833 DE On-Demand Mild ADRB1 44 35 C#C[C@@](C)(CC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881860 CE On-Demand Mild IMDH_CRYPV 41 38 C#C[C@](C)(CC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881861 CE On-Demand Mild IMDH_CRYPV 41 38 CC[C@@](C)(CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880881893 CF On-Demand Mild ADRB1 41 32 CCCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881899 BE On-Demand Mild ADRB1 40 31 CCCONC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881899 BE On-Demand Mild ENPP1 66 31 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@@H]1c1ccccc1 ZINC000880881918 GF On-Demand Mild TSHR 40 30 COC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@H]1c1ccccc1 ZINC000880881919 GF On-Demand Mild TSHR 40 30 COC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881958 DF On-Demand Mild QRFPR 41 35 COC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881958 DF On-Demand Mild ACKR3 46 31 COC[C@@H]1CCCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880881958 DF On-Demand Mild PFKFB3 53 32 C#CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881967 CE On-Demand Mild HTR1B 15 45 C#CC1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880881967 CE On-Demand Mild PDGFRB 35 42 CCC1(CNC(=O)Nc2ccc(OC)c(C#N)c2)COC1 ZINC000880881982 CE On-Demand Mild ADRB1 41 32 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@@H](O)C(C)C ZINC000880882015 DE On-Demand Mild ADRB1 43 33 CC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)[C@H](O)C(C)C ZINC000880882016 DE On-Demand Mild ADRB1 43 33 COC[C@@]1(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882046 DE On-Demand Mild ENPP1 50 32 COC[C@]1(C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882047 DE On-Demand Mild ENPP1 50 32 O=C(Nc1ccccc1C(=O)NCc1cnn(-c2ccccc2)c1)c1ccc(Cl)cc1 ZINC000880882063 IJ On-Demand Anodyne F10 39 48 O=C(Nc1ccccc1C(=O)NCc1cnn(-c2ccccc2)c1)c1ccc(Cl)cc1 ZINC000880882063 IJ On-Demand Anodyne HDAC1 46 41 O=C(Nc1ccccc1C(=O)NCc1cnn(-c2ccccc2)c1)c1ccc(Cl)cc1 ZINC000880882063 IJ On-Demand Anodyne MAPK10 15 41 O=C(Nc1ccccc1C(=O)NCc1cnn(-c2ccccc2)c1)c1ccc(Cl)cc1 ZINC000880882063 IJ On-Demand Anodyne SCN10A 27 40 O=C(Nc1ccccc1C(=O)NCc1cnn(-c2ccccc2)c1)c1ccc(Cl)cc1 ZINC000880882063 IJ On-Demand Anodyne EPHB3 45 32 CCC[C@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880882109 CF On-Demand Mild ADRB1 45 35 CCC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880882110 CF On-Demand Mild ADRB1 45 35 CC[C@H](C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880882127 DF On-Demand Mild P2RY12 15 43 CC[C@H](C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880882127 DF On-Demand Mild PDGFRB 50 43 CC[C@H](C)N1CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880882127 DF On-Demand Mild NPY2R 22 40 CC[C@@H](C)[C@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880882139 DF On-Demand Mild ADRB1 45 35 CC[C@H](C)[C@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880882141 DF On-Demand Mild ADRB1 45 35 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882151 ED On-Demand Mild P2RY12 16 41 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882151 ED On-Demand Mild ENPP1 67 32 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882166 CF On-Demand Mild PDGFRB 44 41 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882166 CF On-Demand Mild QRFPR 40 33 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882167 CF On-Demand Mild PDGFRB 44 41 C#CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882167 CF On-Demand Mild QRFPR 40 33 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880882417 CF On-Demand Mild EPHX2 45 39 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882566 FE On-Demand Mild ACKR3 62 32 CCn1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C ZINC000880882592 CF On-Demand Mild HTR2A 41 43 CCn1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C ZINC000880882592 CF On-Demand Mild HTR2C 15 43 CCn1ncc(NC(=O)Nc2ccc(OC)c(C#N)c2)c1C ZINC000880882592 CF On-Demand Mild ENPP1 62 32 CCC[C@H](CCO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882738 CE On-Demand Mild ADRB1 40 30 CCC[C@@H](CCO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882739 CE On-Demand Mild ADRB1 40 30 CCC1(N2CCOCC2)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880882740 FF On-Demand Mild PDGFRB 31 40 COCc1csc(CNC(=O)Nc2ccc(OC)c(C#N)c2)c1 ZINC000880882755 EG On-Demand Mild ADRB1 41 32 C#CC[C@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882771 CD On-Demand Mild ADRB1 41 31 C#CC[C@@H](COC)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882772 CD On-Demand Mild ADRB1 41 31 CN1CCN(C2CCN(C(=O)Nc3nnc([C@@H]4CCCO4)s3)CC2)CC1 ZINC000880882838 GD On-Demand Anodyne L3MBTL3 46 39 CN1CCN(C2CCN(C(=O)Nc3nnc([C@H]4CCCO4)s3)CC2)CC1 ZINC000880882839 GD On-Demand Anodyne L3MBTL3 46 39 CCN1CC[C@@H]1CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882870 CD On-Demand Mild DRD2 35 43 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C[C@H]1C(F)(F)F ZINC000880882888 GF On-Demand Mild P2RY12 15 44 CCC[C@@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OCC ZINC000880882934 DF On-Demand Mild ADRB1 44 34 CCC[C@H](CNC(=O)Nc1ccc(OC)c(C#N)c1)OCC ZINC000880882935 DF On-Demand Mild ADRB1 44 34 COCC(C)(C)CCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880882969 DF On-Demand Mild ADRB1 45 35 C=CC[C@@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882971 CG On-Demand Mild PDGFRB 41 40 C=CC[C@H]1CCCN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880882972 CG On-Demand Mild PDGFRB 41 40 CCC1(N(C)C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880883078 EF On-Demand Mild HTR1B 17 45 CCC1(N(C)C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880883078 EF On-Demand Mild PDGFRB 40 40 CCC1(N(C)C)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880883078 EF On-Demand Mild ENPP1 60 32 CCOC(=O)[C@@H]1CN(C(=O)Nc2ccc(OC)c(C#N)c2)CCC1(F)F ZINC000880883129 FF On-Demand Mild P2RY12 15 41 COC[C@@H]1CCCN1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883154 DD On-Demand Mild CCR3 15 41 COC[C@@H]1CCCN1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883154 DD On-Demand Mild CASP7 40 34 COC[C@@H]1CCCN1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883154 DD On-Demand Mild QRFPR 40 33 COC[C@@H]1CCCN1NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883154 DD On-Demand Mild ACKR3 44 31 C=CCOCCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883239 CE On-Demand Mild ADRB1 45 34 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883332 FG On-Demand Mild ADRB1 45 38 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883332 FG On-Demand Mild ROCK2 15 46 COC[C@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883332 FG On-Demand Mild TAAR1 27 42 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883333 FG On-Demand Mild ADRB1 45 38 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883333 FG On-Demand Mild ROCK2 15 46 COC[C@@H](NC(=O)Nc1ccc(OC)c(C#N)c1)c1cccc(OC)c1 ZINC000880883333 FG On-Demand Mild TAAR1 27 42 CC[C@@H](O)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883406 CD On-Demand Mild ADRB1 54 43 COC[C@@H](CCNC(=O)Nc1ccc(OC)c(C#N)c1)OC ZINC000880883409 DD On-Demand Mild ADRB1 51 39 COCC1(NC(=O)Nc2ccc(OC)c(C#N)c2)CCCC1 ZINC000880883435 DF On-Demand Mild ENPP1 45 31 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880883443 DD On-Demand Mild PDGFRB 45 42 C#CCC1(O)CCN(C(=O)Nc2ccc(OC)c(C#N)c2)CC1 ZINC000880883443 DD On-Demand Mild S1PR2 29 43 O=C(N[C@@H]1CCC[C@@H]1c1ccccc1)c1cccnc1I ZINC000880883510 GH On-Demand Anodyne GRIA4 15 43 O=C(N[C@@H]1CCC[C@@H]1c1ccccc1)c1cccnc1I ZINC000880883510 GH On-Demand Anodyne EPHX2 16 41 O=C(N[C@@H]1CCC[C@@H]1c1ccccc1)c1cccnc1I ZINC000880883510 GH On-Demand Anodyne G2YM83_BOTF4 46 34 C=CCCSCCNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883533 DF On-Demand Mild ADRB1 43 34 CCc1nccn1C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883543 FG On-Demand Mild ENPP1 61 34 CCc1nccn1C[C@H]1CCCN1C(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883543 FG On-Demand Mild ACKR3 43 30 C#CC[C@H](CO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883548 CD On-Demand Mild ENPP1 54 31 C#CC[C@@H](CO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883549 CD On-Demand Mild ENPP1 54 31 CCC(F)(F)C(C)(C)CNC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880883582 EH On-Demand Mild ADRB1 41 33 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccc(OC)c(C#N)c3)CC2)c1 ZINC000880883630 GH On-Demand Mild TAAR1 29 41 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880883898 FH On-Demand Anodyne NPY5R 32 44 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880883899 FH On-Demand Anodyne NPY5R 32 44 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880883900 FH On-Demand Anodyne NPY5R 32 44 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880883901 FH On-Demand Anodyne NPY5R 32 44 C[C@H]1[C@H](C(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)CCN1C ZINC000880883943 CF On-Demand Anodyne GRIA4 16 44 C[C@@H]1[C@@H](C(=O)N[C@@H]2CCC[C@@H]2c2ccccc2)CCN1C ZINC000880883944 CF On-Demand Anodyne GRIA4 16 44 C=C(C)C[C@H](CO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880884098 CE On-Demand Mild ENPP1 62 32 C=C(C)C[C@@H](CO)NC(=O)Nc1ccc(OC)c(C#N)c1 ZINC000880884099 CE On-Demand Mild ENPP1 62 32 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880884130 GF On-Demand Anodyne EPHX2 15 46 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880884131 GF On-Demand Anodyne EPHX2 15 46 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880884132 GF On-Demand Anodyne EPHX2 15 46 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880884133 GF On-Demand Anodyne EPHX2 15 46 COc1ccc2cc(CNC(=O)Nc3nnc([C@@H]4CCCO4)s3)ccc2c1 ZINC000880884244 GH On-Demand Anodyne ROCK2 17 40 COc1ccc2cc(CNC(=O)Nc3nnc([C@H]4CCCO4)s3)ccc2c1 ZINC000880884247 GH On-Demand Anodyne ROCK2 17 40 O=C(NCc1cccc2ncccc12)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880884253 FG On-Demand Anodyne CDK5 30 45 O=C(NCc1cccc2ncccc12)Nc1nnc([C@H]2CCCO2)s1 ZINC000880884255 FG On-Demand Anodyne CDK5 30 45 COc1ccc(CN(C)C(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)cc1 ZINC000880884299 GH On-Demand Anodyne ROCK2 15 40 COc1cccc(OC)c1CNC(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880884327 GG On-Demand Anodyne ROCK2 19 48 COc1ccc(CN(CCO)C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880884391 FF On-Demand Mild BMP1 23 42 COc1ccc(CN(CCO)C(=O)Nc2ccc(OC)c(C#N)c2)cc1 ZINC000880884391 FF On-Demand Mild ROCK2 16 46 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC(c2ccc(F)cc2)CC1 ZINC000880884410 GH On-Demand Anodyne DGAT1 18 43 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC(c2ccc(F)cc2)CC1 ZINC000880884411 GH On-Demand Anodyne DGAT1 18 43 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880884466 EE On-Demand Mild P2RY12 17 41 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(OC)c(C#N)c2)C1 ZINC000880884466 EE On-Demand Mild ENPP1 57 33 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880884736 GI On-Demand Anodyne TRPM8 17 44 O=C1CC[C@H](c2ccc(C(=O)N[C@@H]3CCO[C@H]3c3ccc(F)c(F)c3)cc2)N1 ZINC000880884870 GG On-Demand Anodyne SSTR3 27 41 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H]3CCO[C@H]3c3ccc(F)c(F)c3)cc2)N1 ZINC000880884871 GG On-Demand Anodyne SSTR3 27 41 CN(C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2)[C@H](CO)Cc1ccccc1 ZINC000880885006 GG On-Demand Anodyne NPY5R 32 44 CN(C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2)[C@@H](CO)Cc1ccccc1 ZINC000880885007 GG On-Demand Anodyne NPY5R 32 44 O=C(NCCc1cccnc1)Nc1nnc([C@H]2CCCO2)s1 ZINC000880885035 DE On-Demand Anodyne NAMPT 37 44 O=C(NCCc1cccnc1)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880885036 DE On-Demand Anodyne NAMPT 37 44 CCCCCCCCNC(=O)Nc1nnc([C@H]2CCCO2)s1 ZINC000880885222 EH On-Demand Mild LASR 43 31 CCCCCCCCNC(=O)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880885223 EH On-Demand Mild LASR 43 31 CCNc1nc(C)c(C(=O)N[C@@H]2CCO[C@H]2c2ccccc2)s1 ZINC000880885230 EG On-Demand Anodyne SCD1 17 42 O=C(N[C@@H]1CCO[C@H]1c1ccc(Cl)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880885290 GG On-Demand Anodyne SIGMAR1 15 40 O=C(N[C@@H]1CCO[C@H]1c1ccc(Cl)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880885290 GG On-Demand Anodyne DPOL_VZVD 24 41 Cn1ncc(Br)c1CC(=O)N[C@@H]1CCO[C@H]1c1ccc(Cl)cc1 ZINC000880885360 GG On-Demand Anodyne P2RX7 16 41 COC(=O)c1cc(-c2csc(NC(=O)COc3ccc(-c4ccccc4)cc3)n2)c[nH]1 ZINC000880885563 IJ On-Demand Anodyne GABRA1 20 41 COC(=O)c1cc(-c2csc(NC(=O)COc3ccc(-c4ccccc4)cc3)n2)c[nH]1 ZINC000880885563 IJ On-Demand Anodyne ROCK1 29 41 COC(=O)c1cc(-c2csc(NC(=O)COc3ccc(-c4ccccc4)cc3)n2)c[nH]1 ZINC000880885563 IJ On-Demand Anodyne ROCK2 36 41 COC(=O)c1cc(-c2csc(NC(=O)COc3ccc(-c4ccccc4)cc3)n2)c[nH]1 ZINC000880885563 IJ On-Demand Anodyne TRPA1 15 44 O=C(COC1CC1)N[C@@H]1CCO[C@H]1c1ccc(Cl)cc1 ZINC000880885635 CE On-Demand Anodyne TRAR 21 41 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@@H](c2ccccc2)CC1 ZINC000880885650 FI On-Demand Anodyne DGAT1 21 45 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@@H](c2ccccc2)CC1 ZINC000880885650 FI On-Demand Anodyne MGEA5 25 40 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@H](c2ccccc2)CC1 ZINC000880885651 FI On-Demand Anodyne DGAT1 21 45 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCC[C@H](c2ccccc2)CC1 ZINC000880885651 FI On-Demand Anodyne MGEA5 25 40 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@@H](c2ccccc2)CC1 ZINC000880885652 FI On-Demand Anodyne DGAT1 21 45 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@@H](c2ccccc2)CC1 ZINC000880885652 FI On-Demand Anodyne MGEA5 25 40 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@H](c2ccccc2)CC1 ZINC000880885653 FI On-Demand Anodyne DGAT1 21 45 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCC[C@H](c2ccccc2)CC1 ZINC000880885653 FI On-Demand Anodyne MGEA5 25 40 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880885772 GG On-Demand Anodyne EPHX2 18 43 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880885772 GG On-Demand Anodyne TRPM8 27 45 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880885773 GG On-Demand Anodyne EPHX2 18 43 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880885773 GG On-Demand Anodyne TRPM8 27 45 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880885774 GG On-Demand Anodyne EPHX2 18 43 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880885774 GG On-Demand Anodyne TRPM8 27 45 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880885775 GG On-Demand Anodyne EPHX2 18 43 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880885775 GG On-Demand Anodyne TRPM8 27 45 O=C(NNc1ccc(OC(F)(F)F)cc1)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880885954 GG On-Demand Reactive EPHX2 41 42 O=C(NNc1ccc(OC(F)(F)F)cc1)Nc1nnc([C@H]2CCCO2)s1 ZINC000880885955 GG On-Demand Reactive EPHX2 41 42 O=C(Nc1nnc([C@H]2CCCO2)s1)NC12CCC(CC1)C2 ZINC000880886067 DF On-Demand Anodyne EPHX2 18 42 O=C(Nc1nnc([C@@H]2CCCO2)s1)NC12CCC(CC1)C2 ZINC000880886069 DF On-Demand Anodyne EPHX2 18 42 CNc1nc(C(=O)N[C@@H]2CCO[C@H]2c2ccc(Cl)cc2)cs1 ZINC000880886414 EG On-Demand Anodyne TRPC6 34 40 CNc1nc(C(=O)N[C@@H]2CCO[C@H]2c2ccc(Cl)cc2)cs1 ZINC000880886414 EG On-Demand Anodyne TRPC3 31 40 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCCC[C@@H]1c1ccccc1 ZINC000880886428 FI On-Demand Anodyne CPT1A 52 35 O=C(Nc1nnc([C@@H]2CCCO2)s1)N1CCCC[C@H]1c1ccccc1 ZINC000880886531 FI On-Demand Anodyne CPT1A 52 35 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCCC[C@@H]1c1ccccc1 ZINC000880886532 FI On-Demand Anodyne CPT1A 52 35 O=C(Nc1nnc([C@H]2CCCO2)s1)N1CCCC[C@H]1c1ccccc1 ZINC000880886533 FI On-Demand Anodyne CPT1A 52 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne PGC 46 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne PAPA1_CARPA 41 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne CCKAR 30 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne CTSK 21 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne CTSL 22 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne REN 57 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne CTSS 15 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886541 GF On-Demand Anodyne FPR1 49 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne PGC 46 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne PAPA1_CARPA 41 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne CCKAR 30 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne CTSK 21 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne CTSL 22 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne REN 57 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne CTSS 15 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880886542 GF On-Demand Anodyne FPR1 49 39 Cc1ccncc1CNC(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880886597 FG On-Demand Anodyne NAMPT 26 49 CC(=O)c1cccc(CNC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)c1 ZINC000880886608 GH On-Demand Anodyne ROCK2 23 43 COc1ccc(N2CCN(C(=O)Nc3nnc([C@@H]4CCCO4)s3)CC2)cc1 ZINC000880886685 GF On-Demand Clean NPBWR1 49 31 COc1ccc(N2CCN(C(=O)Nc3nnc([C@H]4CCCO4)s3)CC2)cc1 ZINC000880886686 GF On-Demand Clean NPBWR1 49 31 COC(=O)c1cc(-c2csc(NC(=O)[C@@H]3Cc4ccccc4CN3C(=O)c3ccccc3)n2)c[nH]1 ZINC000880886788 JI On-Demand Anodyne OPRD1 65 34 COC(=O)c1cc(-c2csc(NC(=O)[C@@H]3Cc4ccccc4CN3C(=O)c3ccccc3)n2)c[nH]1 ZINC000880886788 JI On-Demand Anodyne CFTR 81 45 C[C@@H]1[C@@H](C(=O)N[C@@H]2CCO[C@H]2c2ccc(Cl)cc2)CCN1C ZINC000880887000 DF On-Demand Anodyne SLC6A3 22 40 C[C@H]1[C@H](C(=O)N[C@@H]2CCO[C@H]2c2ccc(Cl)cc2)CCN1C ZINC000880887002 DF On-Demand Anodyne SLC6A3 22 40 O=C(NCc1ccc2ccccc2c1)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880887102 FH On-Demand Anodyne NMT1 38 42 O=C(NCc1ccc2ccccc2c1)Nc1nnc([C@H]2CCCO2)s1 ZINC000880887103 FH On-Demand Anodyne NMT1 38 42 O=C(NCc1ccc(-n2ccnc2)cc1)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880887133 FF On-Demand Anodyne NOS2 42 33 O=C(NCc1ccc(-n2ccnc2)cc1)Nc1nnc([C@H]2CCCO2)s1 ZINC000880887134 FF On-Demand Anodyne NOS2 42 33 COC(=O)c1cc(-c2csc(NC(=O)C(O)(c3ccccc3)c3ccccc3)n2)c[nH]1 ZINC000880887138 IH On-Demand Anodyne GABRA1 22 43 COC(=O)c1cc(-c2csc(NC(=O)C(O)(c3ccccc3)c3ccccc3)n2)c[nH]1 ZINC000880887138 IH On-Demand Anodyne ROCK1 20 41 COC(=O)c1cc(-c2csc(NC(=O)C(O)(c3ccccc3)c3ccccc3)n2)c[nH]1 ZINC000880887138 IH On-Demand Anodyne ROCK2 16 41 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1nnc([C@@H]2CCCO2)s1 ZINC000880887156 GG On-Demand Anodyne CCR3 50 35 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1nnc([C@H]2CCCO2)s1 ZINC000880887157 GG On-Demand Anodyne CCR3 50 35 CC1(C)CCN(C(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880887963 EH On-Demand Anodyne TRPM8 19 40 Cc1cncc(CNC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)c1 ZINC000880888186 FG On-Demand Anodyne NAMPT 35 49 O=C(NCC[C@@H]1CCSC1)c1n[nH]c2ccc(Cl)cc12 ZINC000880888798 DG On-Demand Anodyne ALPL 62 37 O=C(NCC[C@H]1CCSC1)c1n[nH]c2ccc(Cl)cc12 ZINC000880888799 DG On-Demand Anodyne ALPL 62 37 C=CCNc1ncc(C(=O)NCC[C@H]2CCSC2)s1 ZINC000880888808 CF On-Demand Mild SIRT3 40 32 C=CCNc1ncc(C(=O)NCC[C@H]2CCSC2)s1 ZINC000880888808 CF On-Demand Mild SIRT1 40 32 C=CCNc1ncc(C(=O)NCC[C@@H]2CCSC2)s1 ZINC000880888809 CF On-Demand Mild SIRT3 40 32 C=CCNc1ncc(C(=O)NCC[C@@H]2CCSC2)s1 ZINC000880888809 CF On-Demand Mild SIRT1 40 32 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)C1 ZINC000880889102 FE On-Demand Anodyne EPHX2 33 52 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)C1 ZINC000880889103 FE On-Demand Anodyne EPHX2 33 52 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA2 42 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA1 37 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA7 46 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA5B 49 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA4 43 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889145 ED On-Demand Anodyne CA5A 51 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA2 42 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA1 37 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA7 46 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA5B 49 40 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA4 43 41 NS(=O)(=O)c1ccc(Cl)c(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889146 ED On-Demand Anodyne CA5A 51 40 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880889259 GH On-Demand Anodyne NPY5R 21 43 C[C@@H]1CCCN(C(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)[C@@H]1C ZINC000880889288 EH On-Demand Anodyne TRPC6 50 39 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880889289 EH On-Demand Anodyne TRPC6 50 39 CCCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889439 GG On-Demand Anodyne EPHX2 38 41 CCCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889439 GG On-Demand Anodyne CXCR3 21 45 CCCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889439 GG On-Demand Anodyne MCHR1 15 40 Cn1cc(CNC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)cn1 ZINC000880889577 EE On-Demand Anodyne NAMPT 29 40 O=C(NCC[C@@H]1CCSC1)c1ccnc(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889585 GF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@@H]1CCSC1)c1ccnc(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889585 GF On-Demand Anodyne SIRT1 41 34 O=C(NCC[C@H]1CCSC1)c1ccnc(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889586 GF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@H]1CCSC1)c1ccnc(C(=O)NCC[C@H]2CCSC2)c1 ZINC000880889586 GF On-Demand Anodyne SIRT1 41 34 O=C(NCC[C@@H]1CCSC1)c1ccnc(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889587 GF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@@H]1CCSC1)c1ccnc(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889587 GF On-Demand Anodyne SIRT1 41 34 O=C(NCC[C@H]1CCSC1)c1ccnc(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889588 GF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@H]1CCSC1)c1ccnc(C(=O)NCC[C@@H]2CCSC2)c1 ZINC000880889588 GF On-Demand Anodyne SIRT1 41 34 CNc1ncc(C(=O)NCC[C@@H]2CCSC2)s1 ZINC000880889609 CE On-Demand Anodyne SIRT3 43 35 CNc1ncc(C(=O)NCC[C@@H]2CCSC2)s1 ZINC000880889609 CE On-Demand Anodyne SIRT2 47 35 CNc1ncc(C(=O)NCC[C@@H]2CCSC2)s1 ZINC000880889609 CE On-Demand Anodyne SIRT1 43 35 CNc1ncc(C(=O)NCC[C@H]2CCSC2)s1 ZINC000880889610 CE On-Demand Anodyne SIRT3 43 35 CNc1ncc(C(=O)NCC[C@H]2CCSC2)s1 ZINC000880889610 CE On-Demand Anodyne SIRT2 47 35 CNc1ncc(C(=O)NCC[C@H]2CCSC2)s1 ZINC000880889610 CE On-Demand Anodyne SIRT1 43 35 C=C(C)CN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889661 GG On-Demand Mild CXCR3 21 41 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne DRD4 19 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne DRD3 20 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne HDAC1 26 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne HDAC2 22 40 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne MAPK10 17 44 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCc2cnn(-c3ccccc3)c2)cc1OC ZINC000880889730 JI On-Demand Anodyne ABCG2 41 39 CC(C)CN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889851 GG On-Demand Anodyne EPHX2 32 41 CC(C)CN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880889851 GG On-Demand Anodyne CXCR3 21 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(OC2CCC2)CC1 ZINC000880889960 FJ On-Demand Anodyne EPHX2 17 44 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](c2cccnc2)C1 ZINC000880889970 FJ On-Demand Anodyne RBP4 43 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](c2cccnc2)C1 ZINC000880889971 FJ On-Demand Anodyne RBP4 43 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](CO)C1 ZINC000880890002 DF On-Demand Anodyne CACNA1I 50 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](CO)C1 ZINC000880890003 DF On-Demand Anodyne CACNA1I 50 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC(C(F)(F)F)C1 ZINC000880890034 EI On-Demand Anodyne RBP4 52 36 CN(CCN1CCOCC1)C(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880890123 GD On-Demand Anodyne CASR 47 41 NC(=O)[C@@H]1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890168 FH On-Demand Anodyne CACNA1I 47 34 NC(=O)C1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890182 FD On-Demand Anodyne CACNA1H 61 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880890212 EH On-Demand Anodyne PTGES 18 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCC[C@@H](CO)C1 ZINC000880890213 EH On-Demand Anodyne PTGES 18 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCC[C@H](CO)C1 ZINC000880890214 EH On-Demand Anodyne PTGES 18 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCC[C@H](CO)C1 ZINC000880890215 EH On-Demand Anodyne PTGES 18 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880890216 GH On-Demand Anodyne CHRNA4 26 46 COCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880890330 GE On-Demand Anodyne EPHX2 41 39 COCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880890330 GE On-Demand Anodyne CXCR3 21 44 COCCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880890330 GE On-Demand Anodyne MCHR1 20 43 C[C@@H]1CN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CCC1(F)F ZINC000880890364 EJ On-Demand Anodyne CACNA1H 49 38 C[C@H]1CN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CCC1(F)F ZINC000880890365 EJ On-Demand Anodyne CACNA1H 49 38 CS(=O)(=O)CC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890382 GG On-Demand Anodyne EPHX2 15 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCc2nnnn2CC1 ZINC000880890422 FF On-Demand Anodyne EPHX2 18 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCc2nnnn2CC1 ZINC000880890423 FF On-Demand Anodyne EPHX2 18 40 CN1CC[C@@]2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C2)C1 ZINC000880890425 EH On-Demand Anodyne CACNA1H 38 40 O=C(NCC[C@@H]1CCSC1)c1cccnc1I ZINC000880890470 FF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@@H]1CCSC1)c1cccnc1I ZINC000880890470 FF On-Demand Anodyne SIRT1 41 34 O=C(NCC[C@H]1CCSC1)c1cccnc1I ZINC000880890471 FF On-Demand Anodyne SIRT3 41 34 O=C(NCC[C@H]1CCSC1)c1cccnc1I ZINC000880890471 FF On-Demand Anodyne SIRT1 41 34 COC[C@@]1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890525 EI On-Demand Anodyne CACNA1H 48 36 COC[C@]1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890527 EI On-Demand Anodyne CACNA1H 48 36 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890538 FE On-Demand Anodyne EPHX2 40 46 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890540 FE On-Demand Anodyne EPHX2 40 46 C=CCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880890547 FF On-Demand Mild CXCR3 21 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cc(Cl)cc(Cl)c1F)C2 ZINC000880890550 EH On-Demand Anodyne HTR3A 15 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cc(Cl)cc(Cl)c1F)C2 ZINC000880890550 EH On-Demand Anodyne SLC6A3 26 40 COC1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890556 EI On-Demand Anodyne CACNA1H 66 38 COC1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890556 EI On-Demand Anodyne RBP4 19 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H](F)C1 ZINC000880890574 DI On-Demand Anodyne DPP7 15 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H](F)C1 ZINC000880890575 DI On-Demand Anodyne DPP7 15 45 C[C@@H](CO)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890624 EI On-Demand Anodyne CACNA1H 55 37 CN1C(=O)N[C@]2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C2)C1=O ZINC000880890625 GE On-Demand Anodyne CACNA1H 46 39 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C2)C1=O ZINC000880890626 GE On-Demand Anodyne CACNA1H 46 39 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CCNC2=O)CC1 ZINC000880890700 FG On-Demand Anodyne CACNA1H 69 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@H]2COC[C@H]2C1 ZINC000880890707 DG On-Demand Anodyne RBP4 46 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCc2nc(C3CC3)ncc2C1 ZINC000880890741 GI On-Demand Anodyne MAPK1 50 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880890742 GI On-Demand Anodyne RBP4 25 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880890743 GI On-Demand Anodyne RBP4 25 40 O=C(NCC[C@@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890744 CF On-Demand Anodyne SIRT3 43 36 O=C(NCC[C@@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890744 CF On-Demand Anodyne SIRT2 41 36 O=C(NCC[C@@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890744 CF On-Demand Anodyne SIRT1 43 36 O=C(NCC[C@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890745 CF On-Demand Anodyne SIRT3 43 36 O=C(NCC[C@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890745 CF On-Demand Anodyne SIRT2 41 36 O=C(NCC[C@H]1CCSC1)c1cnc(CC2CC2)s1 ZINC000880890745 CF On-Demand Anodyne SIRT1 43 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(COC2)C1 ZINC000880890766 DG On-Demand Anodyne CACNA1H 47 37 CO[C@]1(CO)CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890777 FG On-Demand Anodyne EPHX2 15 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CC[C@@H](O)CC1 ZINC000880890842 DH On-Demand Anodyne EPHX2 25 46 O=C(NCCN1CCCC1=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880890853 EF On-Demand Anodyne CACNA1H 19 40 CN1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1=O ZINC000880890854 DE On-Demand Anodyne P2RX7 15 52 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CC1)OCCO2 ZINC000880890860 EH On-Demand Anodyne CACNA1H 45 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCCC(F)(F)CC1 ZINC000880890897 EJ On-Demand Anodyne CACNA1H 50 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](CF)C1 ZINC000880890899 DH On-Demand Anodyne CACNA1I 51 34 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](CF)C1 ZINC000880890900 DH On-Demand Anodyne CACNA1I 51 34 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880890902 FE On-Demand Anodyne CACNA1H 44 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(CO)(CO)CC1 ZINC000880890911 FF On-Demand Anodyne CACNA1H 56 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(CO)(CO)C1 ZINC000880890923 EE On-Demand Anodyne CACNA1H 41 36 O=C(NCCN1CC[C@@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890938 EE On-Demand Anodyne CACNA1H 21 43 O=C(NCCN1CC[C@@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890938 EE On-Demand Anodyne PLD1 44 36 O=C(NCCN1CC[C@@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890938 EE On-Demand Anodyne PLD2 40 36 O=C(NCCN1CC[C@@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890938 EE On-Demand Anodyne CACNA1I 46 34 O=C(NCCN1CC[C@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890939 EE On-Demand Anodyne CACNA1H 21 43 O=C(NCCN1CC[C@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890939 EE On-Demand Anodyne PLD1 44 36 O=C(NCCN1CC[C@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890939 EE On-Demand Anodyne PLD2 40 36 O=C(NCCN1CC[C@H](O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880890939 EE On-Demand Anodyne CACNA1I 46 34 O=C(NCC[C@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890940 DE On-Demand Anodyne SIRT3 57 39 O=C(NCC[C@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890940 DE On-Demand Anodyne SIRT2 63 39 O=C(NCC[C@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890940 DE On-Demand Anodyne SIRT1 58 39 O=C(NCC[C@@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890941 DE On-Demand Anodyne SIRT3 57 39 O=C(NCC[C@@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890941 DE On-Demand Anodyne SIRT2 63 39 O=C(NCC[C@@H]1CCSC1)c1ccc2c(O)ncnc2c1 ZINC000880890941 DE On-Demand Anodyne SIRT1 58 39 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(F)(F)CC1 ZINC000880890947 EI On-Demand Anodyne CACNA1H 70 40 O=C(NCC[C@@H]1CCSC1)c1cc(C(F)(F)F)ccn1 ZINC000880890957 DF On-Demand Anodyne SIRT3 41 31 O=C(NCC[C@@H]1CCSC1)c1cc(C(F)(F)F)ccn1 ZINC000880890957 DF On-Demand Anodyne SIRT1 41 31 O=C(NCC[C@H]1CCSC1)c1cc(C(F)(F)F)ccn1 ZINC000880890958 DF On-Demand Anodyne SIRT3 41 31 O=C(NCC[C@H]1CCSC1)c1cc(C(F)(F)F)ccn1 ZINC000880890958 DF On-Demand Anodyne SIRT1 41 31 O=C(NCC[C@H]1CCSC1)c1cnc2cc[nH]c2c1 ZINC000880890961 CE On-Demand Anodyne SIRT3 41 33 O=C(NCC[C@H]1CCSC1)c1cnc2cc[nH]c2c1 ZINC000880890961 CE On-Demand Anodyne SIRT1 41 33 O=C(NCC[C@@H]1CCSC1)c1cnc2cc[nH]c2c1 ZINC000880890962 CE On-Demand Anodyne SIRT3 41 33 O=C(NCC[C@@H]1CCSC1)c1cnc2cc[nH]c2c1 ZINC000880890962 CE On-Demand Anodyne SIRT1 41 33 CO[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880890977 EI On-Demand Anodyne RBP4 21 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC(C2CC2)C1 ZINC000880890999 DI On-Demand Anodyne RBP4 46 37 CNS(=O)(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891003 GF On-Demand Anodyne RBP4 28 40 Cn1cnnc1N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891012 FF On-Demand Anodyne RBP4 17 40 Cn1cccc1C(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891013 GG On-Demand Anodyne RBP4 17 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2nccnn2)CC1 ZINC000880891015 FF On-Demand Anodyne FAAH 24 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2nccnn2)CC1 ZINC000880891015 FF On-Demand Anodyne RBP4 17 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880891055 GH On-Demand Anodyne L3MBTL3 55 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880891056 GH On-Demand Anodyne L3MBTL3 55 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCOC1=O ZINC000880891089 DF On-Demand Anodyne LUXR 75 44 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCOC1=O ZINC000880891089 DF On-Demand Anodyne TRAR 88 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCOC1=O ZINC000880891089 DF On-Demand Anodyne LASR 61 38 COC1(C(F)(F)F)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891183 GJ On-Demand Anodyne CACNA1H 68 37 COC1(C(F)(F)F)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891183 GJ On-Demand Anodyne RBP4 24 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCNC1=O ZINC000880891195 DE On-Demand Anodyne GRIN1 21 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCNC1=O ZINC000880891196 DE On-Demand Anodyne GRIN1 21 40 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880891199 FF On-Demand Anodyne CACNA1H 40 36 CC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891202 EH On-Demand Anodyne EPHX2 16 40 CC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891202 EH On-Demand Anodyne RBP4 23 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880891208 EH On-Demand Anodyne RBP4 41 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880891210 EH On-Demand Anodyne RBP4 41 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880891211 EH On-Demand Anodyne RBP4 41 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880891213 EH On-Demand Anodyne RBP4 41 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880891214 EH On-Demand Anodyne RBP4 41 38 COC1(CO)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891230 FG On-Demand Anodyne CACNA1H 67 37 COC[C@]1(CO)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880891241 FF On-Demand Anodyne CACNA1H 41 35 O=C(NCC1CCC(O)CC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880891249 EH On-Demand Anodyne CACNA1I 51 36 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC[S@]1=O ZINC000880891261 FH On-Demand Anodyne CACNA1H 45 37 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC[S@@]1=O ZINC000880891263 FH On-Demand Anodyne CACNA1H 45 37 CON(C)C(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891267 GG On-Demand Anodyne RBP4 21 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880891339 FI On-Demand Anodyne CPT1A 40 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880891340 FI On-Demand Anodyne CPT1A 40 35 CN(C)C1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891351 EI On-Demand Anodyne EPHX2 32 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880891378 GI On-Demand Anodyne CACNA1H 50 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880891378 GI On-Demand Anodyne EPHX2 28 49 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880891379 GI On-Demand Anodyne CACNA1H 50 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880891379 GI On-Demand Anodyne EPHX2 28 49 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891386 GI On-Demand Anodyne EPHX2 51 47 COC(=O)c1cc(-c2csc(NC(=O)Cn3cnc4sc(-c5ccccc5)cc4c3=O)n2)c[nH]1 ZINC000880891419 JI On-Demand Anodyne TRPA1 16 52 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(F)CC1 ZINC000880891503 DI On-Demand Anodyne RBP4 25 40 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CCSC1 ZINC000880891506 EE On-Demand Anodyne PAPA1_CARPA 36 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@@H]1CCSC1 ZINC000880891507 EE On-Demand Anodyne PAPA1_CARPA 36 44 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CCSC1 ZINC000880891508 EE On-Demand Anodyne PAPA1_CARPA 36 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC[C@H]1CCSC1 ZINC000880891509 EE On-Demand Anodyne PAPA1_CARPA 36 44 O=C(NCC1CSC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880891526 DH On-Demand Anodyne CACNA1I 45 33 O=C(NCC[C@@H]1CCSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880891529 EH On-Demand Anodyne PDE4D 16 44 O=C(NCC[C@@H]1CCSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880891529 EH On-Demand Anodyne CACNA1I 41 34 O=C(NCC[C@H]1CCSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880891530 EH On-Demand Anodyne PDE4D 16 44 O=C(NCC[C@H]1CCSC1)c1ccc(OC(F)F)c(Cl)c1 ZINC000880891530 EH On-Demand Anodyne CACNA1I 41 34 CONC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891533 FG On-Demand Anodyne EPHX2 18 42 CONC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891533 FG On-Demand Anodyne RBP4 21 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC(CNC(=O)C(F)(F)F)C1 ZINC000880891543 GG On-Demand Anodyne CACNA1I 46 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H](CF)C1 ZINC000880891555 DI On-Demand Anodyne CACNA1I 40 31 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H](CF)C1 ZINC000880891556 DI On-Demand Anodyne CACNA1I 40 31 CS(=O)(=O)NCC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891571 GF On-Demand Anodyne CACNA1I 52 34 COC(=O)N1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891585 FG On-Demand Anodyne EPHX2 53 49 CO[C@@]1(C)CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891592 EJ On-Demand Anodyne CACNA1H 54 36 N#CC1(c2ccccn2)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891643 GJ On-Demand Mild CACNA1H 55 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CC1)COCCO2 ZINC000880891731 FH On-Demand Anodyne TRPM8 23 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CC[C@H](O)CC1 ZINC000880891733 DH On-Demand Anodyne EPHX2 25 46 O=C(NCC[C@@H]1CCSC1)c1ncccc1-c1ccccn1 ZINC000880891770 DG On-Demand Anodyne SIRT3 42 33 O=C(NCC[C@@H]1CCSC1)c1ncccc1-c1ccccn1 ZINC000880891770 DG On-Demand Anodyne SIRT1 42 33 O=C(NCC[C@H]1CCSC1)c1ncccc1-c1ccccn1 ZINC000880891771 DG On-Demand Anodyne SIRT3 42 33 O=C(NCC[C@H]1CCSC1)c1ncccc1-c1ccccn1 ZINC000880891771 DG On-Demand Anodyne SIRT1 42 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CCCC2=O)CC1 ZINC000880891775 FI On-Demand Anodyne CACNA1H 55 38 O=C(NCC[C@@H]1CCSC1)c1coc(-c2ccccn2)n1 ZINC000880891785 DF On-Demand Anodyne TBXA2R 28 40 O=C(NCC[C@H]1CCSC1)c1coc(-c2ccccn2)n1 ZINC000880891786 DF On-Demand Anodyne TBXA2R 28 40 O=C1NCC2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)O1 ZINC000880891802 FG On-Demand Anodyne CACNA1H 51 36 O=C1NCC2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)O1 ZINC000880891802 FG On-Demand Anodyne TRPM8 26 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](CN2CCOCC2)C1 ZINC000880891830 GG On-Demand Anodyne CACNA1I 42 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880891831 GG On-Demand Anodyne CACNA1I 42 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880891845 GJ On-Demand Anodyne RBP4 32 40 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CCS1(=O)=O ZINC000880891857 GH On-Demand Anodyne CACNA1H 46 37 COC(=O)C1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891861 FF On-Demand Anodyne CACNA1H 69 38 COC(=O)C1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880891861 FF On-Demand Anodyne RBP4 19 40 O=C(NC[C@@H]1CCn2ccnc2C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880891865 FH On-Demand Anodyne CACNA1I 54 35 O=C(NC[C@H]1CCn2ccnc2C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880891866 FH On-Demand Anodyne CACNA1I 54 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(F)(F)C1 ZINC000880891890 DI On-Demand Anodyne CACNA1H 46 38 O=C(NCC[C@H]1CCSC1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880891905 FH On-Demand Anodyne SIRT3 42 33 O=C(NCC[C@H]1CCSC1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880891905 FH On-Demand Anodyne SIRT1 42 33 O=C(NCC[C@@H]1CCSC1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880891906 FH On-Demand Anodyne SIRT3 42 33 O=C(NCC[C@@H]1CCSC1)c1cc2cccc(C(F)(F)F)c2nc1O ZINC000880891906 FH On-Demand Anodyne SIRT1 42 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(c2ccon2)CC1 ZINC000880891928 FJ On-Demand Anodyne SMO 16 42 C[C@@H](O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892001 EH On-Demand Anodyne CACNA1H 49 37 O=C(CC[C@H]1CCc2ccccc21)NCC[C@@H]1CCSC1 ZINC000880892005 DH On-Demand Anodyne NQO2 19 44 O=C(CC[C@H]1CCc2ccccc21)NCC[C@H]1CCSC1 ZINC000880892007 DH On-Demand Anodyne NQO2 19 44 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@H]1CCSC1 ZINC000880892009 DH On-Demand Anodyne NQO2 19 44 O=C(CC[C@@H]1CCc2ccccc21)NCC[C@@H]1CCSC1 ZINC000880892011 DH On-Demand Anodyne NQO2 19 44 O=C(NCCCO)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892043 GF On-Demand Anodyne EPHX2 16 45 O=C(NCCCCCCO)Nc1cc(Cl)cc(Cl)c1F ZINC000880892054 DH On-Demand Anodyne ALPL 29 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@@]2(CCOC2)C1 ZINC000880892076 EG On-Demand Anodyne EPHX2 17 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@]2(CCOC2)C1 ZINC000880892077 EG On-Demand Anodyne EPHX2 17 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(O)(C(F)F)CC1 ZINC000880892098 FH On-Demand Anodyne CACNA1H 55 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(CCO)(CCO)CC1 ZINC000880892149 GH On-Demand Anodyne CACNA1H 41 36 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCSC1)C2 ZINC000880892150 DG On-Demand Anodyne NQO2 32 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCSC1)C2 ZINC000880892150 DG On-Demand Anodyne MTNR1A 43 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@H]1CCSC1)C2 ZINC000880892150 DG On-Demand Anodyne MTNR1B 35 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCSC1)C2 ZINC000880892151 DG On-Demand Anodyne NQO2 32 45 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCSC1)C2 ZINC000880892151 DG On-Demand Anodyne MTNR1A 43 44 COc1ccc2c(c1)CC[C@H](C(=O)NCC[C@@H]1CCSC1)C2 ZINC000880892151 DG On-Demand Anodyne MTNR1B 35 44 CN1CCN(C(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880892156 ED On-Demand Anodyne HTR1B 16 42 CCCCCNC(=O)Nc1ccc2c(c1)NC(=O)C(C)(C)CO2 ZINC000880892166 DG On-Demand Anodyne ASAH1 51 31 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(O)(CO)CC1 ZINC000880892171 EE On-Demand Anodyne CACNA1H 53 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(O)(CO)CC1 ZINC000880892171 EE On-Demand Anodyne S1PR2 26 42 CN1C[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1=O ZINC000880892172 EF On-Demand Anodyne CACNA1I 52 33 CN1C[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1=O ZINC000880892174 EF On-Demand Anodyne CACNA1I 52 33 C[S@](=N)(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892192 FF On-Demand Anodyne RBP4 23 41 CN1CCO[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892212 EF On-Demand Anodyne CACNA1I 41 32 CN1CCO[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892213 EF On-Demand Anodyne CACNA1I 41 32 O=C(NCc1ccsc1C(F)(F)F)c1ncsc1C1CC1 ZINC000880892224 EI On-Demand Anodyne MAP1 56 35 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880892232 GH On-Demand Anodyne CACNA1H 71 42 CN1CCN(C2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)CC1 ZINC000880892250 GG On-Demand Anodyne L3MBTL3 58 39 CSc1nccnc1C(=O)NCc1ccsc1C(F)(F)F ZINC000880892270 EG On-Demand Anodyne MAP1 55 33 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880892295 FH On-Demand Anodyne SLC6A4 30 44 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880892295 FH On-Demand Anodyne SLC6A3 50 41 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880892298 FH On-Demand Anodyne SLC6A4 30 44 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880892298 FH On-Demand Anodyne SLC6A3 50 41 CC(C)(C(N)=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892302 GF On-Demand Anodyne RBP4 17 42 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892307 EH On-Demand Anodyne CACNA1H 44 37 O=C(NCC[C@H]1CCSC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880892384 DF On-Demand Anodyne GABRA1 15 46 O=C(NCC[C@@H]1CCSC1)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880892387 DF On-Demand Anodyne GABRA1 15 46 CCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880892397 FF On-Demand Anodyne EPHX2 36 43 CCN1CCC(NC(=O)Nc2ccc3c(c2)NC(=O)C(C)(C)CO3)CC1 ZINC000880892397 FF On-Demand Anodyne CXCR3 22 43 O=C(NCCO)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892412 GE On-Demand Anodyne EPHX2 20 48 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880892427 DI On-Demand Anodyne RBP4 56 39 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H]2C[C@@H]2C1 ZINC000880892428 DI On-Demand Anodyne RBP4 56 39 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H]2C[C@H]2C1 ZINC000880892429 DI On-Demand Anodyne RBP4 56 39 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H]2C[C@H]2C1 ZINC000880892430 DI On-Demand Anodyne RBP4 56 39 C[C@@H](Cn1cncn1)NC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880892464 EF On-Demand Anodyne HIS3 83 37 O=C(NCCN1CCCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880892487 FF On-Demand Anodyne EPHX2 22 49 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCOC2(CCC2)C1 ZINC000880892489 EH On-Demand Anodyne EPHX2 21 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](CN2CCCC2)C1 ZINC000880892504 FI On-Demand Anodyne CACNA1I 54 33 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](CN2CCCC2)C1 ZINC000880892505 FI On-Demand Anodyne CACNA1I 54 33 CN(C)C[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892521 EH On-Demand Anodyne CACNA1I 60 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2ncc(F)cn2)CC1 ZINC000880892523 GG On-Demand Anodyne RBP4 17 40 COC[C@@H]1CCCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892533 EI On-Demand Anodyne RBP4 21 40 COC[C@@H]1CCCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892533 EI On-Demand Anodyne CACNA1I 42 32 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CCO2)CC1 ZINC000880892541 EH On-Demand Anodyne CACNA1H 45 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC2(CCO2)CC1 ZINC000880892541 EH On-Demand Anodyne TRPM8 25 42 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892555 FH On-Demand Anodyne CACNA1H 15 42 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892555 FH On-Demand Anodyne CACNA1I 72 37 CC(=O)N1CCC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892556 FH On-Demand Anodyne CACNA1H 15 42 CC(=O)N1CCC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892556 FH On-Demand Anodyne CACNA1I 72 37 CN(CCO)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892567 FG On-Demand Anodyne RBP4 27 40 C[C@]1(O)CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892569 DH On-Demand Anodyne EPHX2 15 42 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880892586 GH On-Demand Anodyne CACNA1H 57 36 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880892587 GH On-Demand Anodyne CACNA1H 57 36 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880892588 GH On-Demand Anodyne CACNA1H 57 36 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880892589 GH On-Demand Anodyne CACNA1H 57 36 O=C1NC2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)CO1 ZINC000880892590 FG On-Demand Anodyne CACNA1H 51 36 CC1(CO)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892603 EH On-Demand Anodyne CACNA1H 66 39 COCCO[C@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892609 FG On-Demand Anodyne CACNA1I 40 31 COCCO[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892610 FG On-Demand Anodyne CACNA1I 40 31 Cn1cnc2c1CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)C2 ZINC000880892634 EG On-Demand Anodyne MAPK1 42 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCOC2(CCOCC2)CC1 ZINC000880892657 GH On-Demand Anodyne EPHX2 15 40 CCC1(CO)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892679 EI On-Demand Anodyne CACNA1H 67 37 Cc1nc(CCNC(=O)Nc2cc(Cl)cc(Cl)c2F)n[nH]1 ZINC000880892687 EF On-Demand Anodyne ALPL 45 34 O=C(NCCCCO)Nc1cc(Cl)cc(Cl)c1F ZINC000880892699 CG On-Demand Anodyne ALPL 29 41 O=C(NC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1)C1CC1 ZINC000880892748 FH On-Demand Anodyne EPHX2 39 46 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892749 GG On-Demand Anodyne EPHX2 36 44 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880892750 GG On-Demand Anodyne EPHX2 36 44 CN1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892759 DG On-Demand Anodyne HRH4 15 46 CN1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892759 DG On-Demand Anodyne RBP4 15 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCCOCC1 ZINC000880892772 DH On-Demand Anodyne EPHX2 16 47 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCCOCC1 ZINC000880892773 DH On-Demand Anodyne EPHX2 16 47 C[C@]1(O)CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892774 EH On-Demand Anodyne CACNA1H 52 38 O=C1NC(=O)N2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C[C@H]12 ZINC000880892780 FD On-Demand Anodyne CACNA1H 44 37 O=C1NC(=O)N2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C[C@H]12 ZINC000880892780 FD On-Demand Anodyne SMO 23 41 O=C1NC(=O)N2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C[C@@H]12 ZINC000880892781 FD On-Demand Anodyne CACNA1H 44 37 O=C1NC(=O)N2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)C[C@@H]12 ZINC000880892781 FD On-Demand Anodyne SMO 23 41 C[C@H](O)CN1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892788 FF On-Demand Anodyne CACNA1H 47 39 CN1C(=O)NC2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)C1=O ZINC000880892892 GF On-Demand Anodyne CACNA1H 67 42 C#CCNC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892937 FG On-Demand Mild EPHX2 20 43 C#CCNC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880892937 FG On-Demand Mild CACNA1I 43 30 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@@]2(CCCOC2)C1 ZINC000880892940 FH On-Demand Anodyne EPHX2 18 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCO[C@]2(CCCOC2)C1 ZINC000880892941 FH On-Demand Anodyne EPHX2 18 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCn2c(O)nnc2C1 ZINC000880892973 EE On-Demand Anodyne P2RX7 29 44 C[C@H]1C[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CCO1 ZINC000880893031 EI On-Demand Anodyne CACNA1I 40 31 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](c2ccccn2)C1 ZINC000880893060 FJ On-Demand Anodyne CACNA1H 51 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](c2ccccn2)C1 ZINC000880893060 FJ On-Demand Anodyne EPHX2 19 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](c2ccccn2)C1 ZINC000880893060 FJ On-Demand Anodyne RBP4 57 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](c2ccccn2)C1 ZINC000880893061 FJ On-Demand Anodyne CACNA1H 51 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](c2ccccn2)C1 ZINC000880893061 FJ On-Demand Anodyne EPHX2 19 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](c2ccccn2)C1 ZINC000880893061 FJ On-Demand Anodyne RBP4 57 41 CN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893063 DG On-Demand Anodyne CACNA1H 15 41 CN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893063 DG On-Demand Anodyne CACNA1I 81 41 CN1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893064 DG On-Demand Anodyne CACNA1H 15 41 CN1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893064 DG On-Demand Anodyne CACNA1I 81 41 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cc(Cl)cc(Cl)c1F ZINC000880893081 GH On-Demand Anodyne PIK3CD 33 41 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cc(Cl)cc(Cl)c1F ZINC000880893081 GH On-Demand Anodyne PIK3CB 63 41 O=C(CNC(=O)Nc1cc(Cl)cc(Cl)c1F)NCC1CC1 ZINC000880893138 EF On-Demand Anodyne CACNA1I 51 36 O=C(NCCCCCO)Nc1cc(Cl)cc(Cl)c1F ZINC000880893143 DG On-Demand Anodyne ALPL 29 40 N#CCCN(CCN1CCOCC1)C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880893174 GG On-Demand Mild CASR 57 43 CCc1nnc2n1CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)C2 ZINC000880893218 FG On-Demand Anodyne P2RX7 27 48 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880893235 EH On-Demand Anodyne EPHX2 22 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CC[C@H](CO)CC1 ZINC000880893236 EH On-Demand Anodyne EPHX2 22 43 C[C@H]1C[C@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)CCN1C ZINC000880893263 EH On-Demand Anodyne EPHX2 24 40 COC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893265 EH On-Demand Anodyne RBP4 26 43 COC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893265 EH On-Demand Anodyne PTR1 45 33 COCC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893267 EI On-Demand Anodyne RBP4 23 41 COCC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893267 EI On-Demand Anodyne CACNA1I 47 33 CC(C)c1nnc2n1CCN(C(=O)Nc1cc(Cl)cc(Cl)c1F)C2 ZINC000880893268 FH On-Demand Anodyne P2RX7 27 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(OCCO)CC1 ZINC000880893276 FG On-Demand Anodyne SCD1 15 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N(CCO)CCN1CCOCC1 ZINC000880893283 GE On-Demand Anodyne CASR 60 43 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880893315 GH On-Demand Anodyne EPHX2 35 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880893316 GH On-Demand Anodyne EPHX2 35 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880893317 GH On-Demand Anodyne EPHX2 35 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880893318 GH On-Demand Anodyne EPHX2 35 42 CNC(=O)CC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893328 FH On-Demand Anodyne CACNA1I 44 32 Cn1nccc1C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893329 FI On-Demand Anodyne CACNA1H 48 35 Cn1nccc1C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893329 FI On-Demand Anodyne RBP4 29 40 CC(=O)N(C)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893330 FH On-Demand Anodyne RBP4 27 40 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893344 GF On-Demand Anodyne RBP4 23 40 Cn1cc(CN2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)cn1 ZINC000880893365 GG On-Demand Anodyne FAAH 23 42 N#CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893366 EG On-Demand Mild EPHX2 33 42 N#CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893366 EG On-Demand Mild CXCR3 16 41 CN1CCC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893380 EH On-Demand Anodyne CACNA1H 15 45 CN1CCC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893380 EH On-Demand Anodyne CCR3 38 40 CN1CCC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893380 EH On-Demand Anodyne CACNA1I 75 40 CN(CCN1CCOCC1)C(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880893395 FF On-Demand Anodyne CASR 51 38 CCn1nc2c(cc1=O)CN(C(=O)Nc1cc(Cl)cc(Cl)c1F)CC2 ZINC000880893433 GG On-Demand Anodyne MAPK1 41 37 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](N2CCCC2)C1 ZINC000880893434 EH On-Demand Anodyne L3MBTL3 89 44 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](N2CCCC2)C1 ZINC000880893435 EH On-Demand Anodyne L3MBTL3 89 44 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893454 GF On-Demand Anodyne EPHX2 20 40 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893454 GF On-Demand Anodyne CACNA1I 64 36 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893455 GF On-Demand Anodyne EPHX2 20 40 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893455 GF On-Demand Anodyne CACNA1I 64 36 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893470 FG On-Demand Anodyne CACNA1H 44 37 Cc1noc(C2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)n1 ZINC000880893489 FI On-Demand Anodyne SMO 39 49 Cc1noc(C2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)n1 ZINC000880893489 FI On-Demand Anodyne ETHR 54 35 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880893491 GH On-Demand Anodyne P2RX7 37 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@H](CCO)C1 ZINC000880893492 DG On-Demand Anodyne CACNA1I 45 34 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CC[C@@H](CCO)C1 ZINC000880893493 DG On-Demand Anodyne CACNA1I 45 34 Cc1noc(C)c1CCNC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880893494 EI On-Demand Anodyne P2RX7 19 48 COCCC(=O)N1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893495 GG On-Demand Anodyne EPHX2 45 51 CCOC[C@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893499 EI On-Demand Anodyne CACNA1I 48 34 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccsc1C(F)(F)F ZINC000880893521 GG On-Demand Anodyne PAPA1_CARPA 41 44 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccsc1C(F)(F)F ZINC000880893522 GG On-Demand Anodyne PAPA1_CARPA 41 44 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880893568 GJ On-Demand Anodyne SMO 19 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880893568 GJ On-Demand Anodyne ETHR 21 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880893569 GJ On-Demand Anodyne SMO 19 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880893569 GJ On-Demand Anodyne ETHR 21 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(C(=O)C2CC2)CC1 ZINC000880893570 FG On-Demand Anodyne RBP4 20 41 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCOCC1 ZINC000880893571 DG On-Demand Anodyne EPHX2 21 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2cccnn2)CC1 ZINC000880893583 FG On-Demand Anodyne FAAH 23 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2cccnn2)CC1 ZINC000880893583 FG On-Demand Anodyne RBP4 20 43 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(O)(C(F)(F)F)CC1 ZINC000880893586 GI On-Demand Anodyne CACNA1H 48 37 O=C(NCC1CCS(=O)(=O)CC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880893606 FG On-Demand Anodyne CACNA1I 50 33 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880893617 GH On-Demand Anodyne CXCR3 15 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880893618 GH On-Demand Anodyne CXCR3 15 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(CCO)CC1 ZINC000880893619 FF On-Demand Anodyne HTR4 20 44 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(CCO)CC1 ZINC000880893619 FF On-Demand Anodyne CCR3 26 40 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(CCO)CC1 ZINC000880893619 FF On-Demand Anodyne EPHX2 31 43 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(CCO)CC1 ZINC000880893619 FF On-Demand Anodyne CXCR3 17 42 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893634 EG On-Demand Anodyne EPHX2 39 59 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893635 EG On-Demand Anodyne EPHX2 39 59 COCC1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893672 FG On-Demand Anodyne CACNA1H 71 38 COCC1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893672 FG On-Demand Anodyne S1PR2 27 44 COCC1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893672 FG On-Demand Anodyne RBP4 19 40 C[C@H](O)CN1CCC(CN(C)C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893681 GH On-Demand Anodyne CACNA1I 57 42 Cn1ncc(Br)c1CC(=O)NCc1ccsc1C(F)(F)F ZINC000880893682 GG On-Demand Anodyne P2RX7 22 48 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCn2c(nnc2C2CC2)C1 ZINC000880893685 FH On-Demand Anodyne P2RX7 25 48 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(c2cc[nH]n2)CC1 ZINC000880893686 FI On-Demand Anodyne RBP4 30 41 CC(=O)OC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893696 EH On-Demand Anodyne RBP4 25 40 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893702 GF On-Demand Anodyne SLC6A1 95 37 NC(=O)[C@H]1CCCN(CCCNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893702 GF On-Demand Anodyne CCR3 35 42 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893703 GF On-Demand Anodyne SLC6A1 95 37 NC(=O)[C@@H]1CCCN(CCCNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893703 GF On-Demand Anodyne CCR3 35 42 CN1CCC(CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893715 EH On-Demand Anodyne CACNA1H 18 41 CN1CCC(CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893715 EH On-Demand Anodyne EPHX2 22 40 CN1CCC(CNC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893715 EH On-Demand Anodyne CACNA1I 86 44 NC(=O)C1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893734 EG On-Demand Anodyne EPHX2 22 43 CCC1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893736 EH On-Demand Anodyne CACNA1H 68 38 CCC1(O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893736 EH On-Demand Anodyne S1PR2 28 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCOC2(CCOCC2)C1 ZINC000880893749 FH On-Demand Anodyne EPHX2 18 44 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(Nc2cccnn2)CC1 ZINC000880893761 GI On-Demand Anodyne FAAH 23 42 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880893763 GH On-Demand Anodyne CXCR3 15 40 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880893764 GH On-Demand Anodyne CXCR3 15 40 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C2CC2)CC1 ZINC000880893788 EH On-Demand Anodyne EPHX2 35 43 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880893816 GF On-Demand Anodyne EPHX2 30 40 O=C(NCCN1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880893846 EF On-Demand Anodyne CACNA1H 20 40 O=C(NCCN1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880893846 EF On-Demand Anodyne EPHX2 26 53 C=CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893986 EH On-Demand Mild EPHX2 28 42 C=CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880893986 EH On-Demand Mild CXCR3 16 41 O=C1CC2(CCN(C(=O)Nc3cc(Cl)cc(Cl)c3F)CC2)CN1 ZINC000880894006 FG On-Demand Anodyne CACNA1H 47 36 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880894008 GH On-Demand Anodyne EPHX2 18 40 COCCn1nc(C)c(NC(=O)Nc2cc(Cl)cc(Cl)c2F)c1C ZINC000880894072 GI On-Demand Anodyne P2RX7 16 48 CCCCNC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894093 GI On-Demand Anodyne EPHX2 21 46 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880894132 GH On-Demand Anodyne EPHX2 20 41 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880894133 GH On-Demand Anodyne EPHX2 20 41 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880894134 GH On-Demand Anodyne EPHX2 20 41 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880894135 GH On-Demand Anodyne EPHX2 20 41 COC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894141 EI On-Demand Anodyne CACNA1I 42 32 CN1CCN(C)[C@@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894144 EE On-Demand Anodyne CACNA1I 55 35 CN1CCN(C)[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894145 EE On-Demand Anodyne CACNA1I 55 35 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894165 GF On-Demand Anodyne CACNA1I 41 31 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894166 GF On-Demand Anodyne CACNA1I 41 31 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CC1 ZINC000880894208 CG On-Demand Anodyne EPHX2 39 50 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894263 EG On-Demand Anodyne RBP4 25 40 COC(=O)[C@H]1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894264 EG On-Demand Anodyne RBP4 25 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne TRPV1 20 44 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne P2RX7 43 44 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne SCN2A 17 42 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne EPHX2 16 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne SCN10A 31 54 O=C(NCc1cccnc1N1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894270 GH On-Demand Anodyne STAT6 48 33 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894274 GH On-Demand Anodyne STAT6 43 31 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894274 GH On-Demand Anodyne NAMPT 25 41 O=C(NCCCN1CCCC1=O)Nc1cc(Cl)cc(Cl)c1F ZINC000880894281 EG On-Demand Anodyne TYRO3 20 44 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894302 GG On-Demand Anodyne EPHX2 17 45 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894302 GG On-Demand Anodyne CCR8 72 39 CCN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894313 EH On-Demand Anodyne CACNA1H 15 43 CCN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894313 EH On-Demand Anodyne CCR3 45 38 CCN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880894313 EH On-Demand Anodyne CACNA1I 84 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H]1c1ccccn1 ZINC000880894451 FJ On-Demand Anodyne CACNA1H 54 40 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H]1c1ccccn1 ZINC000880894452 FJ On-Demand Anodyne CACNA1H 54 40 CNC(=O)CN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894455 GE On-Demand Anodyne EPHX2 35 43 CNC(=O)CN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894455 GE On-Demand Anodyne CXCR3 19 42 CS(=O)(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894500 FE On-Demand Anodyne RBP4 23 40 COCC(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894531 FE On-Demand Anodyne RBP4 20 43 COC(=O)c1cc(-c2csc(NC(=O)c3ccc(S(=O)(=O)N(C)OC)cc3)n2)c[nH]1 ZINC000880894641 JE On-Demand Anodyne MPL 44 38 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@H]1c1cccnc1 ZINC000880894654 FJ On-Demand Anodyne CHRNA7 16 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCC[C@@H]1c1cccnc1 ZINC000880894655 FJ On-Demand Anodyne CHRNA7 16 45 CC(=O)N1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894676 EF On-Demand Anodyne RBP4 22 44 O=C(CNC(=O)Nc1cc(Cl)cc(Cl)c1F)NC1CCCC1 ZINC000880894700 EG On-Demand Anodyne EPHX2 15 45 C[C@@H]1[C@@H](C(=O)NCc2ccsc2C(F)(F)F)CCN1C ZINC000880894849 DF On-Demand Anodyne P2RX7 49 37 C[C@H]1[C@H](C(=O)NCc2ccsc2C(F)(F)F)CCN1C ZINC000880894850 DF On-Demand Anodyne P2RX7 49 37 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880894853 FH On-Demand Anodyne EPHX2 46 52 CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894886 EH On-Demand Anodyne HTR4 23 44 CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894886 EH On-Demand Anodyne EPHX2 42 49 CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894886 EH On-Demand Anodyne PDK1 42 30 CCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894886 EH On-Demand Anodyne CXCR3 22 43 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne HTR4 58 42 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne CCR3 28 43 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne EPHX2 36 43 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne PDK1 46 33 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne CXCR3 19 40 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne MCHR1 22 40 COCCN1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894898 FG On-Demand Anodyne CACNA1I 60 40 CN1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894899 DF On-Demand Anodyne HRH4 23 43 CN1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880894899 DF On-Demand Anodyne RBP4 17 43 O=C(NCCCCn1ccnc1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894902 EH On-Demand Anodyne TBXAS1 45 52 O=C(NCCCCn1ccnc1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894902 EH On-Demand Anodyne HMOX2 40 34 O=C(NCCCCn1ccnc1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894902 EH On-Demand Anodyne QPCT 36 49 O=C(NC[C@H]1CCS(=O)(=O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894913 FF On-Demand Anodyne CACNA1I 45 32 O=C(NC[C@@H]1CCS(=O)(=O)C1)Nc1cc(Cl)cc(Cl)c1F ZINC000880894914 FF On-Demand Anodyne CACNA1I 45 32 O=C(Nc1cc(Cl)cc(Cl)c1F)NC1CCSCC1 ZINC000880894940 DI On-Demand Anodyne EPHX2 24 46 CC[C@H](O)CCNC(=O)Nc1cccc(O[C@H](C)CC)n1 ZINC000880894964 CF On-Demand Anodyne ADRB1 40 31 CC[C@H](O)CCNC(=O)Nc1cccc(O[C@@H](C)CC)n1 ZINC000880894966 CF On-Demand Anodyne ADRB1 40 31 CC[C@@H](O)CCNC(=O)Nc1cccc(O[C@H](C)CC)n1 ZINC000880894967 CF On-Demand Anodyne ADRB1 40 31 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2ncccn2)CC1 ZINC000880895123 FG On-Demand Anodyne FAAH 23 42 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCN(c2ncccn2)CC1 ZINC000880895123 FG On-Demand Anodyne RBP4 23 46 COCC(=O)NC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895269 GF On-Demand Anodyne EPHX2 25 40 COCC(=O)NC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895269 GF On-Demand Anodyne RBP4 25 41 CCOC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895271 FH On-Demand Anodyne CACNA1H 40 33 CCOC(=O)C1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895271 FH On-Demand Anodyne EPHX2 16 41 CCOC(=O)C1CCN(C(=O)Nc2cccc(O[C@H](C)CC)n2)CC1 ZINC000880895276 EG On-Demand Anodyne PTR1 44 31 CCOC(=O)C1CCN(C(=O)Nc2cccc(O[C@@H](C)CC)n2)CC1 ZINC000880895277 EG On-Demand Anodyne PTR1 44 31 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCC[C@H](O)C1 ZINC000880895311 DH On-Demand Anodyne EPHX2 17 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCC[C@@H](O)C1 ZINC000880895312 DH On-Demand Anodyne EPHX2 17 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@H]1CCC[C@H](O)C1 ZINC000880895313 DH On-Demand Anodyne EPHX2 17 45 O=C(Nc1cc(Cl)cc(Cl)c1F)N[C@@H]1CCC[C@@H](O)C1 ZINC000880895314 DH On-Demand Anodyne EPHX2 17 45 O=C(NCC1CCOCC1)Nc1cc(Cl)cc(Cl)c1F ZINC000880895406 DH On-Demand Anodyne CACNA1I 54 34 O=C(NCCCO)Nc1cc(Cl)cc(Cl)c1F ZINC000880895408 CF On-Demand Anodyne ALPL 34 41 O=C(Nc1cc(Cl)cc(Cl)c1F)N1CCCC1 ZINC000880895419 CH On-Demand Anodyne RBP4 21 43 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880895427 FH On-Demand Anodyne CCR3 18 44 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 ZINC000880895427 FH On-Demand Anodyne CACNA1I 63 35 Cc1cc([C@@H]2CCCN2C(=O)Nc2cc(Cl)cc(Cl)c2F)on1 ZINC000880895488 FJ On-Demand Anodyne KCNA5 18 45 CC(=O)NCC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895523 FH On-Demand Anodyne EPHX2 19 41 CC(=O)NCC1CCN(C(=O)Nc2cc(Cl)cc(Cl)c2F)CC1 ZINC000880895523 FH On-Demand Anodyne CACNA1I 79 39 O=C(C[C@H]1CCNC1=O)NCCc1ccccc1OCc1ccccc1 ZINC000880895607 FE On-Demand Anodyne PTGER1 20 42 O=C(C[C@H]1CCNC1=O)NCCc1ccccc1OCc1ccccc1 ZINC000880895607 FE On-Demand Anodyne MBTPS1 52 42 O=C(C[C@@H]1CCNC1=O)NCCc1ccccc1OCc1ccccc1 ZINC000880895608 FE On-Demand Anodyne PTGER1 20 42 O=C(C[C@@H]1CCNC1=O)NCCc1ccccc1OCc1ccccc1 ZINC000880895608 FE On-Demand Anodyne MBTPS1 52 42 O=C(COC1CC1)NCCc1ccccc1OCc1ccccc1 ZINC000880895826 EG On-Demand Anodyne PTGER1 40 47 O=C(COC1CC1)NCCc1ccccc1OCc1ccccc1 ZINC000880895826 EG On-Demand Anodyne PTGER3 16 44 O=C(COC1CC1)NCCc1ccccc1OCc1ccccc1 ZINC000880895826 EG On-Demand Anodyne TIMP3 51 33 O=C(COC1CC1)NCCc1ccccc1OCc1ccccc1 ZINC000880895826 EG On-Demand Anodyne MTNR1B 21 41 O=C(COC1CC1)NCCc1ccccc1OCc1ccccc1 ZINC000880895826 EG On-Demand Anodyne MBTPS1 42 42 CCOC[C@H](O)CN1CCN(C(=O)Nc2cccc(O[C@H](C)CC)n2)CC1 ZINC000880895953 GD On-Demand Anodyne ACOX1 49 33 CCOC[C@H](O)CN1CCN(C(=O)Nc2cccc(O[C@@H](C)CC)n2)CC1 ZINC000880895954 GD On-Demand Anodyne ACOX1 49 33 CCc1nc([C@H]2CCCN2C(=O)Nc2cccc(O[C@H](C)CC)n2)no1 ZINC000880896159 FH On-Demand Anodyne CPT1A 52 40 CCc1nc([C@H]2CCCN2C(=O)Nc2cccc(O[C@@H](C)CC)n2)no1 ZINC000880896161 FH On-Demand Anodyne CPT1A 52 40 O=C(NCCc1ccccc1OCc1ccccc1)[C@H]1CCc2nncn2CC1 ZINC000880896216 GG On-Demand Anodyne PTGER1 42 39 O=C(NCCc1ccccc1OCc1ccccc1)[C@@H]1CCc2nncn2CC1 ZINC000880896217 GG On-Demand Anodyne PTGER1 42 39 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc(O[C@H](C)CC)n2)C1 ZINC000880896339 EE On-Demand Anodyne EPHX2 31 48 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc(O[C@H](C)CC)n2)C1 ZINC000880896340 EE On-Demand Anodyne EPHX2 31 48 CCC(=O)N1CC[C@@H](NC(=O)Nc2cccc(O[C@@H](C)CC)n2)C1 ZINC000880896341 EE On-Demand Anodyne EPHX2 31 48 CCC(=O)N1CC[C@H](NC(=O)Nc2cccc(O[C@@H](C)CC)n2)C1 ZINC000880896342 EE On-Demand Anodyne EPHX2 31 48 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896565 DD On-Demand Anodyne PAPA1_CARPA 43 53 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896565 DD On-Demand Anodyne CTSK 18 51 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896565 DD On-Demand Anodyne POLG_HCV1 23 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896566 DD On-Demand Anodyne PAPA1_CARPA 43 53 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896566 DD On-Demand Anodyne CTSK 18 51 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)NCC(C)(C)F ZINC000880896566 DD On-Demand Anodyne POLG_HCV1 23 41 CON=Cc1ccc(C(=O)Nc2cccc(OCC(N)=O)c2)cc1 ZINC000880898141 ED On-Demand Mild ROCK1 45 34 CON=Cc1ccc(C(=O)Nc2cccc(OCC(N)=O)c2)cc1 ZINC000880898141 ED On-Demand Mild PLAU 22 49 CON=Cc1ccc(C(=O)Nc2cccc(OCC(N)=O)c2)cc1 ZINC000880898141 ED On-Demand Mild TAAR1 44 43 CON=Cc1ccc(C(=O)Nc2cccc(OCC(N)=O)c2)cc1 ZINC000880898141 ED On-Demand Mild KCNK3 110 43 CON=Cc1ccc(C(=O)Nc2cccc(OCC(N)=O)c2)cc1 ZINC000880898141 ED On-Demand Mild KCNK9 74 35 CCNc1nc(C)c(C(=O)NCC(C)(C)F)s1 ZINC000880898986 CE On-Demand Anodyne SCD1 15 41 C#Cc1cccc(CNC(=O)Nc2nc(CC(=O)NCCC)cs2)c1 ZINC000880899577 FF On-Demand Mild ROCK2 19 45 COC(=O)c1cc(-c2csc(NC(=O)c3ccc4c(c3)-c3ccccc3C4)n2)c[nH]1 ZINC000880901017 HJ On-Demand Anodyne MPL 67 38 COCCCN(C(=O)/C=C\c1ccc(OC)cc1)c1c(O)nc(=O)n(Cc2ccccc2)c1N ZINC000880901896 JF On-Demand Anodyne PROKR1 59 36 COC(=O)c1cc(-c2csc(NC(=O)c3ccc(Cl)c(S(N)(=O)=O)c3)n2)c[nH]1 ZINC000880902012 IE On-Demand Anodyne MPL 38 42 COC(=O)c1cc(-c2csc(NC(=O)c3ccc(Cl)c(S(N)(=O)=O)c3)n2)c[nH]1 ZINC000880902012 IE On-Demand Anodyne CPT1A 27 40 COC(=O)c1cc(-c2csc(NC(=O)c3ccc(Cl)c(S(N)(=O)=O)c3)n2)c[nH]1 ZINC000880902012 IE On-Demand Anodyne CPT1B 39 40 C#CCC1(O)CCN(C(=O)Nc2cccc(O[C@@H](C)CC)n2)CC1 ZINC000880902325 EF On-Demand Mild S1PR2 27 40 C#CCC1(O)CCN(C(=O)Nc2cccc(O[C@H](C)CC)n2)CC1 ZINC000880902326 EF On-Demand Mild S1PR2 27 40 COC(=O)c1cc(-c2csc(NC(=O)c3cccc(NS(C)(=O)=O)c3)n2)c[nH]1 ZINC000880902679 HF On-Demand Anodyne MPL 57 39 COC(=O)c1cc(-c2csc(NC(=O)c3cccc(NS(C)(=O)=O)c3)n2)c[nH]1 ZINC000880902679 HF On-Demand Anodyne ROCK1 20 48 COC(=O)c1cc(-c2csc(NC(=O)c3cccc(NS(C)(=O)=O)c3)n2)c[nH]1 ZINC000880902679 HF On-Demand Anodyne ROCK2 18 48 CSc1nccnc1C(=O)Nc1nnc(C(F)(F)C(F)(F)F)s1 ZINC000880904814 FF On-Demand Anodyne MAP1 42 33 O=C(Nc1nnc(C(F)(F)C(F)(F)F)s1)c1ncsc1C1CC1 ZINC000880904817 FH On-Demand Anodyne MAP1 80 39 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880905145 GI On-Demand Anodyne SMO 37 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880905145 GI On-Demand Anodyne ETHR 60 45 O=C(COC1CC1)Nc1nnc(-c2cccc(C(F)(F)F)c2)s1 ZINC000880905221 EG On-Demand Anodyne CSNK1D 30 43 CC(C)(CO)[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1cccnc1 ZINC000880905287 FG On-Demand Anodyne NAMPT 20 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Oc2cccc(F)c2)C1 ZINC000880905471 FH On-Demand Anodyne MLNR 15 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Oc2cccc(F)c2)C1 ZINC000880905471 FH On-Demand Anodyne SCD1 22 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Oc2cccc(F)c2)C1 ZINC000880905472 FH On-Demand Anodyne MLNR 15 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Oc2cccc(F)c2)C1 ZINC000880905472 FH On-Demand Anodyne SCD1 22 41 COCCCN(C(=O)/C=C\c1ccc2c(c1)OCO2)c1c(O)nc(=O)n(Cc2ccccc2)c1N ZINC000880905477 JE On-Demand Anodyne DYRK2 45 36 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880905507 GI On-Demand Anodyne SLC18A2 47 34 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880905508 GI On-Demand Anodyne SLC18A2 47 34 O=C(NCCC1CCC1)Nc1cncc(C(F)F)c1 ZINC000880905517 CG On-Demand Anodyne PRMT3 18 45 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cncc(C(F)F)c1 ZINC000880905519 EF On-Demand Anodyne SLC6A3 40 38 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cncc(C(F)F)c1 ZINC000880905520 EF On-Demand Anodyne SLC6A3 40 38 COc1ccccc1[C@H](C)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880905527 DH On-Demand Anodyne KCNK3 37 40 COc1ccccc1[C@H](C)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880905527 DH On-Demand Anodyne KCNK9 33 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccc(F)cc2)CC1 ZINC000880905538 EJ On-Demand Anodyne CACNA1H 42 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccc(F)cc2)CC1 ZINC000880905538 EJ On-Demand Anodyne CCR1 22 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880905682 EI On-Demand Anodyne NPY5R 35 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880905683 EI On-Demand Anodyne NPY5R 35 41 C[C@H]1c2sccc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880905715 DI On-Demand Anodyne TRPM8 22 42 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2cccc(F)c2)CC1 ZINC000880905728 FH On-Demand Anodyne CACNA1H 48 38 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@@H]1Cc1ccccc1 ZINC000880905743 EG On-Demand Anodyne CASR 47 40 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@H]1Cc1ccccc1 ZINC000880905745 EG On-Demand Anodyne CASR 47 40 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880905786 EH On-Demand Anodyne RBP4 45 33 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880905788 EH On-Demand Anodyne RBP4 45 33 O=C(Nc1cncc(C(F)F)c1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880905797 FG On-Demand Anodyne FAAH 22 52 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880905800 FI On-Demand Anodyne EPHX2 22 45 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880905800 FI On-Demand Anodyne SCD1 21 40 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880905800 FI On-Demand Anodyne SCD 23 40 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880905800 FI On-Demand Anodyne TRPM8 36 60 COc1ccc(CN(CCO)C(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880905810 FG On-Demand Anodyne ROCK2 20 47 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880905812 DH On-Demand Anodyne ROCK2 18 44 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880905812 DH On-Demand Anodyne NPY5R 24 40 N#Cc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880905816 FG On-Demand Mild PDGFRB 20 43 O=C(NCc1ccc(CN2CCNC2=O)cc1)Nc1cncc(C(F)F)c1 ZINC000880905847 GF On-Demand Anodyne NAMPT 49 42 CC(C)c1cc(NC(=O)Nc2cncc(C(F)F)c2)ccc1O ZINC000880905851 DI On-Demand Anodyne THRB 39 42 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880905858 GG On-Demand Clean NAMPT 45 39 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880905911 FG On-Demand Anodyne EPHX2 41 39 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2nccnn2)CC1 ZINC000880905932 ED On-Demand Anodyne FAAH 21 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880905957 EH On-Demand Anodyne EPHX2 30 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880905957 EH On-Demand Anodyne SCD1 21 48 CCCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880905959 EI On-Demand Anodyne ROCK2 19 41 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880905965 EH On-Demand Anodyne EPHX2 25 45 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880905966 EH On-Demand Anodyne EPHX2 25 45 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880906032 FI On-Demand Anodyne EPHX2 25 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880906032 FI On-Demand Anodyne SCD1 31 46 O=C(Nc1cncc(C(F)F)c1)N1CCc2nccnc2C1 ZINC000880906040 DE On-Demand Anodyne P2RY14 41 41 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@](F)(c2ccccc2)C1 ZINC000880906042 EJ On-Demand Anodyne EPHX2 27 46 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@](F)(c2ccccc2)C1 ZINC000880906044 EJ On-Demand Anodyne EPHX2 27 46 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880906058 FH On-Demand Anodyne EPHX2 34 41 Cc1cccc2c1CCN2C(=O)Nc1cncc(C(F)F)c1 ZINC000880906060 DH On-Demand Anodyne HTR2C 16 49 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccc(F)cc2F)CC1 ZINC000880906062 FH On-Demand Anodyne NPY2R 85 39 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2cccc(F)c2)CC1 ZINC000880906076 EJ On-Demand Anodyne CACNA1H 56 37 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2cccc(F)c2)CC1 ZINC000880906076 EJ On-Demand Anodyne MCHR1 20 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906099 GD On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906099 GD On-Demand Anodyne CCR3 54 34 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906099 GD On-Demand Anodyne EPHX2 34 46 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906100 GD On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906100 GD On-Demand Anodyne CCR3 54 34 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880906100 GD On-Demand Anodyne EPHX2 34 46 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cc3ccccc3[nH]2)CC1 ZINC000880906143 GH On-Demand Anodyne FAAH 19 43 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880906175 FH On-Demand Anodyne P2RY14 49 40 CN1CCN(C2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)CC1 ZINC000880906209 FE On-Demand Anodyne L3MBTL3 48 38 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880906213 FH On-Demand Anodyne EPHX2 26 54 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880906215 FH On-Demand Anodyne EPHX2 26 54 CN(C[C@@]1(O)CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880906217 GG On-Demand Anodyne NPFFR1 40 33 C[C@@H](c1ccc(Cl)cc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880906229 EJ On-Demand Anodyne UTS2 40 31 C[C@H](c1ccc(Cl)cc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880906238 EJ On-Demand Anodyne UTS2 40 31 N#Cc1cc(F)ccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880906253 GG On-Demand Mild NPY2R 26 42 NC(=O)Cc1cccc2c1CCN(C(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880906275 FF On-Demand Anodyne P2RY14 48 38 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(OC)c1 ZINC000880906284 GG On-Demand Clean PDGFRB 61 47 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880906297 EI On-Demand Anodyne TRPM8 31 46 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCNC2=O)CC1 ZINC000880906305 DE On-Demand Anodyne CACNA1H 45 39 CC(C)(C)OC(=O)CN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880906306 GF On-Demand Anodyne CXCR3 19 44 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(Cl)cn2)CC1 ZINC000880906331 GI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(Cl)cn2)CC1 ZINC000880906331 GI On-Demand Anodyne SCD1 16 44 O=C(NC[C@H]1CCCN(CC2CC2)C1)Nc1cncc(C(F)F)c1 ZINC000880906408 EG On-Demand Anodyne CCR3 76 41 O=C(Nc1cncc(C(F)F)c1)N1CCc2nc(C3CC3)ncc2C1 ZINC000880906414 EG On-Demand Anodyne MAPK1 43 33 O=C(Nc1cncc(C(F)F)c1)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880906434 GI On-Demand Anodyne GRIN2B 19 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880906434 GI On-Demand Anodyne SCD1 25 40 O=C(Nc1cncc(C(F)F)c1)N(CCN1CCOCC1)CC1CC1 ZINC000880906449 FF On-Demand Anodyne CASR 68 55 Cc1ccc(CC2CN(C(=O)Nc3cncc(C(F)F)c3)C2)cc1 ZINC000880906454 EI On-Demand Anodyne CCR3 58 33 O=C(Nc1cncc(C(F)F)c1)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880906464 EI On-Demand Anodyne RBP4 48 36 O=C(NCC1CCN(CC2CC2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906542 EG On-Demand Anodyne CCR3 43 39 O=C(NCC1CCN(CC2CC2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906542 EG On-Demand Anodyne CACNA1I 62 37 O=C(NCC[C@@H](O)COCc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880906559 FG On-Demand Anodyne ADRB1 42 33 N#CCc1cccc2c1CCN(C(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880906619 EH On-Demand Mild P2RY14 50 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880906620 FH On-Demand Anodyne PDGFRB 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880906620 FH On-Demand Anodyne HPGDS 24 42 O=C(Nc1cncc(C(F)F)c1)N1CC(c2ccccc2)C1 ZINC000880906654 DH On-Demand Anodyne RBP4 55 36 C[C@@](CO)(NC(=O)Nc1cncc(C(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000880906670 GI On-Demand Anodyne RIPK1 41 36 C[C@@](CO)(NC(=O)Nc1cncc(C(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000880906670 GI On-Demand Anodyne IMDH_CRYPV 55 36 COc1cccc(OC)c1CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880906701 EG On-Demand Anodyne ROCK2 18 53 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906718 GG On-Demand Anodyne ACHE 22 43 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906718 GG On-Demand Anodyne SIGMAR1 20 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906718 GG On-Demand Anodyne CCR3 66 49 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906718 GG On-Demand Anodyne CACNA1I 61 40 COc1cccc([C@H](CO)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880906777 EF On-Demand Anodyne ROCK1 23 52 O=C(NCc1ccc(N2CCCNC2=O)cc1)Nc1cncc(C(F)F)c1 ZINC000880906820 GG On-Demand Anodyne NAMPT 37 40 O=C(Nc1cncc(C(F)F)c1)N(CCN1CCOCC1)Cc1ccco1 ZINC000880906875 GF On-Demand Anodyne CASR 69 54 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](Oc2ccccc2)C1 ZINC000880906876 EI On-Demand Anodyne EPHX2 24 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](Oc2ccccc2)C1 ZINC000880906877 EI On-Demand Anodyne EPHX2 24 40 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906885 GG On-Demand Anodyne NPFFR2 41 43 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906885 GG On-Demand Anodyne FAAH 15 40 O=C(NCC1(O)CCN(Cc2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880906885 GG On-Demand Anodyne NPFFR1 52 43 CN1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)[C@@H]1c1cccnc1 ZINC000880906914 FG On-Demand Anodyne NAMPT 52 37 COC(=O)[C@@H]1CN(C(=O)Nc2cncc(C(F)F)c2)C[C@H]1c1ccc(O)cc1 ZINC000880906971 GG On-Demand Anodyne SLC6A3 27 40 O=C1C[C@]2(CCCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880906976 GI On-Demand Anodyne EPHX2 28 42 O=C1C[C@@]2(CCCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880906978 GI On-Demand Anodyne EPHX2 28 42 COc1cccc([C@H](CNC(=O)Nc2cncc(C(F)F)c2)OC)c1 ZINC000880906986 FH On-Demand Anodyne ROCK1 19 40 COc1cccc([C@H](CNC(=O)Nc2cncc(C(F)F)c2)OC)c1 ZINC000880906986 FH On-Demand Anodyne MTNR1B 25 40 O=C(Nc1cncc(C(F)F)c1)N1CCc2c(O)cccc2C1 ZINC000880907002 DG On-Demand Anodyne P2RY14 44 39 COc1ccc(N2CC[C@H](NC(=O)Nc3cncc(C(F)F)c3)C2)cc1 ZINC000880907024 FG On-Demand Clean EPHX2 42 38 CN(CCN1CCCCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880907040 DF On-Demand Anodyne CASR 46 40 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild DRD4 17 49 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild SIGMAR1 18 42 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild SSTR5 40 38 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild CCR3 48 51 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild ITGA4 41 31 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild CXCR3 24 43 N#Cc1cccc(CN2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880907041 GH On-Demand Mild MCHR1 55 47 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907047 FG On-Demand Anodyne EPHX2 41 39 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880907076 FH On-Demand Anodyne P2RY14 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCc2cc(Cl)nnc2C1 ZINC000880907077 EG On-Demand Anodyne MAPK1 49 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880907078 GI On-Demand Anodyne EPHX2 19 45 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880907079 GI On-Demand Anodyne EPHX2 19 45 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cncc(C(F)F)c1 ZINC000880907080 GF On-Demand Anodyne CCR3 52 38 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cncc(C(F)F)c1 ZINC000880907080 GF On-Demand Anodyne NAMPT 42 37 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cncc(C(F)F)c1 ZINC000880907081 GF On-Demand Anodyne CCR3 52 38 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cncc(C(F)F)c1 ZINC000880907081 GF On-Demand Anodyne NAMPT 42 37 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Oc2ccccc2)C1 ZINC000880907082 EH On-Demand Anodyne EPHX2 30 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Oc2ccccc2)C1 ZINC000880907082 EH On-Demand Anodyne SCD1 21 48 COc1ccc(N2CC[C@H](CNC(=O)Nc3cncc(C(F)F)c3)C2)cc1 ZINC000880907255 GH On-Demand Clean CCR3 27 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907298 GI On-Demand Anodyne SIRT3 25 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907298 GI On-Demand Anodyne SIRT2 24 41 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907298 GI On-Demand Anodyne SIRT1 24 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880907301 GH On-Demand Anodyne TRPM8 31 44 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880907302 GH On-Demand Anodyne TRPM8 31 44 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880907303 GH On-Demand Anodyne TRPM8 31 44 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880907304 GH On-Demand Anodyne TRPM8 31 44 COCCc1ccc(OC[C@@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907315 GF On-Demand Anodyne ADRB2 36 49 COCCc1ccc(OC[C@@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907315 GF On-Demand Anodyne ADRB1 77 49 COCCc1ccc(OC[C@@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907315 GF On-Demand Anodyne ADRB3 50 44 COCCc1ccc(OC[C@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907316 GF On-Demand Anodyne ADRB2 36 49 COCCc1ccc(OC[C@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907316 GF On-Demand Anodyne ADRB1 77 49 COCCc1ccc(OC[C@H](O)CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880907316 GF On-Demand Anodyne ADRB3 50 44 CC(C)(C)OC(=O)N1CC2(CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)C1 ZINC000880907323 GH On-Demand Anodyne EPHX2 25 40 COC[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1cccc(OC)c1 ZINC000880907326 FH On-Demand Anodyne ROCK1 19 49 COC[C@@H](NC(=O)Nc1cncc(C(F)F)c1)c1cccc(OC)c1 ZINC000880907327 FH On-Demand Anodyne ROCK1 19 49 O=C(CCCc1ccccc1)NCCNC(=O)Nc1cncc(C(F)F)c1 ZINC000880907361 GG On-Demand Anodyne FAAH 40 36 O=C(CCCc1ccccc1)NCCNC(=O)Nc1cncc(C(F)F)c1 ZINC000880907361 GG On-Demand Anodyne CES1D 54 32 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907392 FG On-Demand Anodyne EPHX2 50 44 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907392 FG On-Demand Anodyne CXCR3 15 52 C[C@@H]1CN(C(=O)Nc2cncc(C(F)F)c2)CCc2ccccc21 ZINC000880907402 EI On-Demand Anodyne TRPM8 24 40 C[C@H]1CN(C(=O)Nc2cncc(C(F)F)c2)CCc2ccccc21 ZINC000880907403 EI On-Demand Anodyne TRPM8 24 40 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907471 FG On-Demand Anodyne EPHX2 20 44 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907471 FG On-Demand Anodyne NAMPT 52 36 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907472 FG On-Demand Anodyne EPHX2 20 44 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907472 FG On-Demand Anodyne NAMPT 52 36 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907521 EG On-Demand Anodyne CACNA1I 52 34 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907522 EG On-Demand Anodyne CACNA1I 52 34 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000880907538 EG On-Demand Anodyne ACHE 25 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000880907538 EG On-Demand Anodyne SIGMAR1 37 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccccc2)CC1 ZINC000880907538 EG On-Demand Anodyne FAAH 42 56 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880907553 FF On-Demand Anodyne L3MBTL3 54 37 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880907554 FF On-Demand Anodyne L3MBTL3 54 37 O=C(NCc1cccnc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880907563 EG On-Demand Anodyne TRPV1 30 41 O=C(NCc1cccnc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880907563 EG On-Demand Anodyne SCN2A 20 49 O=C(NCc1cccnc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880907563 EG On-Demand Anodyne SCN10A 35 49 O=C(NCc1cccnc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880907563 EG On-Demand Anodyne NAMPT 46 42 CCN1CC[C@@H](N(CC)C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907566 DF On-Demand Anodyne CCR5 16 45 CCN1CC[C@H](N(CC)C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880907567 DF On-Demand Anodyne CCR5 16 45 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H](CO)Cc1ccccc1 ZINC000880907573 EG On-Demand Anodyne NPY5R 36 48 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H](CO)Cc1ccccc1 ZINC000880907574 EG On-Demand Anodyne NPY5R 36 48 O=C(Nc1cncc(C(F)F)c1)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880907579 DF On-Demand Anodyne PLM2_PLAFA 68 38 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(CO)CC1 ZINC000880907663 DD On-Demand Anodyne S1PR2 28 40 O=C(Nc1cncc(C(F)F)c1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880907679 FJ On-Demand Anodyne KCNH2 39 41 O=C(Nc1cncc(C(F)F)c1)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880907679 FJ On-Demand Anodyne GLRA1 44 36 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1C[C@@H](Oc2ccccc2)C1 ZINC000880907709 EH On-Demand Anodyne EPHX2 38 40 O=C(Nc1cncc(C(F)F)c1)N1C[C@@H]2CCN(Cc3ccccc3)[C@@H]2C1 ZINC000880907716 FH On-Demand Anodyne RBP4 52 34 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880907741 CD On-Demand Anodyne LUXR 72 38 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880907741 CD On-Demand Anodyne TRAR 85 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCOC1=O ZINC000880907741 CD On-Demand Anodyne LASR 58 37 C[C@@H](CNC(=O)Nc1cncc(C(F)F)c1)c1ccccn1 ZINC000880907801 DG On-Demand Anodyne SOAT1 17 40 COC(=O)[C@@H]1CN(C(=O)Nc2cncc(C(F)F)c2)C[C@H]1c1ccccc1 ZINC000880907824 GG On-Demand Anodyne SLC6A3 26 43 CC[C@@H](NC(=O)Nc1cncc(C(F)F)c1)c1ccccc1 ZINC000880907859 DI On-Demand Anodyne TACR3 52 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@](O)(Cc2ccc(F)cc2)C1 ZINC000880907862 FG On-Demand Anodyne S1PR2 30 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@](O)(Cc2ccc(F)cc2)C1 ZINC000880907863 FG On-Demand Anodyne S1PR2 30 43 CN(C)C1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880907887 DG On-Demand Anodyne EPHX2 41 35 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H](CO)c1ccccc1 ZINC000880907890 DG On-Demand Anodyne NPY5R 35 41 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H](CO)c1ccccc1 ZINC000880907891 DG On-Demand Anodyne NPY5R 35 41 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)C(=O)N1c2ccccc2C[C@H]1C ZINC000880907934 FH On-Demand Anodyne TPP2 62 36 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)C(=O)N1c2ccccc2C[C@@H]1C ZINC000880907936 FH On-Demand Anodyne TPP2 62 36 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](F)C1 ZINC000880907950 CF On-Demand Anodyne DPP4 18 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](F)C1 ZINC000880907951 CF On-Demand Anodyne DPP4 18 40 O=C(NC[C@@H](O)c1ccc(C(F)(F)F)cc1)Nc1cncc(C(F)F)c1 ZINC000880907968 GH On-Demand Anodyne EPHX2 15 40 O=C(NC[C@H](O)c1ccc(C(F)(F)F)cc1)Nc1cncc(C(F)F)c1 ZINC000880907969 GH On-Demand Anodyne EPHX2 15 40 CN1CC[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)C1 ZINC000880907974 DF On-Demand Anodyne EPHX2 23 40 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880907978 FG On-Demand Anodyne MTOR 45 36 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880907978 FG On-Demand Anodyne STAT6 61 41 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880907978 FG On-Demand Anodyne NAMPT 48 44 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](c2ccccc2F)C1 ZINC000880907986 EI On-Demand Anodyne RBP4 70 35 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](c2ccccc2F)C1 ZINC000880907987 EI On-Demand Anodyne RBP4 70 35 N#Cc1ccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880908015 GI On-Demand Mild SCD1 18 45 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880908041 GH On-Demand Anodyne EPHX2 21 42 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880908042 GH On-Demand Anodyne EPHX2 21 42 O=C(Nc1cncc(C(F)F)c1)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880908046 FF On-Demand Anodyne CHRNA4 25 43 O=C(Nc1cncc(C(F)F)c1)N[C@@H](CCO)c1ccc(Cl)cc1 ZINC000880908047 FH On-Demand Anodyne UTS2 43 34 O=C(Nc1cncc(C(F)F)c1)N[C@H](CCO)c1ccc(Cl)cc1 ZINC000880908048 FH On-Demand Anodyne UTS2 43 34 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA2 77 43 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA1 69 42 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA7 37 41 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA5B 60 41 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA4 74 43 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA5A 64 41 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne GRM4 40 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA12 49 42 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne CA9 52 42 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne BTK 15 40 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne TAAR1 26 41 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne SHH 25 40 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne MTCA1 45 36 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne P96878_MYCTU 50 36 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne KCNK3 63 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2Cl)c1 ZINC000880908076 GD On-Demand Anodyne KCNK9 60 36 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1Cl ZINC000880908172 FI On-Demand Anodyne PDE5A 33 40 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1Cl ZINC000880908172 FI On-Demand Anodyne PDE6A 43 33 CN1CCC[C@@H](CCNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880908313 DF On-Demand Anodyne CCR3 67 39 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880908328 FJ On-Demand Anodyne PRCP 42 38 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880908329 FJ On-Demand Anodyne PRCP 42 38 O=C(Nc1cncc(C(F)F)c1)N1CC2(CC2)c2ccccc21 ZINC000880908394 DI On-Demand Anodyne P2RY1 16 40 O=C(Nc1cncc(C(F)F)c1)N1CC2(CC2)c2ccccc21 ZINC000880908394 DI On-Demand Anodyne NPY5R 23 40 O=C(Nc1cncc(C(F)F)c1)NC12CCC(CC1)CC2 ZINC000880908405 CH On-Demand Anodyne EPHX2 20 41 O=C1C[C@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908436 FH On-Demand Anodyne ACACA 47 35 O=C1C[C@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908436 FH On-Demand Anodyne EPHX2 28 46 O=C1C[C@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908436 FH On-Demand Anodyne SCD 18 41 O=C1C[C@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908436 FH On-Demand Anodyne TRPM8 29 42 O=C1C[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908437 FH On-Demand Anodyne ACACA 47 35 O=C1C[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908437 FH On-Demand Anodyne EPHX2 28 46 O=C1C[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908437 FH On-Demand Anodyne SCD 18 41 O=C1C[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)Oc2ccccc21 ZINC000880908437 FH On-Demand Anodyne TRPM8 29 42 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](c2ccccc2)C1 ZINC000880908444 EI On-Demand Anodyne RBP4 45 34 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](c2ccccc2)C1 ZINC000880908445 EI On-Demand Anodyne RBP4 45 34 CN(C)S(=O)(=O)c1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880908452 GF On-Demand Anodyne NAMPT 53 45 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880908509 GF On-Demand Anodyne RBP4 45 34 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880908510 GF On-Demand Anodyne RBP4 45 34 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880908511 GF On-Demand Anodyne RBP4 45 34 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880908512 GF On-Demand Anodyne RBP4 45 34 O=C(Nc1cncc(C(F)F)c1)N1CC(c2cccc(C(F)(F)F)c2)C1 ZINC000880908533 FJ On-Demand Anodyne RBP4 46 34 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CC1)OCCc1ccccc12 ZINC000880908550 FI On-Demand Anodyne NPY5R 30 40 Cc1cccc2c1N(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880908560 DH On-Demand Anodyne HTR2C 15 45 O=C(Nc1cncc(C(F)F)c1)NC1CCC(OC(F)F)CC1 ZINC000880908615 EH On-Demand Anodyne EPHX2 44 40 C[C@@H](Cc1cccc(F)c1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880908626 EI On-Demand Anodyne NPY5R 33 46 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880908660 FH On-Demand Anodyne P96878_MYCTU 41 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA2 67 48 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA1 58 40 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA7 40 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA5B 52 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA4 63 48 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA5A 60 38 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA12 42 40 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne CA9 50 48 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne BTK 20 42 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne TAAR1 25 43 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne MTCA1 41 36 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne P96878_MYCTU 43 36 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne KCNK3 62 35 NC(=O)COc1cccc(NC(=O)c2cc(S(N)(=O)=O)ccc2F)c1 ZINC000880908685 FC On-Demand Anodyne KCNK9 56 35 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)nc1 ZINC000880908693 FF On-Demand Anodyne PDGFRB 57 41 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)nc1 ZINC000880908693 FF On-Demand Anodyne FAAH 16 40 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)nc1 ZINC000880908693 FF On-Demand Anodyne DGAT1 31 44 O=C(Nc1cncc(C(F)F)c1)N1CCc2cccc(Cl)c2C1 ZINC000880908824 EI On-Demand Anodyne MAPK1 44 34 O=C(Nc1cncc(C(F)F)c1)N1CCc2cccc(Cl)c2C1 ZINC000880908824 EI On-Demand Anodyne P2RY14 49 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1COc1ccccc1 ZINC000880908835 EI On-Demand Anodyne CHRNA7 17 48 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1COc1ccccc1 ZINC000880908835 EI On-Demand Anodyne CPT1A 91 35 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1COc1ccccc1 ZINC000880908835 EI On-Demand Anodyne CPT2 43 34 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1COc1ccccc1 ZINC000880908835 EI On-Demand Anodyne CHRNA10 69 41 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880908848 EH On-Demand Anodyne PTAFR 37 49 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880908855 FF On-Demand Anodyne EPHX2 27 40 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880908856 FF On-Demand Anodyne EPHX2 27 40 O=C(Nc1cncc(C(F)F)c1)NC1CCC1 ZINC000880908876 BF On-Demand Anodyne EPHX2 42 40 COC(=O)[C@@H]1CN(C(=O)Nc2cncc(C(F)F)c2)C[C@@H]1c1ccccc1 ZINC000880908886 GG On-Demand Anodyne SLC6A3 26 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2noc3cc(F)ccc23)CC1 ZINC000880908930 GJ On-Demand Anodyne HTR2A 26 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2noc3cc(F)ccc23)CC1 ZINC000880908930 GJ On-Demand Anodyne HTR7 25 42 COC(=O)C[C@](C)(NC(=O)Nc1cncc(C(F)F)c1)c1cccc(OC)c1 ZINC000880908970 GH On-Demand Anodyne IMDH_CRYPV 46 39 COC(=O)C[C@@](C)(NC(=O)Nc1cncc(C(F)F)c1)c1cccc(OC)c1 ZINC000880908971 GH On-Demand Anodyne IMDH_CRYPV 46 39 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880908978 EG On-Demand Anodyne EPHX2 33 46 O=C(Nc1cncc(C(F)F)c1)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880908979 EG On-Demand Anodyne EPHX2 33 46 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(CCCO)C1 ZINC000880908992 ED On-Demand Anodyne CCR3 49 33 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(CCCO)C1 ZINC000880908993 ED On-Demand Anodyne CCR3 49 33 O=C(Nc1cncc(C(F)F)c1)N1CCOC2(CCCCC2)C1 ZINC000880909023 EH On-Demand Anodyne EPHX2 17 46 O=C(NCC1(c2ccccn2)CCC1)Nc1cncc(C(F)F)c1 ZINC000880909189 EH On-Demand Anodyne NMBR 45 41 O=C(NCC1(c2ccccn2)CCC1)Nc1cncc(C(F)F)c1 ZINC000880909189 EH On-Demand Anodyne GRPR 24 41 COc1cccc(C2(CNC(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880909196 EH On-Demand Anodyne SOAT1 24 51 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(CCN(Cc3ccccc3)C2)C1 ZINC000880909204 GI On-Demand Anodyne FAAH 19 55 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(CCN(Cc3ccccc3)C2)C1 ZINC000880909204 GI On-Demand Anodyne EPHX2 27 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(CCN(Cc3ccccc3)C2)C1 ZINC000880909205 GI On-Demand Anodyne FAAH 19 55 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(CCN(Cc3ccccc3)C2)C1 ZINC000880909205 GI On-Demand Anodyne EPHX2 27 40 O=C(NCCCCCN1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880909208 EG On-Demand Anodyne CCR3 36 40 O=C(NCCCCCN1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880909208 EG On-Demand Anodyne CHRNA7 23 53 O=C(NC[C@H](CO)C1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880909239 EG On-Demand Anodyne PRMT3 25 41 O=C(NC[C@@H](CO)C1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880909240 EG On-Demand Anodyne PRMT3 25 41 CN(C)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(OCC(N)=O)c2)c1 ZINC000880909261 GD On-Demand Anodyne TAAR1 26 43 CN(C)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(OCC(N)=O)c2)c1 ZINC000880909261 GD On-Demand Anodyne KCNK3 59 35 CN(C)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(OCC(N)=O)c2)c1 ZINC000880909261 GD On-Demand Anodyne KCNK9 55 35 CC(=O)N1CCC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880909318 EE On-Demand Anodyne CCR3 55 32 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880909319 EE On-Demand Anodyne CCR3 55 32 N#Cc1ccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880909321 FH On-Demand Mild EPHX2 23 49 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880909337 GG On-Demand Anodyne BIRC2 18 47 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(C(=O)Cc2ccccc2)C1 ZINC000880909338 GG On-Demand Anodyne BIRC2 18 47 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cncc(C(F)F)c1 ZINC000880909374 FG On-Demand Anodyne CCR3 25 40 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cncc(C(F)F)c1 ZINC000880909374 FG On-Demand Anodyne CACNA1I 63 37 O=C(NCc1cccc(N2CCCS2(=O)=O)c1)Nc1cncc(C(F)F)c1 ZINC000880909402 GF On-Demand Anodyne CDK1 17 41 O=C(Nc1cncc(C(F)F)c1)Nc1cc(C2CC2)[nH]n1 ZINC000880909421 CG On-Demand Anodyne CDK2 15 47 O=C(Nc1cncc(C(F)F)c1)Nc1cc(C2CC2)[nH]n1 ZINC000880909421 CG On-Demand Anodyne PKNB 45 34 O=C(NC[C@@H]1CN(Cc2ccccc2)CCCO1)Nc1cncc(C(F)F)c1 ZINC000880909429 GG On-Demand Anodyne CCR3 29 45 O=C(NC[C@H]1CN(Cc2ccccc2)CCCO1)Nc1cncc(C(F)F)c1 ZINC000880909436 GG On-Demand Anodyne CCR3 29 45 O=C(Nc1cncc(C(F)F)c1)N1CCC(CO)(c2ccccc2)CC1 ZINC000880909562 FH On-Demand Anodyne EPHX2 16 41 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1CN1CCOCC1 ZINC000880909571 EE On-Demand Anodyne CASR 38 40 O=C(Nc1cncc(C(F)F)c1)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880909572 EG On-Demand Anodyne EPHX2 44 46 CN(CCN1CCOC(C)(C)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880909627 EF On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@H]1c1nc2ccccc2s1 ZINC000880909634 GI On-Demand Anodyne CASR 36 40 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@@H]1c1nc2ccccc2s1 ZINC000880909635 GI On-Demand Anodyne CASR 36 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909649 GF On-Demand Anodyne CPT1A 96 39 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909649 GF On-Demand Anodyne CPT2 42 34 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909649 GF On-Demand Anodyne EPHX2 36 44 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909650 GF On-Demand Anodyne CPT1A 96 39 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909650 GF On-Demand Anodyne CPT2 42 34 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)COc2ccccc2)C1 ZINC000880909650 GF On-Demand Anodyne EPHX2 36 44 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880909677 GI On-Demand Anodyne CACNA1H 47 38 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880909677 GI On-Demand Anodyne NPY5R 33 40 Cc1ccncc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880909714 EG On-Demand Anodyne NPY2R 52 34 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCC2)C1 ZINC000880909837 CG On-Demand Anodyne EPHX2 29 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880909849 FG On-Demand Anodyne EPHX2 28 43 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1c1ccccc1 ZINC000880909853 EJ On-Demand Anodyne CPT1A 49 34 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1c1ccccc1 ZINC000880909854 EJ On-Demand Anodyne CPT1A 49 34 O=C(Nc1cncc(C(F)F)c1)N1CCO[C@@]2(CCCOC2)C1 ZINC000880909885 EE On-Demand Anodyne EPHX2 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCO[C@]2(CCCOC2)C1 ZINC000880909887 EE On-Demand Anodyne EPHX2 15 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880909895 FI On-Demand Anodyne EPHX2 32 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880909895 FI On-Demand Anodyne TRPM8 34 53 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880909897 FI On-Demand Anodyne EPHX2 32 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880909897 FI On-Demand Anodyne TRPM8 34 53 COC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880909918 EE On-Demand Anodyne MTOR 26 43 COC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880909918 EE On-Demand Anodyne EPHX2 50 43 COC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880909918 EE On-Demand Anodyne CXCR3 16 42 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2nccc3sccc23)CC1 ZINC000880909970 GH On-Demand Anodyne PDGFRB 49 39 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880910004 FH On-Demand Anodyne NPY2R 54 36 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880910005 FH On-Demand Anodyne NPY2R 54 36 COc1cc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)ccc1F ZINC000880910029 GH On-Demand Anodyne PDGFRB 49 42 O=C(Nc1cncc(C(F)F)c1)N1CCc2cccc(F)c2C1 ZINC000880910040 DH On-Demand Anodyne P2RY14 49 40 O=C(NC[C@H]1CCN(c2ccccc2F)C1)Nc1cncc(C(F)F)c1 ZINC000880910043 FH On-Demand Anodyne NPY2R 56 37 O=C(NC[C@@H]1CCN(c2ccccc2F)C1)Nc1cncc(C(F)F)c1 ZINC000880910044 FH On-Demand Anodyne NPY2R 56 37 CCOC(=O)c1cnn(C2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880910100 GG On-Demand Anodyne P2RY12 19 42 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne AVPR2 17 40 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne KCNQ2 79 42 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne NPY2R 57 33 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne SCN2A 21 48 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne SCN10A 26 48 O=C(NCc1ccccc1N1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880910105 EH On-Demand Anodyne NAMPT 34 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2cc(Cl)c[nH]2)CC1 ZINC000880910134 GG On-Demand Anodyne EPHX2 29 41 O=C(Nc1cncc(C(F)F)c1)N1CCCC2(CCOCC2)C1 ZINC000880910143 EG On-Demand Anodyne EPHX2 28 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(F)(c2ccccc2)CC1 ZINC000880910168 EJ On-Demand Anodyne CACNA1H 46 36 O=C(Nc1cncc(C(F)F)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000880910183 DH On-Demand Anodyne EPHX2 21 49 O=C(Nc1cncc(C(F)F)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000880910184 DH On-Demand Anodyne EPHX2 21 49 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000880910185 DH On-Demand Anodyne EPHX2 21 49 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000880910186 DH On-Demand Anodyne EPHX2 21 49 O=C(Nc1ccc([C@@H]2CCOC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880910196 EI On-Demand Anodyne MTOR 43 39 O=C(Nc1ccc([C@H]2CCOC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880910197 EI On-Demand Anodyne MTOR 43 39 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910231 GI On-Demand Anodyne SLC18A3 28 44 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910231 GI On-Demand Anodyne WNT3A 46 33 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880910247 FG On-Demand Anodyne EPHX2 43 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880910247 FG On-Demand Anodyne CXCR3 20 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC(F)(F)F)CC1 ZINC000880910247 FG On-Demand Anodyne HPGDS 41 45 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(S(=O)(=O)c2ccccc2)C1 ZINC000880910249 GF On-Demand Anodyne EPHX2 32 51 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(S(=O)(=O)c2ccccc2)C1 ZINC000880910249 GF On-Demand Anodyne TGM2 55 46 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(S(=O)(=O)c2ccccc2)C1 ZINC000880910249 GF On-Demand Anodyne F13A1 47 46 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(S(=O)(=O)c2ccccc2)C1 ZINC000880910249 GF On-Demand Anodyne SFRP1 59 37 C[C@@H]1CN(CCCNC(=O)Nc2cncc(C(F)F)c2)CCCO1 ZINC000880910278 EF On-Demand Anodyne CCR3 47 42 O=C(NC[C@@H](O)Cc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880910283 DF On-Demand Anodyne ADRB1 41 31 O=C(NC[C@H](O)Cc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880910285 DF On-Demand Anodyne ADRB1 41 31 CCOC(=O)C1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910333 EG On-Demand Anodyne EPHX2 42 37 CCCN(CCN1CCCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880910335 EG On-Demand Anodyne CASR 60 47 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880910377 EG On-Demand Anodyne EPHX2 22 43 COC[C@@H](O)CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880910381 CD On-Demand Anodyne ADRB1 40 31 C[C@@](CO)(NC(=O)Nc1cncc(C(F)F)c1)c1cccc(O)c1 ZINC000880910421 EF On-Demand Anodyne IMDH_CRYPV 57 35 O=C(Nc1cncc(C(F)F)c1)N1CCCN(c2ccccc2F)CC1 ZINC000880910449 FH On-Demand Anodyne KCNQ2 65 37 O=C(Nc1cncc(C(F)F)c1)N1CCCN(c2ccccc2F)CC1 ZINC000880910449 FH On-Demand Anodyne NPY2R 88 36 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(C(=O)CCC(F)(F)F)C1 ZINC000880910450 GG On-Demand Anodyne EPHX2 25 48 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(C(=O)CCC(F)(F)F)C1 ZINC000880910450 GG On-Demand Anodyne ETHR 47 34 CCCN(CCN1CCCCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880910453 EH On-Demand Anodyne CASR 59 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(c2cccnn2)CC1 ZINC000880910467 EF On-Demand Anodyne EPHX2 33 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@](F)(c2ccccc2)C1 ZINC000880910472 EI On-Demand Anodyne EPHX2 34 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@](F)(c2ccccc2)C1 ZINC000880910473 EI On-Demand Anodyne EPHX2 34 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1c2ccccc2C[C@H]1O ZINC000880910474 DF On-Demand Anodyne PLM2_PLAFA 68 38 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880910475 DF On-Demand Anodyne PLM2_PLAFA 68 38 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880910476 DF On-Demand Anodyne PLM2_PLAFA 68 38 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880910502 GG On-Demand Anodyne EPHX2 43 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880910503 GG On-Demand Anodyne EPHX2 43 42 O=C(Nc1cncc(C(F)F)c1)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880910517 FH On-Demand Anodyne FAAH 19 44 O=C(Nc1cncc(C(F)F)c1)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880910517 FH On-Demand Anodyne RBP4 56 36 COc1cnccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910544 FF On-Demand Anodyne HTR1B 16 48 COc1cnccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910544 FF On-Demand Anodyne PDGFRB 61 48 COc1cnccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910544 FF On-Demand Anodyne RBP4 15 40 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910545 FF On-Demand Anodyne FAAH 17 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(N2CCc3cc(F)ccc32)CC1 ZINC000880910556 GI On-Demand Anodyne SCD1 32 53 O=C(Nc1cncc(C(F)F)c1)N1CCC(N2CCc3cc(F)ccc32)CC1 ZINC000880910556 GI On-Demand Anodyne SCD 22 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](c2cccc(F)c2)C1 ZINC000880910579 EI On-Demand Anodyne CCR5 64 34 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](c2cccc(F)c2)C1 ZINC000880910580 EI On-Demand Anodyne CCR5 64 34 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ncccc2F)CC1 ZINC000880910591 FH On-Demand Anodyne SCD1 19 44 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne DRD4 29 47 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne ACHE 42 44 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne HTR4 32 42 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne SIGMAR1 33 40 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne CCR3 96 44 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910651 FH On-Demand Anodyne CACNA1I 47 37 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne DRD4 29 47 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne ACHE 42 44 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne HTR4 32 42 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne SIGMAR1 33 40 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne CCR3 96 44 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880910652 FH On-Demand Anodyne CACNA1I 47 37 O=C(Nc1cncc(C(F)F)c1)N1CCC(N2CCc3ccccc32)CC1 ZINC000880910664 FI On-Demand Anodyne SCD1 34 56 CN1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880910685 CE On-Demand Anodyne CCR3 40 37 CN1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880910685 CE On-Demand Anodyne CACNA1I 45 32 CN1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880910686 CE On-Demand Anodyne CCR3 40 37 CN1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880910686 CE On-Demand Anodyne CACNA1I 45 32 CC[C@H]1c2ccccc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880910693 EJ On-Demand Anodyne TRPM8 39 44 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880910694 EJ On-Demand Anodyne TRPM8 39 44 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccnc(O)c2C1 ZINC000880910704 DF On-Demand Anodyne MAPK1 45 34 CC(C)(C)OC(=O)N1CCC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910718 GH On-Demand Anodyne EPHX2 50 40 CC(C)(C)OC(=O)N1CCC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910718 GH On-Demand Anodyne GPR119 43 42 CC(C)(C)OC(=O)N1CCC[C@H](NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910719 GH On-Demand Anodyne EPHX2 50 40 CC(C)(C)OC(=O)N1CCC[C@H](NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880910719 GH On-Demand Anodyne GPR119 43 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880910755 GG On-Demand Anodyne CCR3 86 35 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880910756 GG On-Demand Anodyne CCR3 86 35 CN1CCC(N2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)CC1 ZINC000880910757 FF On-Demand Anodyne CXCR3 15 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880910784 FH On-Demand Anodyne EPHX2 24 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880910784 FH On-Demand Anodyne SCD1 18 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880910807 GH On-Demand Anodyne CACNA1H 50 35 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880910807 GH On-Demand Anodyne EPHX2 23 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880910807 GH On-Demand Anodyne TRPM8 28 40 C[C@@](CO)(NC(=O)Nc1cncc(C(F)F)c1)c1ccccc1 ZINC000880910824 DG On-Demand Anodyne IMDH_CRYPV 53 34 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cncc(C(F)F)c1 ZINC000880910830 FF On-Demand Anodyne CASR 44 36 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cncc(C(F)F)c1 ZINC000880910830 FF On-Demand Anodyne MTOR 55 38 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cncc(C(F)F)c1 ZINC000880910830 FF On-Demand Anodyne PIK3CB 46 37 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cncc(C(F)F)c1 ZINC000880910830 FF On-Demand Anodyne STAT6 53 33 O=C(NC[C@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1)c1ccccc1 ZINC000880910847 GH On-Demand Anodyne HCRTR1 20 49 O=C(NC[C@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1)c1ccccc1 ZINC000880910847 GH On-Demand Anodyne PREP 24 40 O=C(Nc1cncc(C(F)F)c1)N1CCO[C@@]2(CCOC2)C1 ZINC000880910848 DE On-Demand Anodyne EPHX2 15 41 O=C(Nc1cncc(C(F)F)c1)N1CCO[C@]2(CCOC2)C1 ZINC000880910849 DE On-Demand Anodyne EPHX2 15 41 O=C(Nc1cncc(C(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880910884 FG On-Demand Anodyne PDGFRB 41 39 O=C(Nc1cncc(C(F)F)c1)N1CCCN(c2ncccc2F)CC1 ZINC000880910884 FG On-Demand Anodyne TRPV1 15 53 O=C(Nc1cncc(C(F)F)c1)N[C@H](CO)Cc1ccccc1 ZINC000880910885 DF On-Demand Anodyne ANPEP 52 32 O=C(Nc1cncc(C(F)F)c1)N[C@@H](CO)Cc1ccccc1 ZINC000880910886 DF On-Demand Anodyne ANPEP 52 32 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccccn2)CC1 ZINC000880910924 EF On-Demand Anodyne FAAH 23 45 O=C(NCCCNC(=O)C1CCC1)Nc1cncc(C(F)F)c1 ZINC000880911021 EE On-Demand Anodyne TBK1 83 38 O=C(Nc1cncc(C(F)F)c1)N1CCc2cc(Cl)ccc2C1 ZINC000880911022 EI On-Demand Anodyne MAPK1 47 37 O=C(Nc1cncc(C(F)F)c1)NC1CC(OCc2ccccc2)C1 ZINC000880911037 EH On-Demand Anodyne EPHX2 19 40 COc1cccc(C2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880911057 FI On-Demand Anodyne MCHR1 21 42 C[C@H]1c2ccccc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880911060 DI On-Demand Anodyne TRPM8 41 46 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880911074 EH On-Demand Anodyne CACNA1H 41 36 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(c2ccccc2)CC1 ZINC000880911074 EH On-Demand Anodyne OPRL1 17 43 O=C(NCc1cccc(C(=O)N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880911090 GF On-Demand Anodyne EPHX2 19 46 O=C(NCc1cccc(C(=O)N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880911090 GF On-Demand Anodyne NAMPT 42 46 O=C(NCCN1CCCOCC1)Nc1cncc(C(F)F)c1 ZINC000880911129 DD On-Demand Anodyne CASR 42 39 O=C(NCCN1CCCOCC1)Nc1cncc(C(F)F)c1 ZINC000880911129 DD On-Demand Anodyne EPHX2 23 46 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne HRH2 46 41 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne HRH3 17 41 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne SIGMAR1 26 45 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne FAAH 49 48 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne MCHR1 17 40 Cn1nnc(C(=O)N2CCN(Cc3cccc(OCc4ccccc4)c3)CC2)n1 ZINC000880911151 GD On-Demand Anodyne CCR8 34 44 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880911160 GH On-Demand Anodyne S1PR2 32 46 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880911188 GH On-Demand Anodyne CACNA1H 56 35 O=C(Nc1cncc(C(F)F)c1)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880911188 GH On-Demand Anodyne S1PR2 29 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(SC)CC1 ZINC000880911189 EE On-Demand Anodyne PAPA1_CARPA 32 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC(SC)CC1 ZINC000880911190 EE On-Demand Anodyne PAPA1_CARPA 32 40 Cc1cc(C)c2c(c1)CN(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880911249 EI On-Demand Anodyne P2RY14 43 39 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880911254 EH On-Demand Anodyne NPY5R 35 48 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880911256 EH On-Demand Anodyne NPY5R 35 48 COCCS(=O)(=O)c1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880911278 GF On-Demand Anodyne PRMT3 18 41 COCCS(=O)(=O)c1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880911278 GF On-Demand Anodyne NAMPT 98 44 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880911293 EE On-Demand Anodyne CCR3 62 40 CCc1nc2ccccc2n1C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880911325 GJ On-Demand Anodyne FPR2 27 47 Cc1ccccc1C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880911347 EJ On-Demand Anodyne RBP4 64 39 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2cccc(F)c2F)CC1 ZINC000880911526 FH On-Demand Anodyne NPY2R 63 35 C[C@@H](CCC1CC1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880911556 CH On-Demand Anodyne CCR3 49 35 CCOC(=O)N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880911558 EE On-Demand Anodyne EPHX2 38 41 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880911559 EE On-Demand Anodyne EPHX2 38 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Cc2ccncc2)C1 ZINC000880911608 EH On-Demand Anodyne CCR3 73 33 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880911609 EH On-Demand Anodyne CCR3 73 33 O=C(NCCC(=O)N1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880911622 EF On-Demand Anodyne PRMT3 17 41 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880911626 FI On-Demand Anodyne DRD4 26 42 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880911626 FI On-Demand Anodyne SIGMAR1 25 41 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880911626 FI On-Demand Anodyne CCR3 56 33 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880911627 FI On-Demand Anodyne DRD4 26 42 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880911627 FI On-Demand Anodyne SIGMAR1 25 41 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880911627 FI On-Demand Anodyne CCR3 56 33 C#CCNS(=O)(=O)c1ccc(C(=O)Nc2nc(-c3c[nH]c(C(=O)OC)c3)cs2)cc1 ZINC000880911645 IE On-Demand Mild MPL 42 37 O=C(NCCCNc1cccc(F)c1)Nc1cncc(C(F)F)c1 ZINC000880911674 EH On-Demand Anodyne TBK1 17 40 CC(C)(C)OC(=O)N1CC[C@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)C1 ZINC000880911710 GH On-Demand Anodyne EPHX2 27 42 CC(C)(C)OC(=O)N1CC[C@@]2(CCN(C(=O)Nc3cncc(C(F)F)c3)C2)C1 ZINC000880911711 GH On-Demand Anodyne EPHX2 27 42 O=C(NCc1ccc(N2CCCS2(=O)=O)cc1)Nc1cncc(C(F)F)c1 ZINC000880911713 GF On-Demand Anodyne CDK1 17 41 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880911738 FG On-Demand Anodyne CACNA1I 59 35 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880911739 FG On-Demand Anodyne CACNA1I 59 35 C[C@@H]1CCCN(C(=O)Nc2cncc(C(F)F)c2)[C@@H]1C ZINC000880911742 CH On-Demand Anodyne TRPC6 50 36 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880911745 CH On-Demand Anodyne TRPC6 50 36 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccc(F)cn2)CC1 ZINC000880911756 FF On-Demand Anodyne DGAT1 30 45 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880911783 FI On-Demand Bother MMP2 15 40 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880911783 FI On-Demand Bother MMP8 31 40 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880911783 FI On-Demand Bother MMP9 16 40 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880911783 FI On-Demand Bother MMP1 22 40 COc1ccccc1COC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880911788 GI On-Demand Anodyne SCD1 22 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880911809 FH On-Demand Anodyne CCR3 22 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880911809 FH On-Demand Anodyne FAAH 36 50 COC(=O)c1cc(-c2csc(NC(=O)c3ccc4c(c3)C[C@@H](c3ccccc3)OC4=O)n2)c[nH]1 ZINC000880911833 JJ On-Demand Anodyne MPL 42 37 COC(=O)c1cc(-c2csc(NC(=O)c3ccc4c(c3)C[C@H](c3ccccc3)OC4=O)n2)c[nH]1 ZINC000880911834 JJ On-Demand Anodyne MPL 42 37 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880911929 EH On-Demand Anodyne GRIN2B 54 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880911929 EH On-Demand Anodyne CCR3 34 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880911929 EH On-Demand Anodyne CHRNA7 56 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880911929 EH On-Demand Anodyne C3AR1 46 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2cccnc2)CC1 ZINC000880911929 EH On-Demand Anodyne ACHP_LYMST 25 40 COc1cc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)ncn1 ZINC000880911934 FE On-Demand Anodyne PDGFRB 56 43 O=C(Nc1cncc(C(F)F)c1)N1CCOC2(CCC2)C1 ZINC000880911955 CF On-Demand Anodyne EPHX2 20 44 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](COc2ccccc2)C1 ZINC000880911996 EH On-Demand Anodyne GRIN2B 29 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](COc2ccccc2)C1 ZINC000880911996 EH On-Demand Anodyne CCR3 16 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](COc2ccccc2)C1 ZINC000880911997 EH On-Demand Anodyne GRIN2B 29 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](COc2ccccc2)C1 ZINC000880911997 EH On-Demand Anodyne CCR3 16 42 O=C(Nc1cncc(C(F)F)c1)N1CCC(OCc2ccccc2F)CC1 ZINC000880911998 GI On-Demand Anodyne SCD1 17 42 O=C(Nc1cncc(C(F)F)c1)NC12CCC(CC1)C2 ZINC000880912005 CG On-Demand Anodyne EPHX2 35 44 O=C(Nc1cncc(C(F)F)c1)N1CC(Cc2ccccc2)C1 ZINC000880912013 DH On-Demand Anodyne CCR3 26 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCOCC1 ZINC000880912017 CF On-Demand Anodyne EPHX2 26 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCOCC1 ZINC000880912018 CF On-Demand Anodyne EPHX2 26 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880912058 GH On-Demand Anodyne CACNA1H 42 35 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880912058 GH On-Demand Anodyne FAAH 15 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880912059 GH On-Demand Anodyne CACNA1H 42 35 O=C(Nc1cncc(C(F)F)c1)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880912059 GH On-Demand Anodyne FAAH 15 43 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880912075 FG On-Demand Anodyne INHA 18 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880912076 FG On-Demand Anodyne INHA 18 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC2CCCC2)CC1 ZINC000880912081 FH On-Demand Anodyne EPHX2 40 36 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC2CCCC2)CC1 ZINC000880912081 FH On-Demand Anodyne CXCR3 19 48 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880912128 GF On-Demand Anodyne MTOR 45 34 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880912128 GF On-Demand Anodyne STAT6 55 35 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880912128 GF On-Demand Anodyne NAMPT 23 42 CS(=O)(=O)N1CCN(C(=O)Nc2cncc(C(F)F)c2)Cc2ccccc21 ZINC000880912133 GF On-Demand Anodyne NPY5R 21 40 O=C(Nc1cncc(C(F)F)c1)N(CCO)CCN1CCOCC1 ZINC000880912246 ED On-Demand Anodyne CASR 74 58 O=C(Nc1cncc(C(F)F)c1)N1CCc2c[nH]nc2C1 ZINC000880912247 CE On-Demand Anodyne MAPK1 42 33 O=C(Nc1cncc(C(F)F)c1)N1CCOC2(CCCCCC2)C1 ZINC000880912250 EH On-Demand Anodyne EPHX2 17 46 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccc(F)c(F)c2C1 ZINC000880912251 EH On-Demand Anodyne MAPK1 41 35 COCCCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880912276 FH On-Demand Anodyne HRH2 30 40 COCCCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880912276 FH On-Demand Anodyne ROCK1 26 40 COCCCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880912276 FH On-Demand Anodyne ROCK2 42 49 COCCCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880912276 FH On-Demand Anodyne PDS 64 35 COCCC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912282 FE On-Demand Anodyne C3AR1 41 38 COCCC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912282 FE On-Demand Anodyne EPHX2 45 46 COCCC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912282 FE On-Demand Anodyne CXCR3 15 43 CCC(=O)N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912296 DE On-Demand Anodyne EPHX2 38 53 CCC(=O)N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912297 DE On-Demand Anodyne EPHX2 38 53 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccccc1[N+](=O)[O-])C1CC1 ZINC000880912298 FI On-Demand Bother COLA 122 44 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880912381 FH On-Demand Anodyne CASR 42 38 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880912381 FH On-Demand Anodyne SIGMAR1 31 42 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880912381 FH On-Demand Anodyne CCR5 42 52 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880912381 FH On-Demand Anodyne MLNR 41 35 CN(C(=O)Nc1cncc(C(F)F)c1)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880912381 FH On-Demand Anodyne MCHR1 30 42 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880912382 FH On-Demand Anodyne CASR 42 38 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880912382 FH On-Demand Anodyne SIGMAR1 31 42 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880912382 FH On-Demand Anodyne CCR5 42 52 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880912382 FH On-Demand Anodyne MLNR 41 35 CN(C(=O)Nc1cncc(C(F)F)c1)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880912382 FH On-Demand Anodyne MCHR1 30 42 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccccc2[C@@H]1CO ZINC000880912383 EG On-Demand Anodyne TRPM8 38 46 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccccc2[C@H]1CO ZINC000880912384 EG On-Demand Anodyne TRPM8 38 46 O=C(Nc1cncc(C(F)F)c1)N[C@H](c1cccnc1)C1CC1 ZINC000880912387 DH On-Demand Anodyne NAMPT 19 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H](c1cccnc1)C1CC1 ZINC000880912388 DH On-Demand Anodyne NAMPT 19 40 CC(C)CN1CCC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912398 EH On-Demand Anodyne CCR3 82 37 CC(C)CN1CCC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912399 EH On-Demand Anodyne CCR3 82 37 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880912412 FF On-Demand Anodyne XIAP 15 49 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880912413 FF On-Demand Anodyne XIAP 15 49 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2O)CC1 ZINC000880912434 EG On-Demand Anodyne NPY2R 67 35 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccc(F)cc2C1 ZINC000880912459 DH On-Demand Anodyne MAPK1 40 35 O=C(Nc1cncc(C(F)F)c1)NC1CCC(F)(F)CC1 ZINC000880912463 DH On-Demand Anodyne EPHX2 29 40 COCC1(O)CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912504 DE On-Demand Anodyne S1PR2 30 42 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne HTR1A 40 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne DRD2 35 43 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne ADRA1D 44 43 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne ADRA1A 37 43 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne ADRA1B 33 43 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912512 FG On-Demand Anodyne DRD3 41 36 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne HTR1A 40 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne DRD2 35 43 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne ADRA1D 44 43 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne ADRA1A 37 43 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne ADRA1B 33 43 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880912513 FG On-Demand Anodyne DRD3 41 36 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912533 GG On-Demand Anodyne SIGMAR1 24 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912533 GG On-Demand Anodyne CCR3 51 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912533 GG On-Demand Anodyne MCHR1 15 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912534 GG On-Demand Anodyne SIGMAR1 24 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912534 GG On-Demand Anodyne CCR3 51 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912534 GG On-Demand Anodyne MCHR1 15 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912535 GG On-Demand Anodyne SIGMAR1 24 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912535 GG On-Demand Anodyne CCR3 51 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@@H]1CO ZINC000880912535 GG On-Demand Anodyne MCHR1 15 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912536 GG On-Demand Anodyne SIGMAR1 24 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912536 GG On-Demand Anodyne CCR3 51 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CN(Cc2ccccc2)CC[C@H]1CO ZINC000880912536 GG On-Demand Anodyne MCHR1 15 41 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880912543 FG On-Demand Clean PDGFRB 54 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880912547 FF On-Demand Anodyne EPHX2 42 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880912548 FF On-Demand Anodyne EPHX2 42 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880912549 FF On-Demand Anodyne EPHX2 42 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880912550 FF On-Demand Anodyne EPHX2 42 37 O=C(Nc1cncc(C(F)F)c1)N1CCc2c(F)cccc2C1 ZINC000880912556 DH On-Demand Anodyne P2RY14 44 39 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880912604 FF On-Demand Anodyne EPHX2 40 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880912605 FF On-Demand Anodyne EPHX2 40 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880912606 FF On-Demand Anodyne EPHX2 40 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880912607 FF On-Demand Anodyne EPHX2 40 37 O=C(Nc1cncc(C(F)F)c1)N[C@H](CO)c1ccc(C(F)(F)F)cc1 ZINC000880912617 GH On-Demand Anodyne EPHX2 15 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H](CO)c1ccc(C(F)(F)F)cc1 ZINC000880912618 GH On-Demand Anodyne EPHX2 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880912644 FF On-Demand Anodyne PDGFRB 48 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ncccc2F)CC1 ZINC000880912644 FF On-Demand Anodyne TRPV1 17 57 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1CN1CCOCC1 ZINC000880912659 EE On-Demand Anodyne CASR 38 40 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880912697 GF On-Demand Anodyne NPFFR2 41 42 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880912697 GF On-Demand Anodyne NPFFR1 51 42 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880912698 GF On-Demand Anodyne NPFFR2 41 42 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880912698 GF On-Demand Anodyne NPFFR1 51 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](N2CCCCC2)C1 ZINC000880912713 DG On-Demand Anodyne L3MBTL3 84 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](N2CCCCC2)C1 ZINC000880912714 DG On-Demand Anodyne L3MBTL3 84 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880912717 GG On-Demand Anodyne FAAH 26 47 O=C(NCC1CCN(C(=O)c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880912722 GH On-Demand Anodyne GRIN2B 49 39 O=C(NCC1CCN(C(=O)c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880912722 GH On-Demand Anodyne EPHX2 25 50 O=C(NCC1CCN(C(=O)c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880912722 GH On-Demand Anodyne NAMPT 19 42 O=C(NCc1ccccc1OCC1CC1)Nc1cncc(C(F)F)c1 ZINC000880912732 EI On-Demand Anodyne ADRB1 41 31 Cn1cc(CNC(=O)Nc2cncc(C(F)F)c2)cn1 ZINC000880912736 CE On-Demand Anodyne NAMPT 37 44 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)CN1CCOCC1 ZINC000880912767 GG On-Demand Anodyne CASR 48 40 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)CN1CCOCC1 ZINC000880912767 GG On-Demand Anodyne TACR2 19 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)CN1CCOCC1 ZINC000880912768 GG On-Demand Anodyne CASR 48 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)CN1CCOCC1 ZINC000880912768 GG On-Demand Anodyne TACR2 19 42 COc1ccc(CN(CCO)C(=O)Nc2cncc(C(F)F)c2)c(OC)c1 ZINC000880912783 GG On-Demand Anodyne ROCK2 17 43 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880912811 GH On-Demand Anodyne GPR119 39 42 CC(C)(C)NC(=O)CN1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912812 GF On-Demand Anodyne CACNA1I 79 51 O=C(Nc1cncc(C(F)F)c1)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880912815 FE On-Demand Anodyne EPHX2 36 41 N#CCCN(CCN1CCOCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880912870 FE On-Demand Mild CASR 70 54 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](OCCCc2ccccc2)C1 ZINC000880912874 GI On-Demand Anodyne FKBP1A 46 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](OCCCc2ccccc2)C1 ZINC000880912875 GI On-Demand Anodyne FKBP1A 46 43 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880912882 FI On-Demand Anodyne CCR5 22 40 O=C(Nc1cncc(C(F)F)c1)N(Cc1cccc([N+](=O)[O-])c1)C1CC1 ZINC000880912894 FI On-Demand Bother CACNA1D 48 32 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1=O ZINC000880912965 GF On-Demand Anodyne CCKAR 30 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1=O ZINC000880912965 GF On-Demand Anodyne CCKBR 42 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1=O ZINC000880912967 GF On-Demand Anodyne CCKAR 30 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1=O ZINC000880912967 GF On-Demand Anodyne CCKBR 42 40 O=C(Nc1cncc(C(F)F)c1)N(CCO)CCc1ccccc1 ZINC000880913026 EG On-Demand Anodyne CASR 40 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(C2CCC2)CC1 ZINC000880913058 DF On-Demand Anodyne HRH3 20 40 O=C(Nc1cncc(C(F)F)c1)N1CCc2cncnc2C1 ZINC000880913059 DE On-Demand Anodyne MAPK1 51 35 O=C(NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1)c1ccccc1 ZINC000880913063 FG On-Demand Anodyne DRD4 15 40 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880913073 GF On-Demand Anodyne P2RX3 25 41 C[C@H](CN1CCN(c2ccccn2)CC1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880913073 GF On-Demand Anodyne PRNP 40 36 O=C(NC[C@H]1CCCN(C(=O)Nc2cncc(C(F)F)c2)C1)c1ccccc1 ZINC000880913177 GH On-Demand Anodyne CACNA1I 59 33 COC(OC)c1ccc(C(=O)N2CCC(SC)CC2)o1 ZINC000880913209 CF On-Demand Anodyne L3MBTL3 17 44 O=C(Nc1cncc(C(F)F)c1)N1CCOC2(CCOCC2)C1 ZINC000880913228 EE On-Demand Anodyne EPHX2 18 44 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne DRD2 15 42 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne DRD4 38 42 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne ACHE 44 41 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne SIGMAR1 41 47 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne CCR3 29 43 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne CCR5 29 53 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(Cc2ccccc2)CC1 ZINC000880913262 FI On-Demand Anodyne MCHR1 42 41 O=C(NCc1ccccc1OC1CCC1)Nc1cncc(C(F)F)c1 ZINC000880913275 EI On-Demand Anodyne PDE4A 19 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880913290 FF On-Demand Anodyne EPHX2 35 45 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880913292 FF On-Demand Anodyne EPHX2 35 45 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne KCNQ2 60 34 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne NPY2R 51 34 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne SCN2A 17 41 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne MTOR 47 39 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne SCN10A 25 52 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne STAT6 54 35 O=C(NCc1ccccc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880913294 FG On-Demand Anodyne NAMPT 24 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880913387 FF On-Demand Anodyne CXCR3 17 43 CN1CCC(CNC(=O)Nc2cncc(C(F)F)c2)(N2CCCCC2)CC1 ZINC000880913428 GG On-Demand Anodyne HCN1 40 36 O=C(Nc1cncc(C(F)F)c1)N1CCOC2(CCCC2)C1 ZINC000880913523 DG On-Demand Anodyne EPHX2 19 44 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913539 EH On-Demand Anodyne NPY5R 33 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880913541 FF On-Demand Anodyne CXCR3 17 43 O=C(Nc1cncc(C(F)F)c1)Nc1ccc(NC[C@@H]2CCCO2)c(F)c1 ZINC000880913568 GI On-Demand Anodyne TNK2 31 44 O=C(Nc1cncc(C(F)F)c1)Nc1ccc(NC[C@H]2CCCO2)c(F)c1 ZINC000880913571 GI On-Demand Anodyne TNK2 31 44 CN1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880913579 CE On-Demand Anodyne CCR3 36 40 CN1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880913579 CE On-Demand Anodyne CACNA1I 62 35 O=C(Nc1cncc(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880913585 FE On-Demand Anodyne CASR 43 39 O=C(Nc1cncc(C(F)F)c1)Nc1cnn(CCN2CCOCC2)c1 ZINC000880913585 FE On-Demand Anodyne EPHX2 24 42 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880913598 GG On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880913599 GG On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880913601 GG On-Demand Anodyne CASR 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCOC[C@H]1C[C@H](O)c1ccccc1 ZINC000880913603 GG On-Demand Anodyne CASR 44 39 CCN1CCC[C@@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880913610 CF On-Demand Anodyne CCR3 53 33 CCN1CCC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880913612 CF On-Demand Anodyne CCR3 53 33 O=C(NCCCCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880913648 EH On-Demand Anodyne CHRNA7 25 55 O=C(NCCCCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880913648 EH On-Demand Anodyne HNMT 41 35 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913718 FI On-Demand Anodyne DRD4 23 40 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913718 FI On-Demand Anodyne ACHE 40 42 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913718 FI On-Demand Anodyne SIGMAR1 33 41 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913718 FI On-Demand Anodyne CCR3 51 36 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913718 FI On-Demand Anodyne CCR5 19 41 CN(C[C@@H](c1cccs1)N1CCOCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880913722 GH On-Demand Anodyne CASR 42 37 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880913726 DG On-Demand Anodyne HTR3A 34 44 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ncnc3ccsc23)CC1 ZINC000880913761 GG On-Demand Anodyne PDGFRB 62 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ncnc3ccsc23)CC1 ZINC000880913761 GG On-Demand Anodyne SIRT3 40 31 COc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1F ZINC000880913762 GH On-Demand Clean PDGFRB 48 42 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1CN1CCOCC1 ZINC000880913769 FF On-Demand Anodyne CASR 44 41 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1CN1CCOCC1 ZINC000880913770 FF On-Demand Anodyne CASR 44 41 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cncc(C(F)F)c1 ZINC000880913783 GF On-Demand Anodyne EPHX2 21 46 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CC1)OCc1ccccc12 ZINC000880913803 FI On-Demand Anodyne NPY5R 35 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880913851 GG On-Demand Anodyne GRIN2B 17 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880913851 GG On-Demand Anodyne C3AR1 49 47 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880913853 GG On-Demand Anodyne GRIN2B 17 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(C(=O)CCc2ccccc2)C1 ZINC000880913853 GG On-Demand Anodyne C3AR1 49 47 C[C@@H](C[C@H](O)c1ccc(F)cc1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880913912 FH On-Demand Anodyne CCR3 52 37 CN(C[C@H](O)CN1CCOCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914062 ED On-Demand Anodyne CASR 46 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](COCc2ccccc2)C1 ZINC000880914096 FI On-Demand Anodyne GRIN2B 51 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880914098 FI On-Demand Anodyne GRIN2B 51 43 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne HTR1A 51 46 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne DRD2 27 46 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne HTR2A 37 41 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne DRD3 37 43 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne CASR 61 46 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne HTR7 65 48 CN(CCN1CCN(c2ccccc2)CC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914117 GG On-Demand Anodyne NPY2R 59 38 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880914128 EI On-Demand Anodyne RBP4 63 42 COc1ccccc1[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880914129 EI On-Demand Anodyne RBP4 63 42 O=C(Nc1cncc(C(F)F)c1)N1CCCN(C2CCCC2)CC1 ZINC000880914155 EH On-Demand Anodyne HRH3 23 42 O=C(Nc1cncc(C(F)F)c1)N1CCCN(C2CCCC2)CC1 ZINC000880914155 EH On-Demand Anodyne L3MBTL3 40 33 COCc1cc(CNC(=O)Nc2cncc(C(F)F)c2)ccc1F ZINC000880914161 EH On-Demand Anodyne ROCK2 15 41 COCCOc1ccc(NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880914162 EH On-Demand Anodyne EPHX2 17 49 COCCOc1ccc(NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880914162 EH On-Demand Anodyne CA12 17 41 COCCOc1ccc(NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880914162 EH On-Demand Anodyne PDGFRA 45 35 COCCOc1ccc(NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880914162 EH On-Demand Anodyne CA9 17 41 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1cncc(C(F)F)c1 ZINC000880914169 FG On-Demand Anodyne NAMPT 40 40 C[C@H](C[C@@H](O)c1ccc(F)cc1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914184 FH On-Demand Anodyne CCR3 52 37 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880914192 GJ On-Demand Anodyne EPHX2 24 50 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880914192 GJ On-Demand Anodyne SCD1 45 67 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880914192 GJ On-Demand Anodyne SCD 30 48 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914198 FG On-Demand Anodyne ACE 23 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914198 FG On-Demand Anodyne MME 17 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914198 FG On-Demand Anodyne NPY1R 28 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914199 FG On-Demand Anodyne ACE 23 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914199 FG On-Demand Anodyne MME 17 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880914199 FG On-Demand Anodyne NPY1R 28 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914223 FG On-Demand Anodyne EPHX2 17 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914224 FG On-Demand Anodyne EPHX2 17 40 C[C@@H](CCc1cccn1C)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914279 DH On-Demand Anodyne CCR3 53 36 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCCCC2)C1 ZINC000880914306 DI On-Demand Anodyne EPHX2 28 44 Cn1ccnc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1=O ZINC000880914307 FD On-Demand Anodyne PDGFRB 42 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880914353 CD On-Demand Anodyne UL80 41 40 Cc1ccc(C[C@@H](C)N(C)C(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880914366 EI On-Demand Anodyne NPY5R 33 46 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880914377 FE On-Demand Anodyne GRM4 45 38 NC(=O)c1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880914384 GE On-Demand Anodyne PRNP 40 33 NC(=O)c1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880914384 GE On-Demand Anodyne STAT6 55 32 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H](N2CCCC2)C1 ZINC000880914422 EH On-Demand Anodyne L3MBTL3 48 36 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H](N2CCCC2)C1 ZINC000880914423 EH On-Demand Anodyne L3MBTL3 48 36 Cc1nc(CN2CCC(CNC(=O)Nc3cncc(C(F)F)c3)CC2)oc1C ZINC000880914429 GH On-Demand Anodyne CCR3 23 41 Cc1nc(CN2CCC(CNC(=O)Nc3cncc(C(F)F)c3)CC2)oc1C ZINC000880914429 GH On-Demand Anodyne CACNA1I 55 35 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880914442 FF On-Demand Anodyne CXCR3 17 42 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880914443 FF On-Demand Anodyne CXCR3 17 42 CN1CCC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880914457 CE On-Demand Anodyne CCR3 75 34 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880914467 DH On-Demand Anodyne CFTR 57 36 C[C@H]1Cc2ccccc2CN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880914468 DH On-Demand Anodyne CFTR 57 36 O=C(Nc1cncc(C(F)F)c1)N1CCc2c(F)ccc(F)c2C1 ZINC000880914507 EH On-Demand Anodyne P2RY14 41 39 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880914679 GG On-Demand Anodyne SIGMAR1 22 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880914679 GG On-Demand Anodyne CCR3 47 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880914680 GG On-Demand Anodyne SIGMAR1 22 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880914680 GG On-Demand Anodyne CCR3 47 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880914681 GG On-Demand Anodyne SIGMAR1 22 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C[C@@H]1CO ZINC000880914681 GG On-Demand Anodyne CCR3 47 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880914683 GG On-Demand Anodyne SIGMAR1 22 40 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C[C@H]1CO ZINC000880914683 GG On-Demand Anodyne CCR3 47 42 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCOCC2)C1 ZINC000880914693 DG On-Demand Anodyne EPHX2 31 40 Cc1ccccc1[C@H](CO)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914703 DG On-Demand Anodyne CTSA 53 32 Cc1ccccc1[C@@H](CO)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880914704 DG On-Demand Anodyne CTSA 53 32 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914712 FG On-Demand Anodyne F13A1 16 41 O=C(Nc1cncc(C(F)F)c1)N(Cc1ccccc1)CC1CCOCC1 ZINC000880914726 GI On-Demand Anodyne CASR 46 42 CC(C)(C)OC(=O)NC1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914737 GH On-Demand Anodyne EPHX2 41 34 COc1ccccc1C[C@@H](C)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914746 EI On-Demand Anodyne NPY5R 35 44 COc1ccccc1C[C@H](C)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914747 EI On-Demand Anodyne NPY5R 35 44 CN(c1ccccc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914751 FI On-Demand Anodyne SFRP1 45 33 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1c1nc(-c2ccccc2)no1 ZINC000880914781 GJ On-Demand Anodyne CPT1A 105 51 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1c1nc(-c2ccccc2)no1 ZINC000880914781 GJ On-Demand Anodyne GRM5 23 54 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@H]1c1nc(-c2ccccc2)no1 ZINC000880914781 GJ On-Demand Anodyne SMO 38 40 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1c1nc(-c2ccccc2)no1 ZINC000880914785 GJ On-Demand Anodyne CPT1A 105 51 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1c1nc(-c2ccccc2)no1 ZINC000880914785 GJ On-Demand Anodyne GRM5 23 54 O=C(Nc1cncc(C(F)F)c1)N1CCCC[C@@H]1c1nc(-c2ccccc2)no1 ZINC000880914785 GJ On-Demand Anodyne SMO 38 40 O=C(NCC1(c2cccc(F)c2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914800 EI On-Demand Anodyne SOAT1 16 44 CCN(Cc1ccc(OC)cc1OC)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914817 FI On-Demand Anodyne ROCK2 17 42 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914818 FI On-Demand Mild ROCK2 30 44 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914818 FI On-Demand Mild PDS 47 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914829 FI On-Demand Mild ROCK2 30 44 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914829 FI On-Demand Mild PDS 47 36 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880914843 FI On-Demand Anodyne CCR2 25 57 COC(=O)C1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914844 EF On-Demand Anodyne EPHX2 41 37 COc1ccnc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)n1 ZINC000880914864 FE On-Demand Anodyne PDGFRB 48 39 CN(CCN1CCOCC1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880914876 DD On-Demand Anodyne CASR 65 50 CCOc1cc(CNC(=O)Nc2cncc(C(F)F)c2)ccc1OC ZINC000880914884 FH On-Demand Anodyne ROCK2 20 49 CCOc1cc(CNC(=O)Nc2cncc(C(F)F)c2)ccc1OC ZINC000880914884 FH On-Demand Anodyne ENPP1 41 33 CCOc1cc(CNC(=O)Nc2cncc(C(F)F)c2)ccc1OC ZINC000880914884 FH On-Demand Anodyne DRTS_TRYCR 48 35 O=C(Nc1cncc(C(F)F)c1)N1CCc2c(Cl)cccc2C1 ZINC000880914887 EI On-Demand Anodyne MAPK1 40 33 O=C(Nc1cncc(C(F)F)c1)N1CCc2c(Cl)cccc2C1 ZINC000880914887 EI On-Demand Anodyne P2RY14 41 38 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Cc2ccc(F)cc2)C1 ZINC000880914890 EI On-Demand Anodyne GRIN2B 43 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](Cc2ccc(F)cc2)C1 ZINC000880914890 EI On-Demand Anodyne CCR3 144 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Cc2ccc(F)cc2)C1 ZINC000880914893 EI On-Demand Anodyne GRIN2B 43 43 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](Cc2ccc(F)cc2)C1 ZINC000880914893 EI On-Demand Anodyne CCR3 144 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000880914904 GG On-Demand Anodyne CASR 55 44 O=C(Nc1cncc(C(F)F)c1)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000880914905 GG On-Demand Anodyne CASR 55 44 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccccc2F)CC1 ZINC000880914911 EJ On-Demand Anodyne RBP4 59 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(-c3ccccc3)no2)CC1 ZINC000880914928 GI On-Demand Anodyne PRCP 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(-c3ccccc3)no2)CC1 ZINC000880914928 GI On-Demand Anodyne GRM5 19 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(-c3ccccc3)no2)CC1 ZINC000880914928 GI On-Demand Anodyne SMO 50 56 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc(-c3ccccc3)no2)CC1 ZINC000880914928 GI On-Demand Anodyne ETHR 64 51 O=C(NC[C@@H](O)COc1ccc(F)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880914929 FF On-Demand Anodyne ADRB1 48 35 O=C(NC[C@H](O)COc1ccc(F)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880914931 FF On-Demand Anodyne ADRB1 48 35 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914932 GH On-Demand Anodyne EPHX2 30 47 CCOc1ccccc1CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880914937 DH On-Demand Anodyne ADRB1 41 31 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880914942 DI On-Demand Anodyne EPHX2 23 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880914942 DI On-Demand Anodyne RBP4 54 35 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](c2ccccc2)C1 ZINC000880914942 DI On-Demand Anodyne ADAM10 22 41 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880914944 DI On-Demand Anodyne EPHX2 23 40 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880914944 DI On-Demand Anodyne RBP4 54 35 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](c2ccccc2)C1 ZINC000880914944 DI On-Demand Anodyne ADAM10 22 41 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne HTR1A 42 45 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne DRD2 32 45 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne ADRA1D 18 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne HTR2A 38 44 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne HTR2C 27 40 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne ADRA1A 19 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne DRD3 52 44 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne HTR7 39 40 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne NPY1R 15 42 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne CCR3 40 43 O=C(NCCCN1CCN(c2ccncc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880914950 GF On-Demand Anodyne CHEK1 41 31 O=C(Nc1cncc(C(F)F)c1)N1CCC2(CCCC2)C1 ZINC000880914960 CH On-Demand Anodyne EPHX2 29 42 COCCCOc1cccc(NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914969 FI On-Demand Anodyne EPHX2 22 44 COCCCOc1cccc(NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880914969 FI On-Demand Anodyne KCNK3 40 33 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1Cc1ccc(F)cc1 ZINC000880914981 EI On-Demand Anodyne CCR3 104 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1Cc1ccc(F)cc1 ZINC000880914982 EI On-Demand Anodyne CCR3 104 40 CCC1(O)CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880914991 CF On-Demand Anodyne S1PR2 31 43 CCCCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915008 EG On-Demand Anodyne EPHX2 38 41 CCCCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915008 EG On-Demand Anodyne CXCR3 18 46 CCn1nc2c(cc1=O)CN(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880915010 EE On-Demand Anodyne P2RY14 48 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCO)CC1 ZINC000880915039 DD On-Demand Anodyne CXCR3 19 46 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880915103 DF On-Demand Anodyne CCR3 25 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(CC2CC2)C1 ZINC000880915103 DF On-Demand Anodyne CXCR3 16 44 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880915104 DF On-Demand Anodyne CCR3 25 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(CC2CC2)C1 ZINC000880915104 DF On-Demand Anodyne CXCR3 16 44 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915108 GG On-Demand Anodyne BMP1 55 36 COc1ccccc1[C@@H](O)CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880915117 EF On-Demand Anodyne ADRB1 41 31 COc1ccccc1[C@@H](O)CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880915117 EF On-Demand Anodyne SOAT1 37 41 O=C(Nc1ccc(F)cc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915169 GI On-Demand Anodyne EPHX2 21 43 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880915173 GG On-Demand Anodyne EPHX2 48 60 O=C(Nc1cncc(C(F)F)c1)N1CCN2CCCC[C@@H]2C1 ZINC000880915176 DF On-Demand Anodyne L3MBTL3 42 35 O=C(Nc1cncc(C(F)F)c1)N1CCN2CCCC[C@H]2C1 ZINC000880915177 DF On-Demand Anodyne L3MBTL3 42 35 COc1ccc(CC[C@@H](C)NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880915182 EI On-Demand Anodyne CCR3 40 33 COc1ccc(CC[C@H](C)NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880915183 EI On-Demand Anodyne CCR3 40 33 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cncc(C(F)F)c1 ZINC000880915186 FG On-Demand Anodyne MAPK14 23 41 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cncc(C(F)F)c1 ZINC000880915186 FG On-Demand Anodyne ROCK2 23 41 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cncc(C(F)F)c1 ZINC000880915186 FG On-Demand Anodyne NAMPT 37 40 CCOc1ccccc1CCNC(=O)Nc1cncc(C(F)F)c1 ZINC000880915190 EH On-Demand Anodyne ADRB1 43 32 N#CCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915204 DE On-Demand Mild CXCR3 18 45 COc1ccccc1[C@@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915211 FJ On-Demand Anodyne FKBP1A 55 37 COc1ccccc1[C@@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915211 FJ On-Demand Anodyne PDE4A 15 40 COc1ccccc1[C@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915212 FJ On-Demand Anodyne FKBP1A 55 37 COc1ccccc1[C@H]1CCCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915212 FJ On-Demand Anodyne PDE4A 15 40 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915213 FH On-Demand Anodyne NAMPT 55 57 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne HTR1A 66 44 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne DRD2 58 49 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne ADRA1D 68 49 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne HTR1B 16 44 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne ADRA1A 61 49 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne ADRA1B 53 49 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne DRD3 58 40 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne HTR7 43 37 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne NPY1R 20 41 COc1ccccc1N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915215 GH On-Demand Anodyne NPY2R 47 34 O=C(Nc1cncc(C(F)F)c1)N1CCC(COc2ccccc2)CC1 ZINC000880915220 FI On-Demand Anodyne GRIN2B 32 46 O=C(Nc1cncc(C(F)F)c1)N1CCC(COc2ccccc2)CC1 ZINC000880915220 FI On-Demand Anodyne FAAH 16 45 O=C(Nc1cncc(C(F)F)c1)N1CCC(COc2ccccc2)CC1 ZINC000880915220 FI On-Demand Anodyne EPHX2 19 40 COc1ccccc1C[C@@H]1CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915223 FI On-Demand Anodyne ACKR3 62 31 COc1ccccc1C[C@H]1CCCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880915224 FI On-Demand Anodyne ACKR3 62 31 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880915226 GH On-Demand Anodyne ROCK2 26 41 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915232 GG On-Demand Anodyne CCR3 46 39 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915232 GG On-Demand Anodyne CXCR3 27 41 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915232 GG On-Demand Anodyne MCHR1 26 41 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915232 GG On-Demand Anodyne NAMPT 46 38 O=C(NCC(=O)N1CCCc2ccccc21)Nc1cncc(C(F)F)c1 ZINC000880915233 FG On-Demand Anodyne AVPR2 37 43 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1Cc1cccc(F)c1 ZINC000880915236 EI On-Demand Anodyne CCR3 20 41 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1Cc1cccc(F)c1 ZINC000880915237 EI On-Demand Anodyne CCR3 20 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000880915241 GG On-Demand Anodyne GRIN2B 24 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000880915241 GG On-Demand Anodyne HRH4 30 53 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000880915241 GG On-Demand Anodyne AKR1C3 18 45 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880915242 EF On-Demand Anodyne CXCR3 17 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880915243 EF On-Demand Anodyne CXCR3 17 42 COc1ccc(N2CCC(NC(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880915259 GH On-Demand Clean EPHX2 49 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880915306 FG On-Demand Anodyne EPHX2 53 53 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880915306 FG On-Demand Anodyne L3MBTL3 40 33 C=CCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915310 DF On-Demand Mild CXCR3 18 45 Cn1cc(CN2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cn1 ZINC000880915311 FE On-Demand Anodyne FAAH 16 40 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880915312 EG On-Demand Anodyne EPHX2 32 41 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(c2ccccc2)C1 ZINC000880915313 EG On-Demand Anodyne EPHX2 32 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(F)cc2F)CC1 ZINC000880915325 GI On-Demand Anodyne EPHX2 15 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(Oc2ccc(F)cc2F)CC1 ZINC000880915325 GI On-Demand Anodyne SCD1 39 49 O=C(Nc1cncc(C(F)F)c1)N1CCC(CCN2CCOCC2)CC1 ZINC000880915335 FF On-Demand Anodyne CASR 42 38 COc1ccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880915362 GI On-Demand Anodyne PRSS2 44 31 COc1ccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880915362 GI On-Demand Anodyne SCD1 21 45 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne ACE 21 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne MME 25 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne MC4R 50 36 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne TRY2_BOVIN 86 37 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne F2R 53 33 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne CYP51A1 21 41 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne PREP 24 53 O=C(Nc1cncc(C(F)F)c1)N[C@@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915364 GG On-Demand Anodyne ST14 61 36 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne ACE 21 41 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne MME 25 41 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne MC4R 50 36 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne TRY2_BOVIN 86 37 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne F2R 53 33 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne CYP51A1 21 41 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne PREP 24 53 O=C(Nc1cncc(C(F)F)c1)N[C@H](Cc1ccccc1)C(=O)N1CCCC1 ZINC000880915365 GG On-Demand Anodyne ST14 61 36 O=C(NCC(=O)N1CCc2ccccc2C1)Nc1cncc(C(F)F)c1 ZINC000880915366 FF On-Demand Anodyne DPP8 15 42 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880915367 FI On-Demand Anodyne PRCP 52 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880915368 FI On-Demand Anodyne PRCP 52 40 CN(C)CCOc1ccccc1CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880915378 FG On-Demand Anodyne ROCK2 19 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915380 ED On-Demand Anodyne EPHX2 27 41 Cc1cccc2c1CC[C@@H]2NC(=O)Nc1cncc(C(F)F)c1 ZINC000880915389 DI On-Demand Anodyne TRPV1 15 52 Cc1cccc2c1CC[C@H]2NC(=O)Nc1cncc(C(F)F)c1 ZINC000880915390 DI On-Demand Anodyne TRPV1 15 52 O=C(NCc1ccc(C(=O)N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915398 GF On-Demand Anodyne MTOR 47 38 O=C(NCc1ccc(C(=O)N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915398 GF On-Demand Anodyne EPHX2 16 48 O=C(NCc1ccc(C(=O)N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915398 GF On-Demand Anodyne NAMPT 50 48 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915423 GH On-Demand Anodyne EPHX2 55 51 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915424 FH On-Demand Anodyne HTR4 21 44 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915424 FH On-Demand Anodyne SIGMAR1 16 41 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915424 FH On-Demand Anodyne CCR3 78 51 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915424 FH On-Demand Anodyne CACNA1I 44 31 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915425 FH On-Demand Anodyne HTR4 21 44 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915425 FH On-Demand Anodyne SIGMAR1 16 41 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915425 FH On-Demand Anodyne CCR3 78 51 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cncc(C(F)F)c1 ZINC000880915425 FH On-Demand Anodyne CACNA1I 44 31 O=C(NCCCOc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915429 EH On-Demand Anodyne ADRB1 42 34 NC(=O)c1ccc(CN(C(=O)Nc2cncc(C(F)F)c2)C2CC2)cc1 ZINC000880915431 FG On-Demand Anodyne GCGR 18 41 NC(=O)c1ccc(CN(C(=O)Nc2cncc(C(F)F)c2)C2CC2)cc1 ZINC000880915431 FG On-Demand Anodyne GIPR 50 41 COCCN(CCc1ccccc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915432 EH On-Demand Anodyne CASR 40 41 CCOc1cccc([C@@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880915459 EI On-Demand Anodyne PDS 51 42 CCOc1cccc([C@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880915460 EI On-Demand Anodyne PDS 51 42 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880915464 FG On-Demand Anodyne DGAT1 24 42 CN1CCN(c2ncccc2CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915467 GE On-Demand Anodyne TRPV1 29 41 CN1CCN(c2ncccc2CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915467 GE On-Demand Anodyne SCN2A 17 41 CN1CCN(c2ncccc2CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915467 GE On-Demand Anodyne SCN10A 27 42 CN1CCN(c2ncccc2CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915467 GE On-Demand Anodyne NAMPT 41 36 CCOc1cc2c(cc1OCC)CN(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880915472 GI On-Demand Anodyne MAPK1 44 32 O=C(NC[C@@H](O)c1ccccc1C(F)(F)F)Nc1cncc(C(F)F)c1 ZINC000880915484 GH On-Demand Anodyne SOAT1 19 42 O=C(NC[C@H](O)c1ccccc1C(F)(F)F)Nc1cncc(C(F)F)c1 ZINC000880915485 GH On-Demand Anodyne SOAT1 19 42 CC(C)(C)OC(=O)N1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915488 GH On-Demand Anodyne MTOR 22 41 CC(C)(C)OC(=O)N1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915488 GH On-Demand Anodyne CACNA1I 58 35 CC(C)(C)OC(=O)N1CCC(CNC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915488 GH On-Demand Anodyne GPR119 44 42 O=C(NC[C@@H](O)C1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880915489 DG On-Demand Anodyne PRMT3 28 52 O=C(NC[C@H](O)C1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880915490 DG On-Demand Anodyne PRMT3 28 52 O=C(NC[C@H]1CCCN(Cc2cccs2)C1)Nc1cncc(C(F)F)c1 ZINC000880915502 GI On-Demand Anodyne CCR3 61 33 O=C(NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1)C1CCCCC1 ZINC000880915511 GH On-Demand Anodyne EPHX2 31 42 N#Cc1c(F)cccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915521 GG On-Demand Mild NPY2R 49 35 O=C(NCCC(=O)N1CCCCCC1)Nc1cncc(C(F)F)c1 ZINC000880915526 EF On-Demand Anodyne PRMT3 17 41 Cc1noc(C2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)n1 ZINC000880915531 EG On-Demand Anodyne SMO 38 44 Cc1noc(C2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)n1 ZINC000880915531 EG On-Demand Anodyne ETHR 54 35 O=C(NCC(=O)N1CCN(c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880915532 GE On-Demand Anodyne NPY2R 41 33 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2n[nH]c(-c3ccccc3)n2)CC1 ZINC000880915542 GI On-Demand Anodyne AKT2 40 35 O=C(NCCCS(=O)(=O)c1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915544 FG On-Demand Anodyne NAMPT 42 45 COc1ccc(N2CCCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880915550 GH On-Demand Clean PDGFRB 51 39 C=C(C)CN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915556 DG On-Demand Mild CXCR3 18 46 Cc1ccccc1CC(=O)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915562 GG On-Demand Anodyne P2RY14 43 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880915576 EF On-Demand Anodyne EPHX2 43 43 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC(F)F)CC1 ZINC000880915576 EF On-Demand Anodyne CXCR3 20 47 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915577 FG On-Demand Anodyne CACNA1I 47 36 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915578 FG On-Demand Anodyne CACNA1I 47 36 O=C(Nc1cncc(C(F)F)c1)N1CC[C@@H](N2CCCC2)C1 ZINC000880915581 DF On-Demand Anodyne L3MBTL3 85 42 O=C(Nc1cncc(C(F)F)c1)N1CC[C@H](N2CCCC2)C1 ZINC000880915582 DF On-Demand Anodyne L3MBTL3 85 42 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915587 FH On-Demand Anodyne MTOR 20 47 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915587 FH On-Demand Anodyne EPHX2 51 42 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915587 FH On-Demand Anodyne GPR119 45 42 C[C@@H](c1ccc(F)cc1)N(C)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915595 DI On-Demand Anodyne NPY5R 26 40 CCN(Cc1cccc(Cl)c1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915605 EJ On-Demand Anodyne ROCK2 17 43 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915609 FF On-Demand Anodyne ADRB2 20 44 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915609 FF On-Demand Anodyne ADRB1 55 44 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915609 FF On-Demand Anodyne GRIN1 25 40 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915610 FF On-Demand Anodyne ADRB2 20 44 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915610 FF On-Demand Anodyne ADRB1 55 44 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cncc(C(F)F)c1 ZINC000880915610 FF On-Demand Anodyne GRIN1 25 40 CCN1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915617 CE On-Demand Anodyne CCR3 40 38 CCN1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915617 CE On-Demand Anodyne CACNA1I 60 34 COCCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915621 EE On-Demand Anodyne EPHX2 44 37 COCCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915621 EE On-Demand Anodyne CXCR3 19 46 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915623 FH On-Demand Anodyne EPHX2 45 50 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915623 FH On-Demand Anodyne CXCR3 16 43 O=C(NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1)c1ccc(F)cc1 ZINC000880915629 GH On-Demand Anodyne SSTR5 40 38 O=C(NCc1ccc(CN2CCCC2=O)cc1)Nc1cncc(C(F)F)c1 ZINC000880915642 FG On-Demand Anodyne NAMPT 40 42 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915655 FH On-Demand Anodyne EPHX2 23 41 O=C(NCCC1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880915656 CH On-Demand Anodyne PRMT3 26 47 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000880915658 GH On-Demand Anodyne FAAH 17 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000880915658 GH On-Demand Anodyne EPHX2 18 45 CC(C)(C)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915659 EG On-Demand Anodyne EPHX2 45 41 CC(C)(C)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915659 EG On-Demand Anodyne CXCR3 16 43 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880915660 GG On-Demand Bother SSTR1 40 43 CN1CCC[C@H](NC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915662 CE On-Demand Anodyne CCR3 55 32 O=C(Nc1cncc(C(F)F)c1)N1CCC(N2CCCCC2)CC1 ZINC000880915667 EH On-Demand Anodyne L3MBTL3 97 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)c(F)c2)CC1 ZINC000880915671 GI On-Demand Anodyne SIGMAR1 19 54 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)c(F)c2)CC1 ZINC000880915671 GI On-Demand Anodyne SSTR5 49 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)c(F)c2)CC1 ZINC000880915671 GI On-Demand Anodyne CCR3 59 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)c(F)c2)CC1 ZINC000880915671 GI On-Demand Anodyne CXCR3 41 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)c(F)c2)CC1 ZINC000880915671 GI On-Demand Anodyne MCHR1 51 47 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccccc2)CC1 ZINC000880915673 EI On-Demand Anodyne RBP4 41 38 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccccc2)CC1 ZINC000880915673 EI On-Demand Anodyne MCHR1 17 48 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2ccccc2)CC1 ZINC000880915673 EI On-Demand Anodyne SMO 21 40 O=C(NC[C@@H](c1ccccc1)N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880915688 GG On-Demand Anodyne CASR 46 40 O=C(NC[C@H](c1ccccc1)N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880915689 GG On-Demand Anodyne CASR 46 40 N#Cc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880915705 GG On-Demand Mild NPY2R 74 42 N#Cc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880915705 GG On-Demand Mild SLC6A9 20 44 O=C(Nc1cccc(F)c1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915728 GI On-Demand Anodyne CACNA1H 41 35 O=C(Nc1cccc(F)c1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915728 GI On-Demand Anodyne SCD1 16 40 CCCN(Cc1ccc(F)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915730 EJ On-Demand Anodyne SOAT1 15 41 CN(C)CCOc1ccc(CCNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880915739 GG On-Demand Anodyne RAF1 17 42 COc1ccnc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880915745 FF On-Demand Anodyne PDGFRB 52 41 O=C(NCC(=O)N1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880915753 DE On-Demand Anodyne PRMT3 20 50 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](Cc2ccccc2)C1 ZINC000880915762 EJ On-Demand Anodyne GRIN2B 49 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](Cc2ccccc2)C1 ZINC000880915762 EJ On-Demand Anodyne CCR3 96 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](Cc2ccccc2)C1 ZINC000880915763 EJ On-Demand Anodyne GRIN2B 49 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](Cc2ccccc2)C1 ZINC000880915763 EJ On-Demand Anodyne CCR3 96 36 CS(=O)(=O)Nc1cccc2c1CCN(C(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880915765 GF On-Demand Anodyne P2RY14 40 38 Cc1cccc2c1CCN(C(=O)Nc1cncc(C(F)F)c1)C2 ZINC000880915768 DH On-Demand Anodyne P2RY14 55 45 O=C(NC1CCCCC1)NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915770 GH On-Demand Anodyne EPHX2 39 44 C[C@@H](Cn1cncn1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880915780 CD On-Demand Anodyne HIS3 79 37 O=C(NCC1CCN(Cc2cccs2)CC1)Nc1cncc(C(F)F)c1 ZINC000880915790 GI On-Demand Anodyne CCR3 37 41 O=C(NCC1CCN(Cc2cccs2)CC1)Nc1cncc(C(F)F)c1 ZINC000880915790 GI On-Demand Anodyne CACNA1I 42 33 O=C(NCc1ccc(N2CCCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880915795 EH On-Demand Clean NAMPT 58 45 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2ccccc2F)CC1 ZINC000880915805 GH On-Demand Anodyne EPHX2 46 45 CN(C)CCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880915821 FG On-Demand Anodyne ROCK2 40 48 CN(C)CCOc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880915821 FG On-Demand Anodyne PDS 61 34 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cncc(C(F)F)c1 ZINC000880915868 EG On-Demand Anodyne NAMPT 51 42 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915877 EI On-Demand Anodyne ROCK2 18 46 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915877 EI On-Demand Anodyne NPY5R 19 40 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cncc(C(F)F)c1 ZINC000880915886 FG On-Demand Anodyne CACNA1I 55 34 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cncc(C(F)F)c1 ZINC000880915887 FG On-Demand Anodyne CACNA1I 55 34 O=C(NC[C@@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915889 EF On-Demand Anodyne ADRB2 33 41 O=C(NC[C@@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915889 EF On-Demand Anodyne ADRB1 65 46 O=C(NC[C@@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915889 EF On-Demand Anodyne ADRB3 42 46 O=C(NC[C@@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915889 EF On-Demand Anodyne PDS 58 34 O=C(NC[C@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915890 EF On-Demand Anodyne ADRB2 33 41 O=C(NC[C@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915890 EF On-Demand Anodyne ADRB1 65 46 O=C(NC[C@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915890 EF On-Demand Anodyne ADRB3 42 46 O=C(NC[C@H](O)COc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880915890 EF On-Demand Anodyne PDS 58 34 CC(C)(C)OC(=O)N1CC[C@@H](CCNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915901 GH On-Demand Anodyne GPR119 36 42 CC(C)(C)OC(=O)N1CC[C@H](CCNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915902 GH On-Demand Anodyne GPR119 36 42 COc1cc2c(cc1OC)CCN(C(=O)Nc1cncc(C(F)F)c1)CC2 ZINC000880915910 GH On-Demand Anodyne PDGFRB 34 40 N#Cc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915913 FG On-Demand Mild NPY2R 55 38 N#Cc1cccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880915915 FH On-Demand Mild CCR3 24 42 N#Cc1cccc(OC2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880915915 FH On-Demand Mild EPHX2 20 51 O=C(Nc1ccc(F)cc1)N[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915918 GH On-Demand Anodyne CCR3 40 43 O=C(Nc1ccc(F)cc1)N[C@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915918 GH On-Demand Anodyne EPHX2 43 43 O=C(Nc1ccc(F)cc1)N[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915919 GH On-Demand Anodyne CCR3 40 43 O=C(Nc1ccc(F)cc1)N[C@@H]1CCN(C(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915919 GH On-Demand Anodyne EPHX2 43 43 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915941 GH On-Demand Anodyne CACNA1I 46 35 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915945 GH On-Demand Anodyne HTR1A 50 39 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915945 GH On-Demand Anodyne ADRA1D 41 35 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915945 GH On-Demand Anodyne DRD3 45 38 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915945 GH On-Demand Anodyne SOAT1 16 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915946 GH On-Demand Anodyne HTR1A 50 39 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915946 GH On-Demand Anodyne ADRA1D 41 35 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915946 GH On-Demand Anodyne DRD3 45 38 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915946 GH On-Demand Anodyne SOAT1 16 40 COc1ccc(C(=O)N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880915951 GG On-Demand Anodyne PDGFRB 47 38 CC(C)(C)OC(=O)N1CCC[C@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915957 GH On-Demand Anodyne CACNA1I 48 32 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915960 GG On-Demand Clean NPY2R 72 36 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915960 GG On-Demand Clean MTOR 41 37 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915960 GG On-Demand Clean STAT6 45 33 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915960 GG On-Demand Clean NAMPT 37 42 CC(C)(C)OC(=O)N1CCC[C@@H](CNC(=O)Nc2cncc(C(F)F)c2)C1 ZINC000880915961 GH On-Demand Anodyne CACNA1I 48 32 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915966 FI On-Demand Anodyne ROCK2 17 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880915966 FI On-Demand Anodyne ENPP1 61 32 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915974 FF On-Demand Anodyne ADRB1 53 38 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915974 FF On-Demand Anodyne PDS 33 40 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915975 FF On-Demand Anodyne ADRB1 53 38 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cncc(C(F)F)c1 ZINC000880915975 FF On-Demand Anodyne PDS 33 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915989 FD On-Demand Anodyne CCR8 45 34 CN(C(=O)Nc1cncc(C(F)F)c1)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880915990 GH On-Demand Anodyne L3MBTL3 45 35 CC(=O)NCC1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880915995 EE On-Demand Anodyne CACNA1I 41 33 CCc1cccc2c1OCC[C@@H]2NC(=O)Nc1cncc(C(F)F)c1 ZINC000880915998 EI On-Demand Anodyne TRPV1 16 43 CCc1cccc2c1OCC[C@H]2NC(=O)Nc1cncc(C(F)F)c1 ZINC000880916000 EI On-Demand Anodyne TRPV1 16 43 CCOC(=O)N1CCCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916004 EF On-Demand Anodyne P2RY12 43 39 COCCN(Cc1ccccc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880916007 EH On-Demand Anodyne CASR 34 40 O=C(NCc1ccc2c(c1)OCCO2)Nc1cncc(C(F)F)c1 ZINC000880916008 EG On-Demand Anodyne NOS2 59 31 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccc(O)cc2C1 ZINC000880916012 DG On-Demand Anodyne MAPK1 44 33 O=C(Nc1cncc(C(F)F)c1)N(Cc1cccnc1)C1CC1 ZINC000880916014 DH On-Demand Anodyne CHRNA7 40 35 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne DRD4 19 45 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne SIGMAR1 21 47 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne SSTR5 51 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne CCR3 42 42 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne EPHX2 40 42 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne CXCR3 27 50 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccncc2)CC1 ZINC000880916023 FG On-Demand Anodyne MCHR1 45 47 O=C(NCc1cccc(NC(=O)C2CCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916024 FI On-Demand Anodyne NAMPT 42 38 O=C(NCCCOc1ccccc1F)Nc1cncc(C(F)F)c1 ZINC000880916036 EH On-Demand Anodyne ADRB1 45 35 O=C(NCCS(=O)(=O)Cc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880916048 FF On-Demand Anodyne NAMPT 37 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1CCc1ccccc1 ZINC000880916049 EJ On-Demand Anodyne FKBP1A 47 45 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1CCc1ccccc1 ZINC000880916049 EJ On-Demand Anodyne SLC18A2 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1CCc1ccccc1 ZINC000880916049 EJ On-Demand Anodyne PREP 67 35 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1CCc1ccccc1 ZINC000880916050 EJ On-Demand Anodyne FKBP1A 47 45 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1CCc1ccccc1 ZINC000880916050 EJ On-Demand Anodyne SLC18A2 44 39 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1CCc1ccccc1 ZINC000880916050 EJ On-Demand Anodyne PREP 67 35 N#Cc1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)nc1 ZINC000880916059 FF On-Demand Mild PDGFRB 29 43 O=C(NCc1cccnc1OCC(F)(F)F)Nc1cncc(C(F)F)c1 ZINC000880916076 GH On-Demand Anodyne SCN10A 18 52 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1ccc(NC(=O)NC2CC2)cc1 ZINC000880916078 GI On-Demand Anodyne EPHX2 44 40 COCCOc1ncccc1CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880916080 FF On-Demand Anodyne SCN10A 30 42 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3cncc(C(F)F)c3)c2)CCO1 ZINC000880916112 GH On-Demand Anodyne CCR3 18 40 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3cncc(C(F)F)c3)c2)CCO1 ZINC000880916113 GH On-Demand Anodyne CCR3 18 40 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916115 GI On-Demand Anodyne ROCK2 22 41 CCCNC(=O)c1cccc(CNC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916119 FG On-Demand Anodyne ROCK2 26 42 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1ccc(NC(=O)C2CC2)cc1 ZINC000880916123 FI On-Demand Anodyne F7 19 49 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne DRD2 16 52 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne DRD4 23 52 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne HTR2A 18 49 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne SIGMAR1 36 42 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne CCR3 71 45 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne CHRNA7 38 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne CXCR3 20 43 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne MCHR1 28 47 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CCc2ccccc2)CC1 ZINC000880916129 FH On-Demand Anodyne ACHP_LYMST 25 41 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880916136 EJ On-Demand Anodyne TRPM8 19 55 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cncc(C(F)F)c1 ZINC000880916137 EJ On-Demand Anodyne TRPM8 19 55 O=C(Nc1cncc(C(F)F)c1)NC1CCN(CC2CC2)CC1 ZINC000880916146 DG On-Demand Anodyne CXCR3 19 50 O=C(NCC1(c2ccccc2)CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916155 FH On-Demand Anodyne SOAT1 16 44 O=C(NCC1(c2ccccc2)CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916155 FH On-Demand Anodyne ICMT 59 38 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916169 FF On-Demand Anodyne MTOR 59 38 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916169 FF On-Demand Anodyne STAT6 48 33 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916169 FF On-Demand Anodyne NAMPT 43 42 C[C@@H](CNC(=O)Nc1cncc(C(F)F)c1)N1CCC[C@@H](C)C1 ZINC000880916175 EG On-Demand Anodyne CCR3 45 34 O=C(Nc1cncc(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880916184 FI On-Demand Anodyne GRIN2B 37 47 O=C(Nc1cncc(C(F)F)c1)N1CCC(OCc2ccccc2)CC1 ZINC000880916184 FI On-Demand Anodyne SCD1 19 45 CCCOc1ncccc1CNC(=O)Nc1cncc(C(F)F)c1 ZINC000880916192 EH On-Demand Anodyne SCN10A 19 42 C[C@H]1CN(c2ccc(CNC(=O)Nc3cncc(C(F)F)c3)cn2)C[C@@H](C)O1 ZINC000880916193 GG On-Demand Anodyne NAMPT 37 44 C[C@H]1CN(c2ccc(CNC(=O)Nc3cncc(C(F)F)c3)cn2)C[C@H](C)O1 ZINC000880916195 GG On-Demand Anodyne NAMPT 37 44 O=C(NCc1ccc(C(=O)N2CCCCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916196 GH On-Demand Anodyne NAMPT 54 58 O=C(NCc1ccc(N2CCC(CO)CC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916210 GH On-Demand Clean NAMPT 40 39 O=C(NCCCOc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880916226 DH On-Demand Anodyne ADRB1 44 36 O=C(NCCCOc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880916226 DH On-Demand Anodyne HRH2 29 45 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1ccc(N2CCOCC2)cc1 ZINC000880916234 GH On-Demand Clean MTOR 54 38 C[C@H](NC(=O)Nc1cncc(C(F)F)c1)c1ccc(N2CCOCC2)cc1 ZINC000880916234 GH On-Demand Clean STAT6 54 33 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H](N2CCCC2)C1 ZINC000880916241 DG On-Demand Anodyne L3MBTL3 48 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H](N2CCCC2)C1 ZINC000880916242 DG On-Demand Anodyne L3MBTL3 48 36 O=C(NCCN1CCCCCC1)Nc1cncc(C(F)F)c1 ZINC000880916254 DG On-Demand Anodyne CHRNA7 19 48 COc1cccc([C@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916264 DH On-Demand Anodyne ROCK1 15 53 COc1cccc([C@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916264 DH On-Demand Anodyne ROCK2 25 42 COc1cccc([C@@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916265 DH On-Demand Anodyne ROCK1 15 53 COc1cccc([C@@H](C)NC(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916265 DH On-Demand Anodyne ROCK2 25 42 O=C(NCc1ccc(N2CCCCCC2)nc1)Nc1cncc(C(F)F)c1 ZINC000880916266 GI On-Demand Anodyne NAMPT 53 43 O=C(NCCN1CCc2ccccc2C1)Nc1cncc(C(F)F)c1 ZINC000880916270 EG On-Demand Anodyne NOD2 41 34 O=C(Nc1cncc(C(F)F)c1)N1CCCN(c2ccccc2)CC1 ZINC000880916274 EH On-Demand Anodyne FAAH 18 40 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916281 GH On-Demand Anodyne EPHX2 32 45 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916281 GH On-Demand Anodyne NAMPT 41 33 CC(C)CN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916285 EG On-Demand Anodyne EPHX2 39 42 CC(C)CN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916285 EG On-Demand Anodyne CXCR3 20 48 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880916302 FG On-Demand Anodyne NPY2R 24 43 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880916302 FG On-Demand Anodyne FAAH 15 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880916302 FG On-Demand Anodyne EPHX2 15 40 N#Cc1ccc(CN2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880916303 FG On-Demand Mild MLNR 24 40 N#Cc1ccc(CN2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880916303 FG On-Demand Mild FAAH 24 45 O=C(NCCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916315 DF On-Demand Anodyne TBXAS1 39 45 O=C(NCCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916315 DF On-Demand Anodyne HMOX2 45 33 O=C(NCCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916315 DF On-Demand Anodyne QPCT 42 54 CCOc1ccc([C@@H](C)NC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880916320 EI On-Demand Anodyne ACACB 24 46 O=C(NCc1ccnc(N2CCCCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916331 FH On-Demand Anodyne NAMPT 48 42 O=C(NC[C@H]1CCN(c2ccc(F)cc2)C1)Nc1cncc(C(F)F)c1 ZINC000880916332 FH On-Demand Anodyne CCR3 81 39 O=C(NC[C@@H]1CCN(c2ccc(F)cc2)C1)Nc1cncc(C(F)F)c1 ZINC000880916333 FH On-Demand Anodyne CCR3 81 39 O=C(Nc1cncc(C(F)F)c1)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000880916336 EG On-Demand Anodyne PANC 40 31 O=C(Nc1cncc(C(F)F)c1)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000880916337 EG On-Demand Anodyne PANC 40 31 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916339 GG On-Demand Anodyne CASR 44 39 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880916339 GG On-Demand Anodyne NAMPT 48 44 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne TRPV1 24 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne PIK3CA 42 41 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne SCN2A 17 42 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne MTOR 66 39 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne PIK3CG 27 41 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne SCN10A 31 53 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne STAT6 55 34 O=C(NCc1cccnc1N1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916340 FF On-Demand Anodyne NAMPT 49 44 O=C(NCc1ccc(N2CCSCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916341 GH On-Demand Clean NAMPT 42 40 CNC(=O)CN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916353 ED On-Demand Anodyne CXCR3 20 46 O=C(NCc1ccc(N2CCC(O)CC2)c(F)c1)Nc1cncc(C(F)F)c1 ZINC000880916355 GG On-Demand Clean NPY2R 68 38 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916359 FG On-Demand Clean MTOR 60 38 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916359 FG On-Demand Clean EPHX2 15 40 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916359 FG On-Demand Clean STAT6 70 41 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cncc(C(F)F)c1 ZINC000880916359 FG On-Demand Clean NAMPT 56 46 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c1 ZINC000880916364 GH On-Demand Anodyne KCNK3 46 38 O=C(Nc1cncc(C(F)F)c1)NC1CCN(c2ccccc2)CC1 ZINC000880916374 EH On-Demand Anodyne EPHX2 42 47 O=C(Nc1cncc(C(F)F)c1)NC1CCN(c2ccccc2)CC1 ZINC000880916374 EH On-Demand Anodyne CXCR3 15 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880916390 FG On-Demand Anodyne SSTR5 40 37 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880916390 FG On-Demand Anodyne CCR3 20 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880916390 FG On-Demand Anodyne EPHX2 36 46 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880916390 FG On-Demand Anodyne CXCR3 21 45 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccccn2)CC1 ZINC000880916390 FG On-Demand Anodyne MCHR1 20 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(C2CCCC2)CC1 ZINC000880916395 DG On-Demand Anodyne HRH3 15 42 CN(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880916398 GF On-Demand Anodyne CYP2C9 15 44 CN(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880916398 GF On-Demand Anodyne PRMT3 18 40 CN(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880916398 GF On-Demand Anodyne NAMPT 101 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000880916399 GG On-Demand Bother NPY2R 54 33 O=C(NCc1ccc(N2CCCCC2)nc1)Nc1cncc(C(F)F)c1 ZINC000880916403 FH On-Demand Anodyne NAMPT 53 43 O=C(NCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880916418 CF On-Demand Anodyne CHRNA7 19 48 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916419 FI On-Demand Anodyne FKBP1A 53 39 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916419 FI On-Demand Anodyne CCR3 16 49 COc1cccc(C[C@@H]2CCCN2C(=O)Nc2cncc(C(F)F)c2)c1 ZINC000880916419 FI On-Demand Anodyne CHRNA7 22 40 O=C(Nc1cncc(C(F)F)c1)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880916425 FG On-Demand Anodyne NPY2R 20 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne DRD4 22 43 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne KCNH2 17 43 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne SIGMAR1 31 51 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne SSTR5 51 44 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne CCR3 135 50 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne MLNR 46 39 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne CYP2D6 16 40 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne CXCR3 35 47 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne MCHR1 55 50 O=C(Nc1cncc(C(F)F)c1)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880916426 GH On-Demand Anodyne CACNA1G 33 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880916433 GF On-Demand Anodyne TGM2 78 41 O=C(Nc1cncc(C(F)F)c1)N1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000880916433 GF On-Demand Anodyne F13A1 97 42 COCCOc1ccc(CNC(=O)Nc2cncc(C(F)F)c2)cc1 ZINC000880916440 FG On-Demand Anodyne ROCK2 18 40 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne HTR1A 89 59 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne DRD2 65 41 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne DRD4 34 43 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne ADRA1D 73 44 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne HTR1D 19 59 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne HTR1B 23 59 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne HTR2A 23 49 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne ADRA1A 68 44 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne ADRA1B 56 44 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne DRD3 67 40 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne PDGFRB 63 48 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne HTR7 56 52 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne NPY2R 69 37 COc1ccccc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916455 FG On-Demand Anodyne RBP4 23 47 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccnc2)CC1 ZINC000880916464 EF On-Demand Anodyne PTAFR 17 53 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccnc2)CC1 ZINC000880916464 EF On-Demand Anodyne CHRNA7 44 34 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccnc2)CC1 ZINC000880916464 EF On-Demand Anodyne FAAH 35 55 CN(C)[C@@H](CNC(=O)Nc1cncc(C(F)F)c1)c1ccccc1 ZINC000880916469 EG On-Demand Anodyne KCNA5 20 41 COc1ccc(CN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880916474 EH On-Demand Anodyne LTA4H 16 40 COc1ccc(CN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880916474 EH On-Demand Anodyne ROCK2 17 44 COc1ccc(CN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880916474 EH On-Demand Anodyne NPY5R 24 42 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880916477 FG On-Demand Anodyne ABCB1B 45 40 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880916477 FG On-Demand Anodyne ABCB1 17 42 COc1cc2c(cc1OC)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880916477 FG On-Demand Anodyne ABCG2 29 41 CC[C@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916481 CF On-Demand Anodyne NPY2R 52 37 O=C(NCCCc1ccccc1)Nc1cncc(C(F)F)c1 ZINC000880916486 DH On-Demand Anodyne AMP1_PLAFQ 22 40 CCOC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916503 EF On-Demand Anodyne EPHX2 51 44 CCOC(=O)N1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916503 EF On-Demand Anodyne CXCR3 17 42 CCOC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916506 FF On-Demand Anodyne NPY2R 50 33 CCOC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916506 FF On-Demand Anodyne EPHX2 63 52 CCOC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916506 FF On-Demand Anodyne CXCR3 18 41 COc1ncccc1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916507 DF On-Demand Anodyne P2RY1 40 38 COc1ncccc1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916507 DF On-Demand Anodyne ROCK2 25 44 CCN(CC)C(=O)CN1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916508 GE On-Demand Anodyne NPY2R 44 35 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916509 GD On-Demand Anodyne CACNA1H 46 39 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916509 GD On-Demand Anodyne NPY2R 42 35 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916513 GG On-Demand Clean NPY2R 40 33 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916513 GG On-Demand Clean EPHB4 46 33 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916513 GG On-Demand Clean STAT6 58 36 CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916514 DE On-Demand Anodyne NPY2R 50 35 CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916514 DE On-Demand Anodyne CCR3 48 41 CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916514 DE On-Demand Anodyne EPHX2 59 47 CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916514 DE On-Demand Anodyne CXCR3 25 46 CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916514 DE On-Demand Anodyne MCHR1 27 41 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916524 FG On-Demand Anodyne CACNA1H 32 40 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916524 FG On-Demand Anodyne NPY2R 71 43 CCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916524 FG On-Demand Anodyne EPHX2 17 45 CCOC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916532 EF On-Demand Anodyne NPY2R 46 34 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880916551 GH On-Demand Anodyne NPY2R 34 40 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880916551 GH On-Demand Anodyne EPHX2 21 40 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880916551 GH On-Demand Anodyne KCNK3 60 39 Cc1cccc(C(=O)N2CCCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880916551 GH On-Demand Anodyne KCNK9 44 38 O=C(NCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916558 CE On-Demand Anodyne TBXAS1 40 45 O=C(NCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916558 CE On-Demand Anodyne HMOX2 45 33 O=C(NCCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880916558 CE On-Demand Anodyne QPCT 58 57 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916560 EG On-Demand Anodyne BMP1 40 34 CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916565 CD On-Demand Anodyne CACNA1H 29 41 CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916565 CD On-Demand Anodyne HTR1D 15 51 CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916565 CD On-Demand Anodyne HTR1B 19 51 CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916565 CD On-Demand Anodyne EPHX2 21 49 O=C(NCc1ccccc1CN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916572 GG On-Demand Anodyne CASR 45 40 O=C(NCc1ccccc1CN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916572 GG On-Demand Anodyne STAT6 42 32 O=C(NCc1ccccc1CN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880916572 GG On-Demand Anodyne NAMPT 26 40 O=C(NC[C@H]1CN(Cc2ccccc2)CCO1)Nc1cncc(C(F)F)c1 ZINC000880916577 GG On-Demand Anodyne DRD4 19 43 O=C(NC[C@H]1CN(Cc2ccccc2)CCO1)Nc1cncc(C(F)F)c1 ZINC000880916577 GG On-Demand Anodyne CCR3 21 47 O=C(NC[C@@H]1CN(Cc2ccccc2)CCO1)Nc1cncc(C(F)F)c1 ZINC000880916578 GG On-Demand Anodyne DRD4 19 43 O=C(NC[C@@H]1CN(Cc2ccccc2)CCO1)Nc1cncc(C(F)F)c1 ZINC000880916578 GG On-Demand Anodyne CCR3 21 47 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916589 FG On-Demand Anodyne F13A1 16 40 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916589 FG On-Demand Anodyne GPR119 34 41 O=C(Nc1cncc(C(F)F)c1)NC1CCCCCC1 ZINC000880916592 CH On-Demand Anodyne EPHX2 44 45 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916611 FD On-Demand Anodyne ABCB1 30 45 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880916614 GH On-Demand Clean CASR 43 39 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880916614 GH On-Demand Clean EPHB4 49 34 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880916614 GH On-Demand Clean STAT6 56 35 CCNC(=O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916634 CD On-Demand Anodyne F7 23 42 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc(N(C)C)c(F)c2)no1 ZINC000880916643 EH On-Demand Anodyne TRPC6 43 30 Cc1nc(CN2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)oc1C ZINC000880916657 GF On-Demand Anodyne FAAH 15 43 O=C(NCCCN1CCCCCC1)Nc1cncc(C(F)F)c1 ZINC000880916665 EG On-Demand Anodyne CCR3 38 41 O=C(NCCCN1CCCCCC1)Nc1cncc(C(F)F)c1 ZINC000880916665 EG On-Demand Anodyne CHRNA7 24 53 O=C(NCCCN1CCCCCC1)Nc1cncc(C(F)F)c1 ZINC000880916665 EG On-Demand Anodyne HNMT 46 32 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880916678 EF On-Demand Anodyne PDGFRB 40 38 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880916678 EF On-Demand Anodyne FAAH 19 40 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccn2)CC1 ZINC000880916678 EF On-Demand Anodyne DGAT1 22 41 CN(Cc1ccc(Cl)nc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916680 EH On-Demand Anodyne NACHRBETA2 17 41 CCCCCNC(=O)Nc1cncc(C(F)F)c1 ZINC000880916690 CG On-Demand Anodyne ASAH1 69 33 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916692 EF On-Demand Anodyne FDFT1 15 44 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916692 EF On-Demand Anodyne EPHX2 21 40 CC(C)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916696 DF On-Demand Anodyne CACNA1H 39 44 CC(C)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916696 DF On-Demand Anodyne NPY2R 41 33 CCCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916733 EG On-Demand Anodyne HTR4 42 41 CCCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916733 EG On-Demand Anodyne CCR3 69 40 CCCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916733 EG On-Demand Anodyne EPHX2 60 49 CCCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916733 EG On-Demand Anodyne CXCR3 22 43 CCCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916733 EG On-Demand Anodyne MCHR1 48 39 CN(C)c1ccc(NC(=O)N[C@@H](CCCO)c2ccccc2)cc1F ZINC000880916745 EH On-Demand Anodyne NPY2R 55 34 CN(C)c1ccc(NC(=O)N[C@@H](CCCO)c2ccccc2)cc1F ZINC000880916745 EH On-Demand Anodyne UTS2 57 38 CN(C)c1ccc(NC(=O)N[C@H](CCCO)c2ccccc2)cc1F ZINC000880916746 EH On-Demand Anodyne NPY2R 55 34 CN(C)c1ccc(NC(=O)N[C@H](CCCO)c2ccccc2)cc1F ZINC000880916746 EH On-Demand Anodyne UTS2 57 38 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@H](S(C)(=O)=O)C2)cc1F ZINC000880916747 FE On-Demand Anodyne EPHX2 44 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](S(C)(=O)=O)C2)cc1F ZINC000880916748 FE On-Demand Anodyne EPHX2 44 41 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@@H](S(C)(=O)=O)C2)cc1F ZINC000880916749 FE On-Demand Anodyne EPHX2 44 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H](S(C)(=O)=O)C2)cc1F ZINC000880916750 FE On-Demand Anodyne EPHX2 44 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880916758 FG On-Demand Anodyne EPHX2 40 44 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne HTR1A 38 51 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne DRD2 33 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne DRD4 19 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne HTR2A 29 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne HTR2C 19 41 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1cncc(C(F)F)c1 ZINC000880916762 GE On-Demand Anodyne DRD3 43 48 O=C(Nc1cncc(C(F)F)c1)NC1CCC(C(F)(F)F)CC1 ZINC000880916767 EI On-Demand Anodyne EPHX2 43 38 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880916774 EG On-Demand Anodyne NPY2R 46 36 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880916774 EG On-Demand Anodyne PRNP 40 34 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2)CC1 ZINC000880916774 EG On-Demand Anodyne FAAH 21 43 CNC(=O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916781 CC On-Demand Anodyne F7 23 43 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916784 GH On-Demand Anodyne TSPO 27 41 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916784 GH On-Demand Anodyne NPY2R 44 34 O=C(Nc1cncc(C(F)F)c1)NC1CCCCC1 ZINC000880916787 CG On-Demand Anodyne EPHX2 44 45 CCOC(=O)CC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916794 FG On-Demand Anodyne EPHX2 20 41 CNC(=O)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916799 FD On-Demand Anodyne DRD4 16 42 CNC(=O)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916799 FD On-Demand Anodyne EPHX2 48 42 CNC(=O)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916799 FD On-Demand Anodyne CXCR3 22 43 CNC(=O)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880916799 FD On-Demand Anodyne MCHR1 21 40 NC(=O)[C@H](c1ccccc1)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916802 GE On-Demand Anodyne NPY2R 60 39 NC(=O)[C@@H](c1ccccc1)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880916803 GE On-Demand Anodyne NPY2R 60 39 CN(C)c1ccc(NC(=O)Nc2cnn(CC3CC3)c2)cc1F ZINC000880916822 DG On-Demand Anodyne PANC 47 35 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1c1nc2ccccc2s1 ZINC000880916828 FJ On-Demand Anodyne UL80 26 41 C[C@@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)CN1CCOCC1 ZINC000880916832 ED On-Demand Anodyne EPHX2 27 47 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1c1nc2ccccc2s1 ZINC000880916833 FJ On-Demand Anodyne UL80 26 41 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880916836 FJ On-Demand Anodyne HTR1D 26 53 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880916836 FJ On-Demand Anodyne HTR1B 24 53 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880916836 FJ On-Demand Anodyne HTR1F 76 44 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880916836 FJ On-Demand Anodyne CCR2 34 57 CN(C)c1ccc(NC(=O)Nc2cnn(CC(=O)N3CCOCC3)c2)cc1F ZINC000880916844 GD On-Demand Anodyne MTOR 64 36 CN(C)c1ccc(NC(=O)Nc2cnn(CC(=O)N3CCOCC3)c2)cc1F ZINC000880916844 GD On-Demand Anodyne EPHX2 23 48 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccsc2)CC1 ZINC000880916847 FG On-Demand Anodyne FAAH 18 41 CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916868 BD On-Demand Anodyne Q25615_ONCVO 48 33 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C1CCOCC1 ZINC000880916879 DG On-Demand Anodyne NPY2R 43 40 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880916882 CE On-Demand Anodyne EPHX2 23 44 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880916883 CE On-Demand Anodyne EPHX2 23 44 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2cccs2)CC1 ZINC000880916890 FG On-Demand Anodyne FAAH 16 41 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916892 GF On-Demand Anodyne CA2 31 42 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916892 GF On-Demand Anodyne CA4 32 42 C[C@@H](c1cccc(S(N)(=O)=O)c1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916892 GF On-Demand Anodyne CA9 21 42 CN(C)C(=O)c1cccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880916906 FF On-Demand Anodyne ROCK2 27 50 CN(CCN1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916914 DD On-Demand Anodyne HTR2A 18 41 CN(CCN1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916914 DD On-Demand Anodyne CASR 59 48 CN(CCN1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916914 DD On-Demand Anodyne EPHX2 28 48 CN(CCN1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880916914 DD On-Demand Anodyne MCHR1 27 40 CN(C)c1ccc(NC(=O)N[C@H]2CCN3CCC[C@H]3C2)cc1F ZINC000880916922 DF On-Demand Anodyne EPHX2 44 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCN3CCC[C@H]3C2)cc1F ZINC000880916927 DF On-Demand Anodyne EPHX2 44 40 CN(C)c1ccc(NC(=O)N[C@H]2CCN3CCC[C@@H]3C2)cc1F ZINC000880916929 DF On-Demand Anodyne EPHX2 44 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCN3CCC[C@@H]3C2)cc1F ZINC000880916931 DF On-Demand Anodyne EPHX2 44 40 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880916935 EF On-Demand Anodyne CACNA1H 64 48 CCN1CCC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916945 DE On-Demand Anodyne NPY2R 40 33 CCN1CCC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916945 DE On-Demand Anodyne CCR3 66 43 CCN1CCC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916945 DE On-Demand Anodyne EPHX2 48 42 CCN1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916947 DE On-Demand Anodyne NPY2R 40 33 CCN1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916947 DE On-Demand Anodyne CCR3 66 43 CCN1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880916947 DE On-Demand Anodyne EPHX2 48 42 CC(=O)Nc1ccc(CCNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880916951 FG On-Demand Anodyne RAF1 17 42 CN(C)c1ccc(NC(=O)N[C@@H]2CC(=O)N(C(C)(C)C)C2)cc1F ZINC000880916981 EE On-Demand Anodyne EPHX2 41 39 CN(C)c1ccc(NC(=O)N[C@H]2CC(=O)N(C(C)(C)C)C2)cc1F ZINC000880916982 EE On-Demand Anodyne EPHX2 41 39 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne SIGMAR1 15 43 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne NPY1R 30 44 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne CCKAR 47 39 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne NPY2R 50 35 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne CCR3 45 36 CN(C)c1ccc(NC(=O)N[C@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880916995 FF On-Demand Anodyne CCKBR 66 38 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne SIGMAR1 15 43 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne NPY1R 30 44 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne CCKAR 47 39 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne NPY2R 50 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne CCR3 45 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(Cc3ccccc3)C2=O)cc1F ZINC000880917000 FF On-Demand Anodyne CCKBR 66 38 COC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917009 DE On-Demand Anodyne EPHX2 16 43 COc1ccc2c(c1)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880917016 EG On-Demand Anodyne HDAC6 30 40 CCC(=O)N1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917017 EE On-Demand Anodyne EPHX2 26 41 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@@H](O)C2)cc1F ZINC000880917018 CE On-Demand Anodyne EPHX2 47 43 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@H](O)C2)cc1F ZINC000880917019 CE On-Demand Anodyne EPHX2 47 43 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H](O)C2)cc1F ZINC000880917020 CE On-Demand Anodyne EPHX2 47 43 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](O)C2)cc1F ZINC000880917021 CE On-Demand Anodyne EPHX2 47 43 CCS(=O)(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917024 FD On-Demand Anodyne NPY2R 44 34 COCCN(Cc1ccccc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917036 EH On-Demand Anodyne LTA4H 19 40 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917037 EE On-Demand Anodyne CACNA1H 30 40 CC(=O)N(C)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917037 EE On-Demand Anodyne EPHX2 37 42 C[C@@H](Cn1cncn1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917046 DD On-Demand Anodyne HIS3 79 36 O=C(CN1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1)Nc1ccccc1 ZINC000880917056 GF On-Demand Anodyne FAAH 16 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(Cc2ccncc2)CC1 ZINC000880917062 EF On-Demand Anodyne FAAH 28 49 O=C(NCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917073 DD On-Demand Anodyne CASR 49 41 O=C(NCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917073 DD On-Demand Anodyne EPHX2 27 49 O=C(NCCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917087 DD On-Demand Anodyne CASR 49 40 O=C(NCCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917087 DD On-Demand Anodyne CCR3 34 40 O=C(NCCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917087 DD On-Demand Anodyne CHRNA7 17 54 O=C(NCCCN1CCOCC1)Nc1cncc(C(F)F)c1 ZINC000880917087 DD On-Demand Anodyne EPHX2 27 43 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1OC ZINC000880917096 FH On-Demand Anodyne MT-ND1 18 42 COc1ccc(CN(C)C(=O)Nc2cncc(C(F)F)c2)cc1OC ZINC000880917096 FH On-Demand Anodyne ENPP1 62 33 O=C(Nc1cncc(C(F)F)c1)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000880917101 GH On-Demand Anodyne CCR3 32 46 O=C(Nc1cncc(C(F)F)c1)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000880917101 GH On-Demand Anodyne FAAH 23 45 CCN(Cc1cccs1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917105 DI On-Demand Anodyne NPY2R 45 35 CC(=O)Nc1cccc([C@@H](C)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917131 FH On-Demand Anodyne F7 15 45 CC(=O)Nc1cccc([C@H](C)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917133 FH On-Demand Anodyne F7 15 45 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne DRD4 39 57 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne CHRM3 18 43 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne SIGMAR1 33 50 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne SSTR5 41 36 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne CCR3 59 56 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne UTS2R 21 42 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne CCR2 21 44 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne EPHX2 30 43 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne CXCR3 26 43 O=C(Nc1cncc(C(F)F)c1)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880917135 EG On-Demand Anodyne MCHR1 36 51 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne DRD4 39 57 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne CHRM3 18 43 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne SIGMAR1 33 50 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne SSTR5 41 36 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne CCR3 59 56 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne UTS2R 21 42 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne CCR2 21 44 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne EPHX2 30 43 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne CXCR3 26 43 O=C(Nc1cncc(C(F)F)c1)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880917137 EG On-Demand Anodyne MCHR1 36 51 O=C(NCCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880917171 DG On-Demand Anodyne CCR3 38 41 O=C(NCCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880917171 DG On-Demand Anodyne CHRNA7 24 53 O=C(NCCCN1CCCCC1)Nc1cncc(C(F)F)c1 ZINC000880917171 DG On-Demand Anodyne HNMT 46 32 Cc1nc(CN2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)cs1 ZINC000880917174 GG On-Demand Anodyne FAAH 16 41 CCOC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917180 EE On-Demand Anodyne P2RY12 40 45 CCOC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917180 EE On-Demand Anodyne NPY2R 54 34 CCOC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917180 EE On-Demand Anodyne TGM2 20 41 CCOC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917180 EE On-Demand Anodyne F13A1 36 41 Cc1noc(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880917186 EF On-Demand Anodyne SMO 40 48 Cc1noc(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880917186 EF On-Demand Anodyne ETHR 55 36 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C2CC2)CC1 ZINC000880917187 DF On-Demand Anodyne CXCR3 15 42 Cc1cc([C@@H]2CCCN2C(=O)Nc2ccc(N(C)C)c(F)c2)on1 ZINC000880917213 EH On-Demand Anodyne KCNA5 17 40 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1c1cccnc1 ZINC000880917214 DH On-Demand Anodyne CHRNA7 21 44 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1c1cccnc1 ZINC000880917216 DH On-Demand Anodyne CHRNA7 21 44 COc1ccc(CN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1OC ZINC000880917229 FH On-Demand Anodyne MT-ND1 19 44 COc1ccc(CN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1OC ZINC000880917229 FH On-Demand Anodyne ENPP1 67 33 C[C@@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)N1CCOCC1 ZINC000880917238 DD On-Demand Anodyne NPY2R 50 33 C[C@@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)N1CCOCC1 ZINC000880917238 DD On-Demand Anodyne EPHX2 23 46 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917242 GG On-Demand Anodyne NPY2R 66 42 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917242 GG On-Demand Anodyne EPHX2 58 53 CCOCCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917243 CF On-Demand Anodyne CCR3 22 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917265 FD On-Demand Anodyne CCR8 82 39 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917265 FD On-Demand Anodyne SFRP1 42 35 COCCN(Cc1ccccn1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917288 EF On-Demand Anodyne GRM4 33 41 CC[C@@H]1CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917289 CG On-Demand Anodyne NPY2R 50 35 CC[C@H]1CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917290 CG On-Demand Anodyne NPY2R 50 35 CN(C)C(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917307 EE On-Demand Anodyne CACNA1H 28 40 CN(C)C(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917307 EE On-Demand Anodyne EPHX2 20 40 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(C(F)F)c1 ZINC000880917315 EH On-Demand Anodyne BMP1 44 36 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1Cc1ccccc1 ZINC000880917316 EI On-Demand Anodyne FKBP1A 39 42 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@H]1Cc1ccccc1 ZINC000880917316 EI On-Demand Anodyne PREP 68 35 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1Cc1ccccc1 ZINC000880917317 EI On-Demand Anodyne FKBP1A 39 42 O=C(Nc1cncc(C(F)F)c1)N1CCC[C@@H]1Cc1ccccc1 ZINC000880917317 EI On-Demand Anodyne PREP 68 35 CCOC(=O)N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917321 EE On-Demand Anodyne P2RY12 51 40 CN(CCOc1ccccc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880917325 DH On-Demand Anodyne LTA4H 21 40 O=C(NCCc1ccc2c(c1)OCO2)Nc1cncc(C(F)F)c1 ZINC000880917327 EG On-Demand Anodyne NOS2 64 37 N#Cc1ccc(CN2CCCN(C(=O)Nc3cncc(C(F)F)c3)CC2)cc1 ZINC000880917328 GH On-Demand Mild FAAH 19 42 O=C(NCc1ccnc(N2CCCC2)c1)Nc1cncc(C(F)F)c1 ZINC000880917333 EG On-Demand Anodyne NAMPT 47 41 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917347 EF On-Demand Anodyne ADRB1 41 34 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917347 EF On-Demand Anodyne KCNK3 51 40 COc1ccccc1[C@@H](O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917347 EF On-Demand Anodyne KCNK9 48 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917356 EF On-Demand Anodyne CCR3 50 44 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917356 EF On-Demand Anodyne EPHX2 50 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917356 EF On-Demand Anodyne CXCR3 21 45 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2F)CC1 ZINC000880917358 FH On-Demand Anodyne NPY2R 103 38 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ccccc2F)CC1 ZINC000880917358 FH On-Demand Anodyne FAAH 19 41 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917360 EF On-Demand Anodyne CCR3 50 44 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917360 EF On-Demand Anodyne EPHX2 50 42 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(F)(F)F)C2)cc1F ZINC000880917360 EF On-Demand Anodyne CXCR3 21 45 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA2 65 42 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne PTGS2 16 42 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA1 55 41 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA7 23 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA4 61 41 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA12 43 45 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne CA9 46 45 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne MTCA1 45 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917373 GF On-Demand Anodyne P96878_MYCTU 57 45 C[C@H](CCc1ccc(O)cc1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880917381 EH On-Demand Anodyne CCR3 41 33 C[C@@H](CCc1ccc(O)cc1)NC(=O)Nc1cncc(C(F)F)c1 ZINC000880917383 EH On-Demand Anodyne CCR3 41 33 CCOCCCNC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917387 GF On-Demand Anodyne EPHX2 17 41 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917392 EE On-Demand Anodyne CCR3 32 41 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917400 DE On-Demand Anodyne TBXAS1 30 40 C[C@@H](Cn1ccnc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917400 DE On-Demand Anodyne QPCT 28 42 O=C(Nc1cncc(C(F)F)c1)N1CCc2ccccc2C1 ZINC000880917403 DH On-Demand Anodyne P2RY14 43 39 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880917430 FG On-Demand Anodyne EPHX2 45 46 CCOC(=O)N1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917442 FF On-Demand Anodyne P2RY12 30 43 CCN(Cc1ccoc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917452 DH On-Demand Anodyne NPY2R 46 35 O=C(Nc1cncc(C(F)F)c1)N1CCN(c2ncnc3sccc23)CC1 ZINC000880917455 GG On-Demand Anodyne PDGFRB 63 45 Cc1nc(C(C)(C)NC(=O)Nc2ccc(N(C)C)c(F)c2)no1 ZINC000880917474 DF On-Demand Anodyne IMDH_CRYPV 54 33 CCN(CC)C(=O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917500 DD On-Demand Anodyne NPY2R 44 35 CC(C)[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917507 CG On-Demand Anodyne CACNA1H 29 42 CC(C)[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917507 CG On-Demand Anodyne NPY2R 61 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917537 DD On-Demand Anodyne UL80 35 41 Cn1ncc2c(N3CCN(C(=O)Nc4cncc(C(F)F)c4)CC3)ncnc21 ZINC000880917538 GE On-Demand Anodyne PDGFRB 61 44 CN(C)c1ccc(NC(=O)Nc2ccc(CCS(C)(=O)=O)cc2)cc1F ZINC000880917542 GG On-Demand Anodyne P96878_MYCTU 45 41 COCC(C)(C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917545 CE On-Demand Anodyne IMDH_CRYPV 44 32 CN(C)c1ccc(NC(=O)N[C@H]2CCOC3(CCOCC3)C2)cc1F ZINC000880917555 FF On-Demand Anodyne ENV 40 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCOC3(CCOCC3)C2)cc1F ZINC000880917558 FF On-Demand Anodyne ENV 40 35 CC[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@H]1N1CCOCC1 ZINC000880917589 FE On-Demand Anodyne EPHX2 15 42 CC[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@@H]1N1CCOCC1 ZINC000880917595 FE On-Demand Anodyne EPHX2 15 42 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917604 ED On-Demand Anodyne CACNA1H 42 39 CC[C@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917604 ED On-Demand Anodyne NPY2R 60 38 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917606 ED On-Demand Anodyne CACNA1H 42 39 CC[C@@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917606 ED On-Demand Anodyne NPY2R 60 38 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc3ccccc3[nH]2)CC1 ZINC000880917619 FI On-Demand Anodyne SMO 31 41 O=C(Nc1cncc(C(F)F)c1)NC1CCN(C(=O)C2CC2)CC1 ZINC000880917630 EF On-Demand Anodyne EPHX2 50 57 O=C(Nc1cncc(C(F)F)c1)N1CCCN(Cc2ccccc2)CC1 ZINC000880917635 FH On-Demand Anodyne ACHE 18 46 O=C(Nc1cncc(C(F)F)c1)N1CCCN(Cc2ccccc2)CC1 ZINC000880917635 FH On-Demand Anodyne FAAH 38 53 O=C(NCC1(c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880917658 DH On-Demand Anodyne KCNA3 41 35 O=C(NCC1(c2ccccc2)CC1)Nc1cncc(C(F)F)c1 ZINC000880917658 DH On-Demand Anodyne SOAT1 17 47 COc1ccc(CN(C(=O)Nc2cncc(C(F)F)c2)C2CC2)cc1 ZINC000880917677 EI On-Demand Anodyne GIPR 38 40 N#Cc1cccnc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917680 FF On-Demand Mild P2RY12 17 48 N#Cc1cccnc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917680 FF On-Demand Mild PDGFRB 44 39 N#Cc1cccnc1N1CCN(C(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917680 FF On-Demand Mild TRPV1 17 65 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2ccccc2)CC1 ZINC000880917686 EJ On-Demand Anodyne GRIN2B 91 43 O=C(Nc1cncc(C(F)F)c1)N1CCC(Cc2ccccc2)CC1 ZINC000880917686 EJ On-Demand Anodyne CCR3 66 44 CCN(Cc1ccncc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917698 DG On-Demand Anodyne NPY2R 41 34 COc1ccc([C@H](CCO)NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880917705 FG On-Demand Anodyne UTS2 64 42 COc1ccc([C@@H](CCO)NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880917708 FG On-Demand Anodyne UTS2 64 42 COCCC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917714 FE On-Demand Anodyne EPHX2 57 52 COCCC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917714 FE On-Demand Anodyne CCR8 42 37 CCN(Cc1ccccc1)C(=O)Nc1cncc(C(F)F)c1 ZINC000880917730 DI On-Demand Anodyne ROCK2 15 42 CCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917731 CF On-Demand Anodyne ASAH1 51 31 O=C(NCCn1ccnc1)Nc1cncc(C(F)F)c1 ZINC000880917734 CE On-Demand Anodyne QPCT 34 49 O=C(Nc1cncc(C(F)F)c1)N1CCC(c2nc3ccccc3s2)CC1 ZINC000880917735 GK On-Demand Anodyne SMO 32 41 COCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917742 CE On-Demand Anodyne EPHX2 15 40 CN1CCN(C(C)(C)CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917746 FE On-Demand Anodyne EPHX2 15 44 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cncc(C(F)F)c1 ZINC000880917758 EG On-Demand Anodyne BMP1 48 35 CCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917766 CF On-Demand Anodyne EPHX2 44 43 CCN1CCC(NC(=O)Nc2cncc(C(F)F)c2)CC1 ZINC000880917766 CF On-Demand Anodyne CXCR3 21 49 CC(=O)c1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880917770 GH On-Demand Anodyne NPY2R 104 39 CC(=O)c1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880917770 GH On-Demand Anodyne PRNP 15 41 CC(=O)c1ccc(N2CCN(C(=O)Nc3cncc(C(F)F)c3)CC2)c(F)c1 ZINC000880917770 GH On-Demand Anodyne SLC6A9 18 44 CCOCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917776 CE On-Demand Anodyne EPHX2 15 41 CC(C)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917781 EG On-Demand Anodyne CCR3 42 39 CC(C)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917781 EG On-Demand Anodyne EPHX2 53 45 CC(C)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917781 EG On-Demand Anodyne CXCR3 24 46 COc1cccc([C@H](CNC(=O)Nc2cncc(C(F)F)c2)N(C)C)c1 ZINC000880917782 FG On-Demand Anodyne ROCK1 31 41 COc1cccc([C@H](CNC(=O)Nc2cncc(C(F)F)c2)N(C)C)c1 ZINC000880917782 FG On-Demand Anodyne MTNR1B 26 40 COc1cccc([C@H](CNC(=O)Nc2cncc(C(F)F)c2)N(C)C)c1 ZINC000880917782 FG On-Demand Anodyne ROCK2 39 41 O=C(NCc1ccccc1CN1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880917784 FH On-Demand Anodyne F2R 51 32 O=C(NCc1ccccc1CN1CCCC1)Nc1cncc(C(F)F)c1 ZINC000880917784 FH On-Demand Anodyne NAMPT 37 41 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917811 EE On-Demand Anodyne NPY5R 33 41 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917813 EE On-Demand Anodyne NPY5R 33 41 C[C@H](CN1CCOCC1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917827 DD On-Demand Anodyne EPHX2 29 47 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917842 FE On-Demand Anodyne ROCK1 18 42 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917842 FE On-Demand Anodyne ROCK2 37 46 CNC(=O)COc1cccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917842 FE On-Demand Anodyne PDS 41 33 C[C@H]1c2ccccc2CN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917843 DI On-Demand Anodyne TRPM8 29 44 CN(C)c1ccc(NC(=O)Nc2ccc(N3CCC(O)CC3)c(C#N)c2)cc1F ZINC000880917845 GG On-Demand Mild NPY2R 85 39 CS[C@@H]1CC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917870 DG On-Demand Anodyne EPHX2 40 39 CS[C@H]1CC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880917872 DG On-Demand Anodyne EPHX2 40 39 CN(C)c1ccc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)cc1F ZINC000880917884 GE On-Demand Anodyne HTR2A 34 45 CN(C)c1ccc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)cc1F ZINC000880917884 GE On-Demand Anodyne CHRNA7 17 42 CN(C)c1ccc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)cc1F ZINC000880917884 GE On-Demand Anodyne MTOR 61 37 CN(C)c1ccc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)cc1F ZINC000880917884 GE On-Demand Anodyne EPHX2 31 52 CN(C)c1ccc(NC(=O)Nc2cnn(CCN3CCOCC3)c2)cc1F ZINC000880917884 GE On-Demand Anodyne STAT6 40 33 COc1ccc([C@@H](O)CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880917897 EF On-Demand Anodyne F7 16 40 COCCN(Cc1cccnc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917902 EF On-Demand Anodyne ROCK2 33 41 Cc1noc(C)c1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917912 DF On-Demand Anodyne P2RX7 15 46 CCCN(CC)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917921 CG On-Demand Anodyne NPY2R 43 36 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917935 FF On-Demand Anodyne CACNA1H 44 39 CCOC(=O)N(C)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917935 FF On-Demand Anodyne NPY2R 44 33 CN(C)c1ccc(NC(=O)N[C@H]2CCCC[C@H]2O)cc1F ZINC000880917937 CE On-Demand Anodyne EPHX2 25 40 CN(C)c1ccc(NC(=O)N[C@H]2CCCC[C@@H]2O)cc1F ZINC000880917939 CE On-Demand Anodyne EPHX2 25 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC[C@@H]2O)cc1F ZINC000880917941 CE On-Demand Anodyne EPHX2 25 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC[C@H]2O)cc1F ZINC000880917943 CE On-Demand Anodyne EPHX2 25 40 CCCCCNC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917945 GG On-Demand Anodyne ASAH1 58 36 C[C@@H]1C[C@@H]1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917947 CF On-Demand Anodyne PRMT3 43 31 C[C@H]1C[C@H]1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917949 CF On-Demand Anodyne PRMT3 43 31 C[C@@H]1C[C@H]1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917953 CF On-Demand Anodyne PRMT3 43 31 CCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917958 DF On-Demand Anodyne CACNA1H 61 44 CCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880917958 DF On-Demand Anodyne S1PR2 32 45 COCc1cc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)ccc1F ZINC000880917969 EG On-Demand Anodyne ROCK2 18 41 CN(C)C(=O)Nc1cccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880917970 FG On-Demand Anodyne ROCK2 25 45 COCCOc1ncccc1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917973 FF On-Demand Anodyne SCN10A 19 40 C[C@@H](CCN(C)C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880917981 CE On-Demand Anodyne UTS2 64 35 C[C@@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918026 GE On-Demand Anodyne CACNA1H 22 40 C[C@@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918026 GE On-Demand Anodyne NPY2R 41 34 C[C@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918027 GE On-Demand Anodyne CACNA1H 22 40 C[C@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918027 GE On-Demand Anodyne NPY2R 41 34 CN(C)c1ccc(NC(=O)N[C@H](c2cccnc2)C2CC2)cc1F ZINC000880918030 EH On-Demand Anodyne NPY2R 48 41 CN(C)c1ccc(NC(=O)N[C@H](c2cccnc2)C2CC2)cc1F ZINC000880918030 EH On-Demand Anodyne NAMPT 17 40 CN(C)c1ccc(NC(=O)N[C@@H](c2cccnc2)C2CC2)cc1F ZINC000880918031 EH On-Demand Anodyne NPY2R 48 41 CN(C)c1ccc(NC(=O)N[C@@H](c2cccnc2)C2CC2)cc1F ZINC000880918031 EH On-Demand Anodyne NAMPT 17 40 CN(C)c1ccc(NC(=O)N[C@H]2CCOC3(CCCC3)C2)cc1F ZINC000880918047 EH On-Demand Anodyne ENV 41 37 CN(C)c1ccc(NC(=O)N[C@@H]2CCOC3(CCCC3)C2)cc1F ZINC000880918048 EH On-Demand Anodyne ENV 41 37 CN(C)c1ccc(NC(=O)Nc2cnn(CC(=O)NC3CC3)c2)cc1F ZINC000880918090 FE On-Demand Anodyne PANC 42 34 Cc1nccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)n1 ZINC000880918095 DE On-Demand Anodyne KIT 17 42 Cc1nccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)n1 ZINC000880918095 DE On-Demand Anodyne BRAF 15 42 COc1ccc(O)c([C@@H](C)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918101 EG On-Demand Clean THRB 28 41 COc1ccc(O)c([C@H](C)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918102 EG On-Demand Clean THRB 28 41 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)C2 ZINC000880918103 FG On-Demand Anodyne P2RY14 45 33 COc1ccnc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880918106 FE On-Demand Anodyne PDGFRB 52 39 COc1ccnc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880918106 FE On-Demand Anodyne FAAH 22 41 COc1ccnc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880918106 FE On-Demand Anodyne MET 18 41 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc1F ZINC000880918113 DE On-Demand Anodyne CCR3 77 45 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc1F ZINC000880918113 DE On-Demand Anodyne EPHX2 45 40 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC3CC3)C2)cc1F ZINC000880918113 DE On-Demand Anodyne CXCR3 19 45 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)cc1F ZINC000880918115 DE On-Demand Anodyne CCR3 77 45 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)cc1F ZINC000880918115 DE On-Demand Anodyne EPHX2 45 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(CC3CC3)C2)cc1F ZINC000880918115 DE On-Demand Anodyne CXCR3 19 45 CN1CCC(N(C)CCN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918120 FE On-Demand Anodyne HTR1F 45 35 CN1CCC(N(C)CCN(C)C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918120 FE On-Demand Anodyne MCHR1 32 40 COCCCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918126 CF On-Demand Anodyne CCR3 15 41 COC(=O)N1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918128 EE On-Demand Anodyne EPHX2 61 49 C[C@@H]1CCCN(C(=O)C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)C1 ZINC000880918135 GG On-Demand Anodyne EPHX2 19 50 CSCC[C@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918141 CG On-Demand Anodyne FPR1 30 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000880918145 FD On-Demand Anodyne EPHX2 49 42 CSCC[C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918146 CG On-Demand Anodyne FPR1 30 40 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000880918147 FD On-Demand Anodyne EPHX2 49 42 CN(C)c1ccc(NC(=O)Nc2cnn(C(C)(C)C)c2)cc1F ZINC000880918154 DG On-Demand Anodyne HTR2A 30 40 C=CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918160 DF On-Demand Mild EPHX2 48 42 C=CCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918160 DF On-Demand Mild CXCR3 22 43 CN1CCC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918164 DE On-Demand Anodyne CCR3 90 43 CN1CCC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918164 DE On-Demand Anodyne EPHX2 15 42 CN1CCC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918164 DE On-Demand Anodyne CACNA1I 52 32 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918177 GE On-Demand Anodyne NPY2R 50 35 C[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918187 CF On-Demand Anodyne CACNA1H 27 40 C[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918187 CF On-Demand Anodyne EPHX2 29 47 C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918189 CF On-Demand Anodyne CACNA1H 27 40 C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918189 CF On-Demand Anodyne EPHX2 29 47 CCN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918194 DE On-Demand Anodyne HTR4 44 33 CCN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918194 DE On-Demand Anodyne NPY2R 51 35 CCN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918194 DE On-Demand Anodyne CCR3 83 40 CCN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918194 DE On-Demand Anodyne CACNA1I 70 35 CCc1cnc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)s1 ZINC000880918195 DG On-Demand Anodyne NPY2R 41 32 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(c3ncccn3)C2)cc1F ZINC000880918220 FE On-Demand Anodyne NPY2R 49 35 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(c3ncccn3)C2)cc1F ZINC000880918220 FE On-Demand Anodyne EPHX2 41 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(c3ncccn3)C2)cc1F ZINC000880918223 FE On-Demand Anodyne NPY2R 49 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(c3ncccn3)C2)cc1F ZINC000880918223 FE On-Demand Anodyne EPHX2 41 40 CN1CCN(C)[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918257 DD On-Demand Anodyne CCR3 40 39 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918258 DD On-Demand Anodyne CCR3 40 39 CN(C)c1ccc(NC(=O)N[C@H]2CCN(c3ccccc3C(N)=O)C2)cc1F ZINC000880918268 GE On-Demand Anodyne NPY2R 68 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(c3ccccc3C(N)=O)C2)cc1F ZINC000880918270 GE On-Demand Anodyne NPY2R 68 36 CNC(=O)CC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918281 EE On-Demand Anodyne EPHX2 18 40 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918366 DE On-Demand Anodyne HTR1F 50 36 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918366 DE On-Demand Anodyne NPY2R 45 33 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918366 DE On-Demand Anodyne CCR3 70 42 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918366 DE On-Demand Anodyne EPHX2 36 42 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918366 DE On-Demand Anodyne CACNA1I 68 37 CN(C)c1ccc(NC(=O)N[C@@H](Cn2ccnc2)C(C)(C)C)cc1F ZINC000880918379 EG On-Demand Anodyne QPCT 24 40 CN(C)c1ccc(NC(=O)N[C@H](Cn2ccnc2)C(C)(C)C)cc1F ZINC000880918380 EG On-Demand Anodyne QPCT 24 40 CN(C)c1ccc(NC(=O)Nc2ccc(N3CCCS3(=O)=O)cc2)cc1F ZINC000880918389 GG On-Demand Anodyne CDK1 16 41 CN1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918404 CE On-Demand Anodyne CCR3 57 39 CN1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918404 CE On-Demand Anodyne EPHX2 50 44 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918407 EE On-Demand Anodyne CACNA1H 40 42 COC(=O)[C@@]1(F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918407 EE On-Demand Anodyne EPHX2 34 43 COc1cccc([C@H](CO)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918409 EF On-Demand Anodyne NPY2R 28 42 COc1cccc([C@H](CO)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918409 EF On-Demand Anodyne ROCK1 17 49 COc1cccc([C@H](CO)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918409 EF On-Demand Anodyne MTNR1A 19 40 COc1cccc([C@H](CO)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918409 EF On-Demand Anodyne MTNR1B 25 40 COc1cccc([C@H](CO)NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918409 EF On-Demand Anodyne TAAR1 21 40 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne DRD4 15 41 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne HTR2A 27 40 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne HTR4 43 37 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne CCR3 59 42 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne EPHX2 59 48 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne CXCR3 22 43 COCCN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918416 EE On-Demand Anodyne MCHR1 44 42 COCCCCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918424 CE On-Demand Anodyne CCR3 17 40 COC(=O)C1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918434 EF On-Demand Anodyne EPHX2 56 44 C[C@@H]([C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1)N1CCOCC1 ZINC000880918445 EE On-Demand Anodyne NPY2R 41 33 C[C@@H]([C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1)N1CCOCC1 ZINC000880918445 EE On-Demand Anodyne EPHX2 20 47 C=C(C)CN(CC)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918459 CG On-Demand Mild NPY2R 41 35 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(N(C)C)c(F)c3)C2)nn1 ZINC000880918460 FF On-Demand Anodyne CCR3 50 34 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(N(C)C)c(F)c3)C2)nn1 ZINC000880918460 FF On-Demand Anodyne EPHX2 29 40 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918483 FG On-Demand Anodyne HRH2 28 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918483 FG On-Demand Anodyne MTNR1A 27 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918483 FG On-Demand Anodyne MTNR1B 25 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918483 FG On-Demand Anodyne EPHX2 24 45 C[C@H](O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918507 DD On-Demand Anodyne CACNA1H 36 41 COCCOc1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cn1 ZINC000880918509 FF On-Demand Anodyne ROCK2 18 41 CN(C)c1ccc(NC(=O)N[C@H](CO)Cc2ccccc2)cc1F ZINC000880918511 EF On-Demand Anodyne MME 45 38 CN(C)c1ccc(NC(=O)N[C@H](CO)Cc2ccccc2)cc1F ZINC000880918511 EF On-Demand Anodyne ANPEP 53 31 CN(C)c1ccc(NC(=O)N[C@@H](CO)Cc2ccccc2)cc1F ZINC000880918513 EF On-Demand Anodyne MME 45 38 CN(C)c1ccc(NC(=O)N[C@@H](CO)Cc2ccccc2)cc1F ZINC000880918513 EF On-Demand Anodyne ANPEP 53 31 COC(=O)N1CCC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918538 EE On-Demand Anodyne EPHX2 50 41 COC(=O)N1CCC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918540 EE On-Demand Anodyne EPHX2 50 41 C=C(C)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918549 EG On-Demand Mild EPHX2 49 43 C=C(C)CN1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918549 EG On-Demand Mild CXCR3 22 43 C[C@@H](O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918550 DF On-Demand Anodyne CACNA1H 38 45 C[C@@H](O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918550 DF On-Demand Anodyne NPY2R 70 38 C[C@@H](O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918550 DF On-Demand Anodyne EPHX2 22 40 CN(C)c1ccc(NC(=O)Nc2cnn(C[C@@H]3CCCO3)c2)cc1F ZINC000880918551 EF On-Demand Anodyne PANC 54 37 CN(C)c1ccc(NC(=O)N[C@H](CCO)c2ccccc2)cc1F ZINC000880918553 EG On-Demand Anodyne NPY2R 58 35 CN(C)c1ccc(NC(=O)N[C@H](CCO)c2ccccc2)cc1F ZINC000880918553 EG On-Demand Anodyne UTS2 63 38 C=CCNC(=O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918602 CD On-Demand Mild F7 24 40 CCOC(=O)N1CC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918616 EE On-Demand Anodyne EPHX2 54 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880918617 EE On-Demand Anodyne EPHX2 54 45 CN(C)c1ccc(NC(=O)Nc2cnn(C[C@H]3CCCO3)c2)cc1F ZINC000880918647 EF On-Demand Anodyne PANC 54 37 COC[C@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccc1 ZINC000880918655 EG On-Demand Anodyne NPY2R 59 35 COC[C@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccc1 ZINC000880918655 EG On-Demand Anodyne TACR3 18 45 COC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccc1 ZINC000880918656 EG On-Demand Anodyne NPY2R 59 35 COC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccc1 ZINC000880918656 EG On-Demand Anodyne TACR3 18 45 CC(=O)NCC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918663 EE On-Demand Anodyne EPHX2 31 43 CC(=O)NCC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918663 EE On-Demand Anodyne CACNA1I 57 32 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918669 GE On-Demand Anodyne TRPV1 23 44 CN1CCN(c2ncccc2CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918669 GE On-Demand Anodyne NPY2R 60 38 CC[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918686 DE On-Demand Anodyne NPY2R 40 36 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918687 DE On-Demand Anodyne NPY2R 40 36 CCN(CC)C(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918702 FG On-Demand Anodyne NPY2R 64 40 COc1ccnc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880918705 FF On-Demand Anodyne PDGFRB 56 44 COc1ccnc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)c1 ZINC000880918705 FF On-Demand Anodyne MET 26 43 C=CC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918812 CG On-Demand Mild CACNA1H 28 40 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccncc1 ZINC000880918821 DH On-Demand Anodyne NPY2R 40 34 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918837 FH On-Demand Anodyne KCNK3 69 37 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880918837 FH On-Demand Anodyne KCNK9 59 37 CN(C)c1ccc(NC(=O)N[C@](C)(CO)c2ccccc2)cc1F ZINC000880918843 EF On-Demand Anodyne IMDH_CRYPV 61 39 CN(C)c1ccc(NC(=O)N[C@@](C)(CO)c2ccccc2)cc1F ZINC000880918844 EF On-Demand Anodyne IMDH_CRYPV 61 39 CN(C)C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880918893 DD On-Demand Anodyne EPHX2 20 40 CCc1nnc2n1CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)C2 ZINC000880918901 EE On-Demand Anodyne P2RX7 17 45 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918915 FD On-Demand Anodyne NPY2R 51 35 C[C@H]1C[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)CCN1C ZINC000880918934 DE On-Demand Anodyne EPHX2 47 39 CCc1noc([C@@H](C)N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880918940 GF On-Demand Anodyne NPY2R 61 49 CCc1noc([C@H](C)N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880918941 GF On-Demand Anodyne NPY2R 61 49 CN(C)c1ccc(NC(=O)N[C@@H]2CC=CCC2)cc1F ZINC000880918957 CG On-Demand Anodyne EPHX2 42 39 CN(C)c1ccc(NC(=O)N[C@H]2CC=CCC2)cc1F ZINC000880918958 CG On-Demand Anodyne EPHX2 42 39 CCN(CC)C(=O)CN1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880918972 GD On-Demand Anodyne NPY2R 50 37 Cc1ccccc1[C@H](CO)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918996 EG On-Demand Anodyne CTSA 60 36 Cc1ccccc1[C@@H](CO)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880918997 EG On-Demand Anodyne CTSA 60 36 COC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919001 DE On-Demand Anodyne CACNA1H 27 40 COC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919001 DE On-Demand Anodyne EPHX2 23 41 C[C@H](O)CN(Cc1ccccc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919008 EG On-Demand Anodyne NPY5R 33 40 CN(CC(=O)N1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919043 ED On-Demand Anodyne EPHX2 20 47 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919046 DF On-Demand Anodyne NPY2R 45 34 CCN1CCC[C@H]1CN(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919046 DF On-Demand Anodyne MCHR1 18 42 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919047 DF On-Demand Anodyne NPY2R 45 34 CCN1CCC[C@@H]1CN(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919047 DF On-Demand Anodyne MCHR1 18 42 CC(=O)N1CCc2cc(NC(=O)Nc3ccc(N(C)C)c(F)c3)ccc21 ZINC000880919048 FG On-Demand Anodyne NPY2R 42 33 CC(=O)N1CCc2cc(NC(=O)Nc3ccc(N(C)C)c(F)c3)ccc21 ZINC000880919048 FG On-Demand Anodyne HSD17B3 47 33 CCOC[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880919050 DG On-Demand Anodyne CCR3 21 45 CCOC[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880919050 DG On-Demand Anodyne EPHX2 15 45 CN(C)C(=O)C1(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CCCC1 ZINC000880919085 FF On-Demand Anodyne PRMT3 42 29 COc1ccc(CN(CCO)C(=O)Nc2ccc(N(C)C)c(F)c2)c(OC)c1 ZINC000880919107 GF On-Demand Anodyne ROCK2 15 42 CN(C)c1ccc(NC(=O)N[C@@H](CS(C)(=O)=O)c2ccccc2)cc1F ZINC000880919123 GF On-Demand Anodyne NPY2R 55 34 CN(C)c1ccc(NC(=O)N[C@H](CS(C)(=O)=O)c2ccccc2)cc1F ZINC000880919124 GF On-Demand Anodyne NPY2R 55 34 CCC1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919141 DF On-Demand Anodyne CACNA1H 60 43 CCC1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919141 DF On-Demand Anodyne NPY2R 47 33 C#CC(C)(C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919144 CE On-Demand Mild IMDH_CRYPV 51 34 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1nnc2n1CCCCC2 ZINC000880919166 FG On-Demand Anodyne NPY2R 45 34 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)c1nnc2n1CCCCC2 ZINC000880919166 FG On-Demand Anodyne CCR3 49 31 C[C@H](C[C@@H](O)c1ccccc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919176 EH On-Demand Anodyne NPY2R 58 35 C[C@H](C[C@@H](O)c1ccccc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919176 EH On-Demand Anodyne F7 15 41 C[C@@H](C[C@H](O)c1ccccc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919178 EH On-Demand Anodyne NPY2R 58 35 C[C@@H](C[C@H](O)c1ccccc1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919178 EH On-Demand Anodyne F7 15 41 CN(C)c1ccc(NC(=O)Nc2cnn(C)c2C(F)F)cc1F ZINC000880919179 EG On-Demand Anodyne HTR2A 39 41 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@@H](CO)CC2)cc1F ZINC000880919187 DF On-Demand Anodyne EPHX2 49 42 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@H](CO)CC2)cc1F ZINC000880919188 DF On-Demand Anodyne EPHX2 49 42 COC(=O)C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880919190 ED On-Demand Anodyne EPHX2 20 41 COC(=O)C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880919191 ED On-Demand Anodyne EPHX2 20 41 CC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@H](C)C1 ZINC000880919193 DD On-Demand Anodyne LIMK1 17 40 CC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@H](C)C1 ZINC000880919193 DD On-Demand Anodyne LIMK2 26 40 CC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@@H](C)C1 ZINC000880919194 DD On-Demand Anodyne LIMK1 17 40 CC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@@H](C)C1 ZINC000880919194 DD On-Demand Anodyne LIMK2 26 40 CN1C(=O)N[C@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1=O ZINC000880919208 ED On-Demand Anodyne CACNA1H 42 42 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1=O ZINC000880919209 ED On-Demand Anodyne CACNA1H 42 42 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919218 FD On-Demand Anodyne EPHX2 23 43 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919220 FD On-Demand Anodyne EPHX2 23 43 C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@@H]1C ZINC000880919290 CG On-Demand Anodyne TRPC6 46 32 C[C@H]1[C@H](C)CCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919291 CG On-Demand Anodyne TRPC6 46 32 C[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@H]1C ZINC000880919292 CG On-Demand Anodyne TRPC6 46 32 C[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)[C@@H]1C ZINC000880919293 CG On-Demand Anodyne TRPC6 46 32 CCN1CC[C@@H](N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@@H]1C ZINC000880919297 EG On-Demand Anodyne NPY2R 42 34 CCN1CC[C@H](N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@H]1C ZINC000880919298 EG On-Demand Anodyne NPY2R 42 34 CCN1CC[C@@H](N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@H]1C ZINC000880919299 EG On-Demand Anodyne NPY2R 42 34 CCN1CC[C@H](N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@@H]1C ZINC000880919300 EG On-Demand Anodyne NPY2R 42 34 CN(C)c1ccc(NC(=O)N[C@H]2CCC(F)(F)C2)cc1F ZINC000880919302 DG On-Demand Anodyne EPHX2 43 38 CN(C)c1ccc(NC(=O)N[C@H]2CCC(F)(F)C2)cc1F ZINC000880919302 DG On-Demand Anodyne ENV 43 38 CN(C)c1ccc(NC(=O)N[C@@H]2CCC(F)(F)C2)cc1F ZINC000880919303 DG On-Demand Anodyne EPHX2 43 38 CN(C)c1ccc(NC(=O)N[C@@H]2CCC(F)(F)C2)cc1F ZINC000880919303 DG On-Demand Anodyne ENV 43 38 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C(=O)N1CCOCC1 ZINC000880919367 FD On-Demand Anodyne NPY2R 55 34 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C(=O)N1CCOCC1 ZINC000880919367 FD On-Demand Anodyne EPHX2 27 49 COCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919375 ED On-Demand Anodyne CACNA1H 73 43 COCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919375 ED On-Demand Anodyne S1PR2 31 44 COc1ccc([C@@H](CO)N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919377 FG On-Demand Anodyne NPY5R 33 40 COc1ccc([C@H](CO)N(C)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919378 FG On-Demand Anodyne NPY5R 33 40 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C3CCOCC3)C2=O)cc1F ZINC000880919383 FD On-Demand Anodyne MTOR 40 36 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C3CCOCC3)C2=O)cc1F ZINC000880919383 FD On-Demand Anodyne EPHX2 24 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C3CCOCC3)C2=O)cc1F ZINC000880919384 FD On-Demand Anodyne MTOR 40 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C3CCOCC3)C2=O)cc1F ZINC000880919384 FD On-Demand Anodyne EPHX2 24 41 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919385 FF On-Demand Anodyne NPY2R 43 36 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919385 FF On-Demand Anodyne CCR3 54 42 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919385 FF On-Demand Anodyne EPHX2 32 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919386 FF On-Demand Anodyne NPY2R 43 36 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919386 FF On-Demand Anodyne CCR3 54 42 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919386 FF On-Demand Anodyne EPHX2 32 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919387 FF On-Demand Anodyne NPY2R 43 36 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919387 FF On-Demand Anodyne CCR3 54 42 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919387 FF On-Demand Anodyne EPHX2 32 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919388 FF On-Demand Anodyne NPY2R 43 36 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919388 FF On-Demand Anodyne CCR3 54 42 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919388 FF On-Demand Anodyne EPHX2 32 42 CC(=O)OC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919390 DE On-Demand Anodyne EPHX2 30 41 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919396 GG On-Demand Anodyne CCR3 32 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919396 GG On-Demand Anodyne EPHX2 27 44 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919397 GG On-Demand Anodyne CCR3 32 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919397 GG On-Demand Anodyne EPHX2 27 44 Cc1c(NC(=O)Nc2ccc(N(C)C)c(F)c2)cnn1C ZINC000880919408 CF On-Demand Anodyne HTR2A 40 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919411 GG On-Demand Anodyne CCR3 35 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919411 GG On-Demand Anodyne EPHX2 30 44 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919412 GG On-Demand Anodyne CCR3 35 40 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919412 GG On-Demand Anodyne EPHX2 30 44 CN(C)c1ccc(NC(=O)N[C@H](C[S@](C)=O)c2ccccc2)cc1F ZINC000880919427 FG On-Demand Anodyne NPY2R 77 38 CN(C)c1ccc(NC(=O)N[C@@H](C[S@@](C)=O)c2ccccc2)cc1F ZINC000880919428 FG On-Demand Anodyne NPY2R 77 38 CN(C)c1ccc(NC(=O)N[C@@H](C[S@](C)=O)c2ccccc2)cc1F ZINC000880919429 FG On-Demand Anodyne NPY2R 77 38 CN(C)c1ccc(NC(=O)N[C@H](C[S@@](C)=O)c2ccccc2)cc1F ZINC000880919430 FG On-Demand Anodyne NPY2R 77 38 CN(C)c1ccc(NC(=O)N[C@@H]2CCCSC2)cc1F ZINC000880919445 CF On-Demand Anodyne EPHX2 40 42 CN(C)c1ccc(NC(=O)N[C@H]2CCCSC2)cc1F ZINC000880919446 CF On-Demand Anodyne EPHX2 40 42 CCc1nc([C@H]2CCCN2C(=O)Nc2ccc(N(C)C)c(F)c2)no1 ZINC000880919471 EG On-Demand Anodyne NPY2R 51 36 CCNS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919478 GF On-Demand Anodyne CA1 15 41 CCNS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919478 GF On-Demand Anodyne CA9 18 42 CCNS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919478 GF On-Demand Anodyne PRMT3 19 42 CCNS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880919478 GF On-Demand Anodyne NAMPT 51 43 Cc1cncc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880919480 DF On-Demand Anodyne ROCK2 18 41 Cc1cncc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)c1 ZINC000880919480 DF On-Demand Anodyne NAMPT 42 56 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919503 EH On-Demand Anodyne NPY5R 36 53 CN(C)c1ccc(NC(=O)N[C@H]2CCOC3(CCCCC3)C2)cc1F ZINC000880919636 EH On-Demand Anodyne ENV 41 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCOC3(CCCCC3)C2)cc1F ZINC000880919637 EH On-Demand Anodyne ENV 41 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCOC3(CCC3)C2)cc1F ZINC000880919638 DG On-Demand Anodyne ENV 42 39 CN(C)c1ccc(NC(=O)N[C@H]2CCOC3(CCC3)C2)cc1F ZINC000880919639 DG On-Demand Anodyne ENV 42 39 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@@H](O)CC2)cc1F ZINC000880919647 CE On-Demand Anodyne EPHX2 56 45 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@@H](O)CC2)cc1F ZINC000880919647 CE On-Demand Anodyne ENV 40 34 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880919667 FE On-Demand Anodyne P2RY14 50 36 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919678 GE On-Demand Anodyne CCR3 25 40 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919678 GE On-Demand Anodyne EPHX2 26 41 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919679 GE On-Demand Anodyne CCR3 25 40 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919679 GE On-Demand Anodyne EPHX2 26 41 CN(C)CC1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919694 EG On-Demand Anodyne EPHX2 53 42 CN(C)c1ccc(NC(=O)N[C@H]2CCN(c3ccccn3)C2)cc1F ZINC000880919699 EF On-Demand Anodyne NPY2R 47 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(c3ccccn3)C2)cc1F ZINC000880919700 EF On-Demand Anodyne NPY2R 47 35 Cc1nsc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n1 ZINC000880919710 FE On-Demand Anodyne FAAH 17 50 CN(C[C@H](O)CN1CCOCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919713 FD On-Demand Anodyne EPHX2 18 41 CN(C)c1ccc(NC(=O)N[C@@H](CO)C[C@@H](O)c2ccccc2)cc1F ZINC000880919717 FE On-Demand Anodyne NPY2R 56 34 CN(C)c1ccc(NC(=O)N[C@H](CO)C[C@@H](O)c2ccccc2)cc1F ZINC000880919718 FE On-Demand Anodyne NPY2R 56 34 CN(C)c1ccc(NC(=O)N[C@@H](CO)C[C@H](O)c2ccccc2)cc1F ZINC000880919719 FE On-Demand Anodyne NPY2R 56 34 CN(C)c1ccc(NC(=O)N[C@H](CO)C[C@H](O)c2ccccc2)cc1F ZINC000880919720 FE On-Demand Anodyne NPY2R 56 34 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC[C@@H]2CO)cc1F ZINC000880919731 DF On-Demand Anodyne CCR3 35 45 CN(C)c1ccc(NC(=O)N[C@H]2CCCC[C@H]2CO)cc1F ZINC000880919732 DF On-Demand Anodyne CCR3 35 45 CN(C)c1ccc(NC(=O)N[C@H]2CCCC[C@@H]2CO)cc1F ZINC000880919733 DF On-Demand Anodyne CCR3 35 45 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC[C@H]2CO)cc1F ZINC000880919734 DF On-Demand Anodyne CCR3 35 45 C[C@@H](O)C(C)(C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919761 CE On-Demand Anodyne IMDH_CRYPV 58 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC(F)(F)C2)cc1F ZINC000880919767 DH On-Demand Anodyne EPHX2 39 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC(F)(F)C2)cc1F ZINC000880919767 DH On-Demand Anodyne ENV 43 39 CN(C)c1ccc(NC(=O)N[C@H]2CCCC(F)(F)C2)cc1F ZINC000880919768 DH On-Demand Anodyne EPHX2 39 41 CN(C)c1ccc(NC(=O)N[C@H]2CCCC(F)(F)C2)cc1F ZINC000880919768 DH On-Demand Anodyne ENV 43 39 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880919784 DE On-Demand Anodyne CACNA1H 36 42 COC(=O)[C@@]1(C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880919784 DE On-Demand Anodyne EPHX2 34 43 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)C3CCCC3)C2)cc1F ZINC000880919791 FF On-Demand Anodyne EPHX2 52 48 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)C3CCCC3)C2)cc1F ZINC000880919792 FF On-Demand Anodyne EPHX2 52 48 CCN(Cc1ccccn1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919828 DG On-Demand Anodyne NPY2R 49 36 CN(C)c1ccc(NC(=O)N[C@@H](CCC#N)c2ccccc2)cc1F ZINC000880919838 EI On-Demand Mild NPY2R 59 34 CN(C)c1ccc(NC(=O)N[C@@H](CCC#N)c2ccccc2)cc1F ZINC000880919838 EI On-Demand Mild UTS2 54 36 CN(C)c1ccc(NC(=O)N[C@H](CCC#N)c2ccccc2)cc1F ZINC000880919839 EI On-Demand Mild NPY2R 59 34 CN(C)c1ccc(NC(=O)N[C@H](CCC#N)c2ccccc2)cc1F ZINC000880919839 EI On-Demand Mild UTS2 54 36 CN1CCC(C)(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919882 DF On-Demand Anodyne EPHX2 16 41 CN1CCC(C)(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919882 DF On-Demand Anodyne MCHR1 15 45 C[C@H](NC(=O)OC(C)(C)C)[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880919904 GH On-Demand Anodyne NPY2R 42 34 COC(=O)C1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919951 ED On-Demand Anodyne CACNA1H 63 43 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(Cc3ccccn3)C2=O)cc1F ZINC000880919979 GF On-Demand Anodyne CCKBR 51 36 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(Cc3ccccn3)C2=O)cc1F ZINC000880919980 GF On-Demand Anodyne CCKBR 51 36 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919986 EG On-Demand Anodyne HTR1F 46 37 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880919986 EG On-Demand Anodyne NPY2R 49 36 CN(C)C(=O)CC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880919998 FF On-Demand Anodyne EPHX2 20 41 CN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920002 CD On-Demand Anodyne CCR3 72 41 CN1CC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920002 CD On-Demand Anodyne CACNA1I 67 34 CN1CC[C@@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920003 CD On-Demand Anodyne CCR3 72 41 CN1CC[C@@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920003 CD On-Demand Anodyne CACNA1I 67 34 CN(C)CCCC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920035 FG On-Demand Anodyne EPHX2 25 43 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920090 EI On-Demand Anodyne TRPC6 43 29 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920092 EI On-Demand Anodyne TRPC6 43 29 CN1CCC(N2CCC(NC(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880920094 GF On-Demand Anodyne HTR1F 46 38 CN1CCC(N2CCC(NC(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880920094 GF On-Demand Anodyne SLC6A5 21 43 CN1CCC(N2CCC(NC(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880920094 GF On-Demand Anodyne EPHX2 47 41 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920138 DE On-Demand Anodyne NPY2R 46 36 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920138 DE On-Demand Anodyne EPHX2 25 40 CN(C)C[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920138 DE On-Demand Anodyne NR1D1 15 40 CN1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920185 CE On-Demand Anodyne EPHX2 17 46 COC1(C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920193 DF On-Demand Anodyne CACNA1H 59 44 CCC1(CC)CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[S@@]1=O ZINC000880920195 FG On-Demand Anodyne NPY2R 55 35 CCC1(CC)CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[S@]1=O ZINC000880920196 FG On-Demand Anodyne NPY2R 55 35 CN(C)c1ccc(NC(=O)N[C@H](CO)Cc2ccc(F)cc2)cc1F ZINC000880920204 EF On-Demand Anodyne CCR3 40 35 CN(C)c1ccc(NC(=O)N[C@@H](CO)Cc2ccc(F)cc2)cc1F ZINC000880920205 EF On-Demand Anodyne CCR3 40 35 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880920278 FF On-Demand Anodyne CACNA1H 51 40 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880920279 FF On-Demand Anodyne CACNA1H 51 40 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880920280 FF On-Demand Anodyne CACNA1H 51 40 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880920281 FF On-Demand Anodyne CACNA1H 51 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCC3(C2)OCCO3)cc1F ZINC000880920306 EF On-Demand Anodyne ENV 41 39 CN(C)c1ccc(NC(=O)N[C@H]2CCCC3(C2)OCCO3)cc1F ZINC000880920307 EF On-Demand Anodyne ENV 41 39 COC[C@@H](O)CCNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920358 CD On-Demand Anodyne ADRB1 42 34 CCc1noc(C)c1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920363 DG On-Demand Anodyne NPY2R 17 42 C[C@H](CO)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920372 CD On-Demand Anodyne NPY5R 35 42 C[C@@H](CO)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920373 CD On-Demand Anodyne NPY5R 35 42 COc1cc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)ncn1 ZINC000880920387 FE On-Demand Anodyne PDGFRB 64 45 COc1cc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)ncn1 ZINC000880920387 FE On-Demand Anodyne LIMK2 21 42 Cc1nc(CN2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)n[nH]1 ZINC000880920388 FD On-Demand Anodyne FAAH 15 41 CO[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920408 DF On-Demand Anodyne EPHX2 23 40 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920426 GH On-Demand Anodyne NPY2R 58 38 CCN(CC)C(=O)CCC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920426 GH On-Demand Anodyne EPHX2 18 41 CCOc1ccccc1OCC(=O)NNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920427 GF On-Demand Reactive KCNK3 38 40 CCOc1ccccc1OCC(=O)NNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920427 GF On-Demand Reactive KCNK9 33 40 CC(=O)N1CCc2c(NC(=O)Nc3ccc(N(C)C)c(F)c3)cccc21 ZINC000880920432 FG On-Demand Anodyne NPY2R 43 35 CC(=O)N1CCc2c(NC(=O)Nc3ccc(N(C)C)c(F)c3)cccc21 ZINC000880920432 FG On-Demand Anodyne P2RY1 48 33 Cc1cc(NC(=O)Nc2ccc(N(C)C)c(F)c2)nn1C ZINC000880920434 CF On-Demand Anodyne FPR2 42 40 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@@H](O)C2(C)C)cc1F ZINC000880920439 CE On-Demand Anodyne ENV 41 39 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](O)C2(C)C)cc1F ZINC000880920440 CE On-Demand Anodyne ENV 41 39 CN(C)c1ccc(NC(=O)N[C@H]2C[C@@H](O)C2(C)C)cc1F ZINC000880920441 CE On-Demand Anodyne ENV 41 39 CN(C)c1ccc(NC(=O)N[C@H]2C[C@H](O)C2(C)C)cc1F ZINC000880920442 CE On-Demand Anodyne ENV 41 39 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920484 FE On-Demand Anodyne NPY2R 40 32 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920484 FE On-Demand Anodyne CCR3 66 40 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920484 FE On-Demand Anodyne EPHX2 20 43 CN1C(=O)NC2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)C1=O ZINC000880920595 FD On-Demand Anodyne CACNA1H 59 43 CN(C)c1ccc(NC(=O)N[C@H](CO)Cc2ccc(O)cc2)cc1F ZINC000880920603 EE On-Demand Anodyne GRIA1 41 32 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920612 EC On-Demand Anodyne CACNA1H 27 43 CN(C)c1nccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)n1 ZINC000880920651 EE On-Demand Anodyne KIT 17 51 CN(C)c1nccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)n1 ZINC000880920651 EE On-Demand Anodyne BRAF 16 51 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920656 FD On-Demand Anodyne NPY2R 45 33 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880920657 FD On-Demand Anodyne NPY2R 45 33 CCC1(O)CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880920705 DG On-Demand Anodyne EPHX2 48 40 CCC1(NC(=O)Nc2ccc(N(C)C)c(F)c2)CCOCC1 ZINC000880920793 DF On-Demand Anodyne EPHX2 17 41 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1 ZINC000880920824 DE On-Demand Anodyne CACNA1H 33 43 CN1CC[C@@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1 ZINC000880920824 DE On-Demand Anodyne EPHX2 35 44 Cc1c(NC(=O)Nc2ccc(N(C)C)c(F)c2)cnn1C1CCOCC1 ZINC000880920856 FG On-Demand Anodyne MTOR 63 35 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCC1(F)F ZINC000880920895 DG On-Demand Anodyne CACNA1H 39 43 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCC1(F)F ZINC000880920896 DG On-Demand Anodyne CACNA1H 39 43 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920914 CE On-Demand Anodyne TRPC6 45 31 C[C@H]1[C@H](O)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920915 CE On-Demand Anodyne TRPC6 45 31 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920917 CE On-Demand Anodyne TRPC6 45 31 CNc1nc(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)cs1 ZINC000880920922 EG On-Demand Anodyne TRPC6 65 51 CNc1nc(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)cs1 ZINC000880920922 EG On-Demand Anodyne TRPC3 56 48 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(S(=O)(=O)N(C)C)C2)cc1F ZINC000880920933 GD On-Demand Anodyne EPHX2 42 40 COC(=O)C[C@](C)(NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccn1 ZINC000880920942 FF On-Demand Anodyne GRM4 32 40 COC(=O)C[C@@](C)(NC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccccn1 ZINC000880920943 FF On-Demand Anodyne GRM4 32 40 CC[C@H]1[C@H](CO)CCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920961 DF On-Demand Anodyne NPY2R 47 36 CC[C@H]1[C@@H](CO)CCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920962 DF On-Demand Anodyne NPY2R 47 36 CC[C@@H]1[C@H](CO)CCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880920963 DF On-Demand Anodyne NPY2R 47 36 CSC1(CNC(=O)Nc2ccc(N(C)C)c(F)c2)CCN(C)CC1 ZINC000880920985 FF On-Demand Anodyne MCHR1 16 44 Cc1nnc(CCNC(=O)Nc2ccc(N(C)C)c(F)c2)s1 ZINC000880920995 DE On-Demand Anodyne PRMT3 61 34 COC[C@]1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921007 ED On-Demand Anodyne CACNA1H 47 42 COC[C@]1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921007 ED On-Demand Anodyne EPHX2 34 41 CN(C)c1ccc(NC(=O)N[C@](C)(CO)c2cccc(O)c2)cc1F ZINC000880921055 EF On-Demand Anodyne IMDH_CRYPV 61 37 CN(C)c1ccc(NC(=O)N[C@@](C)(CO)c2cccc(O)c2)cc1F ZINC000880921056 EF On-Demand Anodyne IMDH_CRYPV 61 37 Cc1ccncc1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921089 DF On-Demand Anodyne NAMPT 33 56 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921095 FF On-Demand Anodyne EPHX2 15 44 CCC[C@]1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921116 DF On-Demand Anodyne CACNA1H 31 40 CCC[C@]1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921116 DF On-Demand Anodyne EPHX2 30 40 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921160 EE On-Demand Anodyne NPY2R 59 35 CN(C[C@@H](O)Cc1ccccc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921220 EF On-Demand Anodyne NPY5R 34 40 CN(C[C@H](O)Cc1ccccc1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921221 EF On-Demand Anodyne NPY5R 34 40 CN(C)c1ccc(NC(=O)N[C@@H]2COc3ccccc3[C@@H]2O)cc1F ZINC000880921263 EF On-Demand Anodyne NPY2R 42 34 CN(C)c1ccc(NC(=O)N[C@@H]2COc3ccccc3[C@H]2O)cc1F ZINC000880921264 EF On-Demand Anodyne NPY2R 42 34 CN(C)c1ccc(NC(=O)N[C@H]2COc3ccccc3[C@H]2O)cc1F ZINC000880921265 EF On-Demand Anodyne NPY2R 42 34 CN(C)c1ccc(NC(=O)N[C@H]2COc3ccccc3[C@@H]2O)cc1F ZINC000880921266 EF On-Demand Anodyne NPY2R 42 34 COCCN(CCOC)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921281 GE On-Demand Anodyne EPHX2 19 40 COC(OC)c1ccc(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)o1 ZINC000880921283 FH On-Demand Anodyne CCR2 22 43 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921321 FD On-Demand Anodyne HLA-DRB1 45 34 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921322 FD On-Demand Anodyne HLA-DRB1 45 34 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921337 EE On-Demand Anodyne CCR3 86 40 CC(=O)N1CCC[C@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921337 EE On-Demand Anodyne EPHX2 20 41 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921338 EE On-Demand Anodyne CCR3 86 40 CC(=O)N1CCC[C@@H](CNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921338 EE On-Demand Anodyne EPHX2 20 41 CN(C)c1ccc(NC(=O)N[C@H]2CC[C@@H](C(=O)N3CCCCC3)C2)cc1F ZINC000880921357 GG On-Demand Anodyne EPHX2 51 47 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne ADRA1D 17 40 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne HTR1D 17 52 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne HTR1B 20 52 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne PDGFRB 65 49 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne NPY2R 74 39 COc1cnccc1N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921384 FF On-Demand Anodyne RBP4 19 41 O=C1NCC[C@@H]1CC(=O)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880921417 EE On-Demand Anodyne CCR2 15 43 O=C1NCC[C@H]1CC(=O)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880921419 EE On-Demand Anodyne CCR2 15 43 CO[C@@]1(C)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921421 DF On-Demand Anodyne EPHX2 34 46 CN(C[C@@H](O)c1cccc(C#N)c1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921512 FF On-Demand Mild MCHR1 26 43 CCO[C@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921516 CF On-Demand Anodyne EPHX2 54 42 CN1CCC[C@@H](CCNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921526 DF On-Demand Anodyne CCR3 85 42 CN1CCC[C@@H](CCNC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921526 DF On-Demand Anodyne PRMT3 24 42 Cc1noc(C)c1C(C)(C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921528 EH On-Demand Anodyne IMDH_CRYPV 56 33 CCn1cc([C@H](C)NC(=O)Nc2ccc(N(C)C)c(F)c2)cn1 ZINC000880921538 DF On-Demand Anodyne NPY2R 51 33 CCc1nnc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)s1 ZINC000880921555 DF On-Demand Anodyne PRMT3 53 34 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880921612 GG On-Demand Anodyne CA2 17 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880921612 GG On-Demand Anodyne CA1 42 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880921612 GG On-Demand Anodyne CA12 31 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880921612 GG On-Demand Anodyne CA9 31 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880921612 GG On-Demand Anodyne P96878_MYCTU 46 40 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@H](C(N)=O)C2)cc1F ZINC000880921617 DD On-Demand Anodyne EPHX2 43 39 COC(=O)[C@@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)CC1CC1 ZINC000880921626 EF On-Demand Anodyne NPY2R 44 35 COC(=O)[C@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)CC1CC1 ZINC000880921627 EF On-Demand Anodyne NPY2R 44 35 CCC(=O)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921632 DD On-Demand Anodyne NPY2R 44 34 O=C1CC[C@H](c2ccc(C(=O)N3CCc4ccc(C(F)(F)F)cc4C3)cc2)N1 ZINC000880921744 GH On-Demand Anodyne CCR2 18 41 O=C1CC[C@@H](c2ccc(C(=O)N3CCc4ccc(C(F)(F)F)cc4C3)cc2)N1 ZINC000880921745 GH On-Demand Anodyne CCR2 18 41 COc1cc(NC(=O)c2ccco2)c(C(=O)NCCc2ccc(Br)s2)cc1OC ZINC000880921763 JI On-Demand Anodyne NQO2 15 42 CN(C)c1ccc(NC(=O)Nc2cnn(Cc3nnc4n3CCCC4)c2)cc1F ZINC000880921772 GF On-Demand Anodyne PANC 53 36 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCCO)C2)cc1F ZINC000880921782 ED On-Demand Anodyne SLC6A1 53 33 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCCO)C2)cc1F ZINC000880921782 ED On-Demand Anodyne CCR3 72 46 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCCO)C2)cc1F ZINC000880921782 ED On-Demand Anodyne EPHX2 42 46 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCCO)C2)cc1F ZINC000880921784 ED On-Demand Anodyne SLC6A1 53 33 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCCO)C2)cc1F ZINC000880921784 ED On-Demand Anodyne CCR3 72 46 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCCO)C2)cc1F ZINC000880921784 ED On-Demand Anodyne EPHX2 42 46 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921808 GF On-Demand Anodyne CACNA1H 33 40 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921808 GF On-Demand Anodyne EPHX2 36 43 CN(C)c1ccc(NC(=O)N[C@H]2CC23CCOCC3)cc1F ZINC000880921814 DF On-Demand Anodyne ENV 40 35 CN(C)c1ccc(NC(=O)N[C@@H]2CC23CCOCC3)cc1F ZINC000880921815 DF On-Demand Anodyne ENV 40 35 CN(C)c1ccc(NC(=O)N[C@@H]2[C@H]3COC[C@H]32)cc1F ZINC000880921816 CD On-Demand Anodyne EPHX2 20 40 CSCC[C@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C(=O)N(C)C ZINC000880921826 FE On-Demand Anodyne FPR1 31 41 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880921834 DE On-Demand Anodyne CCR3 44 34 CON(C)C(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921838 FE On-Demand Anodyne EPHX2 20 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCOC2(C)C)cc1F ZINC000880921850 CF On-Demand Anodyne ENV 40 37 CN(C)c1ccc(NC(=O)N[C@H]2CCOC2(C)C)cc1F ZINC000880921851 CF On-Demand Anodyne ENV 40 37 CN(C)c1ccc(NC(=O)N[C@@H]2CCn3ccnc32)cc1F ZINC000880921863 DE On-Demand Anodyne CCKBR 50 33 CN(C)c1ccc(NC(=O)N[C@H]2CCn3ccnc32)cc1F ZINC000880921864 DE On-Demand Anodyne CCKBR 50 33 CNc1ncc(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)s1 ZINC000880921888 EG On-Demand Anodyne CCR2 26 41 O=C(COC1CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880921942 CF On-Demand Anodyne CCR2 25 44 O=C(COC1CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880921942 CF On-Demand Anodyne LIPG 56 42 CN(C)C(=O)OC1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880921951 FF On-Demand Anodyne EPHX2 27 40 CCOC(=O)[C@@]1(COC)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921963 GF On-Demand Anodyne EPHX2 23 42 CCOC(=O)[C@]1(COC)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880921964 GF On-Demand Anodyne EPHX2 23 42 CCOC(=O)C1([S@@](C)=O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922001 GE On-Demand Anodyne CACNA1H 47 39 CCOC(=O)C1([S@](C)=O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922003 GE On-Demand Anodyne CACNA1H 47 39 O=C([C@@H]1CCc2nncn2CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922025 FF On-Demand Anodyne CCR2 24 42 O=C([C@H]1CCc2nncn2CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922027 FF On-Demand Anodyne CCR2 24 42 COC[C@@]1(C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922058 DF On-Demand Anodyne CACNA1H 43 41 COC[C@]1(C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922060 DF On-Demand Anodyne CACNA1H 43 41 C[C@@H]1CN(CCCNC(=O)Nc2ccc(N(C)C)c(F)c2)CCCO1 ZINC000880922117 FF On-Demand Anodyne CCR3 56 46 C[C@@H]1CN(CCCNC(=O)Nc2ccc(N(C)C)c(F)c2)CCCO1 ZINC000880922117 FF On-Demand Anodyne CHRNA7 19 43 C[C@@H]1CN(CCCNC(=O)Nc2ccc(N(C)C)c(F)c2)CCCO1 ZINC000880922117 FF On-Demand Anodyne EPHX2 20 41 CN(C)c1ccc(NC(=O)N[C@H]2COC(C)(C)C2)cc1F ZINC000880922131 CF On-Demand Anodyne ENV 45 45 CN(C)c1ccc(NC(=O)N[C@@H]2COC(C)(C)C2)cc1F ZINC000880922132 CF On-Demand Anodyne ENV 45 45 CN(C)c1ccc(NC(=O)N[C@H]2CCc3nnnn3CC2)cc1F ZINC000880922185 ED On-Demand Anodyne EPHX2 46 44 CN(C)c1ccc(NC(=O)N[C@@H]2CCc3nnnn3CC2)cc1F ZINC000880922186 ED On-Demand Anodyne EPHX2 46 44 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922195 EF On-Demand Anodyne EPHX2 33 45 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H]2CCO)cc1F ZINC000880922245 DF On-Demand Anodyne CCR3 30 42 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@H]2CCO)cc1F ZINC000880922246 DF On-Demand Anodyne CCR3 30 42 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@@H]2CCO)cc1F ZINC000880922247 DF On-Demand Anodyne CCR3 30 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H]2CCO)cc1F ZINC000880922248 DF On-Demand Anodyne CCR3 30 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H]2CNS(C)(=O)=O)cc1F ZINC000880922267 FD On-Demand Anodyne CCR3 23 41 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@H]2CNS(C)(=O)=O)cc1F ZINC000880922268 FD On-Demand Anodyne CCR3 23 41 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@@H]2CNS(C)(=O)=O)cc1F ZINC000880922269 FD On-Demand Anodyne CCR3 23 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H]2CNS(C)(=O)=O)cc1F ZINC000880922270 FD On-Demand Anodyne CCR3 23 41 O=C([C@@H]1OC[C@@H]2CCC[C@@H]21)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922272 EG On-Demand Anodyne CCR2 30 44 COCCO[C@@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922284 EE On-Demand Anodyne LIPG 26 40 COCCO[C@H]1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922285 EE On-Demand Anodyne LIPG 26 40 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922296 GF On-Demand Anodyne CCR2 25 44 COC1(CO)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922303 ED On-Demand Anodyne CACNA1H 60 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCn3ccnc3C2)cc1F ZINC000880922313 DE On-Demand Anodyne EPHX2 42 39 CN(C)c1ccc(NC(=O)N[C@H]2CCn3ccnc3C2)cc1F ZINC000880922314 DE On-Demand Anodyne EPHX2 42 39 CN(C)C(=O)Nc1ccc(CNC(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880922327 FG On-Demand Anodyne ROCK2 16 41 CN(C)c1ccc(NC(=O)N[C@@H]2CC23CC3)cc1F ZINC000880922427 CF On-Demand Anodyne ENV 42 38 CN(C)c1ccc(NC(=O)N[C@H]2CC23CC3)cc1F ZINC000880922428 CF On-Demand Anodyne ENV 42 38 CC[C@H](C)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922469 DF On-Demand Anodyne CACNA1H 52 41 CC[C@H](C)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922469 DF On-Demand Anodyne NPY2R 67 40 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922499 DI On-Demand Anodyne CCR2 22 43 O=C(C[C@@H]1C[C@H]1C1CC1)N1CCc2ccc(C(F)(F)F)cc2C1 ZINC000880922499 DI On-Demand Anodyne LIPG 47 33 CC(C)C1(O)CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922515 CE On-Demand Anodyne CACNA1H 23 43 CN(C)c1ccc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc1F ZINC000880922518 EH On-Demand Anodyne IMDH_CRYPV 60 37 CN(C)c1ccc(NC(=O)Nc2cccc(C(C)(C)O)c2)cc1F ZINC000880922518 EH On-Demand Anodyne KCNK3 47 33 CC[C@@H](C)n1ncc(NC(=O)Nc2ccc(N(C)C)c(F)c2)c1C ZINC000880922519 EI On-Demand Anodyne NPY2R 46 35 CN(C)c1ccc(NC(=O)N[C@@H](CO)CC2CCC2)cc1F ZINC000880922525 DF On-Demand Anodyne CCR3 47 33 CN(C)c1ccc(NC(=O)N[C@H](CO)CC2CCC2)cc1F ZINC000880922526 DF On-Demand Anodyne CCR3 47 33 Cc1cc(N2CCC[C@H](NC(=O)Nc3ccc(N(C)C)c(F)c3)C2)n(C)n1 ZINC000880922570 FF On-Demand Anodyne CCR3 46 32 CO[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCO1 ZINC000880922617 CD On-Demand Anodyne EPHX2 27 40 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@](C)(O)C2)cc1F ZINC000880922632 CD On-Demand Anodyne EPHX2 40 38 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@](C)(O)C2)cc1F ZINC000880922632 CD On-Demand Anodyne ENV 48 43 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(S(C)(=O)=O)C2)cc1F ZINC000880922646 ED On-Demand Anodyne CCR3 17 45 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(S(C)(=O)=O)C2)cc1F ZINC000880922646 ED On-Demand Anodyne EPHX2 52 53 CN(C)c1ccc(NC(=O)N[C@H]2CCN(S(C)(=O)=O)C2)cc1F ZINC000880922647 ED On-Demand Anodyne CCR3 17 45 CN(C)c1ccc(NC(=O)N[C@H]2CCN(S(C)(=O)=O)C2)cc1F ZINC000880922647 ED On-Demand Anodyne EPHX2 52 53 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H]2CO)cc1F ZINC000880922649 CE On-Demand Anodyne CCR3 31 44 C#CC[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922651 DG On-Demand Mild EPHX2 15 43 C#CC[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922652 DG On-Demand Mild EPHX2 15 43 C[C@H](O)CN(C(=O)Nc1ccc(N(C)C)c(F)c1)C1CC1 ZINC000880922669 CE On-Demand Anodyne MCHR1 25 40 COC[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922677 DG On-Demand Anodyne EPHX2 19 41 C[C@@H]1[C@@H](C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)CCN1C ZINC000880922683 EF On-Demand Anodyne CCR2 30 46 C[C@H]1[C@H](C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)CCN1C ZINC000880922685 EF On-Demand Anodyne CCR2 30 46 CN(C)c1ccc(NC(=O)Nc2cc(C3CC3)[nH]n2)cc1F ZINC000880922696 DG On-Demand Anodyne CDK2 17 52 CN(C)c1ccc(NC(=O)Nc2cc(C3CC3)[nH]n2)cc1F ZINC000880922696 DG On-Demand Anodyne PKNB 66 37 COC[C@@H](O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922747 CD On-Demand Anodyne ADRB1 43 35 COc1nn(C)cc1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922753 DE On-Demand Anodyne HTR2A 33 40 CC[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCCO1 ZINC000880922781 DF On-Demand Anodyne NPY2R 61 34 COCC1CCC(NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880922823 DG On-Demand Anodyne EPHX2 48 43 COc1ccc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)nc1 ZINC000880922826 FF On-Demand Anodyne PDGFRB 60 44 COc1ccc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)nc1 ZINC000880922826 FF On-Demand Anodyne NPY2R 41 39 COc1ccc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)nc1 ZINC000880922826 FF On-Demand Anodyne FAAH 22 41 COc1ccc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)nc1 ZINC000880922826 FF On-Demand Anodyne MET 16 40 COc1ccc(N2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)nc1 ZINC000880922826 FF On-Demand Anodyne DGAT1 35 49 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922827 GE On-Demand Anodyne CACNA1H 32 40 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922827 GE On-Demand Anodyne EPHX2 34 41 COC(=O)CNC(=O)CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922844 EC On-Demand Anodyne F7 22 40 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922854 DE On-Demand Anodyne CHRNA10 58 37 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922854 DE On-Demand Anodyne ACKR3 64 33 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922855 DE On-Demand Anodyne CHRNA10 58 37 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922855 DE On-Demand Anodyne ACKR3 64 33 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922868 DD On-Demand Anodyne EPHX2 46 38 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne CA2 17 45 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne CA1 53 44 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne EPHX2 15 44 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne CA12 33 45 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne CA9 32 45 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne NCE103 20 45 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne MTCA1 39 45 CN(C)c1ccc(NC(=O)Nc2ccc(OCCS(C)(=O)=O)cc2)cc1F ZINC000880922879 GF On-Demand Anodyne P96878_MYCTU 43 45 CCN(C)C(=O)[C@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922916 DD On-Demand Anodyne NPY2R 43 36 CCN(C)C(=O)[C@@H](C)NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880922917 DD On-Demand Anodyne NPY2R 43 36 CCN1CC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1=O ZINC000880922919 DD On-Demand Anodyne EPHX2 29 40 CCN1CC[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1=O ZINC000880922920 DD On-Demand Anodyne EPHX2 29 40 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922988 ED On-Demand Anodyne CACNA1H 28 40 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922988 ED On-Demand Anodyne EPHX2 31 45 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922991 FE On-Demand Anodyne EPHX2 20 40 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880922992 FE On-Demand Anodyne EPHX2 20 40 CCn1c(O)nnc1C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923000 GF On-Demand Anodyne NPY2R 41 33 COCC(COC)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923008 FD On-Demand Anodyne PDGFRB 41 37 COCC(COC)N1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923008 FD On-Demand Anodyne NPY2R 54 36 C[C@H](c1cccc(C#N)c1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923009 EH On-Demand Mild MCHR1 25 43 C[C@@H](c1cccc(C#N)c1)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923010 EH On-Demand Mild MCHR1 25 43 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)(N2CCOCC2)CC1 ZINC000880923024 GD On-Demand Anodyne EPHX2 27 45 CN1CCC(CNC(=O)Nc2ccc(N(C)C)c(F)c2)(N2CCOCC2)CC1 ZINC000880923024 GD On-Demand Anodyne HCN1 44 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H]([S@@](C)=O)C2)cc1F ZINC000880923042 EF On-Demand Anodyne EPHX2 35 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H]([S@](C)=O)C2)cc1F ZINC000880923043 EF On-Demand Anodyne EPHX2 35 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H]([S@](C)=O)C2)cc1F ZINC000880923044 EF On-Demand Anodyne EPHX2 35 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H]([S@@](C)=O)C2)cc1F ZINC000880923046 EF On-Demand Anodyne EPHX2 35 40 CN(CCN1CCCCC1)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923067 DF On-Demand Anodyne MCHR1 39 42 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](O)[C@H]2n2cccn2)cc1F ZINC000880923081 ED On-Demand Anodyne CCKBR 54 34 CCO[C@@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923106 CF On-Demand Anodyne EPHX2 54 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCO[C@H]2c2ccccc2)cc1F ZINC000880923138 EH On-Demand Anodyne EPHX2 16 40 CN(C)c1ccc(NC(=O)Nc2ccn(CC(=O)N3CCOCC3)n2)cc1F ZINC000880923140 GD On-Demand Anodyne EPHX2 23 48 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@@H](N3CCOCC3)C23CCC3)cc1F ZINC000880923142 GF On-Demand Anodyne EPHX2 18 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C[C@H]2O)cc1F ZINC000880923183 GE On-Demand Anodyne F13A1 15 41 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C[C@H]2O)cc1F ZINC000880923184 GE On-Demand Anodyne F13A1 15 41 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)OC(C)(C)C)C[C@@H]2O)cc1F ZINC000880923185 GE On-Demand Anodyne F13A1 15 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)OC(C)(C)C)C[C@@H]2O)cc1F ZINC000880923186 GE On-Demand Anodyne F13A1 15 41 CCC1(N(C)C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923194 EG On-Demand Anodyne CACNA1H 61 44 CCC1(N(C)C)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923194 EG On-Demand Anodyne NPY2R 55 34 C[C@@H](CNC(=O)Nc1ccc(N(C)C)c(F)c1)c1ccc(S(C)(=O)=O)cc1 ZINC000880923206 GG On-Demand Anodyne PRMT3 17 40 C[C@@H](C1CC1)n1cc(NC(=O)Nc2ccc(N(C)C)c(F)c2)cn1 ZINC000880923218 EH On-Demand Anodyne ITK 44 33 CS(=O)(=O)C1CCC(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)CC1 ZINC000880923267 GG On-Demand Anodyne CACNA1B 48 37 CS(=O)(=O)C1CCC(C(=O)N2CCc3ccc(C(F)(F)F)cc3C2)CC1 ZINC000880923267 GG On-Demand Anodyne CCR2 28 44 CC(C)n1ccc(NC(=O)Nc2ccc(N(C)C)c(F)c2)n1 ZINC000880923268 DG On-Demand Anodyne FPR2 43 37 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923270 FD On-Demand Anodyne EPHX2 23 46 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923275 FD On-Demand Anodyne EPHX2 23 46 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C[C@H]1C(=O)N1CCOCC1 ZINC000880923280 GD On-Demand Anodyne EPHX2 16 45 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923282 GG On-Demand Anodyne NPY2R 46 35 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923282 GG On-Demand Anodyne CCR3 36 48 CN(C)c1ccc(NC(=O)N[C@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923282 GG On-Demand Anodyne EPHX2 66 50 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923283 GG On-Demand Anodyne NPY2R 46 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923283 GG On-Demand Anodyne CCR3 36 48 CN(C)c1ccc(NC(=O)N[C@@H]2CCN(C(=O)Nc3ccccc3)C2)cc1F ZINC000880923283 GG On-Demand Anodyne EPHX2 66 50 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[C@@H]1O ZINC000880923285 CE On-Demand Anodyne EPHX2 15 40 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[C@H]1O ZINC000880923286 CE On-Demand Anodyne EPHX2 15 40 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[C@H]1O ZINC000880923287 CE On-Demand Anodyne EPHX2 15 40 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[C@@H]1O ZINC000880923288 CE On-Demand Anodyne EPHX2 15 40 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC[C@@H](C)O1 ZINC000880923355 DF On-Demand Anodyne EPHX2 16 41 CN(C)c1ccc(NC(=O)N[C@H]2COC3(CCC3)C2)cc1F ZINC000880923359 DF On-Demand Anodyne ENV 43 37 CN(C)c1ccc(NC(=O)N[C@@H]2COC3(CCC3)C2)cc1F ZINC000880923360 DF On-Demand Anodyne ENV 43 37 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923401 DF On-Demand Anodyne CACNA1H 45 44 C[C@@H](CO)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923401 DF On-Demand Anodyne NPY2R 64 38 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C(=O)NC ZINC000880923415 CD On-Demand Anodyne NPY2R 40 35 C[C@H]1[C@H](CO)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923468 DF On-Demand Anodyne TRPC6 43 31 C[C@@H]1[C@@H](CO)CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923469 DF On-Demand Anodyne TRPC6 43 31 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](C(N)=O)C2)cc1F ZINC000880923472 CD On-Demand Anodyne EPHX2 41 38 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923475 FG On-Demand Anodyne CACNA1H 53 42 COC1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880923475 FG On-Demand Anodyne TRPM8 28 40 CN(C)c1ccc(NC(=O)N[C@H]2CCCN3CCCC[C@H]23)cc1F ZINC000880923484 EG On-Demand Anodyne CCR3 32 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN3CCCC[C@H]23)cc1F ZINC000880923485 EG On-Demand Anodyne CCR3 32 42 CN(C)c1ccc(NC(=O)N[C@H]2CCCN3CCCC[C@@H]23)cc1F ZINC000880923486 EG On-Demand Anodyne CCR3 32 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN3CCCC[C@@H]23)cc1F ZINC000880923487 EG On-Demand Anodyne CCR3 32 42 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923503 ED On-Demand Anodyne CACNA1H 34 41 CO[C@@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923522 CE On-Demand Anodyne EPHX2 48 41 COC[C@@H]1CCCN1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923553 DE On-Demand Anodyne CCR3 15 43 COC[C@@H]1CCCN1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923553 DE On-Demand Anodyne CASP7 41 34 CN1Cc2ccccc2[C@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1=O ZINC000880923561 FF On-Demand Anodyne CCKBR 43 34 CN1Cc2ccccc2[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1=O ZINC000880923562 FF On-Demand Anodyne CCKBR 43 34 CS[C@@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923586 CF On-Demand Anodyne EPHX2 40 37 CN(C)c1ccc(NC(=O)N[C@H]2C[C@@H]3C[C@@H]3C2)cc1F ZINC000880923629 CF On-Demand Anodyne EPHX2 47 40 CN(C)c1ccc(NC(=O)N[C@H]2C[C@@H]3C[C@@H]3C2)cc1F ZINC000880923629 CF On-Demand Anodyne ENV 41 36 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](O)C2)cc1F ZINC000880923644 CD On-Demand Anodyne EPHX2 47 39 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](O)C2)cc1F ZINC000880923644 CD On-Demand Anodyne ENV 40 35 CN(C)c1ccc(NC(=O)N[C@H]2CCOC2=O)cc1F ZINC000880923651 CD On-Demand Anodyne LUXR 76 43 CN(C)c1ccc(NC(=O)N[C@H]2CCOC2=O)cc1F ZINC000880923651 CD On-Demand Anodyne TRAR 88 41 CN(C)c1ccc(NC(=O)N[C@H]2CCOC2=O)cc1F ZINC000880923651 CD On-Demand Anodyne LASR 60 37 C[C@@H](CCO)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923665 CE On-Demand Anodyne NPY5R 34 41 C[C@H](CCO)N(C)C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923666 CE On-Demand Anodyne NPY5R 34 41 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne NPY1R 28 40 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne CCKAR 64 42 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne NPY2R 45 33 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne PYGL 34 48 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne PYGM 31 48 CN(C)c1ccc(NC(=O)N[C@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923685 FF On-Demand Anodyne CCKBR 82 42 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne NPY1R 28 40 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne CCKAR 64 42 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne NPY2R 45 33 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne PYGL 34 48 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne PYGM 31 48 CN(C)c1ccc(NC(=O)N[C@@H]2Cc3ccccc3N(C)C2=O)cc1F ZINC000880923686 FF On-Demand Anodyne CCKBR 82 42 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@@H](CO)C2)cc1F ZINC000880923689 DF On-Demand Anodyne EPHX2 43 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@H](CO)C2)cc1F ZINC000880923690 DF On-Demand Anodyne EPHX2 43 41 CN(C)c1ccc(NC(=O)N[C@H]2CCC[C@H](CO)C2)cc1F ZINC000880923691 DF On-Demand Anodyne EPHX2 43 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCC[C@@H](CO)C2)cc1F ZINC000880923692 DF On-Demand Anodyne EPHX2 43 41 CCO[C@@]1(C)C[C@H]1NC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880923749 CF On-Demand Anodyne ENV 40 35 CSCC[C@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)C(N)=O ZINC000880923776 ED On-Demand Anodyne FPR1 31 41 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc(N(C)C)c(F)c1)CC2 ZINC000880923787 FG On-Demand Anodyne P2RY14 47 35 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)cc1F ZINC000880923840 ED On-Demand Anodyne CCR3 42 43 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)cc1F ZINC000880923840 ED On-Demand Anodyne EPHX2 46 39 CN(C)c1ccc(NC(=O)N[C@H]2CCN(CC(C)(C)O)C2)cc1F ZINC000880923840 ED On-Demand Anodyne CXCR3 21 42 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880923860 DD On-Demand Anodyne EPHX2 46 38 COC[C@@H]1CCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880924022 CF On-Demand Anodyne MCHR1 15 41 C[C@H]1c2ccccc2OCCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880924039 EH On-Demand Anodyne NPY2R 52 33 CCC1(N2CCCC2)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924053 FH On-Demand Anodyne CACNA1H 44 41 COC(=O)C1=NO[C@@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1 ZINC000880924075 FD On-Demand Anodyne EPHX2 33 40 COC(=O)C1=NO[C@]2(CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)C2)C1 ZINC000880924076 FD On-Demand Anodyne EPHX2 33 40 CCC1(N2CCOCC2)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924083 GG On-Demand Anodyne CACNA1H 35 40 CCC1(N2CCOCC2)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924083 GG On-Demand Anodyne EPHX2 33 40 CCN1CC[C@H](N(CC)C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880924176 DF On-Demand Anodyne NPY2R 46 36 CCN1CC[C@@H](N(CC)C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880924177 DF On-Demand Anodyne NPY2R 46 36 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@@H](C(N)=O)C2)cc1F ZINC000880924187 CD On-Demand Anodyne EPHX2 41 38 CN(C)c1ccc(NC(=O)N[C@@H](c2ccccn2)C2CCC2)cc1F ZINC000880924239 EH On-Demand Anodyne NPY2R 49 35 CN(C)c1ccc(NC(=O)N[C@H](c2ccccn2)C2CCC2)cc1F ZINC000880924240 EH On-Demand Anodyne NPY2R 49 35 CN(C)c1ccc(NC(=O)N[C@H]2C[C@H](O)C2)cc1F ZINC000880924247 CD On-Demand Anodyne EPHX2 47 39 CN(C)c1ccc(NC(=O)N[C@H]2C[C@H](O)C2)cc1F ZINC000880924247 CD On-Demand Anodyne ENV 40 35 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H](CO)C2)cc1F ZINC000880924262 CD On-Demand Anodyne EPHX2 41 37 COCC1CC(NC(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880924264 CE On-Demand Anodyne EPHX2 44 37 COC[C@@H]1CCCN1NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924303 FE On-Demand Mild LGMN 54 33 COC[C@@H]1CCCN1NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924303 FE On-Demand Mild CHRNA10 24 41 COC[C@@H]1CCCN1NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924305 FE On-Demand Mild LGMN 54 33 COC[C@@H]1CCCN1NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924305 FE On-Demand Mild CHRNA10 24 41 COC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924309 EF On-Demand Mild DPP4 23 40 COC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924309 EF On-Demand Mild LGMN 65 35 COC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924309 EF On-Demand Mild CHRNA10 25 41 COC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924311 EF On-Demand Mild DPP4 23 40 COC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924311 EF On-Demand Mild LGMN 65 35 COC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924311 EF On-Demand Mild CHRNA10 25 41 CN1CCN(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880924325 FE On-Demand Anodyne HTR1D 15 42 CN1CCN(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880924325 FE On-Demand Anodyne HTR1B 15 42 CN1CCN(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880924325 FE On-Demand Anodyne HTR1F 40 37 CN1CCN(C2CCN(C(=O)Nc3ccc(N(C)C)c(F)c3)CC2)CC1 ZINC000880924325 FE On-Demand Anodyne L3MBTL3 74 40 COC(=O)C[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924347 EE On-Demand Mild CTSF 47 33 COC(=O)C[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924348 EE On-Demand Mild CTSF 47 33 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880924427 EF On-Demand Anodyne NPY2R 49 33 N#Cc1cccc([C@H](NC(=O)NC/C=C\CO)C(F)(F)F)c1 ZINC000880924458 DE On-Demand Mild CTSF 48 31 N#Cc1cccc([C@H](NC(=O)NC/C=C/CO)C(F)(F)F)c1 ZINC000880924459 DE On-Demand Mild CTSF 48 31 N#Cc1cccc([C@@H](NC(=O)NC/C=C\CO)C(F)(F)F)c1 ZINC000880924460 DE On-Demand Mild CTSF 48 31 N#Cc1cccc([C@@H](NC(=O)NC/C=C/CO)C(F)(F)F)c1 ZINC000880924461 DE On-Demand Mild CTSF 48 31 CO[C@@H]1CC[C@@H](C)N(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880924515 FG On-Demand Mild HCRTR2 19 40 CO[C@@H]1CC[C@@H](C)N(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880924517 FG On-Demand Mild HCRTR2 19 40 COc1ccc(CN(CCO)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880924519 FF On-Demand Anodyne BMP1 21 42 COc1ccc(CN(CCO)C(=O)Nc2ccc(N(C)C)c(F)c2)cc1 ZINC000880924519 FF On-Demand Anodyne ROCK2 16 46 C[C@@H](O)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880924530 FF On-Demand Mild MCHR1 24 40 C[C@@H](O)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880924531 FF On-Demand Mild MCHR1 24 40 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924567 FD On-Demand Mild OPRK1 18 47 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924567 FD On-Demand Mild CCR3 27 48 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924567 FD On-Demand Mild MCHR1 40 48 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924568 FD On-Demand Mild OPRK1 18 47 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924568 FD On-Demand Mild CCR3 27 48 N#Cc1cccc([C@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924568 FD On-Demand Mild MCHR1 40 48 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924569 FD On-Demand Mild OPRK1 18 47 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924569 FD On-Demand Mild CCR3 27 48 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880924569 FD On-Demand Mild MCHR1 40 48 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924570 FD On-Demand Mild OPRK1 18 47 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924570 FD On-Demand Mild CCR3 27 48 N#Cc1cccc([C@@H](NC(=O)NCCN2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880924570 FD On-Demand Mild MCHR1 40 48 C#C[C@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924657 DD On-Demand Mild CTSF 51 32 C#C[C@@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924658 DD On-Demand Mild CTSF 51 32 C#C[C@@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924659 DD On-Demand Mild CTSF 51 32 C#C[C@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924660 DD On-Demand Mild CTSF 51 32 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](c3nccs3)C2)C(F)(F)F)c1 ZINC000880924675 GH On-Demand Mild ETHR 42 35 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](c3nccs3)C2)C(F)(F)F)c1 ZINC000880924676 GH On-Demand Mild ETHR 42 35 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](c3nccs3)C2)C(F)(F)F)c1 ZINC000880924677 GH On-Demand Mild ETHR 42 35 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](c3nccs3)C2)C(F)(F)F)c1 ZINC000880924678 GH On-Demand Mild ETHR 42 35 C[C@@H](O)C1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880924765 EE On-Demand Mild CTSL 15 40 C[C@@H](O)C1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880924768 EE On-Demand Mild CTSL 15 40 CC[C@@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924777 DE On-Demand Mild CTSF 57 35 CC[C@@H](O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924778 DE On-Demand Mild CTSF 57 35 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H]2C2CCOCC2)cc1F ZINC000880924817 DF On-Demand Anodyne EPHX2 19 40 N#Cc1cccc([C@H](NC(=O)N2CCc3ncncc3C2)C(F)(F)F)c1 ZINC000880924822 FF On-Demand Mild MAPK1 42 33 N#Cc1cccc([C@@H](NC(=O)N2CCc3ncncc3C2)C(F)(F)F)c1 ZINC000880924823 FF On-Demand Mild MAPK1 42 33 N#Cc1cccc([C@@H](NC(=O)N2CCC(O)CC2)C(F)(F)F)c1 ZINC000880924835 EE On-Demand Mild MCHR1 28 42 N#Cc1cccc([C@H](NC(=O)N2CCC(O)CC2)C(F)(F)F)c1 ZINC000880924836 EE On-Demand Mild MCHR1 28 42 CCN1CC[C@@H]1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880924837 CE On-Demand Anodyne NPY2R 51 35 CCN1CC[C@@H]1CNC(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880924837 CE On-Demand Anodyne CCR3 44 39 C#CCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924839 DE On-Demand Mild CACNA1H 42 42 C#CCC1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924839 DE On-Demand Mild S1PR2 29 41 N#Cc1cccc([C@H](NC(=O)N2CCC3(CCNC3=O)CC2)C(F)(F)F)c1 ZINC000880924844 GE On-Demand Mild CACNA1H 38 41 N#Cc1cccc([C@@H](NC(=O)N2CCC3(CCNC3=O)CC2)C(F)(F)F)c1 ZINC000880924845 GE On-Demand Mild CACNA1H 38 41 CN(CC(C)(C)S(C)(=O)=O)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924882 GF On-Demand Mild CTSF 68 36 CN(CC(C)(C)S(C)(=O)=O)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924882 GF On-Demand Mild CTSL 17 40 CN(CC(C)(C)S(C)(=O)=O)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924883 GF On-Demand Mild CTSF 68 36 CN(CC(C)(C)S(C)(=O)=O)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924883 GF On-Demand Mild CTSL 17 40 CN(CC1=CCCOC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924895 FG On-Demand Mild CTSF 53 33 CN(CC1=CCCOC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924896 FG On-Demand Mild CTSF 53 33 CC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924910 DF On-Demand Anodyne CACNA1H 32 43 CC(=O)C1CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880924910 DF On-Demand Anodyne EPHX2 27 40 COC(OC)[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924990 EE On-Demand Mild CTSF 53 34 COC(OC)[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924990 EE On-Demand Mild CTSL 18 41 COC(OC)[C@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924991 EE On-Demand Mild CTSF 53 34 COC(OC)[C@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924991 EE On-Demand Mild CTSL 18 41 COC(OC)[C@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924992 EE On-Demand Mild CTSF 53 34 COC(OC)[C@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924992 EE On-Demand Mild CTSL 18 41 COC(OC)[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924993 EE On-Demand Mild CTSF 53 34 COC(OC)[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924993 EE On-Demand Mild CTSL 18 41 CN(C[C@@H]1CC1(C)C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880924996 EH On-Demand Mild CTSF 51 31 CS(=O)(=O)C1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925010 FD On-Demand Mild CTSF 55 34 CS(=O)(=O)C1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925011 FD On-Demand Mild CTSF 55 34 CN(C[C@@H]1CC1(C)C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925019 EH On-Demand Mild CTSF 51 31 C#C[C@@H]1CC[C@@H](NC(=O)Nc2ccc(N(C)C)c(F)c2)CC1 ZINC000880925064 DG On-Demand Mild EPHX2 46 42 N#Cc1cccc([C@@H](NC(=O)NC(CF)CF)C(F)(F)F)c1 ZINC000880925078 DF On-Demand Mild CTSF 50 33 N#Cc1cccc([C@H](NC(=O)NC(CF)CF)C(F)(F)F)c1 ZINC000880925080 DF On-Demand Mild CTSF 50 33 N#Cc1cccc([C@H](NC(=O)NC[C@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925125 GH On-Demand Mild CCR3 46 44 N#Cc1cccc([C@H](NC(=O)NC[C@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925125 GH On-Demand Mild MCHR1 31 42 N#Cc1cccc([C@@H](NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925132 GH On-Demand Mild CCR3 46 44 N#Cc1cccc([C@@H](NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925132 GH On-Demand Mild MCHR1 31 42 N#Cc1cccc([C@@H](NC(=O)NC[C@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925134 GH On-Demand Mild CCR3 46 44 N#Cc1cccc([C@@H](NC(=O)NC[C@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925134 GH On-Demand Mild MCHR1 31 42 N#Cc1cccc([C@H](NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925136 GH On-Demand Mild CCR3 46 44 N#Cc1cccc([C@H](NC(=O)NC[C@@H]2CCCN(CC3CC3)C2)C(F)(F)F)c1 ZINC000880925136 GH On-Demand Mild MCHR1 31 42 CCOC(=O)[C@H](C)C1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925144 GG On-Demand Mild P2RY12 15 40 CCOC(=O)[C@H](C)C1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925144 GG On-Demand Mild CTRB_BOVIN 46 33 CCOC(=O)[C@H](C)C1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925146 GG On-Demand Mild P2RY12 15 40 CCOC(=O)[C@H](C)C1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925146 GG On-Demand Mild CTRB_BOVIN 46 33 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc(N(C)C)c(F)c1 ZINC000880925152 EI On-Demand Anodyne TRPM8 33 48 N#Cc1cccc([C@H](NC(=O)N2CCc3nccnc3C2)C(F)(F)F)c1 ZINC000880925160 FF On-Demand Mild MAPK1 43 34 N#Cc1cccc([C@@H](NC(=O)N2CCc3nccnc3C2)C(F)(F)F)c1 ZINC000880925161 FF On-Demand Mild MAPK1 43 34 CN(C[C@@](C)(O)c1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925163 GH On-Demand Mild CTSF 65 33 CN(C[C@@](C)(O)c1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925165 GH On-Demand Mild CTSF 65 33 N#Cc1cccc([C@@H](NC(=O)N2C[C@H]3CC[C@@H](O)C[C@H]3C2)C(F)(F)F)c1 ZINC000880925190 FF On-Demand Mild RBP4 41 41 N#Cc1cccc([C@H](NC(=O)N2C[C@H]3CC[C@@H](O)C[C@H]3C2)C(F)(F)F)c1 ZINC000880925191 FF On-Demand Mild RBP4 41 41 N#Cc1cccc([C@H](NC(=O)NCC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880925192 FG On-Demand Mild CTSF 52 33 N#Cc1cccc([C@H](NC(=O)NCC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880925192 FG On-Demand Mild MCHR1 18 41 N#Cc1cccc([C@@H](NC(=O)NCC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880925193 FG On-Demand Mild CTSF 52 33 N#Cc1cccc([C@@H](NC(=O)NCC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880925193 FG On-Demand Mild MCHR1 18 41 C[C@@H]1[C@@H](O)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925230 EF On-Demand Mild DPP4 15 40 C[C@@H]1[C@@H](O)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925230 EF On-Demand Mild LGMN 53 35 C[C@@H]1[C@@H](O)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925233 EF On-Demand Mild DPP4 15 40 C[C@@H]1[C@@H](O)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925233 EF On-Demand Mild LGMN 53 35 C[C@@H](CF)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925250 DF On-Demand Mild CTSF 62 36 C[C@@H](CF)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925250 DF On-Demand Mild CTSL 23 40 C[C@@H](CF)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925250 DF On-Demand Mild CTSS 15 40 C[C@@H](CF)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925251 DF On-Demand Mild CTSF 62 36 C[C@@H](CF)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925251 DF On-Demand Mild CTSL 23 40 C[C@@H](CF)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925251 DF On-Demand Mild CTSS 15 40 CC1(CO)CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925272 EE On-Demand Mild CTSF 66 32 CC1(CO)CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925273 EE On-Demand Mild CTSF 66 32 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](Nc3ncccn3)C2)C(F)(F)F)c1 ZINC000880925274 GF On-Demand Mild MAPK1 24 43 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](Nc3ncccn3)C2)C(F)(F)F)c1 ZINC000880925275 GF On-Demand Mild MAPK1 24 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](Nc3ncccn3)C2)C(F)(F)F)c1 ZINC000880925276 GF On-Demand Mild MAPK1 24 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](Nc3ncccn3)C2)C(F)(F)F)c1 ZINC000880925277 GF On-Demand Mild MAPK1 24 43 CNC(=O)OC[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925285 GG On-Demand Mild LGMN 72 36 CNC(=O)OC[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925287 GG On-Demand Mild LGMN 72 36 C[C@@]1(CO)CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C[C@]1(C)CO ZINC000880925369 GE On-Demand Mild CTSF 67 32 C[C@@]1(CO)CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C[C@]1(C)CO ZINC000880925370 GE On-Demand Mild CTSF 67 32 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@H](O)CC2)cc1F ZINC000880925373 CE On-Demand Anodyne EPHX2 56 45 CN(C)c1ccc(NC(=O)N[C@@H]2CC[C@H](O)CC2)cc1F ZINC000880925373 CE On-Demand Anodyne ENV 40 34 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H]3C[C@@H]3C2)C(F)(F)F)c1 ZINC000880925374 DG On-Demand Mild RBP4 49 39 N#Cc1cccc([C@H](NC(=O)N2CC[C@H]3C[C@H]3C2)C(F)(F)F)c1 ZINC000880925375 DG On-Demand Mild RBP4 49 39 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H]3C[C@H]3C2)C(F)(F)F)c1 ZINC000880925376 DG On-Demand Mild RBP4 49 39 N#Cc1cccc([C@H](NC(=O)N2CC[C@H]3C[C@@H]3C2)C(F)(F)F)c1 ZINC000880925377 DG On-Demand Mild RBP4 49 39 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CCO)C(F)(F)F)c1 ZINC000880925423 EF On-Demand Mild DPP4 15 41 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CCO)C(F)(F)F)c1 ZINC000880925423 EF On-Demand Mild LGMN 55 34 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CCO)C(F)(F)F)c1 ZINC000880925424 EF On-Demand Mild DPP4 15 41 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CCO)C(F)(F)F)c1 ZINC000880925424 EF On-Demand Mild LGMN 55 34 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CCO)C(F)(F)F)c1 ZINC000880925425 EF On-Demand Mild DPP4 15 41 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CCO)C(F)(F)F)c1 ZINC000880925425 EF On-Demand Mild LGMN 55 34 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CCO)C(F)(F)F)c1 ZINC000880925426 EF On-Demand Mild DPP4 15 41 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CCO)C(F)(F)F)c1 ZINC000880925426 EF On-Demand Mild LGMN 55 34 CCN1CC[C@@H](N(CC)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925504 FG On-Demand Mild CCR5 42 47 CCN1CC[C@@H](N(CC)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925504 FG On-Demand Mild MCHR1 42 47 CCN1CC[C@H](N(CC)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925505 FG On-Demand Mild CCR5 42 47 CCN1CC[C@H](N(CC)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925505 FG On-Demand Mild MCHR1 42 47 CCN1CC[C@@H](N(CC)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925506 FG On-Demand Mild CCR5 42 47 CCN1CC[C@@H](N(CC)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925506 FG On-Demand Mild MCHR1 42 47 CCN1CC[C@H](N(CC)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925507 FG On-Demand Mild CCR5 42 47 CCN1CC[C@H](N(CC)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925507 FG On-Demand Mild MCHR1 42 47 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)[C@@H]1CCCOC1 ZINC000880925515 DG On-Demand Anodyne NPY2R 24 40 CC[C@@H](NC(=O)Nc1ccc(N(C)C)c(F)c1)[C@H]1CCCOC1 ZINC000880925516 DG On-Demand Anodyne NPY2R 24 40 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925526 GD On-Demand Anodyne HTR2A 23 41 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925526 GD On-Demand Anodyne CCR3 76 42 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925526 GD On-Demand Anodyne EPHX2 56 56 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925527 GD On-Demand Anodyne HTR2A 23 41 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925527 GD On-Demand Anodyne CCR3 76 42 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(CCN3CCOCC3)C2)cc1F ZINC000880925527 GD On-Demand Anodyne EPHX2 56 56 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880925569 DF On-Demand Anodyne EPHX2 19 42 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880925570 DF On-Demand Anodyne EPHX2 19 42 CC(C)[C@H]1CN(C(=O)Nc2ccc(N(C)C)c(F)c2)CCN1C ZINC000880925590 DF On-Demand Anodyne CACNA1H 27 41 CN(C)CC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925655 EF On-Demand Mild CTSF 72 34 CN(C)CC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925656 EF On-Demand Mild CTSF 72 34 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@H]2c2nc[nH]n2)C(F)(F)F)c1 ZINC000880925657 GG On-Demand Mild CPT1A 90 45 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@@H]2c2nc[nH]n2)C(F)(F)F)c1 ZINC000880925658 GG On-Demand Mild CPT1A 90 45 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@H]2c2nc[nH]n2)C(F)(F)F)c1 ZINC000880925659 GG On-Demand Mild CPT1A 90 45 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@@H]2c2nc[nH]n2)C(F)(F)F)c1 ZINC000880925660 GG On-Demand Mild CPT1A 90 45 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](O)CC2)C(F)(F)F)c1 ZINC000880925677 EF On-Demand Mild MCHR1 23 42 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](O)CC2)C(F)(F)F)c1 ZINC000880925678 EF On-Demand Mild MCHR1 23 42 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](O)CC2)C(F)(F)F)c1 ZINC000880925679 EF On-Demand Mild MCHR1 23 42 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](O)CC2)C(F)(F)F)c1 ZINC000880925680 EF On-Demand Mild MCHR1 23 42 CNc1nc(C(=O)N2CCc3nc(COC)ncc3C2)cs1 ZINC000880925685 DD On-Demand Anodyne TRPC6 49 46 CNc1nc(C(=O)N2CCc3nc(COC)ncc3C2)cs1 ZINC000880925685 DD On-Demand Anodyne TRPC3 40 39 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]3C[C@H]32)C(F)(F)F)c1 ZINC000880925694 DG On-Demand Mild LGMN 44 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]3C[C@@H]32)C(F)(F)F)c1 ZINC000880925695 DG On-Demand Mild LGMN 44 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]3C[C@@H]32)C(F)(F)F)c1 ZINC000880925696 DG On-Demand Mild LGMN 44 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]3C[C@H]32)C(F)(F)F)c1 ZINC000880925697 DG On-Demand Mild LGMN 44 33 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880925735 ED On-Demand Anodyne CACNA1H 36 42 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880925735 ED On-Demand Anodyne EPHX2 34 43 N#Cc1cccc([C@H](NC(=O)N2CCC(CCF)CC2)C(F)(F)F)c1 ZINC000880925744 FH On-Demand Mild MCHR1 27 40 CC(C)C1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880925745 EH On-Demand Mild CTSL 16 41 CC(C)C1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880925746 EH On-Demand Mild CTSL 16 41 N#Cc1cccc([C@@H](NC(=O)N2CCC(CCF)CC2)C(F)(F)F)c1 ZINC000880925748 FH On-Demand Mild MCHR1 27 40 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925750 GG On-Demand Mild CTSF 78 38 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925750 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925751 GG On-Demand Mild CTSF 78 38 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925751 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925752 GG On-Demand Mild CTSF 78 38 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925752 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925754 GG On-Demand Mild CTSF 78 38 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)Cc2ccccc2)C(F)(F)F)c1 ZINC000880925754 GG On-Demand Mild CTRB_BOVIN 45 31 CN1C[C@@H]2CCCN(C(=O)N[C@H](c3cccc(C#N)c3)C(F)(F)F)[C@@H]2C1 ZINC000880925833 FF On-Demand Mild LGMN 59 34 CN1C[C@@H]2CCCN(C(=O)N[C@@H](c3cccc(C#N)c3)C(F)(F)F)[C@@H]2C1 ZINC000880925835 FF On-Demand Mild LGMN 59 34 CN(C)c1ccc(NC(=O)N[C@@H]2CC23CCC3)cc1F ZINC000880925851 CF On-Demand Anodyne ENV 42 37 CN(C)c1ccc(NC(=O)N[C@H]2CC23CCC3)cc1F ZINC000880925856 CF On-Demand Anodyne ENV 42 37 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925864 ED On-Demand Mild LUXR 75 43 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925864 ED On-Demand Mild TRAR 87 42 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925864 ED On-Demand Mild LASR 56 39 N#Cc1cccc([C@@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925866 ED On-Demand Mild LUXR 75 43 N#Cc1cccc([C@@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925866 ED On-Demand Mild TRAR 87 42 N#Cc1cccc([C@@H](NC(=O)N[C@H]2CCOC2=O)C(F)(F)F)c1 ZINC000880925866 ED On-Demand Mild LASR 56 39 CC(=O)NC[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925934 GF On-Demand Mild LGMN 47 33 CC(=O)NC[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880925936 GF On-Demand Mild LGMN 47 33 COCC1(O)CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925958 ED On-Demand Mild CTSF 52 34 COCC1(O)CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880925959 ED On-Demand Mild CTSF 52 34 O=C(NCc1ccc(O)cc1)c1cc([N+](=O)[O-])ccc1N1CCCCC1 ZINC000880925977 FG On-Demand Bother WDR5 36 43 COC[C@]1(CO)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926021 FE On-Demand Mild CTSF 46 32 COC[C@]1(CO)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926022 FE On-Demand Mild CTSF 46 32 CC[C@H](C[C@H](C)O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926060 EG On-Demand Mild CTSF 58 36 CC[C@H](C[C@H](C)O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926063 EG On-Demand Mild CTSF 58 36 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880926086 EG On-Demand Anodyne CACNA1H 43 41 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880926086 EG On-Demand Anodyne EPHX2 36 42 COC[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926099 FG On-Demand Mild CPT1A 36 41 COC[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926099 FG On-Demand Mild LGMN 62 35 COC[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926103 FG On-Demand Mild CPT1A 36 41 COC[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926103 FG On-Demand Mild LGMN 62 35 COc1ccc(CN(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880926104 GI On-Demand Mild PTGES 15 43 COc1ccc(CN(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880926106 GI On-Demand Mild PTGES 15 43 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](CC(N)=O)CC2)C(F)(F)F)c1 ZINC000880926107 GF On-Demand Mild LGMN 58 34 C#CC1(F)CN(C(=O)Nc2ccc(N(C)C)c(F)c2)C1 ZINC000880926108 CE On-Demand Mild CACNA1H 27 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](CC(N)=O)CC2)C(F)(F)F)c1 ZINC000880926113 GF On-Demand Mild LGMN 58 34 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](CC(N)=O)CC2)C(F)(F)F)c1 ZINC000880926115 GF On-Demand Mild LGMN 58 34 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](CC(N)=O)CC2)C(F)(F)F)c1 ZINC000880926117 GF On-Demand Mild LGMN 58 34 C[C@@H](Cc1ccccn1)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926125 FG On-Demand Mild CTSF 62 33 C[C@@H](Cc1ccccn1)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926129 FG On-Demand Mild CTSF 62 33 C[C@H](Cc1ccccn1)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926131 FG On-Demand Mild CTSF 62 33 C[C@H](Cc1ccccn1)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926133 FG On-Demand Mild CTSF 62 33 CC[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)(C)O ZINC000880926134 EG On-Demand Mild CTSF 74 36 CC[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)(C)O ZINC000880926136 EG On-Demand Mild CTSF 74 36 COC[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926150 FH On-Demand Mild REN 15 47 COC[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926152 FH On-Demand Mild REN 15 47 CN(C)CCCC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926156 FH On-Demand Mild CTSF 43 32 CN(C)CCCC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926156 FH On-Demand Mild UTS2 42 33 CN(C)CCCC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926158 FH On-Demand Mild CTSF 43 32 CN(C)CCCC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926158 FH On-Demand Mild UTS2 42 33 N#Cc1cccc([C@@H](NC(=O)NCCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926164 EF On-Demand Mild CTSF 67 33 N#Cc1cccc([C@H](NC(=O)NCCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926166 EF On-Demand Mild CTSF 67 33 N#Cc1cccc([C@H](NC(=O)N2CCc3cc(Cl)nnc3C2)C(F)(F)F)c1 ZINC000880926171 GG On-Demand Mild MAPK1 49 35 N#Cc1cccc([C@@H](NC(=O)N2CCc3cc(Cl)nnc3C2)C(F)(F)F)c1 ZINC000880926172 GG On-Demand Mild MAPK1 49 35 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](F)C2)C(F)(F)F)c1 ZINC000880926173 EG On-Demand Mild DPP4 21 45 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](F)C2)C(F)(F)F)c1 ZINC000880926174 EG On-Demand Mild DPP4 21 45 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](F)C2)C(F)(F)F)c1 ZINC000880926175 EG On-Demand Mild DPP4 21 45 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](F)C2)C(F)(F)F)c1 ZINC000880926176 EG On-Demand Mild DPP4 21 45 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@@H]2CCC[C@H]2O)C(F)(F)F)c1 ZINC000880926179 GG On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@H]2CCC[C@@H]2O)C(F)(F)F)c1 ZINC000880926180 GG On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@H]2CCC[C@H]2O)C(F)(F)F)c1 ZINC000880926181 GG On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@@H]2CCC[C@@H]2O)C(F)(F)F)c1 ZINC000880926182 GG On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N(CCO)CC2CC2)C(F)(F)F)c1 ZINC000880926185 EF On-Demand Mild MCHR1 26 42 N#Cc1cccc([C@@H](NC(=O)N(CCO)CC2CC2)C(F)(F)F)c1 ZINC000880926186 EF On-Demand Mild MCHR1 26 42 CCC(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926193 FE On-Demand Mild CTSF 46 31 CCC(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926194 FE On-Demand Mild CTSF 46 31 CN(C[C@H](O)Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926207 GG On-Demand Mild CTSF 79 39 CN(C[C@H](O)Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926207 GG On-Demand Mild CTRB_BOVIN 45 32 CN(C[C@H](O)Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926208 GG On-Demand Mild CTSF 79 39 CN(C[C@H](O)Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926208 GG On-Demand Mild CTRB_BOVIN 45 32 CN(C[C@@H](O)Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926209 GG On-Demand Mild CTSF 79 39 CN(C[C@@H](O)Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926209 GG On-Demand Mild CTRB_BOVIN 45 32 CN(C[C@@H](O)Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926210 GG On-Demand Mild CTSF 79 39 CN(C[C@@H](O)Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926210 GG On-Demand Mild CTRB_BOVIN 45 32 COc1cccc([C@H](CO)NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)c1 ZINC000880926215 GG On-Demand Mild PTGER3 17 44 COc1cccc([C@H](CO)NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)c1 ZINC000880926215 GG On-Demand Mild CTSF 51 32 COc1cccc([C@H](CO)NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)c1 ZINC000880926217 GG On-Demand Mild PTGER3 17 44 COc1cccc([C@H](CO)NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)c1 ZINC000880926217 GG On-Demand Mild CTSF 51 32 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](n3cc(Cl)cn3)C2)C(F)(F)F)c1 ZINC000880926231 GH On-Demand Mild ITGA4 44 31 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](n3cc(Cl)cn3)C2)C(F)(F)F)c1 ZINC000880926232 GH On-Demand Mild ITGA4 44 31 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](n3cc(Cl)cn3)C2)C(F)(F)F)c1 ZINC000880926233 GH On-Demand Mild ITGA4 44 31 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](n3cc(Cl)cn3)C2)C(F)(F)F)c1 ZINC000880926234 GH On-Demand Mild ITGA4 44 31 N#Cc1cccc([C@@H](NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)C(F)(F)F)c1 ZINC000880926279 GE On-Demand Mild CCR3 15 44 N#Cc1cccc([C@H](NC(=O)NCCN2C[C@@H]3CC[C@H](C2)O3)C(F)(F)F)c1 ZINC000880926280 GE On-Demand Mild CCR3 15 44 CC(C)(CO)[C@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C1CC1 ZINC000880926310 FG On-Demand Mild CTSF 77 35 CC(C)(CO)[C@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C1CC1 ZINC000880926312 FG On-Demand Mild CTSF 77 35 N#Cc1cccc([C@H](NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)C(F)(F)F)c1 ZINC000880926314 GG On-Demand Mild PLM2_PLAFA 47 38 N#Cc1cccc([C@@H](NC(=O)N[C@H]2c3ccccc3C[C@@H]2O)C(F)(F)F)c1 ZINC000880926315 GG On-Demand Mild PLM2_PLAFA 47 38 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@@H]2c2cc[nH]n2)C(F)(F)F)c1 ZINC000880926329 GH On-Demand Mild CPT1A 71 43 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@H]2c2cc[nH]n2)C(F)(F)F)c1 ZINC000880926330 GH On-Demand Mild CPT1A 71 43 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@@H]2c2cc[nH]n2)C(F)(F)F)c1 ZINC000880926331 GH On-Demand Mild CPT1A 71 43 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@H]2c2cc[nH]n2)C(F)(F)F)c1 ZINC000880926332 GH On-Demand Mild CPT1A 71 43 C[C@@H](CCCCO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926334 EG On-Demand Mild CTSF 42 33 C[C@@H](CCCCO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926336 EG On-Demand Mild CTSF 42 33 CN(CCN1CCCCC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926355 FG On-Demand Mild CASR 26 42 CN(CCN1CCCCC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926355 FG On-Demand Mild MCHR1 40 46 CN(CCN1CCCCC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926356 FG On-Demand Mild CASR 26 42 CN(CCN1CCCCC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926356 FG On-Demand Mild MCHR1 40 46 C[C@@H]1[C@@H](CO)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926359 FF On-Demand Mild LGMN 65 36 C[C@@H]1[C@@H](CO)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926360 FF On-Demand Mild LGMN 65 36 CCN(C)C(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880926391 GF On-Demand Mild CTSF 40 38 CCN(C)C(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880926392 GF On-Demand Mild CTSF 40 38 C[C@H]1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CCO1 ZINC000880926407 EF On-Demand Mild STK3 20 42 C[C@H]1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CCO1 ZINC000880926408 EF On-Demand Mild STK3 20 42 C[C@@H]1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CCO1 ZINC000880926409 EF On-Demand Mild STK3 20 42 C[C@@H]1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CCO1 ZINC000880926410 EF On-Demand Mild STK3 20 42 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](F)C2)C(F)(F)F)c1 ZINC000880926411 DF On-Demand Mild DPP4 21 49 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](F)C2)C(F)(F)F)c1 ZINC000880926412 DF On-Demand Mild DPP4 21 49 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](F)C2)C(F)(F)F)c1 ZINC000880926413 DF On-Demand Mild DPP4 21 49 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](F)C2)C(F)(F)F)c1 ZINC000880926414 DF On-Demand Mild DPP4 21 49 N#Cc1cccc([C@H](NC(=O)N2C[C@H]3C[C@@H](O)CC[C@H]3C2)C(F)(F)F)c1 ZINC000880926505 FF On-Demand Mild RBP4 41 41 N#Cc1cccc([C@H](NC(=O)N2C[C@H]3C[C@H](O)CC[C@H]3C2)C(F)(F)F)c1 ZINC000880926506 FF On-Demand Mild RBP4 41 41 N#Cc1cccc([C@H](NC(=O)N2C[C@@H]3CC[C@@H](O)C[C@H]3C2)C(F)(F)F)c1 ZINC000880926507 FF On-Demand Mild RBP4 41 41 N#Cc1cccc([C@H](NC(=O)N2C[C@@H]3CC[C@H](O)C[C@H]3C2)C(F)(F)F)c1 ZINC000880926508 FF On-Demand Mild RBP4 41 41 CC[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(=O)NC ZINC000880926539 ED On-Demand Mild CTSF 81 35 CC[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(=O)NC ZINC000880926542 ED On-Demand Mild CTSF 81 35 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926551 GI On-Demand Mild CTSF 67 33 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926552 GI On-Demand Mild CTSF 67 33 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@H](C)C1 ZINC000880926556 GH On-Demand Mild CCR5 16 41 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@H](C)C1 ZINC000880926556 GH On-Demand Mild MCHR1 35 43 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H](C)C1 ZINC000880926557 GH On-Demand Mild CCR5 16 41 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H](C)C1 ZINC000880926557 GH On-Demand Mild MCHR1 35 43 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H](C)C1 ZINC000880926559 GH On-Demand Mild CCR5 16 41 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H](C)C1 ZINC000880926559 GH On-Demand Mild MCHR1 35 43 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@H](C)C1 ZINC000880926560 GH On-Demand Mild CCR5 16 41 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@H](C)C1 ZINC000880926560 GH On-Demand Mild MCHR1 35 43 N#Cc1cccc([C@@H](NC(=O)N2CCCOCC2)C(F)(F)F)c1 ZINC000880926590 EF On-Demand Mild CTSS 23 42 N#Cc1cccc([C@H](NC(=O)N2CCCOCC2)C(F)(F)F)c1 ZINC000880926591 EF On-Demand Mild CTSS 23 42 N#Cc1cccc([C@H](NC(=O)NC23C[C@H]4C[C@@H](CC(O)(C4)C2)C3)C(F)(F)F)c1 ZINC000880926645 GH On-Demand Mild EPHX2 23 41 CCc1nnc2n1CCN(C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C2 ZINC000880926648 GF On-Demand Mild P2RX7 18 48 N#Cc1cccc([C@@H](NC(=O)NC23C[C@H]4C[C@@H](CC(O)(C4)C2)C3)C(F)(F)F)c1 ZINC000880926649 GH On-Demand Mild EPHX2 23 41 CCc1nnc2n1CCN(C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C2 ZINC000880926650 GF On-Demand Mild P2RX7 18 48 N#Cc1cccc([C@H](NC(=O)N2CCc3ccc(O)cc3C2)C(F)(F)F)c1 ZINC000880926656 GH On-Demand Mild AKR1C3 16 41 N#Cc1cccc([C@@H](NC(=O)N2CCc3ccc(O)cc3C2)C(F)(F)F)c1 ZINC000880926658 GH On-Demand Mild AKR1C3 16 41 CCCN(CC(C)(C)O)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926665 FG On-Demand Mild CTSF 41 31 CCCN(CC(C)(C)O)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926666 FG On-Demand Mild CTSF 41 31 CC[C@@](C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926678 EF On-Demand Mild CTSF 50 33 CC[C@@](C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926682 EF On-Demand Mild CTSF 50 33 N#Cc1cccc([C@@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926706 DD On-Demand Mild CTSF 75 35 N#Cc1cccc([C@@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926706 DD On-Demand Mild CTSL 38 42 N#Cc1cccc([C@@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926706 DD On-Demand Mild CTSS 28 42 N#Cc1cccc([C@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926707 DD On-Demand Mild CTSF 75 35 N#Cc1cccc([C@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926707 DD On-Demand Mild CTSL 38 42 N#Cc1cccc([C@H](NC(=O)NCC#CCO)C(F)(F)F)c1 ZINC000880926707 DD On-Demand Mild CTSS 28 42 CCC(CC)(CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926731 EG On-Demand Mild CTSF 49 32 CCC(CC)(CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926733 EG On-Demand Mild CTSF 49 32 CNC(=O)[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926815 ED On-Demand Mild CTSF 68 36 CNC(=O)[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926816 ED On-Demand Mild CTSF 68 36 CCC1(O)CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926819 EE On-Demand Mild CTSF 41 32 CCC1(O)CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926820 EE On-Demand Mild CTSF 41 32 N#Cc1cccc([C@@H](NC(=O)N(CCO)CCc2ccccc2)C(F)(F)F)c1 ZINC000880926838 GG On-Demand Mild CTSF 56 32 N#Cc1cccc([C@H](NC(=O)N(CCO)CCc2ccccc2)C(F)(F)F)c1 ZINC000880926839 GG On-Demand Mild CTSF 56 32 N#Cc1cccc([C@@H](NC(=O)NCC[C@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926844 GH On-Demand Mild CTSF 64 32 N#Cc1cccc([C@@H](NC(=O)NCC[C@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926844 GH On-Demand Mild CTSL 18 40 N#Cc1cccc([C@@H](NC(=O)NCC[C@@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926851 GH On-Demand Mild CTSF 64 32 N#Cc1cccc([C@@H](NC(=O)NCC[C@@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926851 GH On-Demand Mild CTSL 18 40 N#Cc1cccc([C@H](NC(=O)NCC[C@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926853 GH On-Demand Mild CTSF 64 32 N#Cc1cccc([C@H](NC(=O)NCC[C@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926853 GH On-Demand Mild CTSL 18 40 N#Cc1cccc([C@H](NC(=O)NCC[C@@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926855 GH On-Demand Mild CTSF 64 32 N#Cc1cccc([C@H](NC(=O)NCC[C@@H](O)c2ccccc2)C(F)(F)F)c1 ZINC000880926855 GH On-Demand Mild CTSL 18 40 COC[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926867 FG On-Demand Mild REN 16 50 COC[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926867 FG On-Demand Mild LGMN 41 32 COC[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926869 FG On-Demand Mild REN 16 50 COC[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926869 FG On-Demand Mild LGMN 41 32 N#Cc1cccc([C@H](NC(=O)N[C@]2(CO)CCc3ccccc32)C(F)(F)F)c1 ZINC000880926880 GG On-Demand Mild CTSF 41 32 N#Cc1cccc([C@@H](NC(=O)N[C@@]2(CO)CCc3ccccc32)C(F)(F)F)c1 ZINC000880926884 GG On-Demand Mild CTSF 41 32 N#Cc1cccc([C@@H](NC(=O)N[C@]2(CO)CCc3ccccc32)C(F)(F)F)c1 ZINC000880926886 GG On-Demand Mild CTSF 41 32 N#Cc1cccc([C@H](NC(=O)N[C@@]2(CO)CCc3ccccc32)C(F)(F)F)c1 ZINC000880926887 GG On-Demand Mild CTSF 41 32 C[C@@H](CCO)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926913 EE On-Demand Mild CTSF 40 35 C[C@@H](CCO)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926915 EE On-Demand Mild CTSF 40 35 C[C@H](CCO)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926917 EE On-Demand Mild CTSF 40 35 C[C@H](CCO)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926918 EE On-Demand Mild CTSF 40 35 CN(CCO)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926919 DD On-Demand Mild CTSF 49 32 CN(CCO)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926920 DD On-Demand Mild CTSF 49 32 N#Cc1cccc([C@@H](NC(=O)N[C@@H](CCO)c2ccccc2F)C(F)(F)F)c1 ZINC000880926929 GH On-Demand Mild CTSF 43 34 N#Cc1cccc([C@@H](NC(=O)N[C@H](CCO)c2ccccc2F)C(F)(F)F)c1 ZINC000880926934 GH On-Demand Mild CTSF 43 34 N#Cc1cccc([C@H](NC(=O)N[C@@H](CCO)c2ccccc2F)C(F)(F)F)c1 ZINC000880926935 GH On-Demand Mild CTSF 43 34 N#Cc1cccc([C@H](NC(=O)N[C@H](CCO)c2ccccc2F)C(F)(F)F)c1 ZINC000880926937 GH On-Demand Mild CTSF 43 34 CCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926966 DG On-Demand Mild CTSF 53 34 CCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926966 DG On-Demand Mild CTSL 17 44 CCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926968 DG On-Demand Mild CTSF 53 34 CCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880926968 DG On-Demand Mild CTSL 17 44 CN(C)[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926972 EF On-Demand Mild MCHR1 47 40 CN(C)[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926972 EF On-Demand Mild PKNB 17 43 CN(C[C@H]1CCCN1C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926975 FF On-Demand Mild CTSF 41 30 CN(C[C@H]1CCCN1C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926975 FF On-Demand Mild CHRNA10 66 47 CN(C)[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926976 EF On-Demand Mild MCHR1 47 40 CN(C)[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880926976 EF On-Demand Mild PKNB 17 43 CN(C[C@@H]1CCCN1C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926977 FF On-Demand Mild CTSF 41 30 CN(C[C@@H]1CCCN1C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926977 FF On-Demand Mild CHRNA10 66 47 N#Cc1cccc([C@H](NC(=O)N2CCc3cncnc3C2)C(F)(F)F)c1 ZINC000880926978 FF On-Demand Mild MAPK1 54 38 CN(C[C@H]1CCCN1C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926979 FF On-Demand Mild CTSF 41 30 CN(C[C@H]1CCCN1C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926979 FF On-Demand Mild CHRNA10 66 47 N#Cc1cccc([C@@H](NC(=O)N2CCc3cncnc3C2)C(F)(F)F)c1 ZINC000880926980 FF On-Demand Mild MAPK1 54 38 CN(C[C@@H]1CCCN1C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926981 FF On-Demand Mild CTSF 41 30 CN(C[C@@H]1CCCN1C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880926981 FF On-Demand Mild CHRNA10 66 47 C[C@@](CO)(NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C1CC1 ZINC000880926984 EF On-Demand Mild CTSF 46 31 C[C@@](CO)(NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C1CC1 ZINC000880926988 EF On-Demand Mild CTSF 46 31 N#Cc1cccc([C@@H](NC(=O)NCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926994 EE On-Demand Mild CTSF 56 33 N#Cc1cccc([C@@H](NC(=O)NCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926994 EE On-Demand Mild MCHR1 18 41 N#Cc1cccc([C@H](NC(=O)NCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926996 EE On-Demand Mild CTSF 56 33 N#Cc1cccc([C@H](NC(=O)NCC2(CO)CC2)C(F)(F)F)c1 ZINC000880926996 EE On-Demand Mild MCHR1 18 41 N#Cc1cccc([C@H](NC(=O)NCC(Cl)Cl)C(F)(F)F)c1 ZINC000880927001 EG On-Demand Reactive CTSF 42 33 N#Cc1cccc([C@H](NC(=O)NCC(Cl)Cl)C(F)(F)F)c1 ZINC000880927001 EG On-Demand Reactive MCHR1 17 41 N#Cc1cccc([C@@H](NC(=O)NCC(Cl)Cl)C(F)(F)F)c1 ZINC000880927013 EG On-Demand Reactive CTSF 42 33 N#Cc1cccc([C@@H](NC(=O)NCC(Cl)Cl)C(F)(F)F)c1 ZINC000880927013 EG On-Demand Reactive MCHR1 17 41 CC(C)[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927024 EH On-Demand Mild DPP4 16 40 CC(C)[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927024 EH On-Demand Mild LGMN 55 35 CC(C)[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927028 EH On-Demand Mild DPP4 16 40 CC(C)[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927028 EH On-Demand Mild LGMN 55 35 C#C[C@](C)(CC)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927071 DG On-Demand Mild CTSF 46 32 C#C[C@@](C)(CC)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927072 DG On-Demand Mild CTSF 46 32 C#C[C@](C)(CC)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927074 DG On-Demand Mild CTSF 46 32 C#C[C@@](C)(CC)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927076 DG On-Demand Mild CTSF 46 32 N#Cc1cccc([C@H](NC(=O)N[C@@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927077 GE On-Demand Mild CCR3 25 43 N#Cc1cccc([C@H](NC(=O)N[C@@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927077 GE On-Demand Mild MCHR1 29 40 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927078 GE On-Demand Mild CCR3 25 43 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927078 GE On-Demand Mild MCHR1 29 40 N#Cc1cccc([C@@H](NC(=O)N[C@@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927079 GE On-Demand Mild CCR3 25 43 N#Cc1cccc([C@@H](NC(=O)N[C@@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927079 GE On-Demand Mild MCHR1 29 40 N#Cc1cccc([C@@H](NC(=O)N[C@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927080 GE On-Demand Mild CCR3 25 43 N#Cc1cccc([C@@H](NC(=O)N[C@H]2CCCN(CCCO)C2)C(F)(F)F)c1 ZINC000880927080 GE On-Demand Mild MCHR1 29 40 CC(=O)N[C@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927108 FE On-Demand Mild MCHR1 22 43 CC(=O)N[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927109 FE On-Demand Mild MCHR1 22 43 CC(=O)N[C@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927111 FE On-Demand Mild MCHR1 22 43 CC(=O)N[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927112 FE On-Demand Mild MCHR1 22 43 N#Cc1cccc([C@@H](NC(=O)N[C@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927114 GG On-Demand Mild CTSF 78 37 N#Cc1cccc([C@@H](NC(=O)N[C@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927114 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@@H](NC(=O)N[C@@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927118 GG On-Demand Mild CTSF 78 37 N#Cc1cccc([C@@H](NC(=O)N[C@@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927118 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@H](NC(=O)N[C@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927122 GG On-Demand Mild CTSF 78 37 N#Cc1cccc([C@H](NC(=O)N[C@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927122 GG On-Demand Mild CTRB_BOVIN 45 31 CC(C)(C)C1CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927124 EH On-Demand Mild CTSF 45 31 CC(C)(C)C1CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927125 EH On-Demand Mild CTSF 45 31 N#Cc1cccc([C@H](NC(=O)N[C@@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927126 GG On-Demand Mild CTSF 78 37 N#Cc1cccc([C@H](NC(=O)N[C@@H](CO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880927126 GG On-Demand Mild CTRB_BOVIN 45 31 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CN2CCOCC2)C(F)(F)F)c1 ZINC000880927127 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CN2CCOCC2)C(F)(F)F)c1 ZINC000880927128 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CCC(OC3CCC3)CC2)C(F)(F)F)c1 ZINC000880927189 GH On-Demand Mild EPHX2 15 43 N#Cc1cccc([C@@H](NC(=O)N2CCC(OC3CCC3)CC2)C(F)(F)F)c1 ZINC000880927191 GH On-Demand Mild EPHX2 15 43 C[C@H]([C@@H](C)S(C)(=O)=O)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927196 GF On-Demand Mild CTSF 62 39 C[C@H]([C@@H](C)S(C)(=O)=O)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927200 GF On-Demand Mild CTSF 62 39 C[C@@H]([C@@H](C)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)S(C)(=O)=O ZINC000880927202 GF On-Demand Mild CTSF 62 39 C[C@@H]([C@@H](C)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)S(C)(=O)=O ZINC000880927205 GF On-Demand Mild CTSF 62 39 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)C2CCC2)C(F)(F)F)c1 ZINC000880927207 EF On-Demand Mild MCHR1 17 41 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)C2CCC2)C(F)(F)F)c1 ZINC000880927208 EF On-Demand Mild MCHR1 17 41 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)C2CCC2)C(F)(F)F)c1 ZINC000880927209 EF On-Demand Mild MCHR1 17 41 C=CC[C@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927210 DG On-Demand Mild CTSF 76 37 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)C2CCC2)C(F)(F)F)c1 ZINC000880927211 EF On-Demand Mild MCHR1 17 41 C=CC[C@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927213 DG On-Demand Mild CTSF 76 37 C[C@H](CO)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927215 DE On-Demand Mild CTSF 43 34 C[C@H](CO)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927216 DE On-Demand Mild CTSF 43 34 C=CC[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927217 DG On-Demand Mild CTSF 76 37 CO[C@@](C)(CO)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927218 ED On-Demand Mild CTSF 42 32 CO[C@@](C)(CO)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927221 ED On-Demand Mild CTSF 42 32 C=CC[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927222 DG On-Demand Mild CTSF 76 37 COCCN(CCN(C)C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927234 FE On-Demand Mild UTS2 41 31 COCCN(CCN(C)C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927237 FE On-Demand Mild UTS2 41 31 CNC(=O)CN1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927251 GD On-Demand Mild CTSF 66 33 CNC(=O)CN1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927252 GD On-Demand Mild CTSF 66 33 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927255 FE On-Demand Mild CTSF 72 35 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927255 FE On-Demand Mild CTSL 25 40 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927255 FE On-Demand Mild CTSS 18 40 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927256 FE On-Demand Mild CTSF 72 35 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927256 FE On-Demand Mild CTSL 25 40 CNC(=O)[C@@H](C)CN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927256 FE On-Demand Mild CTSS 18 40 N#Cc1cccc([C@H](NC(=O)NCCC2(CO)CCC2)C(F)(F)F)c1 ZINC000880927269 FG On-Demand Mild CTSF 55 33 N#Cc1cccc([C@@H](NC(=O)NCCC2(CO)CCC2)C(F)(F)F)c1 ZINC000880927270 FG On-Demand Mild CTSF 55 33 CC[C@@](C)(NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)c1nccs1 ZINC000880927290 GI On-Demand Mild CTSF 41 32 CC[C@@](C)(NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)c1nccs1 ZINC000880927291 GI On-Demand Mild CTSF 41 32 CCNC(=O)C(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927300 FE On-Demand Mild CTSF 42 32 CCNC(=O)C(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927301 FE On-Demand Mild CTSF 42 32 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)Cc2cccc(F)c2)C(F)(F)F)c1 ZINC000880927311 GG On-Demand Mild CTSF 56 33 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)Cc2cccc(F)c2)C(F)(F)F)c1 ZINC000880927312 GG On-Demand Mild CTSF 56 33 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)Cc2cccc(F)c2)C(F)(F)F)c1 ZINC000880927314 GG On-Demand Mild CTSF 56 33 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)Cc2cccc(F)c2)C(F)(F)F)c1 ZINC000880927315 GG On-Demand Mild CTSF 56 33 COCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927333 EF On-Demand Mild CTSF 67 35 COCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927333 EF On-Demand Mild CTSL 19 40 COCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927335 EF On-Demand Mild CTSF 67 35 COCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927335 EF On-Demand Mild CTSL 19 40 CCN(CC(C)(C)O)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927344 EF On-Demand Mild CTSF 46 32 CCN(CC(C)(C)O)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927345 EF On-Demand Mild CTSF 46 32 CN(CCC#N)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927409 DF On-Demand Mild CTSF 65 34 CN(CCC#N)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927410 DF On-Demand Mild CTSF 65 34 CC[C@H](C[C@H](C)CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927418 FG On-Demand Mild CTSF 49 35 CC[C@H](C[C@H](C)CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927420 FG On-Demand Mild CTSF 49 35 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880927433 DD On-Demand Mild MCHR1 26 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](O)C2)C(F)(F)F)c1 ZINC000880927434 DD On-Demand Mild MCHR1 26 41 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927441 FG On-Demand Mild CCR3 16 43 N#Cc1cccc([C@H](NC(=O)N[C@@H]2CCCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927442 FG On-Demand Mild CCR3 16 43 N#Cc1cccc([C@H](NC(=O)N[C@H]2CCCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927443 FG On-Demand Mild CCR3 16 43 N#Cc1cccc([C@H](NC(=O)N[C@@H]2CCCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927444 FG On-Demand Mild CCR3 16 43 CC(C)(C)CN(CCO)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927447 FG On-Demand Mild CTSF 42 31 CC(C)(C)CN(CCO)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927448 FG On-Demand Mild CTSF 42 31 C#CC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927453 DF On-Demand Mild CTSF 42 32 C#CC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927454 DF On-Demand Mild CTSF 42 32 N#Cc1cccc([C@@H](NC(=O)NCCCCN2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927473 GF On-Demand Mild CCR3 32 43 N#Cc1cccc([C@@H](NC(=O)NCCCCN2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927473 GF On-Demand Mild MCHR1 24 41 N#Cc1cccc([C@@H](NC(=O)NCCCCN2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927474 GF On-Demand Mild CCR3 32 43 N#Cc1cccc([C@@H](NC(=O)NCCCCN2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927474 GF On-Demand Mild MCHR1 24 41 N#Cc1cccc([C@H](NC(=O)NCCCCN2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927475 GF On-Demand Mild CCR3 32 43 N#Cc1cccc([C@H](NC(=O)NCCCCN2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927475 GF On-Demand Mild MCHR1 24 41 N#Cc1cccc([C@H](NC(=O)NCCCCN2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927476 GF On-Demand Mild CCR3 32 43 N#Cc1cccc([C@H](NC(=O)NCCCCN2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927476 GF On-Demand Mild MCHR1 24 41 CS(=O)(=O)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927477 GE On-Demand Mild CTSF 58 34 CS(=O)(=O)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880927478 GE On-Demand Mild CTSF 58 34 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CCCO)C(F)(F)F)c1 ZINC000880927479 FG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CCCO)C(F)(F)F)c1 ZINC000880927480 FG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CCCO)C(F)(F)F)c1 ZINC000880927481 FG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CCCO)C(F)(F)F)c1 ZINC000880927482 FG On-Demand Mild LGMN 48 33 COc1ccccc1[C@@H](O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927499 GG On-Demand Mild CTSF 51 31 COc1ccccc1[C@@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927500 GG On-Demand Mild CTSF 51 31 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@@H]2c2ncc[nH]2)C(F)(F)F)c1 ZINC000880927520 GH On-Demand Mild CPT1A 46 44 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@H]2c2ncc[nH]2)C(F)(F)F)c1 ZINC000880927521 GH On-Demand Mild CPT1A 46 44 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@@H]2c2ncc[nH]2)C(F)(F)F)c1 ZINC000880927522 GH On-Demand Mild CPT1A 46 44 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@H]2c2ncc[nH]2)C(F)(F)F)c1 ZINC000880927523 GH On-Demand Mild CPT1A 46 44 CC[C@@](C)(CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927531 EF On-Demand Mild CTSF 50 33 CC[C@@](C)(CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927532 EF On-Demand Mild CTSF 50 33 N#Cc1cccc([C@H](NC(=O)N2CCN3CCCC[C@@H]3C2)C(F)(F)F)c1 ZINC000880927536 FG On-Demand Mild MCHR1 21 41 N#Cc1cccc([C@H](NC(=O)N2CCN3CCCC[C@H]3C2)C(F)(F)F)c1 ZINC000880927537 FG On-Demand Mild MCHR1 21 41 N#Cc1cccc([C@@H](NC(=O)N2CCN3CCCC[C@@H]3C2)C(F)(F)F)c1 ZINC000880927538 FG On-Demand Mild MCHR1 21 41 N#Cc1cccc([C@@H](NC(=O)N2CCN3CCCC[C@H]3C2)C(F)(F)F)c1 ZINC000880927539 FG On-Demand Mild MCHR1 21 41 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CCOCC3)CC2)C(F)(F)F)c1 ZINC000880927540 GF On-Demand Mild MAPK1 30 42 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CCOCC3)CC2)C(F)(F)F)c1 ZINC000880927540 GF On-Demand Mild MCHR1 17 40 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CCOCC3)CC2)C(F)(F)F)c1 ZINC000880927541 GF On-Demand Mild MAPK1 30 42 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CCOCC3)CC2)C(F)(F)F)c1 ZINC000880927541 GF On-Demand Mild MCHR1 17 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927554 EE On-Demand Mild DPP4 23 42 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927554 EE On-Demand Mild LGMN 58 35 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927555 EE On-Demand Mild DPP4 23 42 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CO)C(F)(F)F)c1 ZINC000880927555 EE On-Demand Mild LGMN 58 35 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927556 EE On-Demand Mild DPP4 23 42 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927556 EE On-Demand Mild LGMN 58 35 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927557 EE On-Demand Mild DPP4 23 42 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CO)C(F)(F)F)c1 ZINC000880927557 EE On-Demand Mild LGMN 58 35 CSC(C)(C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927574 EH On-Demand Mild CTSF 50 33 CSC(C)(C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927575 EH On-Demand Mild CTSF 50 33 CNC(=O)[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927578 FE On-Demand Mild F2 40 37 CNC(=O)[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927578 FE On-Demand Mild CELA1 43 33 CNC(=O)[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927578 FE On-Demand Mild ELANE 52 36 CNC(=O)[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927578 FE On-Demand Mild LGMN 81 41 CNC(=O)[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927578 FE On-Demand Mild WNT3 41 32 CNC(=O)[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927579 FE On-Demand Mild F2 40 37 CNC(=O)[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927579 FE On-Demand Mild CELA1 43 33 CNC(=O)[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927579 FE On-Demand Mild ELANE 52 36 CNC(=O)[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927579 FE On-Demand Mild LGMN 81 41 CNC(=O)[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927579 FE On-Demand Mild WNT3 41 32 CCOC(=O)[C@H](C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927582 FF On-Demand Mild CTSF 57 33 CCOC(=O)[C@H](C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927582 FF On-Demand Mild CTSK 26 40 CCOC(=O)[C@H](C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927582 FF On-Demand Mild CTSL 25 40 CCOC(=O)[C@H](C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927582 FF On-Demand Mild CTSS 19 40 CCOC(=O)[C@H](C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927583 FF On-Demand Mild CTSF 57 33 CCOC(=O)[C@H](C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927583 FF On-Demand Mild CTSK 26 40 CCOC(=O)[C@H](C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927583 FF On-Demand Mild CTSL 25 40 CCOC(=O)[C@H](C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927583 FF On-Demand Mild CTSS 19 40 CCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927762 CF On-Demand Mild CTSF 69 34 CCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927765 CF On-Demand Mild CTSF 69 34 CN(CCN1CCOCC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927768 FE On-Demand Mild CASR 60 54 CN(CCN1CCOCC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927768 FE On-Demand Mild MCHR1 31 43 CN(CCN1CCOCC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927774 FE On-Demand Mild CASR 60 54 CN(CCN1CCOCC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927774 FE On-Demand Mild MCHR1 31 43 CCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CCC1 ZINC000880927795 EH On-Demand Mild CTSL 15 43 CCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CCC1 ZINC000880927799 EH On-Demand Mild CTSL 15 43 CC[C@@H](O)CCNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927830 EF On-Demand Mild CTSF 42 34 CC[C@@H](O)CCNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927832 EF On-Demand Mild CTSF 42 34 CC[C@H](O)CCNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927835 EF On-Demand Mild CTSF 42 34 CC[C@H](O)CCNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927837 EF On-Demand Mild CTSF 42 34 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927862 GF On-Demand Mild CTSF 59 35 N#Cc1cccc([C@H](NC(=O)N2CCC3(CCO3)CC2)C(F)(F)F)c1 ZINC000880927863 FG On-Demand Mild EPHX2 15 43 CCS(=O)(=O)C[C@H](C)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927864 GF On-Demand Mild CTSF 59 35 N#Cc1cccc([C@@H](NC(=O)N2CCC3(CCO3)CC2)C(F)(F)F)c1 ZINC000880927865 FG On-Demand Mild EPHX2 15 43 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927866 GF On-Demand Mild CTSF 59 35 CCS(=O)(=O)C[C@H](C)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927869 GF On-Demand Mild CTSF 59 35 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927889 GG On-Demand Mild CTSF 65 33 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927889 GG On-Demand Mild CTSL 18 40 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927889 GG On-Demand Mild MCHR1 15 43 N#Cc1cccc([C@@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927891 GG On-Demand Mild CTSF 65 33 N#Cc1cccc([C@@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927891 GG On-Demand Mild CTSL 18 40 N#Cc1cccc([C@@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927891 GG On-Demand Mild MCHR1 15 43 N#Cc1cccc([C@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927893 GG On-Demand Mild CTSF 65 33 N#Cc1cccc([C@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927893 GG On-Demand Mild CTSL 18 40 N#Cc1cccc([C@H](NC(=O)NC[C@@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927893 GG On-Demand Mild MCHR1 15 43 N#Cc1cccc([C@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927895 GG On-Demand Mild CTSF 65 33 N#Cc1cccc([C@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927895 GG On-Demand Mild CTSL 18 40 N#Cc1cccc([C@H](NC(=O)NC[C@H](CO)c2ccccc2)C(F)(F)F)c1 ZINC000880927895 GG On-Demand Mild MCHR1 15 43 C[C@H](CS(C)(=O)=O)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927923 GE On-Demand Mild CTSF 64 37 C[C@H](CS(C)(=O)=O)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927923 GE On-Demand Mild CTSL 19 44 C[C@H](CS(C)(=O)=O)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927925 GE On-Demand Mild CTSF 64 37 C[C@H](CS(C)(=O)=O)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927925 GE On-Demand Mild CTSL 19 44 COC[C@@H]1CCCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927964 FH On-Demand Mild REN 17 49 COC[C@@H]1CCCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880927967 FH On-Demand Mild REN 17 49 N#Cc1cccc([C@H](NC(=O)N2CCN(C(=O)C3CC3)CC2)C(F)(F)F)c1 ZINC000880927974 GE On-Demand Mild MCHR1 17 41 N#Cc1cccc([C@@H](NC(=O)N2CCN(C(=O)C3CC3)CC2)C(F)(F)F)c1 ZINC000880927975 GE On-Demand Mild MCHR1 17 41 COCCN(Cc1cccnc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927988 GG On-Demand Mild PTGES 24 47 COCCN(Cc1cccnc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927989 GG On-Demand Mild PTGES 24 47 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880927990 FG On-Demand Mild L3MBTL3 83 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880927991 FG On-Demand Mild L3MBTL3 83 40 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880927992 FG On-Demand Mild L3MBTL3 83 40 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880927993 FG On-Demand Mild L3MBTL3 83 40 COCC[C@@](C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927996 FE On-Demand Mild CTSF 41 31 COCC[C@](C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927997 FE On-Demand Mild CTSF 41 31 COCC[C@@](C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927998 FE On-Demand Mild CTSF 41 31 COCC[C@](C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880927999 FE On-Demand Mild CTSF 41 31 CC[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928038 EH On-Demand Mild DPP4 28 41 CC[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928038 EH On-Demand Mild LGMN 61 35 CC[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928038 EH On-Demand Mild CHRNA10 19 40 CC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928039 EH On-Demand Mild DPP4 28 41 CC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928039 EH On-Demand Mild LGMN 61 35 CC[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928039 EH On-Demand Mild CHRNA10 19 40 CC[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928040 EH On-Demand Mild DPP4 28 41 CC[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928040 EH On-Demand Mild LGMN 61 35 CC[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928040 EH On-Demand Mild CHRNA10 19 40 CC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928041 EH On-Demand Mild DPP4 28 41 CC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928041 EH On-Demand Mild LGMN 61 35 CC[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928041 EH On-Demand Mild CHRNA10 19 40 CCc1nc([C@H]2CCCN2C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)no1 ZINC000880928043 GH On-Demand Mild CPT1A 52 47 CCc1nc([C@H]2CCCN2C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)no1 ZINC000880928044 GH On-Demand Mild CPT1A 52 47 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CC3)CC2)C(F)(F)F)c1 ZINC000880928050 FF On-Demand Mild HRH3 18 41 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CC3)CC2)C(F)(F)F)c1 ZINC000880928050 FF On-Demand Mild MCHR1 21 40 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CC3)CC2)C(F)(F)F)c1 ZINC000880928051 FF On-Demand Mild HRH3 18 41 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CC3)CC2)C(F)(F)F)c1 ZINC000880928051 FF On-Demand Mild MCHR1 21 40 C[S@@](=O)CCCNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928194 EE On-Demand Mild CTSF 57 32 C[S@@](=O)CCCNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928194 EE On-Demand Mild CTSL 18 41 C[S@@](=O)CCCNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928196 EE On-Demand Mild CTSF 57 32 C[S@@](=O)CCCNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928196 EE On-Demand Mild CTSL 18 41 Cc1ccccc1[C@@H](O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928204 GH On-Demand Mild CTSF 65 33 Cc1ccccc1[C@@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928206 GH On-Demand Mild CTSF 65 33 Cc1ccccc1[C@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928207 GH On-Demand Mild CTSF 65 33 CCC1(O)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928224 FG On-Demand Mild S1PR2 25 41 CCC1(O)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928225 FG On-Demand Mild S1PR2 25 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](N3CCCCC3)C2)C(F)(F)F)c1 ZINC000880928226 GG On-Demand Mild L3MBTL3 81 40 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](N3CCCCC3)C2)C(F)(F)F)c1 ZINC000880928227 GG On-Demand Mild L3MBTL3 81 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](N3CCCCC3)C2)C(F)(F)F)c1 ZINC000880928228 GG On-Demand Mild L3MBTL3 81 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](N3CCCCC3)C2)C(F)(F)F)c1 ZINC000880928229 GG On-Demand Mild L3MBTL3 81 40 CC[C@@](C)(CCO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928235 EG On-Demand Mild CTSF 47 32 CC[C@@](C)(CCO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928237 EG On-Demand Mild CTSF 47 32 N#Cc1cccc([C@H](NC(=O)N[C@H]2c3ccccc3C[C@H]2O)C(F)(F)F)c1 ZINC000880928238 GG On-Demand Mild PLM2_PLAFA 47 38 N#Cc1cccc([C@@H](NC(=O)N[C@H]2c3ccccc3C[C@H]2O)C(F)(F)F)c1 ZINC000880928239 GG On-Demand Mild PLM2_PLAFA 47 38 CNC(=O)CCCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928260 FE On-Demand Mild CTSF 45 32 CNC(=O)CCCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928261 FE On-Demand Mild CTSF 45 32 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C[C@H]1C ZINC000880928276 GH On-Demand Mild MCHR1 35 40 CCN1CC[C@H](N(C)C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C[C@@H]1C ZINC000880928277 GH On-Demand Mild MCHR1 35 40 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C[C@@H]1C ZINC000880928278 GH On-Demand Mild MCHR1 35 40 CCN1CC[C@H](N(C)C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C[C@H]1C ZINC000880928279 GH On-Demand Mild MCHR1 35 40 N#Cc1cccc([C@@H](NC(=O)N2CCC(C(F)(F)F)CC2)C(F)(F)F)c1 ZINC000880928288 GI On-Demand Mild MCHR1 20 40 N#Cc1cccc([C@H](NC(=O)N2CCC(C(F)(F)F)CC2)C(F)(F)F)c1 ZINC000880928289 GI On-Demand Mild MCHR1 20 40 CC(C)(C)[C@@H](O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928326 EF On-Demand Mild CTSF 59 36 CC(C)(C)[C@@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928327 EF On-Demand Mild CTSF 59 36 Cc1noc(C2CCN(C(=O)N[C@@H](c3cccc(C#N)c3)C(F)(F)F)CC2)n1 ZINC000880928334 GG On-Demand Mild SMO 41 45 Cc1noc(C2CCN(C(=O)N[C@@H](c3cccc(C#N)c3)C(F)(F)F)CC2)n1 ZINC000880928334 GG On-Demand Mild ETHR 72 42 Cc1noc(C2CCN(C(=O)N[C@H](c3cccc(C#N)c3)C(F)(F)F)CC2)n1 ZINC000880928335 GG On-Demand Mild SMO 41 45 Cc1noc(C2CCN(C(=O)N[C@H](c3cccc(C#N)c3)C(F)(F)F)CC2)n1 ZINC000880928335 GG On-Demand Mild ETHR 72 42 N#Cc1cccc([C@H](NC(=O)N2CCC(c3nccs3)CC2)C(F)(F)F)c1 ZINC000880928336 GI On-Demand Mild ETHR 42 35 N#Cc1cccc([C@@H](NC(=O)N2CCC(c3nccs3)CC2)C(F)(F)F)c1 ZINC000880928337 GI On-Demand Mild ETHR 42 35 N#Cc1cccc([C@H](NC(=O)N(Cc2cccnc2)C2CC2)C(F)(F)F)c1 ZINC000880928338 FH On-Demand Mild PTGES 21 44 N#Cc1cccc([C@@H](NC(=O)N(Cc2cccnc2)C2CC2)C(F)(F)F)c1 ZINC000880928339 FH On-Demand Mild PTGES 21 44 CCOC(=O)N1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928360 GG On-Demand Mild P2RY12 152 44 CCOC(=O)N1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928360 GG On-Demand Mild MCHR1 18 42 CCOC(=O)N1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928361 GG On-Demand Mild P2RY12 152 44 CCOC(=O)N1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928361 GG On-Demand Mild MCHR1 18 42 N#Cc1cccc([C@H](NC(=O)N2CCc3ccccc3[C@H]2CO)C(F)(F)F)c1 ZINC000880928366 GG On-Demand Mild TRPM8 32 49 N#Cc1cccc([C@@H](NC(=O)N2CCc3ccccc3[C@H]2CO)C(F)(F)F)c1 ZINC000880928367 GG On-Demand Mild TRPM8 32 49 N#Cc1cccc([C@H](NC(=O)N2CCc3ccccc3[C@@H]2CO)C(F)(F)F)c1 ZINC000880928368 GG On-Demand Mild TRPM8 32 49 N#Cc1cccc([C@@H](NC(=O)N2CCc3ccccc3[C@@H]2CO)C(F)(F)F)c1 ZINC000880928369 GG On-Demand Mild TRPM8 32 49 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](CN3CCCC3)C2)C(F)(F)F)c1 ZINC000880928384 GG On-Demand Mild MCHR1 41 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](CN3CCCC3)C2)C(F)(F)F)c1 ZINC000880928385 GG On-Demand Mild MCHR1 41 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](CN3CCCC3)C2)C(F)(F)F)c1 ZINC000880928386 GG On-Demand Mild MCHR1 41 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](CN3CCCC3)C2)C(F)(F)F)c1 ZINC000880928387 GG On-Demand Mild MCHR1 41 41 CCCNC(=O)[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928446 GG On-Demand Mild GPBAR1 32 42 CCCNC(=O)[C@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928447 GG On-Demand Mild GPBAR1 32 42 CCCNC(=O)[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928448 GG On-Demand Mild GPBAR1 32 42 CCCNC(=O)[C@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928449 GG On-Demand Mild GPBAR1 32 42 C=CC1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928450 EH On-Demand Mild MCHR1 22 41 C=CC1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928451 EH On-Demand Mild MCHR1 22 41 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CCC3)CC2)C(F)(F)F)c1 ZINC000880928460 FG On-Demand Mild HRH3 20 44 N#Cc1cccc([C@H](NC(=O)N2CCN(C3CCC3)CC2)C(F)(F)F)c1 ZINC000880928460 FG On-Demand Mild MCHR1 22 43 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CCC3)CC2)C(F)(F)F)c1 ZINC000880928461 FG On-Demand Mild HRH3 20 44 N#Cc1cccc([C@@H](NC(=O)N2CCN(C3CCC3)CC2)C(F)(F)F)c1 ZINC000880928461 FG On-Demand Mild MCHR1 22 43 CN(CC(C)(C)O)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928485 EF On-Demand Mild CTSF 50 33 CN(CC(C)(C)O)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928486 EF On-Demand Mild CTSF 50 33 N#Cc1cccc([C@H](NC(=O)N2CCN(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880928491 GG On-Demand Mild DRD4 17 45 N#Cc1cccc([C@H](NC(=O)N2CCN(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880928491 GG On-Demand Mild P2RY12 15 41 N#Cc1cccc([C@@H](NC(=O)N2CCN(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880928493 GG On-Demand Mild DRD4 17 45 N#Cc1cccc([C@@H](NC(=O)N2CCN(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880928493 GG On-Demand Mild P2RY12 15 41 N#Cc1cccc([C@@H](NC(=O)N(CCO)C2CC2)C(F)(F)F)c1 ZINC000880928499 EE On-Demand Mild MCHR1 33 40 N#Cc1cccc([C@H](NC(=O)N(CCO)C2CC2)C(F)(F)F)c1 ZINC000880928502 EE On-Demand Mild MCHR1 33 40 N#Cc1cccc([C@@H](NC(=O)NC2(CO)CC2)C(F)(F)F)c1 ZINC000880928512 DD On-Demand Mild CTSF 56 33 N#Cc1cccc([C@@H](NC(=O)NC2(CO)CC2)C(F)(F)F)c1 ZINC000880928512 DD On-Demand Mild CTSL 18 41 N#Cc1cccc([C@H](NC(=O)NC2(CO)CC2)C(F)(F)F)c1 ZINC000880928513 DD On-Demand Mild CTSF 56 33 N#Cc1cccc([C@H](NC(=O)NC2(CO)CC2)C(F)(F)F)c1 ZINC000880928513 DD On-Demand Mild CTSL 18 41 COc1cccc([C@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)c1 ZINC000880928530 GG On-Demand Mild CTSF 41 32 N#Cc1cccc([C@@H](NC(=O)NC2(CO)CCC2)C(F)(F)F)c1 ZINC000880928535 EE On-Demand Mild CTSF 41 32 N#Cc1cccc([C@H](NC(=O)NC2(CO)CCC2)C(F)(F)F)c1 ZINC000880928536 EE On-Demand Mild CTSF 41 32 CCOCCN1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928547 GF On-Demand Mild P2RY12 16 40 CCOCCN1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928548 GF On-Demand Mild P2RY12 16 40 N#Cc1cccc([C@H](NC(=O)N2CCn3c(nnc3C3CC3)C2)C(F)(F)F)c1 ZINC000880928549 GF On-Demand Mild P2RX7 17 48 N#Cc1cccc([C@@H](NC(=O)N2CCn3c(nnc3C3CC3)C2)C(F)(F)F)c1 ZINC000880928550 GF On-Demand Mild P2RX7 17 48 Cc1ccccc1[C@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928553 GH On-Demand Mild CTSF 61 33 Cc1ccccc1[C@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928553 GH On-Demand Mild CTSA 54 34 Cc1ccccc1[C@@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928554 GH On-Demand Mild CTSF 61 33 Cc1ccccc1[C@@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928554 GH On-Demand Mild CTSA 54 34 Cc1ccccc1[C@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928555 GH On-Demand Mild CTSF 61 33 Cc1ccccc1[C@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928555 GH On-Demand Mild CTSA 54 34 Cc1ccccc1[C@@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928556 GH On-Demand Mild CTSF 61 33 Cc1ccccc1[C@@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928556 GH On-Demand Mild CTSA 54 34 C[C@H](O)CN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928634 DE On-Demand Mild CTSF 51 36 C[C@H](O)CN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928635 DE On-Demand Mild CTSF 51 36 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](Oc3ccccn3)C2)C(F)(F)F)c1 ZINC000880928643 GG On-Demand Mild HCRTR2 16 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](Oc3ccccn3)C2)C(F)(F)F)c1 ZINC000880928644 GG On-Demand Mild HCRTR2 16 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](Oc3ccccn3)C2)C(F)(F)F)c1 ZINC000880928645 GG On-Demand Mild HCRTR2 16 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](Oc3ccccn3)C2)C(F)(F)F)c1 ZINC000880928646 GG On-Demand Mild HCRTR2 16 41 COC(=O)[C@@H]1CC12CCN(C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)CC2 ZINC000880928658 GG On-Demand Mild CACNA1H 42 34 COC(=O)[C@@H]1CC12CCN(C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)CC2 ZINC000880928660 GG On-Demand Mild CACNA1H 42 34 N#Cc1cccc([C@H](NC(=O)NCC2(O)Cc3ccccc3C2)C(F)(F)F)c1 ZINC000880928671 GF On-Demand Mild CTSF 72 34 N#Cc1cccc([C@@H](NC(=O)NCC2(O)Cc3ccccc3C2)C(F)(F)F)c1 ZINC000880928672 GF On-Demand Mild CTSF 72 34 CC(C)(C)OC(=O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928679 FF On-Demand Mild CTSF 54 33 CC(C)(C)OC(=O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928680 FF On-Demand Mild CTSF 54 33 N#Cc1cccc([C@@H](NC(=O)NC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880928685 EF On-Demand Mild CTSF 41 32 N#Cc1cccc([C@H](NC(=O)NC2(CO)CCCC2)C(F)(F)F)c1 ZINC000880928686 EF On-Demand Mild CTSF 41 32 C[C@H](O)CN(Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928687 GH On-Demand Mild CTSF 65 36 C[C@H](O)CN(Cc1ccccc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928687 GH On-Demand Mild PTGES 32 49 C[C@H](O)CN(Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928689 GH On-Demand Mild CTSF 65 36 C[C@H](O)CN(Cc1ccccc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928689 GH On-Demand Mild PTGES 32 49 N#Cc1cccc([C@H](NC(=O)N2CCN3CCC[C@@H]3C2)C(F)(F)F)c1 ZINC000880928697 FF On-Demand Mild MCHR1 21 40 N#Cc1cccc([C@H](NC(=O)N2CCN3CCC[C@H]3C2)C(F)(F)F)c1 ZINC000880928698 FF On-Demand Mild MCHR1 21 40 N#Cc1cccc([C@@H](NC(=O)N2CCN3CCC[C@@H]3C2)C(F)(F)F)c1 ZINC000880928699 FF On-Demand Mild MCHR1 21 40 N#Cc1cccc([C@@H](NC(=O)N2CCN3CCC[C@H]3C2)C(F)(F)F)c1 ZINC000880928700 FF On-Demand Mild MCHR1 21 40 CCC[C@](C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928708 EG On-Demand Mild CTSF 47 33 CCC[C@](C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928710 EG On-Demand Mild CTSF 47 33 CC(C)[C@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928712 EH On-Demand Mild MCHR1 25 40 CC(C)[C@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928714 EH On-Demand Mild MCHR1 25 40 O=C(NCc1ccc(O)cc1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880928721 FF On-Demand Anodyne P2RX7 68 63 O=C(NCc1ccc(O)cc1)[C@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880928721 FF On-Demand Anodyne LNPEP 52 35 O=C(NCc1ccc(O)cc1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880928722 FF On-Demand Anodyne P2RX7 68 63 O=C(NCc1ccc(O)cc1)[C@@H]1CC(=O)N(Cc2ccccc2Cl)C1 ZINC000880928722 FF On-Demand Anodyne LNPEP 52 35 C[C@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928733 DG On-Demand Mild MCHR1 30 40 C[C@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928734 DG On-Demand Mild MCHR1 30 40 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928735 DG On-Demand Mild MCHR1 30 40 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928736 DG On-Demand Mild MCHR1 30 40 N#Cc1cccc([C@@H](NC(=O)N(CCCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880928739 GH On-Demand Mild CTSF 56 32 N#Cc1cccc([C@@H](NC(=O)N(CCCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880928739 GH On-Demand Mild PTGES 29 45 N#Cc1cccc([C@H](NC(=O)N(CCCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880928740 GH On-Demand Mild CTSF 56 32 N#Cc1cccc([C@H](NC(=O)N(CCCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880928740 GH On-Demand Mild PTGES 29 45 N#Cc1cccc([C@@H](NC(=O)N2CCO[C@H](C#N)C2)C(F)(F)F)c1 ZINC000880928741 EE On-Demand Mild STK3 20 42 N#Cc1cccc([C@H](NC(=O)N2CCO[C@H](C#N)C2)C(F)(F)F)c1 ZINC000880928742 EE On-Demand Mild STK3 20 42 N#Cc1cccc([C@@H](NC(=O)N2CCO[C@@H](C#N)C2)C(F)(F)F)c1 ZINC000880928743 EE On-Demand Mild STK3 20 42 N#Cc1cccc([C@H](NC(=O)N2CCO[C@@H](C#N)C2)C(F)(F)F)c1 ZINC000880928744 EE On-Demand Mild STK3 20 42 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880928759 GF On-Demand Mild ITGA4 47 38 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880928760 GF On-Demand Mild ITGA4 47 38 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880928761 GF On-Demand Mild ITGA4 47 38 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880928762 GF On-Demand Mild ITGA4 47 38 CNC(=O)CCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928765 ED On-Demand Mild CTSF 55 33 CNC(=O)CCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928766 ED On-Demand Mild CTSF 55 33 CN(CC(=O)N1CCOCC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928779 GD On-Demand Mild CASR 29 43 CN(CC(=O)N1CCOCC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928780 GD On-Demand Mild CASR 29 43 CN(CCOC(C)(C)C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928821 FH On-Demand Mild CTSF 41 31 CN(CCOC(C)(C)C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928822 FH On-Demand Mild CTSF 41 31 CC1(C)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928823 EH On-Demand Mild CTSF 42 33 CC1(C)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928824 EH On-Demand Mild CTSF 42 33 CCOC(=O)[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928825 GG On-Demand Mild FDFT1 18 41 CCOC(=O)[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928825 GG On-Demand Mild LGMN 45 32 CCOC(=O)[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928826 GG On-Demand Mild FDFT1 18 41 CCOC(=O)[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880928826 GG On-Demand Mild LGMN 45 32 CCC[C@](C)(CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928829 EG On-Demand Mild CTSF 46 33 CCC[C@](C)(CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928831 EG On-Demand Mild CTSF 46 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CN2CCOCC2)C(F)(F)F)c1 ZINC000880928833 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CN2CCOCC2)C(F)(F)F)c1 ZINC000880928834 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@H](O)C(F)(F)F)C(F)(F)F)c1 ZINC000880928835 GG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2[C@H](O)C(F)(F)F)C(F)(F)F)c1 ZINC000880928836 GG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2[C@@H](O)C(F)(F)F)C(F)(F)F)c1 ZINC000880928837 GG On-Demand Mild LGMN 48 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2[C@@H](O)C(F)(F)F)C(F)(F)F)c1 ZINC000880928838 GG On-Demand Mild LGMN 48 33 CC(C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928843 DE On-Demand Mild CTSF 70 34 CC(C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928843 DE On-Demand Mild CTSL 24 40 CC(C)(O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928843 DE On-Demand Mild CTSS 17 40 CC(C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928844 DE On-Demand Mild CTSF 70 34 CC(C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928844 DE On-Demand Mild CTSL 24 40 CC(C)(O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928844 DE On-Demand Mild CTSS 17 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2C2CC2)C(F)(F)F)c1 ZINC000880928847 EH On-Demand Mild LGMN 51 34 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2C2CC2)C(F)(F)F)c1 ZINC000880928848 EH On-Demand Mild LGMN 51 34 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2C2CC2)C(F)(F)F)c1 ZINC000880928849 EH On-Demand Mild LGMN 51 34 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2C2CC2)C(F)(F)F)c1 ZINC000880928850 EH On-Demand Mild LGMN 51 34 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928851 GF On-Demand Mild LGMN 75 38 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928851 GF On-Demand Mild WNT3 40 32 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928852 GF On-Demand Mild LGMN 75 38 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928852 GF On-Demand Mild WNT3 40 32 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928853 GF On-Demand Mild LGMN 75 38 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928853 GF On-Demand Mild WNT3 40 32 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928854 GF On-Demand Mild LGMN 75 38 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2C(=O)NC2CC2)C(F)(F)F)c1 ZINC000880928854 GF On-Demand Mild WNT3 40 32 COC(=O)C[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928857 FF On-Demand Mild LGMN 62 34 COC(=O)C[C@@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928857 FF On-Demand Mild CHRNA10 19 40 COC(=O)C[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928858 FF On-Demand Mild LGMN 62 34 COC(=O)C[C@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928858 FF On-Demand Mild CHRNA10 19 40 COC(=O)C[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928859 FF On-Demand Mild LGMN 62 34 COC(=O)C[C@H]1CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928859 FF On-Demand Mild CHRNA10 19 40 COC(=O)C[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928860 FF On-Demand Mild LGMN 62 34 COC(=O)C[C@@H]1CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928860 FF On-Demand Mild CHRNA10 19 40 COCC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928861 EF On-Demand Mild CTSF 70 34 COCC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928861 EF On-Demand Mild CTSL 28 40 COCC(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928861 EF On-Demand Mild CTSS 22 40 COCC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928862 EF On-Demand Mild CTSF 70 34 COCC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928862 EF On-Demand Mild CTSL 28 40 COCC(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928862 EF On-Demand Mild CTSS 22 40 N#Cc1cccc([C@H](NC(=O)N2CCc3c[nH]nc3C2)C(F)(F)F)c1 ZINC000880928873 EF On-Demand Mild MAPK1 44 35 N#Cc1cccc([C@@H](NC(=O)N2CCc3c[nH]nc3C2)C(F)(F)F)c1 ZINC000880928874 EF On-Demand Mild MAPK1 44 35 C[C@@H](CCS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928887 GE On-Demand Mild CTSF 70 38 C[C@@H](CCS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928887 GE On-Demand Mild CTSL 23 44 C[C@@H](CCS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928888 GE On-Demand Mild CTSF 70 38 C[C@@H](CCS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928888 GE On-Demand Mild CTSL 23 44 C[C@H](CCS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928889 GE On-Demand Mild CTSF 70 38 C[C@H](CCS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928889 GE On-Demand Mild CTSL 23 44 C[C@H](CCS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928890 GE On-Demand Mild CTSF 70 38 C[C@H](CCS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880928890 GE On-Demand Mild CTSL 23 44 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2CN2CCCC2)C(F)(F)F)c1 ZINC000880928912 GG On-Demand Mild LGMN 51 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2CN2CCCC2)C(F)(F)F)c1 ZINC000880928913 GG On-Demand Mild LGMN 51 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2CN2CCCC2)C(F)(F)F)c1 ZINC000880928945 GG On-Demand Mild LGMN 51 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2CN2CCCC2)C(F)(F)F)c1 ZINC000880928946 GG On-Demand Mild LGMN 51 33 CC(=O)N(C)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928971 GF On-Demand Mild MCHR1 31 41 CC(=O)N(C)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880928972 GF On-Demand Mild MCHR1 31 41 N#Cc1cccc([C@@H](NC(=O)N2CCC(O)(C(F)F)CC2)C(F)(F)F)c1 ZINC000880929007 GF On-Demand Mild CTSF 47 33 N#Cc1cccc([C@H](NC(=O)N2CCC(O)(C(F)F)CC2)C(F)(F)F)c1 ZINC000880929008 GF On-Demand Mild CTSF 47 33 CCC(CC)(CCO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929043 FG On-Demand Mild CTSF 56 32 CCC(CC)(CCO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929044 FG On-Demand Mild CTSF 56 32 N#Cc1cccc([C@@H](NC(=O)N2CCC(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880929053 GI On-Demand Mild CACNA1H 29 41 N#Cc1cccc([C@H](NC(=O)N2CCC(c3ccccn3)CC2)C(F)(F)F)c1 ZINC000880929054 GI On-Demand Mild CACNA1H 29 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@](F)(CO)C2)C(F)(F)F)c1 ZINC000880929158 EE On-Demand Mild CTSF 41 33 N#Cc1cccc([C@H](NC(=O)N2CC[C@@](F)(CO)C2)C(F)(F)F)c1 ZINC000880929159 EE On-Demand Mild CTSF 41 33 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@](F)(CO)C2)C(F)(F)F)c1 ZINC000880929160 EE On-Demand Mild CTSF 41 33 N#Cc1cccc([C@@H](NC(=O)N2CC[C@](F)(CO)C2)C(F)(F)F)c1 ZINC000880929161 EE On-Demand Mild CTSF 41 33 Cc1cc([C@@H]2CCCN2C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)no1 ZINC000880929175 GI On-Demand Mild CPT1A 30 40 Cc1cc([C@@H]2CCCN2C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)no1 ZINC000880929177 GI On-Demand Mild CPT1A 30 40 C[C@]1(CO)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929267 EF On-Demand Mild CTSF 41 32 C[C@]1(CO)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929267 EF On-Demand Mild SLC12A5 31 40 C[C@@]1(CO)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929268 EF On-Demand Mild CTSF 41 32 C[C@@]1(CO)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929268 EF On-Demand Mild SLC12A5 31 40 C[C@]1(CO)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929269 EF On-Demand Mild CTSF 41 32 C[C@]1(CO)CCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929269 EF On-Demand Mild SLC12A5 31 40 C[C@@]1(CO)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929270 EF On-Demand Mild CTSF 41 32 C[C@@]1(CO)CCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929270 EF On-Demand Mild SLC12A5 31 40 C[C@@H](O)C(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929271 GD On-Demand Mild CTSF 64 35 C[C@@H](O)C(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929273 GD On-Demand Mild CTSF 64 35 C#CCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929275 CE On-Demand Mild CTSF 42 32 C#CCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929276 CE On-Demand Mild CTSF 42 32 C=CCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929283 CF On-Demand Mild CTSF 65 34 C=CCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929283 CF On-Demand Mild MCHR1 17 40 C=CCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929284 CF On-Demand Mild CTSF 65 34 C=CCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929284 CF On-Demand Mild MCHR1 17 40 N#Cc1cccc([C@@H](NC(=O)NNC(=O)C2CCCC2)C(F)(F)F)c1 ZINC000880929301 FF On-Demand Reactive LGMN 41 33 N#Cc1cccc([C@H](NC(=O)NNC(=O)C2CCCC2)C(F)(F)F)c1 ZINC000880929302 FF On-Demand Reactive LGMN 41 33 N#Cc1cccc([C@H](NC(=O)NC2(CO)Cc3ccccc3C2)C(F)(F)F)c1 ZINC000880929303 GF On-Demand Mild CTSF 72 31 N#Cc1cccc([C@@H](NC(=O)NC2(CO)Cc3ccccc3C2)C(F)(F)F)c1 ZINC000880929304 GF On-Demand Mild CTSF 72 31 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880929309 DD On-Demand Mild MCHR1 26 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](O)C2)C(F)(F)F)c1 ZINC000880929310 DD On-Demand Mild MCHR1 26 41 CC(C)(CS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929315 GE On-Demand Mild CTSF 82 39 CC(C)(CS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929315 GE On-Demand Mild CTSK 38 41 CC(C)(CS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929315 GE On-Demand Mild CTSL 28 44 CC(C)(CS(C)(=O)=O)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929315 GE On-Demand Mild CTSS 21 44 CC(C)(CS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929316 GE On-Demand Mild CTSF 82 39 CC(C)(CS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929316 GE On-Demand Mild CTSK 38 41 CC(C)(CS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929316 GE On-Demand Mild CTSL 28 44 CC(C)(CS(C)(=O)=O)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929316 GE On-Demand Mild CTSS 21 44 C=C(C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929317 CG On-Demand Mild CTSF 60 33 C=C(C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929318 CG On-Demand Mild CTSF 60 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](C(N)=O)C2)C(F)(F)F)c1 ZINC000880929339 FE On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](C(N)=O)C2)C(F)(F)F)c1 ZINC000880929340 FE On-Demand Mild LGMN 41 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](C(N)=O)C2)C(F)(F)F)c1 ZINC000880929341 FE On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](C(N)=O)C2)C(F)(F)F)c1 ZINC000880929342 FE On-Demand Mild LGMN 41 33 N#Cc1cccc([C@H](NC(=O)NOCCO)C(F)(F)F)c1 ZINC000880929452 DD On-Demand Mild CTSF 56 32 N#Cc1cccc([C@@H](NC(=O)NOCCO)C(F)(F)F)c1 ZINC000880929453 DD On-Demand Mild CTSF 56 32 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929454 GH On-Demand Mild CPT1A 44 42 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929454 GH On-Demand Mild LGMN 44 33 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929455 GH On-Demand Mild CPT1A 44 42 N#Cc1cccc([C@H](NC(=O)N2CCCC[C@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929455 GH On-Demand Mild LGMN 44 33 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929456 GH On-Demand Mild CPT1A 44 42 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929456 GH On-Demand Mild LGMN 44 33 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929457 GH On-Demand Mild CPT1A 44 42 N#Cc1cccc([C@@H](NC(=O)N2CCCC[C@H]2c2cn[nH]c2)C(F)(F)F)c1 ZINC000880929457 GH On-Demand Mild LGMN 44 33 CC[C@@H](C)C(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929472 EF On-Demand Reactive CTSF 76 36 CC[C@@H](C)C(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929472 EF On-Demand Reactive CTSK 40 40 CC[C@@H](C)C(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929472 EF On-Demand Reactive CTSL 33 42 CC[C@@H](C)C(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929472 EF On-Demand Reactive CTSS 24 42 CC[C@@H](C)C(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929475 EF On-Demand Reactive CTSF 76 36 CC[C@@H](C)C(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929475 EF On-Demand Reactive CTSK 40 40 CC[C@@H](C)C(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929475 EF On-Demand Reactive CTSL 33 42 CC[C@@H](C)C(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929475 EF On-Demand Reactive CTSS 24 42 CN(CCN1CCOC(C)(C)C1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929484 GF On-Demand Mild CASR 27 42 CN(CCN1CCOC(C)(C)C1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929485 GF On-Demand Mild CASR 27 42 Cn1nccc1[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929490 GH On-Demand Mild CPT1A 34 42 Cn1nccc1[C@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929491 GH On-Demand Mild CPT1A 34 42 Cn1nccc1[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929492 GH On-Demand Mild CPT1A 34 42 Cn1nccc1[C@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929493 GH On-Demand Mild CPT1A 34 42 N#Cc1cccc([C@@H](NC(=O)N2CCC(c3cccnc3)CC2)C(F)(F)F)c1 ZINC000880929502 GI On-Demand Mild PTAFR 15 41 N#Cc1cccc([C@H](NC(=O)N2CCC(c3cccnc3)CC2)C(F)(F)F)c1 ZINC000880929503 GI On-Demand Mild PTAFR 15 41 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)CN2CCOCC2)C(F)(F)F)c1 ZINC000880929510 GD On-Demand Mild CASR 25 43 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)CN2CCOCC2)C(F)(F)F)c1 ZINC000880929511 GD On-Demand Mild CASR 25 43 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)CN2CCOCC2)C(F)(F)F)c1 ZINC000880929512 GD On-Demand Mild CASR 25 43 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)CN2CCOCC2)C(F)(F)F)c1 ZINC000880929513 GD On-Demand Mild CASR 25 43 CN(CC(C)(CO)CO)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929514 FD On-Demand Mild CTSF 42 32 CN(CC(C)(CO)CO)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929515 FD On-Demand Mild CTSF 42 32 N#Cc1cccc([C@@H](NC(=O)NCC2(CO)CCC2)C(F)(F)F)c1 ZINC000880929516 EF On-Demand Mild MCHR1 17 40 N#Cc1cccc([C@H](NC(=O)NCC2(CO)CCC2)C(F)(F)F)c1 ZINC000880929517 EF On-Demand Mild MCHR1 17 40 O=C(NCc1ccc(O)cc1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880929522 HK On-Demand Anodyne HDAC1 30 65 O=C(NCc1ccc(O)cc1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880929522 HK On-Demand Anodyne HDAC2 22 41 O=C(NCc1ccc(O)cc1)c1ccc(CSc2nc3ccccc3s2)cc1 ZINC000880929522 HK On-Demand Anodyne TMPRSS6 43 35 COC[C@@H](O)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929629 ED On-Demand Mild ADRB1 48 33 COC[C@@H](O)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929630 ED On-Demand Mild ADRB1 48 33 CN(C)C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880929650 FF On-Demand Mild MCHR1 42 40 CN(C)C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880929653 FF On-Demand Mild MCHR1 42 40 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](CN3CCOCC3)C2)C(F)(F)F)c1 ZINC000880929695 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](CN3CCOCC3)C2)C(F)(F)F)c1 ZINC000880929696 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](CN3CCOCC3)C2)C(F)(F)F)c1 ZINC000880929697 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](CN3CCOCC3)C2)C(F)(F)F)c1 ZINC000880929698 GF On-Demand Mild CASR 31 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](Oc3ccncc3)C2)C(F)(F)F)c1 ZINC000880929725 GG On-Demand Mild EPHX2 17 43 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](Oc3ccncc3)C2)C(F)(F)F)c1 ZINC000880929726 GG On-Demand Mild EPHX2 17 43 COCC1(O)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929729 FE On-Demand Mild CTSF 47 33 COCC1(O)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929729 FE On-Demand Mild S1PR2 25 40 COCC1(O)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929730 FE On-Demand Mild CTSF 47 33 COCC1(O)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929730 FE On-Demand Mild S1PR2 25 40 N#Cc1cccc([C@@H](NC(=O)NCC(=O)NCC(F)F)C(F)(F)F)c1 ZINC000880929731 FD On-Demand Mild CTSF 42 34 N#Cc1cccc([C@H](NC(=O)NCC(=O)NCC(F)F)C(F)(F)F)c1 ZINC000880929732 FD On-Demand Mild CTSF 42 34 CC(C)(O)CONC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929761 EE On-Demand Mild CTSF 54 32 CC(C)(O)CONC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929761 EE On-Demand Mild CTRB_BOVIN 44 32 CC(C)(O)CONC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929762 EE On-Demand Mild CTSF 54 32 CC(C)(O)CONC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929762 EE On-Demand Mild CTRB_BOVIN 44 32 CC[C@@H](CC#N)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929775 DG On-Demand Mild CTSF 65 34 CC[C@@H](CC#N)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929776 DG On-Demand Mild CTSF 65 34 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@H]1CO ZINC000880929787 EF On-Demand Mild CTSF 46 31 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@H]1CO ZINC000880929787 EF On-Demand Mild LGMN 50 33 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H]1CO ZINC000880929788 EF On-Demand Mild CTSF 46 31 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H]1CO ZINC000880929788 EF On-Demand Mild LGMN 50 33 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H]1CO ZINC000880929789 EF On-Demand Mild CTSF 46 31 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)[C@@H]1CO ZINC000880929789 EF On-Demand Mild LGMN 50 33 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@H]1CO ZINC000880929790 EF On-Demand Mild CTSF 46 31 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)[C@H]1CO ZINC000880929790 EF On-Demand Mild LGMN 50 33 CC(C)(C)C(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929801 EF On-Demand Reactive CTSF 46 32 CC(C)(C)C(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929802 EF On-Demand Reactive CTSF 46 32 COCC[C@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929811 ED On-Demand Mild CTSF 50 31 COCC[C@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929812 ED On-Demand Mild CTSF 50 31 COCC[C@@H](CO)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929813 ED On-Demand Mild CTSF 50 31 COCC[C@@H](CO)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880929814 ED On-Demand Mild CTSF 50 31 N#Cc1cccc([C@H](NC(=O)N2CCc3ccnc(O)c3C2)C(F)(F)F)c1 ZINC000880929920 GG On-Demand Mild MAPK1 42 33 N#Cc1cccc([C@@H](NC(=O)N2CCc3ccnc(O)c3C2)C(F)(F)F)c1 ZINC000880929921 GG On-Demand Mild MAPK1 42 33 Cc1noc(C2CN(C(=O)N[C@H](c3cccc(C#N)c3)C(F)(F)F)C2)n1 ZINC000880929928 FF On-Demand Mild ETHR 42 34 Cc1noc(C2CN(C(=O)N[C@@H](c3cccc(C#N)c3)C(F)(F)F)C2)n1 ZINC000880929929 FF On-Demand Mild ETHR 42 34 CC(C)[C@H](O)C1(CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929930 FG On-Demand Mild CTSF 50 37 CC(C)[C@H](O)C1(CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929930 FG On-Demand Mild MCHR1 19 40 CC(C)[C@H](O)C1(CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929931 FG On-Demand Mild CTSF 50 37 CC(C)[C@H](O)C1(CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880929931 FG On-Demand Mild MCHR1 19 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](CC(N)=O)C2)C(F)(F)F)c1 ZINC000880929980 FE On-Demand Mild LGMN 61 35 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](CC(N)=O)C2)C(F)(F)F)c1 ZINC000880929981 FE On-Demand Mild LGMN 61 35 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](CC(N)=O)C2)C(F)(F)F)c1 ZINC000880929982 FE On-Demand Mild LGMN 61 35 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](CC(N)=O)C2)C(F)(F)F)c1 ZINC000880929983 FE On-Demand Mild LGMN 61 35 CN(CC1(CO)CC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930026 EF On-Demand Mild CTSF 59 33 CN(CC1(CO)CC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930027 EF On-Demand Mild CTSF 59 33 N#Cc1cccc([C@H](NC(=O)N[C@@H]2c3ccccc3C[C@@H]2O)C(F)(F)F)c1 ZINC000880930030 GG On-Demand Mild PLM2_PLAFA 47 38 N#Cc1cccc([C@H](NC(=O)N[C@@H]2c3ccccc3C[C@H]2O)C(F)(F)F)c1 ZINC000880930031 GG On-Demand Mild PLM2_PLAFA 47 38 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](Cc3ccncc3)C2)C(F)(F)F)c1 ZINC000880930044 GH On-Demand Mild CCR3 39 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](Cc3ccncc3)C2)C(F)(F)F)c1 ZINC000880930045 GH On-Demand Mild CCR3 39 43 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](Cc3ccncc3)C2)C(F)(F)F)c1 ZINC000880930046 GH On-Demand Mild CCR3 39 43 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](Cc3ccncc3)C2)C(F)(F)F)c1 ZINC000880930047 GH On-Demand Mild CCR3 39 43 CN(CCO)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930056 GE On-Demand Mild MCHR1 42 37 CN(CCO)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930057 GE On-Demand Mild MCHR1 42 37 O=C(NCc1ccc(O)cc1)c1ccc(OS(=O)(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000880930091 IF On-Demand Bother CA2 15 54 O=C(NCc1ccc(O)cc1)c1ccc(OS(=O)(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000880930091 IF On-Demand Bother CACNA1D 61 38 O=C(NCc1ccc(O)cc1)c1ccc(OS(=O)(=O)c2cccc([N+](=O)[O-])c2)cc1 ZINC000880930091 IF On-Demand Bother ACR 17 40 C[C@@H](CCN1CCN(C)CC1)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930096 GE On-Demand Mild MCHR1 26 43 C[C@@H](CCN1CCN(C)CC1)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930097 GE On-Demand Mild MCHR1 26 43 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CTSB 15 43 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CYSP_TRYCR 38 43 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CTSF 66 43 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CTSK 21 41 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CTSL 17 41 CNC(=O)[C@@H](NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930100 FE On-Demand Mild CTSV 15 43 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CTSB 15 43 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CYSP_TRYCR 38 43 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CTSF 66 43 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CTSK 21 41 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CTSL 17 41 CNC(=O)[C@@H](NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880930101 FE On-Demand Mild CTSV 15 43 CC[C@@H](C)CN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930110 EH On-Demand Mild CTSF 53 35 CC[C@@H](C)CN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930112 EH On-Demand Mild CTSF 53 35 CCC(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930118 DD On-Demand Reactive CTSF 61 33 CCC(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930119 DD On-Demand Reactive CTSF 61 33 CCC1(CO)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930135 FG On-Demand Mild CTSF 50 32 CCC1(CO)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930136 FG On-Demand Mild CTSF 50 32 C=C[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930151 EH On-Demand Mild LGMN 51 34 C=C[C@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930152 EH On-Demand Mild LGMN 51 34 C=C[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930153 EH On-Demand Mild LGMN 51 34 C=C[C@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930154 EH On-Demand Mild LGMN 51 34 C[C@@H](C(N)=O)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930163 ED On-Demand Mild CTSF 48 35 C[C@@H](C(N)=O)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930165 ED On-Demand Mild CTSF 48 35 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)C(F)(F)F)c1 ZINC000880930205 GE On-Demand Mild MCHR1 23 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)C(F)(F)F)c1 ZINC000880930206 GE On-Demand Mild MCHR1 23 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](NC(=O)NC3CC3)C2)C(F)(F)F)c1 ZINC000880930207 GE On-Demand Mild MCHR1 23 41 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](NC(=O)NC3CC3)C2)C(F)(F)F)c1 ZINC000880930208 GE On-Demand Mild MCHR1 23 41 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880930232 FE On-Demand Mild ITGA4 49 39 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880930233 FE On-Demand Mild ITGA4 49 39 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880930234 FE On-Demand Mild ITGA4 49 39 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](n3cncn3)C2)C(F)(F)F)c1 ZINC000880930235 FE On-Demand Mild ITGA4 49 39 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C[C@@H]1F ZINC000880930252 EH On-Demand Mild MCHR1 20 40 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C[C@H]1F ZINC000880930253 EH On-Demand Mild MCHR1 20 40 C[C@@H]1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C[C@H]1F ZINC000880930254 EH On-Demand Mild MCHR1 20 40 C[C@@H]1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C[C@@H]1F ZINC000880930255 EH On-Demand Mild MCHR1 20 40 CN1CC[C@@H](CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930257 EE On-Demand Mild CCR3 26 41 CN1CC[C@@H](CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930257 EE On-Demand Mild CACNA1I 43 35 CN1CC[C@@H](CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930258 EE On-Demand Mild CCR3 26 41 CN1CC[C@@H](CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930258 EE On-Demand Mild CACNA1I 43 35 CN1CC[C@H](CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930259 EE On-Demand Mild CCR3 26 41 CN1CC[C@H](CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930259 EE On-Demand Mild CACNA1I 43 35 CN1CC[C@H](CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930260 EE On-Demand Mild CCR3 26 41 CN1CC[C@H](CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880930260 EE On-Demand Mild CACNA1I 43 35 N#Cc1cccc([C@H](NC(=O)N(CCO)C2CCOCC2)C(F)(F)F)c1 ZINC000880930265 FE On-Demand Mild MCHR1 28 40 N#Cc1cccc([C@@H](NC(=O)N(CCO)C2CCOCC2)C(F)(F)F)c1 ZINC000880930266 FE On-Demand Mild MCHR1 28 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](CN3CCCCC3)C2)C(F)(F)F)c1 ZINC000880930283 GH On-Demand Mild MCHR1 39 42 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](CN3CCCCC3)C2)C(F)(F)F)c1 ZINC000880930284 GH On-Demand Mild MCHR1 39 42 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](CN3CCCCC3)C2)C(F)(F)F)c1 ZINC000880930285 GH On-Demand Mild MCHR1 39 42 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](CN3CCCCC3)C2)C(F)(F)F)c1 ZINC000880930286 GH On-Demand Mild MCHR1 39 42 CN(CCOCCO)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930289 ED On-Demand Mild CTSF 42 32 CN(CCOCCO)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930290 ED On-Demand Mild CTSF 42 32 N#Cc1cccc([C@@H](NC(=O)N[C@H](CO)Cc2ccc(F)cc2)C(F)(F)F)c1 ZINC000880930295 GG On-Demand Mild CTSF 61 32 N#Cc1cccc([C@@H](NC(=O)N[C@@H](CO)Cc2ccc(F)cc2)C(F)(F)F)c1 ZINC000880930296 GG On-Demand Mild CTSF 61 32 N#Cc1cccc([C@H](NC(=O)N[C@H](CO)Cc2ccc(F)cc2)C(F)(F)F)c1 ZINC000880930297 GG On-Demand Mild CTSF 61 32 N#Cc1cccc([C@H](NC(=O)N[C@@H](CO)Cc2ccc(F)cc2)C(F)(F)F)c1 ZINC000880930298 GG On-Demand Mild CTSF 61 32 N#Cc1cccc([C@H](NC(=O)N(CCO)C2CCC2)C(F)(F)F)c1 ZINC000880930299 EF On-Demand Mild MCHR1 34 40 N#Cc1cccc([C@@H](NC(=O)N(CCO)C2CCC2)C(F)(F)F)c1 ZINC000880930300 EF On-Demand Mild MCHR1 34 40 COC(=O)C1(CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930334 FE On-Demand Mild CTSF 68 34 COC(=O)C1(CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930335 FE On-Demand Mild CTSF 68 34 CC1(CO)CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930366 FF On-Demand Mild CTSF 52 33 CC1(CO)CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930367 FF On-Demand Mild CTSF 52 33 N#Cc1cccc([C@H](NC(=O)Nc2cc(C3CC3)[nH]n2)C(F)(F)F)c1 ZINC000880930378 EH On-Demand Mild CDK2 15 50 N#Cc1cccc([C@H](NC(=O)Nc2cc(C3CC3)[nH]n2)C(F)(F)F)c1 ZINC000880930378 EH On-Demand Mild PKNB 80 48 N#Cc1cccc([C@@H](NC(=O)Nc2cc(C3CC3)[nH]n2)C(F)(F)F)c1 ZINC000880930379 EH On-Demand Mild CDK2 15 50 N#Cc1cccc([C@@H](NC(=O)Nc2cc(C3CC3)[nH]n2)C(F)(F)F)c1 ZINC000880930379 EH On-Demand Mild PKNB 80 48 C[C@@H](O)CCCNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930402 EF On-Demand Mild CTSF 62 35 C[C@@H](O)CCCNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930403 EF On-Demand Mild CTSF 62 35 N#Cc1cccc([C@H](NC(=O)NCCF)C(F)(F)F)c1 ZINC000880930404 CE On-Demand Mild CTSF 42 32 N#Cc1cccc([C@@H](NC(=O)NCCF)C(F)(F)F)c1 ZINC000880930405 CE On-Demand Mild CTSF 42 32 CN(C)CCCC1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930412 GH On-Demand Mild MCHR1 36 42 CN(C)CCCC1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930413 GH On-Demand Mild MCHR1 36 42 C=CCCN(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930414 DG On-Demand Mild CTSF 65 34 C=CCCN(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930415 DG On-Demand Mild CTSF 65 34 O=C(C[C@@H]1CCNC1=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880930509 ED On-Demand Anodyne MAPK1 42 36 O=C(C[C@@H]1CCNC1=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880930511 ED On-Demand Anodyne MAPK1 42 36 O=C(C[C@H]1CCNC1=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880930513 ED On-Demand Anodyne MAPK1 42 36 O=C(C[C@H]1CCNC1=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880930515 ED On-Demand Anodyne MAPK1 42 36 NS(=O)(=O)c1cc(NC(=O)N2CCC(CCc3ccccc3)CC2)cs1 ZINC000880930547 GG On-Demand Anodyne GRIN2B 33 41 NS(=O)(=O)c1cc(NC(=O)N2CCC(CCc3ccccc3)CC2)cs1 ZINC000880930547 GG On-Demand Anodyne ST14 56 34 C[C@@H]1C[C@H](c2ccccc2)C(C)(C)N1C(=O)Nc1csc(S(N)(=O)=O)c1 ZINC000880930587 GH On-Demand Anodyne ADAMTS5 47 35 CCn1nc(C)c(CN(C)C(=O)CCCCc2ccc(OC)c(OC)c2)c1C ZINC000880930590 GH On-Demand Anodyne INHA 44 38 N#Cc1cccc([C@H](NC(=O)N2CCCN(C(=O)C3CC3)CC2)C(F)(F)F)c1 ZINC000880930599 GF On-Demand Mild MCHR1 15 40 N#Cc1cccc([C@@H](NC(=O)N2CCCN(C(=O)C3CC3)CC2)C(F)(F)F)c1 ZINC000880930603 GF On-Demand Mild MCHR1 15 40 Cn1c2ccccc2c2cc(C(=O)NCc3ccc(O)cc3)sc21 ZINC000880930606 EI On-Demand Anodyne UL54 69 35 N#Cc1cccc([C@H](NC(=O)NCCCNC(=O)C2CCC2)C(F)(F)F)c1 ZINC000880930610 GF On-Demand Mild TBK1 51 36 N#Cc1cccc([C@@H](NC(=O)NCCCNC(=O)C2CCC2)C(F)(F)F)c1 ZINC000880930614 GF On-Demand Mild TBK1 51 36 O=C1CC[C@H](c2ccc(C(=O)N[C@@H](CCO)c3ccc(Cl)c(F)c3)cc2)N1 ZINC000880930616 GG On-Demand Anodyne UTS2 64 37 O=C1CC[C@H](c2ccc(C(=O)N[C@H](CCO)c3ccc(Cl)c(F)c3)cc2)N1 ZINC000880930619 GG On-Demand Anodyne UTS2 64 37 CN1CCC(C)(CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930632 FG On-Demand Mild MCHR1 33 49 CN1CCC(C)(CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880930633 FG On-Demand Mild MCHR1 33 49 C[C@@](CO)(NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)c1ccccc1 ZINC000880930651 GG On-Demand Mild CTSF 70 33 CNC(C)(C)CNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930652 EE On-Demand Mild CTSF 58 33 CNC(C)(C)CNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930653 EE On-Demand Mild CTSF 58 33 N#Cc1cccc([C@@H](NC(=O)N2CC[C@H](c3ccccn3)C2)C(F)(F)F)c1 ZINC000880930668 FH On-Demand Mild MAP3K12 32 40 N#Cc1cccc([C@@H](NC(=O)N2CC[C@@H](c3ccccn3)C2)C(F)(F)F)c1 ZINC000880930669 FH On-Demand Mild MAP3K12 32 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@H](c3ccccn3)C2)C(F)(F)F)c1 ZINC000880930670 FH On-Demand Mild MAP3K12 32 40 N#Cc1cccc([C@H](NC(=O)N2CC[C@@H](c3ccccn3)C2)C(F)(F)F)c1 ZINC000880930671 FH On-Demand Mild MAP3K12 32 40 COCC1(NC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CCC1 ZINC000880930682 EG On-Demand Mild CTSF 51 34 COCC1(NC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CCC1 ZINC000880930683 EG On-Demand Mild CTSF 51 34 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H](CCO)c3ccc(Cl)c(F)c3)cc2)N1 ZINC000880930738 GG On-Demand Anodyne UTS2 64 37 O=C1CC[C@@H](c2ccc(C(=O)N[C@H](CCO)c3ccc(Cl)c(F)c3)cc2)N1 ZINC000880930740 GG On-Demand Anodyne UTS2 64 37 N#Cc1ccc(CN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C2CC2)cc1 ZINC000880930742 GI On-Demand Mild MCHR1 28 40 N#Cc1ccc(CN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C2CC2)cc1 ZINC000880930746 GI On-Demand Mild MCHR1 28 40 C[C@@H](CO)N(C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930754 DE On-Demand Mild CTSF 43 34 C[C@@H](CO)N(C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930757 DE On-Demand Mild CTSF 43 34 COc1ccc(N2CCC(NC(=O)Nc3cccc4c3NC(=O)CO4)CC2)cc1 ZINC000880930759 GF On-Demand Clean EPHX2 19 41 CN(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880930789 FE On-Demand Anodyne CA2 16 45 CN(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880930789 FE On-Demand Anodyne CA4 15 45 CN(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880930789 FE On-Demand Anodyne UL54 65 36 CN(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880930789 FE On-Demand Anodyne NAMPT 48 35 CC(C)(C)CC(=O)NNC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930804 FF On-Demand Reactive CTSF 54 33 CC(C)(C)CC(=O)NNC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930808 FF On-Demand Reactive CTSF 54 33 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](OCCO)C2)C(F)(F)F)c1 ZINC000880930811 FE On-Demand Mild LGMN 41 32 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](OCCO)C2)C(F)(F)F)c1 ZINC000880930814 FE On-Demand Mild LGMN 41 32 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](OCCO)C2)C(F)(F)F)c1 ZINC000880930818 FE On-Demand Mild LGMN 41 32 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](OCCO)C2)C(F)(F)F)c1 ZINC000880930821 FE On-Demand Mild LGMN 41 32 N#Cc1cccc([C@@H](NC(=O)NCC(F)(F)C(F)F)C(F)(F)F)c1 ZINC000880930832 FG On-Demand Mild CTSF 62 35 N#Cc1cccc([C@H](NC(=O)NCC(F)(F)C(F)F)C(F)(F)F)c1 ZINC000880930835 FG On-Demand Mild CTSF 62 35 C[C@@H](O)C(C)(C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930839 EF On-Demand Mild CTSF 50 35 CC(C)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880930848 DF On-Demand Anodyne CACNA1H 40 41 C[C@@H](O)C(C)(C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930852 EF On-Demand Mild CTSF 50 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CO)C1 ZINC000880930865 CE On-Demand Anodyne CCR3 52 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CO)C1 ZINC000880930867 CE On-Demand Anodyne CCR3 52 33 CN(C)c1ccc(F)cc1NC(=O)NCCCCn1ccnc1 ZINC000880930869 DF On-Demand Anodyne TBXAS1 44 47 CN(C)c1ccc(F)cc1NC(=O)NCCCCn1ccnc1 ZINC000880930869 DF On-Demand Anodyne QPCT 41 52 CCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880930881 CF On-Demand Anodyne CCR3 19 42 C[C@@H](CC#N)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930886 DF On-Demand Mild CTSF 58 35 C[C@@H](CC#N)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930886 DF On-Demand Mild CTSL 23 41 C[C@@H](CC#N)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930886 DF On-Demand Mild CTSS 15 41 C[C@@H](CC#N)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930892 DF On-Demand Mild CTSF 58 35 C[C@@H](CC#N)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930892 DF On-Demand Mild CTSL 23 41 C[C@@H](CC#N)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880930892 DF On-Demand Mild CTSS 15 41 CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880930903 CD On-Demand Anodyne HRH4 18 42 CCN1CC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880930905 DE On-Demand Anodyne CCR3 88 38 CCN1CC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880930905 DE On-Demand Anodyne CACNA1I 67 36 CC(=O)NCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880930910 CD On-Demand Anodyne CCR3 19 41 CN(C)c1ccc(F)cc1NC(=O)N1CCO[C@@H](c2ccccc2)C1 ZINC000880930920 EG On-Demand Anodyne RBP4 46 37 CN(C)c1ccc(F)cc1NC(=O)N1CCO[C@H](c2ccccc2)C1 ZINC000880930921 EG On-Demand Anodyne RBP4 46 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(N2CCCCC2)CC1 ZINC000880930923 EG On-Demand Anodyne L3MBTL3 106 44 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCCC1 ZINC000880930924 DE On-Demand Anodyne DRD4 41 31 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCCC1 ZINC000880930924 DE On-Demand Anodyne CCR3 61 39 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCCC1 ZINC000880930924 DE On-Demand Anodyne PLD2 51 34 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCCC1 ZINC000880930924 DE On-Demand Anodyne MCHR1 15 42 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCOCC2)nc1 ZINC000880930929 FE On-Demand Anodyne DGAT1 23 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCOCC2)nc1 ZINC000880930929 FE On-Demand Anodyne NAMPT 19 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880930932 EE On-Demand Anodyne PDGFRB 32 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880930932 EE On-Demand Anodyne P2RX3 17 44 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880930932 EE On-Demand Anodyne FAAH 24 46 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880930932 EE On-Demand Anodyne RBP4 21 40 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880930933 GG On-Demand Anodyne CCR3 16 41 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880930933 GG On-Demand Anodyne EPHX2 43 46 NS(=O)(=O)c1cc(NC(=O)N2CCC[C@H](c3ccccc3)CC2)cs1 ZINC000880930937 GG On-Demand Anodyne EPHX2 19 40 NS(=O)(=O)c1cc(NC(=O)N2CCC[C@@H](c3ccccc3)CC2)cs1 ZINC000880930940 GG On-Demand Anodyne EPHX2 19 40 CCOCCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880930948 CF On-Demand Anodyne CCR3 20 42 CN(C)c1ccc(F)cc1NC(=O)N(Cc1ccc(C(N)=O)cc1)C1CC1 ZINC000880930965 FG On-Demand Anodyne GCGR 24 40 CN(C)c1ccc(F)cc1NC(=O)N(Cc1ccc(C(N)=O)cc1)C1CC1 ZINC000880930965 FG On-Demand Anodyne GIPR 38 40 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCc3ccccc3C2)ccc1Cl ZINC000880930969 JH On-Demand Anodyne AKR1C3 72 49 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCc3ccccc3C2)ccc1Cl ZINC000880930969 JH On-Demand Anodyne NOD2 46 32 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCc3ccccc3C2)ccc1Cl ZINC000880930969 JH On-Demand Anodyne NAMPT 71 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000880930973 EE On-Demand Anodyne CCR3 17 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000880930973 EE On-Demand Anodyne EPHX2 48 52 CCNC(=O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880930986 FD On-Demand Anodyne SLC27A1 40 31 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)C2CC2)CC1 ZINC000880930991 EE On-Demand Anodyne EPHX2 35 42 CNC(=O)COc1cccc(CNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880930999 FE On-Demand Anodyne ROCK2 25 48 CNC(=O)COc1cccc(CNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880930999 FE On-Demand Anodyne PDS 42 37 COCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931007 CE On-Demand Anodyne CCR3 16 44 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880931010 GG On-Demand Anodyne CCR3 41 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880931010 GG On-Demand Anodyne EPHX2 50 48 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880931010 GG On-Demand Anodyne L3MBTL3 45 34 COc1ccccc1[C@H]1CCCN(C(=O)Nc2cccc3c2NC(=O)CO3)CC1 ZINC000880931044 GH On-Demand Anodyne RBP4 35 43 COc1ccccc1[C@@H]1CCCN(C(=O)Nc2cccc3c2NC(=O)CO3)CC1 ZINC000880931045 GH On-Demand Anodyne RBP4 35 43 CC[C@H](C)NC(=O)[C@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931046 FF On-Demand Mild CTSF 59 36 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931047 FF On-Demand Mild CTSF 59 36 CC[C@H](C)NC(=O)[C@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931048 FF On-Demand Mild CTSF 59 36 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931049 FF On-Demand Mild CTSF 59 36 C[C@@]1(CNC(=O)Nc2cccc3c2NC(=O)CO3)CCN(Cc2ccccc2)C1 ZINC000880931054 GG On-Demand Anodyne NPFFR1 42 36 CN(C)c1ccc(F)cc1NC(=O)NCC1CCC1 ZINC000880931103 CF On-Demand Anodyne CCR3 46 36 CN(C)c1ccc(F)cc1NC(=O)NCCCn1ccnc1 ZINC000880931105 DE On-Demand Anodyne TBXAS1 44 48 CN(C)c1ccc(F)cc1NC(=O)NCCCn1ccnc1 ZINC000880931105 DE On-Demand Anodyne QPCT 43 54 COCCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931106 CE On-Demand Anodyne CCR3 16 46 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCCC2)nc1 ZINC000880931108 FG On-Demand Anodyne SLC27A1 48 38 CN(C)c1ccc(F)cc1NC(=O)NC1CCOCC1 ZINC000880931113 CE On-Demand Anodyne EPHX2 29 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880931115 FF On-Demand Mild P2RY12 17 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880931115 FF On-Demand Mild RBP4 16 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(CC2CC2)CC1 ZINC000880931118 DE On-Demand Anodyne CCR3 45 41 CN(C)C(=O)CCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931121 DD On-Demand Anodyne CCR3 15 40 O=C(CC12C[C@H]3C[C@@H](CC(Br)(C3)C1)C2)NCc1ccc(O)cc1 ZINC000880931133 GI On-Demand Anodyne BOTA 32 45 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931134 FG On-Demand Anodyne MAPK1 47 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931135 FG On-Demand Anodyne MAPK1 47 36 C[C@@H]1CCc2n[nH]cc2[C@H]1C(=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931136 FG On-Demand Anodyne MAPK1 47 36 C[C@@H]1CCc2n[nH]cc2[C@@H]1C(=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931137 FG On-Demand Anodyne MAPK1 47 36 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne CA2 43 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne CA4 47 38 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne CA12 24 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne CA9 26 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne MTCA1 42 40 C[C@@H](c1ccc(S(N)(=O)=O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931152 GF On-Demand Anodyne P96878_MYCTU 47 40 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880931159 FG On-Demand Anodyne MAPK11 35 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880931159 FG On-Demand Anodyne MAPK14 44 43 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880931159 FG On-Demand Anodyne CCR3 39 43 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880931159 FG On-Demand Anodyne ROCK2 19 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(C(=O)NC2CC2)c1 ZINC000880931159 FG On-Demand Anodyne MCHR1 17 44 CCCCN(CCO)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931161 CF On-Demand Anodyne SOAT1 30 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCCC1 ZINC000880931189 CF On-Demand Anodyne CCR3 19 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCCC1 ZINC000880931189 CF On-Demand Anodyne EPHX2 44 51 COc1cc2c(cc1OC)CN(C(=O)Nc1cc(F)ccc1N(C)C)CC2 ZINC000880931193 FG On-Demand Anodyne ABCB1B 43 36 COc1cc2c(cc1OC)CN(C(=O)Nc1cc(F)ccc1N(C)C)CC2 ZINC000880931193 FG On-Demand Anodyne HDAC6 25 40 COc1cc2c(cc1OC)CN(C(=O)Nc1cc(F)ccc1N(C)C)CC2 ZINC000880931193 FG On-Demand Anodyne ABCB1 19 42 CN1CCN(C2CCN(C(=O)Nc3csc(S(N)(=O)=O)c3)CC2)CC1 ZINC000880931196 GC On-Demand Anodyne L3MBTL3 65 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880931199 FE On-Demand Anodyne CCR3 33 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880931200 FE On-Demand Anodyne CCR3 33 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@H](O)C1 ZINC000880931204 CE On-Demand Anodyne EPHX2 21 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@@H](O)C1 ZINC000880931205 CE On-Demand Anodyne EPHX2 21 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@H](O)C1 ZINC000880931206 CE On-Demand Anodyne EPHX2 21 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H](O)C1 ZINC000880931207 CE On-Demand Anodyne EPHX2 21 41 CC(C)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931209 EG On-Demand Anodyne CCR1 29 40 CC(C)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931209 EG On-Demand Anodyne CCR3 52 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(C)(C)C)CC1 ZINC000880931212 EG On-Demand Anodyne EPHX2 41 39 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccc(C#N)cn2)CC1 ZINC000880931214 FF On-Demand Mild PDGFRB 15 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccc(C#N)cn2)CC1 ZINC000880931214 FF On-Demand Mild DGAT1 19 44 CNC(=O)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931228 FD On-Demand Anodyne DRD4 15 41 CNC(=O)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931228 FD On-Demand Anodyne CCR3 52 43 CNC(=O)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931228 FD On-Demand Anodyne MCHR1 19 40 CN(C)c1ccc(F)cc1NC(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000880931238 FE On-Demand Anodyne PIK3CA 17 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000880931238 FE On-Demand Anodyne MTOR 29 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000880931238 FE On-Demand Anodyne PIK3CG 15 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000880931238 FE On-Demand Anodyne EPHB4 52 34 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCCc3ccccc32)ccc1Cl ZINC000880931250 JI On-Demand Anodyne NAMPT 45 38 CSc1nccnc1C(=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931266 FF On-Demand Anodyne MAPK1 45 35 CSc1nccnc1C(=O)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931266 FF On-Demand Anodyne UTS2 42 32 CSc1nccnc1C(=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931267 FF On-Demand Anodyne MAPK1 45 35 CSc1nccnc1C(=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931267 FF On-Demand Anodyne UTS2 42 32 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880931278 HD On-Demand Anodyne UL54 38 43 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880931278 HD On-Demand Anodyne DPOL_VZVD 44 43 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Cl ZINC000880931278 HD On-Demand Anodyne NAMPT 88 54 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880931294 IH On-Demand Anodyne CA2 16 44 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880931294 IH On-Demand Anodyne CA4 16 41 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880931294 IH On-Demand Anodyne LIMK2 20 45 CN(c1ccccc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880931294 IH On-Demand Anodyne NAMPT 49 36 O=C(N[C@@H](CCO)c1ccc(Cl)c(F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880931298 GF On-Demand Anodyne MAPK1 40 39 O=C(N[C@H](CCO)c1ccc(Cl)c(F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880931299 GF On-Demand Anodyne MAPK1 40 39 CCOC(=O)CC1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880931311 GH On-Demand Mild P2RY12 26 42 CCOC(=O)CC1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880931312 GH On-Demand Mild P2RY12 26 42 CN1CCC(CNC(=O)Nc2cccc3c2NC(=O)CO3)(c2ccccc2)CC1 ZINC000880931378 GF On-Demand Anodyne KCNA3 37 41 CN1CCC(CNC(=O)Nc2cccc3c2NC(=O)CO3)(c2ccccc2)CC1 ZINC000880931378 GF On-Demand Anodyne SOAT1 17 44 CCCN(CC1CC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931380 EH On-Demand Mild MCHR1 27 44 CCCN(CC1CC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931381 EH On-Demand Mild MCHR1 27 44 CCN1CCC[C@@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880931402 DE On-Demand Anodyne CCR3 97 47 CCN1CCC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880931403 DE On-Demand Anodyne CCR3 97 47 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCN(CC(F)(F)F)C1 ZINC000880931411 FF On-Demand Anodyne CCR3 76 40 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCN(CC(F)(F)F)C1 ZINC000880931411 FF On-Demand Anodyne CACNA1I 67 37 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880931412 FF On-Demand Anodyne CCR3 76 40 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880931412 FF On-Demand Anodyne CACNA1I 67 37 CN(C)c1ccc(F)cc1NC(=O)NCC1CC1 ZINC000880931414 CE On-Demand Anodyne CCR3 40 36 CN(C)c1ccc(F)cc1NC(=O)NCC1CC1 ZINC000880931414 CE On-Demand Anodyne CACNA1I 41 33 CN(C)c1ccc(F)cc1NC(=O)NCCCO ZINC000880931434 CD On-Demand Anodyne CCR3 19 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2)CC1 ZINC000880931438 EG On-Demand Anodyne HTR1A 16 44 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2)CC1 ZINC000880931438 EG On-Demand Anodyne PDGFRB 17 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2)CC1 ZINC000880931438 EG On-Demand Anodyne HTR7 29 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2)CC1 ZINC000880931438 EG On-Demand Anodyne FAAH 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000880931443 GG On-Demand Anodyne DRD4 21 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000880931443 GG On-Demand Anodyne CCR3 34 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000880931443 GG On-Demand Anodyne MCHR1 27 50 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931448 GG On-Demand Anodyne ASAH1 52 34 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931452 FF On-Demand Anodyne CCR3 29 43 CCOC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880931452 FF On-Demand Anodyne EPHX2 51 42 CN(C)c1ccc(F)cc1NC(=O)N(CCO)Cc1ccccc1 ZINC000880931454 EF On-Demand Anodyne SOAT1 20 43 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(-c3ccccc3F)c(S)nc2c1 ZINC000880931461 HG On-Demand Anodyne POLR1A 43 29 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880931472 FF On-Demand Anodyne NPY2R 21 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C2CC2)CC1 ZINC000880931473 DF On-Demand Anodyne CCR3 27 40 COCCOc1ncccc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931475 FF On-Demand Anodyne P2RX7 23 40 COCCOc1ncccc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931475 FF On-Demand Anodyne P2RY1 31 44 COc1ncccc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931483 DF On-Demand Anodyne P2RX7 24 43 COc1ncccc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931483 DF On-Demand Anodyne P2RY1 36 45 COc1ncccc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931483 DF On-Demand Anodyne ROCK2 16 40 C=CCN(C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880931511 EH On-Demand Mild CTSF 70 36 C=CCN(C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F)C(C)C ZINC000880931512 EH On-Demand Mild CTSF 70 36 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931541 GF On-Demand Mild ADRB2 26 40 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931541 GF On-Demand Mild ADRB1 61 39 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931541 GF On-Demand Mild ADRB3 26 40 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931541 GF On-Demand Mild CTSF 45 30 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931541 GF On-Demand Mild PDS 63 44 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931543 GF On-Demand Mild ADRB2 26 40 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931543 GF On-Demand Mild ADRB1 61 39 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931543 GF On-Demand Mild ADRB3 26 40 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931543 GF On-Demand Mild CTSF 45 30 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931543 GF On-Demand Mild PDS 63 44 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931545 GF On-Demand Mild ADRB2 26 40 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931545 GF On-Demand Mild ADRB1 61 39 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931545 GF On-Demand Mild ADRB3 26 40 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931545 GF On-Demand Mild CTSF 45 30 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931545 GF On-Demand Mild PDS 63 44 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931547 GF On-Demand Mild ADRB2 26 40 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931547 GF On-Demand Mild ADRB1 61 39 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931547 GF On-Demand Mild ADRB3 26 40 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931547 GF On-Demand Mild CTSF 45 30 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)COc2ccccc2)C(F)(F)F)c1 ZINC000880931547 GF On-Demand Mild PDS 63 44 CCOC(=O)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880931570 GG On-Demand Mild P2RY12 24 41 CCOC(=O)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880931572 GG On-Demand Mild P2RY12 24 41 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931575 FI On-Demand Mild CACNA1H 15 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931575 FI On-Demand Mild CPT1A 49 42 Cn1nc2c(c1C(=O)N[C@@H](CCO)c1ccc(Cl)c(F)c1)CSCC2 ZINC000880931578 GF On-Demand Anodyne MAPK1 57 35 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931579 FI On-Demand Mild CACNA1H 15 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931579 FI On-Demand Mild CPT1A 49 42 Cn1nc2c(c1C(=O)N[C@H](CCO)c1ccc(Cl)c(F)c1)CSCC2 ZINC000880931580 GF On-Demand Anodyne MAPK1 57 35 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931581 FI On-Demand Mild CACNA1H 15 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931581 FI On-Demand Mild CPT1A 49 42 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931583 FI On-Demand Mild CACNA1H 15 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2c2ccccn2)C(F)(F)F)c1 ZINC000880931583 FI On-Demand Mild CPT1A 49 42 CS(=O)(=O)C1CCC(C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)CC1 ZINC000880931603 GE On-Demand Anodyne CACNA1B 51 32 CS(=O)(=O)C1CCC(C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)CC1 ZINC000880931605 GE On-Demand Anodyne CACNA1B 51 32 N#Cc1cccc([C@H](NC(=O)N(CCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880931635 GG On-Demand Mild CTSF 62 32 N#Cc1cccc([C@H](NC(=O)N(CCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880931635 GG On-Demand Mild PTGES 30 46 N#Cc1cccc([C@@H](NC(=O)N(CCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880931636 GG On-Demand Mild CTSF 62 32 N#Cc1cccc([C@@H](NC(=O)N(CCO)Cc2ccccc2)C(F)(F)F)c1 ZINC000880931636 GG On-Demand Mild PTGES 30 46 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931671 GH On-Demand Mild BMP1 57 35 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931671 GH On-Demand Mild CTSF 51 33 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931671 GH On-Demand Mild GSK3A 18 40 O=C(COC1CC1)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931672 DE On-Demand Anodyne MAPK1 46 38 O=C(COC1CC1)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880931673 DE On-Demand Anodyne MAPK1 46 38 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931674 GH On-Demand Mild BMP1 57 35 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931674 GH On-Demand Mild CTSF 51 33 CN(Cc1ccc2c(c1)OCO2)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931674 GH On-Demand Mild GSK3A 18 40 C=CCN(CC=C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931676 DH On-Demand Mild CTSF 61 33 C=CCN(CC=C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931681 DH On-Demand Mild CTSF 61 33 CNc1ncc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)s1 ZINC000880931696 EF On-Demand Anodyne MAPK1 45 35 CNc1ncc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)s1 ZINC000880931696 EF On-Demand Anodyne UTS2 41 31 CNc1ncc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)s1 ZINC000880931697 EF On-Demand Anodyne MAPK1 45 35 CNc1ncc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)s1 ZINC000880931697 EF On-Demand Anodyne UTS2 41 31 O=C1CC[C@@H](c2ccc(C(=O)N[C@H](CO)c3cccc(C(F)(F)F)c3)cc2)N1 ZINC000880931698 GG On-Demand Anodyne MTTP 46 36 O=C1CC[C@H](c2ccc(C(=O)N[C@H](CO)c3cccc(C(F)(F)F)c3)cc2)N1 ZINC000880931699 GG On-Demand Anodyne MTTP 46 36 O=C1CC[C@@H](c2ccc(C(=O)N[C@@H](CO)c3cccc(C(F)(F)F)c3)cc2)N1 ZINC000880931700 GG On-Demand Anodyne MTTP 46 36 O=C1CC[C@H](c2ccc(C(=O)N[C@@H](CO)c3cccc(C(F)(F)F)c3)cc2)N1 ZINC000880931701 GG On-Demand Anodyne MTTP 46 36 COc1ccccc1[C@@H](O)CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931708 EF On-Demand Anodyne SOAT1 19 40 Cc1cc([C@@H]2CCCN2C(=O)Nc2cc(F)ccc2N(C)C)on1 ZINC000880931711 EH On-Demand Anodyne KCNA5 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)NCC(F)(F)F)CC1 ZINC000880931719 GF On-Demand Anodyne CACNA1G 39 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN([C@H](C(N)=O)c2ccccc2)CC1 ZINC000880931730 GE On-Demand Anodyne NPY2R 68 38 CN(C)c1ccc(F)cc1NC(=O)N1CCN([C@@H](C(N)=O)c2ccccc2)CC1 ZINC000880931731 GE On-Demand Anodyne NPY2R 68 38 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCc2nc(O)ccc21 ZINC000880931735 EG On-Demand Anodyne TRPV1 18 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCc2nc(O)ccc21 ZINC000880931736 EG On-Demand Anodyne TRPV1 18 42 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CC(=O)NC2CC2)c1 ZINC000880931740 FE On-Demand Anodyne PANC 47 36 CN(Cc1ccc(Cl)nc1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880931741 EH On-Demand Anodyne NACHRBETA2 19 41 CN(C)C(=O)c1cccc(CNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880931744 FF On-Demand Anodyne ROCK2 23 42 COc1ccc(CN(C)C(=O)Nc2cc(F)ccc2N(C)C)cc1OC ZINC000880931752 FH On-Demand Anodyne MT-ND1 19 44 C[C@H](CN1CCOCC1)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880931755 DD On-Demand Anodyne P2RX3 29 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)c2ccccc2)CC1 ZINC000880931766 FI On-Demand Anodyne SLC18A3 40 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)c2ccccc2)CC1 ZINC000880931766 FI On-Demand Anodyne RBP4 40 36 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000880931767 EF On-Demand Anodyne PANC 56 40 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000880931768 EF On-Demand Anodyne PANC 56 40 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCCCCC1=O ZINC000880931782 FF On-Demand Anodyne CCR3 38 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](OCC(F)(F)F)C1 ZINC000880931784 FG On-Demand Anodyne LIPG 40 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](OCC(F)(F)F)C1 ZINC000880931785 FG On-Demand Anodyne LIPG 40 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000880931790 GH On-Demand Anodyne EPHX2 24 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000880931790 GH On-Demand Anodyne RBP4 40 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000880931790 GH On-Demand Anodyne SCD1 16 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880931792 FF On-Demand Anodyne CCR1 23 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880931792 FF On-Demand Anodyne CCR3 26 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880931792 FF On-Demand Anodyne MLNR 41 34 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880931792 FF On-Demand Anodyne FAAH 29 46 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931900 FG On-Demand Anodyne PTGER3 15 42 Cc1nc(C(C)C)ncc1C(=O)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931900 FG On-Demand Anodyne MAPK1 44 37 Cc1nc(C(C)C)ncc1C(=O)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931901 FG On-Demand Anodyne PTGER3 15 42 Cc1nc(C(C)C)ncc1C(=O)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931901 FG On-Demand Anodyne MAPK1 44 37 O=C(NCc1ccc(O)cc1)c1cc(-c2ccco2)nc2ccccc12 ZINC000880931917 EI On-Demand Anodyne ADORA1 22 57 O=C(NCc1ccc(O)cc1)c1cc(-c2ccco2)nc2ccccc12 ZINC000880931917 EI On-Demand Anodyne ADORA2A 32 57 O=C(NCc1ccc(O)cc1)c1cc(-c2ccco2)nc2ccccc12 ZINC000880931917 EI On-Demand Anodyne ADORA2B 15 57 O=C(NCc1ccc(O)cc1)c1cc(-c2ccco2)nc2ccccc12 ZINC000880931917 EI On-Demand Anodyne TACR3 19 62 O=C(NCc1ccc(O)cc1)c1cc(-c2ccco2)nc2ccccc12 ZINC000880931917 EI On-Demand Anodyne UL54 41 33 C[C@@H]1[C@@H](C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)CCN1C ZINC000880931926 EE On-Demand Anodyne MAPK1 49 36 C[C@@H]1[C@@H](C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)CCN1C ZINC000880931926 EE On-Demand Anodyne UTS2 41 31 C[C@@H]1[C@@H](C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)CCN1C ZINC000880931927 EE On-Demand Anodyne MAPK1 49 36 C[C@@H]1[C@@H](C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)CCN1C ZINC000880931927 EE On-Demand Anodyne UTS2 41 31 C=CC(C)(C)CC(=O)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931937 DG On-Demand Mild PDS 40 34 C=CC(C)(C)CC(=O)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880931938 DG On-Demand Mild PDS 40 34 NS(=O)(=O)c1cc(NC(=O)N2CCC(c3cccc(F)c3)CC2)cs1 ZINC000880931939 GF On-Demand Anodyne CACNA1H 46 37 CCN(Cc1ccncc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931958 FH On-Demand Mild CTSF 43 37 CCN(Cc1ccncc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931958 FH On-Demand Mild PTGES 28 42 CCN(Cc1ccncc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931962 FH On-Demand Mild CTSF 43 37 CCN(Cc1ccncc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880931962 FH On-Demand Mild PTGES 28 42 N#Cc1cccc([C@H](NC(=O)N2CCN(CC3CC3)CC2)C(F)(F)F)c1 ZINC000880931984 FF On-Demand Mild MCHR1 41 46 N#Cc1cccc([C@@H](NC(=O)N2CCN(CC3CC3)CC2)C(F)(F)F)c1 ZINC000880931985 FF On-Demand Mild MCHR1 41 46 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H]2c2ccncc2)C(F)(F)F)c1 ZINC000880931994 FI On-Demand Mild TRPM8 16 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H]2c2ccncc2)C(F)(F)F)c1 ZINC000880931998 FI On-Demand Mild TRPM8 16 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H]2c2ccncc2)C(F)(F)F)c1 ZINC000880932001 FI On-Demand Mild TRPM8 16 40 C[C@@H]1[C@@H](C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)CCN1C ZINC000880932002 EE On-Demand Anodyne MTTP 40 33 C[C@@H]1[C@@H](C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)CCN1C ZINC000880932002 EE On-Demand Anodyne CCR2 79 36 C[C@@H]1[C@@H](C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)CCN1C ZINC000880932003 EE On-Demand Anodyne MTTP 40 33 C[C@@H]1[C@@H](C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)CCN1C ZINC000880932003 EE On-Demand Anodyne CCR2 79 36 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H]2c2ccncc2)C(F)(F)F)c1 ZINC000880932004 FI On-Demand Mild TRPM8 16 40 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880932017 IH On-Demand Anodyne CPT1A 38 42 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)N2CCc3ccccc32)c1 ZINC000880932017 IH On-Demand Anodyne CA13 17 40 NS(=O)(=O)c1cc(NC(=O)N2CCC[C@@](F)(c3ccccc3)C2)cs1 ZINC000880932023 GF On-Demand Anodyne EPHX2 22 47 NS(=O)(=O)c1cc(NC(=O)N2CCC[C@](F)(c3ccccc3)C2)cs1 ZINC000880932025 GF On-Demand Anodyne EPHX2 22 47 COc1ccccc1N(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880932033 JH On-Demand Anodyne UL54 47 33 N#Cc1cccc([C@H](NC(=O)N2CCC(N3CCNC3=O)CC2)C(F)(F)F)c1 ZINC000880932046 GE On-Demand Mild CALCRL 27 44 N#Cc1cccc([C@@H](NC(=O)N2CCC(N3CCNC3=O)CC2)C(F)(F)F)c1 ZINC000880932047 GE On-Demand Mild CALCRL 27 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCOc2ccccc21 ZINC000880932086 EH On-Demand Anodyne TRPV1 18 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCOc2ccccc21 ZINC000880932088 EH On-Demand Anodyne TRPV1 18 44 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C2CCCC2)CC1 ZINC000880932110 EF On-Demand Anodyne HRH3 24 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C2CCCC2)CC1 ZINC000880932110 EF On-Demand Anodyne L3MBTL3 52 34 CN(C)c1ccc(F)cc1NC(=O)NC(C1CC1)C1CC1 ZINC000880932115 CG On-Demand Anodyne PYGL 16 42 CC(=O)NCC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932116 EE On-Demand Anodyne CACNA1I 60 33 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(S(C)(=O)=O)CC1 ZINC000880932125 FD On-Demand Anodyne CCR3 23 52 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(S(C)(=O)=O)CC1 ZINC000880932125 FD On-Demand Anodyne NPY5R 15 54 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(S(C)(=O)=O)CC1 ZINC000880932125 FD On-Demand Anodyne EPHX2 47 54 CN(C)c1ccc(F)cc1NC(=O)NCCc1cccnc1 ZINC000880932129 DF On-Demand Anodyne PTAFR 25 42 CN(C)c1ccc(F)cc1NC(=O)NCCc1cccnc1 ZINC000880932129 DF On-Demand Anodyne NAMPT 44 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000880932132 GG On-Demand Anodyne EPHX2 33 45 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000880932132 GG On-Demand Anodyne CACNA1G 50 43 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880932136 GH On-Demand Anodyne TSPO 25 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](N2CCCC2)C1 ZINC000880932137 EF On-Demand Anodyne L3MBTL3 64 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](N2CCCC2)C1 ZINC000880932138 EF On-Demand Anodyne L3MBTL3 64 38 CN(C)c1ccc(F)cc1NC(=O)NC1CC(C)(C)NC(C)(C)C1 ZINC000880932139 EG On-Demand Anodyne ENV 33 47 CN(C)c1ccc(F)cc1NC(=O)NC1CC(C)(C)NC(C)(C)C1 ZINC000880932139 EG On-Demand Anodyne EZH2 45 38 CN(C)c1ccc(F)cc1NC(=O)NCCNC(=O)c1ccco1 ZINC000880932143 EE On-Demand Anodyne KISS1R 59 39 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880932144 FF On-Demand Anodyne CCR3 24 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880932144 FF On-Demand Anodyne FAAH 34 49 CN(C)c1ccc(F)cc1NC(=O)NCCCN(C)S(C)(=O)=O ZINC000880932147 ED On-Demand Anodyne CCR3 15 40 CCOCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880932148 CE On-Demand Anodyne CCR3 19 41 CN(C)c1ccc(F)cc1NC(=O)NCCn1ccnc1 ZINC000880932149 CD On-Demand Anodyne TBXAS1 42 40 CN(C)c1ccc(F)cc1NC(=O)NCCn1ccnc1 ZINC000880932149 CD On-Demand Anodyne QPCT 30 46 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCOCC1 ZINC000880932156 DD On-Demand Anodyne HTR2A 26 44 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCOCC1 ZINC000880932156 DD On-Demand Anodyne ADRA1A 50 37 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCOCC1 ZINC000880932156 DD On-Demand Anodyne CCR3 46 45 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCOCC1 ZINC000880932156 DD On-Demand Anodyne EPHX2 26 47 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932157 FD On-Demand Anodyne CCR8 83 40 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932157 FD On-Demand Anodyne SFRP1 44 35 CCS(=O)(=O)NC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932157 FD On-Demand Anodyne WNT3 44 35 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC2CC2)CC1 ZINC000880932159 EF On-Demand Anodyne SIGMAR1 19 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC2CC2)CC1 ZINC000880932159 EF On-Demand Anodyne CCR3 87 46 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC2CC2)CC1 ZINC000880932159 EF On-Demand Anodyne EPHX2 43 36 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC2CC2)CC1 ZINC000880932159 EF On-Demand Anodyne CXCR3 20 49 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne HTR2A 24 46 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne HTR2C 15 43 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne ADRA1A 43 37 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne DRD3 43 36 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne CCR3 77 48 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC(C(N)=O)CC1 ZINC000880932165 GD On-Demand Anodyne MCHR1 21 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OCc2ccccc2)CC1 ZINC000880932170 FI On-Demand Anodyne GRIN2B 31 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OCc2ccccc2)CC1 ZINC000880932170 FI On-Demand Anodyne RBP4 56 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OCc2ccccc2)CC1 ZINC000880932170 FI On-Demand Anodyne SCD1 22 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cnn(C)c1 ZINC000880932172 CD On-Demand Anodyne PLA2G7 51 38 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(C(=O)N2CCCC2)cc1 ZINC000880932173 GG On-Demand Anodyne L3MBTL3 40 34 CN1CCC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880932175 CE On-Demand Anodyne CCR3 67 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccc(C(N)=O)cn2)CC1 ZINC000880932176 GD On-Demand Anodyne DGAT1 23 45 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CCCC1=O ZINC000880932177 GG On-Demand Anodyne P2RX7 47 41 CSc1nccnc1C(=O)Nc1nc(C2CCCCC2)cs1 ZINC000880932207 EH On-Demand Anodyne MAP1 42 38 O=C(COC1CC1)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880932249 DE On-Demand Anodyne CCR2 45 36 O=C(COC1CC1)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880932250 DE On-Demand Anodyne CCR2 45 36 CNc1nc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)cs1 ZINC000880932262 EF On-Demand Anodyne MAPK1 40 33 CNc1nc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)cs1 ZINC000880932262 EF On-Demand Anodyne UTS2 44 33 CNc1nc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)cs1 ZINC000880932264 EF On-Demand Anodyne MAPK1 40 33 CNc1nc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)cs1 ZINC000880932264 EF On-Demand Anodyne UTS2 44 33 O=C(N[C@@H](CCO)c1ccc(Cl)c(F)c1)[C@@H]1CCc2nncn2CC1 ZINC000880932268 FE On-Demand Anodyne MAPK1 48 37 O=C(N[C@H](CCO)c1ccc(Cl)c(F)c1)[C@@H]1CCc2nncn2CC1 ZINC000880932269 FE On-Demand Anodyne MAPK1 48 37 O=C(N[C@@H](CCO)c1ccc(Cl)c(F)c1)[C@H]1CCc2nncn2CC1 ZINC000880932270 FE On-Demand Anodyne MAPK1 48 37 O=C(N[C@H](CCO)c1ccc(Cl)c(F)c1)[C@H]1CCc2nncn2CC1 ZINC000880932271 FE On-Demand Anodyne MAPK1 48 37 COC(OC)c1ccc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)o1 ZINC000880932274 FG On-Demand Anodyne UTS2 50 33 COC(OC)c1ccc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)o1 ZINC000880932276 FG On-Demand Anodyne UTS2 50 33 O=C(N[C@@H](CO)c1cccc(C(F)(F)F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880932328 GF On-Demand Anodyne CASR 23 43 O=C(N[C@@H](CO)c1cccc(C(F)(F)F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880932328 GF On-Demand Anodyne CCR2 19 40 O=C(N[C@H](CO)c1cccc(C(F)(F)F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880932329 GF On-Demand Anodyne CASR 23 43 O=C(N[C@H](CO)c1cccc(C(F)(F)F)c1)c1ccc(CN2CCOCC2)o1 ZINC000880932329 GF On-Demand Anodyne CCR2 19 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne DRD4 22 52 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne SIGMAR1 17 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne SSTR5 45 37 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne CCR3 61 49 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne EPHX2 29 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccccn2)CC1 ZINC000880932359 FG On-Demand Anodyne MCHR1 36 41 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880932362 EF On-Demand Anodyne FDFT1 18 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880932376 EE On-Demand Anodyne ADRB2 36 43 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880932376 EE On-Demand Anodyne ADRB1 59 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880932376 EE On-Demand Anodyne ADRB3 31 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880932376 EE On-Demand Anodyne TSPO 41 34 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)COc1ccccc1 ZINC000880932376 EE On-Demand Anodyne PDS 50 37 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880932378 EE On-Demand Anodyne ADRB2 36 43 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880932378 EE On-Demand Anodyne ADRB1 59 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880932378 EE On-Demand Anodyne ADRB3 31 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880932378 EE On-Demand Anodyne TSPO 41 34 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)COc1ccccc1 ZINC000880932378 EE On-Demand Anodyne PDS 50 37 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCOCC1 ZINC000880932380 FE On-Demand Anodyne PIK3CA 31 40 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCOCC1 ZINC000880932380 FE On-Demand Anodyne MTOR 42 40 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCOCC1 ZINC000880932380 FE On-Demand Anodyne PIK3CG 21 40 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCOCC1 ZINC000880932380 FE On-Demand Anodyne SCN10A 21 48 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2O)CC1 ZINC000880932384 FF On-Demand Anodyne HTR1A 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2O)CC1 ZINC000880932384 FF On-Demand Anodyne KCNQ2 56 37 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccc2O)CC1 ZINC000880932384 FF On-Demand Anodyne RBP4 21 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880932408 FI On-Demand Anodyne HCRTR1 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880932408 FI On-Demand Anodyne PRCP 60 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880932410 FI On-Demand Anodyne HCRTR1 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880932410 FI On-Demand Anodyne PRCP 60 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCc2c1cnn2C ZINC000880932411 EF On-Demand Anodyne TRPV1 16 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCc2c1cnn2C ZINC000880932412 EF On-Demand Anodyne TRPV1 16 44 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880932414 FE On-Demand Anodyne GRM4 42 39 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880932422 FF On-Demand Anodyne CCR3 27 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880932422 FF On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCOCC1 ZINC000880932424 DD On-Demand Anodyne CCR3 40 38 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCOCC1 ZINC000880932424 DD On-Demand Anodyne EPHX2 25 52 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCOCC1 ZINC000880932424 DD On-Demand Anodyne PLD2 54 33 CN(Cc1cnn(C)c1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880932437 DE On-Demand Anodyne PLA2G7 58 39 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)C(C)(C)C)CC1 ZINC000880932439 FG On-Demand Anodyne CCR3 15 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)C(C)(C)C)CC1 ZINC000880932439 FG On-Demand Anodyne EPHX2 49 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccn2)CC1 ZINC000880932443 EF On-Demand Anodyne DRD4 27 45 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccn2)CC1 ZINC000880932443 EF On-Demand Anodyne PDGFRB 30 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccccn2)CC1 ZINC000880932443 EF On-Demand Anodyne FAAH 21 44 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne DRD4 27 44 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne KCNH2 15 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne SIGMAR1 28 48 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne SSTR5 51 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne CCR3 86 47 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne CXCR3 29 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000880932458 FG On-Demand Anodyne MCHR1 58 47 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncnc3c2cnn3C)CC1 ZINC000880932463 GD On-Demand Anodyne PDGFRB 56 45 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN2CCCC[C@@H]12 ZINC000880932476 DF On-Demand Anodyne CCR3 31 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000880932478 DF On-Demand Anodyne CCR3 31 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN2CCCC[C@H]12 ZINC000880932479 DF On-Demand Anodyne CCR3 31 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN2CCCC[C@H]12 ZINC000880932480 DF On-Demand Anodyne CCR3 31 40 COCCn1cc(NC(=O)Nc2cc(F)ccc2N(C)C)cn1 ZINC000880932486 DE On-Demand Anodyne PANC 43 36 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880932496 FG On-Demand Clean MTOR 22 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCOCC2)cc1 ZINC000880932496 FG On-Demand Clean STAT6 50 35 CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932519 DE On-Demand Anodyne SIGMAR1 15 41 CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932519 DE On-Demand Anodyne CCR3 64 46 CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932519 DE On-Demand Anodyne EPHX2 40 40 CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932519 DE On-Demand Anodyne CXCR3 21 40 CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880932519 DE On-Demand Anodyne MCHR1 22 41 Cc1cccc2c1OCC[C@@H]2NC(=O)Nc1cccc2c1NC(=O)CO2 ZINC000880932561 FF On-Demand Anodyne TRPV1 20 51 N#Cc1cccc([C@@H](NC(=O)N[C@@H]2c3ccccc3C[C@@H]2O)C(F)(F)F)c1 ZINC000880932589 GG On-Demand Mild PLM2_PLAFA 47 38 C[C@@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932593 EH On-Demand Mild LGMN 55 34 C[C@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932594 EH On-Demand Mild LGMN 55 34 C[C@@H]1CCCCN1C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932595 EH On-Demand Mild LGMN 55 34 Cc1cc([C@@H]2CCCN2C(=O)Nc2cccc3c2NC(=O)CO3)no1 ZINC000880932596 EF On-Demand Anodyne KCNA5 15 44 COC(OC)c1ccc(C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)o1 ZINC000880932606 FG On-Demand Anodyne PDS 40 35 COC(OC)c1ccc(C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)o1 ZINC000880932607 FG On-Demand Anodyne PDS 40 35 NS(=O)(=O)c1cc(NC(=O)N2CC3(CN(Cc4ccccc4)C3)C2)cs1 ZINC000880932624 GD On-Demand Anodyne FAAH 17 45 Cn1nnc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)n1 ZINC000880932626 DC On-Demand Anodyne MAPK1 47 35 Cn1nnc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)n1 ZINC000880932626 DC On-Demand Anodyne UTS2 44 33 Cn1nnc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)n1 ZINC000880932627 DC On-Demand Anodyne MAPK1 47 35 Cn1nnc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)n1 ZINC000880932627 DC On-Demand Anodyne UTS2 44 33 Cc1cccc2c1CCN(C(=O)Nc1csc(S(N)(=O)=O)c1)C2 ZINC000880932667 FE On-Demand Anodyne P2RY14 50 37 NS(=O)(=O)c1cc(NC(=O)N2CC[C@@]3(CCc4ccccc43)C2)cs1 ZINC000880932683 GF On-Demand Anodyne NPY5R 30 46 NS(=O)(=O)c1cc(NC(=O)N2CC[C@]3(CCc4ccccc43)C2)cs1 ZINC000880932684 GF On-Demand Anodyne NPY5R 30 46 CNc1ncc(C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)s1 ZINC000880932685 EF On-Demand Anodyne MAPK1 40 38 CNc1ncc(C(=O)N[C@@H](CO)c2cccc(C(F)(F)F)c2)s1 ZINC000880932685 EF On-Demand Anodyne PDS 41 32 CNc1ncc(C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)s1 ZINC000880932686 EF On-Demand Anodyne MAPK1 40 38 CNc1ncc(C(=O)N[C@H](CO)c2cccc(C(F)(F)F)c2)s1 ZINC000880932686 EF On-Demand Anodyne PDS 41 32 C[C@H]1CCCCN1C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932696 EH On-Demand Mild LGMN 55 34 CCOC(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932704 GF On-Demand Mild P2RY12 169 46 CCOC(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932704 GF On-Demand Mild MCHR1 22 44 CCOC(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932705 GF On-Demand Mild P2RY12 169 46 CCOC(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932705 GF On-Demand Mild MCHR1 22 44 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild CTSF 61 33 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild CTSK 22 44 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild CTSL 30 44 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild MTNR1A 20 40 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild CTSS 20 44 COc1ccc([C@@H](O)CNC(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932709 GG On-Demand Mild FFAR1 18 40 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild CTSF 61 33 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild CTSK 22 44 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild CTSL 30 44 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild MTNR1A 20 40 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild CTSS 20 44 COc1ccc([C@@H](O)CNC(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)cc1 ZINC000880932711 GG On-Demand Mild FFAR1 18 40 CC(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932755 FE On-Demand Mild CTSF 71 33 CC(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932756 FE On-Demand Mild CTSF 71 33 N#Cc1cccc([C@@H](NC(=O)N2CCC(N3CCCCC3)CC2)C(F)(F)F)c1 ZINC000880932760 GH On-Demand Mild MCHR1 20 41 N#Cc1cccc([C@@H](NC(=O)N2CCC(N3CCCCC3)CC2)C(F)(F)F)c1 ZINC000880932760 GH On-Demand Mild L3MBTL3 92 43 N#Cc1cccc([C@H](NC(=O)N2CCC(N3CCCCC3)CC2)C(F)(F)F)c1 ZINC000880932761 GH On-Demand Mild MCHR1 20 41 N#Cc1cccc([C@H](NC(=O)N2CCC(N3CCCCC3)CC2)C(F)(F)F)c1 ZINC000880932761 GH On-Demand Mild L3MBTL3 92 43 CS(=O)(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932780 GD On-Demand Mild CTSF 55 34 CS(=O)(=O)N1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932780 GD On-Demand Mild MCHR1 17 41 CS(=O)(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932781 GD On-Demand Mild CTSF 55 34 CS(=O)(=O)N1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932781 GD On-Demand Mild MCHR1 17 41 CCCN(CCC)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932795 EH On-Demand Mild CTSF 57 33 C=CCN(c1ccc(OC)cc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880932817 JI On-Demand Mild BMP1 64 38 C=CCN(c1ccc(OC)cc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880932817 JI On-Demand Mild MMP9 28 40 C=CCN(c1ccc(OC)cc1)S(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880932817 JI On-Demand Mild CA9 16 41 NS(=O)(=O)c1cc(NC(=O)N2CCC(c3ccc(F)cc3)CC2)cs1 ZINC000880932826 GF On-Demand Anodyne CACNA1H 29 40 Cc1coc(C(=O)N[C@H](CCO)c2ccc(Cl)c(F)c2)c1 ZINC000880932846 DG On-Demand Anodyne UTS2 59 37 Cc1coc(C(=O)N[C@@H](CCO)c2ccc(Cl)c(F)c2)c1 ZINC000880932847 DG On-Demand Anodyne UTS2 59 37 CCCN(CCC)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932857 EH On-Demand Mild CTSF 57 33 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932866 GG On-Demand Mild MCHR1 19 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932866 GG On-Demand Mild L3MBTL3 42 36 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932867 GG On-Demand Mild MCHR1 19 40 N#Cc1cccc([C@@H](NC(=O)N2CCC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932867 GG On-Demand Mild L3MBTL3 42 36 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932868 GG On-Demand Mild MCHR1 19 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932868 GG On-Demand Mild L3MBTL3 42 36 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932869 GG On-Demand Mild MCHR1 19 40 N#Cc1cccc([C@H](NC(=O)N2CCC[C@@H](N3CCCC3)C2)C(F)(F)F)c1 ZINC000880932869 GG On-Demand Mild L3MBTL3 42 36 CN(C)C(=O)C1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932883 GF On-Demand Mild MCHR1 23 41 CN(C)C(=O)C1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932884 GF On-Demand Mild MCHR1 23 41 CN1CCN(C2CCN(C(=O)Nc3cccc4c3NC(=O)CO4)CC2)CC1 ZINC000880932899 FD On-Demand Anodyne L3MBTL3 44 38 CC(=O)NCC1CCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932913 GF On-Demand Mild CACNA1I 48 32 CC(=O)NCC1CCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)CC1 ZINC000880932914 GF On-Demand Mild CACNA1I 48 32 CN(Cc1ccoc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932915 EH On-Demand Mild CTSF 41 32 CN(Cc1ccoc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932916 EH On-Demand Mild CTSF 41 32 CC(=O)N[C@@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880932976 FE On-Demand Mild MCHR1 20 40 CC(=O)N[C@H]1CCCN(C(=O)N[C@@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880932977 FE On-Demand Mild MCHR1 20 40 CC(=O)N[C@@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880932978 FE On-Demand Mild MCHR1 20 40 CC(=O)N[C@H]1CCCN(C(=O)N[C@H](c2cccc(C#N)c2)C(F)(F)F)C1 ZINC000880932979 FE On-Demand Mild MCHR1 20 40 CN(CC1CC1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932995 DG On-Demand Mild CTSF 40 35 CN(CC1CC1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880932996 DG On-Demand Mild CTSF 40 35 CN(Cc1ccsc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933011 FI On-Demand Mild CTSF 51 32 CN(Cc1ccsc1)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933011 FI On-Demand Mild HSD17B2 17 40 CN(Cc1ccsc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933012 FI On-Demand Mild CTSF 51 32 CN(Cc1ccsc1)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933012 FI On-Demand Mild HSD17B2 17 40 CN(CC(=O)NC(C)(C)C)C(=O)N[C@@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933067 FF On-Demand Mild CTSF 42 31 CN(CC(=O)NC(C)(C)C)C(=O)N[C@H](c1cccc(C#N)c1)C(F)(F)F ZINC000880933068 FF On-Demand Mild CTSF 42 31 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933109 GE On-Demand Mild CCR3 19 43 N#Cc1cccc([C@H](NC(=O)NC[C@@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933109 GE On-Demand Mild MCHR1 18 45 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933110 GE On-Demand Mild CCR3 19 43 N#Cc1cccc([C@H](NC(=O)NC[C@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933110 GE On-Demand Mild MCHR1 18 45 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933111 GE On-Demand Mild CCR3 19 43 N#Cc1cccc([C@@H](NC(=O)NC[C@@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933111 GE On-Demand Mild MCHR1 18 45 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933112 GE On-Demand Mild CCR3 19 43 N#Cc1cccc([C@@H](NC(=O)NC[C@H](O)CN2CCCCC2)C(F)(F)F)c1 ZINC000880933112 GE On-Demand Mild MCHR1 18 45 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(S(C)(=O)=O)CC1 ZINC000880933180 FD On-Demand Anodyne CCR3 63 41 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(S(C)(=O)=O)CC1 ZINC000880933180 FD On-Demand Anodyne NPY5R 15 45 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(S(C)(=O)=O)CC1 ZINC000880933180 FD On-Demand Anodyne CACNA1I 60 34 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(c2ccccc2C(N)=O)C1 ZINC000880933183 GE On-Demand Anodyne CCR3 23 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(c2ccccc2C(N)=O)C1 ZINC000880933184 GE On-Demand Anodyne CCR3 23 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(CC(F)F)CC1 ZINC000880933186 EE On-Demand Anodyne CACNA1H 41 36 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCC[C@@H]2C1 ZINC000880933187 DE On-Demand Anodyne HRH3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCC[C@@H]2C1 ZINC000880933187 DE On-Demand Anodyne L3MBTL3 42 35 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCC[C@H]2C1 ZINC000880933188 DE On-Demand Anodyne HRH3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCC[C@H]2C1 ZINC000880933188 DE On-Demand Anodyne L3MBTL3 42 35 CC(=O)N1CCc2cc(NC(=O)Nc3cc(F)ccc3N(C)C)ccc21 ZINC000880933206 FG On-Demand Anodyne HSD17B3 43 29 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(CC2CC2)C1 ZINC000880933223 DE On-Demand Anodyne CCR3 102 51 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(CC2CC2)C1 ZINC000880933223 DE On-Demand Anodyne CXCR3 15 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(CC2CC2)C1 ZINC000880933224 DE On-Demand Anodyne CCR3 102 51 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(CC2CC2)C1 ZINC000880933224 DE On-Demand Anodyne CXCR3 15 43 COC(=O)N1CCC[C@@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933235 EE On-Demand Anodyne CCR3 39 45 COC(=O)N1CCC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933236 EE On-Demand Anodyne CCR3 39 45 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880933237 EF On-Demand Anodyne CCR1 33 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880933237 EF On-Demand Anodyne CCR3 62 44 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880933237 EF On-Demand Anodyne EPHX2 41 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)F)CC1 ZINC000880933237 EF On-Demand Anodyne CXCR3 21 40 CN(C)c1ccc(F)cc1NC(=O)N(C)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880933248 GH On-Demand Anodyne CCR3 17 42 CN(C)c1ccc(F)cc1NC(=O)N(C)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880933248 GH On-Demand Anodyne L3MBTL3 58 37 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880933249 FF On-Demand Anodyne CCR3 47 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880933250 FF On-Demand Anodyne CCR3 47 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CN1CCCC1 ZINC000880933251 EF On-Demand Anodyne CCR3 33 49 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CN1CCCC1 ZINC000880933251 EF On-Demand Anodyne ACKR3 46 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CN1CCCC1 ZINC000880933252 EF On-Demand Anodyne CCR3 33 49 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CN1CCCC1 ZINC000880933252 EF On-Demand Anodyne ACKR3 46 32 Cc1noc(C)c1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880933256 DF On-Demand Anodyne P2RX7 31 50 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880933264 EF On-Demand Anodyne CCR3 58 48 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880933264 EF On-Demand Anodyne HPGDS 34 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880933265 EF On-Demand Anodyne CCR3 58 48 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880933265 EF On-Demand Anodyne HPGDS 34 40 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCCCC1=O ZINC000880933269 EE On-Demand Anodyne CCR3 41 41 Cc1noc(C)c1CCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880933270 DF On-Demand Anodyne P2RX7 22 49 CN(CCN1CCOCC1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933283 DD On-Demand Anodyne CASR 54 41 CN(CCN1CCOCC1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933283 DD On-Demand Anodyne EPHX2 20 42 CN(C)c1ccc(F)cc1NC(=O)N1CCCC[C@H](N2CCCC2)C1 ZINC000880933286 EG On-Demand Anodyne L3MBTL3 64 38 CN(C)c1ccc(F)cc1NC(=O)N1CCCC[C@@H](N2CCCC2)C1 ZINC000880933287 EG On-Demand Anodyne L3MBTL3 64 38 COC(=O)C1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933288 DE On-Demand Anodyne PTR1 44 32 C[C@@H](Cn1cncn1)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880933293 DD On-Demand Anodyne HIS3 79 37 CN(C)c1ccc(F)cc1NC(=O)NCCO ZINC000880933299 BD On-Demand Anodyne ALPL 26 40 CN(C)c1ccc(F)cc1NC(=O)NCC1(N2CCCC2)CCOCC1 ZINC000880933300 FF On-Demand Anodyne HCN1 58 38 CN(C)c1ccc(F)cc1NC(=O)NCC1(N2CCCC2)CCOCC1 ZINC000880933300 FF On-Demand Anodyne HCN4 48 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)C2CCCCC2)CC1 ZINC000880933312 GH On-Demand Anodyne EPHX2 37 46 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2nccn2C)CC1 ZINC000880933315 FD On-Demand Anodyne FAAH 15 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933316 GG On-Demand Anodyne ACACB 15 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933316 GG On-Demand Anodyne CACNA1I 63 35 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933317 GG On-Demand Anodyne ACACB 15 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933317 GG On-Demand Anodyne CACNA1I 63 35 CN1CCC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933334 DE On-Demand Anodyne CCR3 103 42 CN1CCC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933334 DE On-Demand Anodyne CACNA1I 49 36 CN(C[C@@H]1CCN(C(=O)Nc2cc(F)ccc2N(C)C)C1)C(=O)OC(C)(C)C ZINC000880933336 GH On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)Cc1ccccc1 ZINC000880933347 EF On-Demand Anodyne MME 64 38 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)Cc1ccccc1 ZINC000880933347 EF On-Demand Anodyne ANPEP 71 33 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)Cc1ccccc1 ZINC000880933347 EF On-Demand Anodyne PIN1 25 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)Cc1ccccc1 ZINC000880933348 EF On-Demand Anodyne MME 64 38 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)Cc1ccccc1 ZINC000880933348 EF On-Demand Anodyne ANPEP 71 33 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)Cc1ccccc1 ZINC000880933348 EF On-Demand Anodyne PIN1 25 41 CCCCCN(CCO)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933373 DF On-Demand Anodyne SOAT1 38 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880933379 FF On-Demand Anodyne NPY1R 24 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880933379 FF On-Demand Anodyne CCR3 51 39 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880933380 FF On-Demand Anodyne NPY1R 24 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880933380 FF On-Demand Anodyne CCR3 51 39 C[C@@H](O)C1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933389 DF On-Demand Anodyne CACNA1H 40 36 CN(C)c1ccc(F)cc1NC(=O)NCCCS(=O)(=O)c1ccccc1 ZINC000880933397 GF On-Demand Anodyne CCR3 24 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CCO)C1 ZINC000880933400 DF On-Demand Anodyne CCR3 41 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CCO)C1 ZINC000880933401 DF On-Demand Anodyne CCR3 41 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C2CCC2)CC1 ZINC000880933404 DF On-Demand Anodyne HRH3 26 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C2CCC2)CC1 ZINC000880933404 DF On-Demand Anodyne L3MBTL3 52 34 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1C ZINC000880933407 CE On-Demand Anodyne CCR3 59 38 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1C ZINC000880933407 CE On-Demand Anodyne CHRNA10 59 39 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1C ZINC000880933407 CE On-Demand Anodyne ACKR3 71 37 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN1C ZINC000880933408 CE On-Demand Anodyne CCR3 59 38 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN1C ZINC000880933408 CE On-Demand Anodyne CHRNA10 59 39 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN1C ZINC000880933408 CE On-Demand Anodyne ACKR3 71 37 CCCCN(CCOC)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933410 DG On-Demand Anodyne SOAT1 27 42 COc1ccnc(N2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)n1 ZINC000880933418 FE On-Demand Anodyne FAAH 23 45 O=C(NCc1ccc(O)cc1)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1 ZINC000880933423 HF On-Demand Anodyne KCNA3 15 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCC1 ZINC000880933431 CF On-Demand Anodyne EPHX2 46 48 COCCN(Cc1ccccc1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933436 EH On-Demand Anodyne SOAT1 18 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CCS(C)(=O)=O)CC1 ZINC000880933441 GD On-Demand Anodyne CCR3 61 46 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CCN2CCOCC2)CC1 ZINC000880933442 GF On-Demand Anodyne CCR3 45 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CCN2CCOCC2)CC1 ZINC000880933442 GF On-Demand Anodyne EPHX2 25 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](N2CCCC2)C1 ZINC000880933447 DF On-Demand Anodyne L3MBTL3 93 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](N2CCCC2)C1 ZINC000880933448 DF On-Demand Anodyne L3MBTL3 93 43 CN(C)c1ccc(F)cc1NC(=O)NCCCc1cnn(C)c1 ZINC000880933450 DE On-Demand Anodyne PLA2G7 53 35 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880933455 EF On-Demand Anodyne PLM1_PLAFA 45 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880933455 EF On-Demand Anodyne PLM2_PLAFA 68 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1c2ccccc2C[C@H]1O ZINC000880933456 EF On-Demand Anodyne PLM1_PLAFA 45 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1c2ccccc2C[C@H]1O ZINC000880933456 EF On-Demand Anodyne PLM2_PLAFA 68 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880933457 FG On-Demand Anodyne KCNQ2 61 38 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880933457 FG On-Demand Anodyne MTOR 19 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1N1CCOCC1 ZINC000880933457 FG On-Demand Anodyne SCN10A 15 46 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCC[C@@H](C(N)=O)C1 ZINC000880933462 FD On-Demand Anodyne SLC6A1 121 38 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCC[C@@H](C(N)=O)C1 ZINC000880933462 FD On-Demand Anodyne CCR3 79 47 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCC[C@H](C(N)=O)C1 ZINC000880933463 FD On-Demand Anodyne SLC6A1 121 38 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCC[C@H](C(N)=O)C1 ZINC000880933463 FD On-Demand Anodyne CCR3 79 47 C=CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933497 DF On-Demand Mild CCR3 52 43 C=CCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933497 DF On-Demand Mild MCHR1 17 40 COc1ccc(CN(CCO)C(=O)Nc2cc(F)ccc2N(C)C)c(OC)c1 ZINC000880933501 GF On-Demand Anodyne TSPO 39 40 CN(C)c1ccc(F)cc1NC(=O)NCC(=O)N1CCc2ccccc2C1 ZINC000880933515 FF On-Demand Anodyne DPP8 19 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2cccnn2)CC1 ZINC000880933516 EE On-Demand Anodyne FAAH 23 46 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CCO)CC1 ZINC000880933517 DD On-Demand Anodyne SIGMAR1 15 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CCO)CC1 ZINC000880933517 DD On-Demand Anodyne CCR3 79 46 CN(C)c1ccc(F)cc1NC(=O)N1CCc2cncnc2C1 ZINC000880933527 DE On-Demand Anodyne MAPK1 51 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880933537 GI On-Demand Anodyne HTR1D 20 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880933537 GI On-Demand Anodyne HTR1B 18 46 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880933537 GI On-Demand Anodyne HTR1F 76 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880933537 GI On-Demand Anodyne CCR2 22 50 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880933537 GI On-Demand Anodyne LIMK2 19 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933539 GH On-Demand Anodyne ACACB 15 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933539 GH On-Demand Anodyne CACNA1I 45 34 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933540 GH On-Demand Anodyne ACACB 15 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)OC(C)(C)C)C1 ZINC000880933540 GH On-Demand Anodyne CACNA1I 45 34 CN1CCC(CNC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933542 DE On-Demand Anodyne CCR3 67 40 CN1CCC(CNC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933542 DE On-Demand Anodyne CACNA1I 65 38 CN(C)c1ccc(F)cc1NC(=O)N(CCO)CCc1ccccc1 ZINC000880933561 EF On-Demand Anodyne SOAT1 24 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2C(N)=O)CC1 ZINC000880933566 GD On-Demand Anodyne FAAH 20 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2C(N)=O)CC1 ZINC000880933566 GD On-Demand Anodyne RBP4 23 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880933576 GF On-Demand Anodyne CCR3 24 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880933576 GF On-Demand Anodyne EPHX2 49 56 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C[C@@H]2CCCO2)CC1 ZINC000880933578 FE On-Demand Anodyne CCR3 21 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(C[C@H]2CCCO2)CC1 ZINC000880933579 FE On-Demand Anodyne CCR3 21 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCSCC1 ZINC000880933580 CF On-Demand Anodyne EPHX2 33 40 Cc1noc(C2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)n1 ZINC000880933588 EF On-Demand Anodyne SMO 39 45 Cc1noc(C2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)n1 ZINC000880933588 EF On-Demand Anodyne ETHR 55 39 C=C(C)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933601 EG On-Demand Mild CCR3 53 43 C=C(C)CN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933601 EG On-Demand Mild EPHX2 33 41 COCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933604 EE On-Demand Anodyne DRD2 17 45 COCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933604 EE On-Demand Anodyne CCR3 70 52 COCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933604 EE On-Demand Anodyne MCHR1 27 42 CCOCCN(CC)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933605 CF On-Demand Anodyne SOAT1 18 41 CN(C)c1ccc(F)cc1NC(=O)NCC(=O)NC1CCCC1 ZINC000880933610 DE On-Demand Anodyne EPHX2 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2cnn(C)c2)CC1 ZINC000880933614 FD On-Demand Anodyne PLA2G7 54 34 CN(C)c1ccc(F)cc1NC(=O)NCCCCC#N ZINC000880933615 CF On-Demand Mild CCR3 15 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)(F)F)CC1 ZINC000880933620 FG On-Demand Anodyne CCR3 51 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)(F)F)CC1 ZINC000880933620 FG On-Demand Anodyne EPHX2 45 39 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)(F)F)CC1 ZINC000880933620 FG On-Demand Anodyne CXCR3 22 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC(F)(F)F)CC1 ZINC000880933620 FG On-Demand Anodyne HPGDS 38 45 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](N(C)C)C1 ZINC000880933621 CE On-Demand Anodyne RBP4 42 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](N(C)C)C1 ZINC000880933621 CE On-Demand Anodyne MCHR1 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](N(C)C)C1 ZINC000880933622 CE On-Demand Anodyne RBP4 42 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](N(C)C)C1 ZINC000880933622 CE On-Demand Anodyne MCHR1 18 40 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCCC[C@H]2C1 ZINC000880933627 DF On-Demand Anodyne HRH3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCCC[C@H]2C1 ZINC000880933627 DF On-Demand Anodyne L3MBTL3 59 37 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCCC[C@@H]2C1 ZINC000880933628 DF On-Demand Anodyne HRH3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN2CCCC[C@@H]2C1 ZINC000880933628 DF On-Demand Anodyne L3MBTL3 59 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)NC2CCCCC2)CC1 ZINC000880933632 GH On-Demand Anodyne EPHX2 36 51 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000880933637 FD On-Demand Anodyne CCR3 36 45 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000880933637 FD On-Demand Anodyne EPHX2 30 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000880933638 FD On-Demand Anodyne CCR3 36 45 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000880933638 FD On-Demand Anodyne EPHX2 30 41 CC[C@@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933644 CG On-Demand Anodyne ACKR3 45 32 CC[C@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933645 CG On-Demand Anodyne ACKR3 45 32 COC[C@H](NC(=O)Nc1cc(F)ccc1N(C)C)c1ccccc1 ZINC000880933657 EG On-Demand Anodyne TACR3 16 43 COC[C@@H](NC(=O)Nc1cc(F)ccc1N(C)C)c1ccccc1 ZINC000880933658 EG On-Demand Anodyne TACR3 16 43 COc1ccc2c(c1)CN(C(=O)Nc1cc(F)ccc1N(C)C)CC2 ZINC000880933663 EG On-Demand Anodyne HDAC6 32 45 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CCN2CCOCC2)c1 ZINC000880933669 GE On-Demand Anodyne HTR2A 24 45 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CCN2CCOCC2)c1 ZINC000880933669 GE On-Demand Anodyne PIK3CA 18 42 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CCN2CCOCC2)c1 ZINC000880933669 GE On-Demand Anodyne MTOR 29 42 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CCN2CCOCC2)c1 ZINC000880933669 GE On-Demand Anodyne EPHX2 26 47 CCCN(CC)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880933673 CG On-Demand Anodyne SOAT1 22 40 COC[C@@H]1CCCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933679 DF On-Demand Anodyne CCR3 49 44 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCN(S(C)(=O)=O)CC1 ZINC000880933698 GC On-Demand Anodyne CCR3 49 43 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCN(S(C)(=O)=O)CC1 ZINC000880933698 GC On-Demand Anodyne PLD2 42 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CNC(=O)OC(C)(C)C)CC1 ZINC000880933699 GH On-Demand Anodyne ACACB 15 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CNC(=O)OC(C)(C)C)CC1 ZINC000880933699 GH On-Demand Anodyne CACNA1I 59 34 CN1CCN(c2ncccc2CNC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933701 GE On-Demand Anodyne TRPV1 27 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)C1CC1 ZINC000880933710 CD On-Demand Anodyne PYGL 16 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)C1CC1 ZINC000880933711 CD On-Demand Anodyne PYGL 16 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)Nc2ccccc2)CC1 ZINC000880933723 GH On-Demand Anodyne CCR3 56 51 CN(C)c1ccc(F)cc1NC(=O)N1CCC(NC(=O)Nc2ccccc2)CC1 ZINC000880933723 GH On-Demand Anodyne EPHX2 59 46 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(CS(C)(=O)=O)c1 ZINC000880933724 GF On-Demand Anodyne ROCK2 16 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](N2CCCCC2)C1 ZINC000880933758 EF On-Demand Anodyne L3MBTL3 92 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](N2CCCCC2)C1 ZINC000880933759 EF On-Demand Anodyne L3MBTL3 92 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OC2CCCC2)CC1 ZINC000880933778 EH On-Demand Anodyne SCD1 17 40 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(N2CCCS2(=O)=O)cc1 ZINC000880933780 GG On-Demand Anodyne CDK1 17 43 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCSCC1 ZINC000880933790 EE On-Demand Anodyne DRD4 40 31 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCSCC1 ZINC000880933790 EE On-Demand Anodyne CCR3 45 39 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCSCC1 ZINC000880933790 EE On-Demand Anodyne UTS2R 16 42 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCSCC1 ZINC000880933790 EE On-Demand Anodyne PLD2 51 34 CCOC[C@H]1CCCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933806 DG On-Demand Anodyne CCR3 31 43 CC(=O)Nc1cccc(OCCNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933808 FG On-Demand Anodyne HRH2 25 42 CC(=O)Nc1cccc(OCCNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933808 FG On-Demand Anodyne MTNR1A 26 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933808 FG On-Demand Anodyne MTNR1B 24 45 CC(=O)Nc1cccc(OCCNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933808 FG On-Demand Anodyne EPHX2 19 42 CN(C)c1ccc(F)cc1NC(=O)N(CCCO)CC(C)(C)C ZINC000880933825 EG On-Demand Anodyne SOAT1 21 45 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CO ZINC000880933830 CD On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CO ZINC000880933831 CD On-Demand Anodyne ACKR3 45 32 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933846 FH On-Demand Anodyne KCNK3 47 36 CO[C@@H](C)C(=O)Nc1cccc(NC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880933846 FH On-Demand Anodyne KCNK9 46 36 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880933848 EE On-Demand Anodyne CCR3 48 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1[C@@H]1CCCN1C ZINC000880933871 EF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1[C@H]1CCCN1C ZINC000880933872 EF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1[C@@H]1CCCN1C ZINC000880933873 EF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1[C@H]1CCCN1C ZINC000880933874 EF On-Demand Anodyne ACKR3 45 32 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cc(F)ccc1N(C)C)CC2 ZINC000880933878 EF On-Demand Anodyne CACNA1H 53 41 COC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933884 EE On-Demand Anodyne CCR3 28 43 COC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933884 EE On-Demand Anodyne NPY5R 16 43 COC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933884 EE On-Demand Anodyne EPHX2 51 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)C(C)(C)C)C1 ZINC000880933890 GG On-Demand Anodyne CACNA1I 52 34 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)C(C)(C)C)C1 ZINC000880933891 GG On-Demand Anodyne CACNA1I 52 34 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(CC#N)CC1 ZINC000880933892 DE On-Demand Mild CCR3 53 43 CN(C)c1ccc(F)cc1NC(=O)NCC(=O)NC1CCCCC1 ZINC000880933896 EE On-Demand Anodyne EPHX2 17 41 COCCCOC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933932 FF On-Demand Anodyne SCD1 17 41 COCCn1nc(C)c(NC(=O)Nc2cc(F)ccc2N(C)C)c1C ZINC000880933941 EF On-Demand Anodyne P2RX7 17 49 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933955 FD On-Demand Anodyne CCR1 32 40 CCOC[C@H](O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880933955 FD On-Demand Anodyne ABCB1 28 40 C[C@@H](CCN(C)C)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880933969 CE On-Demand Anodyne UTS2 59 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CCCO ZINC000880933978 DF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CCCO ZINC000880933979 DF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Cc2cnn(C)c2)C1 ZINC000880933997 EF On-Demand Anodyne CCR3 114 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Cc2cnn(C)c2)C1 ZINC000880933998 EF On-Demand Anodyne CCR3 114 37 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CCO)c1ccccc1 ZINC000880934055 EG On-Demand Anodyne UTS2 54 38 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCC[C@H]1CO ZINC000880934103 DF On-Demand Anodyne CCR3 43 47 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCC[C@@H]1CO ZINC000880934104 DF On-Demand Anodyne CCR3 43 47 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCC[C@H]1CO ZINC000880934105 DF On-Demand Anodyne CCR3 43 47 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCC[C@@H]1CO ZINC000880934106 DF On-Demand Anodyne CCR3 43 47 CN(C)c1ccc(F)cc1NC(=O)NC1C[C@@H]2CCC[C@H](C1)N2C ZINC000880934107 EG On-Demand Anodyne HTR3A 32 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OCC2CC2)CC1 ZINC000880934131 EG On-Demand Anodyne SCD1 17 40 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(Cc2cnn(C)c2)CC1 ZINC000880934138 FE On-Demand Anodyne PLA2G7 46 34 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(Cc2cnn(C)c2)CC1 ZINC000880934138 FE On-Demand Anodyne CCR3 17 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(N)=O)(c2ccccc2)CC1 ZINC000880934139 GF On-Demand Anodyne CACNA1H 52 34 Cc1ccccc1[C@H](CO)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934140 EG On-Demand Anodyne CTSA 60 38 Cc1ccccc1[C@@H](CO)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934141 EG On-Demand Anodyne CTSA 60 38 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3cc(F)ccc3N(C)C)C2)nn1 ZINC000880934143 FF On-Demand Anodyne CCR3 51 30 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](CO)c1ccccc1 ZINC000880934152 EF On-Demand Anodyne SOAT1 22 40 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](CO)c1ccccc1 ZINC000880934153 EF On-Demand Anodyne SOAT1 22 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2ncc[nH]2)CC1 ZINC000880934159 EG On-Demand Anodyne HTR2B 19 44 CN(C)C(=O)Nc1cccc(CNC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880934160 FG On-Demand Anodyne ROCK2 21 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(F)(F)F)CC1 ZINC000880934164 EH On-Demand Anodyne RBP4 41 37 C[C@H]1C[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)CCN1C ZINC000880934201 DE On-Demand Anodyne CCR3 23 41 CCOC[C@H]1CCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880934248 DF On-Demand Anodyne CCR3 24 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCCC2)C1 ZINC000880934257 DH On-Demand Anodyne EPHX2 26 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1C(=O)NCc1ccco1 ZINC000880934266 FF On-Demand Anodyne P2RX7 19 46 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1C(=O)NCc1ccco1 ZINC000880934267 FF On-Demand Anodyne P2RX7 19 46 CCCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934278 EG On-Demand Anodyne DRD2 19 40 CCCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934278 EG On-Demand Anodyne SIGMAR1 15 40 CCCCN1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934278 EG On-Demand Anodyne CCR3 86 44 CN(C)c1ccc(F)cc1NC(=O)NCCCC(F)(F)F ZINC000880934293 DG On-Demand Anodyne CCR3 15 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCc2c(O)cccc21 ZINC000880934296 EG On-Demand Anodyne TRPV1 19 46 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCc2c(O)cccc21 ZINC000880934297 EG On-Demand Anodyne TRPV1 19 46 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)c2ccccc2)CC1 ZINC000880934300 GH On-Demand Anodyne GRIN2B 51 36 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)c2ccccc2)CC1 ZINC000880934300 GH On-Demand Anodyne CCR3 74 39 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)c2ccccc2)CC1 ZINC000880934300 GH On-Demand Anodyne EPHX2 18 50 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)c2ccccc2)CC1 ZINC000880934300 GH On-Demand Anodyne CACNA1I 61 36 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)c2ccccc2)CC1 ZINC000880934300 GH On-Demand Anodyne ACKR3 43 30 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C2CCCC2)CC1 ZINC000880934316 EG On-Demand Anodyne CCR3 29 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C2CCCC2)CC1 ZINC000880934316 EG On-Demand Anodyne EPHX2 36 41 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CC2CC2)c1 ZINC000880934320 DG On-Demand Anodyne CCR3 49 34 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CC2CC2)c1 ZINC000880934320 DG On-Demand Anodyne PANC 52 38 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](N2CCOCC2)C1 ZINC000880934321 ED On-Demand Anodyne L3MBTL3 41 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](N2CCOCC2)C1 ZINC000880934322 ED On-Demand Anodyne L3MBTL3 41 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CO)C1 ZINC000880934323 CD On-Demand Anodyne CCR3 32 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CO)C1 ZINC000880934324 CD On-Demand Anodyne CCR3 32 41 CN(C)c1ccc(F)cc1NC(=O)N1CCOC2(CCCCC2)C1 ZINC000880934327 EG On-Demand Anodyne EPHX2 15 43 CC[C@@H](NC(=O)Nc1cc(F)ccc1N(C)C)c1nnc2n1CCCCC2 ZINC000880934337 FG On-Demand Anodyne CCR3 43 31 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880934345 FE On-Demand Anodyne CCR3 85 45 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880934345 FE On-Demand Anodyne PLD1 42 39 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCC(N(C)C)CC1 ZINC000880934345 FE On-Demand Anodyne PLD2 58 39 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC[C@H]1CO ZINC000880934350 FE On-Demand Anodyne CCR3 52 41 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC[C@H]1CO ZINC000880934350 FE On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC[C@@H]1CO ZINC000880934351 FE On-Demand Anodyne CCR3 52 41 CN(C)c1ccc(F)cc1NC(=O)NCCCCN1CCC[C@@H]1CO ZINC000880934351 FE On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N(CCC#N)CCN1CCOCC1 ZINC000880934368 FD On-Demand Mild CASR 60 45 CCC1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934371 DF On-Demand Anodyne CACNA1H 45 37 CCC1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934371 DF On-Demand Anodyne S1PR2 31 45 C[C@H](O)CN1CCC(CN(C)C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880934374 FE On-Demand Anodyne CCR3 34 42 CN(Cc1nccs1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880934395 DG On-Demand Anodyne MAP1 43 36 CN(C)c1ccc(F)cc1NC(=O)N1CC(Cc2ccccc2)C1 ZINC000880934424 EH On-Demand Anodyne CCR3 73 42 CN(C)c1ccc(F)cc1NC(=O)N1CC(Cc2ccccc2)C1 ZINC000880934424 EH On-Demand Anodyne RBP4 53 39 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(C2CCCC2)CC1 ZINC000880934426 EG On-Demand Anodyne HRH3 26 45 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(C2CCCC2)CC1 ZINC000880934426 EG On-Demand Anodyne L3MBTL3 55 35 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CC(=O)N2CCOCC2)c1 ZINC000880934430 GD On-Demand Anodyne PIK3CA 16 41 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(CC(=O)N2CCOCC2)c1 ZINC000880934430 GD On-Demand Anodyne MTOR 29 41 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934435 EG On-Demand Anodyne TRPV1 16 41 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(N2CCC(O)CC2)c(C#N)c1 ZINC000880934459 GG On-Demand Mild NPY2R 46 39 CN(C)c1ccc(F)cc1NC(=O)N1CCn2c(nnc2-c2ccccc2)C1 ZINC000880934461 GG On-Demand Anodyne P2RX7 31 56 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CN2CCCC2)C1 ZINC000880934470 EF On-Demand Anodyne CCR3 79 46 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CN2CCCC2)C1 ZINC000880934471 EF On-Demand Anodyne CCR3 79 46 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880934474 FF On-Demand Anodyne CCR3 51 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880934474 FF On-Demand Anodyne CXCR3 16 42 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880934475 FF On-Demand Anodyne CCR3 51 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880934475 FF On-Demand Anodyne CXCR3 16 42 C[C@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934499 FD On-Demand Anodyne CCR3 22 40 C[C@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934501 FD On-Demand Anodyne CCR3 22 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)c2ccccc2)C1 ZINC000880934507 GH On-Demand Anodyne CCR3 59 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)c2ccccc2)C1 ZINC000880934507 GH On-Demand Anodyne PREP 23 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)c2ccccc2)C1 ZINC000880934507 GH On-Demand Anodyne CACNA1I 64 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CNC(=O)c2ccccc2)C1 ZINC000880934507 GH On-Demand Anodyne ACKR3 49 30 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)c2ccccc2)C1 ZINC000880934508 GH On-Demand Anodyne CCR3 59 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)c2ccccc2)C1 ZINC000880934508 GH On-Demand Anodyne PREP 23 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)c2ccccc2)C1 ZINC000880934508 GH On-Demand Anodyne CACNA1I 64 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CNC(=O)c2ccccc2)C1 ZINC000880934508 GH On-Demand Anodyne ACKR3 49 30 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880934582 DD On-Demand Anodyne LGMN 64 35 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880934612 FF On-Demand Anodyne CCR3 19 43 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880934613 FF On-Demand Anodyne CCR3 19 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](Cn2ccnn2)C1 ZINC000880934617 EE On-Demand Anodyne CCR3 54 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](Cn2ccnn2)C1 ZINC000880934618 EE On-Demand Anodyne CCR3 54 33 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CCC#N)c1ccccc1 ZINC000880934632 EI On-Demand Mild UTS2 47 36 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CCC#N)c1ccccc1 ZINC000880934633 EI On-Demand Mild UTS2 47 36 CN(C)c1ccc(F)cc1NC(=O)NCCOc1ncccc1F ZINC000880934644 EF On-Demand Anodyne P2RY1 32 45 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880934659 EH On-Demand Anodyne NPY5R 21 50 CN(C)c1ccc(F)cc1NC(=O)N(CCCO)Cc1ccccc1 ZINC000880934699 EG On-Demand Anodyne SOAT1 26 46 COc1cccc([C@H](CO)NC(=O)Nc2cc(F)ccc2N(C)C)c1 ZINC000880934774 EF On-Demand Anodyne ROCK2 15 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CCCO)c1ccccc1 ZINC000880934797 EH On-Demand Anodyne UTS2 50 36 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CCCO)c1ccccc1 ZINC000880934798 EH On-Demand Anodyne UTS2 50 36 CN(C)c1ccc(F)cc1NC(=O)NCCC[S@](C)=O ZINC000880934802 DD On-Demand Anodyne CCR3 21 40 CN(C)c1ccc(F)cc1NC(=O)NCCC[S@@](C)=O ZINC000880934803 DD On-Demand Anodyne CCR3 21 40 C[C@H]1c2ccccc2CN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880934808 DI On-Demand Anodyne TRPM8 20 43 CN(C)c1ccc(F)cc1NC(=O)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880934813 FF On-Demand Anodyne P2RX7 24 41 CN(Cc1ccc(S(C)(=O)=O)cc1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880934863 GF On-Demand Anodyne PTGS2 23 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Nc2cccnn2)CC1 ZINC000880934872 FF On-Demand Anodyne FAAH 23 45 CC[C@@H]1CN(S(C)(=O)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934899 GE On-Demand Anodyne CCR3 44 41 CC[C@@H]1CN(S(C)(=O)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880934900 GE On-Demand Anodyne CCR3 44 41 CN1C(=O)N[C@]2(CCN(C(=O)Nc3cc(F)ccc3N(C)C)C2)C1=O ZINC000880934910 ED On-Demand Anodyne CACNA1H 35 40 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3cc(F)ccc3N(C)C)C2)C1=O ZINC000880934911 ED On-Demand Anodyne CACNA1H 35 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880934929 FE On-Demand Anodyne EPHX2 41 37 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880934930 FE On-Demand Anodyne EPHX2 41 37 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880934931 FE On-Demand Anodyne EPHX2 41 37 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880934932 FE On-Demand Anodyne EPHX2 41 37 CN(C)c1ccc(F)cc1NC(=O)N[C@H](C(N)=O)C(C)(C)C ZINC000880934958 DD On-Demand Anodyne FCER2 15 42 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(c2ccccn2)C1 ZINC000880934967 EF On-Demand Anodyne CCR3 21 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(c2ccccn2)C1 ZINC000880934968 EF On-Demand Anodyne CCR3 21 44 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880934981 GG On-Demand Anodyne CCR3 44 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CC(=O)N(Cc2ccccc2)C1 ZINC000880934982 GG On-Demand Anodyne CCR3 44 35 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880934985 GF On-Demand Anodyne SLC18A3 41 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880934985 GF On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880934986 GF On-Demand Anodyne SLC18A3 41 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880934986 GF On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880934987 GF On-Demand Anodyne SLC18A3 41 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880934987 GF On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880934988 GF On-Demand Anodyne SLC18A3 41 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880934988 GF On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880934992 FH On-Demand Anodyne GRIN2B 51 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880934992 FH On-Demand Anodyne CCR3 68 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880934992 FH On-Demand Anodyne CHRNA7 52 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Cc2cccnc2)CC1 ZINC000880934992 FH On-Demand Anodyne C3AR1 42 42 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880934998 FD On-Demand Anodyne CCR3 64 40 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880934999 FD On-Demand Anodyne CCR3 64 40 Cc1noc(C)c1CCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935009 EG On-Demand Anodyne P2RX7 15 48 CC[C@H]1CCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935025 CG On-Demand Anodyne CCR3 32 41 CNC(=O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935087 EC On-Demand Anodyne SLC27A1 41 31 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](C2CC2)C1 ZINC000880935151 CG On-Demand Anodyne RBP4 53 39 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](C2CC2)C1 ZINC000880935152 CG On-Demand Anodyne RBP4 53 39 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)CN1CCOCC1 ZINC000880935153 EC On-Demand Anodyne KIT 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)CN1CCOCC1 ZINC000880935153 EC On-Demand Anodyne PHKG1 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)CN1CCOCC1 ZINC000880935153 EC On-Demand Anodyne CAMK1G 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)CN1CCOCC1 ZINC000880935153 EC On-Demand Anodyne CIT 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H](O)CN1CCOCC1 ZINC000880935153 EC On-Demand Anodyne SRMS 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)CN1CCOCC1 ZINC000880935154 EC On-Demand Anodyne KIT 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)CN1CCOCC1 ZINC000880935154 EC On-Demand Anodyne PHKG1 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)CN1CCOCC1 ZINC000880935154 EC On-Demand Anodyne CAMK1G 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)CN1CCOCC1 ZINC000880935154 EC On-Demand Anodyne CIT 15 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H](O)CN1CCOCC1 ZINC000880935154 EC On-Demand Anodyne SRMS 15 46 CN(C)c1ccc(F)cc1NC(=O)N1CCOC2(CCOCC2)C1 ZINC000880935158 EE On-Demand Anodyne EPHX2 15 43 CN(C)c1ccc(F)cc1NC(=O)NCC1CN(C(=O)OC(C)(C)C)C1 ZINC000880935165 FF On-Demand Anodyne CACNA1I 49 33 CN(C)c1ccc(F)cc1NC(=O)NCC1CN(C(=O)OC(C)(C)C)C1 ZINC000880935165 FF On-Demand Anodyne GPR119 18 40 COc1ccc([C@H](CCO)NC(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880935191 FG On-Demand Anodyne UTS2 57 40 COc1ccc([C@@H](CCO)NC(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880935192 FG On-Demand Anodyne UTS2 57 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C)(O)CC1 ZINC000880935210 CE On-Demand Anodyne CACNA1H 57 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2ccccn2)CC1 ZINC000880935229 EH On-Demand Anodyne RBP4 55 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C#N)(c2ccccn2)CC1 ZINC000880935275 FG On-Demand Mild CACNA1H 47 38 CCCN(CCCN(C)C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880935280 DG On-Demand Anodyne SOAT1 27 42 CC1CN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935284 CE On-Demand Anodyne RBP4 52 39 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne HTR1A 34 45 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne ADRA1D 30 42 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne HTR1D 15 46 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne HTR1B 17 46 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne ADRA1A 27 42 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne PDGFRB 45 43 COc1cnccc1N1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935313 FF On-Demand Anodyne RBP4 20 43 CN(C)c1ccc(F)cc1NC(=O)NCCCCCO ZINC000880935330 CE On-Demand Anodyne CCR3 17 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(F)(F)CC1 ZINC000880935340 DG On-Demand Anodyne CACNA1H 55 40 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@@H](O)C1 ZINC000880935345 GF On-Demand Anodyne OPRK1 21 42 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@@H](O)C1 ZINC000880935345 GF On-Demand Anodyne CCR3 70 43 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@@H](O)C1 ZINC000880935345 GF On-Demand Anodyne MCHR1 21 43 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@H](O)C1 ZINC000880935346 GF On-Demand Anodyne OPRK1 21 42 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@H](O)C1 ZINC000880935346 GF On-Demand Anodyne CCR3 70 43 CN(C)c1ccc(F)cc1NC(=O)NCc1ccccc1CN1CC[C@H](O)C1 ZINC000880935346 GF On-Demand Anodyne MCHR1 21 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)CNC(=O)O2 ZINC000880935395 ED On-Demand Anodyne CACNA1H 49 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)CNC(=O)O2 ZINC000880935395 ED On-Demand Anodyne TRPM8 23 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(C(F)F)CC1 ZINC000880935396 EF On-Demand Anodyne CACNA1H 46 38 COC1(C)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935401 DF On-Demand Anodyne CACNA1H 43 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880935406 FE On-Demand Anodyne CCR3 27 46 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CN2CCOCC2)C1 ZINC000880935407 FE On-Demand Anodyne CCR3 27 46 COC[C@@H]1CCCCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935418 DG On-Demand Anodyne CCR3 34 42 CN(C)c1ccc(F)cc1NC(=O)N1CCOC2(CCOCC2)CC1 ZINC000880935441 FF On-Demand Anodyne TRPM8 16 43 CC(=O)N1CCC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935491 EE On-Demand Anodyne CCR3 102 40 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935492 EE On-Demand Anodyne CCR3 102 40 CN(C)c1ccc(F)cc1NC(=O)N(CCCO)Cc1ccccn1 ZINC000880935494 EF On-Demand Anodyne SOAT1 26 40 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)C(F)(F)F)CC1 ZINC000880935498 GF On-Demand Anodyne CCR3 44 38 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)C(F)(F)F)CC1 ZINC000880935498 GF On-Demand Anodyne EPHX2 18 45 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C(=O)C(F)(F)F)CC1 ZINC000880935498 GF On-Demand Anodyne CACNA1I 62 36 CN(C)c1ccc(F)cc1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880935521 FD On-Demand Anodyne CASR 64 47 CN(C)c1ccc(F)cc1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880935521 FD On-Demand Anodyne EPHX2 18 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880935534 GD On-Demand Anodyne CCR3 15 43 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880935534 GD On-Demand Anodyne EPHX2 39 52 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@](C)(O)CC1 ZINC000880935554 DF On-Demand Anodyne CACNA1H 41 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@](C)(O)CC1 ZINC000880935556 DF On-Demand Anodyne CACNA1H 41 36 COC(=O)C1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880935566 ED On-Demand Anodyne CACNA1H 45 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](c2ncc(C(F)(F)F)[nH]2)C1 ZINC000880935579 GI On-Demand Anodyne RBP4 56 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](c2ncc(C(F)(F)F)[nH]2)C1 ZINC000880935581 GI On-Demand Anodyne RBP4 56 38 CN(C)c1ccc(F)cc1NC(=O)NCCCF ZINC000880935629 CE On-Demand Anodyne CCR3 18 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935635 GG On-Demand Anodyne CCR3 49 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935638 GG On-Demand Anodyne CCR3 49 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2cccnc2)CC1 ZINC000880935642 EH On-Demand Anodyne CACNA1H 42 33 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880935658 EG On-Demand Anodyne CCR3 119 38 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Cc2ccncc2)C1 ZINC000880935659 EG On-Demand Anodyne CCR3 119 38 COC[C@@H](C)n1ccc(NC(=O)Nc2cc(F)ccc2N(C)C)n1 ZINC000880935666 EF On-Demand Anodyne GCK 21 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880935675 GH On-Demand Anodyne S1PR2 30 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCOCC1 ZINC000880935685 CF On-Demand Anodyne EPHX2 20 43 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCOCC1 ZINC000880935686 CF On-Demand Anodyne EPHX2 20 43 CN(C)c1ccc(F)cc1NC(=O)NCCCOCCO ZINC000880935688 CD On-Demand Anodyne CCR3 21 40 CCCCN(CCCO)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880935700 DF On-Demand Anodyne SOAT1 30 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)Cc1ccc(O)cc1 ZINC000880935717 EE On-Demand Anodyne YARS 74 33 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(CCc3ccccc3)c(S)nc2c1 ZINC000880935726 IH On-Demand Anodyne HDAC8 15 49 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(CCc3ccccc3)c(S)nc2c1 ZINC000880935726 IH On-Demand Anodyne HDAC6 19 49 CN1CC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935731 CD On-Demand Anodyne CCR3 71 38 CN1CC[C@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935731 CD On-Demand Anodyne CACNA1I 67 35 CN1CC[C@@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935732 CD On-Demand Anodyne CCR3 71 38 CN1CC[C@@H](CNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880935732 CD On-Demand Anodyne CACNA1I 67 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCO2)CC1 ZINC000880935746 DF On-Demand Anodyne TRPM8 23 44 CCn1cccc(CNC(=O)Nc2cc(F)ccc2N(C)C)c1=O ZINC000880935772 EE On-Demand Anodyne P2RX7 45 40 CN(C)c1ccc(F)cc1NC(=O)NCC1(N2CCOCC2)CC1 ZINC000880935811 ED On-Demand Anodyne HCN1 56 35 CN(C)c1ccc(F)cc1NC(=O)NCC1(N2CCOCC2)CC1 ZINC000880935811 ED On-Demand Anodyne HCN4 47 32 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2nc(N)ns2)CC1 ZINC000880935851 FD On-Demand Anodyne FAAH 15 47 CN1C(=O)NC2(CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)C1=O ZINC000880935872 FD On-Demand Anodyne CACNA1H 53 41 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935876 FF On-Demand Anodyne CCR3 72 43 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935876 FF On-Demand Anodyne EPHX2 15 40 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935879 FF On-Demand Anodyne CCR3 72 43 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935879 FF On-Demand Anodyne EPHX2 15 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935881 FF On-Demand Anodyne CCR3 72 43 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935881 FF On-Demand Anodyne EPHX2 15 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935883 FF On-Demand Anodyne CCR3 72 43 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880935883 FF On-Demand Anodyne EPHX2 15 40 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCOCC1 ZINC000880935900 DD On-Demand Anodyne EPHX2 22 48 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCCOCC1 ZINC000880935900 DD On-Demand Anodyne PLD2 49 31 CN(C)c1ccc(F)cc1NC(=O)N1CCOC2(CCC2)C1 ZINC000880935921 DF On-Demand Anodyne EPHX2 15 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](NC(=O)NC2CC2)C1 ZINC000880935924 ED On-Demand Anodyne CCR3 26 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](NC(=O)NC2CC2)C1 ZINC000880935924 ED On-Demand Anodyne EPHX2 40 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCC2)C1 ZINC000880935925 CG On-Demand Anodyne EPHX2 26 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](NC(=O)NC2CC2)C1 ZINC000880935926 ED On-Demand Anodyne CCR3 26 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](NC(=O)NC2CC2)C1 ZINC000880935926 ED On-Demand Anodyne EPHX2 40 36 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880935951 FF On-Demand Anodyne CCR3 28 42 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880935951 FF On-Demand Anodyne EPHX2 38 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880935953 FF On-Demand Anodyne CCR3 28 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880935953 FF On-Demand Anodyne EPHX2 38 41 CN1CCC(N2CCC(NC(=O)Nc3cc(F)ccc3N(C)C)CC2)CC1 ZINC000880935956 GF On-Demand Anodyne SLC6A5 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(N2CC=CC2)CC1 ZINC000880936004 EF On-Demand Anodyne L3MBTL3 47 34 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(CCS(C)(=O)=O)cc1 ZINC000880936019 GG On-Demand Anodyne CA12 20 40 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(CCS(C)(=O)=O)cc1 ZINC000880936019 GG On-Demand Anodyne CA9 20 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@H]1CCO ZINC000880936039 DF On-Demand Anodyne CCR3 38 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H]1CCO ZINC000880936040 DF On-Demand Anodyne CCR3 38 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@H]1CCO ZINC000880936041 DF On-Demand Anodyne CCR3 38 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@@H]1CCO ZINC000880936042 DF On-Demand Anodyne CCR3 38 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880936063 GH On-Demand Anodyne EPHX2 19 40 COC1(CO)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936076 ED On-Demand Anodyne CACNA1H 48 35 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)CC1CCC1 ZINC000880936091 DF On-Demand Anodyne CCR3 56 34 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)CC1CCC1 ZINC000880936092 DF On-Demand Anodyne CCR3 56 34 CN(C)c1ccc(F)cc1NC(=O)NCCCCO ZINC000880936095 CD On-Demand Anodyne CCR3 19 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCC2)CC1 ZINC000880936116 DH On-Demand Anodyne CACNA1H 45 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Oc2ncccc2F)CC1 ZINC000880936131 GH On-Demand Anodyne SCD1 23 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880936144 GI On-Demand Anodyne CACNA1H 59 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880936144 GI On-Demand Anodyne NPY5R 31 41 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1S(C)(=O)=O ZINC000880936163 FD On-Demand Anodyne CCR3 47 36 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880936168 DE On-Demand Anodyne CCR3 33 45 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880936168 DE On-Demand Anodyne EPHX2 37 47 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880936169 DE On-Demand Anodyne CCR3 33 45 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880936169 DE On-Demand Anodyne EPHX2 37 47 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CC[C@@H](O)CC1 ZINC000880936177 CE On-Demand Anodyne EPHX2 37 40 CN(C)c1ccc(F)cc1NC(=O)N1CCOC2(CCCC2)C1 ZINC000880936179 DG On-Demand Anodyne EPHX2 15 43 COCCC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936189 FE On-Demand Anodyne CCR3 23 47 COCCC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936189 FE On-Demand Anodyne EPHX2 43 44 COCCC(=O)N1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936189 FE On-Demand Anodyne CCR8 42 37 CN(C)c1ccc(F)cc1NC(=O)N(C)C1CCN(S(C)(=O)=O)CC1 ZINC000880936197 FD On-Demand Anodyne NPY5R 15 62 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OCCO)CC1 ZINC000880936199 ED On-Demand Anodyne SCD1 19 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H]1Cc1ccccc1 ZINC000880936204 EH On-Demand Anodyne CCR3 69 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H]1Cc1ccccc1 ZINC000880936205 EH On-Demand Anodyne CCR3 69 41 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(Cc2nnc3n2CCC3)cc1 ZINC000880936247 GH On-Demand Anodyne CCR3 56 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880936249 FG On-Demand Anodyne EPHX2 18 52 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880936250 FG On-Demand Anodyne EPHX2 18 52 CN(C)c1ccc(F)cc1NC(=O)N1CC(C2CCCC2)C1 ZINC000880936308 DH On-Demand Anodyne RBP4 46 39 CN(C)c1ccc(F)cc1NC(=O)NCC1(c2ccccn2)CCC1 ZINC000880936340 EH On-Demand Anodyne NMBR 44 40 CN(C)c1ccc(F)cc1NC(=O)NCC1(c2ccccn2)CCC1 ZINC000880936340 EH On-Demand Anodyne GRPR 23 40 CN(C)c1ccc(F)cc1NC(=O)Nc1cccc(C(C)(C)O)c1 ZINC000880936350 EH On-Demand Anodyne RIPK1 40 33 CN(C)c1ccc(F)cc1NC(=O)Nc1cccc(C(C)(C)O)c1 ZINC000880936350 EH On-Demand Anodyne IMDH_CRYPV 40 31 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880936351 GG On-Demand Anodyne CCR3 56 52 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880936351 GG On-Demand Anodyne EPHX2 45 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880936352 GG On-Demand Anodyne CCR3 56 52 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880936352 GG On-Demand Anodyne EPHX2 45 43 CN(C)c1ccc(F)cc1NC(=O)Nc1cnn(Cc2nnc3n2CCCC3)c1 ZINC000880936358 GF On-Demand Anodyne PANC 54 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880936359 GF On-Demand Anodyne CACNA1I 61 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880936363 EG On-Demand Anodyne RBP4 55 36 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880936364 EG On-Demand Anodyne RBP4 55 36 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C2CC2)CC1 ZINC000880936388 EF On-Demand Anodyne CCR3 59 38 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C2CC2)CC1 ZINC000880936388 EF On-Demand Anodyne CACNA1I 61 35 CCOC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880936418 FD On-Demand Anodyne HLA-DRB1 45 33 CCOC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880936419 FD On-Demand Anodyne HLA-DRB1 45 33 CN(C)c1ccc(F)cc1NC(=O)N1CCc2ccccc2[C@H]1CO ZINC000880936460 EG On-Demand Anodyne TRPM8 41 43 CN(C)c1ccc(F)cc1NC(=O)N1CCc2ccccc2[C@@H]1CO ZINC000880936461 EG On-Demand Anodyne TRPM8 41 43 CC(=O)OC1CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936501 DE On-Demand Anodyne SCD1 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCC[C@H]1C(N)=O ZINC000880936530 DE On-Demand Anodyne CCR3 25 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCC[C@@H]1C(N)=O ZINC000880936531 DE On-Demand Anodyne CCR3 25 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCC[C@@H]1C(N)=O ZINC000880936532 DE On-Demand Anodyne CCR3 25 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCC[C@H]1C(N)=O ZINC000880936533 DE On-Demand Anodyne CCR3 25 41 COCC1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936636 ED On-Demand Anodyne CACNA1H 53 36 COCC1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936636 ED On-Demand Anodyne S1PR2 31 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CS(N)(=O)=O)C1 ZINC000880936647 FD On-Demand Anodyne CCR3 53 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CS(N)(=O)=O)C1 ZINC000880936648 FD On-Demand Anodyne CCR3 53 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CN1CCOCC1 ZINC000880936653 FE On-Demand Anodyne CCR3 15 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CN1CCOCC1 ZINC000880936654 FE On-Demand Anodyne CCR3 15 44 C[C@H](CO)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880936659 CD On-Demand Anodyne NPY5R 23 40 C[C@@H](CO)N(C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880936660 CD On-Demand Anodyne NPY5R 23 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(C(F)(F)F)CC1 ZINC000880936661 EF On-Demand Anodyne CACNA1H 44 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(C(F)(F)F)CC1 ZINC000880936661 EF On-Demand Anodyne TRPM8 20 42 CCC1(CO)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936667 DF On-Demand Anodyne CACNA1H 42 36 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880936671 GG On-Demand Anodyne CCR3 48 43 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880936672 GG On-Demand Anodyne CCR3 48 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccn2)C1 ZINC000880936674 EF On-Demand Anodyne HCRTR1 18 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccn2)C1 ZINC000880936674 EF On-Demand Anodyne HCRTR2 27 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880936675 EF On-Demand Anodyne HCRTR1 18 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880936675 EF On-Demand Anodyne HCRTR2 27 41 COC(=O)C[C@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880936717 DE On-Demand Anodyne ACKR3 58 33 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880936718 DE On-Demand Anodyne ACKR3 58 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)OCc1ccccc12 ZINC000880936722 FH On-Demand Anodyne NPY5R 31 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880936727 FF On-Demand Anodyne PDGFRB 34 41 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880936727 FF On-Demand Anodyne TRPV1 15 48 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880936727 FF On-Demand Anodyne FAAH 21 42 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2F)CC1 ZINC000880936727 FF On-Demand Anodyne RBP4 20 46 C[C@@H]1CN(CCCNC(=O)Nc2cc(F)ccc2N(C)C)CCCO1 ZINC000880936730 FF On-Demand Anodyne CCR3 53 45 C[C@H](O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)[C@H](C)C1 ZINC000880936744 ED On-Demand Anodyne CCR1 34 40 C[C@H](O)CN1CCN(C(=O)Nc2cc(F)ccc2N(C)C)[C@@H](C)C1 ZINC000880936746 ED On-Demand Anodyne CCR1 34 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880936756 GH On-Demand Anodyne CACNA1H 49 34 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CC(C)(C)C(N)=O)C1 ZINC000880936782 FG On-Demand Anodyne CCR3 54 31 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CC(C)(C)C(N)=O)C1 ZINC000880936783 FG On-Demand Anodyne CCR3 54 31 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CN2CCOCC2)C1 ZINC000880936788 FE On-Demand Anodyne CCR3 53 47 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CN2CCOCC2)C1 ZINC000880936789 FE On-Demand Anodyne CCR3 53 47 CN(C)c1ccc(F)cc1NC(=O)NCC(C)(C)c1ccccn1 ZINC000880936797 EG On-Demand Anodyne P2RY1 25 40 CN(C)c1ccc(F)cc1NC(=O)N(CCN1CCOCC1)Cc1ccco1 ZINC000880936799 GF On-Demand Anodyne CASR 58 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880936808 EF On-Demand Anodyne EPHX2 18 42 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880936824 GG On-Demand Anodyne EPHX2 29 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(S(=O)(=O)N(C)C)C1 ZINC000880936848 GD On-Demand Anodyne CCR3 25 42 COC[C@@H]1CCCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880936856 DF On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1C[C@H]2CCCC[C@H]2C1 ZINC000880936874 DH On-Demand Anodyne RBP4 47 39 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(c2ncccc2F)CC1 ZINC000880936882 GG On-Demand Anodyne FAAH 20 40 CN(C)c1ccc(F)cc1NC(=O)N1CCCN(c2ncccc2F)CC1 ZINC000880936882 GG On-Demand Anodyne RBP4 18 49 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000880936904 GI On-Demand Anodyne SLC18A3 33 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1 ZINC000880936904 GI On-Demand Anodyne WNT3A 47 34 CN(C)c1ccc(F)cc1NC(=O)NCCCc1nc[nH]n1 ZINC000880936918 DD On-Demand Anodyne CCR3 18 41 COC[C@@H]1CCCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880936932 DG On-Demand Anodyne CCR3 25 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CO)(c2ccccc2)CC1 ZINC000880936939 FG On-Demand Anodyne CACNA1H 51 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CO)(c2ccccc2)CC1 ZINC000880936939 FG On-Demand Anodyne RBP4 45 36 O=C(CCc1nc(O)c2cnn(-c3ccccc3)c2n1)NCc1ccc(O)cc1 ZINC000880937008 GE On-Demand Anodyne HCAR2 30 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CCO)Cc1ccccc1 ZINC000880937013 EG On-Demand Anodyne MME 52 36 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CCO)Cc1ccccc1 ZINC000880937013 EG On-Demand Anodyne ANPEP 56 32 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CCO)Cc1ccccc1 ZINC000880937014 EG On-Demand Anodyne MME 52 36 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CCO)Cc1ccccc1 ZINC000880937014 EG On-Demand Anodyne ANPEP 56 32 CN(C)c1ccc(F)cc1NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880937033 FF On-Demand Anodyne CHRNA4 26 48 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN1CCCO ZINC000880937065 ED On-Demand Anodyne CCR3 49 43 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN1CCCO ZINC000880937065 ED On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1CCCO ZINC000880937066 ED On-Demand Anodyne CCR3 49 43 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN1CCCO ZINC000880937066 ED On-Demand Anodyne ACKR3 45 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)OCCc1ccccc12 ZINC000880937076 GH On-Demand Anodyne NPY5R 26 42 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne DRD2 38 41 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne HTR2A 28 43 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne ADRA1A 44 36 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne DRD3 65 41 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne CCR3 59 44 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne CHRNA7 20 56 CN(C)c1ccc(F)cc1NC(=O)NCCCCCN1CCCC1 ZINC000880937087 EG On-Demand Anodyne HNMT 40 33 CN(C)c1ccc(F)cc1NC(=O)Nc1cc(C2CC2)[nH]n1 ZINC000880937089 DG On-Demand Anodyne CDK2 18 50 CN(C)c1ccc(F)cc1NC(=O)Nc1cc(C2CC2)[nH]n1 ZINC000880937089 DG On-Demand Anodyne NTRK1 19 41 CN(C)c1ccc(F)cc1NC(=O)Nc1cc(C2CC2)[nH]n1 ZINC000880937089 DG On-Demand Anodyne PKNB 71 42 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(N2CCOCC2)c1 ZINC000880937093 FG On-Demand Anodyne STAT6 44 38 CCSCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880937132 CG On-Demand Anodyne CCR3 19 43 CN(C)c1ccc(F)cc1NC(=O)N(C)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880937152 EF On-Demand Anodyne GLRA1 41 31 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C)(C#N)CC1 ZINC000880937157 DG On-Demand Mild CACNA1H 40 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H]1CCO ZINC000880937169 CE On-Demand Anodyne ACKR3 46 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H]1CCO ZINC000880937170 CE On-Demand Anodyne ACKR3 46 33 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880937173 EF On-Demand Anodyne PLM1_PLAFA 45 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880937173 EF On-Demand Anodyne PLM2_PLAFA 68 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880937174 EF On-Demand Anodyne PLM1_PLAFA 45 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880937174 EF On-Demand Anodyne PLM2_PLAFA 68 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C)(NC(=O)OC(C)(C)C)CC1 ZINC000880937239 GH On-Demand Anodyne CACNA1H 42 34 CN(C)c1ccc(F)cc1NC(=O)N1CCC(Oc2cncc(Cl)n2)CC1 ZINC000880937243 GG On-Demand Anodyne SCD1 24 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880937244 FG On-Demand Anodyne CACNA1H 56 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880937244 FG On-Demand Anodyne OPRL1 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880937244 FG On-Demand Anodyne CCR1 21 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880937247 FG On-Demand Anodyne CACNA1H 40 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880937248 FG On-Demand Anodyne CACNA1H 40 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](F)C1 ZINC000880937283 CE On-Demand Anodyne DPP4 21 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](F)C1 ZINC000880937284 CE On-Demand Anodyne DPP4 21 42 CN(C)c1ccc(F)cc1NC(=O)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880937288 EG On-Demand Anodyne EPHX2 51 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H](C1CC1)C(F)(F)F ZINC000880937293 DG On-Demand Anodyne PYGL 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](C1CC1)C(F)(F)F ZINC000880937294 DG On-Demand Anodyne PYGL 16 40 CN(C)c1ccc(F)cc1NC(=O)NC1CCC(OC(F)F)CC1 ZINC000880937320 EH On-Demand Anodyne EPHX2 39 43 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccc(F)cn2)CC1 ZINC000880937358 FF On-Demand Anodyne DGAT1 27 49 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ccc(F)cn2)CC1 ZINC000880937358 FF On-Demand Anodyne SLC27A1 44 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCC[C@H]1O ZINC000880937409 CE On-Demand Anodyne CCR3 29 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCC[C@@H]1O ZINC000880937410 CE On-Demand Anodyne CCR3 29 41 CN(C)c1ccc(F)cc1NC(=O)NCCN1CCNC(=O)C1 ZINC000880937420 DC On-Demand Anodyne PLD2 55 34 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(S(=O)(=O)N(C)C)c1 ZINC000880937422 GE On-Demand Anodyne ROCK2 16 42 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(S(=O)(=O)N(C)C)c1 ZINC000880937422 GE On-Demand Anodyne NAMPT 20 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880937431 EE On-Demand Anodyne CCR3 33 45 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880937432 EE On-Demand Anodyne CCR3 33 45 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880937455 GH On-Demand Anodyne CACNA1H 49 35 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880937463 FE On-Demand Anodyne CCR1 26 41 CN(C)C[C@@H]1CCN(C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880937515 DE On-Demand Anodyne CCR3 36 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880937545 GH On-Demand Anodyne CACNA1H 60 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880937552 EG On-Demand Anodyne CCR3 71 46 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CN2CCCCC2)C1 ZINC000880937553 EG On-Demand Anodyne CCR3 71 46 CN(C)c1ccc(F)cc1NC(=O)N1CCN(Cc2ccccn2)CC1 ZINC000880937576 FF On-Demand Anodyne FAAH 21 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880937580 FH On-Demand Anodyne NPY5R 25 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880937581 FH On-Demand Anodyne NPY5R 25 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(F)(F)C1 ZINC000880937599 CF On-Demand Anodyne CACNA1H 41 38 COc1cc(N2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)ncn1 ZINC000880937683 FE On-Demand Anodyne PDGFRB 51 40 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880937697 FE On-Demand Anodyne CCR3 63 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)C1CCOCC1 ZINC000880937709 ED On-Demand Anodyne PYGL 17 42 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)C1CCOCC1 ZINC000880937710 ED On-Demand Anodyne PYGL 17 42 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc2c(c1)C(=O)NCC2 ZINC000880937712 FE On-Demand Anodyne CSNK1G2 43 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)COC(=O)N2 ZINC000880937760 ED On-Demand Anodyne CACNA1H 49 36 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)Nc2ccc(Br)cc2)c1 ZINC000880937773 JJ On-Demand Anodyne RPA1 28 41 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(C(C)(C)O)cc1 ZINC000880937774 EG On-Demand Anodyne TRPV1 20 42 CN(C)c1ccc(F)cc1NC(=O)NCc1nnnn1CC1CC1 ZINC000880937775 ED On-Demand Anodyne CCR3 40 30 O=C(Cn1cnc2sc(-c3ccccc3)cc2c1=O)NCc1ccc(O)cc1 ZINC000880937778 GG On-Demand Anodyne F2 18 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccc2)C1 ZINC000880937841 EH On-Demand Anodyne PRSS2 45 31 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccc2)C1 ZINC000880937841 EH On-Demand Anodyne CCR3 38 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccc2)C1 ZINC000880937841 EH On-Demand Anodyne EPHX2 26 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccc2)C1 ZINC000880937841 EH On-Demand Anodyne RBP4 52 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](Oc2ccccc2)C1 ZINC000880937841 EH On-Demand Anodyne SCD1 18 46 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN(C(=O)C(F)(F)F)C1 ZINC000880937881 GF On-Demand Anodyne CCR3 56 38 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncc(F)cn2)CC1 ZINC000880937883 FE On-Demand Anodyne FAAH 20 40 CN(C)c1ccc(F)cc1NC(=O)NCCCCCCO ZINC000880937888 CF On-Demand Anodyne CCR3 17 43 CN(C)c1ccc(F)cc1NC(=O)NCCCNC(=O)C1CCC1 ZINC000880937897 EE On-Demand Anodyne TBK1 69 40 C[C@@H](C1CC1)n1cc(NC(=O)Nc2cc(F)ccc2N(C)C)cn1 ZINC000880937925 EH On-Demand Anodyne ITK 49 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCn2ccnc2C1 ZINC000880937937 EE On-Demand Anodyne CCR3 44 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCn2ccnc2C1 ZINC000880937938 EE On-Demand Anodyne CCR3 44 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CC(N)=O)C1 ZINC000880937939 DE On-Demand Anodyne CCR3 63 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CC(N)=O)C1 ZINC000880937940 DE On-Demand Anodyne CCR3 63 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C)(CO)CC1 ZINC000880937944 DF On-Demand Anodyne CACNA1H 45 37 CN(C)c1ccc(F)cc1NC(=O)NCc1cnc(N2CCOCC2)c(F)c1 ZINC000880937955 GF On-Demand Anodyne PIK3CA 20 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cnc(N2CCOCC2)c(F)c1 ZINC000880937955 GF On-Demand Anodyne MTOR 32 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cnc(N2CCOCC2)c(F)c1 ZINC000880937955 GF On-Demand Anodyne STAT6 50 35 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(N2CCOCC2)n1 ZINC000880937966 FE On-Demand Anodyne PIK3CA 25 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(N2CCOCC2)n1 ZINC000880937966 FE On-Demand Anodyne MTOR 26 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(N2CCOCC2)n1 ZINC000880937966 FE On-Demand Anodyne PIK3CG 16 41 CN(C)c1ccc(F)cc1NC(=O)NCc1cccc(N2CCOCC2)n1 ZINC000880937966 FE On-Demand Anodyne PIK3CB 64 39 CN(C)c1ccc(F)cc1NC(=O)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880937999 EF On-Demand Anodyne CPT1A 49 38 CN(C)c1ccc(F)cc1NC(=O)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880938000 EF On-Demand Anodyne CPT1A 49 38 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880938025 DE On-Demand Anodyne PLA2G7 44 33 C[C@@H](Cc1cnn(C)c1)NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880938025 DE On-Demand Anodyne CCR3 44 34 CN(C)c1ccc(F)cc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880938026 DF On-Demand Anodyne SLC6A3 19 42 CN(C)c1ccc(F)cc1NC(=O)NC1C[C@@H]2CC[C@H](C1)N2C ZINC000880938026 DF On-Demand Anodyne GLRA1 40 30 C[C@@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)CCN(C2CCC2)C1 ZINC000880938032 EG On-Demand Anodyne HRH3 16 40 C[C@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)CCN(C2CCC2)C1 ZINC000880938033 EG On-Demand Anodyne HRH3 16 40 COc1ccc(-c2nnc(S)n2CCC(=O)NCc2ccc(O)cc2)cc1 ZINC000880938056 GF On-Demand Anodyne HTR7 15 41 COc1ccc(-c2nnc(S)n2CCC(=O)NCc2ccc(O)cc2)cc1 ZINC000880938056 GF On-Demand Anodyne PROKR1 56 38 COc1ccc(N2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)nc1 ZINC000880938239 FF On-Demand Anodyne PDGFRB 50 39 COc1ccc(N2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)nc1 ZINC000880938239 FF On-Demand Anodyne DGAT1 29 49 COc1ccc(N2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)nc1 ZINC000880938239 FF On-Demand Anodyne SLC27A1 46 38 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880938338 ED On-Demand Anodyne SLC6A1 42 35 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880938338 ED On-Demand Anodyne CCR3 95 48 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCCO)C1 ZINC000880938338 ED On-Demand Anodyne BIRC2 33 41 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880938339 ED On-Demand Anodyne SLC6A1 42 35 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880938339 ED On-Demand Anodyne CCR3 95 48 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCCO)C1 ZINC000880938339 ED On-Demand Anodyne BIRC2 33 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN(C2CCC2)CC1 ZINC000880938364 EG On-Demand Anodyne EPHX2 41 39 CN(C)c1ccc(F)cc1NC(=O)NCCN1C[C@@H]2CC[C@H](C1)O2 ZINC000880938373 ED On-Demand Anodyne CCR3 41 37 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2ncccc2[N+](=O)[O-])CC1 ZINC000880938421 GF On-Demand Bother RBP4 16 41 CN(C)c1ccc(F)cc1NC(=O)N1CC(C(F)(F)F)C1 ZINC000880938422 DF On-Demand Anodyne RBP4 53 39 CN(C)c1ccc(F)cc1NC(=O)N(C)[C@@H](CO)c1ccccc1 ZINC000880938509 EG On-Demand Anodyne NPY5R 32 42 CN(C)c1ccc(F)cc1NC(=O)N(C)[C@H](CO)c1ccccc1 ZINC000880938510 EG On-Demand Anodyne NPY5R 32 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H]1CO ZINC000880938513 CE On-Demand Anodyne CCR3 40 45 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880938514 FG On-Demand Anodyne CACNA1H 47 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880938514 FG On-Demand Anodyne EPHX2 20 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880938515 FG On-Demand Anodyne CACNA1H 47 34 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880938515 FG On-Demand Anodyne EPHX2 20 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)C1CCCC1 ZINC000880938543 DF On-Demand Anodyne PYGL 16 47 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)C1CCCC1 ZINC000880938544 DF On-Demand Anodyne PYGL 16 47 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCC(O)CC2)CC1 ZINC000880938557 EG On-Demand Anodyne CACNA1H 49 38 CN(C)c1ccc(F)cc1NC(=O)NCCCCF ZINC000880938560 CF On-Demand Anodyne CCR3 18 44 CN(C)c1ccc(F)cc1NC(=O)NCc1nn(C)cc1Cl ZINC000880938566 EF On-Demand Anodyne P2RX7 39 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(C(N)=O)CC1 ZINC000880938573 DC On-Demand Anodyne CACNA1H 53 37 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880938579 GG On-Demand Anodyne CA12 25 41 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880938579 GG On-Demand Anodyne CA9 23 41 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880938579 GG On-Demand Anodyne P96878_MYCTU 41 39 CCc1noc(C)c1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880938594 DG On-Demand Anodyne P2RX7 17 44 CN(C)c1ccc(F)cc1NC(=O)NCCCCN(C)C1CC1 ZINC000880938596 DF On-Demand Anodyne CCR3 29 44 Cc1ccncc1CNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880938601 DF On-Demand Anodyne P2RX7 32 41 CN(C)c1ccc(F)cc1NC(=O)N1CC(C2CC2)C1 ZINC000880938613 CF On-Demand Anodyne RBP4 48 40 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCCN1CCO ZINC000880938648 ED On-Demand Anodyne CCR3 41 41 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCCN1CCO ZINC000880938649 ED On-Demand Anodyne CCR3 41 41 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN(C(=O)C(F)(F)F)C1 ZINC000880938668 GF On-Demand Anodyne CCR3 56 38 COCC1CCC(NC(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880938669 DG On-Demand Anodyne CCR3 16 41 CN1CCC[C@@H](CCNC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880938675 DF On-Demand Anodyne CCR3 90 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880938687 EG On-Demand Anodyne SCD1 18 42 CN(C)c1ccc(F)cc1NC(=O)N(CCO)CCOCCO ZINC000880938705 EC On-Demand Anodyne SOAT1 17 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H]1N1CC[C@@H](O)C1 ZINC000880938762 FE On-Demand Anodyne CCR3 27 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H]1N1CC[C@H](O)C1 ZINC000880938763 FE On-Demand Anodyne CCR3 27 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H](CO)C1CCC1 ZINC000880938861 CE On-Demand Anodyne PYGL 16 45 CN(C)c1ccc(F)cc1NC(=O)N[C@@H](CO)C1CCC1 ZINC000880938862 CE On-Demand Anodyne PYGL 16 45 CN(C)c1ccc(F)cc1NC(=O)NCc1nccc(C(F)(F)F)n1 ZINC000880938879 FG On-Demand Anodyne TRPV1 41 36 CN(C)c1ccc(F)cc1NC(=O)NCc1c(C2CC2)cnn1C ZINC000880938880 EF On-Demand Anodyne P2RX7 17 41 CN(C)c1ccc(F)cc1NC(=O)NCC1(N2CCOCC2)CCOCC1 ZINC000880938911 GD On-Demand Anodyne HCN1 48 38 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880938930 GF On-Demand Anodyne CCR1 31 40 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880938930 GF On-Demand Anodyne CCR3 96 44 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880938930 GF On-Demand Anodyne MLNR 63 38 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@@H](O)C2)cc1 ZINC000880938930 GF On-Demand Anodyne MCHR1 33 46 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880938931 GF On-Demand Anodyne CCR1 31 40 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880938931 GF On-Demand Anodyne CCR3 96 44 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880938931 GF On-Demand Anodyne MLNR 63 38 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(CN2CC[C@H](O)C2)cc1 ZINC000880938931 GF On-Demand Anodyne MCHR1 33 46 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880938938 ED On-Demand Anodyne CCR3 25 51 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880938938 ED On-Demand Anodyne EPHX2 34 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880938939 ED On-Demand Anodyne CCR3 25 51 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880938939 ED On-Demand Anodyne EPHX2 34 41 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880938941 EG On-Demand Anodyne CCR3 53 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCN(C(C)(C)C)C1 ZINC000880938941 EG On-Demand Anodyne CACNA1I 61 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880938942 EG On-Demand Anodyne CCR3 53 35 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCN(C(C)(C)C)C1 ZINC000880938942 EG On-Demand Anodyne CACNA1I 61 35 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880939002 GF On-Demand Anodyne CCR3 51 37 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(C2CCOCC2)CC1 ZINC000880939002 GF On-Demand Anodyne CACNA1I 58 34 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@H](CO)C1 ZINC000880939009 DF On-Demand Anodyne CCR3 22 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880939010 DF On-Demand Anodyne CCR3 22 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCC[C@H](CO)C1 ZINC000880939011 DF On-Demand Anodyne CCR3 22 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCC[C@@H](CO)C1 ZINC000880939012 DF On-Demand Anodyne CCR3 22 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1COCc2ccccc21 ZINC000880939108 EG On-Demand Anodyne TRPV1 18 43 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1COCc2ccccc21 ZINC000880939109 EG On-Demand Anodyne TRPV1 18 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](C(=O)NCc2ccccc2)C1 ZINC000880939128 GG On-Demand Anodyne CCR3 42 38 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](C(=O)NCc2ccccc2)C1 ZINC000880939128 GG On-Demand Anodyne EPHX2 25 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](C(=O)NCc2ccccc2)C1 ZINC000880939128 GG On-Demand Anodyne CACNA1G 48 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](C(=O)NCc2ccccc2)C1 ZINC000880939129 GG On-Demand Anodyne CCR3 42 38 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](C(=O)NCc2ccccc2)C1 ZINC000880939129 GG On-Demand Anodyne EPHX2 25 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](C(=O)NCc2ccccc2)C1 ZINC000880939129 GG On-Demand Anodyne CACNA1G 48 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN2CCCC[C@@H]12 ZINC000880939158 EG On-Demand Anodyne CCR3 42 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN2CCCC[C@H]12 ZINC000880939159 EG On-Demand Anodyne CCR3 42 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN2CCCC[C@H]12 ZINC000880939160 EG On-Demand Anodyne CCR3 42 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN2CCCC[C@@H]12 ZINC000880939161 EG On-Demand Anodyne CCR3 42 44 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](C2CCC2)C1 ZINC000880939165 DH On-Demand Anodyne RBP4 45 38 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](C2CCC2)C1 ZINC000880939166 DH On-Demand Anodyne RBP4 45 38 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880939173 DE On-Demand Anodyne CHRNA10 60 40 CN(C[C@H]1CCCN1C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880939173 DE On-Demand Anodyne ACKR3 68 36 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880939174 DE On-Demand Anodyne CHRNA10 60 40 CN(C[C@@H]1CCCN1C)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880939174 DE On-Demand Anodyne ACKR3 68 36 CN1CCC(CNC(=O)Nc2cc(F)ccc2N(C)C)(N2CCOCC2)CC1 ZINC000880939175 GD On-Demand Anodyne HCN1 45 35 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880939195 FF On-Demand Anodyne PYGL 33 55 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1Cc2ccccc2N(C)C1=O ZINC000880939195 FF On-Demand Anodyne PYGM 31 55 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CN2CCCC2=O)C1 ZINC000880939196 EE On-Demand Anodyne CCR3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CN2CCCC2=O)C1 ZINC000880939197 EE On-Demand Anodyne CCR3 17 41 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CCCN(CC2CC2)C1 ZINC000880939254 EG On-Demand Anodyne CCR3 131 47 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CCCN(CC2CC2)C1 ZINC000880939255 EG On-Demand Anodyne CCR3 131 47 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880939256 EH On-Demand Anodyne PRSS2 45 31 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880939256 EH On-Demand Anodyne CCR3 38 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880939256 EH On-Demand Anodyne EPHX2 26 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880939256 EH On-Demand Anodyne RBP4 52 37 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880939256 EH On-Demand Anodyne SCD1 18 46 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880939296 FF On-Demand Anodyne PYGL 33 55 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1Cc2ccccc2N(C)C1=O ZINC000880939296 FF On-Demand Anodyne PYGM 31 55 CN(C)c1ccc(F)cc1NC(=O)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880939331 DF On-Demand Anodyne RBP4 42 41 CN(C)c1ccc(F)cc1NC(=O)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880939332 DF On-Demand Anodyne RBP4 42 41 CN(C)c1ccc(F)cc1NC(=O)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880939333 DF On-Demand Anodyne RBP4 42 41 CN(C)c1ccc(F)cc1NC(=O)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880939334 DF On-Demand Anodyne RBP4 42 41 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880939335 GG On-Demand Anodyne ACHE 23 42 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880939335 GG On-Demand Anodyne HTR4 45 39 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880939335 GG On-Demand Anodyne SIGMAR1 25 46 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880939335 GG On-Demand Anodyne CCR3 100 50 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(Cc2ccncc2)CC1 ZINC000880939335 GG On-Demand Anodyne CACNA1I 68 43 CCN1CC[C@H](N(CC)C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880939339 DF On-Demand Anodyne CCR5 15 40 CCN1CC[C@@H](N(CC)C(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880939340 DF On-Demand Anodyne CCR5 15 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)CC2(F)F ZINC000880939341 EH On-Demand Anodyne CACNA1H 44 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880939377 FF On-Demand Anodyne L3MBTL3 67 38 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880939378 FF On-Demand Anodyne L3MBTL3 67 38 COC1(C(F)(F)F)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880939385 FG On-Demand Anodyne CACNA1H 46 35 COC1(C(F)(F)F)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880939385 FG On-Demand Anodyne TRPM8 23 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCOC1=O ZINC000880939395 CD On-Demand Anodyne LUXR 76 41 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCOC1=O ZINC000880939395 CD On-Demand Anodyne TRAR 88 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCOC1=O ZINC000880939395 CD On-Demand Anodyne LASR 60 37 CN(C)c1ccc(F)cc1NC(=O)N1C[C@H]2COC[C@H]2C1 ZINC000880939414 CE On-Demand Anodyne RBP4 47 39 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880939420 ED On-Demand Anodyne CCR3 55 47 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCCC2=O)CC1 ZINC000880939421 EG On-Demand Anodyne CACNA1H 44 36 CCn1nc(C)c(CN(C)C(=O)Nc2cc(F)ccc2N(C)C)c1C ZINC000880939423 EG On-Demand Anodyne P2RX7 18 47 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880939432 EE On-Demand Anodyne HCRTR1 18 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCNC2=O)CC1 ZINC000880939454 EE On-Demand Anodyne CACNA1H 64 39 CN(C)c1ccc(F)cc1NC(=O)NC[C@H]1CN(Cc2ccncc2)CCO1 ZINC000880939456 GE On-Demand Anodyne CCR3 28 45 CN(C)c1ccc(F)cc1NC(=O)NC[C@@H]1CN(Cc2ccncc2)CCO1 ZINC000880939457 GE On-Demand Anodyne CCR3 28 45 CN(C)c1ccc(F)cc1NC(=O)N1CCC(C)(F)CC1 ZINC000880939489 CG On-Demand Anodyne CACNA1H 49 39 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(CO)CC1 ZINC000880939554 DD On-Demand Anodyne CACNA1H 46 37 CN(C)c1ccc(F)cc1NC(=O)N1CCC(O)(CO)CC1 ZINC000880939554 DD On-Demand Anodyne S1PR2 30 43 CN(C)c1ccc(F)cc1NC(=O)NCCCCS(C)(=O)=O ZINC000880939555 ED On-Demand Anodyne CCR3 15 41 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne CA2 15 45 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne CA1 44 39 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne P2RY1 43 34 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne CA12 26 45 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne CA9 25 45 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne NCE103 18 42 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne MTCA1 22 42 CN(C)c1ccc(F)cc1NC(=O)Nc1ccc(OCCS(C)(=O)=O)cc1 ZINC000880939571 GF On-Demand Anodyne P96878_MYCTU 21 42 CN(C)c1ccc(F)cc1NC(=O)N1CCc2cc(Cl)nnc2C1 ZINC000880939576 EF On-Demand Anodyne MAPK1 45 35 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880939589 FH On-Demand Anodyne CACNA1H 49 39 CN(C)c1ccc(F)cc1NC(=O)NC1CCC(N(C)C)CC1 ZINC000880939598 DF On-Demand Anodyne AVPR1A 33 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCC(N(C)C)CC1 ZINC000880939598 DF On-Demand Anodyne EPHX2 43 40 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCCC1 ZINC000880939602 FG On-Demand Anodyne KCNQ2 44 38 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCCC1 ZINC000880939602 FG On-Demand Anodyne TRPV1 34 42 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCCC1 ZINC000880939602 FG On-Demand Anodyne SCN2A 19 45 CN(C)c1ccc(F)cc1NC(=O)NCc1cccnc1N1CCCC1 ZINC000880939602 FG On-Demand Anodyne SCN10A 19 45 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939604 GH On-Demand Anodyne ACACA 41 36 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939604 GH On-Demand Anodyne NPY5R 16 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939604 GH On-Demand Anodyne EPHX2 20 49 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939604 GH On-Demand Anodyne TRPM8 20 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939605 GH On-Demand Anodyne ACACA 41 36 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939605 GH On-Demand Anodyne NPY5R 16 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939605 GH On-Demand Anodyne EPHX2 20 49 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(CC(=O)c3ccccc3O2)C1 ZINC000880939605 GH On-Demand Anodyne TRPM8 20 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880939643 GG On-Demand Anodyne TRPM8 31 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880939644 GG On-Demand Anodyne TRPM8 31 41 CN(C)c1ccc(F)cc1NC(=O)N1CCc2nc(C3CC3)ncc2C1 ZINC000880939648 FG On-Demand Anodyne MAPK1 43 35 CN(C)c1ccc(F)cc1NC(=O)N1CCn2c(nnc2-c2cn(C)cn2)C1 ZINC000880939657 GD On-Demand Anodyne P2RX7 23 44 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(CC2CC2)CC1 ZINC000880939670 EG On-Demand Anodyne CCR3 87 42 CN(C)c1ccc(F)cc1NC(=O)NCC1CCN(CC2CC2)CC1 ZINC000880939670 EG On-Demand Anodyne CACNA1I 68 38 NC(=O)COc1cccc(NC(=O)c2cccnc2-n2cccn2)c1 ZINC000880939671 ED On-Demand Anodyne GRM4 28 41 NC(=O)COc1cccc(NC(=O)c2cccnc2-n2cccn2)c1 ZINC000880939671 ED On-Demand Anodyne KCNK3 66 37 NC(=O)COc1cccc(NC(=O)c2cccnc2-n2cccn2)c1 ZINC000880939671 ED On-Demand Anodyne KCNK9 51 37 CN(C)c1ccc(F)cc1NC(=O)N1CCN(c2nccnn2)CC1 ZINC000880939677 ED On-Demand Anodyne FAAH 25 48 CN(C)c1ccc(F)cc1NC(=O)N1CC(c2ccccc2)C1 ZINC000880939688 DH On-Demand Anodyne RBP4 58 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CCF)C1 ZINC000880939717 DG On-Demand Anodyne CCR3 49 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CCF)C1 ZINC000880939718 DG On-Demand Anodyne CCR3 49 33 COc1ccc(-n2c(C)cc(C(=O)NCc3ccc(O)cc3)c2C)cc1 ZINC000880939733 FH On-Demand Clean SLC6A5 18 44 COc1ccc(-n2c(C)cc(C(=O)NCc3ccc(O)cc3)c2C)cc1 ZINC000880939733 FH On-Demand Clean AKR1B10 32 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CCO)(CCO)CC1 ZINC000880939736 FE On-Demand Anodyne CACNA1H 44 36 CN(C)c1ccc(F)cc1NC(=O)NCc1ccc(N2CCC(O)CC2)cc1 ZINC000880939737 GG On-Demand Clean CCR3 52 35 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880939772 GG On-Demand Anodyne TRPM8 31 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880939773 GG On-Demand Anodyne TRPM8 31 41 C[C@@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)[C@H](C)CN1CCO ZINC000880939780 ED On-Demand Anodyne CCR1 20 40 C[C@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)[C@H](C)CN1CCO ZINC000880939782 ED On-Demand Anodyne CCR1 20 40 C[C@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)[C@@H](C)CN1CCO ZINC000880939783 ED On-Demand Anodyne CCR1 20 40 CN(C)c1ccc(F)cc1NC(=O)N(C)[C@H](CO)Cc1ccccc1 ZINC000880939792 EF On-Demand Anodyne NPY5R 33 45 CN(C)c1ccc(F)cc1NC(=O)N(C)[C@@H](CO)Cc1ccccc1 ZINC000880939793 EF On-Demand Anodyne NPY5R 33 45 C=CCOCCCNC(=O)Nc1cc(F)ccc1N(C)C ZINC000880939831 CF On-Demand Mild CCR3 17 40 CCC1(N(C)C)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880939947 EG On-Demand Anodyne CACNA1H 45 37 CN(C)c1ccc(F)cc1NC(=O)NCc1nc(O)c2c(n1)CCOC2 ZINC000880939948 FD On-Demand Anodyne WNT3A 53 34 CN1CCN(C2CCN(C(=O)Nc3cc(F)ccc3N(C)C)CC2)CC1 ZINC000880939957 FE On-Demand Anodyne L3MBTL3 65 40 CN(C)c1ccc(F)cc1NC(=O)NCc1c(Br)cnn1C ZINC000880939997 FF On-Demand Anodyne HTR2A 19 40 CN(C)c1ccc(F)cc1NC(=O)N1CCc2nc(C(C)(C)C)ncc2C1 ZINC000880940008 FH On-Demand Anodyne MAPK1 43 36 COc1ccccc1[C@@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)CCO1 ZINC000880940025 FH On-Demand Anodyne RBP4 42 39 COc1ccccc1[C@H]1CN(C(=O)Nc2cc(F)ccc2N(C)C)CCO1 ZINC000880940026 FH On-Demand Anodyne RBP4 42 39 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@H]2CCOC2)CC1 ZINC000880940050 FE On-Demand Anodyne CCR3 17 41 CN(C)c1ccc(F)cc1NC(=O)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880940051 FE On-Demand Anodyne CCR3 17 41 CN(C)c1ccc(F)cc1NC(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880940061 FF On-Demand Anodyne RBP4 45 37 COCC1CC(NC(=O)Nc2cc(F)ccc2N(C)C)C1 ZINC000880940078 CE On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)NCCN1CC[C@@H](O)C1 ZINC000880940151 DD On-Demand Anodyne CCR3 81 40 CN(C)c1ccc(F)cc1NC(=O)NCCN1CC[C@H](O)C1 ZINC000880940152 DD On-Demand Anodyne CCR3 81 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)OC(C)(C)C)C[C@@H]1O ZINC000880940174 GE On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)OC(C)(C)C)C[C@@H]1O ZINC000880940174 GE On-Demand Anodyne GPR119 30 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)OC(C)(C)C)C[C@@H]1O ZINC000880940175 GE On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)OC(C)(C)C)C[C@@H]1O ZINC000880940175 GE On-Demand Anodyne GPR119 30 42 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)OC(C)(C)C)C[C@H]1O ZINC000880940176 GE On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCN(C(=O)OC(C)(C)C)C[C@H]1O ZINC000880940176 GE On-Demand Anodyne GPR119 30 42 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)OC(C)(C)C)C[C@H]1O ZINC000880940177 GE On-Demand Anodyne CCR3 16 40 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCN(C(=O)OC(C)(C)C)C[C@H]1O ZINC000880940177 GE On-Demand Anodyne GPR119 30 42 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2nnnn2C)CC1 ZINC000880940178 ED On-Demand Anodyne CCR3 41 32 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880940181 GH On-Demand Anodyne SMO 38 43 CN(C)c1ccc(F)cc1NC(=O)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880940181 GH On-Demand Anodyne ETHR 61 44 COCCN(CC1CCN(C)CC1)C(=O)Nc1cc(F)ccc1N(C)C ZINC000880940190 FF On-Demand Anodyne ACKR3 45 31 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CCF)CC1 ZINC000880940222 DG On-Demand Anodyne RBP4 41 38 COC[C@@H]1CCCN1NC(=O)Nc1cc(F)ccc1N(C)C ZINC000880940230 DE On-Demand Anodyne CCR3 20 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](OC2CCC2)CC1 ZINC000880940251 EH On-Demand Anodyne SCD1 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880940252 EH On-Demand Anodyne SCD1 17 41 CN(C)c1ccc(F)cc1NC(=O)N1CCCC(F)(F)CC1 ZINC000880940262 DH On-Demand Anodyne CACNA1H 41 37 CN(C)c1ccc(F)cc1NC(=O)N(CCN1CCOCC1)CC1CC1 ZINC000880940294 FE On-Demand Anodyne CASR 59 43 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H]2C[C@@H]2C1 ZINC000880940297 CF On-Demand Anodyne RBP4 57 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H]2C[C@H]2C1 ZINC000880940298 CF On-Demand Anodyne RBP4 57 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H]2C[C@H]2C1 ZINC000880940299 CF On-Demand Anodyne RBP4 57 42 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H]2C[C@@H]2C1 ZINC000880940300 CF On-Demand Anodyne RBP4 57 42 COC[C@@H]1CCCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880940319 CF On-Demand Anodyne ACKR3 59 34 CN(C)c1ccc(F)cc1NC(=O)NCCCN1CCC[C@H]1C(N)=O ZINC000880940327 FD On-Demand Anodyne CCR3 52 41 CN(C)c1ccc(F)cc1NC(=O)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880940338 GF On-Demand Anodyne ETHR 41 34 CN(C)c1ccc(F)cc1NC(=O)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880940339 GF On-Demand Anodyne ETHR 41 34 CN(C)c1ccc(F)cc1NC(=O)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880940352 DG On-Demand Anodyne RBP4 47 39 CN1CCN(C(=O)Nc2cnc3ccccc3c2Br)CCC1=O ZINC000880940372 GF On-Demand Anodyne PDGFRB 25 40 CN1CC[C@@]2(CCN(C(=O)Nc3cnc4ccccc4c3Br)C2)C1 ZINC000880940415 GH On-Demand Anodyne EPHX2 21 41 COC(=O)C[C@@H](C)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880940431 FG On-Demand Anodyne ANPEP 16 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CCCCO2)CC1 ZINC000880940509 EG On-Demand Anodyne TRPM8 16 41 C[C@H]1c2sccc2CCN1C(=O)Nc1cc(F)ccc1N(C)C ZINC000880940593 EI On-Demand Anodyne TRPM8 24 46 O=C(Nc1cnc2ccccc2c1Br)N1C[C@H]2COC[C@H]2C1 ZINC000880940616 FG On-Demand Anodyne RBP4 48 36 O=C(Nc1cnc2ccccc2c1Br)N1CC(C(F)(F)F)C1 ZINC000880940638 FI On-Demand Anodyne RBP4 57 38 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@@H]2CCCC23CC3)c1 ZINC000880940677 EE On-Demand Anodyne CA2 32 44 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@@H]2CCCC23CC3)c1 ZINC000880940677 EE On-Demand Anodyne CA1 29 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@@H]2CCCC23CC3)c1 ZINC000880940677 EE On-Demand Anodyne CA4 34 44 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@@H]2CCCC23CC3)c1 ZINC000880940677 EE On-Demand Anodyne CA9 19 44 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@H]2CCCC23CC3)c1 ZINC000880940678 EE On-Demand Anodyne CA2 32 44 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@H]2CCCC23CC3)c1 ZINC000880940678 EE On-Demand Anodyne CA1 29 42 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@H]2CCCC23CC3)c1 ZINC000880940678 EE On-Demand Anodyne CA4 34 44 NS(=O)(=O)c1ccc(Cl)c(C(=O)N[C@H]2CCCC23CC3)c1 ZINC000880940678 EE On-Demand Anodyne CA9 19 44 CN(C)c1ccc(F)cc1NC(=O)N1CCC2(CC1)COCCO2 ZINC000880940679 EE On-Demand Anodyne TRPM8 18 42 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880940691 GF On-Demand Anodyne CCR8 71 34 CC(=O)N[C@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880940692 GF On-Demand Anodyne CCR8 71 34 O=C(Nc1cnc2ccccc2c1Br)N[C@H]1CCC[C@@H]1O ZINC000880940705 FG On-Demand Anodyne CDK5 23 41 O=C(Nc1cnc2ccccc2c1Br)N[C@@H]1CCC[C@H]1O ZINC000880940706 FG On-Demand Anodyne CDK5 23 41 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@@H](F)C1 ZINC000880940716 EH On-Demand Anodyne RBP4 53 34 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@H](F)C1 ZINC000880940717 EH On-Demand Anodyne RBP4 53 34 CN1CC[C@H]2CN(C(=O)Nc3cnc4ccccc4c3Br)CC[C@H]21 ZINC000880940754 GH On-Demand Anodyne CCR8 43 30 CN1CC[C@H]2CN(C(=O)Nc3cnc4ccccc4c3Br)CC[C@@H]21 ZINC000880940755 GH On-Demand Anodyne CCR8 43 30 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880940760 JH On-Demand Bother KCNMA1 19 41 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880940760 JH On-Demand Bother PTGDR 35 47 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880940760 JH On-Demand Bother PTGDR2 27 47 O=C(Nc1cnc2ccccc2c1Br)NC1CCC1 ZINC000880940770 DH On-Demand Anodyne EPHX2 19 46 O=C(Nc1cnc2ccccc2c1Br)NC1CCC1 ZINC000880940770 DH On-Demand Anodyne CDK5 29 44 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880940774 FG On-Demand Anodyne RBP4 40 36 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880940775 FG On-Demand Anodyne RBP4 40 36 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@H](CF)C1 ZINC000880940784 CG On-Demand Anodyne CCR3 55 33 CN(C)c1ccc(F)cc1NC(=O)N1CCC[C@@H](CF)C1 ZINC000880940785 CG On-Demand Anodyne CCR3 55 33 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc3ccccc3c1Br)C2 ZINC000880940843 GH On-Demand Anodyne HTR3A 34 43 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnc3ccccc3c1Br)C2 ZINC000880940843 GH On-Demand Anodyne GLRA1 44 41 O=C(Nc1cnc2ccccc2c1Br)N1CCC2(COC2)C1 ZINC000880940851 FG On-Demand Anodyne EPHX2 22 42 O=C(Nc1cnc2ccccc2c1Br)N1CC(C2CC2)C1 ZINC000880940890 EH On-Demand Anodyne RBP4 55 37 CC[C@@H](NC(=O)Nc1cnc2ccccc2c1Br)C(=O)NC ZINC000880940918 FF On-Demand Anodyne ANPEP 19 43 CC[C@@H](NC(=O)Nc1cnc2ccccc2c1Br)C(=O)NC ZINC000880940918 FF On-Demand Anodyne TACR3 40 40 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnc2ccccc2c1Br ZINC000880940930 FG On-Demand Anodyne UL80 24 42 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnc2ccccc2c1Br ZINC000880940931 FG On-Demand Anodyne UL80 24 42 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnc2ccccc2c1Br ZINC000880940933 FG On-Demand Anodyne UL80 24 42 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)Nc2cc(Cl)ccc2Cl)c1 ZINC000880940962 JK On-Demand Anodyne PTGDR 32 45 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)Nc2cc(Cl)ccc2Cl)c1 ZINC000880940962 JK On-Demand Anodyne PTGDR2 25 45 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880941024 CE On-Demand Anodyne EPHX2 37 40 C#CCC1(O)CCN(C(=O)Nc2cc(F)ccc2N(C)C)CC1 ZINC000880941035 DE On-Demand Mild S1PR2 29 41 CS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880941037 JG On-Demand Anodyne CA4 15 42 CS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880941037 JG On-Demand Anodyne MAPK9 26 42 CS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880941037 JG On-Demand Anodyne GHSR 17 42 CS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880941037 JG On-Demand Anodyne MAPK8 24 42 O=C(NCCN1CC[C@@H](O)C1)Nc1cnc2ccccc2c1Br ZINC000880941122 GE On-Demand Anodyne UTS2R 17 42 O=C(NCCN1CC[C@H](O)C1)Nc1cnc2ccccc2c1Br ZINC000880941123 GE On-Demand Anodyne UTS2R 17 42 CN1C(=O)CC[C@@H](NC(=O)Nc2cnc3ccccc3c2Br)C1=O ZINC000880941124 GE On-Demand Anodyne CCKBR 17 40 CN1C(=O)CC[C@H](NC(=O)Nc2cnc3ccccc3c2Br)C1=O ZINC000880941125 GE On-Demand Anodyne CCKBR 17 40 O=C(NCCCC1(O)CCC1)Nc1cnc2ccccc2c1Br ZINC000880941150 GH On-Demand Anodyne UTS2R 15 40 O=C(NCCN1CCCC1=O)Nc1cnc2ccccc2c1Br ZINC000880941157 GF On-Demand Anodyne UTS2R 17 41 COc1ccc(CN(CCO)C(=O)Nc2cc(F)ccc2N(C)C)cc1 ZINC000880941202 FF On-Demand Anodyne ROCK2 15 40 COC[C@@H](O)CNC(=O)Nc1cnc2ccccc2c1Br ZINC000880941210 FE On-Demand Anodyne ADRB1 43 37 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941212 GD On-Demand Anodyne CCR3 105 44 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941212 GD On-Demand Anodyne EPHX2 30 45 CN(C)c1ccc(F)cc1NC(=O)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941212 GD On-Demand Anodyne BIRC2 32 40 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941213 GD On-Demand Anodyne CCR3 105 44 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941213 GD On-Demand Anodyne EPHX2 30 45 CN(C)c1ccc(F)cc1NC(=O)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880941213 GD On-Demand Anodyne BIRC2 32 40 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@@H](CF)C1 ZINC000880941225 CF On-Demand Anodyne CCR3 30 41 CN(C)c1ccc(F)cc1NC(=O)N1CC[C@H](CF)C1 ZINC000880941226 CF On-Demand Anodyne CCR3 30 41 O=C(Nc1cnc2ccccc2c1Br)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880941244 GH On-Demand Anodyne RBP4 62 37 O=C(Nc1cnc2ccccc2c1Br)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880941245 GH On-Demand Anodyne RBP4 62 37 O=C(Nc1cnc2ccccc2c1Br)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880941246 GH On-Demand Anodyne RBP4 62 37 O=C(Nc1cnc2ccccc2c1Br)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880941247 GH On-Demand Anodyne RBP4 62 37 O=C(Nc1cnc2ccccc2c1Br)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880941248 GH On-Demand Anodyne RBP4 62 37 COC[C@@H](C)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880941249 EG On-Demand Anodyne ANPEP 15 40 COC[C@H](C)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880941250 EG On-Demand Anodyne ANPEP 15 40 CCC[C@H](NC(=O)Nc1cnc2ccccc2c1Br)C(N)=O ZINC000880941273 FF On-Demand Anodyne ANPEP 16 41 O=C(CNC(=O)Nc1cnc2ccccc2c1Br)NC1CC1 ZINC000880941287 FE On-Demand Anodyne TNKS 58 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(N(C)C(C)=O)CC1 ZINC000880941302 FE On-Demand Anodyne RBP4 40 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCN(S(C)(=O)=O)CC1 ZINC000880941308 GD On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](C2OCCO2)C1 ZINC000880941310 FF On-Demand Anodyne RBP4 40 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](C2OCCO2)C1 ZINC000880941312 FF On-Demand Anodyne RBP4 40 40 CN(C)c1ccc(F)cc1NC(=O)N1CCC(CO)(CO)CC1 ZINC000880941313 ED On-Demand Anodyne CACNA1H 45 38 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941321 GG On-Demand Anodyne RBP4 40 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](OCC)C1 ZINC000880941324 EG On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](OCC)C1 ZINC000880941324 EG On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](OCC)C1 ZINC000880941326 EG On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](OCC)C1 ZINC000880941326 EG On-Demand Anodyne TLR4 15 40 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@@H]2C[C@@H]2C1 ZINC000880941338 EH On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@@H]2C[C@H]2C1 ZINC000880941343 EH On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@H]2C[C@H]2C1 ZINC000880941345 EH On-Demand Anodyne RBP4 58 39 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@H]2C[C@@H]2C1 ZINC000880941346 EH On-Demand Anodyne RBP4 58 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880941364 FE On-Demand Anodyne P2RY12 38 47 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880941364 FE On-Demand Anodyne PDGFRB 37 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccn2)CC1 ZINC000880941364 FE On-Demand Anodyne FAAH 27 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CO)C1 ZINC000880941365 DE On-Demand Anodyne CCR3 74 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CO)C1 ZINC000880941365 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CO)C1 ZINC000880941367 DE On-Demand Anodyne CCR3 74 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CO)C1 ZINC000880941367 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nnc(NC)cc2C1 ZINC000880941370 FE On-Demand Anodyne P2RY14 40 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)OC)CC1 ZINC000880941419 FE On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)OC)CC1 ZINC000880941419 FE On-Demand Anodyne PTR1 47 35 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC)C(C)C ZINC000880941433 CG On-Demand Anodyne TLR4 15 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880941434 GF On-Demand Anodyne TLR4 16 42 NC(=O)c1cc2cc(NC(=O)COC3CC3)ccc2[nH]1 ZINC000880941445 CD On-Demand Anodyne PYGL 72 42 NC(=O)c1cc2cc(NC(=O)COC3CC3)ccc2[nH]1 ZINC000880941445 CD On-Demand Anodyne ENPP1 66 32 CC1(C)CC[C@@H](CC(=O)Nc2ccc3[nH]c(C(N)=O)cc3c2)OC1 ZINC000880941447 EF On-Demand Anodyne ENPP1 40 32 O=C(Cn1c(S)nc2ccccc2c1=O)NCc1ccc(O)cc1 ZINC000880941452 ED On-Demand Anodyne F2 22 42 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@@H](N2CCCC2)C1 ZINC000880941460 GH On-Demand Anodyne L3MBTL3 86 44 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@H](N2CCCC2)C1 ZINC000880941461 GH On-Demand Anodyne L3MBTL3 86 44 CC1CN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941464 DG On-Demand Anodyne RBP4 54 37 CNC(=O)[C@@H]1CCC[C@H]1NC(=O)Nc1cnc2ccccc2c1Br ZINC000880941488 GG On-Demand Anodyne ADAM17 19 42 CNC(=O)[C@@H]1CCC[C@@H]1NC(=O)Nc1cnc2ccccc2c1Br ZINC000880941490 GG On-Demand Anodyne ADAM17 19 42 COC[C@@H](O)CCNC(=O)Nc1cnc2ccccc2c1Br ZINC000880941491 FF On-Demand Anodyne ADRB1 42 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880941501 GF On-Demand Anodyne TLR4 16 42 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC)CCCO ZINC000880941502 DE On-Demand Anodyne SOAT1 24 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)C(C)C)CC1 ZINC000880941515 FE On-Demand Anodyne P2RY12 46 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CCO)CC1 ZINC000880941526 EF On-Demand Anodyne RBP4 41 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(N(C)C)CC1 ZINC000880941533 EF On-Demand Anodyne RBP4 42 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880941537 GF On-Demand Anodyne P2RY12 23 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(Cc2ccncc2)CC1 ZINC000880941537 GF On-Demand Anodyne FAAH 25 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)N(C)C)CC1 ZINC000880941552 FD On-Demand Anodyne P2RY12 24 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](O)C1 ZINC000880941553 DD On-Demand Anodyne CCR3 41 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](O)C1 ZINC000880941554 DD On-Demand Anodyne CCR3 41 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2cc(C#N)ccn2)CC1 ZINC000880941559 GF On-Demand Mild P2RY12 35 48 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne EGFR 20 42 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne CNR2 15 42 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne CASR 41 37 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne UTS2R 21 46 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne HNMT 52 36 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne PTGDS 43 38 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne EPHX2 21 46 O=C(NCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880941561 GE On-Demand Anodyne HPGDS 26 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](Cc2noc(C)n2)C1 ZINC000880941566 GG On-Demand Anodyne CCR3 90 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](Cc2noc(C)n2)C1 ZINC000880941567 GG On-Demand Anodyne CCR3 90 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(c2nc(C)no2)CC1 ZINC000880941573 GG On-Demand Anodyne SMO 38 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(c2nc(C)no2)CC1 ZINC000880941573 GG On-Demand Anodyne ETHR 63 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000880941576 FD On-Demand Anodyne P2RY12 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000880941576 FD On-Demand Anodyne RBP4 35 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000880941576 FD On-Demand Anodyne TLR4 18 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(CC(C)(C)O)CC1 ZINC000880941578 FD On-Demand Anodyne P2RY12 23 40 O=C(Nc1cnc2ccccc2c1Br)N1CCOCC1 ZINC000880941585 EF On-Demand Anodyne NPY5R 17 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](c2cc[nH]n2)C1 ZINC000880941587 FG On-Demand Anodyne CCR3 44 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](c2cc[nH]n2)C1 ZINC000880941588 FG On-Demand Anodyne CCR3 44 33 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC)Cc1ccncc1 ZINC000880941770 EG On-Demand Anodyne SOAT1 17 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880941785 GF On-Demand Anodyne P2RY12 23 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(Cc2cccnc2)CC1 ZINC000880941785 GF On-Demand Anodyne FAAH 32 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(N(C)C(=O)OCC)CC1 ZINC000880941790 GG On-Demand Anodyne RBP4 40 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(C)=O)CC1 ZINC000880941791 ED On-Demand Anodyne P2RY12 26 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1CC1 ZINC000880941815 CF On-Demand Anodyne TLR4 16 44 O=C(CCCNC(=O)Nc1cnc2ccccc2c1Br)NC1CC1 ZINC000880941827 GG On-Demand Anodyne TNKS 61 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(NC(=O)C2CC2)CC1 ZINC000880941833 GF On-Demand Anodyne EPHX2 39 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(NC(=O)C2CC2)CC1 ZINC000880941833 GF On-Demand Anodyne CCR8 48 34 COC(=O)[C@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941834 GG On-Demand Anodyne CCR8 42 38 COC(=O)[C@@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941836 GG On-Demand Anodyne CCR8 42 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1c1cc(C)no1 ZINC000880941848 FH On-Demand Anodyne KCNA5 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1c1cc(C)no1 ZINC000880941850 FH On-Demand Anodyne KCNA5 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCN(C(=O)C(C)C)CC1 ZINC000880941856 GF On-Demand Anodyne P2RY12 37 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCCN(C)C1 ZINC000880941888 FF On-Demand Anodyne CCR3 82 36 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCCN(C)C1 ZINC000880941890 FF On-Demand Anodyne CCR3 82 36 CCN1CCC(NC(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880941899 GH On-Demand Anodyne DRD4 15 45 CCN1CCC(NC(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880941899 GH On-Demand Anodyne SIGMAR1 17 40 CCN1CCC(NC(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880941899 GH On-Demand Anodyne EPHX2 35 41 CCN1CCC(NC(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880941899 GH On-Demand Anodyne CCR8 45 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CCO)C1 ZINC000880941908 EF On-Demand Anodyne CCR3 67 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CCO)C1 ZINC000880941910 EF On-Demand Anodyne CCR3 67 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880941912 GF On-Demand Anodyne P2RY12 28 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880941912 GF On-Demand Anodyne TLR4 16 43 COCCN(CC1CCN(C)CC1)C(=O)CNC(=O)c1ccc(O)cc1 ZINC000880941934 FC On-Demand Anodyne CACNA1I 53 34 COCCN(CC1CCN(C)CC1)C(=O)CNC(=O)c1ccc(O)cc1 ZINC000880941934 FC On-Demand Anodyne ACKR3 56 31 Cc1noc(C2CN(C(=O)Nc3cnc4ccccc4c3Br)C2)n1 ZINC000880941936 GG On-Demand Anodyne SMO 39 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCS(=O)(=O)[C@@H](C)C1 ZINC000880941939 FD On-Demand Anodyne RBP4 40 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCS(=O)(=O)[C@H](C)C1 ZINC000880941941 FD On-Demand Anodyne RBP4 40 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)Cc1cnn(C)c1 ZINC000880941947 EE On-Demand Anodyne PLA2G7 53 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC12CC2 ZINC000880941955 EE On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCCC12CC2 ZINC000880941957 EE On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H]1CCCC12CC2 ZINC000880941959 EE On-Demand Anodyne PAPA1_CARPA 33 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H]1CCCC12CC2 ZINC000880941960 EE On-Demand Anodyne PAPA1_CARPA 33 41 O=C(NCCN1C(=O)CCC1=O)Nc1cnc2ccccc2c1Br ZINC000880941963 GE On-Demand Anodyne UTS2R 17 41 O=C(N[C@@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941964 CE On-Demand Anodyne JAK3 20 46 O=C(N[C@@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941964 CE On-Demand Anodyne JAK1 16 46 O=C(N[C@@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941964 CE On-Demand Anodyne TYK2 24 46 O=C(N[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941965 CE On-Demand Anodyne JAK3 20 46 O=C(N[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941965 CE On-Demand Anodyne JAK1 16 46 O=C(N[C@H]1CCCC12CC2)c1cccn2nccc12 ZINC000880941965 CE On-Demand Anodyne TYK2 24 46 O=C(Nc1cnc2ccccc2c1Br)N1CCC2(CCOCC2)C1 ZINC000880941966 GI On-Demand Anodyne EPHX2 25 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941967 GG On-Demand Anodyne EPHX2 31 49 CCC(=O)N1CC[C@@H](NC(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941967 GG On-Demand Anodyne CCR8 74 38 CCC(=O)N1CC[C@H](NC(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941968 GG On-Demand Anodyne EPHX2 31 49 CCC(=O)N1CC[C@H](NC(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880941968 GG On-Demand Anodyne CCR8 74 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(c2ncc[nH]2)CC1 ZINC000880941982 FG On-Demand Anodyne HTR2B 18 41 COc1ccc(-c2nnc(S)n2CC(=O)NCc2ccc(O)cc2)cc1 ZINC000880941989 FE On-Demand Anodyne AVPR1B 44 36 COc1ccc(-c2nnc(S)n2CC(=O)NCc2ccc(O)cc2)cc1 ZINC000880941989 FE On-Demand Anodyne PROKR1 62 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)C(C)(C)C)CC1 ZINC000880941992 GF On-Demand Anodyne P2RY12 25 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CC(C)(C)C ZINC000880942013 EF On-Demand Anodyne SOAT1 18 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)c2ccco2)CC1 ZINC000880942024 GF On-Demand Anodyne P2RY12 21 40 C[C@H]1[C@H](C(=O)Nc2ccc3[nH]c(C(N)=O)cc3c2)CCN1C ZINC000880942067 DD On-Demand Anodyne PYGL 50 39 C[C@@H]1[C@@H](C(=O)Nc2ccc3[nH]c(C(N)=O)cc3c2)CCN1C ZINC000880942069 DD On-Demand Anodyne PYGL 50 39 COCCN(CC1CCN(C)CC1)C(=O)c1c[nH]c2ccccc2c1=O ZINC000880942095 FD On-Demand Anodyne HTR4 40 43 COCCN(CC1CCN(C)CC1)C(=O)c1c[nH]c2ccccc2c1=O ZINC000880942095 FD On-Demand Anodyne HTR1F 61 35 COCCN(CC1CCN(C)CC1)C(=O)c1c[nH]c2ccccc2c1=O ZINC000880942095 FD On-Demand Anodyne CFTR 36 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](CCO)C1 ZINC000880942097 DE On-Demand Anodyne CCR3 37 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](CCO)C1 ZINC000880942099 DE On-Demand Anodyne CCR3 37 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880942117 GF On-Demand Mild P2RY12 46 56 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880942117 GF On-Demand Mild PDGFRB 37 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ncccc2C#N)CC1 ZINC000880942117 GF On-Demand Mild RBP4 18 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(NC(C)C)CC1 ZINC000880942172 FF On-Demand Anodyne CCR8 58 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1C2CCC1CC2 ZINC000880942173 DG On-Demand Anodyne TLR4 15 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)O[C@H](C)C1 ZINC000880942174 DF On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)O[C@H](C)C1 ZINC000880942175 DF On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)O[C@@H](C)C1 ZINC000880942176 DF On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC1 ZINC000880942182 CF On-Demand Anodyne P2RY12 26 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2cnc(C(C)C)nc2C1 ZINC000880942203 GH On-Demand Anodyne MAPK1 59 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2cnc(C(C)C)nc2C1 ZINC000880942203 GH On-Demand Anodyne P2RY14 40 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C#N)CC1 ZINC000880942224 DF On-Demand Mild P2RY12 31 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1CO ZINC000880942227 DD On-Demand Anodyne TLR4 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1CO ZINC000880942228 DD On-Demand Anodyne TLR4 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCC[C@@H]2C1 ZINC000880942229 EE On-Demand Anodyne CCR3 20 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCC[C@H]2C1 ZINC000880942230 EE On-Demand Anodyne CCR3 20 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(CC)CC1 ZINC000880942249 EF On-Demand Anodyne S1PR2 32 45 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CC1CC1 ZINC000880942250 DE On-Demand Anodyne TLR4 15 42 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1CCC1 ZINC000880942256 CG On-Demand Anodyne TLR4 17 45 CN1CCN(C(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880942261 EF On-Demand Anodyne HTR3A 21 41 CN1CCN(C(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880942261 EF On-Demand Anodyne PDGFRB 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCO[C@H](CC)C1 ZINC000880942262 DF On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCO[C@@H](CC)C1 ZINC000880942263 DF On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCOCC1 ZINC000880942272 CD On-Demand Anodyne P2RY12 23 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CO)CC1 ZINC000880942273 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCCC[C@H]2C1 ZINC000880942280 EF On-Demand Anodyne CCR3 17 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCCC[C@H]2C1 ZINC000880942280 EF On-Demand Anodyne L3MBTL3 51 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCCC[C@@H]2C1 ZINC000880942281 EF On-Demand Anodyne CCR3 17 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2CCCC[C@@H]2C1 ZINC000880942281 EF On-Demand Anodyne L3MBTL3 51 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C)CC1 ZINC000880942284 DD On-Demand Anodyne P2RY12 27 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1C(=O)NC1CC1 ZINC000880942289 FE On-Demand Anodyne CCR3 18 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1C(=O)NC1CC1 ZINC000880942289 FE On-Demand Anodyne LGMN 93 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1C(=O)NC1CC1 ZINC000880942290 FE On-Demand Anodyne CCR3 18 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1C(=O)NC1CC1 ZINC000880942290 FE On-Demand Anodyne LGMN 93 37 COCCN(CC1CCN(C)CC1)C(=O)c1ccc2c(O)nc(S)nc2c1 ZINC000880942310 GE On-Demand Anodyne ACKR3 62 32 CC(=O)NCCCNC(=O)Nc1cnc2ccccc2c1Br ZINC000880942315 FF On-Demand Anodyne MTNR1A 51 43 CC(=O)NCCCNC(=O)Nc1cnc2ccccc2c1Br ZINC000880942315 FF On-Demand Anodyne MTNR1B 49 43 O=C(NCCCN1CCCC1=O)Nc1cnc2ccccc2c1Br ZINC000880942319 GG On-Demand Anodyne TYRO3 21 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CCCO ZINC000880942326 ED On-Demand Anodyne SOAT1 25 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1C(=O)N(C)C ZINC000880942338 FE On-Demand Anodyne LGMN 59 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1C(=O)N(C)C ZINC000880942339 FE On-Demand Anodyne LGMN 59 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](O)C1 ZINC000880942361 CD On-Demand Anodyne RBP4 39 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](O)C1 ZINC000880942361 CD On-Demand Anodyne TLR4 15 40 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(F)cc2C(=O)OCC)CC1 ZINC000880942370 GD On-Demand Anodyne ACOX1 40 34 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc(F)cc2C(=O)OCC)CC1 ZINC000880942370 GD On-Demand Anodyne ABCB1 43 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)[C@@H]2CCCO2)CC1 ZINC000880942381 GD On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)[C@H]2CCCO2)CC1 ZINC000880942382 GD On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](NC(=O)C(C)C)C1 ZINC000880942385 GF On-Demand Anodyne CCR3 44 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](NC(=O)C(C)C)C1 ZINC000880942385 GF On-Demand Anodyne BIRC2 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](NC(=O)C(C)C)C1 ZINC000880942386 GF On-Demand Anodyne CCR3 44 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](NC(=O)C(C)C)C1 ZINC000880942386 GF On-Demand Anodyne BIRC2 34 40 COCCN(CC1CCN(C)CC1)C(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880942387 GG On-Demand Anodyne CACNA1I 51 35 COCCN(CC1CCN(C)CC1)C(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880942387 GG On-Demand Anodyne ACKR3 65 35 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)C1CC1 ZINC000880942391 DD On-Demand Anodyne TLR4 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(Nc2cccnn2)CC1 ZINC000880942407 GF On-Demand Anodyne FAAH 27 42 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CCN1CCOCC1 ZINC000880942414 FD On-Demand Anodyne CASR 50 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CCN1CCOCC1 ZINC000880942414 FD On-Demand Anodyne EPHX2 18 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)CC1 ZINC000880942415 DD On-Demand Anodyne RBP4 40 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)CC1 ZINC000880942415 DD On-Demand Anodyne TLR4 15 40 COCCN(CC1CCN(C)CC1)C(=O)c1ccc2nc[nH]c2c1 ZINC000880942422 ED On-Demand Anodyne ACKR3 72 36 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC)C1CC1 ZINC000880942426 CG On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCCOC)Cc1ccncc1 ZINC000880942427 GG On-Demand Anodyne SOAT1 23 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1c1cccnc1 ZINC000880942444 FH On-Demand Anodyne CHRNA7 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1c1cccnc1 ZINC000880942445 FH On-Demand Anodyne CHRNA7 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCCCO1 ZINC000880942447 EG On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCCCO1 ZINC000880942448 EG On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(C)C)CC1 ZINC000880942449 EF On-Demand Anodyne P2RY12 27 42 COc1cccc([C@H](O)C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)c1 ZINC000880942458 GH On-Demand Anodyne MTNR1B 16 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCCO1 ZINC000880942471 DF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCCO1 ZINC000880942473 DF On-Demand Anodyne TLR4 15 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2nccnn2)CC1 ZINC000880942479 ED On-Demand Anodyne FAAH 24 44 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1ccc3c(n1)CCCC3)CC2 ZINC000880942483 FH On-Demand Anodyne P2RY14 44 31 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880942503 FH On-Demand Anodyne EPHX2 18 52 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880942504 FH On-Demand Anodyne EPHX2 18 52 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne EGFR 25 45 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne CASR 42 36 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne BCHE 15 41 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne CCR3 25 42 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne UTS2R 18 41 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne HNMT 75 40 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne EPHX2 23 42 O=C(NCCCN1CCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942551 GF On-Demand Anodyne HPGDS 22 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CC(C)(C)S(C)(=O)=O ZINC000880942557 FE On-Demand Anodyne TLR4 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1CCC(CO)CC1 ZINC000880942560 FG On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC=C(C)C1 ZINC000880942563 DG On-Demand Anodyne TLR4 15 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(C(C)C)C1 ZINC000880942566 DG On-Demand Anodyne RBP4 28 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(C2CCOCC2)C1 ZINC000880942583 FF On-Demand Anodyne RBP4 47 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2cccc(NC(C)=O)c2C1 ZINC000880942586 GH On-Demand Anodyne P2RY14 45 38 COCCN(CC1CCN(C)CC1)C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880942589 GE On-Demand Anodyne HTR1F 46 33 COCCN(CC1CCN(C)CC1)C(=O)c1cc2cc(F)ccc2[nH]c1=O ZINC000880942589 GE On-Demand Anodyne ACKR3 53 35 C[C@@H](CC[S@](C)=O)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942598 GG On-Demand Anodyne ANPEP 17 41 C[C@@H](CC[S@@](C)=O)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942600 GG On-Demand Anodyne ANPEP 17 41 C[C@H](CC[S@](C)=O)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942602 GG On-Demand Anodyne ANPEP 17 41 C[C@H](CC[S@@](C)=O)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942603 GG On-Demand Anodyne ANPEP 17 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CCN(C)C1CC1 ZINC000880942604 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2ncnc(OCC)c2C1 ZINC000880942606 GF On-Demand Anodyne P2RY14 49 38 O=C(NCCNC(=O)C1CC1)Nc1cnc2ccccc2c1Br ZINC000880942633 GF On-Demand Anodyne MTNR1A 19 42 O=C(NCCNC(=O)C1CC1)Nc1cnc2ccccc2c1Br ZINC000880942633 GF On-Demand Anodyne MTNR1B 15 42 COc1cc(NC(=O)c2ccccc2)c(C(=O)NCCc2ccc(Br)s2)cc1OC ZINC000880942645 JJ On-Demand Anodyne GPR35 48 38 COCCN(CC1CCN(C)CC1)C(=O)CN(C(C)=O)c1ccccc1 ZINC000880942650 FD On-Demand Anodyne ACKR3 56 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1CCO ZINC000880942655 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1CCO ZINC000880942657 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](C(F)(F)F)[C@H](CO)C1 ZINC000880942663 GG On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](C(F)(F)F)[C@H](CO)C1 ZINC000880942665 GG On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880942667 GG On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880942669 GG On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)C1CCC1 ZINC000880942677 DE On-Demand Anodyne TLR4 16 44 COCCN(CC1CCN(C)CC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880942687 GE On-Demand Anodyne HTR1F 58 39 COCCN(CC1CCN(C)CC1)C(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880942687 GE On-Demand Anodyne ACKR3 40 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880942698 FF On-Demand Anodyne RBP4 57 46 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880942700 FF On-Demand Anodyne RBP4 57 46 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880942702 FF On-Demand Anodyne RBP4 57 46 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880942703 FF On-Demand Anodyne RBP4 57 46 CCOC(=O)c1cc(F)ccc1NC(=O)N(C[C@H](C)O)C1CC1 ZINC000880942710 DE On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C[C@@H](C)O)C1CC1 ZINC000880942712 DE On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@@H]2CCOC2)C1 ZINC000880942714 EF On-Demand Anodyne RBP4 41 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@H]2CCOC2)C1 ZINC000880942716 EF On-Demand Anodyne RBP4 41 42 O=C(Nc1cnc2ccccc2c1Br)N1CCN(CCO)CC1 ZINC000880942717 GE On-Demand Anodyne FAAH 21 40 O=C(Nc1cnc2ccccc2c1Br)N1CCN(CCO)CC1 ZINC000880942717 GE On-Demand Anodyne HNMT 50 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2nncn2C)CC1 ZINC000880942720 GD On-Demand Anodyne P2RY12 23 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C)C(=O)C1 ZINC000880942726 DD On-Demand Anodyne P2RY12 21 40 O=C(NCc1ccc(O)cc1)c1ccc(Cl)c(S(=O)(=O)Nc2ccc(F)cc2)c1 ZINC000880942736 IH On-Demand Anodyne SGK1 46 33 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne EGFR 19 40 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne BCHE 15 40 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne UTS2R 20 44 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne HNMT 80 38 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne EPHX2 20 44 O=C(NCCN1CCCOCC1)Nc1cnc2ccccc2c1Br ZINC000880942737 GF On-Demand Anodyne HPGDS 24 43 C[C@H](CCO)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942748 EF On-Demand Anodyne ANPEP 18 42 C[C@@H](CCO)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880942749 EF On-Demand Anodyne ANPEP 18 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCn2c(nnc2C(C)(C)C)C1 ZINC000880942755 GF On-Demand Anodyne P2RX7 23 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C)(O)CC1 ZINC000880942768 DE On-Demand Anodyne CACNA1H 41 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C)(O)CC1 ZINC000880942768 DE On-Demand Anodyne S1PR2 30 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nn(CC)c(=O)cc2C1 ZINC000880942770 GE On-Demand Anodyne P2RY14 44 37 O=C(Nc1ccc2c(n1)CCCC2)N1CC(c2ccccc2)C1 ZINC000880942845 DH On-Demand Anodyne RBP4 45 32 COCCN(CC1CCN(C)CC1)C(=O)c1ccc(Oc2cc(C)ccn2)cc1 ZINC000880942943 GH On-Demand Anodyne ACKR3 62 31 O=C(NCC(=O)N1CCCCC1)Nc1cnc2ccccc2c1Br ZINC000880942978 GG On-Demand Anodyne PREP 20 43 O=C(NCC(=O)N1CCCCC1)Nc1cnc2ccccc2c1Br ZINC000880942978 GG On-Demand Anodyne PRMT3 18 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OCC)CC1 ZINC000880942979 EG On-Demand Anodyne RBP4 40 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OCC)CC1 ZINC000880942979 EG On-Demand Anodyne SCD1 19 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nn(C)c(=O)cc2C1 ZINC000880942985 FD On-Demand Anodyne P2RY14 40 35 CCOC(=O)c1cc(F)ccc1NC(=O)NOC1CCC1 ZINC000880942987 CF On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](O)[C@H](C)C1 ZINC000880942989 DD On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)[C@@H](O)C1 ZINC000880942991 DD On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)[C@H](O)C1 ZINC000880942993 DD On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)[C@@H](O)C1 ZINC000880942995 DD On-Demand Anodyne RBP4 27 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(C)(=O)=O)[C@H](C)C1 ZINC000880942997 GD On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2[C@H](CCCN2C)C1 ZINC000880942999 FF On-Demand Anodyne RBP4 46 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2[C@H](CCCN2C)C1 ZINC000880943001 FF On-Demand Anodyne RBP4 46 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2[C@@H](CCCN2C)C1 ZINC000880943003 FF On-Demand Anodyne RBP4 46 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2[C@@H](CCCN2C)C1 ZINC000880943005 FF On-Demand Anodyne RBP4 46 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2C(=O)N(CC)C(=O)[C@@H]2C1 ZINC000880943017 GD On-Demand Anodyne SMO 31 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN2C(=O)N(CC)C(=O)[C@H]2C1 ZINC000880943019 GD On-Demand Anodyne SMO 31 40 O=C(Nc1cnc2ccccc2c1Br)N1CCN2CCC[C@@H]2C1 ZINC000880943030 GG On-Demand Anodyne HRH3 18 40 O=C(Nc1cnc2ccccc2c1Br)N1CCN2CCC[C@H]2C1 ZINC000880943032 GG On-Demand Anodyne HRH3 18 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCOCCO)C1CCC1 ZINC000880943037 FE On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)C[C@@H](O)C1 ZINC000880943039 DE On-Demand Anodyne RBP4 48 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)C[C@H](O)C1 ZINC000880943041 DE On-Demand Anodyne RBP4 48 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](O)C[C@@H](C)C1 ZINC000880943042 DE On-Demand Anodyne RBP4 48 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)C[C@@H](O)C1 ZINC000880943044 DE On-Demand Anodyne RBP4 48 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CC(C)(C)CO ZINC000880943055 EE On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)[C@@H]1CCN(S(C)(=O)=O)C1 ZINC000880943056 GD On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)[C@H]1CCN(S(C)(=O)=O)C1 ZINC000880943058 GD On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2CC[C@H](C1)O2 ZINC000880943060 DE On-Demand Anodyne RBP4 33 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880943062 GG On-Demand Anodyne P2RY12 20 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880943062 GG On-Demand Anodyne RBP4 42 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880943064 GG On-Demand Anodyne P2RY12 20 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880943064 GG On-Demand Anodyne RBP4 42 42 CCOC(=O)c1cc(F)ccc1NC(=O)NOC1CCOCC1 ZINC000880943068 EE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]2CN(C)C[C@H]21 ZINC000880943071 EF On-Demand Anodyne CCR3 47 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nccnc2C1 ZINC000880943075 EE On-Demand Anodyne P2RY14 49 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2[C@@H](CO)[C@@H]2C1 ZINC000880943083 DD On-Demand Anodyne RBP4 33 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)C(O)[C@H](C)C1 ZINC000880943085 EE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)[C@@H](O)[C@H](C)C1 ZINC000880943087 EE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)C(O)[C@@H](C)C1 ZINC000880943089 EE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)[C@@H](C)O)CC1 ZINC000880943090 FD On-Demand Anodyne P2RY12 42 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(C(=O)[C@H](C)O)CC1 ZINC000880943091 FD On-Demand Anodyne P2RY12 42 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nc(COC)ncc2C1 ZINC000880943107 GF On-Demand Anodyne P2RY14 44 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@@H](C)C(=O)OCC)C1 ZINC000880943108 FF On-Demand Anodyne RBP4 35 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@H](C)C(=O)OCC)C1 ZINC000880943110 FF On-Demand Anodyne RBP4 35 43 CNc1nc(C(=O)N(CCOC)CC2CCN(C)CC2)cs1 ZINC000880943113 ED On-Demand Anodyne TRPC6 42 34 NC(=O)c1cc(F)ccc1N1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880943132 GF On-Demand Anodyne SLC27A1 41 34 O=C(Nc1ccc2c(n1)CCCC2)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880943148 FF On-Demand Anodyne ETHR 40 34 O=C(Nc1ccc2c(n1)CCCC2)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880943149 FF On-Demand Anodyne ETHR 40 34 O=C(NNc1ccc(F)cn1)Nc1ccc2c(n1)CCCC2 ZINC000880943162 DF On-Demand Reactive SLC27A1 42 35 Cn1nnnc1C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880943179 ED On-Demand Anodyne HTR1F 57 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](NC(=O)N(C)C)C1 ZINC000880943193 GE On-Demand Anodyne CCR3 30 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](NC(=O)N(C)C)C1 ZINC000880943196 GE On-Demand Anodyne CCR3 30 40 NC(=O)Cc1cccc2c1CCN(C(=O)Nc1ccc3c(n1)CCCC3)C2 ZINC000880943212 FF On-Demand Anodyne P2RY14 41 31 CC[C@H]1CCC[C@@]1(C)C(=O)Nc1ccc2[nH]c(C(N)=O)cc2c1 ZINC000880943321 DG On-Demand Anodyne PYGL 51 38 CC[C@@H]1CCC[C@@]1(C)C(=O)Nc1ccc2[nH]c(C(N)=O)cc2c1 ZINC000880943323 DG On-Demand Anodyne PYGL 51 38 CC[C@H]1CCC[C@]1(C)C(=O)Nc1ccc2[nH]c(C(N)=O)cc2c1 ZINC000880943326 DG On-Demand Anodyne PYGL 51 38 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880943350 FF On-Demand Anodyne HTR1F 59 33 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H](N2CCOCC2)C1 ZINC000880943418 ED On-Demand Anodyne L3MBTL3 61 38 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H](N2CCOCC2)C1 ZINC000880943419 ED On-Demand Anodyne L3MBTL3 61 38 O=C(Cn1c(SC(F)F)nc2ccccc21)NCc1ccc(O)cc1 ZINC000880943436 FG On-Demand Anodyne FABI 49 32 Cc1csc([C@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C2)n1 ZINC000880943439 EH On-Demand Anodyne HTR1F 42 32 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc3c(n1)CCCC3)CC2 ZINC000880943462 FH On-Demand Anodyne P2RY14 45 32 C[C@@H](CCCO)NC(=O)Nc1cnc2ccccc2c1Br ZINC000880943517 FG On-Demand Anodyne ANPEP 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880943528 GF On-Demand Anodyne CHRNA4 25 47 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2OCC[C@@H]2C1 ZINC000880943530 EF On-Demand Anodyne RBP4 46 41 CCCN(CC(C)(C)O)C(=O)Nc1ccc(F)cc1C(=O)OCC ZINC000880943532 EG On-Demand Anodyne SOAT1 18 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CC#N)C1 ZINC000880943534 EG On-Demand Mild P2RY12 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CC#N)C1 ZINC000880943534 EG On-Demand Mild CCR3 44 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CC#N)C1 ZINC000880943536 EG On-Demand Mild P2RY12 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CC#N)C1 ZINC000880943536 EG On-Demand Mild CCR3 44 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nc(C3CC3)ncc2C1 ZINC000880943538 GG On-Demand Anodyne MAPK1 42 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nc(C3CC3)ncc2C1 ZINC000880943538 GG On-Demand Anodyne P2RY14 44 35 COCCN(CC1CCN(C)CC1)C(=O)CC[C@H]1CCCCN1C ZINC000880943539 EE On-Demand Anodyne ACKR3 66 34 COCCN(CC1CCN(C)CC1)C(=O)CC[C@@H]1CCCCN1C ZINC000880943540 EE On-Demand Anodyne ACKR3 66 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2nc(C)ns2)CC1 ZINC000880943548 GF On-Demand Anodyne P2RY12 29 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCN(C(=O)CC(C)C)CC1 ZINC000880943554 GG On-Demand Anodyne P2RY12 20 40 CN1CC[C@H](NC(=O)Nc2cnc3ccccc3c2Br)C1=O ZINC000880943557 FE On-Demand Anodyne TRPV1 16 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CCNC(C)=O)C1 ZINC000880943564 GF On-Demand Anodyne CCR3 67 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CCNC(C)=O)C1 ZINC000880943566 GF On-Demand Anodyne CCR3 67 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2cccc(C#N)n2)CC1 ZINC000880943568 GF On-Demand Mild P2RY12 44 49 COCCN(CC1CCN(C)CC1)C(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880943570 FE On-Demand Anodyne ACKR3 44 31 COCCN(CC1CCN(C)CC1)C(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880943572 FE On-Demand Anodyne ACKR3 44 31 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nnc(OC)cc2C1 ZINC000880943578 FE On-Demand Anodyne P2RY14 43 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1C(=O)NC ZINC000880943582 ED On-Demand Anodyne LGMN 104 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1C(=O)NC ZINC000880943584 ED On-Demand Anodyne LGMN 104 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880943589 EF On-Demand Anodyne RBP4 54 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2COC[C@H]2C1 ZINC000880943591 EF On-Demand Anodyne RBP4 54 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2COC[C@@H]2C1 ZINC000880943594 EF On-Demand Anodyne RBP4 54 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2COC[C@H]2C1 ZINC000880943596 EF On-Demand Anodyne RBP4 54 42 COCCN(CC1CCN(C)CC1)C(=O)c1cc2ccccc2cc1F ZINC000880943608 FG On-Demand Anodyne CHRNA10 40 32 COCCN(CC1CCN(C)CC1)C(=O)c1cc2ccccc2cc1F ZINC000880943608 FG On-Demand Anodyne ACKR3 67 35 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H](O)C1CC1 ZINC000880943620 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H](O)C1CC1 ZINC000880943621 DE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@H]1c1nc(C)no1 ZINC000880943625 GG On-Demand Anodyne CPT1A 84 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@@H]1c1nc(C)no1 ZINC000880943626 GG On-Demand Anodyne CPT1A 84 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2cc(Cl)nnc2C1 ZINC000880943634 GG On-Demand Anodyne MAPK1 47 35 CCOC(=O)c1cc(F)ccc1NC(=O)NOC1CCCC1 ZINC000880943635 DF On-Demand Anodyne TLR4 17 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@H](F)C(=O)OCC)C1 ZINC000880943636 FE On-Demand Anodyne RBP4 35 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC([C@@H](F)C(=O)OCC)C1 ZINC000880943637 FE On-Demand Anodyne RBP4 35 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](OC)CC1 ZINC000880943638 EG On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](OC)CC1 ZINC000880943639 EG On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1CC(O)C1 ZINC000880943642 DD On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](S(C)(=O)=O)C1 ZINC000880943643 FE On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](S(C)(=O)=O)C1 ZINC000880943644 FE On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CCO)CC1 ZINC000880943654 FG On-Demand Anodyne CCR3 44 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CCO)CC1 ZINC000880943655 FG On-Demand Anodyne CCR3 44 38 Cn1ncc(NC(=O)Nc2ccc3c(n2)CCCC3)c1C1CC1 ZINC000880943673 DG On-Demand Anodyne HTR1F 53 34 O=C(NCc1nc(-c2ccncc2)cs1)Nc1ccc2c(n1)CCCC2 ZINC000880943693 FH On-Demand Anodyne ROCK1 23 48 O=C(NCc1nc(-c2ccncc2)cs1)Nc1ccc2c(n1)CCCC2 ZINC000880943693 FH On-Demand Anodyne ROCK2 16 48 CN1CCC[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1=O ZINC000880943714 DD On-Demand Anodyne HTR1F 53 36 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCCN(CCN2CCOCC2)C1 ZINC000880943761 GD On-Demand Anodyne EPHX2 18 44 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCCN(CCN2CCOCC2)C1 ZINC000880943762 GD On-Demand Anodyne EPHX2 18 44 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC13CC3)C2 ZINC000880943810 CG On-Demand Anodyne MTNR1A 26 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@@H]1CCCC13CC3)C2 ZINC000880943810 CG On-Demand Anodyne MTNR1B 25 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCC13CC3)C2 ZINC000880943812 CG On-Demand Anodyne MTNR1A 26 40 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCCC13CC3)C2 ZINC000880943812 CG On-Demand Anodyne MTNR1B 25 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc2ccccc2c1Br ZINC000880943815 GF On-Demand Anodyne UL80 29 45 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnc2ccccc2c1Br ZINC000880943815 GF On-Demand Anodyne PREP 48 38 C=CC(C)(C)CC(=O)Nc1ccc2[nH]c(C(N)=O)cc2c1 ZINC000880943816 CF On-Demand Mild ENPP1 57 33 O=C(Nc1cnc2ccccc2c1Br)N[C@@H]1CCCCNC1=O ZINC000880943826 GF On-Demand Anodyne CDK5 23 40 O=C(Nc1cnc2ccccc2c1Br)N[C@H]1CCCCNC1=O ZINC000880943827 GF On-Demand Anodyne CDK5 23 40 O=C(N[C@H]1CCCC12CC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880943836 DF On-Demand Anodyne GABRA1 18 43 O=C(N[C@H]1CCCC12CC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880943836 DF On-Demand Anodyne GABRA2 16 43 O=C(N[C@@H]1CCCC12CC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880943837 DF On-Demand Anodyne GABRA1 18 43 O=C(N[C@@H]1CCCC12CC2)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880943837 DF On-Demand Anodyne GABRA2 16 43 O=C(N[C@H]1CCCC12CC2)c1cccnc1I ZINC000880943841 EF On-Demand Anodyne G2YM83_BOTF4 52 32 O=C(N[C@@H]1CCCC12CC2)c1cccnc1I ZINC000880943842 EF On-Demand Anodyne G2YM83_BOTF4 52 32 O=C(Nc1cnc2ccccc2c1Br)N1CC(CC(F)(F)F)C1 ZINC000880943843 GI On-Demand Anodyne RBP4 55 36 O=C(CNC(=O)Nc1cnc2ccccc2c1Br)NC1CCCC1 ZINC000880943846 GG On-Demand Anodyne TNKS 45 31 O=C(Nc1cnc2ccccc2c1Br)N1CC(C2CCOCC2)C1 ZINC000880943866 GH On-Demand Anodyne RBP4 46 34 COCCN(CC1CCN(C)CC1)C(=O)c1cc(C(F)(F)F)ccn1 ZINC000880943904 FF On-Demand Anodyne LIPG 47 36 COCCN(CC1CCN(C)CC1)C(=O)c1cc(C(F)(F)F)ccn1 ZINC000880943904 FF On-Demand Anodyne ACKR3 60 31 CN1CC[C@H]2CN(C(=O)Nc3ccc4c(n3)CCCC4)CC[C@H]21 ZINC000880943909 DF On-Demand Anodyne HTR1F 54 31 CN1CC[C@H]2CN(C(=O)Nc3ccc4c(n3)CCCC4)CC[C@@H]21 ZINC000880943912 DF On-Demand Anodyne HTR1F 54 31 CCOC(=O)c1cc(F)ccc1NC(=O)NOCCOC ZINC000880943916 DD On-Demand Anodyne PYGL 17 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCN(C(C)=O)C1 ZINC000880943924 FE On-Demand Anodyne CCR3 53 35 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCN(C(C)=O)C1 ZINC000880943926 FE On-Demand Anodyne CCR3 53 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880943929 GF On-Demand Anodyne L3MBTL3 57 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880943931 GF On-Demand Anodyne L3MBTL3 57 35 O=C(Nc1cnc2ccccc2c1Br)N1CC([C@@H]2CCOC2)C1 ZINC000880943942 GG On-Demand Anodyne RBP4 45 34 O=C(Nc1cnc2ccccc2c1Br)N1CC([C@H]2CCOC2)C1 ZINC000880943946 GG On-Demand Anodyne RBP4 45 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2cnccc2C#N)CC1 ZINC000880943949 GF On-Demand Mild P2RY12 38 50 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2C[C@@H]2C1 ZINC000880943954 DF On-Demand Anodyne RBP4 60 48 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2C[C@H]2C1 ZINC000880943956 DF On-Demand Anodyne RBP4 60 48 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2C[C@H]2C1 ZINC000880943959 DF On-Demand Anodyne RBP4 60 48 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2C[C@@H]2C1 ZINC000880943961 DF On-Demand Anodyne RBP4 60 48 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](OC)C1 ZINC000880943966 DF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](OC)C1 ZINC000880943969 DF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CN2CCOCC2)C1 ZINC000880943978 GF On-Demand Anodyne CCR3 73 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(c2ccc(C#N)nc2)CC1 ZINC000880943984 GF On-Demand Mild P2RY12 35 46 CCCCN(CCCO)C(=O)Nc1ccc(F)cc1C(=O)OCC ZINC000880943989 EG On-Demand Anodyne SOAT1 30 44 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880944010 GF On-Demand Anodyne HTR7 18 42 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880944010 GF On-Demand Anodyne CCKBR 25 44 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(-c3ccccc3)c(O)nc2c1 ZINC000880944010 GF On-Demand Anodyne NAMPT 44 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880944032 EF On-Demand Anodyne CCR3 45 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880944033 EF On-Demand Anodyne CCR3 45 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](OCCO)C1 ZINC000880944035 FE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](OCCO)C1 ZINC000880944036 FE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(=O)N(C)CC1 ZINC000880944038 ED On-Demand Anodyne P2RY12 23 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CC1CCOCC1 ZINC000880944045 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CCOC)CC1 ZINC000880944049 FG On-Demand Anodyne RBP4 38 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](O)[C@H](OC)C1 ZINC000880944060 ED On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(CCO)CC1 ZINC000880944061 ED On-Demand Anodyne P2RY12 22 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880944073 GI On-Demand Anodyne SMO 37 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880944073 GI On-Demand Anodyne ETHR 55 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(CCC#N)CC1 ZINC000880944081 EE On-Demand Mild P2RY12 27 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2ncncc2C1 ZINC000880944089 EE On-Demand Anodyne P2RY12 16 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2ncncc2C1 ZINC000880944089 EE On-Demand Anodyne P2RY14 50 38 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C(C)C ZINC000880944094 CF On-Demand Anodyne TLR4 15 41 O=C(NCc1ccc(O)cc1)c1ccc2c(c1)-c1ccccc1C2 ZINC000880944096 DH On-Demand Anodyne NAMPT 24 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCS(C)(=O)=O)C1CC1 ZINC000880944099 FE On-Demand Anodyne TLR4 17 46 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880944130 EE On-Demand Anodyne L3MBTL3 58 33 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880944132 EE On-Demand Anodyne L3MBTL3 58 33 CN1CCN(C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)CC1 ZINC000880944161 FE On-Demand Anodyne HTR1F 69 36 CN1CCN(C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)CC1 ZINC000880944161 FE On-Demand Anodyne L3MBTL3 84 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(N2CCN(C)CC2)CC1 ZINC000880944234 GE On-Demand Anodyne L3MBTL3 55 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880944250 CF On-Demand Anodyne DPP4 21 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880944250 CF On-Demand Anodyne DPP7 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880944250 CF On-Demand Anodyne RBP4 40 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880944250 CF On-Demand Anodyne CCR8 46 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H](F)C1 ZINC000880944250 CF On-Demand Anodyne TLR4 15 40 COCC1CCN(C(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880944252 GH On-Demand Anodyne PTPN2 21 40 COCC1CCN(C(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880944252 GH On-Demand Anodyne PTPN1 18 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880944255 CF On-Demand Anodyne DPP4 21 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880944255 CF On-Demand Anodyne DPP7 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880944255 CF On-Demand Anodyne RBP4 40 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880944255 CF On-Demand Anodyne CCR8 46 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](F)C1 ZINC000880944255 CF On-Demand Anodyne TLR4 15 40 C[C@@H]1[C@H](C(=O)NNC(=O)Nc2ccc3c(n2)CCCC3)CCCN1C ZINC000880944261 ED On-Demand Reactive HTR1F 46 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(NC2CCOCC2)CC1 ZINC000880944263 GF On-Demand Anodyne CCR8 43 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(NC2CCOCC2)CC1 ZINC000880944263 GF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2ncsc2C1 ZINC000880944297 EG On-Demand Anodyne P2RY14 46 38 C#CCC1(O)CCN(C(=O)Nc2ccc(F)cc2C(=O)OCC)CC1 ZINC000880944300 EE On-Demand Mild S1PR2 30 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nc(C(C)C)ncc2C1 ZINC000880944302 GH On-Demand Anodyne MAPK1 48 38 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2nc(C(C)C)ncc2C1 ZINC000880944302 GH On-Demand Anodyne P2RY14 47 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CCF)C1 ZINC000880944311 EH On-Demand Anodyne CCR3 76 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](CCF)C1 ZINC000880944311 EH On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CCF)C1 ZINC000880944313 EH On-Demand Anodyne CCR3 76 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](CCF)C1 ZINC000880944313 EH On-Demand Anodyne RBP4 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCO[C@H](CF)C1 ZINC000880944315 EE On-Demand Anodyne RBP4 33 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCO[C@@H](CF)C1 ZINC000880944317 EE On-Demand Anodyne RBP4 33 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880944334 GD On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880944336 GD On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880944338 GD On-Demand Anodyne RBP4 47 41 COC(=O)c1cc(NC(=O)/C=C\c2cccnc2)ccc1F ZINC000880944339 DF On-Demand Anodyne BTK 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880944340 GD On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880944342 GD On-Demand Anodyne CASR 62 45 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880944342 GD On-Demand Anodyne SOAT1 22 44 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCO)CCN1CCOCC1 ZINC000880944342 GD On-Demand Anodyne EPHX2 15 41 COCCN(CC1CCN(C)CC1)C(=O)c1cnc2cc[nH]c2c1 ZINC000880944361 ED On-Demand Anodyne ACKR3 64 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@@H](COC)C1 ZINC000880944364 FG On-Demand Anodyne CCR3 37 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@H](COC)C1 ZINC000880944365 FG On-Demand Anodyne CCR3 37 40 C#CCNC(=O)C1CCN(C(=O)Nc2ccc(F)cc2C(=O)OCC)CC1 ZINC000880944385 GD On-Demand Mild P2RY12 21 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(CO)CC1 ZINC000880944389 ED On-Demand Anodyne S1PR2 32 45 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)[C@@H]1CCCC[C@H]1O ZINC000880944393 EF On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(C2CC2)C1 ZINC000880944406 DF On-Demand Anodyne RBP4 57 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(C2CC2)C1 ZINC000880944406 DF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCCCO)C1CC1 ZINC000880944429 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC2(CC2)C1 ZINC000880944431 DG On-Demand Anodyne EPHX2 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)S(=O)(=O)[C@H](C)C1 ZINC000880944432 FE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)S(=O)(=O)[C@H](C)C1 ZINC000880944433 FE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)S(=O)(=O)[C@@H](C)C1 ZINC000880944434 FE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2NC(=O)CC[C@@H]2C1 ZINC000880944446 FE On-Demand Anodyne RBP4 53 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2NC(=O)CC[C@H]2C1 ZINC000880944447 FE On-Demand Anodyne RBP4 53 41 O=C(NNC(=O)C1CCC1)Nc1cnc2ccccc2c1Br ZINC000880944467 FF On-Demand Reactive CDK5 23 42 COC(=O)C1CCN(C(=O)Nc2cnc3ccccc3c2Br)CC1 ZINC000880944469 GG On-Demand Anodyne PTR1 46 33 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@]2(CCOC2)C1 ZINC000880944474 GH On-Demand Anodyne EPHX2 25 40 O=C(Nc1cnc2ccccc2c1Br)N1CC[C@@]2(CCOC2)C1 ZINC000880944475 GH On-Demand Anodyne EPHX2 25 40 COCCO[C@@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880944494 GG On-Demand Anodyne CCR8 43 33 COCCO[C@H]1CCN(C(=O)Nc2cnc3ccccc3c2Br)C1 ZINC000880944495 GG On-Demand Anodyne CCR8 43 33 O=C(Nc1cnc2ccccc2c1Br)N1C[C@H](O)[C@H](O)C1 ZINC000880944513 FD On-Demand Anodyne RBP4 51 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2NC(=O)CC[C@@H]2C1 ZINC000880944522 FE On-Demand Anodyne RBP4 53 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2NC(=O)CC[C@H]2C1 ZINC000880944523 FE On-Demand Anodyne RBP4 53 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC2(CCN(C)C2=O)CC1 ZINC000880944525 GE On-Demand Anodyne CACNA1H 48 37 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCOC)CC1CCN(C)CC1 ZINC000880944530 GF On-Demand Anodyne ACKR3 45 31 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)NOC)CC1 ZINC000880944534 FD On-Demand Anodyne P2RY12 23 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880944535 EF On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880944537 EF On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880944538 EF On-Demand Anodyne RBP4 47 41 CN(CCN1CCOCC1)C(=O)Nc1cnc2ccccc2c1Br ZINC000880944539 GF On-Demand Anodyne CNR2 15 41 CN(CCN1CCOCC1)C(=O)Nc1cnc2ccccc2c1Br ZINC000880944539 GF On-Demand Anodyne CASR 56 42 CN(CCN1CCOCC1)C(=O)Nc1cnc2ccccc2c1Br ZINC000880944539 GF On-Demand Anodyne PTGDS 42 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880944540 EF On-Demand Anodyne RBP4 47 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C[C@H]1CCC(=O)N1)C(C)C ZINC000880944541 FF On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(C[C@@H]1CCC(=O)N1)C(C)C ZINC000880944543 FF On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)[C@@H]1CCSC1 ZINC000880944544 EF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)[C@H]1CCSC1 ZINC000880944546 EF On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880944547 FG On-Demand Anodyne GLRA1 43 33 COCCN(CC1CCN(C)CC1)C(=O)c1ccc2c(O)ncnc2c1 ZINC000880944552 FD On-Demand Anodyne ACKR3 69 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](S(C)(=O)=O)CC1 ZINC000880944553 GE On-Demand Anodyne TLR4 16 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](S(C)(=O)=O)CC1 ZINC000880944554 GE On-Demand Anodyne TLR4 16 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](CC)[C@@H](O)C1 ZINC000880944563 DE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](O)[C@@H](CC)C1 ZINC000880944564 DE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](O)[C@H](CC)C1 ZINC000880944565 DE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](O)[C@H](CC)C1 ZINC000880944566 DE On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@@H](S(C)(=O)=O)C1 ZINC000880944570 GE On-Demand Anodyne P2RY12 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@@H](S(C)(=O)=O)C1 ZINC000880944570 GE On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@H](S(C)(=O)=O)C1 ZINC000880944571 GE On-Demand Anodyne P2RY12 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCC[C@H](S(C)(=O)=O)C1 ZINC000880944571 GE On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C)(C#N)CC1 ZINC000880944572 EG On-Demand Mild P2RY12 25 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC(C)(C)O)C1CC1 ZINC000880944573 EF On-Demand Anodyne TLR4 15 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(C(=O)NC)C1 ZINC000880944577 DD On-Demand Anodyne RBP4 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C1CCN(OC)CC1 ZINC000880944586 FE On-Demand Anodyne TLR4 15 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](CO)C[C@@H](C)C1 ZINC000880944587 EE On-Demand Anodyne RBP4 41 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)C[C@@H](CO)C1 ZINC000880944588 EE On-Demand Anodyne RBP4 41 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)C[C@H](CO)C1 ZINC000880944589 EE On-Demand Anodyne RBP4 41 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)C[C@@H](CO)C1 ZINC000880944590 EE On-Demand Anodyne RBP4 41 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880944593 DG On-Demand Anodyne RBP4 41 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880944593 DG On-Demand Anodyne TLR4 15 40 COCCN(CC1CCN(C)CC1)C(=O)c1n[nH]c2ccc(Cl)cc12 ZINC000880944599 FF On-Demand Anodyne CACNA1I 48 33 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(CC(F)(F)F)C1 ZINC000880944607 EG On-Demand Anodyne RBP4 55 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(F)(F)CC1 ZINC000880944608 EG On-Demand Anodyne CACNA1H 49 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(F)(F)CC1 ZINC000880944608 EG On-Demand Anodyne S1PR2 29 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(CCCO)C1CC1 ZINC000880944610 DE On-Demand Anodyne TLR4 15 41 C=CCN(C(=O)Nc1ccc(F)cc1C(=O)OCC)C1CC1 ZINC000880944630 DG On-Demand Mild TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(COC)CC1 ZINC000880944654 FE On-Demand Anodyne S1PR2 31 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCc2ccnc(O)c2C1 ZINC000880944655 FF On-Demand Anodyne P2RY14 44 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880944656 GG On-Demand Anodyne RBP4 42 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC2(CCNC2=O)CC1 ZINC000880944667 FE On-Demand Anodyne CACNA1H 59 35 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880944669 GD On-Demand Anodyne P2RY12 32 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880944669 GD On-Demand Anodyne RBP4 37 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880944669 GD On-Demand Anodyne TLR4 16 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H]1c1nc(C)cs1 ZINC000880944672 GI On-Demand Anodyne TRPC6 45 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1c1nc(C)cs1 ZINC000880944673 GI On-Demand Anodyne TRPC6 45 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880944681 GH On-Demand Anodyne P2RY12 28 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880944681 GH On-Demand Anodyne CCR1 18 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880944681 GH On-Demand Anodyne S1PR2 29 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880944681 GH On-Demand Anodyne RBP4 40 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880944683 FH On-Demand Anodyne P2RY12 24 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880944683 FH On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OC2CCC2)CC1 ZINC000880944683 FH On-Demand Anodyne SCD1 19 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)CCCn1ccnc1 ZINC000880944698 EF On-Demand Anodyne TBXAS1 41 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCOC2(CCN(C)CC2)C1 ZINC000880944699 GE On-Demand Anodyne EPHX2 18 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CC#N)CC1 ZINC000880944709 EG On-Demand Mild P2RY12 30 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H]2NC(=O)OC[C@H]2C1 ZINC000880944710 FD On-Demand Anodyne RBP4 40 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](c2nccn2C)C1 ZINC000880944713 FG On-Demand Anodyne CCR3 54 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](c2nccn2C)C1 ZINC000880944714 FG On-Demand Anodyne CCR3 54 37 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)S(=O)(=O)[C@@H](CC)C1 ZINC000880944716 GE On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H](C)S(=O)(=O)[C@H](CC)C1 ZINC000880944717 GE On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](C)S(=O)(=O)[C@H](CC)C1 ZINC000880944718 GE On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@H](CC)S(=O)(=O)[C@H](C)C1 ZINC000880944719 GE On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N(C1CC1)[C@H](C)CS(C)(=O)=O ZINC000880944720 GE On-Demand Anodyne TLR4 17 45 CCOC(=O)c1cc(F)ccc1NC(=O)N(C1CC1)[C@@H](C)CS(C)(=O)=O ZINC000880944721 GE On-Demand Anodyne TLR4 17 45 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(OCCO)CC1 ZINC000880944722 FE On-Demand Anodyne SCD1 18 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC(Cc2ccco2)C1 ZINC000880944740 EG On-Demand Anodyne RBP4 27 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1C[C@@H]2CCCC[C@@H]21 ZINC000880944745 DG On-Demand Anodyne TLR4 15 41 COCCN(CC1CCN(C)CC1)C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880944746 GG On-Demand Anodyne CACNA1I 53 36 COCCN(CC1CCN(C)CC1)C(=O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880944746 GG On-Demand Anodyne ACKR3 68 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CCF)CC1 ZINC000880944809 EH On-Demand Anodyne RBP4 50 42 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1[C@H](C)O ZINC000880944810 DE On-Demand Anodyne CCR3 46 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H]1[C@@H](C)O ZINC000880944811 DE On-Demand Anodyne CCR3 46 32 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCC[C@@H]1O ZINC000880944813 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@H]1CCC[C@H]1O ZINC000880944814 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCC[C@@H]1O ZINC000880944815 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(C)C[C@@H]1CCC[C@H]1O ZINC000880944816 EF On-Demand Anodyne TLR4 15 41 CCOC(=O)c1cc(F)ccc1NC(=O)N(CC)CCOCCO ZINC000880944818 ED On-Demand Anodyne SOAT1 17 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](COC)CC1 ZINC000880944822 FG On-Demand Anodyne CCR3 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](COC)CC1 ZINC000880944823 FG On-Demand Anodyne CCR3 34 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC2(CC1)CC2(F)F ZINC000880944825 FH On-Demand Anodyne S1PR2 28 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C(C)(C)O)CC1 ZINC000880944829 FG On-Demand Anodyne RBP4 40 39 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(C)(F)CC1 ZINC000880944834 EG On-Demand Anodyne S1PR2 28 40 COCCN(CC1CCN(C)CC1)C(=O)c1cc(C)cnc1Cl ZINC000880944847 EE On-Demand Anodyne CACNA1I 52 35 CCOC(=O)c1cc(F)ccc1NC(=O)N(C1CC1)C1CC1 ZINC000880944851 DG On-Demand Anodyne TLR4 16 44 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880944856 EC On-Demand Anodyne RBP4 39 41 CCOC(=O)c1cc(F)ccc1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880944856 EC On-Demand Anodyne TLR4 15 40 CCn1c(=O)c2ccccc2n(CC(=O)NCc2ccc(O)cc2)c1=O ZINC000880944857 FD On-Demand Anodyne F2 19 40 CCn1c(=O)c2ccccc2n(CC(=O)NCc2ccc(O)cc2)c1=O ZINC000880944857 FD On-Demand Anodyne FABI 53 34 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(Cc3ccccc3Cl)c(S)nc2c1 ZINC000880944862 JI On-Demand Anodyne PTGES 17 40 O=C(NCc1ccc(O)cc1)c1ccc2c(=O)n(Cc3ccccc3Cl)c(S)nc2c1 ZINC000880944862 JI On-Demand Anodyne NAMPT 41 36 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CS(C)(=O)=O)CC1 ZINC000880944863 GE On-Demand Anodyne CCR8 40 34 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(CS(C)(=O)=O)CC1 ZINC000880944863 GE On-Demand Anodyne TLR4 16 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(C(F)F)CC1 ZINC000880944864 FF On-Demand Anodyne P2RY12 20 40 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC(O)(C(F)F)CC1 ZINC000880944864 FF On-Demand Anodyne S1PR2 30 43 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@@H](C(=O)NC(C)C)C1 ZINC000880944868 GF On-Demand Anodyne CCR3 43 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCC[C@H](C(=O)NC(C)C)C1 ZINC000880944869 GF On-Demand Anodyne CCR3 43 32 CCOC(=O)c1cc(F)ccc1NC(=O)N1CCCN(C(=O)C2CC2)CC1 ZINC000880944874 GE On-Demand Anodyne TLR4 16 42 CN1C[C@@H]2CCCN(C(=O)Nc3ccc4c(n3)CCCC4)[C@@H]2C1 ZINC000880944916 DF On-Demand Anodyne HTR1F 60 34 O=C(Nc1ccc2c(n1)CCCC2)N1CCc2cc(Cl)nnc2C1 ZINC000880944926 EF On-Demand Anodyne MAPK1 42 36 Cn1ncc(C2CC2)c1CNC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880944937 EF On-Demand Anodyne HTR1F 67 41 O=C(Nc1ccc2c(n1)CCCC2)Nc1n[nH]cc1C1CC1 ZINC000880944950 CG On-Demand Anodyne HTR1F 63 37 O=C(Nc1ccc2c(n1)CCCC2)N1CCC2(CCCC2=O)CC1 ZINC000880944960 EG On-Demand Anodyne NPY5R 32 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCOC1=O ZINC000880944981 CD On-Demand Anodyne LUXR 75 43 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCOC1=O ZINC000880944981 CD On-Demand Anodyne TRAR 89 43 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCOC1=O ZINC000880944981 CD On-Demand Anodyne LASR 59 40 Cn1ncc(C2CCC2)c1CNC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880945013 EG On-Demand Anodyne HTR1F 63 40 CC(=O)c1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880945158 DG On-Demand Anodyne ROCK2 25 41 CN(C(=O)Nc1ccc2c(n1)CCCC2)[C@H](CO)Cc1ccccc1 ZINC000880945177 EG On-Demand Anodyne NPY5R 21 42 CN(C(=O)Nc1ccc2c(n1)CCCC2)[C@@H](CO)Cc1ccccc1 ZINC000880945178 EG On-Demand Anodyne NPY5R 21 42 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880945181 GG On-Demand Anodyne TRPM8 28 41 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880945182 GG On-Demand Anodyne TRPM8 28 41 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880945183 GG On-Demand Anodyne TRPM8 28 41 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880945184 GG On-Demand Anodyne TRPM8 28 41 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880945217 ED On-Demand Anodyne EPHX2 26 45 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880945218 ED On-Demand Anodyne EPHX2 26 45 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880945228 FG On-Demand Anodyne EPHX2 39 41 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880945277 DF On-Demand Anodyne PLM1_PLAFA 41 39 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880945390 FF On-Demand Anodyne L3MBTL3 76 39 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880945391 FF On-Demand Anodyne L3MBTL3 76 39 Cc1nnc([C@@H]2CCCN(C(=O)Nc3ccc4c(n3)CCCC4)C2)o1 ZINC000880945629 EG On-Demand Anodyne HTR1F 40 32 CN(C[C@@H]1CCCN1C)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880945674 DF On-Demand Anodyne HTR1F 50 31 CN(C[C@H]1CCCN1C)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880945675 DF On-Demand Anodyne HTR1F 50 31 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880945687 FG On-Demand Anodyne EPHX2 17 46 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880945688 FG On-Demand Anodyne EPHX2 17 46 CN1CCC(CNC(=O)Nc2ccc3c(n2)CCCC3)(N2CCOCC2)CC1 ZINC000880945689 GD On-Demand Anodyne HCN1 76 40 CN1CCC(CNC(=O)Nc2ccc3c(n2)CCCC3)(N2CCOCC2)CC1 ZINC000880945689 GD On-Demand Anodyne HCN4 51 32 CN1CCO[C@@H]2CN(C(=O)Nc3ccc4c(n3)CCCC4)C[C@@H]21 ZINC000880945703 DD On-Demand Anodyne HTR1F 58 32 O=C(Nc1ccc2c(n1)CCCC2)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880945736 FF On-Demand Anodyne CHRNA4 26 44 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CCCS2(=O)=O)CC1 ZINC000880945796 GD On-Demand Anodyne HTR1F 44 32 CN1CCC[C@@H](CCNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880945847 DF On-Demand Anodyne HTR1F 41 39 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880945865 EG On-Demand Anodyne HTR1F 49 33 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880945867 EG On-Demand Anodyne HTR1F 49 33 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccc2c(n1)CCCC2 ZINC000880945950 CG On-Demand Anodyne CDK2 16 50 O=C(Nc1cc(C2CC2)[nH]n1)Nc1ccc2c(n1)CCCC2 ZINC000880945950 CG On-Demand Anodyne PKNB 79 40 COC(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880945995 EE On-Demand Anodyne EPHX2 39 43 CC(=O)Nc1ccc(CNC(=O)Nc2ccc3c(n2)CCCC3)cn1 ZINC000880946018 EF On-Demand Anodyne MAPK1 15 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc3c(n1)CCCC3)C2 ZINC000880946029 DF On-Demand Anodyne HTR4 17 40 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1ccc3c(n1)CCCC3)C2 ZINC000880946029 DF On-Demand Anodyne GLRA1 41 30 Cn1nc(NC(=O)Nc2ccc3c(n2)CCCC3)cc1C1CC1 ZINC000880946084 DG On-Demand Anodyne HTR1F 49 35 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCCN(CCCO)C1 ZINC000880946111 ED On-Demand Anodyne CCR3 21 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCCN(CCCO)C1 ZINC000880946113 ED On-Demand Anodyne CCR3 21 40 O=C(Nc1ccc2c(n1)CCCC2)N1[C@H]2CC[C@H]1c1ccccc12 ZINC000880946150 DI On-Demand Anodyne HTR1F 44 33 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880946158 FG On-Demand Anodyne NPY5R 28 40 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880946159 FG On-Demand Anodyne NPY5R 28 40 CNC(=O)COc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880946365 FE On-Demand Anodyne ROCK1 19 41 CNC(=O)COc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880946365 FE On-Demand Anodyne ROCK2 33 42 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(CC(F)(F)F)CC1 ZINC000880946399 FG On-Demand Anodyne CXCR3 19 42 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(CC(F)(F)F)CC1 ZINC000880946399 FG On-Demand Anodyne HPGDS 39 44 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCCN(C(=O)CCC(F)(F)F)C1 ZINC000880946406 GG On-Demand Anodyne ETHR 56 37 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880946467 GF On-Demand Anodyne RBP4 53 32 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880946468 GF On-Demand Anodyne RBP4 53 32 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880946469 GF On-Demand Anodyne RBP4 53 32 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880946470 GF On-Demand Anodyne RBP4 53 32 O=C(Nc1ccc2c(n1)CCCC2)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880946471 EG On-Demand Anodyne EPHX2 39 42 CS(=O)(=O)c1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880946478 FF On-Demand Anodyne NAMPT 50 38 O=C(Nc1ccc2c(n1)CCCC2)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880946636 EF On-Demand Anodyne CPT1A 66 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880946638 EF On-Demand Anodyne CPT1A 66 35 O=C(Nc1ccc2c(n1)CCCC2)NN1CCCCC1 ZINC000880946656 CE On-Demand Anodyne CNR1 51 32 O=C(NCc1ccc(F)cn1)Nc1ccc2c(n1)CCCC2 ZINC000880946860 DF On-Demand Anodyne SLC27A1 44 37 CC(C)(C)OC(=O)N1CCCN(Cc2cn(Cc3ncc[nH]3)nn2)CC1 ZINC000880946869 FD On-Demand Anodyne KDM1A 20 45 CC(C)(O)CN1CC[C@H](NC(=O)c2n[nH]c3ccc(Cl)cc23)C1 ZINC000880946877 ED On-Demand Anodyne DRD4 22 40 CC(C)(O)CN1CC[C@H](NC(=O)c2n[nH]c3ccc(Cl)cc23)C1 ZINC000880946877 ED On-Demand Anodyne PLD1 40 34 CC(C)(O)CN1CC[C@H](NC(=O)c2n[nH]c3ccc(Cl)cc23)C1 ZINC000880946877 ED On-Demand Anodyne MCHR1 31 47 CC(C)(O)CN1CC[C@H](NC(=O)c2n[nH]c3ccc(Cl)cc23)C1 ZINC000880946877 ED On-Demand Anodyne CACNA1I 41 32 COCCC(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880946950 FE On-Demand Anodyne EPHX2 33 45 CC(C)(C)OC(=O)N1CCN(Cc2cn(Cc3ncc[nH]3)nn2)CC1 ZINC000880946963 ED On-Demand Anodyne KDM1A 21 47 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880947024 FD On-Demand Anodyne HCN1 65 39 O=C(NCC1(N2CCOCC2)CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880947024 FD On-Demand Anodyne HCN4 50 32 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880947082 FG On-Demand Anodyne CCR3 36 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880947085 FG On-Demand Anodyne CCR3 36 42 C[C@H](NC(=O)Nc1ccc2c(n1)CCCC2)[C@H]1CN(C)CCO1 ZINC000880947091 DD On-Demand Anodyne HTR1F 42 33 C[C@H](NC(=O)Nc1ccc2c(n1)CCCC2)[C@@H]1CN(C)CCO1 ZINC000880947093 DD On-Demand Anodyne HTR1F 42 33 O=C(NCCCCc1cn(Cc2ncc[nH]2)nn1)OCc1ccccc1 ZINC000880947097 FE On-Demand Anodyne CYSP_TRYCR 42 33 O=C(NCCCCc1cn(Cc2ncc[nH]2)nn1)OCc1ccccc1 ZINC000880947097 FE On-Demand Anodyne CAPN2 58 33 O=C(NCCCCc1cn(Cc2ncc[nH]2)nn1)OCc1ccccc1 ZINC000880947097 FE On-Demand Anodyne NPR 47 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CCCCC2=O)CC1 ZINC000880947127 FF On-Demand Anodyne L3MBTL3 42 32 Cc1cncc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880947156 CF On-Demand Anodyne NAMPT 23 48 CN1CCO[C@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C[C@H]21 ZINC000880947167 ED On-Demand Anodyne HTR1F 66 34 CN1CCO[C@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C[C@@H]21 ZINC000880947171 ED On-Demand Anodyne HTR1F 66 34 CN1CCO[C@@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C[C@H]21 ZINC000880947174 ED On-Demand Anodyne HTR1F 66 34 CN1CCO[C@@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C[C@@H]21 ZINC000880947177 ED On-Demand Anodyne HTR1F 66 34 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880947184 FG On-Demand Anodyne CCR3 30 43 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880947187 FG On-Demand Anodyne CCR3 30 43 COC(=O)[C@@H]1CCCN(Cc2cn(Cc3ncc(Cl)n3C)nn2)C1 ZINC000880947188 FD On-Demand Anodyne SLC6A1 45 33 CN(C(=O)Nc1ccc2c(n1)CCCC2)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880947209 EG On-Demand Anodyne GLRA1 40 31 CC(=O)c1cccc(OCc2cn(C3CCCC3)nn2)c1 ZINC000880947281 CG On-Demand Anodyne VCP 42 37 Cn1nccc1[C@H]1CCCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880947480 EG On-Demand Anodyne HTR1F 43 32 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880947481 EG On-Demand Anodyne HTR1F 43 32 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1c2ccccc2C[C@H]1O ZINC000880947534 DF On-Demand Anodyne PLM1_PLAFA 41 39 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880947535 DF On-Demand Anodyne PLM1_PLAFA 41 39 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880947536 DF On-Demand Anodyne PLM1_PLAFA 41 39 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA2 65 81 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA6 29 44 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA1 49 81 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA7 41 45 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA13 50 45 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA4 46 81 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA14 20 40 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA12 26 48 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CA9 26 48 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne CYNT 27 51 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne NCE103 21 41 NS(=O)(=O)c1cc(C(=O)NCc2ccc(O)cc2)ccc1Cl ZINC000880947603 ED On-Demand Anodyne A6YCJ1_9METZ 20 40 O=C(CCNS(=O)(=O)/C=C\c1ccccc1)NCc1ccc(O)cc1 ZINC000880947610 FD On-Demand Anodyne CA5A 15 40 O=C(NCCN1CCCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880947648 DD On-Demand Anodyne EPHX2 18 42 O=C(NCCN1CCCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880947648 DD On-Demand Anodyne HPGDS 23 40 O=C(NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1)C1CC1 ZINC000880947684 EE On-Demand Anodyne EPHX2 28 41 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(Cc2ccccn2)CC1 ZINC000880947705 FF On-Demand Anodyne FAAH 18 44 O=C(NCC1(N2CCOCC2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880947720 ED On-Demand Anodyne HCN1 69 36 O=C(NCC1(N2CCOCC2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880947720 ED On-Demand Anodyne HCN4 51 32 Nc1ccc(CNC(=O)Nc2ccc3c(n2)CCCC3)cn1 ZINC000880947722 CE On-Demand Anodyne NAMPT 17 47 Cn1ccnc1[C@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880947827 EF On-Demand Anodyne HTR1F 67 35 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880947828 EF On-Demand Anodyne HTR1F 67 35 O=C(Nc1cc(C2CCOCC2)[nH]n1)Nc1ccc2c(n1)CCCC2 ZINC000880947932 EG On-Demand Anodyne PKNB 49 34 O=C(Nc1ccc2c(n1)CCCC2)N[C@H](CO)Cc1ccccc1 ZINC000880947987 EF On-Demand Anodyne MME 30 41 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948080 EF On-Demand Anodyne CCR3 52 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948082 EF On-Demand Anodyne CCR3 52 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948085 EF On-Demand Anodyne CCR3 52 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948087 EF On-Demand Anodyne CCR3 52 40 COC(=O)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880948089 DE On-Demand Anodyne PTR1 45 32 COC(OC)c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)o1 ZINC000880948093 ED On-Demand Anodyne SSTR5 41 35 COC(OC)c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)o1 ZINC000880948093 ED On-Demand Anodyne MCHR1 28 41 CC(=O)c1cccc(OCc2cn(Cc3c(C)noc3C)nn2)c1 ZINC000880948099 EF On-Demand Anodyne NR1H4 55 38 CC(=O)c1cccc(OCc2cn(Cc3c(C)noc3C)nn2)c1 ZINC000880948099 EF On-Demand Anodyne FIMH 17 40 CC(=O)OC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880948127 DF On-Demand Anodyne HTR1F 40 34 CC(=O)c1cccc(OCc2cn([C@H](C)C(=O)NC3CC3)nn2)c1 ZINC000880948132 ED On-Demand Anodyne PLG 15 40 CC(=O)c1cccc(OCc2cn([C@H](C)C(=O)NC3CC3)nn2)c1 ZINC000880948132 ED On-Demand Anodyne FAAH 17 42 CC(=O)c1cccc(OCc2cn([C@@H](C)C(=O)NC3CC3)nn2)c1 ZINC000880948133 ED On-Demand Anodyne PLG 15 40 CC(=O)c1cccc(OCc2cn([C@@H](C)C(=O)NC3CC3)nn2)c1 ZINC000880948133 ED On-Demand Anodyne FAAH 17 42 Cc1cccc(C(=O)NNC(=O)Nc2ccc3c(n2)CCCC3)n1 ZINC000880948234 EE On-Demand Reactive SORT1 22 44 Cc1nc(CNC(=O)Nc2ccc3c(n2)CCCC3)nc2ccccc12 ZINC000880948293 EH On-Demand Anodyne ACHE 46 38 Cc1nc(CNC(=O)Nc2ccc3c(n2)CCCC3)nc2ccccc12 ZINC000880948293 EH On-Demand Anodyne BCHE 70 37 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948297 EG On-Demand Anodyne HTR1F 43 36 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948298 EG On-Demand Anodyne HTR1F 43 36 CNCC(=O)Nc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880948321 FD On-Demand Anodyne HDAC10 28 50 CNCC(=O)Nc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880948321 FD On-Demand Anodyne HDAC3 33 50 CNCC(=O)Nc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880948321 FD On-Demand Anodyne HDAC6 26 50 CC(=O)c1cccc(OCc2cn(C3CCCCC3)nn2)c1 ZINC000880948325 CH On-Demand Anodyne FAAH 15 42 CC(=O)c1cccc(OCc2cn(C3CCCCC3)nn2)c1 ZINC000880948325 CH On-Demand Anodyne VCP 41 36 Cc1coc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c1 ZINC000880948418 CD On-Demand Anodyne DRD4 21 43 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne HTR1A 23 43 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne DRD2 32 45 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne DRD4 41 44 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne DRD3 37 44 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne HTR4 47 41 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne HTR7 22 46 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne SSTR5 22 40 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne CCR3 19 45 COc1ccccc1-c1ccc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)c(O)n1 ZINC000880948447 GE On-Demand Anodyne MCHR1 15 40 CS(=O)(=O)Nc1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880948483 DD On-Demand Anodyne TRPV1 32 47 CS(=O)(=O)Nc1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880948483 DD On-Demand Anodyne NAMPT 47 38 CS(=O)(=O)Nc1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880948483 DD On-Demand Anodyne KCNK3 57 35 CN1[C@H]2CC[C@H]1CC(N1CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC1)C2 ZINC000880948488 GF On-Demand Anodyne HTR1F 44 32 CC(C)(C)OC(=O)N1CCC(c2cn(Cc3ncc[nH]3)nn2)CC1 ZINC000880948489 EE On-Demand Anodyne GPR119 41 42 O=C(CCc1ccccc1)NNC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880948656 EF On-Demand Reactive HCAR2 41 42 O=C(NNC(=O)c1ccccn1)Nc1ccc2c(n1)CCCC2 ZINC000880948660 DD On-Demand Reactive GRM4 57 37 CN1CC[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1=O ZINC000880948689 CD On-Demand Anodyne HTR1F 57 36 COc1ccc2c(c1)CC[C@H](C(=O)N[C@H]1CCN(CC(C)(C)O)C1)C2 ZINC000880948831 ED On-Demand Anodyne MCHR1 16 43 CN1CCC(N2CCC(NC(=O)Nc3ccc4c(n3)CCCC4)CC2)CC1 ZINC000880948853 FF On-Demand Anodyne HTR1F 75 39 CN1CCC(N2CCC(NC(=O)Nc3ccc4c(n3)CCCC4)CC2)CC1 ZINC000880948853 FF On-Demand Anodyne SLC6A5 19 41 C[C@@H]1CN(C(=O)Nc2ccc3c(n2)CCCC3)CC[C@@H]1N1CCN(C)CC1 ZINC000880948895 FE On-Demand Anodyne HTR1F 42 32 C[C@H]1CN(C(=O)Nc2ccc3c(n2)CCCC3)CC[C@@H]1N1CCN(C)CC1 ZINC000880948896 FE On-Demand Anodyne HTR1F 42 32 C[C@H]1CN(C(=O)Nc2ccc3c(n2)CCCC3)CC[C@H]1N1CCN(C)CC1 ZINC000880948982 FE On-Demand Anodyne HTR1F 42 32 C[C@@H]1CN(C(=O)Nc2ccc3c(n2)CCCC3)CC[C@H]1N1CCN(C)CC1 ZINC000880948983 FE On-Demand Anodyne HTR1F 42 32 C[C@@H](C1CCN(C)CC1)N(C)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880949050 EG On-Demand Anodyne HTR1F 66 35 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880949098 EE On-Demand Anodyne CCR3 44 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880949115 GH On-Demand Anodyne TRPM8 27 40 CCOc1ccccc1OS(=O)(=O)c1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880949150 IG On-Demand Anodyne HCN1 42 30 CCOc1ccccc1OS(=O)(=O)c1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880949150 IG On-Demand Anodyne KCNK3 31 40 CCOc1ccccc1OS(=O)(=O)c1cccc(C(=O)NCc2ccc(O)cc2)c1 ZINC000880949150 IG On-Demand Anodyne KCNK9 20 40 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880949154 GE On-Demand Anodyne EPHX2 28 50 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2ncc(F)cn2)CC1 ZINC000880949188 FE On-Demand Anodyne FAAH 22 41 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2ncc(F)cn2)CC1 ZINC000880949188 FE On-Demand Anodyne SLC27A1 46 37 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2cn[nH]c2)CC1 ZINC000880949217 EG On-Demand Anodyne HTR1F 55 34 O[C@]1(c2cn(CCOc3ccccc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880949316 CE On-Demand Anodyne ALOX5AP 40 40 O[C@@]1(c2cn(CCOc3ccccc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880949317 CE On-Demand Anodyne ALOX5AP 40 40 O=C(NCCCNC(=O)C1CCC1)Nc1ccc2c(n1)CCCC2 ZINC000880949331 EE On-Demand Anodyne TBK1 82 36 CC(=O)c1cccc(OCc2cn(Cc3nc(C)no3)nn2)c1 ZINC000880949332 DD On-Demand Anodyne NR1H4 45 34 CC(=O)c1cccc(OCc2cn(Cc3nc(C)no3)nn2)c1 ZINC000880949332 DD On-Demand Anodyne FIMH 17 40 CC(=O)N1CCN(Cc2cn(CCOc3ccccc3)nn2)CC1 ZINC000880949352 ED On-Demand Anodyne LTA4H 40 37 CC(=O)N1CCN(Cc2cn(CCOc3ccccc3)nn2)CC1 ZINC000880949352 ED On-Demand Anodyne HRH3 26 42 CC(=O)N1CCN(Cc2cn(CCOc3ccccc3)nn2)CC1 ZINC000880949352 ED On-Demand Anodyne FAAH 24 40 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1ccc2c(n1)CCCC2 ZINC000880949395 GF On-Demand Anodyne STAT6 56 35 Cc1ccccc1[C@H](CO)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880949401 EG On-Demand Anodyne CTSA 43 32 Cc1ccccc1[C@@H](CO)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880949402 EG On-Demand Anodyne CTSA 43 32 CNc1nc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)cs1 ZINC000880949423 CC On-Demand Anodyne MAPKAPK2 20 44 CNc1nc(C(=O)N[C@H]2CCN(CC(C)(C)O)C2)cs1 ZINC000880949423 CC On-Demand Anodyne TRPC6 43 33 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H](CO)Cc1ccccc1 ZINC000880949428 EF On-Demand Anodyne MME 30 41 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc3c(n1)CCCC3)CC2 ZINC000880949465 FE On-Demand Anodyne P2RY14 44 33 O=C(NNc1ncccc1Cl)Nc1ccc2c(n1)CCCC2 ZINC000880949563 DG On-Demand Reactive PPIA 23 40 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880949564 HF On-Demand Anodyne LNPEP 45 36 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880949564 HF On-Demand Anodyne EPHX2 27 51 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 ZINC000880949564 HF On-Demand Anodyne TMPRSS11D 57 33 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880949566 HF On-Demand Anodyne LNPEP 45 36 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880949566 HF On-Demand Anodyne EPHX2 27 51 O=C(NCc1ccc(O)cc1)C1CCN(S(=O)(=O)/C=C\c2ccccc2)CC1 ZINC000880949566 HF On-Demand Anodyne TMPRSS11D 57 33 CC(=O)N(CC(=O)N[C@H]1CCN(CC(C)(C)O)C1)c1ccccc1 ZINC000880949675 ED On-Demand Anodyne DRD4 22 40 CC(=O)N(CC(=O)N[C@H]1CCN(CC(C)(C)O)C1)c1ccccc1 ZINC000880949675 ED On-Demand Anodyne SIGMAR1 18 44 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880949683 EH On-Demand Anodyne NPY5R 32 42 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880949684 EH On-Demand Anodyne NPY5R 32 42 CN1CC[C@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880949720 CE On-Demand Anodyne HTR1F 67 42 CN1CC[C@@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880949721 CE On-Demand Anodyne HTR1F 67 42 O=C(Nc1ccc2c(n1)CCCC2)N(CCO)CCN1CCOCC1 ZINC000880949899 ED On-Demand Anodyne CASR 65 50 CC(=O)c1cccc(OCc2cn([C@H](C)c3nc(C(C)C)no3)nn2)c1 ZINC000880950037 FG On-Demand Anodyne NR1H4 66 38 CC(=O)c1cccc(OCc2cn([C@@H](C)c3nc(C(C)C)no3)nn2)c1 ZINC000880950038 FG On-Demand Anodyne NR1H4 66 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880950040 DD On-Demand Anodyne XIAP 25 40 CC(=O)c1cccc(OCc2cn([C@H](C)C(=O)C3CC3)nn2)c1 ZINC000880950098 DF On-Demand Anodyne NR1H4 40 35 CC(=O)c1cccc(OCc2cn([C@@H](C)C(=O)C3CC3)nn2)c1 ZINC000880950099 DF On-Demand Anodyne NR1H4 40 35 CC(=O)c1cccc(OCc2cn([C@H]3CCN(C)C3=O)nn2)c1 ZINC000880950119 DD On-Demand Anodyne DRD4 40 30 CC(=O)c1cccc(OCc2cn([C@@H]3CCN(C)C3=O)nn2)c1 ZINC000880950120 DD On-Demand Anodyne DRD4 40 30 COc1ccccc1[C@@](N)(C(=O)N[C@H]1CCN(CC(C)(C)O)C1)C(F)(F)F ZINC000880950159 GD On-Demand Anodyne DRD2 19 42 COc1ccccc1[C@@](N)(C(=O)N[C@H]1CCN(CC(C)(C)O)C1)C(F)(F)F ZINC000880950159 GD On-Demand Anodyne DRD4 25 42 COc1ccccc1[C@@](N)(C(=O)N[C@H]1CCN(CC(C)(C)O)C1)C(F)(F)F ZINC000880950159 GD On-Demand Anodyne DRD3 16 42 CC1(C)CCC[C@H](Cn2cc(CNC(=O)OCc3ccccc3)nn2)O1 ZINC000880950193 FG On-Demand Anodyne PREP 22 40 CC1(C)CCC[C@H](Cn2cc(CNC(=O)OCc3ccccc3)nn2)O1 ZINC000880950193 FG On-Demand Anodyne CAPN2 46 35 CC1(C)CCC[C@H](Cn2cc(CNC(=O)OCc3ccccc3)nn2)O1 ZINC000880950193 FG On-Demand Anodyne NPR 59 34 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880950210 FF On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880950211 FF On-Demand Anodyne EPHX2 26 40 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H](N2CC=CC2)C1 ZINC000880950249 DE On-Demand Anodyne L3MBTL3 45 36 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H](N2CC=CC2)C1 ZINC000880950251 DE On-Demand Anodyne L3MBTL3 45 36 COc1cccc(OCc2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880950256 EE On-Demand Anodyne FIMH 15 40 CC(=O)c1cccc(OCc2cn([C@H]3C[C@H](C)O[C@H](C)C3)nn2)c1 ZINC000880950278 EG On-Demand Anodyne FIMH 15 41 CC(=O)c1cccc(OCc2cn([C@@H]3C[C@H](C)O[C@H](C)C3)nn2)c1 ZINC000880950279 EG On-Demand Anodyne FIMH 15 41 CNC(=O)CNc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880950281 FD On-Demand Anodyne HDAC10 19 44 CNC(=O)CNc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880950281 FD On-Demand Anodyne HDAC3 22 44 CNC(=O)CNc1cccc(-c2cn(Cc3ncc(Cl)n3C)nn2)c1 ZINC000880950281 FD On-Demand Anodyne HDAC6 18 44 O=C(Nc1ccc2c(n1)CCCC2)N1CCc2ccccc2[C@H]1CO ZINC000880950283 EG On-Demand Anodyne TRPM8 26 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCc2ccccc2[C@@H]1CO ZINC000880950285 EG On-Demand Anodyne TRPM8 26 40 O=C(/C=C\c1cccnc1)Nc1ccc(NC(=O)NCc2ccco2)cc1 ZINC000880950302 FH On-Demand Anodyne CYP2C9 15 41 O=C(/C=C\c1cccnc1)Nc1ccc(NC(=O)NCc2ccco2)cc1 ZINC000880950302 FH On-Demand Anodyne NAMPT 62 53 CC(=O)c1cccc(OCc2cn(Cc3noc(C(C)C)n3)nn2)c1 ZINC000880950317 EF On-Demand Anodyne NR1H4 59 38 CC(=O)c1cccc(OCc2cn(Cc3cc(C)on3)nn2)c1 ZINC000880950371 DE On-Demand Anodyne NR1H4 50 36 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CC=CC2)CC1 ZINC000880950409 EF On-Demand Anodyne L3MBTL3 69 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCCN(C2CCCC2)CC1 ZINC000880950421 EG On-Demand Anodyne L3MBTL3 64 36 CNC(=O)CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880950433 EC On-Demand Anodyne SLC27A1 46 39 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2cnc[nH]2)CC1 ZINC000880950438 EG On-Demand Anodyne HTR1F 57 34 CC1(C)CCC[C@H](Cn2cc(-c3ccc(CO)nc3)nn2)O1 ZINC000880950471 DE On-Demand Anodyne FIMH 15 40 O=C(Nc1cnn(CC2CC2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880950476 DG On-Demand Anodyne PANC 41 31 COC(=O)[C@@H](C)n1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880950484 DF On-Demand Anodyne ESRRA 18 42 COC(=O)[C@@H](C)n1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880950484 DF On-Demand Anodyne MAP3K5 47 35 c1c([C@H]2CCCCO2)nnn1C[C@@H]1CCCO1 ZINC000880950492 BD On-Demand Anodyne PDE8B 54 45 c1c([C@@H]2CCCCO2)nnn1C[C@@H]1CCCO1 ZINC000880950493 BD On-Demand Anodyne PDE8B 54 45 c1c([C@@H]2CCCCO2)nnn1C[C@H]1CCCO1 ZINC000880950494 BD On-Demand Anodyne PDE8B 54 45 c1c([C@H]2CCCCO2)nnn1C[C@H]1CCCO1 ZINC000880950495 BD On-Demand Anodyne PDE8B 54 45 O=C(c1ccc(Cl)cc1)c1cn(C[C@H]2CCCO2)nn1 ZINC000880950512 CE On-Demand Anodyne PDE8B 52 36 O=C(c1ccc(Cl)cc1)c1cn(C[C@@H]2CCCO2)nn1 ZINC000880950513 CE On-Demand Anodyne PDE8B 52 36 CN(C)C(=O)Nc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880950524 FG On-Demand Anodyne ROCK2 23 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@H](CCO)c1ccccc1 ZINC000880950539 EG On-Demand Anodyne TACR3 16 42 CN1CCC(N(C)CCN(C)C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880950630 FE On-Demand Anodyne HTR1F 65 35 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(=O)CN)c3)nn2)O1 ZINC000880950748 EE On-Demand Anodyne HDAC10 23 43 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(=O)CN)c3)nn2)O1 ZINC000880950748 EE On-Demand Anodyne HDAC3 27 43 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(=O)CN)c3)nn2)O1 ZINC000880950748 EE On-Demand Anodyne HDAC6 22 43 COCCNC(=O)c1cn(C[C@H]2CCCC(C)(C)O2)nn1 ZINC000880950767 CD On-Demand Anodyne LGALS3 20 41 COCCNC(=O)c1cn(C[C@@H]2CCCC(C)(C)O2)nn1 ZINC000880950768 CD On-Demand Anodyne LGALS3 20 41 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2ncc[nH]2)CC1 ZINC000880950779 EG On-Demand Anodyne HTR1F 57 36 CC1(C)CCC[C@H](Cn2cc(COc3cccc(CO)c3)nn2)O1 ZINC000880950793 EF On-Demand Anodyne DRTS_LEIMA 29 40 CC1(C)CCC[C@H](Cn2cc(COc3cccc(CO)c3)nn2)O1 ZINC000880950793 EF On-Demand Anodyne FIMH 15 41 CC(=O)N1CCN(Cc2cn(C[C@@H]3CCCCO3)nn2)CC1 ZINC000880950878 DC On-Demand Anodyne PDE8B 51 38 CC(=O)N1CCN(Cc2cn(C[C@H]3CCCCO3)nn2)CC1 ZINC000880950879 DC On-Demand Anodyne PDE8B 51 38 O[C@H](c1ccc(Cl)cc1)c1cn(C[C@@H]2CCCCO2)nn1 ZINC000880950908 DF On-Demand Anodyne PDE8B 46 37 O[C@@H](c1ccc(Cl)cc1)c1cn(C[C@H]2CCCCO2)nn1 ZINC000880950909 DF On-Demand Anodyne PDE8B 46 37 O[C@H](c1ccc(Cl)cc1)c1cn(C[C@H]2CCCCO2)nn1 ZINC000880950910 DF On-Demand Anodyne PDE8B 46 37 O[C@@H](c1ccc(Cl)cc1)c1cn(C[C@@H]2CCCCO2)nn1 ZINC000880950911 DF On-Demand Anodyne PDE8B 46 37 NC(=O)c1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880950916 DE On-Demand Anodyne ROCK2 22 48 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(N)=O)c3)nn2)O1 ZINC000880950977 EF On-Demand Anodyne HDAC10 20 41 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(N)=O)c3)nn2)O1 ZINC000880950977 EF On-Demand Anodyne HDAC3 23 41 CC1(C)CCC[C@H](Cn2cc(-c3cccc(NC(N)=O)c3)nn2)O1 ZINC000880950977 EF On-Demand Anodyne HDAC6 18 41 O=S1(=O)CCN(Cc2cn(C[C@H]3CCCCO3)nn2)CC1 ZINC000880950988 DC On-Demand Anodyne PDE8B 48 35 O=S1(=O)CCN(Cc2cn(C[C@@H]3CCCCO3)nn2)CC1 ZINC000880950989 DC On-Demand Anodyne PDE8B 48 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(C2CC2)CC1 ZINC000880950996 DE On-Demand Anodyne L3MBTL3 61 36 O=C(NCc1cccnc1-n1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880951006 EF On-Demand Anodyne NOS2 70 31 C[C@H]1C[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)CCN1C ZINC000880951025 DF On-Demand Anodyne HTR1F 52 33 O=C(Nc1ccc2c(n1)CCCC2)N1CCn2c(nnc2-c2ccccc2)C1 ZINC000880951036 FG On-Demand Anodyne P2RX7 28 45 Cn1nc2c(c1-c1cn(C[C@H]3CCCO3)nn1)CCCC2 ZINC000880951037 CD On-Demand Anodyne PDE8B 42 33 Cn1nc2c(c1-c1cn(C[C@@H]3CCCO3)nn1)CCCC2 ZINC000880951038 CD On-Demand Anodyne PDE8B 42 33 CC1(C)CCC[C@H](Cn2cc(CNC(=O)Nc3ccc(F)c(F)c3)nn2)O1 ZINC000880951042 GG On-Demand Anodyne PRMT3 44 31 CC(=O)c1cccc(OCc2cn(C[C@@H]3CCCCO3)nn2)c1 ZINC000880951076 DF On-Demand Anodyne PDE8B 46 42 CC(=O)c1cccc(OCc2cn(C[C@H]3CCCCO3)nn2)c1 ZINC000880951077 DF On-Demand Anodyne PDE8B 46 42 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(Nc2cccnn2)CC1 ZINC000880951095 FF On-Demand Anodyne FAAH 22 40 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951108 FE On-Demand Anodyne HDAC10 23 43 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951108 FE On-Demand Anodyne HDAC3 27 43 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951108 FE On-Demand Anodyne HDAC6 22 43 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951109 FE On-Demand Anodyne HDAC10 23 43 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951109 FE On-Demand Anodyne HDAC3 27 43 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880951109 FE On-Demand Anodyne HDAC6 22 43 N#CCCN(CCN1CCOCC1)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880951156 FE On-Demand Mild CASR 61 47 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1ccc3c(n1)CCCC3)C2 ZINC000880951158 EG On-Demand Anodyne HTR3A 37 42 Cn1nc2c(c1-c1cn(C[C@H]3CCCCO3)nn1)CCCC2 ZINC000880951182 DE On-Demand Anodyne PDE8B 49 37 Cn1nc2c(c1-c1cn(C[C@@H]3CCCCO3)nn1)CCCC2 ZINC000880951183 DE On-Demand Anodyne PDE8B 49 37 c1c([C@@H]2CCCCO2)nnn1C[C@@H]1CCCCO1 ZINC000880951189 CE On-Demand Anodyne PDE8B 54 44 c1c([C@H]2CCCCO2)nnn1C[C@H]1CCCCO1 ZINC000880951190 CE On-Demand Anodyne PDE8B 54 44 c1c([C@H]2CCCCO2)nnn1C[C@@H]1CCCCO1 ZINC000880951191 CE On-Demand Anodyne PDE8B 54 44 c1c([C@@H]2CCCCO2)nnn1C[C@H]1CCCCO1 ZINC000880951192 CE On-Demand Anodyne PDE8B 54 44 CC1(C)CCC[C@H](Cn2cc(CN3C(=O)C(=O)c4ccccc43)nn2)O1 ZINC000880951213 FE On-Demand Anodyne ALDH1A1 44 37 CN(CCN1CCOCC1)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880951375 DD On-Demand Anodyne CASR 55 43 CC1(C)CCC[C@H](Cn2cc(COc3ccc(CO)cc3)nn2)O1 ZINC000880951431 EF On-Demand Anodyne FIMH 15 42 O[C@@]1(c2cn(C[C@@H]3CCCCO3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880951440 CD On-Demand Anodyne PDE8B 41 34 O[C@]1(c2cn(C[C@@H]3CCCCO3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880951441 CD On-Demand Anodyne PDE8B 41 34 O[C@]1(c2cn(C[C@H]3CCCCO3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880951442 CD On-Demand Anodyne PDE8B 41 34 O[C@@]1(c2cn(C[C@H]3CCCCO3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880951443 CD On-Demand Anodyne PDE8B 41 34 O=C(c1ccc(Cl)cc1)c1cn(C[C@H]2CCCCO2)nn1 ZINC000880951458 DF On-Demand Anodyne PDE8B 54 39 O=C(c1ccc(Cl)cc1)c1cn(C[C@@H]2CCCCO2)nn1 ZINC000880951459 DF On-Demand Anodyne PDE8B 54 39 O=C(NCc1ccc(CN2CCC(O)CC2)cc1)Nc1ccc2c(n1)CCCC2 ZINC000880951506 GG On-Demand Anodyne SIGMAR1 18 41 c1cncc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880951514 DE On-Demand Anodyne FIMH 15 47 c1cncc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880951515 DE On-Demand Anodyne FIMH 15 47 CN(C(=O)Nc1ccc2c(n1)CCCC2)C1CCN(C(=O)c2ccccc2)CC1 ZINC000880951518 GH On-Demand Anodyne L3MBTL3 67 38 c1ccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)cc1 ZINC000880951553 DF On-Demand Anodyne FIMH 15 42 c1ccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)cc1 ZINC000880951554 DF On-Demand Anodyne FIMH 15 42 O=C(NCCCN1CCOC1=O)Nc1ccc2c(n1)CCCC2 ZINC000880951557 DD On-Demand Anodyne TYRO3 15 40 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H](N2CCCCC2)C1 ZINC000880951597 EG On-Demand Anodyne L3MBTL3 101 44 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H](N2CCCCC2)C1 ZINC000880951598 EG On-Demand Anodyne L3MBTL3 101 44 COCCNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880951623 GD On-Demand Anodyne CA2 15 42 O=C1C(=O)N(Cc2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)c2ccccc21 ZINC000880951625 GD On-Demand Anodyne ALDH1A1 42 35 O=C1C(=O)N(Cc2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)c2ccccc21 ZINC000880951626 GD On-Demand Anodyne ALDH1A1 42 35 Cc1ccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)cc1 ZINC000880951635 EG On-Demand Anodyne FIMH 15 44 Cc1ccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)cc1 ZINC000880951638 EG On-Demand Anodyne FIMH 15 44 O=C(Nc1ccc2c(n1)CCCC2)N1CCN2CCCC[C@H]2C1 ZINC000880951681 DF On-Demand Anodyne L3MBTL3 66 38 O=C(Nc1ccc2c(n1)CCCC2)N1CCN2CCCC[C@@H]2C1 ZINC000880951682 DF On-Demand Anodyne L3MBTL3 66 38 O=C(NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1)C1CCCCC1 ZINC000880951685 GH On-Demand Anodyne EPHX2 25 44 COc1ccc2c(c1)CN(C(=O)Nc1ccc3c(n1)CCCC3)CC2 ZINC000880951691 EH On-Demand Anodyne HDAC6 23 40 O=C(NCCN1CCCS1(=O)=O)Nc1ccc2c(n1)CCCC2 ZINC000880951697 ED On-Demand Anodyne HTR1F 27 40 O=C(NOCc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880951701 CG On-Demand Anodyne SLC12A5 44 33 O=C(NCCCN1CCCCC1=O)Nc1ccc2c(n1)CCCC2 ZINC000880951709 EE On-Demand Anodyne TYRO3 20 42 CN1CCC[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951743 CE On-Demand Anodyne HTR1F 57 36 CC(=O)Nc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880951744 EG On-Demand Anodyne ROCK2 25 49 COCCCCNC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880951745 CF On-Demand Anodyne BCHE 45 33 CCCCCCn1cc([C@@H](O)c2ccc(Cl)cc2)nn1 ZINC000880951752 CH On-Demand Anodyne SOAT1 19 41 CCCCCCn1cc([C@H](O)c2ccc(Cl)cc2)nn1 ZINC000880951753 CH On-Demand Anodyne SOAT1 19 41 COCCCCCNC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880951765 CF On-Demand Anodyne BCHE 53 35 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@H](N2CCCC2)C1 ZINC000880951768 DF On-Demand Anodyne L3MBTL3 104 45 O=C(Nc1ccc2c(n1)CCCC2)N1CC[C@@H](N2CCCC2)C1 ZINC000880951769 DF On-Demand Anodyne L3MBTL3 104 45 O=C(NCc1ccc(C(=O)N2CCOCC2)cc1)Nc1ccc2c(n1)CCCC2 ZINC000880951803 GF On-Demand Anodyne NAMPT 15 42 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951857 FD On-Demand Anodyne EPHX2 17 40 CC(=O)c1cccc(OCc2cn(CCO)nn2)c1 ZINC000880951896 CD On-Demand Anodyne FIMH 17 40 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951910 FG On-Demand Anodyne ACACB 16 42 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951910 FG On-Demand Anodyne CACNA1I 41 32 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951912 FG On-Demand Anodyne ACACB 16 42 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880951912 FG On-Demand Anodyne CACNA1I 41 32 CCS(=O)(=O)NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880951921 FD On-Demand Anodyne CCR8 81 38 O=C(CNC(=O)Nc1ccc2c(n1)CCCC2)Nc1cccnc1 ZINC000880951929 EE On-Demand Anodyne NAMPT 34 40 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne DRD4 21 53 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne SIGMAR1 21 46 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne SSTR5 62 37 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne CCR3 26 40 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne CXCR3 27 44 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccncc2)CC1 ZINC000880951953 FG On-Demand Anodyne MCHR1 37 45 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880951999 GE On-Demand Anodyne HDAC10 22 41 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880951999 GE On-Demand Anodyne HDAC3 25 41 CNCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880951999 GE On-Demand Anodyne HDAC6 19 41 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880952000 GE On-Demand Anodyne HDAC10 22 41 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880952000 GE On-Demand Anodyne HDAC3 25 41 CNCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)c1 ZINC000880952000 GE On-Demand Anodyne HDAC6 19 41 COc1ccc(-c2cn(C[C@@H]3CCC4(CCOCC4)CO3)nn2)cn1 ZINC000880952002 EE On-Demand Anodyne PDE5A 45 34 COc1ccc(-c2cn(C[C@H]3CCC4(CCOCC4)CO3)nn2)cn1 ZINC000880952003 EE On-Demand Anodyne PDE5A 45 34 CN1CCO[C@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880952034 DD On-Demand Anodyne HTR1F 40 38 CN1CCO[C@@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880952035 DD On-Demand Anodyne HTR1F 40 38 Cn1cc(CN2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)cn1 ZINC000880952065 FE On-Demand Anodyne FAAH 15 41 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2cccnn2)CC1 ZINC000880952113 EE On-Demand Anodyne FAAH 23 42 CNc1nc(C(=O)N2CC(C)(C)[C@H]2c2ccco2)cs1 ZINC000880952118 CG On-Demand Anodyne TRPC6 58 37 CNc1nc(C(=O)N2CC(C)(C)[C@H]2c2ccco2)cs1 ZINC000880952118 CG On-Demand Anodyne TRPC3 52 37 CNc1nc(C(=O)N2CC(C)(C)[C@@H]2c2ccco2)cs1 ZINC000880952119 CG On-Demand Anodyne TRPC6 58 37 CNc1nc(C(=O)N2CC(C)(C)[C@@H]2c2ccco2)cs1 ZINC000880952119 CG On-Demand Anodyne TRPC3 52 37 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)c2ccccc2F)CC1 ZINC000880952136 GH On-Demand Anodyne EPHX2 32 41 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952168 EF On-Demand Anodyne ADRB2 42 43 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952168 EF On-Demand Anodyne ADRB1 68 43 O=C(NC[C@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952168 EF On-Demand Anodyne ADRB3 38 43 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952169 EF On-Demand Anodyne ADRB2 42 43 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952169 EF On-Demand Anodyne ADRB1 68 43 O=C(NC[C@@H](O)COc1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952169 EF On-Demand Anodyne ADRB3 38 43 O=C(NCCCCn1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880952178 DF On-Demand Anodyne TBXAS1 47 45 O=C(NCCCCn1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880952178 DF On-Demand Anodyne QPCT 51 50 N#Cc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880952276 DG On-Demand Mild ROCK2 18 45 O=C(NCCNC(=O)c1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952319 EF On-Demand Anodyne ACHE 34 44 O=C(NCCNC(=O)c1ccccc1)Nc1ccc2c(n1)CCCC2 ZINC000880952319 EF On-Demand Anodyne BCHE 54 44 O=C(NCc1cccc(O)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952323 CF On-Demand Anodyne ROCK2 20 46 O=C(NCc1cccc(O)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952323 CF On-Demand Anodyne PKN1 15 46 O=C(NCc1cccc(O)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952323 CF On-Demand Anodyne IKBKE 15 46 O=C(NCc1cccc(O)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952323 CF On-Demand Anodyne PAK1 15 46 O=C(NCc1cccc(O)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952323 CF On-Demand Anodyne DMPK 15 46 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880952325 GG On-Demand Anodyne EPHX2 39 56 CCOC(=O)N1CCCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952374 EF On-Demand Anodyne P2RY12 52 35 O=C(NCc1ccc(Cl)nc1)Nc1ccc2c(n1)CCCC2 ZINC000880952393 DG On-Demand Anodyne NAMPT 17 47 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(CCO)CC1 ZINC000880952426 DD On-Demand Anodyne SLC6A5 16 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCN(CC2CC2)C1 ZINC000880952448 DF On-Demand Anodyne CCR3 48 36 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCN(CC2CC2)C1 ZINC000880952449 DF On-Demand Anodyne CCR3 48 36 C=C(C)CN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952450 EG On-Demand Mild CXCR3 19 40 O=C(Nc1ccccc1)NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952451 GH On-Demand Anodyne EPHX2 57 43 CN1CCC(CNC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952475 DE On-Demand Anodyne HTR1F 72 44 CN1CCC(CNC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952475 DE On-Demand Anodyne CACNA1I 40 37 O=C(Nc1ccc2c(n1)CCCC2)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880952495 EF On-Demand Anodyne CCR3 20 40 O=C(Nc1ccc2c(n1)CCCC2)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880952496 EF On-Demand Anodyne CCR3 20 40 O=C(CNC(=O)Nc1ccc2c(n1)CCCC2)NCc1ccccc1 ZINC000880952521 EE On-Demand Anodyne BCHE 49 32 COCCn1cc(NC(=O)Nc2ccc3c(n2)CCCC3)cn1 ZINC000880952525 DE On-Demand Anodyne PANC 50 33 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952558 GH On-Demand Anodyne EPHX2 28 49 COCCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952567 EE On-Demand Anodyne HTR4 55 40 COCCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952567 EE On-Demand Anodyne HTR1F 42 32 COCCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952567 EE On-Demand Anodyne SSTR5 40 34 COCCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952567 EE On-Demand Anodyne CXCR3 17 40 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952582 EF On-Demand Anodyne PANC 52 34 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952583 EF On-Demand Anodyne PANC 52 34 Cc1noc(C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)n1 ZINC000880952596 EG On-Demand Anodyne HTR1F 42 32 Cc1noc(C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)n1 ZINC000880952596 EG On-Demand Anodyne SMO 41 42 Cc1noc(C2CCN(C(=O)Nc3ccc4c(n3)CCCC4)CC2)n1 ZINC000880952596 EG On-Demand Anodyne ETHR 54 35 CCCCNC(=O)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952606 FG On-Demand Anodyne TBK1 47 33 CCCCCN(CCO)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952618 DF On-Demand Anodyne SOAT1 21 41 CN1CCN(C)[C@@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880952624 DD On-Demand Anodyne HTR1F 44 37 CN1CCN(C)[C@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880952625 DD On-Demand Anodyne HTR1F 44 37 Cc1nc(CN2CCC(CNC(=O)Nc3ccc4c(n3)CCCC4)CC2)oc1C ZINC000880952626 GH On-Demand Anodyne HTR4 52 36 Cc1nc(CN2CCC(CNC(=O)Nc3ccc4c(n3)CCCC4)CC2)oc1C ZINC000880952626 GH On-Demand Anodyne CACNA1I 54 38 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne OPRM1 42 42 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne MME 44 37 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne ANPEP 44 32 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne FCER2 62 39 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne CTSB 15 41 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne NPFFR2 62 37 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne CAPNS1 45 30 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne HLA-DRB1 52 36 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne MMP11 50 32 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne CAPN1 32 41 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne ACE2 40 33 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne MC1R 40 36 NC(=O)[C@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952637 EE On-Demand Anodyne NPFFR1 68 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne OPRM1 42 42 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne MME 44 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne ANPEP 44 32 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne FCER2 62 39 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne CTSB 15 41 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne NPFFR2 62 37 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne CAPNS1 45 30 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne HLA-DRB1 52 36 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne MMP11 50 32 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne CAPN1 32 41 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne ACE2 40 33 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne MC1R 40 36 NC(=O)[C@@H](Cc1ccccc1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952638 EE On-Demand Anodyne NPFFR1 68 37 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@H](N2CCCC2)C1 ZINC000880952639 EG On-Demand Anodyne L3MBTL3 73 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCC[C@@H](N2CCCC2)C1 ZINC000880952641 EG On-Demand Anodyne L3MBTL3 73 40 CCC(CC)C(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952656 FH On-Demand Anodyne EPHX2 35 45 Cc1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)n1 ZINC000880952705 CF On-Demand Anodyne SORT1 19 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(N2CCCCC2)CC1 ZINC000880952716 EG On-Demand Anodyne L3MBTL3 116 45 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne ALDH2 45 31 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne MAOB 56 50 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne RAF1 24 41 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne MTNR1A 57 41 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne MTNR1B 55 41 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne HSD17B3 18 50 COc1ccc2c(C)c(CCC(=O)NCc3ccc(O)cc3)c(=O)oc2c1 ZINC000880952717 FG On-Demand Anodyne NQO1 67 51 CCCCCCn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880952720 CD On-Demand Anodyne GBA 15 48 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880952726 FF On-Demand Anodyne HCN1 65 39 O=C(NCC1(N2CCCC2)CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880952726 FF On-Demand Anodyne HCN4 50 32 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880952729 FE On-Demand Anodyne EPHX2 23 42 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccccn2)CC1 ZINC000880952758 FG On-Demand Anodyne SIGMAR1 15 42 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccccn2)CC1 ZINC000880952758 FG On-Demand Anodyne SSTR5 51 35 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccccn2)CC1 ZINC000880952758 FG On-Demand Anodyne EPHX2 17 41 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(Cc2ccccn2)CC1 ZINC000880952758 FG On-Demand Anodyne CXCR3 20 44 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880952762 GG On-Demand Anodyne EPHX2 38 48 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880952762 GG On-Demand Anodyne L3MBTL3 71 35 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(CC2CC2)CC1 ZINC000880952763 EF On-Demand Anodyne CXCR3 15 41 CS(=O)(=O)N1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880952778 ED On-Demand Anodyne NPY5R 17 40 CN1CCC[C@H](CNC(=O)Nc2ccc3c(n2)CCCC3)C1 ZINC000880952829 DE On-Demand Anodyne HTR1F 51 40 CNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880952867 FD On-Demand Anodyne CA2 20 46 CNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880952867 FD On-Demand Anodyne CA1 17 46 CNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880952867 FD On-Demand Anodyne CA4 19 46 CNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880952867 FD On-Demand Anodyne CA9 18 40 CNS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880952867 FD On-Demand Anodyne NAMPT 53 34 C[C@@H](Cn1cncn1)NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880952871 DD On-Demand Anodyne HIS3 79 35 C[C@H](NC(=O)Nc1ccc2c(n1)CCCC2)c1cccnc1 ZINC000880952882 CG On-Demand Anodyne KCNA5 17 40 O=C(Nc1ccc2c(n1)CCCC2)N1CCN2CCC[C@H]2C1 ZINC000880952916 DE On-Demand Anodyne L3MBTL3 49 36 O=C(Nc1ccc2c(n1)CCCC2)N1CCN2CCC[C@@H]2C1 ZINC000880952917 DE On-Demand Anodyne L3MBTL3 49 36 Fc1ccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cn1 ZINC000880953005 EH On-Demand Anodyne FIMH 18 40 Fc1ccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cn1 ZINC000880953006 EH On-Demand Anodyne FIMH 18 40 Fc1ccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cn1 ZINC000880953007 EH On-Demand Anodyne FIMH 18 40 Fc1ccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cn1 ZINC000880953008 EH On-Demand Anodyne FIMH 18 40 COC(=O)[C@@H]1CCCN(Cc2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)C1 ZINC000880953042 GF On-Demand Anodyne SLC6A1 111 36 COC(=O)[C@@H]1CCCN(Cc2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)C1 ZINC000880953043 GF On-Demand Anodyne SLC6A1 111 36 COC(=O)[C@@H]1CCCN(Cc2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)C1 ZINC000880953044 GF On-Demand Anodyne SLC6A1 111 36 COC(=O)[C@@H]1CCCN(Cc2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)C1 ZINC000880953045 GF On-Demand Anodyne SLC6A1 111 36 Cn1cc([C@@H]2CCN(C(=O)Nc3ccc4c(n3)CCCC4)C2)cn1 ZINC000880953066 EF On-Demand Anodyne HTR1F 62 34 N#Cc1ccc(Cn2cc(CCCCNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880953083 GG On-Demand Mild CAPN2 47 33 N#Cc1ccc(Cn2cc(CCCCNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880953083 GG On-Demand Mild NPR 49 35 O=C(NCCN1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953105 DD On-Demand Anodyne EPHX2 20 44 CC(C)(C)OC(=O)N1CCC(O)(c2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953121 GG On-Demand Anodyne KDM1A 19 50 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2ncccn2)CC1 ZINC000880953125 EE On-Demand Anodyne FAAH 23 42 CCNC(=O)CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953127 ED On-Demand Anodyne SLC27A1 47 38 CO[C@@H]1CN(C(=O)OC(C)(C)C)C[C@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953140 GF On-Demand Mild KDM1A 16 43 CN(Cc1ccc(Cl)nc1)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880953144 EH On-Demand Anodyne NACHRBETA2 19 41 CC(C)(C)OC(=O)NCCSCc1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953180 FF On-Demand Mild KDM1A 17 45 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953182 ED On-Demand Anodyne DRD4 33 45 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953182 ED On-Demand Anodyne SIGMAR1 15 53 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953182 ED On-Demand Anodyne LSS 18 47 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953182 ED On-Demand Anodyne FAAH 23 49 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880953182 ED On-Demand Anodyne KDM1A 16 43 N#Cc1cccnc1N1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953188 FF On-Demand Mild P2RY12 15 41 CC(=O)Nc1cccc(NC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880953236 DH On-Demand Anodyne KCNK3 66 35 CC(=O)Nc1cccc(NC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880953236 DH On-Demand Anodyne KCNK9 60 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(C2CCC2)CC1 ZINC000880953276 DF On-Demand Anodyne L3MBTL3 57 36 CC(C)(C)OC(=O)N1CC(O)(c2cn(Cc3ccc(Cl)cc3)nn2)C1 ZINC000880953302 FE On-Demand Anodyne KDM1A 18 47 CC(C)(C)OC(=O)N1CCCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953303 GF On-Demand Mild GPR119 18 43 CC(C)(C)OC(=O)N1CCCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953303 GF On-Demand Mild KDM1A 21 54 CO[C@@H]1CN(C(=O)OC(C)(C)C)C[C@H]1c1cn(Cc2ccc(Cl)cc2)nn1 ZINC000880953312 GG On-Demand Anodyne KDM1A 17 46 CC(C)(C)OC(=O)N1CCC(c2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953313 FG On-Demand Mild GPR119 48 45 CC(C)(C)OC(=O)N1CCC(c2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953313 FG On-Demand Mild KDM1A 18 48 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880953329 FF On-Demand Anodyne EPHX2 25 41 CCOC(=O)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953333 EF On-Demand Anodyne PTR1 45 32 CCOC(=O)N1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953361 EE On-Demand Anodyne P2RY12 58 35 O=C(Nc1cnn(Cc2ccncc2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880953387 EG On-Demand Anodyne RPS6KA3 18 45 O=C(Nc1cnn(Cc2ccncc2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880953387 EG On-Demand Anodyne PANC 45 35 O=C(Nc1ccc2c(n1)CCCC2)N1CCc2cncnc2C1 ZINC000880953448 DE On-Demand Anodyne MAPK1 47 38 CCOC[C@H](O)CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953461 FD On-Demand Anodyne ACOX1 51 39 CC1(C)CCC[C@H](Cn2cc(-c3cccnc3)nn2)O1 ZINC000880953469 CF On-Demand Anodyne FIMH 16 50 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880953509 EF On-Demand Anodyne HTR1F 40 34 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1ccc2c(n1)CCCC2 ZINC000880953510 EF On-Demand Anodyne HTR1F 40 34 CCCn1cc(COc2ccc(N)cc2)nn1 ZINC000880953512 BD On-Demand Clean FIMH 15 41 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne HTR1A 64 51 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne DRD2 60 45 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne DRD4 31 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne ADRA1D 23 40 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne HTR2A 50 43 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne HTR2C 30 43 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne ADRA1A 26 40 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne DRD3 73 48 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne HTR7 44 42 O=C(NCCCN1CCN(c2ncccn2)CC1)Nc1ccc2c(n1)CCCC2 ZINC000880953536 GE On-Demand Anodyne CCR3 22 40 CN(Cc1cn(Cc2ccc(C#N)cc2)nn1)C(=O)OC(C)(C)C ZINC000880953562 EF On-Demand Mild KDM1A 15 42 CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953563 CD On-Demand Anodyne HTR1F 53 34 CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953563 CD On-Demand Anodyne HRH4 15 42 O=C(NCc1cccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880953567 CF On-Demand Anodyne NAMPT 88 48 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953572 GF On-Demand Mild SIGMAR1 21 41 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953572 GF On-Demand Mild SSTR5 44 37 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953572 GF On-Demand Mild MCHR1 33 41 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953572 GF On-Demand Mild KDM1A 17 43 CN(Cc1cn(Cc2ccc(Cl)cc2)nn1)C(=O)OC(C)(C)C ZINC000880953586 EG On-Demand Anodyne KDM1A 17 45 O=C(NCCCN1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953588 DD On-Demand Anodyne BCHE 19 42 O=C(NCCCN1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953588 DD On-Demand Anodyne CHRNA7 15 46 O=C(NCCCN1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953588 DD On-Demand Anodyne EPHX2 21 42 N#Cc1ccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953607 EI On-Demand Mild FIMH 15 40 N#Cc1ccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953616 EI On-Demand Mild FIMH 15 40 Cn1cnnc1C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953617 EF On-Demand Anodyne HTR1F 60 34 N#Cc1ccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953618 EI On-Demand Mild FIMH 15 40 N#Cc1ccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953621 EI On-Demand Mild FIMH 15 40 CCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953677 DF On-Demand Anodyne EPHX2 33 40 CCN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953677 DF On-Demand Anodyne CXCR3 22 41 Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880953687 EH On-Demand Anodyne FIMH 18 40 CC(C)(C)OC(=O)N1CCC[C@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880953688 FG On-Demand Mild GPR119 27 47 CC(C)(C)OC(=O)N1CCC[C@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880953688 FG On-Demand Mild KDM1A 16 44 Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880953689 EH On-Demand Anodyne FIMH 18 40 CC(C)(C)OC(=O)N1CCC[C@@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880953690 FG On-Demand Mild GPR119 27 47 CC(C)(C)OC(=O)N1CCC[C@@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880953690 FG On-Demand Mild KDM1A 16 44 Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880953691 EH On-Demand Anodyne FIMH 18 40 CCCn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880953692 CD On-Demand Anodyne G2YM83_BOTF4 76 39 Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880953693 EH On-Demand Anodyne FIMH 18 40 NCc1ccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953703 EH On-Demand Anodyne FIMH 18 41 NCc1ccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953706 EH On-Demand Anodyne FIMH 18 41 NCc1ccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953708 EH On-Demand Anodyne FIMH 18 41 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CASP3 18 42 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne BMP1 20 40 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne KLK3 78 36 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CTSB 67 46 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne PAPA1_CARPA 73 37 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CYSP_TRYCR 53 38 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CTSK 41 45 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CTSL 46 38 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne GBA 15 41 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CAPNS1 67 40 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CTSS 19 42 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne GHSR 33 44 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CAPN1 88 46 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CASP1 21 41 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne CAPN2 136 46 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne NPR 87 43 CCCn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880953709 CE On-Demand Anodyne PDS 46 34 NCc1ccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953710 EH On-Demand Anodyne FIMH 18 41 NCc1ccc(OCc2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953741 GH On-Demand Anodyne FIMH 15 46 NCc1ccc(OCc2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880953744 GH On-Demand Anodyne FIMH 15 46 NCc1ccc(OCc2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953745 GH On-Demand Anodyne FIMH 15 46 NCc1ccc(OCc2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880953746 GH On-Demand Anodyne FIMH 15 46 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc2c(n1)CCCC2 ZINC000880953747 FF On-Demand Anodyne NAMPT 23 43 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1ccc2c(n1)CCCC2 ZINC000880953747 FF On-Demand Anodyne SLC27A1 43 37 O=C(NCCCn1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880953760 CE On-Demand Anodyne TBXAS1 46 46 O=C(NCCCn1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880953760 CE On-Demand Anodyne QPCT 58 52 CCCn1cc(COc2ccc([C@@H](C)O)cc2)nn1 ZINC000880953766 CE On-Demand Anodyne FIMH 15 41 CCCn1cc(COc2ccc([C@H](C)O)cc2)nn1 ZINC000880953768 CE On-Demand Anodyne FIMH 15 41 O=C(Nc1ccc2c(n1)CCCC2)NC1CCN(C(=O)C2CC2)CC1 ZINC000880953780 EE On-Demand Anodyne EPHX2 37 50 O=C(NCCn1ccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880953803 CD On-Demand Anodyne QPCT 39 44 CC(C)(C)OC(=O)NCC(=O)NCc1cn(Cc2ccc(Cl)cc2)nn1 ZINC000880953805 GE On-Demand Anodyne KDM1A 18 46 Cn1ncc2c(N3CCN(C(=O)Nc4ccc5c(n4)CCCC5)CC3)ncnc21 ZINC000880953808 GD On-Demand Anodyne PDGFRB 56 38 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953813 FG On-Demand Mild DPP4 19 43 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953813 FG On-Demand Mild DPP8 22 43 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953813 FG On-Demand Mild DPP9 23 43 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953813 FG On-Demand Mild KDM1A 16 43 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953814 FG On-Demand Mild DPP4 19 43 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953814 FG On-Demand Mild DPP8 22 43 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953814 FG On-Demand Mild DPP9 23 43 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(Cc2ccc(C#N)cc2)nn1 ZINC000880953814 FG On-Demand Mild KDM1A 16 43 CC(C)(C)OC(=O)N1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953841 GE On-Demand Mild GPR119 27 46 CC(C)(C)OC(=O)N1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953841 GE On-Demand Mild KDM1A 22 58 O=C(NCc1ccc(-n2ccnc2)nc1)Nc1ccc2c(n1)CCCC2 ZINC000880953844 EF On-Demand Anodyne NOS2 85 35 O=C(NCc1ccc(-n2ccnc2)nc1)Nc1ccc2c(n1)CCCC2 ZINC000880953844 EF On-Demand Anodyne NAMPT 34 55 CC(=O)N1CCN(Cc2cn(Cc3ccc(C#N)cc3)nn2)CC1 ZINC000880953855 DC On-Demand Mild KDM1A 15 41 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953862 FF On-Demand Anodyne MTOR 46 43 O=C(NCc1cccnc1N1CCOCC1)Nc1ccc2c(n1)CCCC2 ZINC000880953862 FF On-Demand Anodyne SCN10A 20 46 N#Cc1ccc(Cn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880953872 DD On-Demand Mild KCNJ1 19 43 CCCn1cc(COc2cccc(N)c2)nn1 ZINC000880953873 BD On-Demand Anodyne DRTS_LEIMA 43 34 CCCn1cc(COc2cccc(N)c2)nn1 ZINC000880953873 BD On-Demand Anodyne FIMH 15 41 CNC(=O)CN1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880953875 ED On-Demand Anodyne CXCR3 17 41 O=C(Nc1cnn(Cc2ccccn2)c1)Nc1ccc2c(n1)CCCC2 ZINC000880953910 EG On-Demand Anodyne PANC 45 32 O=C(NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1)c1ccc(F)cc1 ZINC000880953981 GH On-Demand Anodyne HTR1F 46 39 O=C(NC1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1)c1ccc(F)cc1 ZINC000880953981 GH On-Demand Anodyne CCR3 19 46 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(Cc2ccncc2)CC1 ZINC000880953984 FF On-Demand Anodyne FAAH 24 44 CCCC[C@@H](CC)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880954020 EG On-Demand Anodyne G2YM83_BOTF4 67 35 CCCC[C@H](CC)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880954021 EG On-Demand Anodyne G2YM83_BOTF4 67 35 CCOC(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880954028 EF On-Demand Anodyne EPHX2 39 43 CCOC(=O)N1CCC(NC(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880954028 EF On-Demand Anodyne CCR8 24 41 O=C(NCc1ccc(O)cc1)c1cccnc1S ZINC000880954037 CE On-Demand Anodyne NAMPT 40 38 O=C(NCCCN1CCCCCC1=O)Nc1ccc2c(n1)CCCC2 ZINC000880954043 EF On-Demand Anodyne TYRO3 20 41 O=C(NCCCN1CCCC1=O)Nc1ccc2c(n1)CCCC2 ZINC000880954047 DE On-Demand Anodyne TYRO3 21 44 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(c2ccccn2)CC1 ZINC000880954049 EF On-Demand Anodyne SLC27A1 36 48 CC(=O)N1CCN(Cc2cn(Cc3ccc([N+](=O)[O-])cc3)nn2)CC1 ZINC000880954066 EC On-Demand Bother KDM1A 15 40 CC(=O)N1CCN(Cc2cn(Cc3ccc([N+](=O)[O-])cc3)nn2)CC1 ZINC000880954066 EC On-Demand Bother KCNJ1 30 46 OCc1cccc(OCc2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954103 GH On-Demand Anodyne FIMH 24 48 OCc1cccc(OCc2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954104 GH On-Demand Anodyne FIMH 24 48 OCc1cccc(OCc2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954105 GH On-Demand Anodyne FIMH 24 48 OCc1cccc(OCc2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954106 GH On-Demand Anodyne FIMH 24 48 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1Cl ZINC000880954126 JI On-Demand Anodyne CA2 19 45 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1Cl ZINC000880954126 JI On-Demand Anodyne CA1 17 45 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1Cl ZINC000880954126 JI On-Demand Anodyne CA4 18 43 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1Cl ZINC000880954126 JI On-Demand Anodyne UL54 61 36 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1Cl ZINC000880954126 JI On-Demand Anodyne NAMPT 44 36 CCN(Cc1nc(O)c2ccccc2n1)C(=O)Nc1ccc2c(n1)CCCC2 ZINC000880954183 GH On-Demand Anodyne BCHE 54 35 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880954187 GH On-Demand Anodyne EPHX2 32 44 O=C(NCc1ccccc1)C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880954187 GH On-Demand Anodyne TMPRSS11D 47 31 COC(=O)C1CCC(c2cn(Cc3ccc(Cl)cc3)nn2)CC1 ZINC000880954192 EG On-Demand Anodyne SIGMAR1 16 42 NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880954197 CC On-Demand Anodyne MMP8 18 46 CC(C)(C)OC(=O)N1CC[C@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880954202 FF On-Demand Mild GPR119 38 48 CC(C)(C)OC(=O)N1CC[C@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880954202 FF On-Demand Mild KDM1A 17 45 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880954203 FF On-Demand Mild GPR119 38 48 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(Cc3ccc(C#N)cc3)nn2)C1 ZINC000880954203 FF On-Demand Mild KDM1A 17 45 O=C(Nc1ccc2c(n1)CCCC2)N1CCN(Cc2cccnc2)CC1 ZINC000880954214 FF On-Demand Anodyne FAAH 30 45 CN(C)C(=O)c1cccc(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880954223 FF On-Demand Anodyne ROCK2 24 41 O=C(NCc1ccncc1)Nc1ccc2c(n1)CCCC2 ZINC000880954228 CF On-Demand Anodyne NAMPT 48 36 O=C(NCCc1cccnc1)Nc1ccc2c(n1)CCCC2 ZINC000880954247 CF On-Demand Anodyne NAMPT 39 48 O=C(CN1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1)N1CCCC1 ZINC000880954250 FD On-Demand Anodyne SLC27A1 42 34 O=[N+]([O-])c1ccc(Cn2cc([C@@H]3CCCCO3)nn2)cc1 ZINC000880954265 CE On-Demand Bother KCNJ1 18 43 O=[N+]([O-])c1ccc(Cn2cc([C@H]3CCCCO3)nn2)cc1 ZINC000880954266 CE On-Demand Bother KCNJ1 18 43 COC(=O)Cn1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880954312 DD On-Demand Anodyne MAP3K5 48 36 CC1(C)CCC[C@H](Cn2cc(CNC(=O)c3cccnc3Cl)nn2)O1 ZINC000880954389 FF On-Demand Anodyne G2YM83_BOTF4 74 38 CC1(C)CCC[C@H](Cn2cc(COc3cccc(C#N)c3)nn2)O1 ZINC000880954423 EG On-Demand Mild CHRNA10 25 43 C[C@H](O)c1ccc(OCc2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880954426 GI On-Demand Anodyne FIMH 15 46 C[C@H](O)c1ccc(OCc2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880954427 GI On-Demand Anodyne FIMH 15 46 C[C@H](O)c1ccc(OCc2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880954428 GI On-Demand Anodyne FIMH 15 46 C[C@H](O)c1ccc(OCc2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880954429 GI On-Demand Anodyne FIMH 15 46 CCCn1cc(COc2cccc(C(C)=O)c2)nn1 ZINC000880954566 CE On-Demand Anodyne FIMH 17 40 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954619 GG On-Demand Anodyne HDAC10 26 46 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954619 GG On-Demand Anodyne HDAC3 30 46 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954619 GG On-Demand Anodyne HDAC6 24 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954621 GG On-Demand Anodyne HDAC10 26 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954621 GG On-Demand Anodyne HDAC3 30 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880954621 GG On-Demand Anodyne HDAC6 24 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954623 GG On-Demand Anodyne HDAC10 26 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954623 GG On-Demand Anodyne HDAC3 30 46 NCC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954623 GG On-Demand Anodyne HDAC6 24 46 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954626 GG On-Demand Anodyne HDAC10 26 46 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954626 GG On-Demand Anodyne HDAC3 30 46 NCC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880954626 GG On-Demand Anodyne HDAC6 24 46 CC(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880954806 CC On-Demand Anodyne G2YM83_BOTF4 73 37 COc1ccc(O)c(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880955023 EF On-Demand Clean MTNR1A 40 41 COc1ccc(O)c(CNC(=O)Nc2ccc3c(n2)CCCC3)c1 ZINC000880955023 EF On-Demand Clean MTNR1B 32 41 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955036 GH On-Demand Anodyne HDAC10 25 44 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955036 GH On-Demand Anodyne HDAC3 27 44 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955036 GH On-Demand Anodyne HDAC6 22 44 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955037 GH On-Demand Anodyne HDAC10 25 44 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955037 GH On-Demand Anodyne HDAC3 27 44 NC(=O)Nc1cccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955037 GH On-Demand Anodyne HDAC6 22 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955038 GH On-Demand Anodyne HDAC10 25 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955038 GH On-Demand Anodyne HDAC3 27 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)c1 ZINC000880955038 GH On-Demand Anodyne HDAC6 22 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955039 GH On-Demand Anodyne HDAC10 25 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955039 GH On-Demand Anodyne HDAC3 27 44 NC(=O)Nc1cccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)c1 ZINC000880955039 GH On-Demand Anodyne HDAC6 22 44 O=C(Nc1ccc2c(n1)CCCC2)N1CCC(c2cc[nH]n2)CC1 ZINC000880955049 EG On-Demand Anodyne HTR1F 51 35 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880955064 JH On-Demand Bother KCNMA1 25 45 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880955064 JH On-Demand Bother PTGDR 22 42 COc1ccc([N+](=O)[O-])cc1NS(=O)(=O)c1ccc(Cl)c(C(=O)NCc2ccc(O)cc2)c1 ZINC000880955064 JH On-Demand Bother PTGDR2 20 42 COc1cccc(OCc2cn(C[C@@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880955065 EG On-Demand Anodyne FIMH 15 40 COc1cccc(OCc2cn(C[C@H]3CCCC(C)(C)O3)nn2)c1 ZINC000880955066 EG On-Demand Anodyne FIMH 15 40 c1ccc([C@@H]2CCC[C@H](Cn3cc(-c4cncnc4)nn3)O2)cc1 ZINC000880955067 DG On-Demand Anodyne FIMH 18 40 c1ccc([C@H]2CCC[C@@H](Cn3cc(-c4cncnc4)nn3)O2)cc1 ZINC000880955068 DG On-Demand Anodyne FIMH 18 40 c1ccc([C@H]2CCC[C@H](Cn3cc(-c4cncnc4)nn3)O2)cc1 ZINC000880955069 DG On-Demand Anodyne FIMH 18 40 c1ccc([C@@H]2CCC[C@@H](Cn3cc(-c4cncnc4)nn3)O2)cc1 ZINC000880955070 DG On-Demand Anodyne FIMH 18 40 CCCn1cc(CON)nn1 ZINC000880955370 AC On-Demand Anodyne GBA 15 40 CCCn1cc(-c2ccc([C@@H](O)C(F)(F)F)cc2)nn1 ZINC000880955380 CF On-Demand Anodyne FIMH 17 40 CCCn1cc(-c2ccc([C@H](O)C(F)(F)F)cc2)nn1 ZINC000880955381 CF On-Demand Anodyne FIMH 17 40 CC(=O)N1CCN(Cc2cn(Cc3ccc(Br)cc3)nn2)CC1 ZINC000880955409 GD On-Demand Anodyne KDM1A 16 42 CC1(C)CCC[C@H](Cn2cc(-c3ccccc3)nn2)O1 ZINC000880955416 CG On-Demand Anodyne FIMH 16 45 Cn1nccc1C1CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880955427 EG On-Demand Anodyne HTR1F 61 34 COCCNC(=O)c1cn(C[C@@H]2CCC[C@H](c3ccccc3)O2)nn1 ZINC000880955461 ED On-Demand Anodyne LGALS3 26 41 COCCNC(=O)c1cn(C[C@H]2CCC[C@H](c3ccccc3)O2)nn1 ZINC000880955462 ED On-Demand Anodyne LGALS3 26 41 COCCNC(=O)c1cn(C[C@@H]2CCC[C@@H](c3ccccc3)O2)nn1 ZINC000880955463 ED On-Demand Anodyne LGALS3 26 41 COCCNC(=O)c1cn(C[C@H]2CCC[C@@H](c3ccccc3)O2)nn1 ZINC000880955464 ED On-Demand Anodyne LGALS3 26 41 OCc1ccc(-c2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cn1 ZINC000880955514 FG On-Demand Anodyne FIMH 24 43 OCc1ccc(-c2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cn1 ZINC000880955516 FG On-Demand Anodyne FIMH 24 43 OCc1ccc(-c2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cn1 ZINC000880955518 FG On-Demand Anodyne FIMH 24 43 OCc1ccc(-c2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cn1 ZINC000880955520 FG On-Demand Anodyne FIMH 24 43 CCCn1cc(COc2ccc(Br)nc2)nn1 ZINC000880955549 CE On-Demand Anodyne FIMH 15 40 O=C(CN1C(=O)COc2ccc(Cl)cc21)NCc1ccc(O)cc1 ZINC000880955589 EE On-Demand Anodyne PIK3CG 21 43 OCCOCc1cn(C[C@@H]2CCC[C@H](c3ccccc3)O2)nn1 ZINC000880955713 DE On-Demand Anodyne FIMH 34 44 OCCOCc1cn(C[C@H]2CCC[C@H](c3ccccc3)O2)nn1 ZINC000880955714 DE On-Demand Anodyne FIMH 34 44 OCCOCc1cn(C[C@@H]2CCC[C@@H](c3ccccc3)O2)nn1 ZINC000880955715 DE On-Demand Anodyne FIMH 34 44 OCCOCc1cn(C[C@H]2CCC[C@@H](c3ccccc3)O2)nn1 ZINC000880955716 DE On-Demand Anodyne FIMH 34 44 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2ccc3c(n2)CCCC3)CC1 ZINC000880955717 GG On-Demand Anodyne NPY5R 31 41 OCc1ccc(OCc2cn(C[C@@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880955735 GH On-Demand Anodyne FIMH 23 50 OCc1ccc(OCc2cn(C[C@H]3CCC[C@H](c4ccccc4)O3)nn2)cc1 ZINC000880955736 GH On-Demand Anodyne FIMH 23 50 OCc1ccc(OCc2cn(C[C@@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880955737 GH On-Demand Anodyne FIMH 23 50 OCc1ccc(OCc2cn(C[C@H]3CCC[C@@H](c4ccccc4)O3)nn2)cc1 ZINC000880955738 GH On-Demand Anodyne FIMH 23 50 c1ccc([C@@H]2CCC[C@@H](Cn3cc(-c4cccnc4)nn3)O2)cc1 ZINC000880955796 DH On-Demand Anodyne FIMH 22 52 c1ccc([C@H]2CCC[C@H](Cn3cc(-c4cccnc4)nn3)O2)cc1 ZINC000880955797 DH On-Demand Anodyne FIMH 22 52 c1ccc([C@@H]2CCC[C@H](Cn3cc(-c4cccnc4)nn3)O2)cc1 ZINC000880955798 DH On-Demand Anodyne FIMH 22 52 c1ccc([C@H]2CCC[C@@H](Cn3cc(-c4cccnc4)nn3)O2)cc1 ZINC000880955799 DH On-Demand Anodyne FIMH 22 52 CC(=O)Cn1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880955854 DC On-Demand Anodyne KDM1A 22 51 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCCC2)ccc1Br ZINC000880955863 IF On-Demand Anodyne NAMPT 95 50 CCC[C@H](NC(=O)Nc1cc(CC)ccc1Br)C(N)=O ZINC000880955973 EF On-Demand Anodyne ANPEP 16 42 COCCNC(=O)c1cn(CC(=O)Nc2ccc(SC(F)F)cc2)nn1 ZINC000880956038 GD On-Demand Anodyne LGALS3 24 40 CC(=O)N1CCN(Cc2cn(Cc3ccccc3Cl)nn2)CC1 ZINC000880956100 ED On-Demand Anodyne DRD4 21 40 CC(=O)N1CCN(Cc2cn(Cc3ccccc3Cl)nn2)CC1 ZINC000880956100 ED On-Demand Anodyne SIGMAR1 15 48 CC(=O)N1CCN(Cc2cn(Cc3ccccc3Cl)nn2)CC1 ZINC000880956100 ED On-Demand Anodyne FAAH 15 40 CC(=O)Cn1cc(CN2CCC(NC(=O)OC(C)(C)C)CC2)nn1 ZINC000880956117 ED On-Demand Anodyne SSTR5 46 36 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)cc3Cl)nn2)CC1 ZINC000880956142 FE On-Demand Anodyne KDM1A 17 42 c1ccc([C@@H]2CCC[C@@H](Cn3cc(-c4ccncc4)nn3)O2)cc1 ZINC000880956244 DH On-Demand Anodyne FIMH 16 43 c1ccc([C@H]2CCC[C@H](Cn3cc(-c4ccncc4)nn3)O2)cc1 ZINC000880956245 DH On-Demand Anodyne FIMH 16 43 c1ccc([C@@H]2CCC[C@H](Cn3cc(-c4ccncc4)nn3)O2)cc1 ZINC000880956246 DH On-Demand Anodyne FIMH 16 43 c1ccc([C@H]2CCC[C@@H](Cn3cc(-c4ccncc4)nn3)O2)cc1 ZINC000880956247 DH On-Demand Anodyne FIMH 16 43 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne CTSB 43 38 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne CYSP_TRYCR 48 37 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne CAPNS1 59 35 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne GHSR 24 44 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne CAPN1 63 38 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne CAPN2 104 38 CC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880956394 EE On-Demand Anodyne NPR 65 40 CC(=O)N1CCN(Cc2cn(Cc3cccc(Cl)c3)nn2)CC1 ZINC000880956439 ED On-Demand Anodyne DRD2 15 44 CC(=O)N1CCN(Cc2cn(Cc3cccc(Cl)c3)nn2)CC1 ZINC000880956439 ED On-Demand Anodyne DRD4 32 43 CC(=O)N1CCN(Cc2cn(Cc3cccc(Cl)c3)nn2)CC1 ZINC000880956439 ED On-Demand Anodyne SIGMAR1 22 52 CC(=O)N1CCN(Cc2cn(Cc3cccc(Cl)c3)nn2)CC1 ZINC000880956439 ED On-Demand Anodyne FAAH 32 54 CC(=O)N1CCN(Cc2cn(Cc3cccc(Cl)c3)nn2)CC1 ZINC000880956439 ED On-Demand Anodyne CDC7 16 40 CC(=O)Cn1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880956562 CE On-Demand Anodyne MAP3K5 47 35 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne KLK3 64 34 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CTSB 48 40 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CYSP_TRYCR 45 35 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CTSK 28 40 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CAPNS1 61 36 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CAPN1 68 40 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne CAPN2 109 40 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne NPR 67 38 CC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880956654 CD On-Demand Anodyne PDS 45 34 CCOc1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880956692 JI On-Demand Anodyne ADRB2 17 44 CCOc1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880956692 JI On-Demand Anodyne ADRB1 21 44 CCOc1ccc(NS(=O)(=O)c2ccc(Cl)c(C(=O)NCc3ccc(O)cc3)c2)cc1 ZINC000880956692 JI On-Demand Anodyne ADRB3 26 50 CC(=O)Cn1cc([C@@H]2CCN(C(=O)OC(C)(C)C)C2)nn1 ZINC000880956695 CD On-Demand Anodyne GPR119 42 40 CC(=O)Cn1cc([C@H]2CCN(C(=O)OC(C)(C)C)C2)nn1 ZINC000880956696 CD On-Demand Anodyne GPR119 42 40 CC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880956698 CD On-Demand Anodyne MMP8 19 48 CC(=O)N1CCN(Cc2cn(Cc3ccc(F)cc3)nn2)CC1 ZINC000880956820 DD On-Demand Anodyne SIGMAR1 23 41 CC(=O)N1CCN(Cc2cn(Cc3ccc(F)cc3)nn2)CC1 ZINC000880956820 DD On-Demand Anodyne MLNR 48 38 CC(=O)N1CCN(Cc2cn(Cc3ccc(F)cc3)nn2)CC1 ZINC000880956820 DD On-Demand Anodyne KDM1A 16 42 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)c(Cl)c3)nn2)CC1 ZINC000880956844 FE On-Demand Anodyne DRD4 19 43 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)c(Cl)c3)nn2)CC1 ZINC000880956844 FE On-Demand Anodyne OPRK1 21 43 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)c(Cl)c3)nn2)CC1 ZINC000880956844 FE On-Demand Anodyne SIGMAR1 20 67 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)c(Cl)c3)nn2)CC1 ZINC000880956844 FE On-Demand Anodyne CCR3 15 41 CC(=O)N1CCN(Cc2cn(Cc3ccc(Cl)c(Cl)c3)nn2)CC1 ZINC000880956844 FE On-Demand Anodyne KDM1A 16 41 CC(=O)Cn1cc(CN2CCCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880956861 ED On-Demand Anodyne KDM1A 21 48 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Br ZINC000880956879 JE On-Demand Anodyne DPOL_VZVD 40 38 O=C(NCc1ccc(O)cc1)c1cc(S(=O)(=O)N2CCOCC2)ccc1Br ZINC000880956879 JE On-Demand Anodyne NAMPT 77 52 CC(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880956921 DD On-Demand Anodyne GPR119 47 44 CC(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880956921 DD On-Demand Anodyne KDM1A 17 40 CC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880956933 CC On-Demand Anodyne PAOX 17 40 O=C(Cn1cc(CN2CCC[C@H]2CO)nn1)Nc1ccc(SC(F)F)cc1 ZINC000880957359 GE On-Demand Anodyne AURKC 15 40 O=C(Cn1cc(CN2CCC[C@@H]2CO)nn1)Nc1ccc(SC(F)F)cc1 ZINC000880957360 GE On-Demand Anodyne AURKC 15 40 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(F)c(Cl)c2)nn1 ZINC000880957386 ED On-Demand Anodyne MAP3K8 38 40 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(F)c(Cl)c3)nn2)CC1 ZINC000880957404 GD On-Demand Anodyne NPY2R 19 40 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(F)c(Cl)c3)nn2)CC1 ZINC000880957404 GD On-Demand Anodyne ERBB4 44 34 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(F)c(Cl)c3)nn2)CC1 ZINC000880957404 GD On-Demand Anodyne MCHR1 27 42 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(F)c(Cl)c3)nn2)CC1 ZINC000880957404 GD On-Demand Anodyne MAP3K8 45 38 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957408 FG On-Demand Anodyne HDAC10 19 40 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957408 FG On-Demand Anodyne HDAC3 19 40 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957408 FG On-Demand Anodyne HDAC6 15 40 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957409 FG On-Demand Anodyne HDAC10 19 40 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957409 FG On-Demand Anodyne HDAC3 19 40 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(C(F)(F)F)c3)nn2)C1 ZINC000880957409 FG On-Demand Anodyne HDAC6 15 40 O=[N+]([O-])c1cccc(Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880957418 ED On-Demand Bother KCNJ1 23 44 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957436 EE On-Demand Mild HDAC10 20 42 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957436 EE On-Demand Mild HDAC3 22 42 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957436 EE On-Demand Mild HDAC6 18 45 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957437 EE On-Demand Mild HDAC10 20 42 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957437 EE On-Demand Mild HDAC3 22 42 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957437 EE On-Demand Mild HDAC6 18 45 CC(C)(C)OC(=O)NCc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957440 GF On-Demand Anodyne HDAC6 17 41 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne HDAC10 21 40 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne HDAC3 21 40 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne HDAC6 18 45 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne SLC1A1 25 41 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne SLC1A3 24 41 C[C@H](N)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957455 DD On-Demand Anodyne SLC1A2 36 41 CN(C(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1)c1ccccc1 ZINC000880957603 GG On-Demand Anodyne GPR119 43 42 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957641 DE On-Demand Anodyne MAP3K8 47 36 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957642 DE On-Demand Anodyne MAP3K8 47 36 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957645 FG On-Demand Anodyne HDAC10 20 40 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957645 FG On-Demand Anodyne HDAC3 20 40 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957645 FG On-Demand Anodyne HDAC6 17 43 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957647 GE On-Demand Anodyne CASR 26 48 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957647 GE On-Demand Anodyne LCK 15 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957647 GE On-Demand Anodyne EPHX2 31 55 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957672 EE On-Demand Anodyne HDAC10 20 41 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957672 EE On-Demand Anodyne HDAC3 22 41 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880957672 EE On-Demand Anodyne HDAC6 18 43 COC(=O)Cc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957762 ED On-Demand Anodyne HDAC10 21 41 COC(=O)Cc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957762 ED On-Demand Anodyne HDAC3 22 41 COC(=O)Cc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880957762 ED On-Demand Anodyne HDAC6 19 44 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957774 FF On-Demand Anodyne MAP3K8 32 40 O=C(Cn1cc(CC2(O)CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957799 FD On-Demand Anodyne ERBB4 48 37 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)c3cccnc3Cl)nn2)C1 ZINC000880957800 GD On-Demand Anodyne G2YM83_BOTF4 70 39 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)c3cccnc3Cl)nn2)C1 ZINC000880957802 GD On-Demand Anodyne G2YM83_BOTF4 70 39 COC(=O)Cc1cn(CC(=O)N(c2ccccc2)C(C)C)nn1 ZINC000880957812 DD On-Demand Anodyne CCKAR 15 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne EGFR 26 45 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne ERBB2 21 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne CHRNA7 17 43 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne EPHX2 25 48 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne ERBB4 49 44 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne EPHA6 22 43 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880957894 GD On-Demand Anodyne MAP3K8 59 46 CN(C(=O)Cn1cc(CN2CCOC2=O)nn1)c1ccccc1 ZINC000880957959 DC On-Demand Anodyne TSPO 25 41 COC(=O)Cc1cn(CC(=O)N(C)c2ccccc2)nn1 ZINC000880957974 CC On-Demand Anodyne TSPO 24 43 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880958030 EE On-Demand Anodyne CCR3 22 40 CC(=O)c1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880958031 EE On-Demand Anodyne CCR3 22 40 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958078 DE On-Demand Anodyne ERBB4 40 33 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958078 DE On-Demand Anodyne MCHR1 27 41 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958090 GF On-Demand Anodyne HDAC6 15 40 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958093 EE On-Demand Anodyne HDAC6 16 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958093 EE On-Demand Anodyne CCR2 41 35 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958094 EE On-Demand Anodyne HDAC6 16 41 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958094 EE On-Demand Anodyne CCR2 41 35 NOCc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880958108 DD On-Demand Anodyne HDAC10 19 40 NOCc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880958108 DD On-Demand Anodyne HDAC3 21 40 NOCc1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880958108 DD On-Demand Anodyne HDAC6 18 45 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)c1 ZINC000880958110 FE On-Demand Anodyne CASR 15 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)c1 ZINC000880958110 FE On-Demand Anodyne KCNK3 47 33 CC(=O)c1cccc(NC(=O)Cn2cc([C@H](O)c3ccccc3)nn2)c1 ZINC000880958111 FE On-Demand Anodyne CASR 15 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@H](O)c3ccccc3)nn2)c1 ZINC000880958111 FE On-Demand Anodyne KCNK3 47 33 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958126 DE On-Demand Anodyne ERBB4 46 32 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958127 DE On-Demand Anodyne ERBB4 46 32 CC[C@H](O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880958131 EE On-Demand Anodyne HDAC6 17 44 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958193 EE On-Demand Anodyne HDAC6 16 43 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958194 EE On-Demand Anodyne HDAC6 16 43 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(CC)ccc2Br)C1 ZINC000880958249 FG On-Demand Anodyne EPHX2 40 59 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(CC)ccc2Br)C1 ZINC000880958250 FG On-Demand Anodyne EPHX2 40 59 CC[C@@](C)(O)c1cn(CC(=O)Nc2cccc(C(F)(F)F)c2)nn1 ZINC000880958257 EF On-Demand Anodyne HDAC6 16 44 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958281 FF On-Demand Anodyne MCHR1 27 40 CC(C)(C)OC(=O)NCc1cn(CC(=O)Nc2ccc(F)c(Cl)c2)nn1 ZINC000880958304 GF On-Demand Anodyne MAP3K8 59 43 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958306 FG On-Demand Anodyne HDAC6 15 40 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958306 FG On-Demand Anodyne CCR2 46 38 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958307 FG On-Demand Anodyne HDAC6 15 40 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958307 FG On-Demand Anodyne CCR2 46 38 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958311 EF On-Demand Anodyne MCHR1 23 40 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958311 EF On-Demand Anodyne MAP3K8 43 36 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958312 EF On-Demand Anodyne MCHR1 23 40 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958312 EF On-Demand Anodyne MAP3K8 43 36 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958315 FG On-Demand Anodyne HDAC10 28 42 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958315 FG On-Demand Anodyne HDAC3 28 42 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958315 FG On-Demand Anodyne HDAC6 26 48 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958325 FD On-Demand Anodyne HDAC6 16 41 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958365 FD On-Demand Anodyne ERBB4 52 36 CC(=O)c1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880958379 FD On-Demand Anodyne CASR 40 47 CC(=O)c1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880958379 FD On-Demand Anodyne EPHX2 27 44 CC(=O)N1CCN(Cc2cn(Cc3cccc([N+](=O)[O-])c3)nn2)CC1 ZINC000880958387 EC On-Demand Bother FAAH 25 58 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne KLK3 46 31 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne PREP 48 47 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne CAPN1 41 35 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne CAPN2 63 35 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne TGM2 26 40 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)OCc1ccccc1 ZINC000880958414 FE On-Demand Anodyne NPR 59 34 O=C(Cn1cc(CNC(=O)C(F)(F)F)nn1)Nc1cccc(C(F)(F)F)c1 ZINC000880958499 GE On-Demand Anodyne HDAC6 15 44 CC(=O)c1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880958502 EE On-Demand Anodyne HDAC10 16 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880958502 EE On-Demand Anodyne HDAC3 18 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880958502 EE On-Demand Anodyne CCKBR 33 40 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880958503 EE On-Demand Anodyne HDAC10 16 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880958503 EE On-Demand Anodyne HDAC3 18 41 CC(=O)c1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880958503 EE On-Demand Anodyne CCKBR 33 40 O=[N+]([O-])c1cccc(Cn2cc([C@@H]3CCOC3)nn2)c1 ZINC000880958504 CD On-Demand Bother LUXR 17 44 O=[N+]([O-])c1cccc(Cn2cc([C@H]3CCOC3)nn2)c1 ZINC000880958505 CD On-Demand Bother LUXR 17 44 CN(C(=O)Cn1cc(CCCOc2cccnc2F)nn1)c1ccccc1 ZINC000880958527 FE On-Demand Anodyne MMP8 18 45 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958551 ED On-Demand Anodyne ERBB4 47 34 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1ccc(F)c(Cl)c1 ZINC000880958552 ED On-Demand Anodyne ERBB4 47 34 CC[C@@H]1CCCCN1C(=O)Cn1cc(Cn2cnc(-c3ccccc3)c2N)nn1 ZINC000880958649 GF On-Demand Anodyne CPT1A 61 35 CC[C@H]1CCCCN1C(=O)Cn1cc(Cn2cnc(-c3ccccc3)c2N)nn1 ZINC000880958650 GF On-Demand Anodyne CPT1A 61 35 CC[C@H]1CCCCN1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880958732 EE On-Demand Clean CPT1A 63 37 CC[C@@H]1CCCCN1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880958733 EE On-Demand Clean CPT1A 63 37 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CA2 15 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne ACE 66 51 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TYR 46 54 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne OPRM1 100 53 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne OPRD1 94 53 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CELA1 23 44 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MME 160 54 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne ANPEP 93 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TACR1 25 68 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSD 21 52 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTRA_BOVIN 53 35 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne FCER2 102 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne GRB2 48 46 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CASP3 20 58 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne BMP1 26 52 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NPY1R 35 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne KLK3 96 50 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSB 116 76 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PAPA1_CARPA 119 68 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CYSP_TRYCR 84 58 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CCKAR 49 53 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NTSR1 43 36 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSG 42 35 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSK 55 69 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSL 96 69 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CPA1 34 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CACNA1B 53 36 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PGA 37 44 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NPFFR2 50 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TIMP3 86 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TACR3 23 59 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NAALAD2 24 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CAPNS1 92 54 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP2 26 45 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP3 31 53 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP8 34 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne GRIA1 95 51 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne ECE1 39 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne HLA-DRB1 86 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CELA2A 51 35 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne REN 61 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne REN1 23 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne LNPEP 51 36 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne LGMN 15 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP11 77 38 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne F11 21 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne FURIN 65 52 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PTPRA 43 36 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne YARS 82 46 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CCKBR 26 43 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTSS 43 69 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CAPN1 145 62 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP9 33 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CASP1 36 54 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CTRC 27 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CAPN2 181 76 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne ACE2 84 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MC1R 53 37 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PLAU 24 43 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CASP6 15 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne CASP9 31 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TGM2 23 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne LAP3 47 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TPSAB1 57 52 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PROC 60 48 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne MMP1 36 56 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne FPR1 77 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NPR 92 45 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne AMP1_PLAFQ 57 46 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne XIAP 29 41 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PSMB5 83 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne BLA1_STEMA 62 36 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne QRFPR 41 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne KDM1A 16 55 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne NPFFR1 70 47 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne TMPRSS11D 34 45 O=C(N[C@H](Cc1ccccc1)C(=O)NCc1ccc(O)cc1)OCc1ccccc1 ZINC000880958741 HH On-Demand Anodyne PDS 52 36 CC[C@H]1CCCCN1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880958781 EE On-Demand Anodyne CPT1A 96 40 CC[C@@H]1CCCCN1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880958782 EE On-Demand Anodyne CPT1A 96 40 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CCCOc3cccnc3F)nn2)C1 ZINC000880958809 GE On-Demand Anodyne MMP8 17 44 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CCCOc3cccnc3F)nn2)C1 ZINC000880958811 GE On-Demand Anodyne MMP8 17 44 CC[C@@H]1CCCCN1C(=O)Cn1cc(COc2cccc(C(C)=O)c2)nn1 ZINC000880958825 FF On-Demand Anodyne CPT1A 101 37 CC[C@H]1CCCCN1C(=O)Cn1cc(COc2cccc(C(C)=O)c2)nn1 ZINC000880958826 FF On-Demand Anodyne CPT1A 101 37 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880958831 FD On-Demand Anodyne P2RY1 49 37 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880958831 FD On-Demand Anodyne EPHX2 51 37 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958845 GF On-Demand Anodyne EPHX2 50 38 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958846 GF On-Demand Anodyne EPHX2 50 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958867 FE On-Demand Anodyne P2RY1 41 35 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958867 FE On-Demand Anodyne EPHX2 54 41 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958868 FE On-Demand Anodyne P2RY1 41 35 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880958868 FE On-Demand Anodyne EPHX2 54 41 COC(=O)Cc1cn(CC(=O)N(C)Cc2ccccc2)nn1 ZINC000880958893 DC On-Demand Anodyne TSPO 15 40 O=C(NCc1cn(CC(=O)N2CCCCCC2)nn1)c1cccnc1Cl ZINC000880958897 GD On-Demand Anodyne G2YM83_BOTF4 66 34 O=C1CCC[C@@H](c2cn(CC(=O)Nc3ccc(OC(F)(F)F)cc3)nn2)C1 ZINC000880958918 GG On-Demand Anodyne EPHX2 49 42 O=C1CCC[C@@H](c2cn(CC(=O)Nc3ccc(OC(F)(F)F)cc3)nn2)C1 ZINC000880958918 GG On-Demand Anodyne TRAR 26 41 O=C1CCC[C@H](c2cn(CC(=O)Nc3ccc(OC(F)(F)F)cc3)nn2)C1 ZINC000880958919 GG On-Demand Anodyne EPHX2 49 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3ccc(OC(F)(F)F)cc3)nn2)C1 ZINC000880958919 GG On-Demand Anodyne TRAR 26 41 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958935 GE On-Demand Anodyne KLK3 55 32 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958935 GE On-Demand Anodyne PREP 32 47 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958935 GE On-Demand Anodyne CAPN1 45 36 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958935 GE On-Demand Anodyne CAPN2 70 36 C[C@@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958935 GE On-Demand Anodyne NPR 60 34 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958936 GE On-Demand Anodyne KLK3 55 32 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958936 GE On-Demand Anodyne PREP 32 47 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958936 GE On-Demand Anodyne CAPN1 45 36 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958936 GE On-Demand Anodyne CAPN2 70 36 C[C@H]1C[C@@H](C)CN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880958936 GE On-Demand Anodyne NPR 60 34 CC[C@H]1CCCCN1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880958937 FF On-Demand Anodyne CPT1A 63 35 CC[C@H]1CCCCN1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880958938 FF On-Demand Anodyne CPT1A 63 35 CC[C@@H]1CCCCN1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880958939 FF On-Demand Anodyne CPT1A 63 35 CC[C@@H]1CCCCN1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880958940 FF On-Demand Anodyne CPT1A 63 35 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880958960 EE On-Demand Anodyne P2RY1 47 35 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880958960 EE On-Demand Anodyne EPHX2 51 43 CC[C@@H]1CCCCN1C(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880958977 DE On-Demand Anodyne CPT1A 44 34 CC[C@H]1CCCCN1C(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880958978 DE On-Demand Anodyne CPT1A 44 34 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(CC(=O)N2CCCCCC2)nn1 ZINC000880959000 GF On-Demand Anodyne PREP 25 46 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(CC(=O)N2CCCCCC2)nn1 ZINC000880959001 GF On-Demand Anodyne PREP 25 46 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne ACE 19 41 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne FKBP1A 30 42 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne ELANE 24 40 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne CTRA_BOVIN 59 31 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne TRY1_BOVIN 51 32 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne CTSG 41 31 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne CPT1A 64 35 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne PREP 57 45 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne CELA2A 48 31 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne CAPN2 65 35 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne NPR 58 32 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959017 GE On-Demand Anodyne TMPRSS11D 40 35 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne ACE 19 41 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne FKBP1A 30 42 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne ELANE 24 40 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne CTRA_BOVIN 59 31 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne TRY1_BOVIN 51 32 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne CTSG 41 31 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne CPT1A 64 35 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne PREP 57 45 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne CELA2A 48 31 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne CAPN2 65 35 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne NPR 58 32 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880959018 GE On-Demand Anodyne TMPRSS11D 40 35 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959019 GD On-Demand Anodyne P2RY1 44 35 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959019 GD On-Demand Anodyne EPHX2 55 43 CC(C)(C)OC(=O)N1CCC(c2cn(CC(=O)N3CCCCCC3)nn2)CC1 ZINC000880959048 GF On-Demand Anodyne GPR119 39 40 CC[C@@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880959065 EE On-Demand Anodyne PREP 43 34 CC[C@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880959066 EE On-Demand Anodyne PREP 43 34 CC[C@@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880959067 EE On-Demand Anodyne PREP 43 34 CC[C@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880959068 EE On-Demand Anodyne PREP 43 34 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959069 FE On-Demand Anodyne P2RY1 56 39 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959069 FE On-Demand Anodyne EPHX2 54 41 CC[C@H]1CCCCN1C(=O)Cn1cc(C(=O)c2ccc(OC)cc2)nn1 ZINC000880959070 FE On-Demand Anodyne CPT1A 54 40 CC[C@@H]1CCCCN1C(=O)Cn1cc(C(=O)c2ccc(OC)cc2)nn1 ZINC000880959071 FE On-Demand Anodyne CPT1A 54 40 C[C@H](N)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959096 ED On-Demand Anodyne P2RY1 51 36 C[C@H](N)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959096 ED On-Demand Anodyne EPHX2 51 39 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959106 FE On-Demand Anodyne P2RY1 48 36 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959106 FE On-Demand Anodyne EPHX2 52 41 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959236 GF On-Demand Anodyne P2RY1 55 40 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959236 GF On-Demand Anodyne EPHX2 54 41 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959248 FD On-Demand Anodyne P2RY1 56 36 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959248 FD On-Demand Anodyne EPHX2 52 39 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959249 FD On-Demand Anodyne P2RY1 56 36 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880959249 FD On-Demand Anodyne EPHX2 52 39 CC(=O)N1CCN(Cc2cn(CC(=O)N(C)Cc3ccccc3)nn2)CC1 ZINC000880959278 FC On-Demand Anodyne FAAH 16 40 CC[C@@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2Cl)nn1 ZINC000880959305 EF On-Demand Anodyne CPT1A 55 35 CC[C@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2Cl)nn1 ZINC000880959306 EF On-Demand Anodyne CPT1A 55 35 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959317 FE On-Demand Mild P2RY1 47 35 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959317 FE On-Demand Mild EPHX2 48 36 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959318 FE On-Demand Mild P2RY1 47 35 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880959318 FE On-Demand Mild EPHX2 48 36 CC[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880959325 GE On-Demand Anodyne G2YM83_BOTF4 67 35 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1nnn(C)n1 ZINC000880959327 DC On-Demand Anodyne DRD4 18 52 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1nnn(C)n1 ZINC000880959328 DC On-Demand Anodyne DRD4 18 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1nnn(C)n1 ZINC000880959329 DC On-Demand Anodyne DRD4 18 52 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1nnn(C)n1 ZINC000880959330 DC On-Demand Anodyne DRD4 18 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)CN1CCCCS1(=O)=O ZINC000880959337 GD On-Demand Anodyne DRD4 18 45 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)CN1CCCCS1(=O)=O ZINC000880959338 GD On-Demand Anodyne DRD4 18 45 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)CN1CCCCS1(=O)=O ZINC000880959339 GD On-Demand Anodyne DRD4 18 45 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)CN1CCCCS1(=O)=O ZINC000880959340 GD On-Demand Anodyne DRD4 18 45 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880959341 GF On-Demand Anodyne DRD4 35 49 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880959342 GF On-Demand Anodyne DRD4 35 49 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880959343 GF On-Demand Anodyne DRD4 35 49 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc(CN2CCOCC2)o1 ZINC000880959344 GF On-Demand Anodyne DRD4 35 49 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)Nc1cccc2ccccc12 ZINC000880959364 GD On-Demand Anodyne PTPN22 30 46 Cc1ccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)cc1 ZINC000880959367 GF On-Demand Anodyne GPR119 34 44 Cc1ccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)cc1 ZINC000880959367 GF On-Demand Anodyne KDM1A 16 43 Cc1ccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)cc1 ZINC000880959368 GF On-Demand Anodyne GPR119 34 44 Cc1ccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)cc1 ZINC000880959368 GF On-Demand Anodyne KDM1A 16 43 CC[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880959386 GE On-Demand Anodyne G2YM83_BOTF4 67 35 O=C(CN1CCCCS1(=O)=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880959407 FC On-Demand Anodyne CPT1A 50 34 COc1ccc(C)cc1NC(=O)Cn1cc([C@@H](O)c2ccc(C)cc2)nn1 ZINC000880959464 FF On-Demand Anodyne ENPP1 54 30 COc1ccc(C)cc1NC(=O)Cn1cc([C@H](O)c2ccc(C)cc2)nn1 ZINC000880959465 FF On-Demand Anodyne ENPP1 54 30 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc(CC(C)(C)O)nn2)C1 ZINC000880959466 EC On-Demand Anodyne FDFT1 22 40 COC(=O)Cc1cn(CC(=O)Nc2cccc(C)c2)nn1 ZINC000880959470 CC On-Demand Anodyne KCNK3 61 38 COC(=O)Cc1cn(CC(=O)Nc2cccc(C)c2)nn1 ZINC000880959470 CC On-Demand Anodyne KCNK9 50 36 Cc1cccc(NC(=O)Cn2cc(CCCCCCO)nn2)c1 ZINC000880959475 DE On-Demand Anodyne KCNK3 43 35 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCc2ccc(Cl)cc2)nn1 ZINC000880959477 GF On-Demand Anodyne F2 15 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959482 GF On-Demand Anodyne CNR2 24 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959482 GF On-Demand Anodyne EPHX2 48 45 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959483 GF On-Demand Anodyne CNR2 24 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959483 GF On-Demand Anodyne EPHX2 48 45 Nc1ccc(OCc2cn(CC(=O)NC34CC5CC(CC(C5)C3)C4)nn2)cc1 ZINC000880959486 GF On-Demand Clean EPHX2 56 40 Cc1cccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959490 GF On-Demand Anodyne CCKAR 30 41 Cc1cccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959490 GF On-Demand Anodyne CCKBR 51 41 Cc1cccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959490 GF On-Demand Anodyne GPR119 31 46 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959491 GF On-Demand Anodyne CCKAR 30 41 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959491 GF On-Demand Anodyne CCKBR 51 41 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1 ZINC000880959491 GF On-Demand Anodyne GPR119 31 46 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959504 FE On-Demand Anodyne CNR2 26 41 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959504 FE On-Demand Anodyne EPHX2 52 44 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959505 FE On-Demand Anodyne CNR2 26 41 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959505 FE On-Demand Anodyne EPHX2 52 44 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCOC3)nn2)c1 ZINC000880959506 CD On-Demand Anodyne CCKAR 27 40 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCOC3)nn2)c1 ZINC000880959506 CD On-Demand Anodyne CCKBR 49 37 Cc1cccc(NC(=O)Cn2cc([C@H]3CCOC3)nn2)c1 ZINC000880959507 CD On-Demand Anodyne CCKAR 27 40 Cc1cccc(NC(=O)Cn2cc([C@H]3CCOC3)nn2)c1 ZINC000880959507 CD On-Demand Anodyne CCKBR 49 37 Cc1ccc(NC(=O)Cn2cc(CON)nn2)cc1C ZINC000880959508 CC On-Demand Anodyne ENPP1 66 32 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959515 GE On-Demand Anodyne LTA4H 17 46 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959516 GE On-Demand Anodyne LTA4H 17 46 COC(=O)Cc1cn(CC(=O)Nc2ccc(C)c(C)c2)nn1 ZINC000880959521 DD On-Demand Anodyne ENPP1 69 34 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc(C[C@H](O)c3ccccc3)nn2)C1 ZINC000880959533 GD On-Demand Anodyne FDFT1 26 42 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc(C[C@@H](O)c3ccccc3)nn2)C1 ZINC000880959535 GD On-Demand Anodyne FDFT1 26 42 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne PDGFRB 23 45 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne CCR3 15 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne HDAC10 16 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne MTNR1A 26 44 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne MTNR1B 33 44 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne HDAC3 18 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne HDAC6 15 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne CCKBR 18 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne FLT4 24 45 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(OC)c3)nn2)CC1 ZINC000880959537 FE On-Demand Anodyne FPR2 15 43 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)C3CC3)nn2)C1 ZINC000880959539 EC On-Demand Anodyne FDFT1 22 40 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)C3CC3)nn2)C1 ZINC000880959540 EC On-Demand Anodyne FDFT1 22 40 Cc1ccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)cc1 ZINC000880959561 GG On-Demand Anodyne GPR119 41 48 Cc1ccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)cc1 ZINC000880959561 GG On-Demand Anodyne KDM1A 17 46 CN(CC(=O)N1CCN(C(=O)N2CCCCC2)CC1)C1=NS(=O)(=O)c2ccccc21 ZINC000880959564 IC On-Demand Anodyne KCNA3 34 42 C#CCC(CC#C)C(=O)NC[C@@H]1CN(Cc2ccccc2)C[C@@H]1C ZINC000880959577 DF On-Demand Mild DRD4 18 51 C#CCC(CC#C)C(=O)NC[C@H]1CN(Cc2ccccc2)C[C@@H]1C ZINC000880959578 DF On-Demand Mild DRD4 18 51 C#CCC(CC#C)C(=O)NC[C@H]1CN(Cc2ccccc2)C[C@H]1C ZINC000880959579 DF On-Demand Mild DRD4 18 51 C#CCC(CC#C)C(=O)NC[C@@H]1CN(Cc2ccccc2)C[C@H]1C ZINC000880959580 DF On-Demand Mild DRD4 18 51 COC(=O)Cc1cn(CC(=O)Nc2ccc(Br)c(C)c2)nn1 ZINC000880959581 FD On-Demand Anodyne IMDH_CRYPV 17 43 Cc1ccc(NC(=O)Cn2cc(CN(C)C(=O)OC(C)(C)C)nn2)cc1 ZINC000880959583 FF On-Demand Anodyne KDM1A 15 42 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccccc1Oc1ccccc1 ZINC000880959587 GH On-Demand Anodyne CPT1A 50 35 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccccc1Oc1ccccc1 ZINC000880959588 GH On-Demand Anodyne CPT1A 50 35 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@@H]1C ZINC000880959597 EE On-Demand Anodyne DRD2 15 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@@H]1C ZINC000880959597 EE On-Demand Anodyne DRD4 39 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@@H]1C ZINC000880959597 EE On-Demand Anodyne ACHE 31 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@@H]1C ZINC000880959597 EE On-Demand Anodyne SIGMAR1 38 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@@H]1C ZINC000880959597 EE On-Demand Anodyne CCR5 19 40 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCN(C)[C@H]1C ZINC000880959598 EE On-Demand Anodyne DRD2 15 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCN(C)[C@H]1C ZINC000880959598 EE On-Demand Anodyne DRD4 39 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCN(C)[C@H]1C ZINC000880959598 EE On-Demand Anodyne ACHE 31 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCN(C)[C@H]1C ZINC000880959598 EE On-Demand Anodyne SIGMAR1 38 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCN(C)[C@H]1C ZINC000880959598 EE On-Demand Anodyne CCR5 19 40 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@H]1C ZINC000880959599 EE On-Demand Anodyne DRD2 15 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@H]1C ZINC000880959599 EE On-Demand Anodyne DRD4 39 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@H]1C ZINC000880959599 EE On-Demand Anodyne ACHE 31 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@H]1C ZINC000880959599 EE On-Demand Anodyne SIGMAR1 38 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCN(C)[C@H]1C ZINC000880959599 EE On-Demand Anodyne CCR5 19 40 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc2ccccc12 ZINC000880959617 GE On-Demand Anodyne PRKDC 70 37 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc2ccccc12 ZINC000880959617 GE On-Demand Anodyne ADCY5 17 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc2ccccc12 ZINC000880959617 GE On-Demand Anodyne PTGDS 38 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc2ccccc12 ZINC000880959617 GE On-Demand Anodyne PTPN22 40 44 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc3ccccc23)nn1 ZINC000880959621 ED On-Demand Anodyne PTPN22 20 43 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1cccc2ccccc12 ZINC000880959631 FG On-Demand Anodyne PTPN22 24 46 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccccc1Cl ZINC000880959635 ED On-Demand Anodyne EPHB3 50 36 CC[C@@](C)(O)c1cn(CC(=O)Nc2cccc3ccccc23)nn1 ZINC000880959648 DF On-Demand Anodyne PTPN22 29 45 Cc1cccc(NC(=O)Cn2cc(CN[C@H]3CCCc4ccccc43)nn2)c1 ZINC000880959655 GG On-Demand Anodyne CCKAR 23 40 Cc1cccc(NC(=O)Cn2cc(CN[C@H]3CCCc4ccccc43)nn2)c1 ZINC000880959655 GG On-Demand Anodyne CCKBR 40 38 Cc1cccc(NC(=O)Cn2cc(CN[C@@H]3CCCc4ccccc43)nn2)c1 ZINC000880959656 GG On-Demand Anodyne CCKAR 23 40 Cc1cccc(NC(=O)Cn2cc(CN[C@@H]3CCCc4ccccc43)nn2)c1 ZINC000880959656 GG On-Demand Anodyne CCKBR 40 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959661 GF On-Demand Anodyne TSHR 42 32 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959661 GF On-Demand Anodyne LTA4H 39 49 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959661 GF On-Demand Anodyne ADAM17 18 45 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959662 GF On-Demand Anodyne TSHR 42 32 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959662 GF On-Demand Anodyne LTA4H 39 49 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959662 GF On-Demand Anodyne ADAM17 18 45 CC[C@H](O)c1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880959663 DD On-Demand Anodyne EPHX2 57 45 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)c3ccccc3)nn2)C1 ZINC000880959674 FD On-Demand Anodyne FDFT1 32 47 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)C1 ZINC000880959676 FD On-Demand Anodyne FDFT1 32 47 Cc1cccc(NC(=O)Cn2cc(C3CC4(C3)OCCO4)nn2)c1 ZINC000880959678 ED On-Demand Anodyne CCKAR 27 40 Cc1cccc(NC(=O)Cn2cc(C3CC4(C3)OCCO4)nn2)c1 ZINC000880959678 ED On-Demand Anodyne CCKBR 45 37 Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1C ZINC000880959679 FD On-Demand Anodyne PRKDC 44 34 Cc1ccc(NC(=O)Cn2cc(C(C)(C)NC(=O)OC(C)(C)C)nn2)cc1C ZINC000880959680 GG On-Demand Anodyne ENPP1 54 32 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(Cl)c(Cl)c1 ZINC000880959693 GE On-Demand Anodyne EPHX2 23 42 O=C(Cn1cc(C2(O)CCC2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959697 ED On-Demand Anodyne EPHX2 44 37 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)c3ccc(F)cc3)nn2)C1 ZINC000880959711 GD On-Demand Anodyne FDFT1 25 44 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)c3ccc(F)cc3)nn2)C1 ZINC000880959713 GD On-Demand Anodyne FDFT1 25 44 CC(C)(C)OC(=O)NCc1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880959716 GE On-Demand Anodyne EPHX2 60 42 Cc1cccc(NC(=O)Cn2cc(CC3(O)CCOCC3)nn2)c1 ZINC000880959717 ED On-Demand Anodyne KCNK3 42 34 Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880959722 ED On-Demand Anodyne EGFR 15 41 Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880959722 ED On-Demand Anodyne CASR 37 43 Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880959722 ED On-Demand Anodyne EPHX2 25 44 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(C)c(C)c2)nn1 ZINC000880959724 DD On-Demand Anodyne ENPP1 61 32 COc1ccc(C)cc1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880959740 GF On-Demand Anodyne MMP8 24 41 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccccc3Cl)nn2)CC1 ZINC000880959764 GD On-Demand Anodyne EPHB3 46 34 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(F)c1 ZINC000880959772 FD On-Demand Anodyne CHRNA7 18 45 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)c(F)c1 ZINC000880959772 FD On-Demand Anodyne EPHX2 24 50 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccccc1Cl ZINC000880959773 DD On-Demand Anodyne EPHB3 56 38 N#Cc1ccc(Cl)cc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880959774 GD On-Demand Mild MAP3K8 38 42 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1cccc2ccccc12 ZINC000880959786 DF On-Demand Anodyne PTPN22 36 46 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1cccc2ccccc12 ZINC000880959787 DF On-Demand Anodyne PTPN22 36 46 Cc1ccc(NC(=O)Cn2cc(CNC(=O)OC(C)(C)C)nn2)cc1 ZINC000880959789 EE On-Demand Anodyne KDM1A 16 43 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959801 FE On-Demand Anodyne DRD4 18 43 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959801 FE On-Demand Anodyne SIGMAR1 21 47 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959801 FE On-Demand Anodyne PDE8B 47 33 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959801 FE On-Demand Anodyne CACNA1G 38 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959802 FE On-Demand Anodyne DRD4 18 43 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959802 FE On-Demand Anodyne SIGMAR1 21 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959802 FE On-Demand Anodyne PDE8B 47 33 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959802 FE On-Demand Anodyne CACNA1G 38 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959803 FE On-Demand Anodyne DRD4 18 43 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959803 FE On-Demand Anodyne SIGMAR1 21 47 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959803 FE On-Demand Anodyne PDE8B 47 33 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1CCc2nncn2CC1 ZINC000880959803 FE On-Demand Anodyne CACNA1G 38 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959804 FE On-Demand Anodyne DRD4 18 43 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959804 FE On-Demand Anodyne SIGMAR1 21 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959804 FE On-Demand Anodyne PDE8B 47 33 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@@H]1CCc2nncn2CC1 ZINC000880959804 FE On-Demand Anodyne CACNA1G 38 41 COC(OC)c1ccc(C(=O)NC[C@@H]2CN(Cc3ccccc3)C[C@@H]2C)o1 ZINC000880959814 FG On-Demand Anodyne DRD4 26 55 COC(OC)c1ccc(C(=O)NC[C@@H]2CN(Cc3ccccc3)C[C@@H]2C)o1 ZINC000880959814 FG On-Demand Anodyne NOD2 40 36 COC(OC)c1ccc(C(=O)NC[C@@H]2CN(Cc3ccccc3)C[C@H]2C)o1 ZINC000880959815 FG On-Demand Anodyne DRD4 26 55 COC(OC)c1ccc(C(=O)NC[C@@H]2CN(Cc3ccccc3)C[C@H]2C)o1 ZINC000880959815 FG On-Demand Anodyne NOD2 40 36 COC(OC)c1ccc(C(=O)NC[C@H]2CN(Cc3ccccc3)C[C@@H]2C)o1 ZINC000880959816 FG On-Demand Anodyne DRD4 26 55 COC(OC)c1ccc(C(=O)NC[C@H]2CN(Cc3ccccc3)C[C@@H]2C)o1 ZINC000880959816 FG On-Demand Anodyne NOD2 40 36 COC(OC)c1ccc(C(=O)NC[C@H]2CN(Cc3ccccc3)C[C@H]2C)o1 ZINC000880959817 FG On-Demand Anodyne DRD4 26 55 COC(OC)c1ccc(C(=O)NC[C@H]2CN(Cc3ccccc3)C[C@H]2C)o1 ZINC000880959817 FG On-Demand Anodyne NOD2 40 36 Cc1ccc(NC(=O)Cn2cc([C@@H]3CCCN3C(=O)OC(C)(C)C)nn2)cc1 ZINC000880959823 GG On-Demand Anodyne KDM1A 15 41 Cc1ccc(NC(=O)Cn2cc([C@H]3CCCN3C(=O)OC(C)(C)C)nn2)cc1 ZINC000880959824 GG On-Demand Anodyne KDM1A 15 41 C[C@H](N)c1cn(CC(=O)Nc2ccc(C(C)(C)C)cc2)nn1 ZINC000880959826 DE On-Demand Anodyne DOT1L 40 31 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccccc1Cl ZINC000880959843 DE On-Demand Anodyne EPHB3 41 34 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccccc1Cl ZINC000880959844 DE On-Demand Anodyne EPHB3 41 34 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccccc1Cl ZINC000880959850 EF On-Demand Anodyne EPHB3 46 33 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccccc1Cl ZINC000880959851 EF On-Demand Anodyne EPHB3 46 33 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959859 FF On-Demand Anodyne TSHR 49 33 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959859 FF On-Demand Anodyne LTA4H 39 51 COc1ccc(C)cc1NC(=O)Cn1cc(CCNC(C)=O)nn1 ZINC000880959861 EC On-Demand Anodyne NQO2 59 37 COc1ccc(C)cc1NC(=O)Cn1cc(CCNC(C)=O)nn1 ZINC000880959861 EC On-Demand Anodyne MTNR1B 42 39 Cc1cccc(NC(=O)Cn2cc(CN3CCOC3=O)nn2)c1 ZINC000880959870 DD On-Demand Anodyne KCNK3 49 36 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959884 GE On-Demand Anodyne ADRB1 29 40 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959884 GE On-Demand Anodyne TSHR 49 34 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959884 GE On-Demand Anodyne ADRB3 23 40 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880959884 GE On-Demand Anodyne LTA4H 36 48 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959888 GF On-Demand Anodyne CNR2 23 40 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959888 GF On-Demand Anodyne EPHX2 44 42 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959889 GF On-Demand Anodyne CNR2 23 40 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880959889 GF On-Demand Anodyne EPHX2 44 42 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959895 GH On-Demand Anodyne TSHR 55 33 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959895 GH On-Demand Anodyne LTA4H 33 46 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959895 GH On-Demand Anodyne ADAM17 21 46 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959895 GH On-Demand Anodyne CPT1A 42 37 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959896 GH On-Demand Anodyne TSHR 55 33 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959896 GH On-Demand Anodyne LTA4H 33 46 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959896 GH On-Demand Anodyne ADAM17 21 46 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880959896 GH On-Demand Anodyne CPT1A 42 37 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc(-c3cccnc3Cl)nn2)C1 ZINC000880959914 GD On-Demand Anodyne FDFT1 23 40 Cc1cccc(NC(=O)Cn2cc([C@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1C ZINC000880959919 GG On-Demand Anodyne CCR8 41 33 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCN(C(=O)OC(C)(C)C)C3)nn2)c1C ZINC000880959920 GG On-Demand Anodyne CCR8 41 33 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne PIK3CA 42 45 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne CHRNA7 15 52 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne PRNP 39 46 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne JAK2 15 45 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne MAPKAPK5 40 35 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne MTOR 66 45 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne PIK3CG 30 45 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne STAT6 76 39 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne DGAT1 15 40 O=C(Cn1cc(-c2cccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880959971 FD On-Demand Anodyne NAMPT 26 44 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc4ccccc34)nn2)CC1 ZINC000880959986 GH On-Demand Anodyne PTPN22 21 43 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)Nc1ccccc1Cl ZINC000880959996 GC On-Demand Anodyne EPHB3 42 34 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960000 GG On-Demand Anodyne DRD4 29 50 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960000 GG On-Demand Anodyne ACHE 22 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960000 GG On-Demand Anodyne DRD3 15 50 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960001 GG On-Demand Anodyne DRD4 29 50 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960001 GG On-Demand Anodyne ACHE 22 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960001 GG On-Demand Anodyne DRD3 15 50 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960002 GG On-Demand Anodyne DRD4 29 50 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960002 GG On-Demand Anodyne ACHE 22 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@@H]2CCC(=O)N2)cc1 ZINC000880960002 GG On-Demand Anodyne DRD3 15 50 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960003 GG On-Demand Anodyne DRD4 29 50 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960003 GG On-Demand Anodyne ACHE 22 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)c1ccc([C@H]2CCC(=O)N2)cc1 ZINC000880960003 GG On-Demand Anodyne DRD3 15 50 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne GHRHR 46 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne P2RY12 122 36 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne CTSK 23 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne CTSL 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960029 GD On-Demand Anodyne FPR1 48 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne GHRHR 46 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne P2RY12 122 36 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne PAPA1_CARPA 35 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne CTSK 23 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne CTSL 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880960030 GD On-Demand Anodyne FPR1 48 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccccc1Cl ZINC000880960034 DE On-Demand Anodyne EPHB3 53 33 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccccc1Cl ZINC000880960035 DE On-Demand Anodyne EPHB3 53 33 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1cccc2ccccc12 ZINC000880960050 EG On-Demand Anodyne PTPN22 29 45 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1cccc2ccccc12 ZINC000880960051 EG On-Demand Anodyne PTPN22 29 45 Cc1cccc(NC(=O)Cn2cc(CC(C)(C)O)nn2)c1 ZINC000880960106 CD On-Demand Anodyne KCNK3 53 36 Cc1cccc(NC(=O)Cn2cc(CC(C)(C)O)nn2)c1 ZINC000880960106 CD On-Demand Anodyne KCNK9 41 36 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960107 FG On-Demand Anodyne EPHX2 52 45 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960107 FG On-Demand Anodyne TRAR 26 42 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960108 FG On-Demand Anodyne EPHX2 52 45 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960108 FG On-Demand Anodyne TRAR 26 42 CC(C)c1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880960126 FE On-Demand Anodyne CHRNA7 16 45 CC(C)c1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880960126 FE On-Demand Anodyne EPHX2 20 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccccc1Cl ZINC000880960135 FD On-Demand Anodyne EPHB3 53 38 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@](C)(O)CC)nn2)C1 ZINC000880960145 EC On-Demand Anodyne FDFT1 22 40 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@](C)(O)CC)nn2)C1 ZINC000880960146 EC On-Demand Anodyne FDFT1 22 40 O=C(Cn1cc([C@H](O)C2CC2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880960150 ED On-Demand Anodyne EPHX2 46 42 O=C(Cn1cc([C@@H](O)C2CC2)nn1)NC12CC3CC(CC(C3)C1)C2 ZINC000880960151 ED On-Demand Anodyne EPHX2 46 42 Cc1cccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)c1 ZINC000880960157 GG On-Demand Anodyne CCKAR 32 43 Cc1cccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)c1 ZINC000880960157 GG On-Demand Anodyne CCKBR 54 43 Cc1cccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)c1 ZINC000880960157 GG On-Demand Anodyne GPR119 37 49 Cc1cccc(NC(=O)Cn2cc(C3CCN(C(=O)OC(C)(C)C)CC3)nn2)c1 ZINC000880960157 GG On-Demand Anodyne KDM1A 17 40 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960166 GE On-Demand Anodyne DRD4 18 47 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960166 GE On-Demand Anodyne SIGMAR1 21 46 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960166 GE On-Demand Anodyne PDE8B 52 35 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960168 GE On-Demand Anodyne DRD4 18 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960168 GE On-Demand Anodyne SIGMAR1 21 46 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960168 GE On-Demand Anodyne PDE8B 52 35 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960169 GE On-Demand Anodyne DRD4 18 47 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960169 GE On-Demand Anodyne SIGMAR1 21 46 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960169 GE On-Demand Anodyne PDE8B 52 35 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960171 GE On-Demand Anodyne DRD4 18 47 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960171 GE On-Demand Anodyne SIGMAR1 21 46 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)C1CCC(S(C)(=O)=O)CC1 ZINC000880960171 GE On-Demand Anodyne PDE8B 52 35 Cc1cccc(NC(=O)Cn2cc(CNC(=O)C(F)(F)F)nn2)c1 ZINC000880960182 ED On-Demand Anodyne KCNK3 45 35 Cc1ccc(NC(=O)Cn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880960186 FF On-Demand Anodyne MMP13 15 45 Cc1ccc(NC(=O)Cn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880960186 FF On-Demand Anodyne MMP8 25 44 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)CC)nn2)C1 ZINC000880960204 DC On-Demand Anodyne FDFT1 23 42 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)CC)nn2)C1 ZINC000880960206 DC On-Demand Anodyne FDFT1 23 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(C)c2)nn1 ZINC000880960207 DC On-Demand Anodyne KCNK3 47 35 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1cccc2ccccc12 ZINC000880960219 FE On-Demand Anodyne PTPN22 30 47 Cc1cccc(NC(=O)Cn2cc(C3(O)CCCCC3)nn2)c1 ZINC000880960234 DE On-Demand Anodyne KCNK3 40 34 O=C(Cn1cc([C@@H](O)C2CC2)nn1)NCc1ccc(Cl)cc1 ZINC000880960235 DD On-Demand Anodyne UL54 56 32 O=C(Cn1cc([C@H](O)C2CC2)nn1)NCc1ccc(Cl)cc1 ZINC000880960236 DD On-Demand Anodyne UL54 56 32 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne PDGFRB 35 49 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne MTNR1A 33 45 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne MTNR1B 35 47 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne FLT4 30 49 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne FLT3 15 48 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne FPR2 15 43 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne TAAR1 31 42 COC(=O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960239 DC On-Demand Anodyne ENPP1 50 32 Cc1cccc(NC(=O)Cn2cc(CN3CCS(=O)(=O)CC3)nn2)c1 ZINC000880960242 FC On-Demand Anodyne KCNK3 45 34 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1cccc2ccccc12 ZINC000880960246 FF On-Demand Anodyne PTPN22 29 45 NOCc1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880960252 DC On-Demand Anodyne EPHX2 65 40 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccccc1Cl ZINC000880960274 EF On-Demand Anodyne EPHB3 56 37 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1cccc2ccccc12 ZINC000880960275 ED On-Demand Anodyne PTPN22 23 44 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1cccc2ccccc12 ZINC000880960276 ED On-Demand Anodyne PTPN22 23 44 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960301 GE On-Demand Anodyne DRD4 17 47 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960301 GE On-Demand Anodyne SIGMAR1 22 44 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960301 GE On-Demand Anodyne PDE8B 56 36 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960302 GE On-Demand Anodyne DRD4 17 47 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960302 GE On-Demand Anodyne SIGMAR1 22 44 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960302 GE On-Demand Anodyne PDE8B 56 36 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc(C(C)(C)O)nn2)C1 ZINC000880960305 DC On-Demand Anodyne FDFT1 24 42 Cc1cccc(NC(=O)Cn2cc(COc3ccccc3[C@H](C)O)nn2)c1 ZINC000880960307 FF On-Demand Anodyne KCNK3 50 37 Cc1cccc(NC(=O)Cn2cc(COc3ccccc3[C@H](C)O)nn2)c1 ZINC000880960307 FF On-Demand Anodyne KCNK9 54 37 Cc1cccc(NC(=O)Cn2cc(COc3ccccc3[C@@H](C)O)nn2)c1 ZINC000880960308 FF On-Demand Anodyne KCNK3 50 37 Cc1cccc(NC(=O)Cn2cc(COc3ccccc3[C@@H](C)O)nn2)c1 ZINC000880960308 FF On-Demand Anodyne KCNK9 54 37 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880960309 GF On-Demand Anodyne LTA4H 30 47 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880960310 GF On-Demand Anodyne LTA4H 30 47 CN(Cc1cn(CC(=O)NCc2ccc(Cl)cc2)nn1)C(=O)OC(C)(C)C ZINC000880960311 GF On-Demand Anodyne UL54 50 31 Cc1cccc(NC(=O)Cn2cc(CON)nn2)c1 ZINC000880960312 CC On-Demand Anodyne KCNK3 51 36 Cc1cccc(NC(=O)Cn2cc(CON)nn2)c1 ZINC000880960312 CC On-Demand Anodyne KCNK9 41 36 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1ccc(Cl)cc1 ZINC000880960313 GD On-Demand Anodyne CCR4 17 40 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1ccc(Cl)cc1 ZINC000880960313 GD On-Demand Anodyne UL54 26 45 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1ccc(Cl)cc1 ZINC000880960313 GD On-Demand Anodyne DPOL_VZVD 44 45 Cc1ccc(NC(=O)Cn2cc(COc3ccccc3[C@H](C)O)nn2)cc1C ZINC000880960315 GG On-Demand Anodyne ENPP1 40 31 Cc1ccc(NC(=O)Cn2cc(COc3ccccc3[C@@H](C)O)nn2)cc1C ZINC000880960316 GG On-Demand Anodyne ENPP1 40 31 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960327 DD On-Demand Mild PDGFRB 21 46 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960327 DD On-Demand Mild MTNR1A 18 42 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960327 DD On-Demand Mild MTNR1B 24 43 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960327 DD On-Demand Mild FLT4 24 46 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960327 DD On-Demand Mild ENPP1 50 32 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960328 DD On-Demand Mild PDGFRB 21 46 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960328 DD On-Demand Mild MTNR1A 18 42 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960328 DD On-Demand Mild MTNR1B 24 43 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960328 DD On-Demand Mild FLT4 24 46 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960328 DD On-Demand Mild ENPP1 50 32 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccc(C)c3)nn2)CC1 ZINC000880960337 FC On-Demand Anodyne KCNK3 48 35 CC[C@@](C)(O)c1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880960339 ED On-Demand Anodyne EPHX2 58 40 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960351 GE On-Demand Anodyne DRD4 17 47 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960351 GE On-Demand Anodyne SIGMAR1 22 44 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960351 GE On-Demand Anodyne PDE8B 56 36 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960352 FE On-Demand Anodyne EPHX2 54 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960352 FE On-Demand Anodyne MCHR1 17 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960352 FE On-Demand Anodyne TRAR 38 45 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960353 GE On-Demand Anodyne DRD4 17 47 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960353 GE On-Demand Anodyne SIGMAR1 22 44 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880960353 GE On-Demand Anodyne PDE8B 56 36 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960354 FE On-Demand Anodyne EPHX2 54 41 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960354 FE On-Demand Anodyne MCHR1 17 41 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960354 FE On-Demand Anodyne TRAR 38 45 O=C(Cn1cc(CCCCCCO)nn1)NCc1ccc(Cl)cc1 ZINC000880960375 FE On-Demand Anodyne UL54 29 42 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccc(Cl)cc3)nn2)CC1 ZINC000880960389 GC On-Demand Anodyne DRD4 21 41 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccc(Cl)cc3)nn2)CC1 ZINC000880960389 GC On-Demand Anodyne LSS 15 40 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccc(Cl)cc3)nn2)CC1 ZINC000880960389 GC On-Demand Anodyne FAAH 17 42 COc1ccc(C)cc1NC(=O)Cn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880960446 GC On-Demand Anodyne SLC9A1 57 32 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccccc2Cl)nn1 ZINC000880960450 DD On-Demand Anodyne EPHB3 50 35 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccc4ccccc34)nn2)CC1 ZINC000880960480 GD On-Demand Anodyne PTPN22 39 46 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc2ccccc12 ZINC000880960491 FG On-Demand Anodyne PTPN22 29 45 Cc1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1Cl ZINC000880960493 GE On-Demand Anodyne EPHX2 24 40 O=C(Cn1cc([C@]2(O)CCOC2)nn1)Nc1ccccc1Cl ZINC000880960525 DD On-Demand Anodyne EPHB3 49 36 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)Nc1ccccc1Cl ZINC000880960526 DD On-Demand Anodyne EPHB3 49 36 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960542 DE On-Demand Anodyne DRD4 26 52 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960542 DE On-Demand Anodyne SIGMAR1 36 41 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960542 DE On-Demand Anodyne TIMP3 50 32 C[C@@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960542 DE On-Demand Anodyne MBTPS1 40 32 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960543 DE On-Demand Anodyne DRD4 26 52 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960543 DE On-Demand Anodyne SIGMAR1 36 41 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960543 DE On-Demand Anodyne TIMP3 50 32 C[C@H]1CN(Cc2ccccc2)C[C@H]1CNC(=O)COC1CC1 ZINC000880960543 DE On-Demand Anodyne MBTPS1 40 32 Cc1ccc(NC(=O)Cn2cc(COc3ccc([C@H](C)O)cc3)nn2)cc1C ZINC000880960544 GG On-Demand Anodyne ENPP1 40 32 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960545 DE On-Demand Anodyne DRD4 26 52 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960545 DE On-Demand Anodyne SIGMAR1 36 41 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960545 DE On-Demand Anodyne TIMP3 50 32 C[C@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960545 DE On-Demand Anodyne MBTPS1 40 32 Cc1ccc(NC(=O)Cn2cc(COc3ccc([C@@H](C)O)cc3)nn2)cc1C ZINC000880960546 GG On-Demand Anodyne ENPP1 40 32 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960547 DE On-Demand Anodyne DRD4 26 52 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960547 DE On-Demand Anodyne SIGMAR1 36 41 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960547 DE On-Demand Anodyne TIMP3 50 32 C[C@@H]1CN(Cc2ccccc2)C[C@@H]1CNC(=O)COC1CC1 ZINC000880960547 DE On-Demand Anodyne MBTPS1 40 32 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccccc1Cl ZINC000880960549 EF On-Demand Anodyne EPHB3 55 34 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1cccc2ccccc12 ZINC000880960559 DE On-Demand Anodyne PTPN22 43 49 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)c3ccc(C)cc3)nn2)C1 ZINC000880960576 GD On-Demand Anodyne FDFT1 25 43 O=C(Cn1cc(CN2CCOC2=O)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960618 GD On-Demand Anodyne EPHX2 49 39 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(C)c3)nn2)CC1 ZINC000880960634 FF On-Demand Anodyne HDAC2 15 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(C)c3)nn2)CC1 ZINC000880960634 FF On-Demand Anodyne HDAC3 24 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(C)c3)nn2)CC1 ZINC000880960634 FF On-Demand Anodyne HDAC6 20 41 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(C)c3)nn2)CC1 ZINC000880960634 FF On-Demand Anodyne CCKBR 51 36 COC(=O)C1CCC(c2cn(CC(=O)Nc3ccc(C)c(C)c3)nn2)CC1 ZINC000880960649 FF On-Demand Anodyne ENPP1 55 33 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCN3C(=O)OC(C)(C)C)nn2)c1 ZINC000880960650 GG On-Demand Anodyne CCKAR 31 41 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCN3C(=O)OC(C)(C)C)nn2)c1 ZINC000880960650 GG On-Demand Anodyne CCKBR 49 41 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCN3C(=O)OC(C)(C)C)nn2)c1 ZINC000880960651 GG On-Demand Anodyne CCKAR 31 41 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCN3C(=O)OC(C)(C)C)nn2)c1 ZINC000880960651 GG On-Demand Anodyne CCKBR 49 41 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960652 GE On-Demand Anodyne EPHX2 54 38 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1ccc(OC(F)(F)F)cc1 ZINC000880960652 GE On-Demand Anodyne TRAR 26 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960655 DC On-Demand Anodyne PDGFRB 24 47 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960655 DC On-Demand Anodyne MTNR1A 22 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960655 DC On-Demand Anodyne MTNR1B 26 44 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(OC)c2)nn1 ZINC000880960655 DC On-Demand Anodyne FLT4 25 47 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880960658 GG On-Demand Anodyne TSHR 42 33 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880960658 GG On-Demand Anodyne LTA4H 36 50 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880960658 GG On-Demand Anodyne ADORA2B 17 40 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OCc3ccccc3)cc2)nn1 ZINC000880960658 GG On-Demand Anodyne S1PR4 22 40 C=C[C@](C)(O)c1cn(CC(=O)Nc2cccc(C)c2)nn1 ZINC000880960670 CD On-Demand Mild KCNK3 45 34 C=C[C@@](C)(O)c1cn(CC(=O)Nc2cccc(C)c2)nn1 ZINC000880960671 CD On-Demand Mild KCNK3 45 34 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880960673 GF On-Demand Anodyne CNR2 20 40 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC23CC4CC(CC(C4)C2)C3)nn1 ZINC000880960673 GF On-Demand Anodyne EPHX2 48 43 Cc1cccc(NC(=O)Cn2cc(C3(O)CCC3)nn2)c1 ZINC000880960692 CD On-Demand Anodyne KCNK3 43 35 Cc1cccc(NC(=O)Cn2cc([C@@H](O)C3CC3)nn2)c1 ZINC000880960702 CD On-Demand Anodyne KCNK3 51 36 Cc1cccc(NC(=O)Cn2cc([C@@H](O)C3CC3)nn2)c1 ZINC000880960702 CD On-Demand Anodyne KCNK9 41 36 Cc1cccc(NC(=O)Cn2cc([C@H](O)C3CC3)nn2)c1 ZINC000880960703 CD On-Demand Anodyne KCNK3 51 36 Cc1cccc(NC(=O)Cn2cc([C@H](O)C3CC3)nn2)c1 ZINC000880960703 CD On-Demand Anodyne KCNK9 41 36 Cc1cccc(NC(=O)Cn2cc([C@@](C)(O)Cc3ccccc3)nn2)c1 ZINC000880960714 FF On-Demand Anodyne CCKBR 41 35 Cc1cccc(NC(=O)Cn2cc([C@@](C)(O)Cc3ccccc3)nn2)c1 ZINC000880960714 FF On-Demand Anodyne KCNK3 47 36 Cc1cccc(NC(=O)Cn2cc([C@](C)(O)Cc3ccccc3)nn2)c1 ZINC000880960715 FF On-Demand Anodyne CCKBR 41 35 Cc1cccc(NC(=O)Cn2cc([C@](C)(O)Cc3ccccc3)nn2)c1 ZINC000880960715 FF On-Demand Anodyne KCNK3 47 36 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880960722 DE On-Demand Anodyne CCKAR 30 41 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880960722 DE On-Demand Anodyne HDAC2 15 42 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880960722 DE On-Demand Anodyne HDAC3 25 42 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880960722 DE On-Demand Anodyne HDAC6 19 42 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCC(=O)C3)nn2)c1 ZINC000880960722 DE On-Demand Anodyne CCKBR 56 39 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880960723 DE On-Demand Anodyne CCKAR 30 41 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880960723 DE On-Demand Anodyne HDAC2 15 42 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880960723 DE On-Demand Anodyne HDAC3 25 42 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880960723 DE On-Demand Anodyne HDAC6 19 42 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCC(=O)C3)nn2)c1 ZINC000880960723 DE On-Demand Anodyne CCKBR 56 39 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)C1 ZINC000880960728 GD On-Demand Anodyne FDFT1 25 42 CCOC(=O)[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)C1 ZINC000880960730 GD On-Demand Anodyne FDFT1 25 42 COC[C@@H](O)Cc1cn(CC(=O)NCc2ccc(Cl)cc2)nn1 ZINC000880960734 EC On-Demand Anodyne UL54 50 32 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880960738 FD On-Demand Anodyne P2RY1 47 35 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)nn1 ZINC000880960738 FD On-Demand Anodyne EPHX2 49 37 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880960739 DE On-Demand Anodyne CCKBR 47 36 Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880960739 DE On-Demand Anodyne KCNK3 45 34 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880960740 DE On-Demand Anodyne CCKBR 47 36 Cc1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880960740 DE On-Demand Anodyne KCNK3 45 34 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880960742 GF On-Demand Anodyne LTA4H 32 50 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(OCc2ccccc2)cc1 ZINC000880960742 GF On-Demand Anodyne ADAM17 21 43 C=C[C@@](C)(O)c1cn(CC(=O)N2CCC[C@H](C(=O)OCC)C2)nn1 ZINC000880960743 EC On-Demand Mild FDFT1 18 40 C=C[C@](C)(O)c1cn(CC(=O)N2CCC[C@H](C(=O)OCC)C2)nn1 ZINC000880960744 EC On-Demand Mild FDFT1 18 40 C=C[C@@](C)(O)c1cn(CC(=O)N2CCC[C@@H](C(=O)OCC)C2)nn1 ZINC000880960745 EC On-Demand Mild FDFT1 18 40 C=C[C@](C)(O)c1cn(CC(=O)N2CCC[C@@H](C(=O)OCC)C2)nn1 ZINC000880960746 EC On-Demand Mild FDFT1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](NC2CCOCC2)C1 ZINC000880960760 FF On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](NC2CCOCC2)C1 ZINC000880960761 FF On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CF)C1 ZINC000880960762 CF On-Demand Anodyne RBP4 76 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CF)C1 ZINC000880960763 CF On-Demand Anodyne RBP4 76 45 Cn1cc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960767 FD On-Demand Anodyne MTOR 80 39 Cn1cc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960767 FD On-Demand Anodyne MAPK10 16 42 Cn1cc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960767 FD On-Demand Anodyne STAT6 60 35 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960771 FD On-Demand Anodyne MTOR 78 39 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960771 FD On-Demand Anodyne STAT6 55 34 C[C@@H]1CC[C@H](O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880960775 DE On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]2CCCC[C@@H]21 ZINC000880960778 DH On-Demand Anodyne EPHX2 15 44 CCNCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960784 EC On-Demand Anodyne MTOR 57 40 CCNCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960784 EC On-Demand Anodyne STAT6 56 35 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne PIK3CA 31 40 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne HDAC6 18 41 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne MTOR 55 40 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne PIK3CG 29 40 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne PIK3CB 17 43 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne STAT6 74 43 O=C(Cn1cc(-c2cc(F)cc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960785 GF On-Demand Anodyne DGAT1 15 42 CCC(C)(C)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960791 FE On-Demand Anodyne MTOR 63 38 CCC(C)(C)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960791 FE On-Demand Anodyne STAT6 56 34 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960793 FD On-Demand Anodyne MTOR 72 38 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960793 FD On-Demand Anodyne STAT6 53 32 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960794 FD On-Demand Anodyne MTOR 72 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960794 FD On-Demand Anodyne STAT6 53 32 O=C(Cn1cc([C@@H]2CCCC[C@@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960799 GD On-Demand Anodyne MTOR 56 36 O=C(Cn1cc([C@@H]2CCCC[C@@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960799 GD On-Demand Anodyne STAT6 53 34 O=C(Cn1cc([C@H]2CCCC[C@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960800 GD On-Demand Anodyne MTOR 56 36 O=C(Cn1cc([C@H]2CCCC[C@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960800 GD On-Demand Anodyne STAT6 53 34 O=C(Cn1cc([C@H]2CCCC[C@@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960801 GD On-Demand Anodyne MTOR 56 36 O=C(Cn1cc([C@H]2CCCC[C@@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960801 GD On-Demand Anodyne STAT6 53 34 O=C(Cn1cc([C@@H]2CCCC[C@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960802 GD On-Demand Anodyne MTOR 56 36 O=C(Cn1cc([C@@H]2CCCC[C@H]2O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960802 GD On-Demand Anodyne STAT6 53 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2nccs2)C1 ZINC000880960804 EH On-Demand Anodyne RBP4 80 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2nccs2)C1 ZINC000880960805 EH On-Demand Anodyne RBP4 80 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CF)C1 ZINC000880960806 DG On-Demand Anodyne RBP4 69 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CF)C1 ZINC000880960807 DG On-Demand Anodyne RBP4 69 44 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(C(F)(F)F)nc1 ZINC000880960811 GI On-Demand Anodyne TRPV1 19 55 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)cc1Cl ZINC000880960812 GD On-Demand Anodyne EPHX2 16 40 O=C(/C=C\c1cccnc1)N1CCN(C(=O)N2CCCCC2)CC1 ZINC000880960816 ED On-Demand Anodyne C3AR1 33 59 C#CC1(F)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880960819 CE On-Demand Mild RBP4 58 42 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960822 FD On-Demand Mild MTOR 47 36 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960822 FD On-Demand Mild STAT6 61 35 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960823 FD On-Demand Mild MTOR 47 36 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960823 FD On-Demand Mild STAT6 61 35 O=C(Cn1cc(-c2cc(F)ccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960824 GF On-Demand Anodyne MTOR 19 40 O=C(Cn1cc(-c2cc(F)ccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960824 GF On-Demand Anodyne PIK3CB 15 46 O=C(Cn1cc(-c2cc(F)ccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960824 GF On-Demand Anodyne STAT6 69 42 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne JAK2 15 48 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne HDAC10 25 42 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne HDAC3 29 42 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne HDAC6 23 42 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne MTOR 54 37 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne FLT3 15 40 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne STAT6 58 35 CNc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960825 GE On-Demand Anodyne DGAT1 17 40 CC[C@H](O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960831 ED On-Demand Anodyne PIK3CA 29 40 CC[C@H](O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960831 ED On-Demand Anodyne MTOR 61 40 CC[C@H](O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960831 ED On-Demand Anodyne PIK3CG 30 40 CC[C@H](O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960831 ED On-Demand Anodyne STAT6 53 32 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960837 GD On-Demand Anodyne PIK3CA 24 40 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960837 GD On-Demand Anodyne MTOR 40 38 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960837 GD On-Demand Anodyne STAT6 55 34 O=C(Cn1cc(-c2ccsc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960844 FE On-Demand Anodyne MTOR 56 39 O=C(Cn1cc(-c2ccsc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960844 FE On-Demand Anodyne STAT6 52 33 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(Cl)c2)nn1 ZINC000880960845 ED On-Demand Mild ENPP1 76 37 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(Cl)c2)nn1 ZINC000880960846 ED On-Demand Mild ENPP1 76 37 C[C@H](O)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960849 FD On-Demand Anodyne MTOR 52 42 C[C@H](O)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960849 FD On-Demand Anodyne PIK3CG 29 42 C[C@H](O)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960849 FD On-Demand Anodyne STAT6 52 32 O=C(Cn1cc(CNC2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960855 GE On-Demand Anodyne MTOR 45 35 O=C(Cn1cc(CNC2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960855 GE On-Demand Anodyne STAT6 56 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@]1(c2ccccc2)C[C@@H](O)C1 ZINC000880960858 FG On-Demand Anodyne TRPV1 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CCSC[C@@H]1C1CC1 ZINC000880960861 EG On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCSC[C@H]1C1CC1 ZINC000880960862 EG On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCn2cnc(C(F)(F)F)c2C1 ZINC000880960863 GG On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880960865 GI On-Demand Anodyne RBP4 67 43 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880960865 GI On-Demand Anodyne SFRP1 50 33 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@H]2C1 ZINC000880960865 GI On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880960866 GI On-Demand Anodyne RBP4 67 43 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880960866 GI On-Demand Anodyne SFRP1 50 33 O=C(Nc1cnccc1C(F)(F)F)N1Cc2ccccc2N2CCC[C@@H]2C1 ZINC000880960866 GI On-Demand Anodyne WNT3 40 33 NC(=O)C1(N2CCCCC2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880960867 GE On-Demand Anodyne RBP4 48 38 Nc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960870 GE On-Demand Anodyne MTOR 40 36 Nc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880960870 GE On-Demand Anodyne STAT6 58 38 COC(=O)c1ccc2c(c1)CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880960871 GG On-Demand Anodyne RBP4 45 36 COCCNCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960872 GC On-Demand Anodyne STAT6 46 32 CC(C)(C)[C@@H](O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960874 GD On-Demand Anodyne MTOR 53 39 CC(C)(C)[C@@H](O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960874 GD On-Demand Anodyne STAT6 54 33 NCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960876 EC On-Demand Anodyne MTOR 45 37 NCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960876 EC On-Demand Anodyne STAT6 59 36 O=C(Cn1cc(CC2(O)CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960879 GD On-Demand Anodyne STAT6 54 33 O=C(Nc1cnccc1C(F)(F)F)N1CCCSC[C@H]1c1ccccc1 ZINC000880960882 GJ On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCSC[C@@H]1c1ccccc1 ZINC000880960883 GJ On-Demand Anodyne RBP4 58 41 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne PRNP 40 32 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne JAK2 15 45 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne HDAC10 22 41 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne HDAC3 24 41 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne HDAC6 21 41 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne MTOR 43 39 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne PIK3CB 18 44 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne STAT6 55 35 O=C(Cn1cc(-c2cccc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960884 GG On-Demand Anodyne DGAT1 18 41 CCOc1ccccc1NC(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880960885 EE On-Demand Anodyne HCN1 57 37 CCOc1ccccc1NC(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880960885 EE On-Demand Anodyne HCN4 47 36 O=C(Cn1cc(C[C@@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960886 GD On-Demand Anodyne MTOR 46 35 O=C(Cn1cc(C[C@@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960886 GD On-Demand Anodyne STAT6 51 31 O=C(Cn1cc(C[C@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960887 GD On-Demand Anodyne MTOR 46 35 O=C(Cn1cc(C[C@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960887 GD On-Demand Anodyne STAT6 51 31 O=C(Cn1cc(-c2cccs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960892 FE On-Demand Anodyne PIK3CA 21 40 O=C(Cn1cc(-c2cccs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960892 FE On-Demand Anodyne MTOR 34 40 O=C(Cn1cc(-c2cccs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960892 FE On-Demand Anodyne PIK3CG 22 40 O=C(Cn1cc(-c2cccs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960892 FE On-Demand Anodyne STAT6 58 35 O=C(Cn1cc(-c2ccccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960895 GF On-Demand Anodyne MTOR 47 37 O=C(Cn1cc(-c2ccccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960895 GF On-Demand Anodyne STAT6 78 40 O=C(Cn1cc(-c2ccccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960895 GF On-Demand Anodyne DGAT1 16 48 O=C(Cn1cc(C2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960896 FF On-Demand Anodyne MTOR 66 36 O=C(Cn1cc(C2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960896 FF On-Demand Anodyne STAT6 54 34 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880960899 DD On-Demand Mild ENPP1 61 32 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880960900 DD On-Demand Mild ENPP1 61 32 O=C1CCC(c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)CC1 ZINC000880960901 GD On-Demand Anodyne MTOR 50 35 O=C1CCC(c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)CC1 ZINC000880960901 GD On-Demand Anodyne STAT6 52 33 CNc1nc(C(=O)N2C[C@@H](O)[C@H](Oc3ccccc3)C2)cs1 ZINC000880960903 DD On-Demand Anodyne TRPC6 61 42 CNc1nc(C(=O)N2C[C@@H](O)[C@H](Oc3ccccc3)C2)cs1 ZINC000880960903 DD On-Demand Anodyne TRPC3 53 42 O=C(Cn1cc(C2CCNCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960904 FD On-Demand Anodyne MTOR 51 38 O=C(Cn1cc(C2CCNCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960904 FD On-Demand Anodyne STAT6 57 33 COC(=O)[C@@H]1C[C@H](NC(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880960907 GH On-Demand Anodyne TRPV1 29 41 COC(=O)[C@@H]1C[C@H](NC(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880960907 GH On-Demand Anodyne RBP4 74 40 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960911 GD On-Demand Anodyne CASR 46 37 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960911 GD On-Demand Anodyne MTOR 53 39 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960911 GD On-Demand Anodyne STAT6 63 37 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960912 GD On-Demand Anodyne CASR 46 37 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960912 GD On-Demand Anodyne MTOR 53 39 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960912 GD On-Demand Anodyne STAT6 63 37 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne PDE5A 40 34 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne PIK3CA 49 42 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne PRNP 40 34 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne JAK2 19 43 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne MAPKAPK5 40 35 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne MTOR 83 42 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne PIK3CG 43 42 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880960914 GD On-Demand Anodyne STAT6 65 37 O=C(NC[C@@H](O)C(F)(F)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880960919 FF On-Demand Mild TRPV1 15 47 O=C(NC[C@H](O)C(F)(F)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880960920 FF On-Demand Mild TRPV1 15 47 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960921 FD On-Demand Anodyne MTOR 71 37 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960921 FD On-Demand Anodyne STAT6 52 33 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960922 FD On-Demand Anodyne MTOR 71 37 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960922 FD On-Demand Anodyne STAT6 52 33 COC[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880960930 CE On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)CC2(CCOCC2)C1 ZINC000880960933 FE On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)CC2(CCOCC2)C1 ZINC000880960934 FE On-Demand Anodyne RBP4 54 39 O=C(NC[C@@H](O)c1cccc(C(F)(F)F)c1)Nc1cnccc1C(F)(F)F ZINC000880960935 GH On-Demand Anodyne TRPV1 32 54 O=C(NC[C@H](O)c1cccc(C(F)(F)F)c1)Nc1cnccc1C(F)(F)F ZINC000880960936 GH On-Demand Anodyne TRPV1 32 54 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960938 GD On-Demand Anodyne STAT6 55 34 C#CCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880960939 EE On-Demand Mild RBP4 58 41 O=C(NC[C@@H]1C=CCC1)Nc1cnccc1C(F)(F)F ZINC000880960947 CG On-Demand Anodyne TRPV1 16 46 O=C(NC[C@H]1C=CCC1)Nc1cnccc1C(F)(F)F ZINC000880960948 CG On-Demand Anodyne TRPV1 16 46 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC)c(Cl)c2)nn1 ZINC000880960951 ED On-Demand Anodyne GRM4 15 47 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC)c(Cl)c2)nn1 ZINC000880960951 ED On-Demand Anodyne ENPP1 77 38 CCN(CC)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960963 FD On-Demand Anodyne MTOR 51 37 CCN(CC)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960963 FD On-Demand Anodyne STAT6 52 32 CCN1CC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880960966 DE On-Demand Anodyne TRPV1 16 42 O=C(Cn1cc(CC2(O)CCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960968 FD On-Demand Anodyne STAT6 55 34 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880960982 GD On-Demand Anodyne STAT6 52 32 CC[C@@](C)(O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960998 FD On-Demand Anodyne MTOR 46 36 CC[C@@](C)(O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880960998 FD On-Demand Anodyne STAT6 54 33 O=C(Cn1cc(-c2cncnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961001 FD On-Demand Anodyne MTOR 65 38 O=C(Cn1cc(-c2cncnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961001 FD On-Demand Anodyne STAT6 60 36 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne PIK3CA 52 44 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne JAK2 21 47 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne MTOR 98 44 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne PIK3CG 43 44 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne PIK3CB 15 42 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne STAT6 64 37 COc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961003 GE On-Demand Anodyne DGAT1 16 40 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961004 FD On-Demand Anodyne MTOR 54 37 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961004 FD On-Demand Anodyne STAT6 61 35 O=C(Cn1cc(CN2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961006 GD On-Demand Anodyne MTOR 44 36 O=C(Cn1cc(CN2CCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961006 GD On-Demand Anodyne STAT6 58 33 O=C(Cn1cc(C2(F)COC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961013 FC On-Demand Anodyne MTOR 40 36 O=C(Cn1cc(C2(F)COC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961013 FC On-Demand Anodyne STAT6 61 35 CCC[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961014 FD On-Demand Anodyne MTOR 44 40 CCC[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961014 FD On-Demand Anodyne PIK3CG 24 40 CCC[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961014 FD On-Demand Anodyne STAT6 54 33 CCC[C@@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961015 FD On-Demand Anodyne MTOR 44 40 CCC[C@@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961015 FD On-Demand Anodyne PIK3CG 24 40 CCC[C@@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961015 FD On-Demand Anodyne STAT6 54 33 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(F)c(F)cc2C1 ZINC000880961020 FH On-Demand Anodyne RBP4 56 40 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961022 EF On-Demand Anodyne RBP4 68 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C(C)(C)C1 ZINC000880961024 DH On-Demand Anodyne RBP4 49 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C(C)(C)C1 ZINC000880961025 DH On-Demand Anodyne RBP4 49 41 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961029 FG On-Demand Anodyne RBP4 54 39 CC(=O)CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961030 FD On-Demand Anodyne MTOR 43 37 CC(=O)CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961030 FD On-Demand Anodyne STAT6 52 32 CCOc1ccccc1NC(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880961033 DD On-Demand Anodyne HCN1 50 34 CCOc1ccccc1NC(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880961033 DD On-Demand Anodyne HCN4 42 33 C[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961035 EC On-Demand Anodyne MTOR 59 44 C[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961035 EC On-Demand Anodyne PIK3CG 31 44 C[C@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961035 EC On-Demand Anodyne STAT6 56 35 O=C(Cn1cc(-c2ccc(F)cn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961036 GD On-Demand Anodyne STAT6 72 40 O=C(Cn1cc(-c2ccc(F)cn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961036 GD On-Demand Anodyne SLC27A1 43 34 O=C1CCC[C@H](c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)C1 ZINC000880961037 GD On-Demand Anodyne STAT6 51 32 O=C1CCC[C@@H](c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)C1 ZINC000880961038 GD On-Demand Anodyne STAT6 51 32 CC[C@@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961040 ED On-Demand Anodyne MTOR 50 39 CC[C@@H](N)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961040 ED On-Demand Anodyne STAT6 55 34 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(F)cc1F ZINC000880961042 FD On-Demand Anodyne EPHX2 18 49 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)CC(F)F ZINC000880961043 EH On-Demand Anodyne TRPV1 20 45 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(F)F ZINC000880961046 CF On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ncncc2C1 ZINC000880961060 DE On-Demand Anodyne RBP4 60 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961061 FD On-Demand Anodyne MTOR 64 39 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961061 FD On-Demand Anodyne STAT6 53 34 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961062 FD On-Demand Anodyne MTOR 64 39 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961062 FD On-Demand Anodyne STAT6 53 34 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1(C)C ZINC000880961063 DF On-Demand Anodyne RBP4 60 43 O=C(Nc1cnccc1C(F)(F)F)N1CC(CC2CCOCC2)C1 ZINC000880961065 EG On-Demand Anodyne RBP4 59 43 CNC(C)(C)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961066 FD On-Demand Anodyne MTOR 59 38 CNC(C)(C)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961066 FD On-Demand Anodyne STAT6 60 34 Cc1nn(C)cc1-c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961068 GD On-Demand Anodyne STAT6 52 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC(F)CC1 ZINC000880961073 CG On-Demand Anodyne TRPV1 19 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(F)CC1 ZINC000880961073 CG On-Demand Anodyne RBP4 81 47 O=C(Cn1cc(C[C@@H]2CCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961082 FC On-Demand Anodyne STAT6 57 32 O=C(Cn1cc(C[C@H]2CCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961083 FC On-Demand Anodyne STAT6 57 32 NCCSCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961090 GC On-Demand Anodyne STAT6 55 33 O=C(Cn1cc([C@@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961097 FC On-Demand Anodyne PIK3CA 42 39 O=C(Cn1cc([C@@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961097 FC On-Demand Anodyne MTOR 102 39 O=C(Cn1cc([C@@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961097 FC On-Demand Anodyne STAT6 51 33 O=C(Cn1cc([C@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961098 FC On-Demand Anodyne PIK3CA 42 39 O=C(Cn1cc([C@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961098 FC On-Demand Anodyne MTOR 102 39 O=C(Cn1cc([C@H]2COCCN2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961098 FC On-Demand Anodyne STAT6 51 33 NCCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961099 EC On-Demand Anodyne MTOR 43 36 NCCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961099 EC On-Demand Anodyne STAT6 57 36 COC(=O)[C@@]1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961100 ED On-Demand Anodyne RBP4 54 39 O=C(Cn1cc(-c2cncs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961102 FD On-Demand Anodyne MTOR 53 36 O=C(Cn1cc(-c2cncs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961102 FD On-Demand Anodyne STAT6 54 35 Cn1c(S)nnc1[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961103 GF On-Demand Anodyne RBP4 61 41 Cn1c(S)nnc1[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961104 GF On-Demand Anodyne RBP4 61 41 CCOc1ccccc1NC(=O)Cn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880961105 GC On-Demand Anodyne SSTR5 41 35 O=C(Cn1cc(-c2cncc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961107 GE On-Demand Anodyne MTOR 51 39 O=C(Cn1cc(-c2cncc(Cl)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961107 GE On-Demand Anodyne STAT6 56 35 N#Cc1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880961117 DE On-Demand Mild CCR3 15 41 N#Cc1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880961118 DE On-Demand Mild CCR3 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCCO2)CC1 ZINC000880961119 EH On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCCO2)CC1 ZINC000880961119 EH On-Demand Anodyne RBP4 55 39 NCc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880961132 GD On-Demand Anodyne HDAC10 20 42 NCc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880961132 GD On-Demand Anodyne HDAC3 22 42 NCc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880961132 GD On-Demand Anodyne HDAC6 19 42 NCc1cccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)c1 ZINC000880961132 GD On-Demand Anodyne STAT6 65 39 O=C(Cn1cc(Cn2ccnc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961138 FC On-Demand Anodyne STAT6 55 32 CCOc1ccccc1NC(=O)Cn1cc([C@]2(O)CCOC2)nn1 ZINC000880961143 EC On-Demand Anodyne HCN1 42 35 CCOc1ccccc1NC(=O)Cn1cc([C@@]2(O)CCOC2)nn1 ZINC000880961144 EC On-Demand Anodyne HCN1 42 35 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne PIK3CA 42 44 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne PRNP 38 42 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne JAK2 16 47 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne HDAC6 18 40 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne MTOR 77 44 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne PIK3CG 33 44 O=C(Cn1cc(-c2ccncc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961150 FD On-Demand Anodyne STAT6 54 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H](O)CC1 ZINC000880961155 DF On-Demand Anodyne TRPV1 26 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H](O)CC1 ZINC000880961155 DF On-Demand Anodyne EPHX2 45 48 CC(=O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961158 EC On-Demand Anodyne PIK3CA 35 40 CC(=O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961158 EC On-Demand Anodyne MTOR 68 40 CC(=O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961158 EC On-Demand Anodyne PIK3CG 34 40 CC(=O)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961158 EC On-Demand Anodyne STAT6 60 34 O=C(Cn1cc([C@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961161 FD On-Demand Anodyne MTOR 49 36 O=C(Cn1cc([C@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961161 FD On-Demand Anodyne STAT6 46 32 O=C(Cn1cc([C@@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961162 FD On-Demand Anodyne MTOR 49 36 O=C(Cn1cc([C@@H]2CCCNC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961162 FD On-Demand Anodyne STAT6 46 32 O=C(Cn1cc(C[C@@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961170 FD On-Demand Anodyne MTOR 52 37 O=C(Cn1cc(C[C@@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961170 FD On-Demand Anodyne STAT6 52 32 O=C(Cn1cc(C[C@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961171 FD On-Demand Anodyne MTOR 52 37 O=C(Cn1cc(C[C@H](O)C2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961171 FD On-Demand Anodyne STAT6 52 32 CCOc1ccccc1NC(=O)Cn1cc([C@@H]2CCCCO2)nn1 ZINC000880961172 EF On-Demand Anodyne SSTR5 40 34 CCOc1ccccc1NC(=O)Cn1cc([C@H]2CCCCO2)nn1 ZINC000880961173 EF On-Demand Anodyne SSTR5 40 34 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H](C2CCOCC2)C1 ZINC000880961174 FI On-Demand Anodyne RBP4 69 46 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H](C2CCOCC2)C1 ZINC000880961175 FI On-Demand Anodyne RBP4 69 46 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961179 FD On-Demand Anodyne MTOR 40 41 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961179 FD On-Demand Anodyne PIK3CG 25 41 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961179 FD On-Demand Anodyne STAT6 50 31 O=C(Cn1cc(C2CCCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961182 GG On-Demand Anodyne MTOR 66 36 O=C(Cn1cc(C2CCCCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961182 GG On-Demand Anodyne STAT6 54 34 C[C@H]1[C@H](C(=O)N2C[C@@H](O)[C@H](Oc3ccccc3)C2)CCN1C ZINC000880961186 DC On-Demand Anodyne CHRNA10 15 40 C[C@@H]1[C@@H](C(=O)N2C[C@@H](O)[C@H](Oc3ccccc3)C2)CCN1C ZINC000880961187 DC On-Demand Anodyne CHRNA10 15 40 CCc1nccn1Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961189 GD On-Demand Anodyne STAT6 60 33 CC#CCNCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961192 FC On-Demand Mild STAT6 56 35 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@]2(O)C1 ZINC000880961194 CD On-Demand Anodyne RBP4 58 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@]2(O)C1 ZINC000880961195 CD On-Demand Anodyne RBP4 58 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@@]2(O)C1 ZINC000880961196 CD On-Demand Anodyne RBP4 58 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@@]2(O)C1 ZINC000880961197 CD On-Demand Anodyne RBP4 58 43 CN(C)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1n1ccnn1 ZINC000880961198 FD On-Demand Anodyne RBP4 54 39 O=C(NC[C@H]1CCC2(CCOCC2)CO1)Nc1cnccc1C(F)(F)F ZINC000880961201 FG On-Demand Anodyne TRPV1 18 41 COc1ccc(CN(CCO)C(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880961203 FG On-Demand Anodyne ROCK2 21 43 C[C@H]1c2sccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880961208 EI On-Demand Anodyne TRPM8 41 45 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961209 FD On-Demand Anodyne MTOR 49 36 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961209 FD On-Demand Anodyne STAT6 58 33 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880961212 DC On-Demand Anodyne CA9 18 43 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880961212 DC On-Demand Anodyne ENPP1 61 32 COC(=O)Cc1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880961212 DC On-Demand Anodyne IMDH_CRYPV 23 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OC)c(Cl)c2)nn1 ZINC000880961217 FD On-Demand Anodyne ENPP1 73 36 Cn1nccc1-c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961218 FD On-Demand Anodyne MTOR 60 37 Cn1nccc1-c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961218 FD On-Demand Anodyne STAT6 57 33 O=C(Cn1cc(CSCCO)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961225 GC On-Demand Anodyne STAT6 51 32 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne PIK3CA 39 40 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne JAK2 15 45 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne HDAC6 17 43 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne MTOR 72 40 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne PIK3CG 33 40 NCc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961230 GD On-Demand Anodyne STAT6 64 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CC[C@H]1c1ccccc12 ZINC000880961235 EJ On-Demand Anodyne RBP4 92 48 N#CCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961236 ED On-Demand Mild STAT6 52 32 O=C(Cn1cc(CCN2CCNCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961237 GC On-Demand Anodyne PIK3CA 21 41 O=C(Cn1cc(CCN2CCNCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961237 GC On-Demand Anodyne STAT6 58 33 CCC1(N2CCCCC2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961238 GI On-Demand Anodyne RBP4 46 38 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1c1ccncc1 ZINC000880961239 FG On-Demand Anodyne RBP4 60 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1c1ccncc1 ZINC000880961239 FG On-Demand Anodyne SMO 19 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1c1ccncc1 ZINC000880961240 FG On-Demand Anodyne RBP4 60 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1c1ccncc1 ZINC000880961240 FG On-Demand Anodyne SMO 19 42 O=C(Cn1cc(-c2ccccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961250 FD On-Demand Anodyne PRNP 60 44 O=C(Cn1cc(-c2ccccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961250 FD On-Demand Anodyne MTOR 63 37 O=C(Cn1cc(-c2ccccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961250 FD On-Demand Anodyne STAT6 69 39 O=C(Cn1cc(-c2ccccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961250 FD On-Demand Anodyne DGAT1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(NC2CCOCC2)CC1 ZINC000880961260 FF On-Demand Anodyne RBP4 70 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(NC2CCOCC2)CC1 ZINC000880961260 FF On-Demand Anodyne SFRP1 53 35 N#Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880961261 FD On-Demand Mild CASR 25 48 N#Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880961261 FD On-Demand Mild CCR3 18 42 N#Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880961261 FD On-Demand Mild EPHX2 20 42 N#Cc1cccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880961261 FD On-Demand Mild MCHR1 27 40 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne PIK3CA 40 39 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne JAK2 15 44 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne MAPKAPK5 42 38 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne HDAC6 15 40 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne MTOR 79 39 O=C(Cn1cc(-c2ccc(F)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961264 GD On-Demand Anodyne STAT6 71 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C=C[C@H]1C2 ZINC000880961266 CF On-Demand Anodyne RBP4 55 41 O=C(Cn1cc(-c2cccnc2Cl)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961267 GE On-Demand Anodyne STAT6 60 36 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@H]1CN2c1ccccc1 ZINC000880961269 FH On-Demand Anodyne RBP4 74 46 NCCCCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961273 FD On-Demand Anodyne STAT6 56 34 O=C(Cn1cc(-c2nccs2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961274 FD On-Demand Anodyne STAT6 58 35 COC(=O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961279 FC On-Demand Anodyne PIK3CA 31 40 COC(=O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961279 FC On-Demand Anodyne MTOR 56 40 COC(=O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961279 FC On-Demand Anodyne PIK3CG 30 40 COC(=O)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961279 FC On-Demand Anodyne STAT6 56 36 CC(C)(CO)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccnc1 ZINC000880961283 FG On-Demand Anodyne TRPV1 20 44 O=C(Cn1cc(CCCO)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961287 EC On-Demand Anodyne MTOR 44 39 O=C(Cn1cc(CCCO)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961287 EC On-Demand Anodyne STAT6 53 33 O=C(Cn1cc(C(=O)C2CCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961288 FD On-Demand Anodyne MTOR 59 36 O=C(Cn1cc(C(=O)C2CCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961288 FD On-Demand Anodyne STAT6 53 32 N[C@@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961292 GD On-Demand Anodyne CASR 46 37 N[C@@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961292 GD On-Demand Anodyne PIK3CA 23 40 N[C@@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961292 GD On-Demand Anodyne MTOR 46 40 N[C@@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961292 GD On-Demand Anodyne PIK3CG 26 40 N[C@@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961292 GD On-Demand Anodyne STAT6 65 38 N[C@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961293 GD On-Demand Anodyne CASR 46 37 N[C@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961293 GD On-Demand Anodyne PIK3CA 23 40 N[C@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961293 GD On-Demand Anodyne MTOR 46 40 N[C@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961293 GD On-Demand Anodyne PIK3CG 26 40 N[C@H](c1ccccc1)c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961293 GD On-Demand Anodyne STAT6 65 38 O=C(Nc1cnccc1C(F)(F)F)NC1(c2ncccn2)CCC1 ZINC000880961303 EG On-Demand Anodyne TRPV1 19 42 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne PIK3CA 45 47 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne PRNP 44 37 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne JAK2 18 47 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne HDAC6 17 42 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne MTOR 91 47 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne PIK3CG 38 42 Cc1ccc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cc1 ZINC000880961304 GF On-Demand Anodyne STAT6 58 35 NC(=O)[C@H](F)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961305 EE On-Demand Anodyne RBP4 67 41 NC(=O)[C@@H](F)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961306 EE On-Demand Anodyne RBP4 67 41 O=C(Cn1cc(-c2c(F)cccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961311 GF On-Demand Anodyne STAT6 62 41 O=C(Cn1cc(-c2c(F)cccc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961311 GF On-Demand Anodyne DGAT1 15 46 O=C(Cn1cc(-c2cncc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961312 GD On-Demand Anodyne HDAC6 18 40 O=C(Cn1cc(-c2cncc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961312 GD On-Demand Anodyne MTOR 46 38 O=C(Cn1cc(-c2cncc(F)c2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961312 GD On-Demand Anodyne STAT6 69 40 CCOc1ccccc1NC(=O)Cn1cc(C2(O)CCOCC2)nn1 ZINC000880961317 ED On-Demand Anodyne HCN1 43 37 Cc1ccsc1-c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961318 GF On-Demand Anodyne STAT6 51 33 CCCn1cc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880961324 GE On-Demand Anodyne MTOR 69 38 CCCn1cc(-c2cn(CC(=O)Nc3ccc(N4CCOCC4)cc3)nn2)cn1 ZINC000880961324 GE On-Demand Anodyne STAT6 57 33 O=C(Cn1cc(Cn2cccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961325 FC On-Demand Anodyne MTOR 46 35 O=C(Cn1cc(Cn2cccn2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961325 FC On-Demand Anodyne STAT6 62 33 CN(C)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961326 FC On-Demand Anodyne PIK3CA 35 40 CN(C)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961326 FC On-Demand Anodyne MTOR 68 40 CN(C)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961326 FC On-Demand Anodyne PIK3CG 29 40 CN(C)CCc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961326 FC On-Demand Anodyne STAT6 55 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)CC1 ZINC000880961335 CE On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)CC1 ZINC000880961335 CE On-Demand Anodyne RBP4 82 46 O=C(Cn1cc(-c2cnccc2Cl)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961338 GE On-Demand Anodyne STAT6 60 37 C/C=C\c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961341 ED On-Demand Anodyne MTOR 55 38 C/C=C\c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961341 ED On-Demand Anodyne STAT6 54 33 C/C=C/c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961342 ED On-Demand Anodyne MTOR 55 38 C/C=C/c1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961342 ED On-Demand Anodyne STAT6 54 33 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961345 FD On-Demand Anodyne STAT6 52 32 COC(=O)C1CCC(c2cn(CC(=O)Nc3ccc(OC)cc3)nn2)CC1 ZINC000880961346 FE On-Demand Anodyne MTNR1B 16 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCC2(CC1)COC2 ZINC000880961347 EG On-Demand Anodyne EPHX2 32 44 O=C(NCC1(CC2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880961352 DH On-Demand Anodyne TRPV1 22 48 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961354 GD On-Demand Anodyne JAK2 15 45 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961354 GD On-Demand Anodyne MAPKAPK5 40 35 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961354 GD On-Demand Anodyne MTOR 58 38 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961354 GD On-Demand Anodyne STAT6 69 38 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961355 FD On-Demand Anodyne MTOR 44 38 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961355 FD On-Demand Anodyne STAT6 56 34 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961356 GC On-Demand Anodyne MTOR 55 38 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961356 GC On-Demand Anodyne STAT6 64 34 O=C(Cn1cc(CN2CCCCC2=O)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961357 GD On-Demand Anodyne STAT6 50 31 O=C(Cn1cc(CNC2CCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961362 GD On-Demand Anodyne MTOR 50 35 O=C(Cn1cc(CNC2CCCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961362 GD On-Demand Anodyne STAT6 56 35 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961365 GD On-Demand Anodyne STAT6 51 33 O=C(Cn1cc(-c2cccnc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961367 GD On-Demand Anodyne MTOR 40 37 O=C(Cn1cc(-c2cccnc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961367 GD On-Demand Anodyne STAT6 67 36 O=C(Cn1cc(CN2CCNCC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961369 GC On-Demand Anodyne STAT6 57 32 O=C(Cn1cc(-c2ccncc2F)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961370 GD On-Demand Anodyne STAT6 81 39 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(OC)cc2)nn1 ZINC000880961376 DC On-Demand Anodyne ENPP1 54 30 O=C(Cn1cc(CNC2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961379 FD On-Demand Anodyne MTOR 58 36 O=C(Cn1cc(CNC2CC2)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961379 FD On-Demand Anodyne STAT6 55 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)COCCO2 ZINC000880961381 EF On-Demand Anodyne RBP4 55 39 CN(CCO)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961387 FC On-Demand Anodyne MTOR 51 36 CN(CCO)Cc1cn(CC(=O)Nc2ccc(N3CCOCC3)cc2)nn1 ZINC000880961387 FC On-Demand Anodyne STAT6 53 32 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961388 GD On-Demand Anodyne MTOR 50 35 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961388 GD On-Demand Anodyne STAT6 51 31 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961389 GD On-Demand Anodyne MTOR 50 35 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1ccc(N2CCOCC2)cc1 ZINC000880961389 GD On-Demand Anodyne STAT6 51 31 CC(C)c1cc(NC(=O)Nc2cnccc2C(F)(F)F)ccc1O ZINC000880961393 EJ On-Demand Anodyne TRPV1 24 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)[C@@H](CO)C1 ZINC000880961396 DD On-Demand Anodyne RBP4 79 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)[C@H](CO)C1 ZINC000880961397 DD On-Demand Anodyne RBP4 79 48 COC(=O)C[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961402 DE On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880961408 FI On-Demand Anodyne RBP4 98 55 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880961408 FI On-Demand Anodyne SMO 25 45 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2cnccc2C(F)(F)F)C3)c1 ZINC000880961412 GE On-Demand Anodyne P2RX7 37 47 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880961415 ED On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2cccs2)C1 ZINC000880961419 EH On-Demand Anodyne RBP4 70 44 O=C(Nc1cnccc1C(F)(F)F)NC1CC2(CSC2)C1 ZINC000880961424 DG On-Demand Anodyne TRPV1 21 40 O=C(Nc1cnccc1C(F)(F)F)NC1CC2(CSC2)C1 ZINC000880961424 DG On-Demand Anodyne EPHX2 15 40 O=C(NCc1ccnc(N2CCSCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880961425 GG On-Demand Anodyne TRPV1 19 47 C=C[C@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961426 FE On-Demand Mild GRIN2B 84 44 C=C[C@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961426 FE On-Demand Mild SIGMAR1 19 43 C=C[C@@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961427 FE On-Demand Mild GRIN2B 84 44 C=C[C@@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961427 FE On-Demand Mild SIGMAR1 19 43 O=C(NCC1CC=CC1)Nc1cnccc1C(F)(F)F ZINC000880961429 CG On-Demand Anodyne TRPV1 23 47 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880961430 GG On-Demand Mild RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CCC[C@]2(CO)C1 ZINC000880961431 EF On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2cccc(F)c2C1 ZINC000880961434 FH On-Demand Anodyne RBP4 54 39 O=C(NCC[C@@H](O)C(F)F)Nc1cnccc1C(F)(F)F ZINC000880961435 DE On-Demand Anodyne TRPV1 15 46 O=C(NCC[C@H](O)C(F)F)Nc1cnccc1C(F)(F)F ZINC000880961436 DE On-Demand Anodyne TRPV1 15 46 NC(=O)[C@@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961437 DD On-Demand Anodyne EPHX2 20 42 NC(=O)C1CC(NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961438 DD On-Demand Anodyne EPHX2 20 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1C(F)(F)F ZINC000880961439 DG On-Demand Anodyne TRPV1 26 41 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cn1 ZINC000880961444 GF On-Demand Mild RBP4 42 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880961450 FH On-Demand Anodyne RBP4 69 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880961450 FH On-Demand Anodyne SFRP1 51 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880961450 FH On-Demand Anodyne WNT3 58 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880961451 FH On-Demand Anodyne RBP4 69 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880961451 FH On-Demand Anodyne SFRP1 51 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880961451 FH On-Demand Anodyne WNT3 58 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880961452 FH On-Demand Anodyne RBP4 69 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880961452 FH On-Demand Anodyne SFRP1 51 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880961452 FH On-Demand Anodyne WNT3 58 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@H](O)c1ccccc1 ZINC000880961453 FH On-Demand Anodyne RBP4 69 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@H](O)c1ccccc1 ZINC000880961453 FH On-Demand Anodyne SFRP1 51 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@H](O)c1ccccc1 ZINC000880961453 FH On-Demand Anodyne WNT3 58 36 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961458 DG On-Demand Mild TRPV1 20 40 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961458 DG On-Demand Mild EPHX2 37 47 O=C(NC[C@H](O)Cc1cccc(Cl)c1)Nc1cnccc1C(F)(F)F ZINC000880961459 FG On-Demand Anodyne TRPV1 27 49 O=C(NC[C@@H](O)Cc1cccc(Cl)c1)Nc1cnccc1C(F)(F)F ZINC000880961460 FG On-Demand Anodyne TRPV1 27 49 NOCc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961462 ED On-Demand Anodyne GRIN2B 89 47 C/C=C\C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961463 EI On-Demand Anodyne RBP4 57 41 C/C=C/C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961464 EI On-Demand Anodyne RBP4 57 41 C/C=C/C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961465 EI On-Demand Anodyne RBP4 57 41 C/C=C\C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961466 EI On-Demand Anodyne RBP4 57 41 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961467 ED On-Demand Anodyne RBP4 56 40 CC[C@@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961472 FE On-Demand Anodyne GRIN2B 85 43 CC[C@@](C)(O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961472 FE On-Demand Anodyne CCR3 25 40 O=C(NC[C@@H]1C[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961475 CD On-Demand Anodyne TRPV1 19 46 O=C(NCC1CC(O)C1)Nc1cnccc1C(F)(F)F ZINC000880961476 CD On-Demand Anodyne TRPV1 19 46 O=C(NC[C@H]1C[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961477 CD On-Demand Anodyne TRPV1 19 46 CO[C@@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961478 CE On-Demand Anodyne EPHX2 35 40 O=C(Nc1cnccc1C(F)(F)F)NC1CC(CO)(CO)C1 ZINC000880961480 DD On-Demand Anodyne TRPV1 24 43 O=C(Nc1cnccc1C(F)(F)F)NC1CC(CO)(CO)C1 ZINC000880961480 DD On-Demand Anodyne EPHX2 23 40 O=C(NC[C@@H]1CCO[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961481 FH On-Demand Anodyne TRPV1 21 46 O=C(NC[C@@H]1CCO[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961481 FH On-Demand Anodyne RBP4 46 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2nccs2)CC1 ZINC000880961484 FI On-Demand Anodyne RBP4 66 41 C[C@H]1C[C@H](CO)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880961491 DF On-Demand Anodyne RBP4 40 38 C[C@H](N)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961498 ED On-Demand Anodyne GRIN2B 84 44 C[C@H](N)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961498 ED On-Demand Anodyne SIGMAR1 15 41 C[C@H](N)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961498 ED On-Demand Anodyne GRIN2C 17 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CO[C@@H](C2CC2)C1 ZINC000880961501 DF On-Demand Anodyne EPHX2 19 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CO[C@H](C2CC2)C1 ZINC000880961502 DF On-Demand Anodyne EPHX2 19 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CO[C@@H](C2CC2)C1 ZINC000880961503 DF On-Demand Anodyne EPHX2 19 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CO[C@H](C2CC2)C1 ZINC000880961504 DF On-Demand Anodyne EPHX2 19 40 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880961510 FH On-Demand Anodyne RBP4 70 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880961511 FH On-Demand Anodyne RBP4 70 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H](C(F)(F)F)O1 ZINC000880961512 FH On-Demand Anodyne RBP4 70 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H](C(F)(F)F)O1 ZINC000880961513 FH On-Demand Anodyne RBP4 70 42 CC(C)(C)OC(=O)N1C[C@@H]2C[C@H]1CN2C(=O)Nc1cnccc1C(F)(F)F ZINC000880961516 GG On-Demand Anodyne RBP4 48 40 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCCO2)C1 ZINC000880961519 DE On-Demand Anodyne RBP4 41 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)[C@H](C(F)(F)F)C1 ZINC000880961522 FF On-Demand Anodyne RBP4 75 45 O=C(Nc1cnccc1C(F)(F)F)N1CC(CNC(=O)C(F)(F)F)C1 ZINC000880961523 FE On-Demand Anodyne RBP4 66 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880961524 FI On-Demand Anodyne EPHX2 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880961524 FI On-Demand Anodyne RBP4 68 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880961524 FI On-Demand Anodyne SFRP1 43 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)CC1 ZINC000880961524 FI On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)CC1 ZINC000880961525 FI On-Demand Anodyne EPHX2 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)CC1 ZINC000880961525 FI On-Demand Anodyne RBP4 68 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)CC1 ZINC000880961525 FI On-Demand Anodyne SFRP1 43 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)CC1 ZINC000880961525 FI On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880961526 DD On-Demand Anodyne RBP4 85 48 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961533 EH On-Demand Anodyne RBP4 57 41 O=C(NC[C@H](CO)c1ccc(Cl)cc1)Nc1cnccc1C(F)(F)F ZINC000880961538 FH On-Demand Anodyne TRPV1 20 48 O=C(NC[C@@H](CO)c1ccc(Cl)cc1)Nc1cnccc1C(F)(F)F ZINC000880961539 FH On-Demand Anodyne TRPV1 20 48 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961540 GF On-Demand Anodyne GRIN2B 81 45 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961540 GF On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961540 GF On-Demand Anodyne GRIN2C 18 43 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961541 GF On-Demand Anodyne GRIN2B 81 45 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961541 GF On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961541 GF On-Demand Anodyne GRIN2C 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CCc2cnccn2)CC1 ZINC000880961542 GE On-Demand Anodyne RBP4 54 39 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961543 GH On-Demand Anodyne RBP4 47 38 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](C(F)F)CC1 ZINC000880961548 EF On-Demand Anodyne RBP4 72 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](C(F)F)CC1 ZINC000880961549 EF On-Demand Anodyne RBP4 72 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CC[C@@H](O)[C@@H]21 ZINC000880961550 DE On-Demand Anodyne RBP4 56 41 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)C(F)(F)F ZINC000880961552 EF On-Demand Anodyne TRPV1 15 47 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)C(F)(F)F ZINC000880961554 EF On-Demand Anodyne TRPV1 15 47 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961563 GF On-Demand Anodyne GRIN2B 71 42 O=C(Nc1cnccc1C(F)(F)F)N1OC2CCC1CC2 ZINC000880961564 DG On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)N1Cc2cccnc2N2C[C@H](O)C[C@H]2C1 ZINC000880961566 GE On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCSCC2)CC1 ZINC000880961571 FI On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCCC2=O)C1 ZINC000880961572 FG On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCCC2=O)C1 ZINC000880961573 FG On-Demand Anodyne RBP4 56 41 CN1Cc2ccccc2[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961574 FG On-Demand Anodyne TRPV1 21 43 CN1Cc2ccccc2[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961574 FG On-Demand Anodyne ABL2 42 34 CN1Cc2ccccc2[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961574 FG On-Demand Anodyne RBP4 48 38 CN1Cc2ccccc2[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961575 FG On-Demand Anodyne TRPV1 21 43 CN1Cc2ccccc2[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961575 FG On-Demand Anodyne ABL2 42 34 CN1Cc2ccccc2[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961575 FG On-Demand Anodyne RBP4 48 38 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCCCO1 ZINC000880961578 EH On-Demand Anodyne TRPV1 20 42 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCCCO1 ZINC000880961579 EH On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880961581 FH On-Demand Anodyne EPHX2 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880961581 FH On-Demand Anodyne RBP4 70 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880961582 FH On-Demand Anodyne EPHX2 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880961582 FH On-Demand Anodyne RBP4 70 44 O=C(NCCOC(F)(F)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880961583 FG On-Demand Mild TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880961590 GH On-Demand Anodyne EPHX2 27 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880961590 GH On-Demand Anodyne RBP4 64 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880961591 GH On-Demand Anodyne EPHX2 27 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880961591 GH On-Demand Anodyne RBP4 64 42 COc1ccccc1[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880961600 GH On-Demand Anodyne RBP4 92 46 CS[C@@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961602 DG On-Demand Anodyne EPHX2 23 40 C=CC[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961603 CH On-Demand Mild RBP4 72 43 C=CC[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961604 CH On-Demand Mild RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CC[C@H](C1)O2 ZINC000880961605 DE On-Demand Anodyne RBP4 85 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCNC2=O)CC1 ZINC000880961606 EE On-Demand Anodyne RBP4 55 39 COC(=O)[C@@]1(C)CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880961607 EF On-Demand Anodyne RBP4 55 40 CCOC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCC1(F)F ZINC000880961610 GG On-Demand Anodyne RBP4 56 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COC[C@H]1O ZINC000880961614 CC On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1CC1(CC1)C2 ZINC000880961615 EI On-Demand Anodyne RBP4 40 38 COC[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880961618 DF On-Demand Anodyne RBP4 40 36 CCC(F)(F)C(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961619 EI On-Demand Anodyne TRPV1 19 46 CONC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961620 EE On-Demand Anodyne RBP4 68 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880961623 GD On-Demand Anodyne RBP4 88 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(F)(F)F)C1 ZINC000880961625 EH On-Demand Anodyne RBP4 68 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(F)(F)F)C1 ZINC000880961626 EH On-Demand Anodyne RBP4 68 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](C(F)F)C1 ZINC000880961627 EF On-Demand Anodyne RBP4 75 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](C(F)F)C1 ZINC000880961628 EF On-Demand Anodyne RBP4 75 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2)CC1 ZINC000880961630 FH On-Demand Anodyne TRPV1 25 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2)CC1 ZINC000880961630 FH On-Demand Anodyne RBP4 59 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2)CC1 ZINC000880961630 FH On-Demand Anodyne MLYCD 17 41 O=C(NC[C@@H]1CCO[C@H]1c1cn[nH]c1)Nc1cnccc1C(F)(F)F ZINC000880961632 FF On-Demand Anodyne TRPV1 15 43 Cn1ncc(NC(=O)Nc2cnccc2C(F)(F)F)c1C1CC1 ZINC000880961633 EG On-Demand Anodyne FLT1 17 45 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961637 GH On-Demand Anodyne RBP4 65 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961637 GH On-Demand Anodyne SFRP1 43 35 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961637 GH On-Demand Anodyne WNT3 40 32 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961638 GH On-Demand Anodyne RBP4 65 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961638 GH On-Demand Anodyne SFRP1 43 35 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961638 GH On-Demand Anodyne WNT3 40 32 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961639 GH On-Demand Anodyne RBP4 65 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961639 GH On-Demand Anodyne SFRP1 43 35 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1C(=O)OC(C)(C)C ZINC000880961639 GH On-Demand Anodyne WNT3 40 32 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961640 GH On-Demand Anodyne RBP4 65 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961640 GH On-Demand Anodyne SFRP1 43 35 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C(=O)OC(C)(C)C ZINC000880961640 GH On-Demand Anodyne WNT3 40 32 O=C(Nc1cnccc1C(F)(F)F)N1CCc2nc(C3CC3)ncc2C1 ZINC000880961643 FG On-Demand Anodyne RBP4 55 39 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCC1(C)C ZINC000880961646 EG On-Demand Anodyne RBP4 60 42 COc1ccc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)cc1 ZINC000880961648 GH On-Demand Anodyne RBP4 57 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CC1)CC2 ZINC000880961651 DH On-Demand Anodyne RBP4 58 41 Cc1csc([C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880961652 FH On-Demand Anodyne RBP4 72 42 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)C(=O)N1CCCC1 ZINC000880961654 FF On-Demand Anodyne TRPV1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880961657 FI On-Demand Anodyne NPY5R 36 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880961657 FI On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880961658 FI On-Demand Anodyne NPY5R 36 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880961658 FI On-Demand Anodyne RBP4 58 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc2c(c1)OCO2 ZINC000880961659 FC On-Demand Anodyne EPHX2 21 51 C[C@@H]1CC[C@H](O)[C@H]([C@H]2CCCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961661 GI On-Demand Anodyne RBP4 47 39 C[C@@H]1CC[C@H](O)[C@@H]([C@H]2CCCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961662 GI On-Demand Anodyne RBP4 47 39 C[C@@H]1CC[C@H](O)[C@@H]([C@@H]2CCCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961663 GI On-Demand Anodyne RBP4 47 39 C[C@@H]1CC[C@H](O)[C@H]([C@@H]2CCCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961664 GI On-Demand Anodyne RBP4 47 39 Cc1cccc2c1OCC[C@@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961673 FI On-Demand Anodyne TRPV1 42 59 CCC1(N2CCCC2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961674 FH On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](CCF)C1 ZINC000880961679 DF On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](CCF)C1 ZINC000880961680 DF On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CC(O)(c2ccc(F)cc2)C1 ZINC000880961681 FF On-Demand Anodyne RBP4 48 39 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961689 GH On-Demand Anodyne RBP4 58 41 CCC1(N(C)C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961690 EG On-Demand Anodyne RBP4 63 41 O=C(Nc1cnccc1C(F)(F)F)NC1CN(c2ccncn2)C1 ZINC000880961691 ED On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)NC1CN(c2ccncn2)C1 ZINC000880961691 ED On-Demand Anodyne EPHX2 17 40 CS(=O)(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961694 FD On-Demand Anodyne RBP4 66 42 CS(=O)(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961694 FD On-Demand Anodyne SFRP1 118 37 CS(=O)(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961694 FD On-Demand Anodyne WNT3 82 36 CS(=O)(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961695 FD On-Demand Anodyne RBP4 66 42 CS(=O)(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961695 FD On-Demand Anodyne SFRP1 118 37 CS(=O)(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961695 FD On-Demand Anodyne WNT3 82 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CC[C@@H](C1)[S@@]2=O ZINC000880961703 EF On-Demand Anodyne RBP4 69 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CC[C@@H](C1)[S@]2=O ZINC000880961704 EF On-Demand Anodyne RBP4 69 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC12CCC2 ZINC000880961705 CG On-Demand Anodyne TRPV1 16 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC12CCC2 ZINC000880961706 CG On-Demand Anodyne TRPV1 16 40 CN1CCN(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CC1 ZINC000880961709 FE On-Demand Anodyne RBP4 68 41 CN1CCN(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CC1 ZINC000880961709 FE On-Demand Anodyne L3MBTL3 54 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C(N)=O)O1 ZINC000880961712 ED On-Demand Anodyne RBP4 66 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C(N)=O)O1 ZINC000880961713 ED On-Demand Anodyne RBP4 66 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C(N)=O)O1 ZINC000880961714 ED On-Demand Anodyne RBP4 66 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C(N)=O)O1 ZINC000880961715 ED On-Demand Anodyne RBP4 66 43 CCO[C@@]1(C)C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961718 DF On-Demand Anodyne TRPV1 21 40 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccncc1 ZINC000880961719 DG On-Demand Anodyne TRPV1 20 53 O=C(Nc1cnccc1C(F)(F)F)N1CCC(F)(F)CC1 ZINC000880961721 DG On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(F)(F)CC1 ZINC000880961721 DG On-Demand Anodyne RBP4 61 44 O=C(NCc1ccc(CN2CCNC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880961729 GF On-Demand Anodyne TRPV1 18 49 O=C(NCc1ccc(CN2CCNC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880961729 GF On-Demand Anodyne NAMPT 65 39 Cn1cncc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961737 CE On-Demand Anodyne TRPV1 19 49 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961738 GI On-Demand Anodyne SLC18A2 43 31 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961738 GI On-Demand Anodyne RBP4 39 41 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961739 GI On-Demand Anodyne SLC18A2 43 31 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880961739 GI On-Demand Anodyne RBP4 39 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000880961743 GG On-Demand Anodyne SFRP1 109 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](S(=O)(=O)c2ccccc2)C1 ZINC000880961743 GG On-Demand Anodyne WNT3 72 34 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2COC[C@H]2C1 ZINC000880961745 DE On-Demand Anodyne RBP4 85 52 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1C1CC1 ZINC000880961746 DE On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1C1CC1 ZINC000880961747 DE On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1C1CC1 ZINC000880961748 DE On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1C1CC1 ZINC000880961749 DE On-Demand Anodyne RBP4 62 42 COC(=O)Cc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961750 FD On-Demand Anodyne GRIN2B 85 43 COC(=O)Cc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961750 FD On-Demand Anodyne SIGMAR1 23 42 COC(=O)Cc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880961750 FD On-Demand Anodyne CCR3 37 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880961751 GH On-Demand Anodyne TRPV1 27 52 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880961751 GH On-Demand Anodyne RIPK1 40 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880961752 GH On-Demand Anodyne TRPV1 27 52 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)c1cccc(C(F)(F)F)c1 ZINC000880961752 GH On-Demand Anodyne RIPK1 40 35 O=C(NCCO)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961754 FD On-Demand Anodyne RBP4 65 40 O=C(Cn1cc([C@@H](O)C2CC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961756 FE On-Demand Anodyne GRIN2B 77 44 O=C(Cn1cc([C@H](O)C2CC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961757 FE On-Demand Anodyne GRIN2B 77 44 C[C@@H](O)C1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961760 CE On-Demand Anodyne TRPV1 15 41 C[C@@H](Cc1ccccn1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961770 DG On-Demand Anodyne TRPV1 20 45 C[C@H](Cc1ccccn1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961772 DG On-Demand Anodyne TRPV1 20 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](C(F)(F)F)CC1 ZINC000880961773 FG On-Demand Anodyne RBP4 72 43 CC[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961774 CD On-Demand Anodyne TRPV1 22 47 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](C(F)(F)F)CC1 ZINC000880961775 FG On-Demand Anodyne RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C2CCC2)C1 ZINC000880961776 EI On-Demand Anodyne RBP4 90 50 O=C(NCc1cc2c(nc1O)CCCC2)Nc1cnccc1C(F)(F)F ZINC000880961777 FG On-Demand Anodyne TRPV1 25 50 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C2CCC2)C1 ZINC000880961778 EI On-Demand Anodyne RBP4 90 50 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961780 FH On-Demand Anodyne TRPV1 23 41 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961780 FH On-Demand Anodyne RAF1 18 41 COc1ccccc1[C@@H]1C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961780 FH On-Demand Anodyne RBP4 46 38 O=C1CCC2=C(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)N1 ZINC000880961784 EF On-Demand Anodyne RBP4 47 38 O=C(NC[C@@H]1CC[C@@H]2C[C@H]2C1)Nc1cnccc1C(F)(F)F ZINC000880961787 DH On-Demand Anodyne TRPV1 18 45 O=C(NC[C@@H]1CC[C@@H]2C[C@@H]2C1)Nc1cnccc1C(F)(F)F ZINC000880961789 DH On-Demand Anodyne TRPV1 18 45 O=C(NC[C@@H]1CC[C@H]2C[C@H]2C1)Nc1cnccc1C(F)(F)F ZINC000880961791 DH On-Demand Anodyne TRPV1 18 45 O=C(NC[C@@H]1CC[C@H]2C[C@@H]2C1)Nc1cnccc1C(F)(F)F ZINC000880961793 DH On-Demand Anodyne TRPV1 18 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CC[C@@H](C1)S2 ZINC000880961794 EH On-Demand Anodyne RBP4 73 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H](O)C1 ZINC000880961807 CD On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H](O)C1 ZINC000880961807 CD On-Demand Anodyne EPHX2 33 43 C#C[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961809 CD On-Demand Mild TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880961810 GI On-Demand Anodyne RBP4 66 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880961810 GI On-Demand Anodyne SMO 41 54 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880961810 GI On-Demand Anodyne ETHR 66 49 C[C@@](CO)(Cc1ccccc1F)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961811 FG On-Demand Anodyne TRPV1 15 44 C#C[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880961818 CD On-Demand Mild TRPV1 17 43 C#CC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961820 DG On-Demand Mild RBP4 81 46 C#CC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961822 DG On-Demand Mild RBP4 81 46 O=C(NC/C=C/CO)Nc1cnccc1C(F)(F)F ZINC000880961827 CD On-Demand Anodyne TRPV1 20 47 O=C(NC/C=C\CO)Nc1cnccc1C(F)(F)F ZINC000880961828 CD On-Demand Anodyne TRPV1 20 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne EPHX2 39 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne RBP4 95 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne SCD1 31 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne SFRP1 111 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne SCD 27 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccc2)C1 ZINC000880961831 FH On-Demand Anodyne WNT3 80 35 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)C[C@H]1Br ZINC000880961833 FG On-Demand Reactive TRPV1 26 47 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1Br ZINC000880961835 FG On-Demand Reactive TRPV1 26 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1C(F)(F)F ZINC000880961836 DG On-Demand Anodyne RBP4 59 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1C(F)(F)F ZINC000880961837 DG On-Demand Anodyne RBP4 59 41 CC(C)(C)N1C[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880961838 FF On-Demand Anodyne TRPV1 15 40 CC(C)(C)N1C[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880961839 FF On-Demand Anodyne TRPV1 15 40 O=C(Cn1cc(-c2ccc(F)nc2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961840 GF On-Demand Anodyne GRIN2B 75 42 Cn1ncc(C2CC2)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961842 EG On-Demand Anodyne TRPV1 20 42 O=C(NCC[C@@H]1CC1(F)F)Nc1cnccc1C(F)(F)F ZINC000880961844 DG On-Demand Anodyne TRPV1 19 47 O=C(NCC[C@H]1CC1(F)F)Nc1cnccc1C(F)(F)F ZINC000880961845 DG On-Demand Anodyne TRPV1 19 47 O=C(NC[C@H]1CCCN(CC2CC2)C1)Nc1cnccc1C(F)(F)F ZINC000880961856 FG On-Demand Anodyne CCR3 76 38 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H](CO)Cc1ccccc1 ZINC000880961858 FG On-Demand Anodyne TRPV1 15 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H](CO)Cc1ccccc1 ZINC000880961858 FG On-Demand Anodyne NPY5R 28 45 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H](CO)Cc1ccccc1 ZINC000880961858 FG On-Demand Anodyne GPR142 57 34 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H](CO)Cc1ccccc1 ZINC000880961859 FG On-Demand Anodyne TRPV1 15 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H](CO)Cc1ccccc1 ZINC000880961859 FG On-Demand Anodyne NPY5R 28 45 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H](CO)Cc1ccccc1 ZINC000880961859 FG On-Demand Anodyne GPR142 57 34 O=C(NCCO[C@@H]1CC1(F)F)Nc1cnccc1C(F)(F)F ZINC000880961862 EF On-Demand Anodyne TRPV1 16 44 O=C(NCCO[C@H]1CC1(F)F)Nc1cnccc1C(F)(F)F ZINC000880961863 EF On-Demand Anodyne TRPV1 16 44 CN(C)S(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961872 GD On-Demand Anodyne RBP4 65 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](F)C1 ZINC000880961873 CG On-Demand Anodyne RBP4 72 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](F)C1 ZINC000880961873 CG On-Demand Anodyne SFRP1 70 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](F)C1 ZINC000880961873 CG On-Demand Anodyne WNT3 61 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](F)C1 ZINC000880961874 CG On-Demand Anodyne RBP4 72 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](F)C1 ZINC000880961874 CG On-Demand Anodyne SFRP1 70 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](F)C1 ZINC000880961874 CG On-Demand Anodyne WNT3 61 34 O=C(Nc1cnccc1C(F)(F)F)N(CCN1CCOCC1)CC1CC1 ZINC000880961875 FF On-Demand Anodyne CASR 57 47 O=C(NC[C@@H]1CCN1Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961878 FG On-Demand Anodyne TRPV1 24 43 O=C(NC[C@@H]1CCN1Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961878 FG On-Demand Anodyne RBP4 49 39 O=C(NC[C@H]1CCN1Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961879 FG On-Demand Anodyne TRPV1 24 43 O=C(NC[C@H]1CCN1Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961879 FG On-Demand Anodyne RBP4 49 39 CC1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnccc1C(F)(F)F ZINC000880961884 DH On-Demand Anodyne RBP4 48 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1Cc1ccccc1 ZINC000880961889 FH On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1Cc1ccccc1 ZINC000880961890 FH On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CCF)C1 ZINC000880961891 DH On-Demand Anodyne RBP4 76 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CCF)C1 ZINC000880961892 DH On-Demand Anodyne RBP4 76 46 CN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880961896 DD On-Demand Anodyne TRPV1 25 40 O=C(NCCN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961900 DD On-Demand Anodyne TRPV1 16 41 O=C(NCCN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961900 DD On-Demand Anodyne CCR3 19 45 O=C(NCCN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961901 DD On-Demand Anodyne TRPV1 16 41 O=C(NCCN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880961901 DD On-Demand Anodyne CCR3 19 45 COCC(C)(C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961906 DG On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H]2C[C@@H]2C1 ZINC000880961909 CG On-Demand Anodyne EPHX2 35 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H]2C[C@H]2C1 ZINC000880961910 CG On-Demand Anodyne EPHX2 35 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H]2C[C@H]2C1 ZINC000880961911 CG On-Demand Anodyne EPHX2 35 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H]2C[C@@H]2C1 ZINC000880961912 CG On-Demand Anodyne EPHX2 35 44 O=C(NCCCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880961913 DH On-Demand Anodyne TRPV1 25 47 O=C(NCCCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880961913 DH On-Demand Anodyne CCR3 18 44 C[C@]1(NC(=O)C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961920 GF On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2cccc(F)c2)C1 ZINC000880961921 FH On-Demand Anodyne EPHX2 25 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2cccc(F)c2)C1 ZINC000880961921 FH On-Demand Anodyne RBP4 67 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2cccc(F)c2)C1 ZINC000880961922 FH On-Demand Anodyne EPHX2 25 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2cccc(F)c2)C1 ZINC000880961922 FH On-Demand Anodyne RBP4 67 42 CCC1(N2CCOCC2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961923 GG On-Demand Anodyne RBP4 45 37 O=C(NC[C@H]1CCC12CCOCC2)Nc1cnccc1C(F)(F)F ZINC000880961924 EG On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2cc(F)ccc2C1 ZINC000880961926 FH On-Demand Anodyne RBP4 47 37 CS(=O)(=O)NC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961929 EC On-Demand Anodyne RBP4 78 45 CS(=O)(=O)NC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961929 EC On-Demand Anodyne SFRP1 44 34 COC(=O)c1oc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1C ZINC000880961930 FG On-Demand Anodyne TRPV1 21 47 O=C(NC[C@H]1CC2(CCOCC2)CO1)Nc1cnccc1C(F)(F)F ZINC000880961931 FF On-Demand Anodyne TRPV1 18 41 O=C(NC[C@@H]1CC2(CCOCC2)CO1)Nc1cnccc1C(F)(F)F ZINC000880961932 FF On-Demand Anodyne TRPV1 18 41 O=C(NCC[C@@H](O)COCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880961933 GG On-Demand Anodyne TRPV1 16 44 O=C(Cn1cc(C2(O)CCCCC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961934 GF On-Demand Anodyne GRIN2B 74 43 C[C@@]1(CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]1(C)CO ZINC000880961935 ED On-Demand Anodyne TRPV1 16 41 C[C@@]1(CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]1(C)CO ZINC000880961935 ED On-Demand Anodyne RBP4 66 43 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H]2C[C@@H]2C1 ZINC000880961937 DH On-Demand Anodyne TRPV1 19 46 CCn1ncc(NC(=O)Nc2cnccc2C(F)(F)F)c1C ZINC000880961940 DG On-Demand Anodyne TRPV1 17 41 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1CC(CCO)C2 ZINC000880961941 EG On-Demand Anodyne RBP4 45 38 C[C@@H]1CC(F)(F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880961942 DH On-Demand Anodyne RBP4 41 38 C[C@H]1CC(F)(F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880961943 DH On-Demand Anodyne RBP4 41 38 O=C(Nc1cnn(CCF)c1)Nc1cnccc1C(F)(F)F ZINC000880961947 DF On-Demand Anodyne TRPV1 19 44 Cc1nonc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880961948 DE On-Demand Anodyne TRPV1 19 48 C[S@](=N)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961958 FD On-Demand Anodyne RBP4 69 47 C[S@](=N)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961958 FD On-Demand Anodyne SFRP1 47 34 CC(C)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880961960 EF On-Demand Anodyne RBP4 67 44 N#Cc1cc(F)ccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961966 GG On-Demand Mild NPY2R 29 42 N#Cc1cc(F)ccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961966 GG On-Demand Mild RBP4 53 37 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880961967 EH On-Demand Anodyne TRPV1 17 44 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880961967 EH On-Demand Anodyne ROCK2 21 40 O=C(Cn1cc(CC2(O)CCOCC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961968 GD On-Demand Anodyne GRIN2B 65 41 N#C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C1CC1 ZINC000880961969 EE On-Demand Mild RBP4 67 44 N#C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C1CC1 ZINC000880961970 EE On-Demand Mild RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCF)CC1 ZINC000880961971 DH On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCF)CC1 ZINC000880961971 DH On-Demand Anodyne EPHX2 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCF)CC1 ZINC000880961971 DH On-Demand Anodyne RBP4 81 46 C#CCNS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880961973 GC On-Demand Mild RBP4 60 43 COC(=O)C1(O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880961974 DC On-Demand Anodyne RBP4 54 40 NC(=O)Cc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880961977 GF On-Demand Anodyne RBP4 54 40 O=C(Cn1cc(-c2cccnc2F)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880961978 GF On-Demand Anodyne GRIN2B 78 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880961985 FH On-Demand Anodyne TRPV1 26 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@H]1c1ccccc1 ZINC000880961985 FH On-Demand Anodyne RBP4 40 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(CO)CC1 ZINC000880961986 ED On-Demand Anodyne RBP4 65 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccc(F)cc1 ZINC000880961987 EH On-Demand Anodyne TRPV1 18 40 O=C(NCc1cccc2c1CCOC2)Nc1cnccc1C(F)(F)F ZINC000880961993 FG On-Demand Anodyne TRPV1 30 53 O=C(NCCC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880961994 CG On-Demand Anodyne TRPV1 24 46 O=C(NCCSCCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962077 FH On-Demand Anodyne TRPV1 15 45 N#CCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962078 EE On-Demand Mild RBP4 54 39 O=C(Cn1cc(C2(O)CCC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962080 FE On-Demand Anodyne GRIN2B 75 44 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962081 FI On-Demand Anodyne TRPV1 16 41 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962081 FI On-Demand Anodyne RBP4 47 37 C[C@H]1c2ccc(F)cc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962081 FI On-Demand Anodyne TRPM8 46 47 O=C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCCCCCN1 ZINC000880962088 FG On-Demand Anodyne RBP4 53 39 O=C(NCC[C@@H](O)C1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880962090 EG On-Demand Anodyne TRPV1 15 43 O=C(NCC[C@H](O)C1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880962091 EG On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@H](O)C[C@H]1C2 ZINC000880962094 DE On-Demand Anodyne RBP4 53 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@@H](O)C[C@H]1C2 ZINC000880962095 DE On-Demand Anodyne RBP4 53 40 COc1ccc([C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)cc1F ZINC000880962096 GI On-Demand Anodyne RBP4 76 50 CC(C)c1cc([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n[nH]1 ZINC000880962098 GI On-Demand Anodyne RBP4 68 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)[C@H](Oc2ccccc2)C1 ZINC000880962102 FF On-Demand Anodyne RBP4 87 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880962108 GH On-Demand Anodyne TRPV1 19 52 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc3[nH]ccc23)CC1 ZINC000880962108 GH On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC(F)(F)CC1 ZINC000880962115 DH On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880962118 GI On-Demand Anodyne TRPV1 18 53 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)c1ccc(Cl)c(F)c1 ZINC000880962119 GI On-Demand Anodyne TRPV1 18 53 CCOC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962129 EE On-Demand Anodyne RBP4 59 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880962131 FH On-Demand Anodyne EPHX2 40 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880962131 FH On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880962131 FH On-Demand Anodyne LIPG 28 45 CCN1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880962132 DD On-Demand Anodyne TRPV1 25 40 CCN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880962133 DD On-Demand Anodyne TRPV1 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@H](O)c1ccccc1 ZINC000880962134 GI On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@H](O)c1ccccc1 ZINC000880962134 GI On-Demand Anodyne SFRP1 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@H](O)c1ccccc1 ZINC000880962134 GI On-Demand Anodyne WNT3 55 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880962135 GI On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880962135 GI On-Demand Anodyne SFRP1 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@H](O)c1ccccc1 ZINC000880962135 GI On-Demand Anodyne WNT3 55 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880962136 GI On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880962136 GI On-Demand Anodyne SFRP1 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1[C@@H](O)c1ccccc1 ZINC000880962136 GI On-Demand Anodyne WNT3 55 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880962137 GI On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880962137 GI On-Demand Anodyne SFRP1 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1[C@@H](O)c1ccccc1 ZINC000880962137 GI On-Demand Anodyne WNT3 55 35 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880962139 EI On-Demand Anodyne RBP4 93 49 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880962140 EI On-Demand Anodyne RBP4 93 49 COc1ccccc1[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962147 EH On-Demand Anodyne TRPV1 16 49 CC(C)(C)OC(=O)CCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962150 FH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N(C1CC1)C1CC1 ZINC000880962151 CG On-Demand Anodyne TRPV1 21 40 COc1ccc(OC)c([C@H](O)[C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880962154 GG On-Demand Anodyne RAF1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](CO)C1 ZINC000880962157 CD On-Demand Anodyne TRPV1 21 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](CO)C1 ZINC000880962157 CD On-Demand Anodyne EPHX2 25 41 O=C(NC[C@H]1CCCC12CC2)Nc1cnccc1C(F)(F)F ZINC000880962161 DH On-Demand Anodyne TRPV1 17 45 Cc1cccc2c1CCN2C(=O)Nc1cnccc1C(F)(F)F ZINC000880962163 DI On-Demand Anodyne HTR2C 15 47 Cc1cccc2c1CCN2C(=O)Nc1cnccc1C(F)(F)F ZINC000880962163 DI On-Demand Anodyne TRPV1 26 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2ccccc2)C1 ZINC000880962166 DH On-Demand Anodyne TRPV1 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2ccccc2)C1 ZINC000880962166 DH On-Demand Anodyne RBP4 103 56 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2ccccc2)C1 ZINC000880962166 DH On-Demand Anodyne SMO 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCO)(CCO)CC1 ZINC000880962170 FE On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880962176 EG On-Demand Anodyne RBP4 88 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880962177 EG On-Demand Anodyne RBP4 88 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CSC[C@H]2C1 ZINC000880962178 EG On-Demand Anodyne RBP4 88 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880962179 EG On-Demand Anodyne RBP4 88 48 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2nc(C3CC3)no2)O1 ZINC000880962180 GG On-Demand Anodyne RBP4 54 39 CN1CC[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@@H]21 ZINC000880962183 EF On-Demand Anodyne RBP4 88 47 CN1CC[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@H]21 ZINC000880962184 EF On-Demand Anodyne RBP4 88 47 O=C(NNCC(F)(F)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962188 FF On-Demand Reactive TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880962193 GF On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880962193 GF On-Demand Anodyne SMO 30 48 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880962193 GF On-Demand Anodyne ETHR 59 37 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880962194 GF On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880962194 GF On-Demand Anodyne SMO 30 48 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880962194 GF On-Demand Anodyne ETHR 59 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)[C@H](n2ccnn2)C1 ZINC000880962195 ED On-Demand Anodyne RBP4 58 42 N#CCc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962198 FH On-Demand Mild RBP4 54 39 N#CCc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962198 FH On-Demand Mild P2RY14 44 38 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc3c(c2)OCO3)nn1 ZINC000880962199 DD On-Demand Mild DYRK2 49 34 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc3c(c2)OCO3)nn1 ZINC000880962200 DD On-Demand Mild DYRK2 49 34 C[C@]1(C(F)(F)F)CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962203 FG On-Demand Anodyne RBP4 54 39 CC[C@H](O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880962209 EE On-Demand Anodyne GRIN2B 79 44 CC[C@H](O)c1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880962209 EE On-Demand Anodyne GRIN2C 18 40 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)c1ccccc1 ZINC000880962211 FH On-Demand Anodyne TRPV1 18 49 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)c1ccccc1 ZINC000880962212 FH On-Demand Anodyne TRPV1 18 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880962214 FD On-Demand Anodyne RBP4 87 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880962215 FD On-Demand Anodyne RBP4 87 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880962216 FD On-Demand Anodyne RBP4 87 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880962217 FD On-Demand Anodyne RBP4 87 48 O=C1OC[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]12 ZINC000880962226 DD On-Demand Anodyne RBP4 73 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cn1ccnc1 ZINC000880962227 EF On-Demand Anodyne RBP4 40 37 Cn1ncc(Br)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962228 GF On-Demand Anodyne HTR2A 20 43 Cn1ncc(Br)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962228 GF On-Demand Anodyne TRPV1 18 48 Cn1ncc(Br)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962228 GF On-Demand Anodyne P2RX7 18 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880962229 DH On-Demand Anodyne RBP4 85 52 O=C(Cn1cc(CCCCCCO)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962230 GF On-Demand Anodyne GRIN2B 78 44 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962231 FG On-Demand Anodyne EPHX2 45 42 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962231 FG On-Demand Anodyne GPR119 43 42 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962231 FG On-Demand Anodyne SFRP1 123 45 CC(C)(C)OC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962231 FG On-Demand Anodyne WNT3 84 40 O=C(Cn1cc(C2(O)CCOCC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962232 GD On-Demand Anodyne GRIN2B 74 42 CC(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962235 DF On-Demand Anodyne RBP4 73 44 CC(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962235 DF On-Demand Anodyne SFRP1 59 33 CC(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962235 DF On-Demand Anodyne WNT3 58 33 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962236 DF On-Demand Anodyne RBP4 73 44 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962236 DF On-Demand Anodyne SFRP1 59 33 CC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962236 DF On-Demand Anodyne WNT3 58 33 N#Cc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962237 GH On-Demand Mild TRPV1 21 42 N#Cc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962237 GH On-Demand Mild EPHX2 40 41 N#Cc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962237 GH On-Demand Mild SFRP1 75 36 NC(=O)C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962244 ED On-Demand Anodyne RBP4 57 42 NC(=O)C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962245 ED On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccco2)C1 ZINC000880962248 EG On-Demand Anodyne RBP4 81 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@H]1c1ccncc1 ZINC000880962254 FG On-Demand Anodyne TRPV1 30 41 CCN(CC)C(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962255 DE On-Demand Anodyne TRPV1 21 47 C[C@@](CO)(Cc1ccc(F)cc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962256 FG On-Demand Anodyne TRPV1 16 43 COc1cccc([C@H](CNC(=O)Nc2cnccc2C(F)(F)F)OC)c1 ZINC000880962258 FH On-Demand Anodyne TRPV1 27 46 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(O)cccc2C1 ZINC000880962265 EG On-Demand Anodyne RBP4 58 43 CC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962266 DF On-Demand Anodyne TRPV1 16 43 CC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962266 DF On-Demand Anodyne RBP4 75 44 CC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962266 DF On-Demand Anodyne SFRP1 61 35 CC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962266 DF On-Demand Anodyne WNT3 50 33 C/C=C\CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962269 CF On-Demand Anodyne TRPV1 23 50 C/C=C/CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962270 CF On-Demand Anodyne TRPV1 23 50 O=C(Nc1cnccc1C(F)(F)F)N1Cc2cccnc2N2CCC[C@H]2C1 ZINC000880962275 GH On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1Cc2cccnc2N2CCC[C@H]2C1 ZINC000880962275 GH On-Demand Anodyne RBP4 60 40 Cc1cncc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880962276 FI On-Demand Anodyne WNT3 40 31 Cc1cncc([C@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880962277 FI On-Demand Anodyne WNT3 40 31 C[C@@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962280 DF On-Demand Anodyne TRPV1 15 41 C[C@@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962280 DF On-Demand Anodyne RBP4 79 43 O=C(Nc1cnccc1C(F)(F)F)N1CCn2ccnc2C1 ZINC000880962288 DE On-Demand Anodyne RBP4 55 40 Cc1ccccc1[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962289 DI On-Demand Anodyne TRPV1 19 53 CCOC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C(F)(F)F ZINC000880962298 GG On-Demand Anodyne RBP4 56 41 CN(C)C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1CN(C)C ZINC000880962299 FE On-Demand Anodyne RBP4 76 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2CC[C@@H](C1)S2(=O)=O ZINC000880962308 FE On-Demand Anodyne RBP4 76 44 Cn1nnnc1C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962310 FE On-Demand Anodyne RBP4 73 42 O=C(Nc1cnccc1C(F)(F)F)N1CCn2ncc(Br)c2C1 ZINC000880962311 GG On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@H]2CCCO2)CC1 ZINC000880962313 FG On-Demand Anodyne RBP4 61 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@@H]2CCCO2)CC1 ZINC000880962314 FG On-Demand Anodyne RBP4 61 39 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1CC(O)(c1ccccc1)C2 ZINC000880962315 GI On-Demand Anodyne RBP4 56 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC12CC2 ZINC000880962316 CH On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC12CC2 ZINC000880962317 CH On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H](c1ccccn1)C1CCC1 ZINC000880962318 FI On-Demand Anodyne TRPV1 16 52 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](c1ccccn1)C1CCC1 ZINC000880962319 FI On-Demand Anodyne TRPV1 16 52 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880962327 GG On-Demand Anodyne RBP4 89 46 COC(=O)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880962328 GG On-Demand Anodyne RBP4 89 46 O=C(Cn1cc([C@]2(O)CCOC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962329 FD On-Demand Anodyne GRIN2B 66 41 O=C(Cn1cc([C@@]2(O)CCOC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962330 FD On-Demand Anodyne GRIN2B 66 41 C[C@H]1CCC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)O1 ZINC000880962331 DG On-Demand Anodyne TRPV1 15 41 O=C(NCCCC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962335 DH On-Demand Anodyne TRPV1 20 44 O=C(NCCCC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962335 DH On-Demand Anodyne CCR3 23 44 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CC[C@@H](C2)C1 ZINC000880962336 CG On-Demand Anodyne RBP4 90 50 CCC(CC)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962339 FG On-Demand Anodyne TRPV1 20 44 CCC(CC)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962339 FG On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@@H]2CCOC2)CC1 ZINC000880962340 EE On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@H]2CCOC2)CC1 ZINC000880962341 EE On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2CCC2)CC1 ZINC000880962342 EI On-Demand Anodyne TRPV1 19 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2CCC2)CC1 ZINC000880962342 EI On-Demand Anodyne RBP4 79 47 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880962343 EF On-Demand Anodyne RBP4 70 42 O=C(NCC1CCC(O)CC1)Nc1cnccc1C(F)(F)F ZINC000880962344 DF On-Demand Anodyne TRPV1 25 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCNC2=O)C1 ZINC000880962345 FE On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCNC2=O)C1 ZINC000880962346 FE On-Demand Anodyne RBP4 58 41 COc1cccc(OC)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962348 FG On-Demand Anodyne TRPV1 33 53 COc1cccc(OC)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962348 FG On-Demand Anodyne RAF1 24 42 COc1cccc(OC)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962348 FG On-Demand Anodyne ROCK2 22 42 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C1(CO)CC1 ZINC000880962351 DE On-Demand Anodyne TRPV1 19 44 CO[C@@](C)(CNC(=O)Nc1cnccc1C(F)(F)F)COCc1ccccc1 ZINC000880962353 GH On-Demand Anodyne TRPV1 18 43 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962355 GF On-Demand Anodyne TRPV1 15 47 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962355 GF On-Demand Anodyne CCR3 31 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962355 GF On-Demand Anodyne MCHR1 28 40 O=C(NCc1ccc(CN2CC[C@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962355 GF On-Demand Anodyne NAMPT 65 39 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962356 GF On-Demand Anodyne TRPV1 15 47 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962356 GF On-Demand Anodyne CCR3 31 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962356 GF On-Demand Anodyne MCHR1 28 40 O=C(NCc1ccc(CN2CC[C@@H](O)C2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962356 GF On-Demand Anodyne NAMPT 65 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2C[C@H]2C1 ZINC000880962361 CF On-Demand Anodyne TRPV1 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2C[C@H]2C1 ZINC000880962361 CF On-Demand Anodyne RBP4 99 56 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2C[C@@H]2C1 ZINC000880962362 CF On-Demand Anodyne TRPV1 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2C[C@@H]2C1 ZINC000880962362 CF On-Demand Anodyne RBP4 99 56 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2C[C@H]2C1 ZINC000880962363 CF On-Demand Anodyne TRPV1 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2C[C@H]2C1 ZINC000880962363 CF On-Demand Anodyne RBP4 99 56 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880962364 CF On-Demand Anodyne TRPV1 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2C[C@@H]2C1 ZINC000880962364 CF On-Demand Anodyne RBP4 99 56 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)C1(F)F ZINC000880962365 EH On-Demand Anodyne RBP4 80 48 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)C1(F)F ZINC000880962366 EH On-Demand Anodyne RBP4 80 48 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)C1(F)F ZINC000880962367 EH On-Demand Anodyne RBP4 80 48 O=C(NOCC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962370 CF On-Demand Anodyne TRPV1 17 40 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962374 FF On-Demand Mild IMDH_CRYPV 25 43 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962375 FF On-Demand Mild IMDH_CRYPV 25 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)C(F)(F)C1 ZINC000880962380 EE On-Demand Anodyne RBP4 67 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](O)C(F)(F)C1 ZINC000880962381 EE On-Demand Anodyne RBP4 67 42 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962389 FG On-Demand Anodyne EPHX2 54 48 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962389 FG On-Demand Anodyne RBP4 43 41 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962389 FG On-Demand Anodyne SFRP1 103 37 CC(C)(C)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962389 FG On-Demand Anodyne WNT3 79 36 COC(=O)[C@@]12CCCC[C@@H]1CN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962394 FG On-Demand Anodyne RBP4 40 37 CCn1nncc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962395 DE On-Demand Anodyne TRPV1 16 47 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880962397 FF On-Demand Anodyne IMDH_CRYPV 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880962401 FF On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCOCC2)CC1 ZINC000880962401 FF On-Demand Anodyne L3MBTL3 57 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880962402 FF On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCOCC2)CC1 ZINC000880962402 FF On-Demand Anodyne L3MBTL3 57 38 COc1ccc(N2CC[C@H](NC(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880962405 GH On-Demand Clean TRPV1 18 44 COc1ccc(N2CC[C@H](NC(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880962405 GH On-Demand Clean EPHX2 46 41 CO[C@@](C)(CO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962407 DD On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COC(=O)C1 ZINC000880962413 CD On-Demand Anodyne EPHX2 18 40 O=C(NCCCc1ccco1)Nc1cnccc1C(F)(F)F ZINC000880962419 DG On-Demand Anodyne TRPV1 15 45 CO[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962420 DD On-Demand Anodyne RBP4 68 43 CO[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962421 DD On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CC[C@@H](O)C2)CC1 ZINC000880962427 FE On-Demand Anodyne RBP4 67 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CC[C@H](O)C2)CC1 ZINC000880962428 FE On-Demand Anodyne RBP4 67 43 Cc1nc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n[nH]1 ZINC000880962429 FD On-Demand Anodyne ABL1 42 36 Cc1nc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n[nH]1 ZINC000880962429 FD On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880962435 GI On-Demand Anodyne EPHX2 30 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880962435 GI On-Demand Anodyne RBP4 68 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cccc(F)c2)CC1 ZINC000880962435 GI On-Demand Anodyne SCD1 39 44 CC(C)(CO)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880962437 FH On-Demand Anodyne TRPV1 20 47 Cc1ccccc1CC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962438 EI On-Demand Anodyne TRPV1 22 42 Cc1ccccc1CC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962438 EI On-Demand Anodyne RBP4 84 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(CO)C1 ZINC000880962441 DD On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](CC(F)(F)F)C1 ZINC000880962443 FG On-Demand Anodyne RBP4 67 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](CC(F)(F)F)C1 ZINC000880962444 FG On-Demand Anodyne RBP4 67 43 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962447 FH On-Demand Anodyne TRPV1 22 51 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962447 FH On-Demand Anodyne ROCK1 21 45 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962447 FH On-Demand Anodyne TAAR1 19 40 COC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962448 FH On-Demand Anodyne TRPV1 22 51 COC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962448 FH On-Demand Anodyne ROCK1 21 45 COC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(OC)c1 ZINC000880962448 FH On-Demand Anodyne TAAR1 19 40 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)CC(F)(F)F ZINC000880962449 EI On-Demand Anodyne TRPV1 21 47 O=C(NCC[C@@H]1CCCOC1)Nc1cnccc1C(F)(F)F ZINC000880962450 DG On-Demand Anodyne TRPV1 15 42 O=C(NCC[C@H]1CCCOC1)Nc1cnccc1C(F)(F)F ZINC000880962451 DG On-Demand Anodyne TRPV1 15 42 C[C@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N(C)C ZINC000880962454 DF On-Demand Anodyne TRPV1 15 44 C[C@@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N(C)C ZINC000880962455 DF On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne NPY5R 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne EPHX2 21 52 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne SCD1 31 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne SCD 38 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCc3ccccc3O2)CC1 ZINC000880962456 GI On-Demand Anodyne TRPM8 45 63 O=C1CCC[C@H](c2cn(CC(=O)N3CCC(Cc4ccccc4)CC3)nn2)C1 ZINC000880962457 GF On-Demand Anodyne GRIN2B 66 41 O=C1CCC[C@@H](c2cn(CC(=O)N3CCC(Cc4ccccc4)CC3)nn2)C1 ZINC000880962458 GF On-Demand Anodyne GRIN2B 66 41 CC1=NO[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962459 DE On-Demand Anodyne TRPV1 15 44 C[C@H](N)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962462 EF On-Demand Anodyne SLC1A1 31 41 C[C@H](N)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962462 EF On-Demand Anodyne SLC1A3 31 41 C[C@H](N)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962462 EF On-Demand Anodyne SLC1A2 38 41 C[C@H](N)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962462 EF On-Demand Anodyne IMDH_CRYPV 27 45 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962463 GF On-Demand Anodyne GRIN2B 65 41 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962464 GF On-Demand Anodyne GRIN2B 65 41 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962465 GE On-Demand Anodyne GRIN2B 65 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(C2CC2)C1 ZINC000880962468 EF On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(C2CC2)C1 ZINC000880962469 EF On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880962477 EG On-Demand Anodyne TRPV1 35 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H](O)c2ccccc21 ZINC000880962477 EG On-Demand Anodyne RBP4 81 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880962478 EG On-Demand Anodyne TRPV1 35 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H](O)c2ccccc21 ZINC000880962478 EG On-Demand Anodyne RBP4 81 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880962479 EG On-Demand Anodyne TRPV1 35 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](O)c2ccccc21 ZINC000880962479 EG On-Demand Anodyne RBP4 81 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880962480 EG On-Demand Anodyne TRPV1 35 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](O)c2ccccc21 ZINC000880962480 EG On-Demand Anodyne RBP4 81 44 C=C[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962481 CD On-Demand Mild TRPV1 17 43 Cc1ncoc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962484 DF On-Demand Anodyne TRPV1 27 50 CC(C)(C)CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962488 FG On-Demand Anodyne TRPV1 17 44 CC(C)(C)CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962488 FG On-Demand Anodyne RBP4 60 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CS(=O)(=O)Cc2ccccc21 ZINC000880962489 GF On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CS(=O)(=O)Cc2ccccc21 ZINC000880962489 GF On-Demand Anodyne RBP4 42 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CS(=O)(=O)Cc2ccccc21 ZINC000880962490 GF On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CS(=O)(=O)Cc2ccccc21 ZINC000880962490 GF On-Demand Anodyne RBP4 42 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCCOC2)C1 ZINC000880962496 EG On-Demand Anodyne RBP4 41 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCCOC2)C1 ZINC000880962497 EG On-Demand Anodyne RBP4 41 38 COc1ccc2c(c1)CN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962498 EH On-Demand Anodyne RBP4 46 37 O=C(NC[C@@H](CO)CC1CC1)Nc1cnccc1C(F)(F)F ZINC000880962501 DF On-Demand Anodyne TRPV1 17 44 O=C(NC[C@H](CO)CC1CC1)Nc1cnccc1C(F)(F)F ZINC000880962502 DF On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccsc2)C1 ZINC000880962503 EH On-Demand Anodyne RBP4 62 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCOCC2)C1 ZINC000880962506 EE On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCOCC2)C1 ZINC000880962507 EE On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H]2CCCCO2)CC1 ZINC000880962508 FH On-Demand Anodyne RBP4 70 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H]2CCCCO2)CC1 ZINC000880962509 FH On-Demand Anodyne RBP4 70 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962511 GE On-Demand Anodyne IMDH_CRYPV 21 42 CCn1ncc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880962512 DE On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]([C@@H]2CCCCO2)C1 ZINC000880962513 FH On-Demand Anodyne RBP4 64 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]([C@H]2CCCCO2)C1 ZINC000880962514 FH On-Demand Anodyne RBP4 64 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]([C@H]2CCCCO2)C1 ZINC000880962515 FH On-Demand Anodyne RBP4 64 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]([C@@H]2CCCCO2)C1 ZINC000880962516 FH On-Demand Anodyne RBP4 64 44 COc1cccc([C@]2(C)CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)c1 ZINC000880962519 GI On-Demand Anodyne RBP4 53 37 O=C(CCn1c(S)nnc1-c1cccs1)N1CC(c2ccccc2)C1 ZINC000880962522 FG On-Demand Anodyne ETHR 48 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Cn2ccnn2)C1 ZINC000880962523 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Cn2ccnn2)C1 ZINC000880962524 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(O)C1=O ZINC000880962526 DD On-Demand Mild RBP4 36 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(O)C1=O ZINC000880962527 DD On-Demand Mild RBP4 36 40 O=C(NCCS(=O)(=O)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962563 FE On-Demand Anodyne TRPV1 16 47 CC(C)(C)OC(=O)C1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962564 GI On-Demand Anodyne RBP4 52 38 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C1CC1 ZINC000880962565 FF On-Demand Anodyne RBP4 72 44 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2ccc(O)cc2C1 ZINC000880962566 FG On-Demand Anodyne RBP4 54 39 O=C(Cn1cc(CN2CCOC2=O)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962570 GD On-Demand Anodyne GRIN2B 58 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOC(C2CC2)(C2CC2)C1 ZINC000880962572 FH On-Demand Anodyne RBP4 57 40 COc1ccc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)cc1F ZINC000880962576 GJ On-Demand Anodyne RBP4 40 41 O=C(NCC(O)(C1CC1)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880962581 EF On-Demand Anodyne TRPV1 22 46 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1NC(=O)C(F)(F)F ZINC000880962592 GG On-Demand Anodyne RBP4 66 42 C[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)CS1(=O)=O ZINC000880962597 FE On-Demand Anodyne EPHX2 27 40 C[C@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)CS1(=O)=O ZINC000880962598 FE On-Demand Anodyne EPHX2 27 40 C[C@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)CS1(=O)=O ZINC000880962599 FE On-Demand Anodyne EPHX2 27 40 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880962603 CG On-Demand Anodyne TRPV1 19 47 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne ACHE 29 46 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne TRPV1 17 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne SIGMAR1 25 43 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne CCR3 54 44 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne MCHR1 30 41 O=C(NCC1CCN(Cc2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962612 GH On-Demand Anodyne CACNA1I 64 43 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962613 EG On-Demand Anodyne TRPV1 22 42 CC(C)(C)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962613 EG On-Demand Anodyne CACNA1I 42 35 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962614 EG On-Demand Anodyne TRPV1 22 42 CC(C)(C)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962614 EG On-Demand Anodyne CACNA1I 42 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2n[nH]cc2C1 ZINC000880962623 EF On-Demand Anodyne RBP4 54 40 O=C(NC[C@H](n1cccn1)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962624 FG On-Demand Anodyne TRPV1 17 44 O=C(NC[C@@H](n1cccn1)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962625 FG On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880962631 GJ On-Demand Anodyne RBP4 57 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880962631 GJ On-Demand Anodyne SFRP1 42 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2O[C@H](c3ccccc3)C[C@@H]21 ZINC000880962631 GJ On-Demand Anodyne WNT3 46 34 O=C(NCc1ccc(N2CCCNC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880962632 GG On-Demand Anodyne NAMPT 49 38 C[C@H]1c2ccccc2OCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962635 FI On-Demand Anodyne RBP4 77 42 N#CC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962636 DG On-Demand Mild RBP4 58 42 N#CC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962637 DG On-Demand Mild RBP4 58 42 O=C(NCCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880962638 CG On-Demand Anodyne TRPV1 27 48 O=C(NCCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880962638 CG On-Demand Anodyne CCR3 22 45 COC(=O)[C@@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962641 DE On-Demand Anodyne EPHX2 32 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)C1 ZINC000880962642 EH On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)C1 ZINC000880962642 EH On-Demand Anodyne SFRP1 43 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC2CCC2)C1 ZINC000880962642 EH On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)C1 ZINC000880962643 EH On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)C1 ZINC000880962643 EH On-Demand Anodyne SFRP1 43 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC2CCC2)C1 ZINC000880962643 EH On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](O)C1 ZINC000880962644 CE On-Demand Anodyne RBP4 78 46 CCO[C@@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962645 DF On-Demand Anodyne EPHX2 40 38 CCC[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)OCC ZINC000880962646 DG On-Demand Anodyne TRPV1 15 42 CCC[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)OCC ZINC000880962647 DG On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(COC2)C1 ZINC000880962650 DE On-Demand Anodyne EPHX2 31 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(COC2)C1 ZINC000880962650 DE On-Demand Anodyne RBP4 56 41 Cc1cncc(CCNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880962653 EF On-Demand Anodyne TRPV1 18 48 CO[C@]1(CO)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962656 EE On-Demand Anodyne RBP4 57 41 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962659 GG On-Demand Anodyne IMDH_CRYPV 30 46 O=C(Nc1cnccc1C(F)(F)F)N1CC(CC2CC2)C1 ZINC000880962661 CG On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(CC2CC2)C1 ZINC000880962661 CG On-Demand Anodyne RBP4 85 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCC2=O)CC1 ZINC000880962662 EG On-Demand Anodyne NPY5R 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCC2=O)CC1 ZINC000880962662 EG On-Demand Anodyne RBP4 57 41 O=C(NC[C@@H]1C[C@H](c2ccccc2)CO1)Nc1cnccc1C(F)(F)F ZINC000880962665 FH On-Demand Anodyne TRPV1 16 45 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCC1=O ZINC000880962666 DD On-Demand Anodyne TRPV1 17 44 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCC1=O ZINC000880962666 DD On-Demand Anodyne RBP4 61 41 CON(C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962667 CD On-Demand Anodyne TRPV1 17 45 Cn1nccc1[C@@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962676 GF On-Demand Anodyne RBP4 64 41 Cn1nccc1[C@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962677 GF On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCNC1=O ZINC000880962678 CD On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCNC1=O ZINC000880962679 CD On-Demand Anodyne TRPV1 26 41 O=C(NCC(Cl)Cl)Nc1cnccc1C(F)(F)F ZINC000880962683 DG On-Demand Reactive TRPV1 23 49 CC1CC(CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962689 CG On-Demand Anodyne TRPV1 27 45 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962690 GG On-Demand Clean TRPV1 21 49 O=C(NCc1ccc(N2CCC(O)CC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962690 GG On-Demand Clean NAMPT 72 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)C1 ZINC000880962691 DH On-Demand Anodyne RBP4 53 41 O=C(NCC1=CCCC1)Nc1cnccc1C(F)(F)F ZINC000880962694 CG On-Demand Anodyne TRPV1 17 52 O=C(Nc1cnccc1C(F)(F)F)N(CC1CC1)CC1CC1 ZINC000880962697 DH On-Demand Anodyne TRPV1 21 42 N#CCC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962699 ED On-Demand Mild RBP4 55 41 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1(F)F ZINC000880962700 DG On-Demand Anodyne TRPV1 28 51 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN2CCCC[C@H]12 ZINC000880962703 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN2CCCC[C@@H]12 ZINC000880962704 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN2CCCC[C@@H]12 ZINC000880962705 EG On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN2CCCC[C@H]12 ZINC000880962706 EG On-Demand Anodyne EPHX2 15 40 O=C(NCC1(O)CCC(F)(F)CC1)Nc1cnccc1C(F)(F)F ZINC000880962707 FG On-Demand Anodyne TRPV1 16 47 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccn1 ZINC000880962708 DG On-Demand Anodyne TRPV1 23 47 O=C(Nc1cnccc1C(F)(F)F)N1CC2CC1(c1ccccc1)C2 ZINC000880962714 EI On-Demand Anodyne RBP4 77 43 NOCc1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880962715 ED On-Demand Anodyne IMDH_CRYPV 26 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@]23CCCC[C@@]2(COC3)C1 ZINC000880962717 FH On-Demand Anodyne RBP4 49 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@]23CCCC[C@]2(COC3)C1 ZINC000880962718 FH On-Demand Anodyne RBP4 49 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@]23CCCC[C@]2(COC3)C1 ZINC000880962719 FH On-Demand Anodyne RBP4 49 39 Cn1ncc(C2CCC2)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962720 FG On-Demand Anodyne TRPV1 17 41 O=C(NCC1SCCS1)Nc1cnccc1C(F)(F)F ZINC000880962726 DG On-Demand Anodyne TRPV1 18 46 O=C(Cn1cc([C@@H]2CCCCO2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962727 FG On-Demand Anodyne GRIN2B 70 42 O=C(Cn1cc([C@H]2CCCCO2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880962728 FG On-Demand Anodyne GRIN2B 70 42 Cc1cnc(CCNC(=O)Nc2cnccc2C(F)(F)F)c(C)c1 ZINC000880962729 EG On-Demand Anodyne TRPV1 15 45 Cc1cnc(CCNC(=O)Nc2cnccc2C(F)(F)F)c(C)c1 ZINC000880962729 EG On-Demand Anodyne RAF1 25 42 O=C(NCCOCCF)Nc1cnccc1C(F)(F)F ZINC000880962732 CE On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nccnn2)CC1 ZINC000880962738 FD On-Demand Anodyne TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nccnn2)CC1 ZINC000880962738 FD On-Demand Anodyne FAAH 22 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nccnn2)CC1 ZINC000880962738 FD On-Demand Anodyne RBP4 55 39 O=C(NCC1CCN(CC2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962739 FG On-Demand Anodyne TRPV1 20 44 O=C(NCC1CCN(CC2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962739 FG On-Demand Anodyne CCR3 45 44 O=C(NCC1CCN(CC2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962739 FG On-Demand Anodyne CACNA1I 61 38 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]1(C)CO ZINC000880962740 DF On-Demand Anodyne RBP4 62 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]1(C)CO ZINC000880962741 DF On-Demand Anodyne RBP4 62 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]1(C)CO ZINC000880962742 DF On-Demand Anodyne RBP4 62 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]1(C)CO ZINC000880962743 DF On-Demand Anodyne RBP4 62 42 C[C@H]1c2ccccc2CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962744 DI On-Demand Anodyne RBP4 83 43 C[C@H]1c2ccccc2CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962744 DI On-Demand Anodyne TRPM8 32 41 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)C(=O)OC(C)(C)C ZINC000880962747 EG On-Demand Anodyne TRPV1 15 43 C[C@H]1c2ccccc2C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962757 EH On-Demand Anodyne TRPV1 33 42 C[C@H]1c2ccccc2C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962757 EH On-Demand Anodyne RBP4 57 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@](C)(C(F)F)O1 ZINC000880962761 FG On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2F)C1 ZINC000880962762 FI On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2F)C1 ZINC000880962762 FI On-Demand Anodyne RBP4 110 53 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2F)C1 ZINC000880962762 FI On-Demand Anodyne SFRP1 47 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2F)C1 ZINC000880962763 FI On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2F)C1 ZINC000880962763 FI On-Demand Anodyne RBP4 110 53 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2F)C1 ZINC000880962763 FI On-Demand Anodyne SFRP1 47 34 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2cccc(C(F)(F)F)c2)C1 ZINC000880962766 GJ On-Demand Anodyne TRPV1 27 45 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2cccc(C(F)(F)F)c2)C1 ZINC000880962766 GJ On-Demand Anodyne CCR2 35 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2cccc(C(F)(F)F)c2)C1 ZINC000880962766 GJ On-Demand Anodyne RBP4 84 47 CNc1ncc(C(=O)N2CC(c3ccccc3)C2)s1 ZINC000880962767 CE On-Demand Anodyne MGEA5 33 43 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCOC2)C1 ZINC000880962768 DE On-Demand Anodyne RBP4 48 39 O=C(NC[C@@H](O)C1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962770 DE On-Demand Anodyne TRPV1 17 44 O=C(NC[C@H](O)C1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962771 DE On-Demand Anodyne TRPV1 17 44 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CCC(=O)N1 ZINC000880962774 DD On-Demand Anodyne TRPV1 16 44 CC(C)(C)C1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962779 DH On-Demand Anodyne RBP4 79 48 CC[C@H]1CN(C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962782 DF On-Demand Anodyne RBP4 53 39 CC[C@@H]1CN(C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962783 DF On-Demand Anodyne RBP4 53 39 CC[C@H](C)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880962788 DG On-Demand Anodyne TRPV1 15 43 CC[C@@H](C)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880962790 DG On-Demand Anodyne TRPV1 15 43 O=C(Nc1ccc([C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962792 FI On-Demand Anodyne TRPV1 18 44 O=C(Nc1ccc([C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962792 FI On-Demand Anodyne PIK3CA 15 40 O=C(Nc1ccc([C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962792 FI On-Demand Anodyne MTOR 40 40 O=C(Nc1ccc([C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962793 FI On-Demand Anodyne TRPV1 18 44 O=C(Nc1ccc([C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962793 FI On-Demand Anodyne PIK3CA 15 40 O=C(Nc1ccc([C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880962793 FI On-Demand Anodyne MTOR 40 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCC(O)CC2)CC1 ZINC000880962796 FH On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](O)C1 ZINC000880962798 CD On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H](O)C1 ZINC000880962798 CD On-Demand Anodyne EPHX2 33 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2ccccc2CC1 ZINC000880962800 EI On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2ccccc2CC1 ZINC000880962800 EI On-Demand Anodyne RBP4 73 45 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2ccccc2CC1 ZINC000880962800 EI On-Demand Anodyne TRPM8 46 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccc(Cl)cc2)C1 ZINC000880962801 GI On-Demand Anodyne RBP4 59 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccc(Cl)cc2)C1 ZINC000880962802 GI On-Demand Anodyne RBP4 59 41 Cc1cnc(CCNC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880962804 EF On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCn2ccnc21 ZINC000880962807 DF On-Demand Anodyne RBP4 37 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCn2ccnc21 ZINC000880962808 DF On-Demand Anodyne RBP4 37 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(C(=O)N2CCCC2)C1 ZINC000880962814 GE On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(C(=O)N2CCCC2)C1 ZINC000880962815 GE On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](C1)[C@H]1C=C[C@H]2CC1 ZINC000880962816 EH On-Demand Anodyne RBP4 86 46 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@H]3C=C[C@@H](CC3)[C@H]2C1 ZINC000880962817 EH On-Demand Anodyne RBP4 86 46 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H]3C=C[C@@H](CC3)[C@H]2C1 ZINC000880962818 EH On-Demand Anodyne RBP4 86 46 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(N)=O ZINC000880962819 CD On-Demand Anodyne TRPV1 16 48 COC[C@]1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962820 DF On-Demand Anodyne RBP4 41 38 COC[C@@]1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962821 DF On-Demand Anodyne RBP4 41 38 O=C(Nc1cnccc1C(F)(F)F)N1CC(C2CCCCC2)C1 ZINC000880962824 EI On-Demand Anodyne RBP4 87 51 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCCc1ccccc12 ZINC000880962828 GI On-Demand Anodyne NPY5R 32 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCCc1ccccc12 ZINC000880962828 GI On-Demand Anodyne RBP4 56 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@](C)(C(F)F)O1 ZINC000880962830 FG On-Demand Anodyne RBP4 53 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@](C)(C(F)F)O1 ZINC000880962831 FG On-Demand Anodyne RBP4 53 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@](C)(C(F)F)O1 ZINC000880962832 FG On-Demand Anodyne RBP4 53 39 Cn1cccc1C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962834 GE On-Demand Anodyne RBP4 63 41 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880962837 GH On-Demand Anodyne IMDH_CRYPV 22 41 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880962838 GH On-Demand Anodyne IMDH_CRYPV 22 41 O=C(NCC1CCN(C2CCOCC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880962839 GG On-Demand Anodyne NAMPT 23 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)[C@@H]1O ZINC000880962840 DF On-Demand Anodyne RBP4 78 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)C1O ZINC000880962841 DF On-Demand Anodyne RBP4 78 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)C1O ZINC000880962842 DF On-Demand Anodyne RBP4 78 47 O=C1CC[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@H]2N1 ZINC000880962843 EE On-Demand Anodyne RBP4 87 50 O=C1CC[C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@@H]2N1 ZINC000880962844 EE On-Demand Anodyne RBP4 87 50 O=C1CC[C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@H]2N1 ZINC000880962845 EE On-Demand Anodyne RBP4 87 50 O=C1CC[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@@H]2N1 ZINC000880962846 EE On-Demand Anodyne RBP4 87 50 CN(C)CCC[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880962847 FF On-Demand Anodyne RBP4 59 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(O)C[C@H]2C1 ZINC000880962855 DE On-Demand Anodyne RBP4 61 44 O=C1CCCN1C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962857 FF On-Demand Anodyne RBP4 57 41 O=C1CCCN1C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962858 FF On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)NN1CCc2ccccc2C1 ZINC000880962859 EG On-Demand Anodyne TRPV1 20 41 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962864 GH On-Demand Anodyne RBP4 57 41 CCSC1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962865 DH On-Demand Anodyne TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(CO)CC1 ZINC000880962866 DD On-Demand Anodyne RBP4 61 43 COCC(COC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880962869 DD On-Demand Anodyne TRPV1 17 45 N#Cc1sccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962870 GG On-Demand Mild RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CC2)c2ccccc21 ZINC000880962874 EI On-Demand Anodyne P2RY1 43 43 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CC2)c2ccccc21 ZINC000880962874 EI On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCC2(CC1)CC2(F)F ZINC000880962875 EI On-Demand Anodyne EPHX2 33 44 C[C@@]12COC[C@H]1CN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962877 DF On-Demand Anodyne RBP4 55 40 C[C@@]12COC[C@@H]1CN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962879 DF On-Demand Anodyne RBP4 55 40 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H](C)O1 ZINC000880962881 DG On-Demand Anodyne RBP4 82 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C[C@H](O)C[C@H]2C1 ZINC000880962882 ED On-Demand Anodyne RBP4 68 46 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962892 DE On-Demand Anodyne RBP4 47 39 C[C@H]1[C@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962892 DE On-Demand Anodyne WNT3 40 31 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962893 DE On-Demand Anodyne RBP4 47 39 C[C@@H]1[C@@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962893 DE On-Demand Anodyne WNT3 40 31 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962894 DE On-Demand Anodyne RBP4 47 39 C[C@H]1[C@@H](O)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962894 DE On-Demand Anodyne WNT3 40 31 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC2CC2)nn1 ZINC000880962901 DD On-Demand Anodyne SIGMAR1 15 42 C=CC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962904 DH On-Demand Mild RBP4 61 42 C=CC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962905 DH On-Demand Mild RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1C1CC1 ZINC000880962906 CG On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1C1CC1 ZINC000880962907 CG On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCCCC2)C1 ZINC000880962910 DH On-Demand Anodyne RBP4 56 41 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NCCc1ccccc1 ZINC000880962914 GF On-Demand Anodyne ANPEP 22 45 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NCCc1ccccc1 ZINC000880962914 GF On-Demand Anodyne TRPV1 24 52 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NCCc1ccccc1 ZINC000880962914 GF On-Demand Anodyne BRS3 21 42 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NCCc1ccccc1 ZINC000880962914 GF On-Demand Anodyne AMP1_PLAFQ 20 40 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880962916 EF On-Demand Anodyne RBP4 55 39 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880962917 EF On-Demand Anodyne RBP4 55 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(=O)N1 ZINC000880962922 DD On-Demand Anodyne RBP4 57 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(=O)N1 ZINC000880962924 DD On-Demand Anodyne RBP4 57 41 CN1C[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880962932 DD On-Demand Anodyne TRPV1 16 42 CN1C[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880962933 DD On-Demand Anodyne TRPV1 16 42 O=C(NCC[C@@H]1CC1(Cl)Cl)Nc1cnccc1C(F)(F)F ZINC000880962934 EH On-Demand Anodyne TRPV1 18 46 O=C(NCC[C@H]1CC1(Cl)Cl)Nc1cnccc1C(F)(F)F ZINC000880962935 EH On-Demand Anodyne TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@@H]2CCOC2)CC1 ZINC000880962937 FE On-Demand Anodyne EPHX2 37 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@H]2CCOC2)CC1 ZINC000880962938 FE On-Demand Anodyne EPHX2 37 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)C1CCC1 ZINC000880962939 DE On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)C1CCC1 ZINC000880962940 DE On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)NC1CC(CO)C1 ZINC000880962941 CD On-Demand Anodyne TRPV1 21 41 O=C(Nc1cnccc1C(F)(F)F)NC1CC(CO)C1 ZINC000880962941 CD On-Demand Anodyne EPHX2 25 41 C[C@H]1CCC(C)(C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880962947 DH On-Demand Anodyne RBP4 42 37 O=C(NCC1(CO)CCCC1)Nc1cnccc1C(F)(F)F ZINC000880962948 DF On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccon2)CC1 ZINC000880962951 EG On-Demand Anodyne RBP4 73 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccon2)CC1 ZINC000880962951 EG On-Demand Anodyne SMO 22 49 CC(C)(C)C(F)(F)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962952 EH On-Demand Anodyne TRPV1 22 48 Cn1cnnc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962953 FD On-Demand Anodyne TRPV1 15 45 Cn1cnnc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880962953 FD On-Demand Anodyne RBP4 53 38 O=C(NCCC1SCCS1)Nc1cnccc1C(F)(F)F ZINC000880962954 EG On-Demand Anodyne TRPV1 16 44 CO[C@@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962957 CE On-Demand Anodyne TRPV1 19 46 O=C(NCC[S@@](=O)CC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962959 FF On-Demand Anodyne TRPV1 15 45 O=C(NCC[S@](=O)CC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880962960 FF On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1C1CCC1 ZINC000880962961 EI On-Demand Anodyne RBP4 55 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(CCS(=O)(=O)C2)C1 ZINC000880962966 GF On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(CCS(=O)(=O)C2)C1 ZINC000880962967 GF On-Demand Anodyne RBP4 40 37 NC(=O)[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962968 DD On-Demand Anodyne TRPV1 18 40 NC(=O)[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880962968 DD On-Demand Anodyne EPHX2 28 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCCCCCC1 ZINC000880962969 DI On-Demand Anodyne TRPV1 19 47 O=C(Nc1cnccc1C(F)(F)F)N1CCCCCCCC1 ZINC000880962969 DI On-Demand Anodyne RBP4 69 46 O=C(NOC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880962970 CF On-Demand Anodyne TRPV1 20 42 O=C(Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CC1 ZINC000880962971 ED On-Demand Anodyne CCR2 68 42 O=C(Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CC1 ZINC000880962972 ED On-Demand Anodyne CCR2 68 42 Cc1ncsc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962974 EG On-Demand Anodyne RAF1 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CO)CC1 ZINC000880962976 DF On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CO)CC1 ZINC000880962976 DF On-Demand Anodyne SFRP1 47 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CO)CC1 ZINC000880962976 DF On-Demand Anodyne WNT3 47 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CO)CC1 ZINC000880962977 DF On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CO)CC1 ZINC000880962977 DF On-Demand Anodyne SFRP1 47 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CO)CC1 ZINC000880962977 DF On-Demand Anodyne WNT3 47 33 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962982 EF On-Demand Anodyne EPHX2 33 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880962982 EF On-Demand Anodyne GLRA1 43 39 O=C(NC[C@H](O)Cc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880962983 FF On-Demand Anodyne TRPV1 26 53 O=C(NC[C@@H](O)Cc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880962984 FF On-Demand Anodyne TRPV1 26 53 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880962988 GG On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880962988 GG On-Demand Anodyne RBP4 81 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880962989 GG On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](c2ccccc2)[C@](F)(CO)C1 ZINC000880962989 GG On-Demand Anodyne RBP4 81 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880962990 GG On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](c2ccccc2)[C@@](F)(CO)C1 ZINC000880962990 GG On-Demand Anodyne RBP4 81 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC2CCCCC2)CC1 ZINC000880962991 FI On-Demand Anodyne RBP4 72 43 CC/C=C\CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962994 CG On-Demand Anodyne TRPV1 21 47 CC/C=C/CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880962995 CG On-Demand Anodyne TRPV1 21 47 O=C(NCC#CCO)Nc1cnccc1C(F)(F)F ZINC000880962996 CD On-Demand Mild TRPV1 23 49 CN(C)CC(C)(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963000 DF On-Demand Anodyne TRPV1 17 45 CCNC(=O)C(C)(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963001 DE On-Demand Anodyne TRPV1 18 44 CCC1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963003 CG On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)NC12CCC(CC1)CC2 ZINC000880963010 DH On-Demand Anodyne TRPV1 17 42 O=C(Nc1cnccc1C(F)(F)F)NC12CCC(CC1)CC2 ZINC000880963010 DH On-Demand Anodyne EPHX2 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CCO ZINC000880963011 DE On-Demand Anodyne RBP4 46 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CCO ZINC000880963012 DE On-Demand Anodyne RBP4 46 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2c(O)cccc21 ZINC000880963014 EH On-Demand Anodyne TRPV1 41 57 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2c(O)cccc21 ZINC000880963014 EH On-Demand Anodyne RBP4 46 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2c(O)cccc21 ZINC000880963015 EH On-Demand Anodyne TRPV1 41 57 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2c(O)cccc21 ZINC000880963015 EH On-Demand Anodyne RBP4 46 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](F)C1 ZINC000880963016 CF On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](F)C1 ZINC000880963016 CF On-Demand Anodyne RBP4 91 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](F)C1 ZINC000880963016 CF On-Demand Anodyne SFRP1 64 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](F)C1 ZINC000880963016 CF On-Demand Anodyne WNT3 46 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](F)C1 ZINC000880963017 CF On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](F)C1 ZINC000880963017 CF On-Demand Anodyne RBP4 91 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](F)C1 ZINC000880963017 CF On-Demand Anodyne SFRP1 64 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](F)C1 ZINC000880963017 CF On-Demand Anodyne WNT3 46 34 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(OC(F)F)CC1 ZINC000880963024 FH On-Demand Anodyne EPHX2 48 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1C1CCC1 ZINC000880963026 EI On-Demand Anodyne RBP4 55 41 C[S@](=O)[C@@H]1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963036 EF On-Demand Anodyne EPHX2 21 43 C[C@@H](F)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963037 CF On-Demand Anodyne TRPV1 18 47 C[S@](=O)[C@H]1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963038 EF On-Demand Anodyne EPHX2 21 43 C[S@](=O)[C@@H]1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963040 EF On-Demand Anodyne EPHX2 21 43 C[S@](=O)[C@H]1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963042 EF On-Demand Anodyne EPHX2 21 43 O=C(NCc1nc(C2CC2)n[nH]1)Nc1cnccc1C(F)(F)F ZINC000880963043 EE On-Demand Anodyne TRPV1 24 43 COC1(CO)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963044 EE On-Demand Anodyne RBP4 66 43 Cc1ccncc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963046 DG On-Demand Anodyne TRPV1 19 48 Cc1ccncc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963046 DG On-Demand Anodyne RAF1 24 41 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N(C)C ZINC000880963047 CE On-Demand Anodyne TRPV1 20 46 C=CC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963049 CG On-Demand Mild TRPV1 26 48 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1CC(Oc1ccccc1)C2 ZINC000880963050 GJ On-Demand Anodyne RBP4 77 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccccc21 ZINC000880963055 DH On-Demand Anodyne TRPV1 39 54 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccccc21 ZINC000880963055 DH On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccccc21 ZINC000880963055 DH On-Demand Anodyne TRPM8 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCOC2=O)CC1 ZINC000880963059 FF On-Demand Anodyne RBP4 64 40 COC[C@@H](O)Cc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880963061 FD On-Demand Anodyne GRIN2B 71 41 COC[C@@H](O)Cc1cn(CC(=O)N2CCC(Cc3ccccc3)CC2)nn1 ZINC000880963061 FD On-Demand Anodyne CCR3 31 40 O=C(NCc1cccnc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880963081 FG On-Demand Anodyne TRPV1 63 55 O=C(NCc1cccnc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880963081 FG On-Demand Anodyne SCN2A 19 47 O=C(NCc1cccnc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880963081 FG On-Demand Anodyne SCN10A 28 47 O=C(NCc1cccnc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880963081 FG On-Demand Anodyne NAMPT 53 41 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne TRPV1 29 47 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne RAF1 43 39 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne KDR 18 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne EPHX2 17 40 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne P96878_MYCTU 40 37 CCS(=O)(=O)Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880963082 GH On-Demand Anodyne NAMPT 51 38 COC(=O)N(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963084 CD On-Demand Reactive TRPV1 15 41 CC(C)(C)N1CC[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963085 EG On-Demand Anodyne TRPV1 19 43 NC(=O)c1cccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)c1 ZINC000880963086 GG On-Demand Anodyne ROCK2 24 40 CC(C)(C)N1CC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963087 EG On-Demand Anodyne TRPV1 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880963089 GI On-Demand Anodyne RBP4 63 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccc(F)cc2)CC1 ZINC000880963089 GI On-Demand Anodyne LIPG 38 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880963090 EF On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1c2ccccc2C[C@@H]1O ZINC000880963090 EF On-Demand Anodyne RBP4 49 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COC[C@H]1O ZINC000880963092 CC On-Demand Anodyne TRPV1 24 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)C1=O ZINC000880963093 DF On-Demand Anodyne TRPV1 15 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)C1=O ZINC000880963093 DF On-Demand Anodyne RBP4 78 47 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)C1(O)CCCC1 ZINC000880963094 EH On-Demand Anodyne TRPV1 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccco2)CC1 ZINC000880963099 EI On-Demand Anodyne RBP4 81 46 O=C(NC[C@@H]1C[C@H]1C1CC1)Nc1cnccc1C(F)(F)F ZINC000880963100 CG On-Demand Anodyne TRPV1 17 44 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880963102 FG On-Demand Anodyne IMDH_CRYPV 20 42 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880963103 FG On-Demand Anodyne IMDH_CRYPV 20 42 C=C[C@@H](C)ONC(=O)Nc1cnccc1C(F)(F)F ZINC000880963107 CF On-Demand Mild TRPV1 15 40 C=C[C@H](C)ONC(=O)Nc1cnccc1C(F)(F)F ZINC000880963108 CF On-Demand Mild TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2COC[C@H]2C1 ZINC000880963111 DF On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2COC[C@H]2C1 ZINC000880963111 DF On-Demand Anodyne RBP4 90 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2COC[C@@H]2C1 ZINC000880963112 DF On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2COC[C@@H]2C1 ZINC000880963112 DF On-Demand Anodyne RBP4 90 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2COC[C@H]2C1 ZINC000880963113 DF On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2COC[C@H]2C1 ZINC000880963113 DF On-Demand Anodyne RBP4 90 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880963114 DF On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2COC[C@@H]2C1 ZINC000880963114 DF On-Demand Anodyne RBP4 90 49 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)S(C)(=O)=O ZINC000880963120 ED On-Demand Anodyne TRPV1 22 45 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880963121 FG On-Demand Anodyne IMDH_CRYPV 18 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000880963122 FG On-Demand Anodyne IMDH_CRYPV 18 41 N#CCC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963123 CE On-Demand Mild RBP4 74 45 COCc1csc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880963124 EH On-Demand Anodyne TRPV1 21 45 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963125 FG On-Demand Anodyne EPHX2 45 42 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963125 FG On-Demand Anodyne GPR119 43 42 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963125 FG On-Demand Anodyne SFRP1 123 45 CC(C)(C)OC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963125 FG On-Demand Anodyne WNT3 84 40 N#Cc1cccc(C2(NC(=O)Nc3cnccc3C(F)(F)F)CCOCC2)c1 ZINC000880963129 GH On-Demand Mild MCHR1 19 40 COC(=O)Cc1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880963130 GE On-Demand Anodyne IMDH_CRYPV 30 46 CO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963131 DG On-Demand Anodyne RBP4 68 44 CO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963131 DG On-Demand Anodyne SFRP1 47 33 CO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963131 DG On-Demand Anodyne WNT3 42 32 C[C@H](N)c1cn(CC(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)nn1 ZINC000880963140 GD On-Demand Anodyne MC4R 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccc(O)cc21 ZINC000880963141 EH On-Demand Anodyne TRPV1 36 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2ccc(O)cc21 ZINC000880963142 EH On-Demand Anodyne TRPV1 36 50 CC[C@@H](C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963143 CH On-Demand Anodyne TRPV1 18 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C=Cc3ccccc3O2)CC1 ZINC000880963145 GJ On-Demand Anodyne NPY5R 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C=Cc3ccccc3O2)CC1 ZINC000880963145 GJ On-Demand Anodyne RBP4 56 39 CCn1c(O)nnc1C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963146 GF On-Demand Anodyne RBP4 72 42 Cc1ccc(CC2CN(C(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880963147 EI On-Demand Anodyne RBP4 62 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880963150 EF On-Demand Anodyne RBP4 95 53 COC1CC(CCNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963152 DG On-Demand Anodyne TRPV1 19 42 CCNC(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963153 CD On-Demand Anodyne TRPV1 20 47 O=C(Cn1cc([C@@H]2CCOC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880963157 FE On-Demand Anodyne GRIN2B 71 42 O=C(Cn1cc([C@H]2CCOC2)nn1)N1CCC(Cc2ccccc2)CC1 ZINC000880963158 FE On-Demand Anodyne GRIN2B 71 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](CC(F)(F)F)O1 ZINC000880963170 FH On-Demand Anodyne RBP4 57 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](CC(F)(F)F)O1 ZINC000880963171 FH On-Demand Anodyne RBP4 57 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](CC(F)(F)F)O1 ZINC000880963172 FH On-Demand Anodyne RBP4 57 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](CC(F)(F)F)O1 ZINC000880963173 FH On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CCCC[C@@H]21 ZINC000880963175 CH On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCOC2=O)C1 ZINC000880963176 EE On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCOC2=O)C1 ZINC000880963177 EE On-Demand Anodyne RBP4 61 41 C=CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963179 CF On-Demand Mild TRPV1 16 47 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnccc1C(F)(F)F ZINC000880963182 DH On-Demand Mild RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C1)CC2(F)F ZINC000880963184 DG On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C1)CC2(F)F ZINC000880963185 DG On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880963186 FH On-Demand Anodyne TRPV1 22 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1[C@@H]2c3ccc(F)cc3C[C@H]21 ZINC000880963187 FH On-Demand Anodyne TRPV1 22 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@H]21 ZINC000880963188 FH On-Demand Anodyne TRPV1 22 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2Cc3cc(F)ccc3[C@@H]21 ZINC000880963189 FH On-Demand Anodyne TRPV1 22 44 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963190 FH On-Demand Anodyne TRPV1 18 42 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963190 FH On-Demand Anodyne RBP4 99 49 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963190 FH On-Demand Anodyne SFRP1 114 38 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963190 FH On-Demand Anodyne SMO 22 40 CN(c1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963190 FH On-Demand Anodyne WNT3 83 36 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963191 FH On-Demand Anodyne TRPV1 18 42 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963191 FH On-Demand Anodyne RBP4 99 49 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963191 FH On-Demand Anodyne SFRP1 114 38 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963191 FH On-Demand Anodyne SMO 22 40 CN(c1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963191 FH On-Demand Anodyne WNT3 83 36 C=CC(C)(C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963192 DH On-Demand Mild TRPV1 17 44 CC[C@H](O)c1cn(CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)nn1 ZINC000880963194 FG On-Demand Anodyne IMDH_CRYPV 24 44 O=C(NCCS(=O)(=O)CC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880963195 GE On-Demand Anodyne TRPV1 15 46 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1S(C)(=O)=O ZINC000880963196 FD On-Demand Anodyne HSD11B1 22 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1S(C)(=O)=O ZINC000880963196 FD On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CCc2nccnc2C1 ZINC000880963198 DE On-Demand Anodyne RBP4 56 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1CO ZINC000880963203 DF On-Demand Anodyne RBP4 76 43 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1CO ZINC000880963204 DF On-Demand Anodyne RBP4 76 43 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1CO ZINC000880963205 DF On-Demand Anodyne RBP4 76 43 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1CO ZINC000880963206 DF On-Demand Anodyne RBP4 76 43 CO[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1cnn[nH]1 ZINC000880963207 FD On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880963208 GH On-Demand Anodyne CCR5 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880963208 GH On-Demand Anodyne RBP4 90 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880963208 GH On-Demand Anodyne SFRP1 63 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880963208 GH On-Demand Anodyne SMO 25 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)[C@H](CO)C1 ZINC000880963208 GH On-Demand Anodyne WNT3 47 32 O=C(NC[C@@H]1Cc2ccccc2CO1)Nc1cnccc1C(F)(F)F ZINC000880963211 FG On-Demand Anodyne TRPV1 21 45 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963213 FG On-Demand Anodyne TRPV1 20 49 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963213 FG On-Demand Anodyne P2RX7 21 43 Cn1ncc(C(F)(F)F)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963213 FG On-Demand Anodyne FLT1 16 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C(=O)N1CCOCC1 ZINC000880963217 GE On-Demand Anodyne RBP4 65 44 C[C@]1(C#N)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963219 CF On-Demand Mild RBP4 55 39 C[C@@]1(C#N)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963220 CF On-Demand Mild RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C=CCC1 ZINC000880963221 CF On-Demand Anodyne TRPV1 22 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C=CCC1 ZINC000880963222 CF On-Demand Anodyne TRPV1 22 41 CC[C@@](C)(NC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880963227 DH On-Demand Anodyne TRPV1 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880963231 GH On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880963231 GH On-Demand Anodyne NPY5R 22 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(c2ccccc2)CC1 ZINC000880963231 GH On-Demand Anodyne RBP4 93 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC[C@H]1O ZINC000880963232 DF On-Demand Anodyne EPHX2 15 44 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc2O1 ZINC000880963233 FH On-Demand Anodyne RBP4 75 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc2O1 ZINC000880963234 FH On-Demand Anodyne RBP4 75 43 CCC1(CNC(=O)Nc2cnccc2C(F)(F)F)COC1 ZINC000880963235 DF On-Demand Anodyne TRPV1 21 49 CN(C[C@H](O)Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880963236 FG On-Demand Anodyne TRPV1 15 42 CN(C[C@H](O)Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880963236 FG On-Demand Anodyne GPR142 56 34 CN(C[C@@H](O)Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880963237 FG On-Demand Anodyne TRPV1 15 42 CN(C[C@@H](O)Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880963237 FG On-Demand Anodyne GPR142 56 34 O=C(Nc1cnccc1C(F)(F)F)N1CC(F)(F)C(F)(F)C1 ZINC000880963245 EG On-Demand Mild TRPV1 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(F)(F)C(F)(F)C1 ZINC000880963245 EG On-Demand Mild RBP4 59 44 C[C@@H](CCCO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963252 DF On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne TRPV1 17 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne EPHX2 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne RBP4 99 52 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne SFRP1 109 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne SMO 22 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccccc2)C1 ZINC000880963253 EJ On-Demand Anodyne WNT3 77 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne TRPV1 17 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne EPHX2 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne RBP4 99 52 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne SFRP1 109 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne SMO 22 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccccc2)C1 ZINC000880963255 EJ On-Demand Anodyne WNT3 77 36 Cc1cccc2c1N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880963256 DI On-Demand Anodyne HTR2C 15 48 Cc1cccc2c1N(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880963256 DI On-Demand Anodyne RBP4 47 39 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN(C)C(=O)OC(C)(C)C)nn1 ZINC000880963261 GF On-Demand Anodyne DRD4 24 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN(C)C(=O)OC(C)(C)C)nn1 ZINC000880963261 GF On-Demand Anodyne TPP2 50 34 C=CCC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963262 DH On-Demand Mild TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2cccc(Cl)c2)C1 ZINC000880963268 FI On-Demand Anodyne TRPV1 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2cccc(Cl)c2)C1 ZINC000880963268 FI On-Demand Anodyne RBP4 80 46 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)O1 ZINC000880963273 ED On-Demand Anodyne RBP4 57 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)OC(C)(C)C)nn1 ZINC000880963283 FE On-Demand Anodyne DRD4 25 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)OC(C)(C)C)nn1 ZINC000880963283 FE On-Demand Anodyne TPP2 60 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(C1)CC2(F)F ZINC000880963290 EH On-Demand Anodyne RBP4 56 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(C1)CC2(F)F ZINC000880963294 EH On-Demand Anodyne RBP4 56 39 C[C@@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963295 FI On-Demand Anodyne RBP4 49 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963297 EI On-Demand Anodyne TRPV1 18 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963297 EI On-Demand Anodyne RBP4 95 50 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963297 EI On-Demand Anodyne TRPM8 44 44 C[C@H]1C[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963298 FI On-Demand Anodyne RBP4 49 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963300 EI On-Demand Anodyne TRPV1 18 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963300 EI On-Demand Anodyne RBP4 95 50 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCc2ccccc21 ZINC000880963300 EI On-Demand Anodyne TRPM8 44 44 O=C(NOCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880963302 CF On-Demand Anodyne TRPV1 25 43 NC(=O)[C@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963306 DD On-Demand Anodyne EPHX2 20 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)NC1CC1 ZINC000880963309 CB On-Demand Anodyne AVPR1B 17 40 N#C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880963311 FH On-Demand Mild RBP4 83 47 N#C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880963311 FH On-Demand Mild SMO 20 42 CNc1nc(C(=O)N2CC(c3ccccc3)C2)cs1 ZINC000880963312 CE On-Demand Anodyne TRPC6 66 43 CNc1nc(C(=O)N2CC(c3ccccc3)C2)cs1 ZINC000880963312 CE On-Demand Anodyne TRPC3 59 43 O=C(NCCC1CC(F)(F)C1)Nc1cnccc1C(F)(F)F ZINC000880963315 DH On-Demand Anodyne TRPV1 17 46 C[C@@H](CF)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963318 CF On-Demand Anodyne TRPV1 21 48 C[C@H]1CC[C@@H](O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963320 DE On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1nc[nH]n1 ZINC000880963322 EF On-Demand Anodyne CPT1A 58 38 C[C@H]1CC[C@H](O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963323 DE On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1nc[nH]n1 ZINC000880963324 EF On-Demand Anodyne CPT1A 58 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(Cc2ccc(F)cc2)C1 ZINC000880963327 GG On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(Cc2ccc(F)cc2)C1 ZINC000880963328 GG On-Demand Anodyne RBP4 47 37 CO[C@H]1c2ccccc2C[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963329 FH On-Demand Anodyne TRPV1 21 40 COC(=O)Cc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880963332 DC On-Demand Anodyne DRD4 28 52 COC(=O)Cc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880963332 DC On-Demand Anodyne TPP2 67 37 COC(=O)Cc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880963333 DC On-Demand Anodyne DRD4 28 52 COC(=O)Cc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880963333 DC On-Demand Anodyne TPP2 67 37 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)C(F)(F)F)nn1 ZINC000880963335 FD On-Demand Anodyne DRD4 25 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)C(F)(F)F)nn1 ZINC000880963335 FD On-Demand Anodyne TPP2 58 34 C[C@@H]1C[C@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963336 DE On-Demand Anodyne RBP4 82 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccccc2)nn1 ZINC000880963338 EE On-Demand Anodyne DRD4 28 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccccc2)nn1 ZINC000880963338 EE On-Demand Anodyne TPP2 60 35 C[C@H]1C[C@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963339 DE On-Demand Anodyne RBP4 82 49 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1c1ccc(F)cc1 ZINC000880963341 FH On-Demand Anodyne TRPM8 31 43 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1c1ccc(F)cc1 ZINC000880963343 FH On-Demand Anodyne TRPM8 31 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](O)CC1 ZINC000880963344 DE On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](O)CC1 ZINC000880963344 DE On-Demand Anodyne SFRP1 56 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](O)CC1 ZINC000880963344 DE On-Demand Anodyne WNT3 53 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccccc2)nn1 ZINC000880963345 EE On-Demand Anodyne DRD4 28 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccccc2)nn1 ZINC000880963345 EE On-Demand Anodyne TPP2 60 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](O)CC1 ZINC000880963346 DE On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](O)CC1 ZINC000880963346 DE On-Demand Anodyne SFRP1 56 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](O)CC1 ZINC000880963346 DE On-Demand Anodyne WNT3 53 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne EPHX2 39 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne RBP4 95 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne SCD1 31 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne SFRP1 111 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne SCD 27 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccc2)C1 ZINC000880963350 FH On-Demand Anodyne WNT3 80 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccncn2)CC1 ZINC000880963351 FG On-Demand Anodyne RBP4 76 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne ABL1 42 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne ACHE 26 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne TRPV1 27 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne SIGMAR1 36 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne P2RX7 18 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne ABL2 42 35 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne FAAH 45 59 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccc2)CC1 ZINC000880963353 FG On-Demand Anodyne RBP4 88 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CC(F)(F)F)C1 ZINC000880963354 FI On-Demand Anodyne RBP4 70 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CC(F)(F)F)C1 ZINC000880963355 FI On-Demand Anodyne RBP4 70 44 COC1(C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963362 FH On-Demand Anodyne RBP4 57 40 C=C(C)CONC(=O)Nc1cnccc1C(F)(F)F ZINC000880963369 CF On-Demand Mild TRPV1 15 41 O=C1O[C@H]2C[C@H]1N(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880963370 DD On-Demand Anodyne RBP4 48 41 Cn1ncc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880963375 DD On-Demand Anodyne TRPV1 20 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H]1CO ZINC000880963376 DE On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ccc([N+](=O)[O-])cc2)C1 ZINC000880963377 GI On-Demand Bother RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ccc([N+](=O)[O-])cc2)C1 ZINC000880963379 GI On-Demand Bother RBP4 62 42 C[C@@H]1CN(CC(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963384 GG On-Demand Anodyne RBP4 59 43 O=C1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)[C@H](c2ccccc2)N1 ZINC000880963386 GG On-Demand Anodyne TRPV1 22 40 Cn1cnc(CCNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880963388 DE On-Demand Anodyne TRPV1 15 45 N#CC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963389 CE On-Demand Mild RBP4 77 47 C[C@@H](CCO)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963390 DF On-Demand Anodyne TRPV1 16 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@@H](O)c2ccccn2)nn1 ZINC000880963392 FD On-Demand Anodyne DRD4 25 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@@H](O)c2ccccn2)nn1 ZINC000880963392 FD On-Demand Anodyne TPP2 58 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@H](O)c2ccccn2)nn1 ZINC000880963394 FD On-Demand Anodyne DRD4 25 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@H](O)c2ccccn2)nn1 ZINC000880963394 FD On-Demand Anodyne TPP2 58 34 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)OCC1CC1 ZINC000880963399 EG On-Demand Anodyne TRPV1 22 44 O=C(Nc1ccc(COCCO)cc1)Nc1cnccc1C(F)(F)F ZINC000880963400 FG On-Demand Anodyne TRPV1 20 46 O=C(Nc1ccc(COCCO)cc1)Nc1cnccc1C(F)(F)F ZINC000880963400 FG On-Demand Anodyne RAF1 43 38 O=C(Nc1cnccc1C(F)(F)F)N1CCS[C@H](c2ccccc2)C1 ZINC000880963401 FI On-Demand Anodyne RBP4 90 49 O=C(Nc1cnccc1C(F)(F)F)N1CCS[C@H](c2ccccc2)C1 ZINC000880963401 FI On-Demand Anodyne SMO 25 46 O=C(Nc1cnccc1C(F)(F)F)N1CCS[C@@H](c2ccccc2)C1 ZINC000880963402 FI On-Demand Anodyne RBP4 90 49 O=C(Nc1cnccc1C(F)(F)F)N1CCS[C@@H](c2ccccc2)C1 ZINC000880963402 FI On-Demand Anodyne SMO 25 46 NC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C(F)(F)F ZINC000880963403 FE On-Demand Anodyne RBP4 74 45 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963409 FD On-Demand Anodyne TRPV1 17 43 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963409 FD On-Demand Anodyne EPHX2 46 43 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963409 FD On-Demand Anodyne SFRP1 72 34 CS(=O)(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963409 FD On-Demand Anodyne WNT3 45 32 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963410 FD On-Demand Anodyne TRPV1 17 43 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963410 FD On-Demand Anodyne EPHX2 46 43 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963410 FD On-Demand Anodyne SFRP1 72 34 CS(=O)(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963410 FD On-Demand Anodyne WNT3 45 32 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880963413 FE On-Demand Anodyne DRD4 25 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880963413 FE On-Demand Anodyne TPP2 42 31 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880963414 FE On-Demand Anodyne DRD4 25 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880963414 FE On-Demand Anodyne TPP2 42 31 CNC(=O)C[C@@]1(O)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963422 FD On-Demand Anodyne RBP4 40 36 CNC(=O)C[C@]1(O)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963423 FD On-Demand Anodyne RBP4 40 36 CCC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963428 DE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](n2cc(CO)nn2)C1 ZINC000880963429 FD On-Demand Anodyne RBP4 57 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](n2cc(CO)nn2)C1 ZINC000880963430 FD On-Demand Anodyne RBP4 57 40 C[C@H](CCO)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963431 DF On-Demand Anodyne TRPV1 16 44 O=C(Nc1cnccc1C(F)(F)F)NC1(Cc2ccccc2)CCOCC1 ZINC000880963436 GI On-Demand Anodyne TRPV1 15 42 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1ccccc1 ZINC000880963441 GH On-Demand Anodyne RBP4 83 46 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1ccccc1 ZINC000880963441 GH On-Demand Anodyne SMO 18 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C(=O)c1cscn1 ZINC000880963443 GF On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)NC(CF)CF ZINC000880963444 CF On-Demand Anodyne TRPV1 20 46 O=C(NCCOCC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880963445 EG On-Demand Anodyne TRPV1 15 42 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880963446 GF On-Demand Anodyne PDGFRB 44 37 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880963446 GF On-Demand Anodyne TRPV1 20 46 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880963446 GF On-Demand Anodyne FAAH 18 47 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880963446 GF On-Demand Anodyne RBP4 49 46 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880963446 GF On-Demand Anodyne DGAT1 32 44 CO[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1O ZINC000880963448 DD On-Demand Anodyne RBP4 76 45 CN(C)C(=O)OC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963449 FF On-Demand Anodyne RBP4 72 42 O=C(NC[C@H](CO)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880963450 EG On-Demand Anodyne TRPV1 15 44 O=C(NC[C@@H](CO)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880963451 EG On-Demand Anodyne TRPV1 15 44 CC[C@H](C)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963453 EG On-Demand Anodyne TRPV1 15 43 CC[C@H](C)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963453 EG On-Demand Anodyne RBP4 60 40 O=C(NCCOC(=O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880963454 DE On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCOCC2)C1 ZINC000880963457 DF On-Demand Anodyne RBP4 55 40 CCO[C@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963461 DF On-Demand Anodyne EPHX2 40 38 CCC1(NC(=O)Nc2cnccc2C(F)(F)F)CCCC1 ZINC000880963462 DH On-Demand Anodyne TRPV1 16 43 O=C(NCC1=CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880963465 CH On-Demand Anodyne TRPV1 16 51 CC(C)(C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)C(N)=O ZINC000880963466 FG On-Demand Anodyne RBP4 62 42 CC(C)(C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)C(N)=O ZINC000880963467 FG On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)NN1CCCCC1 ZINC000880963468 CF On-Demand Anodyne TRPV1 19 41 CC(C)(C)OC(=O)N1CCN(Cc2cn(CC(=O)NC3CC3)nn2)CC1 ZINC000880963469 FC On-Demand Anodyne KDM1A 20 46 CCC(C)(C)OCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963470 DG On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CCCO)C1 ZINC000880963473 DF On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CCCO)C1 ZINC000880963474 DF On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H](C1CC1)[C@H](CO)C1CC1 ZINC000880963475 EG On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](C1CC1)[C@@H](CO)C1CC1 ZINC000880963476 EG On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](C1CC1)[C@H](CO)C1CC1 ZINC000880963477 EG On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H](C1CC1)[C@@H](CO)C1CC1 ZINC000880963478 EG On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C2CCC2)CC1 ZINC000880963481 EG On-Demand Anodyne EPHX2 48 46 CC[C@@H]1CN(CC)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963488 EG On-Demand Anodyne RBP4 46 38 COC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963491 EG On-Demand Anodyne RBP4 66 42 COC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963491 EG On-Demand Anodyne WNT3 42 31 O=C(NOCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880963493 CF On-Demand Anodyne TRPV1 25 43 CCc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)co1 ZINC000880963494 DF On-Demand Anodyne TRPV1 19 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](C2CC2)[C@H]1C1CC1 ZINC000880963499 EH On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](C2CC2)[C@@H]1C1CC1 ZINC000880963500 EH On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](C2CC2)[C@@H]1C1CC1 ZINC000880963501 EH On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](C2CC2)[C@H]1C1CC1 ZINC000880963502 EH On-Demand Anodyne RBP4 61 41 C[C@@H](Cc1cccc(O)c1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963503 EH On-Demand Anodyne TRPV1 35 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H]3C=C[C@@H](C3)[C@H]2C1 ZINC000880963505 DG On-Demand Anodyne RBP4 84 48 CCC1(CC)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963506 DH On-Demand Anodyne TRPV1 15 43 CCC1(CC)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963506 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)c2ccccc21 ZINC000880963509 EG On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)c2ccccc21 ZINC000880963509 EG On-Demand Anodyne RBP4 84 44 O=C(NC[C@@H]1CC[C@@H](c2ccccc2)O1)Nc1cnccc1C(F)(F)F ZINC000880963510 FI On-Demand Anodyne TRPV1 19 46 O=C(NC[C@H]1CC[C@@H](c2ccccc2)O1)Nc1cnccc1C(F)(F)F ZINC000880963511 FI On-Demand Anodyne TRPV1 19 46 O=C(NC[C@H]1CC[C@H](c2ccccc2)O1)Nc1cnccc1C(F)(F)F ZINC000880963512 FI On-Demand Anodyne TRPV1 19 46 O=C(NC[C@@H]1CC[C@H](c2ccccc2)O1)Nc1cnccc1C(F)(F)F ZINC000880963513 FI On-Demand Anodyne TRPV1 19 46 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C(=O)OC(C)(C)C ZINC000880963518 FH On-Demand Anodyne RBP4 58 42 O=C(NCCN1CCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880963521 DD On-Demand Anodyne TRPV1 15 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880963527 GF On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880963527 GF On-Demand Anodyne TPP2 49 32 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880963528 GF On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880963528 GF On-Demand Anodyne TPP2 49 32 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](CO)c2ccccc21 ZINC000880963530 EG On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](CO)c2ccccc21 ZINC000880963530 EG On-Demand Anodyne RBP4 84 44 CC(C)(CO)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880963531 EG On-Demand Anodyne TRPV1 17 45 COC[C@]1(CO)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963535 ED On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CC(C(F)(F)F)C1 ZINC000880963544 DG On-Demand Anodyne RBP4 88 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC=C(Cl)C1 ZINC000880963554 DG On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCc2sc(Cl)cc2C1 ZINC000880963555 FI On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CCSC2(CCC2)CC1 ZINC000880963562 EH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](C1)C2(F)F ZINC000880963563 DF On-Demand Anodyne RBP4 78 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@H](C1)C2(F)F ZINC000880963564 DF On-Demand Anodyne RBP4 78 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H](C1)C2(F)F ZINC000880963565 DF On-Demand Anodyne RBP4 78 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CC2(O)CCOCC2)nn1 ZINC000880963591 FD On-Demand Anodyne DRD4 25 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CC2(O)CCOCC2)nn1 ZINC000880963591 FD On-Demand Anodyne TPP2 45 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O[C@@H]2CCOC2)CC1 ZINC000880963592 FF On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O[C@H]2CCOC2)CC1 ZINC000880963593 FF On-Demand Anodyne RBP4 65 40 CN1C[C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)[C@@H]2C1 ZINC000880963594 EF On-Demand Anodyne RBP4 68 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CCN(Cc3ccccc3)[C@@H]2C1 ZINC000880963595 GH On-Demand Anodyne RBP4 93 51 COC(=O)[C@@]1(C)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963596 EF On-Demand Anodyne RBP4 45 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CCCC[C@H]2C1 ZINC000880963598 DH On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CCCC[C@H]2C1 ZINC000880963598 DH On-Demand Anodyne RBP4 94 52 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)C1 ZINC000880963606 EE On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)C1 ZINC000880963606 EE On-Demand Anodyne RBP4 67 44 Cc1ccccc1C1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963607 EI On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne SLC9A1 35 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne CCR2 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne EPHX2 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne RBP4 94 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccnc2)C1 ZINC000880963612 EH On-Demand Anodyne SMO 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne SLC9A1 35 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne CCR2 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne EPHX2 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne RBP4 94 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccnc2)C1 ZINC000880963613 EH On-Demand Anodyne SMO 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC12CCCC2 ZINC000880963619 CH On-Demand Anodyne RBP4 40 38 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880963625 EE On-Demand Anodyne DRD4 27 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880963625 EE On-Demand Anodyne TPP2 55 34 CC(=O)N1CCN(Cc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)CC1 ZINC000880963627 GC On-Demand Anodyne DRD4 38 57 CC(=O)N1CCN(Cc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)CC1 ZINC000880963627 GC On-Demand Anodyne TPP2 49 34 CC(=O)N1CCN(Cc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)CC1 ZINC000880963628 GC On-Demand Anodyne DRD4 38 57 CC(=O)N1CCN(Cc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)CC1 ZINC000880963628 GC On-Demand Anodyne TPP2 49 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)OCC(F)(F)F)nn1 ZINC000880963629 GE On-Demand Anodyne DRD4 24 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CNC(=O)OCC(F)(F)F)nn1 ZINC000880963629 GE On-Demand Anodyne TPP2 60 36 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H](C2CCC2)C1 ZINC000880963636 EG On-Demand Anodyne RBP4 76 46 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H](C2CCC2)C1 ZINC000880963637 EG On-Demand Anodyne RBP4 76 46 CC(C)(C)OC(=O)[C@]1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963639 FH On-Demand Anodyne RBP4 41 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@@H]2C1 ZINC000880963641 EH On-Demand Anodyne RBP4 92 51 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880963642 EH On-Demand Anodyne RBP4 92 51 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@H]3CC[C@@H](C3)[C@H]2C1 ZINC000880963643 EH On-Demand Anodyne RBP4 92 51 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(C(F)F)C1 ZINC000880963646 EE On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(C(F)F)C1 ZINC000880963647 EE On-Demand Anodyne RBP4 55 40 CCNc1nc(C)c(C(=O)N2CC(c3ccccc3)C2)s1 ZINC000880963656 DG On-Demand Anodyne SCD1 15 40 CS(=O)(=O)CC1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963658 GF On-Demand Anodyne EPHX2 40 42 CCC(CC)(CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880963669 DG On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccnc(F)c2)CC1 ZINC000880963671 FF On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccnc(F)c2)CC1 ZINC000880963671 FF On-Demand Anodyne RBP4 56 39 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCC2)[C@@H]1c1ccccc1 ZINC000880963713 FJ On-Demand Anodyne RBP4 69 42 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCC2)[C@H]1c1ccccc1 ZINC000880963728 FJ On-Demand Anodyne RBP4 69 42 O=C(NCCC1(CO)CC1)Nc1cnccc1C(F)(F)F ZINC000880963759 DE On-Demand Anodyne TRPV1 15 47 O=C(NCCN1C[C@@H]2CC[C@H](C1)O2)Nc1cnccc1C(F)(F)F ZINC000880963760 EE On-Demand Anodyne TRPV1 15 41 N#Cc1ccncc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963767 GF On-Demand Mild RBP4 54 39 C=C(C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963770 CG On-Demand Mild TRPV1 26 52 O=C(NC[C@H]1Cc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880963777 EG On-Demand Anodyne TRPV1 18 47 O=C(NC[C@@H]1Cc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880963778 EG On-Demand Anodyne TRPV1 18 47 O=C(NC[C@H]1CSc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880963786 FI On-Demand Anodyne TRPV1 16 45 O=C(NC[C@@H]1CSc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880963787 FI On-Demand Anodyne TRPV1 16 45 CC(C)C1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963790 CG On-Demand Anodyne TRPV1 17 42 CC(C)(C)OC(=O)N1CCC(c2cn(CC(=O)NC3CC3)nn2)CC1 ZINC000880963791 ED On-Demand Anodyne GPR119 44 41 CCc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)n[nH]1 ZINC000880963793 DE On-Demand Anodyne TRPV1 22 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCCCO2 ZINC000880963871 EF On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)C12CCCC2 ZINC000880963872 EG On-Demand Anodyne RBP4 41 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](O)C12CCCC2 ZINC000880963873 EG On-Demand Anodyne RBP4 41 38 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN(C2CCC2)C1 ZINC000880963874 FG On-Demand Anodyne RBP4 59 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN(C2CCC2)C1 ZINC000880963875 FG On-Demand Anodyne RBP4 59 42 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CC1 ZINC000880963876 CC On-Demand Anodyne MME 42 36 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CC1 ZINC000880963876 CC On-Demand Anodyne SIGMAR1 17 44 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CC1 ZINC000880963877 CC On-Demand Anodyne MME 42 36 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CC1 ZINC000880963877 CC On-Demand Anodyne SIGMAR1 17 44 O=C(Nc1cnccc1C(F)(F)F)NC1(Cc2cccc(F)c2)CCOCC1 ZINC000880963880 GI On-Demand Anodyne TRPV1 23 42 CCC[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880963883 DG On-Demand Anodyne TRPV1 15 43 CCC[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880963884 DG On-Demand Anodyne TRPV1 15 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)N1C ZINC000880963885 DF On-Demand Anodyne TRPV1 15 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)N1C ZINC000880963885 DF On-Demand Anodyne RBP4 79 47 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963888 FE On-Demand Anodyne RBP4 64 41 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963888 FE On-Demand Anodyne SFRP1 48 35 CN(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963888 FE On-Demand Anodyne WNT3 41 35 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963889 FE On-Demand Anodyne RBP4 64 41 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963889 FE On-Demand Anodyne SFRP1 48 35 CN(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963889 FE On-Demand Anodyne WNT3 41 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne TRPV1 24 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne PIM1 29 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne EPHX2 35 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne PIM3 19 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2F)C1 ZINC000880963892 FH On-Demand Anodyne SFRP1 74 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne TRPV1 24 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne PIM1 29 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne EPHX2 35 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne PIM3 19 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2F)C1 ZINC000880963893 FH On-Demand Anodyne SFRP1 74 35 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](C1)[C@H]1C=C[C@H]2O1 ZINC000880963894 EF On-Demand Anodyne RBP4 80 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2[C@H]3C=C[C@@H](O3)[C@H]2C1 ZINC000880963895 EF On-Demand Anodyne RBP4 80 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@H]3C=C[C@@H](O3)[C@H]2C1 ZINC000880963896 EF On-Demand Anodyne RBP4 80 45 Cc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880963899 DI On-Demand Anodyne TRPV1 24 62 CC[C@@](C)(CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880963903 DG On-Demand Anodyne TRPV1 17 44 CO[C@H]1COCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963907 EE On-Demand Anodyne TRPV1 16 41 C=C(CC)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963914 CG On-Demand Mild TRPV1 20 47 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccn1 ZINC000880963915 EH On-Demand Anodyne TRPV1 28 53 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(CCSC2)C1 ZINC000880963916 EH On-Demand Anodyne RBP4 54 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(CCSC2)C1 ZINC000880963917 EH On-Demand Anodyne RBP4 54 37 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(CCCO)C1 ZINC000880963926 EE On-Demand Anodyne EPHX2 29 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(CCCO)C1 ZINC000880963926 EE On-Demand Anodyne BIRC2 31 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(CCCO)C1 ZINC000880963927 EE On-Demand Anodyne EPHX2 29 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(CCCO)C1 ZINC000880963927 EE On-Demand Anodyne BIRC2 31 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)n2)CC1 ZINC000880963928 FF On-Demand Anodyne TRPV1 27 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)n2)CC1 ZINC000880963928 FF On-Demand Anodyne RBP4 58 41 CS(=O)(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963932 FE On-Demand Anodyne RBP4 69 43 CS(=O)(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963932 FE On-Demand Anodyne SFRP1 69 34 CS(=O)(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880963932 FE On-Demand Anodyne WNT3 58 33 Cn1cc(Br)c(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880963936 GF On-Demand Anodyne TRPV1 15 46 CC1(C)CCC[C@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963938 EG On-Demand Anodyne TRPV1 17 45 CC1(C)CCC[C@@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963939 EG On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](n2cc(CO)nn2)C1 ZINC000880963940 FE On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](n2cc(CO)nn2)C1 ZINC000880963941 FE On-Demand Anodyne RBP4 54 39 C#C[C@](C)(CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963944 CG On-Demand Mild TRPV1 19 44 C#C[C@@](C)(CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880963945 CG On-Demand Mild TRPV1 19 44 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne MAPK14 15 42 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne TRPV1 32 52 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne EPHX2 18 44 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne CARM1 55 35 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne STAT6 57 42 O=C(NCc1cccc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880963947 GG On-Demand Anodyne NAMPT 61 44 O=C(NC[C@H]1CCC[C@@H]1O)Nc1cnccc1C(F)(F)F ZINC000880963953 DE On-Demand Anodyne TRPV1 19 44 CC(CO)(CO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880963962 DD On-Demand Anodyne TRPV1 21 47 CCOC(=O)[C@@H](F)C1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963965 EE On-Demand Anodyne RBP4 68 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880963966 CE On-Demand Anodyne RBP4 78 45 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963970 FF On-Demand Anodyne RBP4 60 42 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963970 FF On-Demand Anodyne SFRP1 55 35 CN(C)C(=O)O[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880963970 FF On-Demand Anodyne WNT3 49 35 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)(C)O ZINC000880963972 DF On-Demand Anodyne TRPV1 17 51 O=C(Nc1cnccc1C(F)(F)F)N(CCN1CCOCC1)Cc1ccco1 ZINC000880963974 GG On-Demand Anodyne CASR 57 45 CC[C@H](O)c1cn(CC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)nn1 ZINC000880963983 GG On-Demand Anodyne NPY5R 15 55 CC[C@H](O)c1cn(CC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)nn1 ZINC000880963983 GG On-Demand Anodyne IMDH_CRYPV 46 34 CC[C@H]1[C@H](CO)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963986 DF On-Demand Anodyne RBP4 46 38 CC[C@@H]1[C@H](CO)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963987 DF On-Demand Anodyne RBP4 46 38 CC[C@H]1[C@@H](CO)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880963988 DF On-Demand Anodyne RBP4 46 38 C[C@H]1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)O1 ZINC000880963994 DF On-Demand Anodyne TRPV1 20 42 C[C@H]1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)O1 ZINC000880963995 DF On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1C(F)F ZINC000880963997 CF On-Demand Anodyne RBP4 54 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1C(F)F ZINC000880963998 CF On-Demand Anodyne RBP4 54 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(c2ccc(Cl)cc2)C1 ZINC000880964001 FI On-Demand Anodyne RBP4 83 47 O=C(NCCc1cccc(C(F)(F)F)n1)Nc1cnccc1C(F)(F)F ZINC000880964008 GH On-Demand Anodyne TRPV1 33 53 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc(F)cc1F ZINC000880964013 FJ On-Demand Anodyne RBP4 49 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc(F)cc1F ZINC000880964014 FJ On-Demand Anodyne RBP4 49 37 CN1CC[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1 ZINC000880964029 EF On-Demand Anodyne EPHX2 28 40 CN1CC[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1 ZINC000880964029 EF On-Demand Anodyne RBP4 55 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)N1CCO ZINC000880964032 EE On-Demand Anodyne RBP4 77 46 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NC1CC1 ZINC000880964037 DD On-Demand Anodyne MMP8 18 45 C[C@@H]1CCC[C@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964049 DF On-Demand Anodyne TRPV1 17 44 C[C@H]1CCC[C@@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964050 DF On-Demand Anodyne TRPV1 17 44 C[C@H]1CCC[C@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964051 DF On-Demand Anodyne TRPV1 17 44 Nc1cccc(OCc2cn(CC(=O)NC3CC3)nn2)c1 ZINC000880964052 CC On-Demand Anodyne FAAH 16 40 Nc1cccc(OCc2cn(CC(=O)NC3CC3)nn2)c1 ZINC000880964052 CC On-Demand Anodyne FIMH 15 41 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NC ZINC000880964055 DD On-Demand Anodyne TRPV1 20 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H](C1CCC1)C1CC1 ZINC000880964059 DH On-Demand Anodyne TRPV1 15 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](C1CCC1)C1CC1 ZINC000880964060 DH On-Demand Anodyne TRPV1 15 49 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne CTSB 35 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne CTSK 27 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne PREP 27 44 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne CAPNS1 52 33 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne CAPN1 59 37 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne CAPN2 96 37 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CC1 ZINC000880964068 EC On-Demand Anodyne NPR 60 33 O=C1CC[C@@H](N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CCN1 ZINC000880964069 GD On-Demand Anodyne RBP4 54 39 O=C1CC[C@H](N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CCN1 ZINC000880964070 GD On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](Nc2ccccn2)CC1 ZINC000880964071 GI On-Demand Anodyne TRPV1 32 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](Nc2ccccn2)CC1 ZINC000880964071 GI On-Demand Anodyne PRKD1 42 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](Nc2ccccn2)CC1 ZINC000880964071 GI On-Demand Anodyne EPHX2 39 47 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CC2)C1 ZINC000880964073 CF On-Demand Anodyne RBP4 59 43 CO[C@@H](C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964077 CF On-Demand Anodyne TRPV1 17 44 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C1CCCC1 ZINC000880964079 DH On-Demand Anodyne TRPV1 19 51 O=C1NC(=O)[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]12 ZINC000880964080 EC On-Demand Anodyne RBP4 77 46 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880964084 GJ On-Demand Anodyne PRCP 40 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880964084 GJ On-Demand Anodyne RBP4 40 36 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880964085 GJ On-Demand Anodyne PRCP 40 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880964085 GJ On-Demand Anodyne RBP4 40 36 O=C(Cn1cc(-c2ccc(Cl)cc2F)nn1)NC1CC1 ZINC000880964090 CE On-Demand Anodyne MAPK13 52 31 CNS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964093 FD On-Demand Anodyne RBP4 70 46 CNS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964093 FD On-Demand Anodyne SFRP1 68 35 CNS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964093 FD On-Demand Anodyne WNT3 55 33 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne DRD2 16 40 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne HRH2 22 41 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne DRD3 35 40 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne TRPV1 15 43 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne CCR3 25 49 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne CHRNA7 22 54 O=C(NCCCCCN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880964095 EG On-Demand Anodyne HNMT 53 37 O=C(NC[C@H]1CCCC[C@@H]1O)Nc1cnccc1C(F)(F)F ZINC000880964097 DF On-Demand Anodyne TRPV1 19 44 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1(Cl)Cl ZINC000880964098 EH On-Demand Anodyne TRPV1 23 47 O=C(NCCc1cc(C(F)(F)F)ccn1)Nc1cnccc1C(F)(F)F ZINC000880964105 GH On-Demand Anodyne TRPV1 25 57 O=C(NCCc1cc(C(F)(F)F)ccn1)Nc1cnccc1C(F)(F)F ZINC000880964105 GH On-Demand Anodyne RAF1 30 40 O=C(NCCc1cc(C(F)(F)F)ccn1)Nc1cnccc1C(F)(F)F ZINC000880964105 GH On-Demand Anodyne RIPK1 44 34 O=C(NC[C@H]1CCCCC1(F)F)Nc1cnccc1C(F)(F)F ZINC000880964108 EI On-Demand Anodyne TRPV1 15 44 CC(C)(C)C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964110 EI On-Demand Anodyne RBP4 81 45 CC(C)(C)C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964110 EI On-Demand Anodyne SFRP1 96 36 CC(C)(C)C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964110 EI On-Demand Anodyne WNT3 75 33 CC(C)(C)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964111 EI On-Demand Anodyne RBP4 81 45 CC(C)(C)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964111 EI On-Demand Anodyne SFRP1 96 36 CC(C)(C)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964111 EI On-Demand Anodyne WNT3 75 33 O=C(Cn1cc(COc2ccc(Br)nc2)nn1)NC1CC1 ZINC000880964115 FD On-Demand Anodyne FIMH 20 42 CC1(CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964119 CD On-Demand Anodyne TRPV1 15 40 CC1(CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964119 CD On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCC2)CC1 ZINC000880964122 EI On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880964123 GF On-Demand Anodyne CHRNA4 26 48 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@H](C1)c1cccc(=O)n1C2 ZINC000880964123 GF On-Demand Anodyne RBP4 77 45 CC(C)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCCO1 ZINC000880964124 EG On-Demand Anodyne RBP4 70 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880964127 DD On-Demand Anodyne DRD4 28 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880964127 DD On-Demand Anodyne TPP2 58 34 C[C@@H](CO)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964131 EF On-Demand Anodyne RBP4 74 41 O=C(NC[C@H]1C[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880964135 EI On-Demand Anodyne TRPV1 22 49 O=C(NC[C@H]1C[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880964135 EI On-Demand Anodyne RBP4 47 40 O=C(NC[C@@H]1C[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880964137 EI On-Demand Anodyne TRPV1 22 49 O=C(NC[C@@H]1C[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880964137 EI On-Demand Anodyne RBP4 47 40 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)S1(=O)=O ZINC000880964146 FE On-Demand Anodyne RBP4 77 46 O=C(NC[C@]1(CO)CCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880964147 FG On-Demand Anodyne TRPV1 17 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)S1(=O)=O ZINC000880964148 FE On-Demand Anodyne RBP4 77 46 O=C(NC[C@@]1(CO)CCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880964149 FG On-Demand Anodyne TRPV1 17 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)S1(=O)=O ZINC000880964150 FE On-Demand Anodyne RBP4 77 46 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC(F)(F)F ZINC000880964153 EH On-Demand Anodyne TRPV1 19 46 CN1C(=O)N[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1=O ZINC000880964157 FD On-Demand Anodyne RBP4 42 39 CN1C(=O)N[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1=O ZINC000880964158 FD On-Demand Anodyne RBP4 42 39 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1 ZINC000880964175 FE On-Demand Anodyne DRD4 26 56 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1 ZINC000880964175 FE On-Demand Anodyne TPP2 62 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1 ZINC000880964177 FE On-Demand Anodyne DRD4 26 56 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1 ZINC000880964177 FE On-Demand Anodyne TPP2 62 34 O=C(NCCOCC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880964179 DG On-Demand Anodyne TRPV1 15 42 C#C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880964180 CF On-Demand Mild TRPV1 15 46 C#C[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880964182 CF On-Demand Mild TRPV1 15 46 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)S1(=O)=O ZINC000880964186 FF On-Demand Anodyne RBP4 61 44 Cn1cnnc1[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880964187 FD On-Demand Anodyne RBP4 59 39 Cn1cnnc1[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880964189 FD On-Demand Anodyne RBP4 59 39 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)S1(=O)=O ZINC000880964190 FF On-Demand Anodyne RBP4 61 44 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964193 FI On-Demand Anodyne TBXAS1 30 41 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964193 FI On-Demand Anodyne PTAFR 36 51 C[C@@H](CCCc1cccnc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964193 FI On-Demand Anodyne TRPV1 21 43 CCCN(CCN1CCCC1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880964194 EG On-Demand Anodyne CASR 44 38 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@@](C)(O)c2cccs2)nn1 ZINC000880964195 GF On-Demand Anodyne DRD4 23 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@](C)(O)c2cccs2)nn1 ZINC000880964199 GF On-Demand Anodyne DRD4 23 44 CO[C@@](C)(C1CC1)[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964207 EG On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(C(F)(F)F)CC1 ZINC000880964210 FG On-Demand Anodyne RBP4 56 40 CO[C@@](C)(C1CC1)[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964212 EG On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(C(F)(F)F)CC1 ZINC000880964213 FG On-Demand Anodyne RBP4 56 40 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)cc1 ZINC000880964214 GF On-Demand Anodyne DRD4 24 49 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)cc1 ZINC000880964214 GF On-Demand Anodyne TPP2 54 33 COCC(C)(C)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964215 EH On-Demand Anodyne TRPV1 17 42 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)cc1 ZINC000880964217 GF On-Demand Anodyne DRD4 24 49 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)cc1 ZINC000880964217 GF On-Demand Anodyne TPP2 54 33 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)C1(O)CCOCC1 ZINC000880964223 FF On-Demand Anodyne TRPV1 16 43 O=C(NCC1(C(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880964228 EH On-Demand Anodyne TRPV1 24 51 C[C@@](CO)(NC(=O)Nc1cnccc1C(F)(F)F)c1cccc(O)c1 ZINC000880964230 FF On-Demand Anodyne TRPV1 29 46 COCC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964234 DF On-Demand Anodyne TRPV1 21 45 C#C[C@H](CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964236 CF On-Demand Mild TRPV1 21 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1 ZINC000880964237 GF On-Demand Anodyne DRD4 32 57 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1 ZINC000880964237 GF On-Demand Anodyne TPP2 63 32 C#C[C@@H](CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964238 CF On-Demand Mild TRPV1 21 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1 ZINC000880964239 GF On-Demand Anodyne DRD4 32 57 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1 ZINC000880964239 GF On-Demand Anodyne TPP2 63 32 CS(=O)(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CCCC1 ZINC000880964240 FF On-Demand Anodyne TRPV1 17 45 CN1CCC[C@@H](CCNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964245 EF On-Demand Anodyne TRPV1 15 40 O=C(Cn1cc(C(=O)c2ccc(C(F)(F)F)cc2)nn1)NC1CC1 ZINC000880964252 ED On-Demand Anodyne CCR2 42 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1F ZINC000880964255 EH On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1F ZINC000880964255 EH On-Demand Anodyne RBP4 52 40 COC(=O)[C@H](F)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964257 DD On-Demand Anodyne TRPV1 18 45 CC[C@@H](C)CONC(=O)Nc1cnccc1C(F)(F)F ZINC000880964260 CG On-Demand Anodyne TRPV1 15 43 CC[C@H](C)CONC(=O)Nc1cnccc1C(F)(F)F ZINC000880964262 CG On-Demand Anodyne TRPV1 15 43 CN(C[C@@](C)(O)c1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880964270 FG On-Demand Anodyne TRPV1 16 41 CN1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1cccnc1 ZINC000880964283 GG On-Demand Anodyne TRPV1 17 41 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnccc4C(F)(F)F)[C@H]1[C@H]3C2 ZINC000880964284 EF On-Demand Anodyne RBP4 55 41 C#C[C@@H]1COCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880964285 CD On-Demand Mild RBP4 53 39 CO[C@@H]1[C@@H]2C[C@H]3[C@@H](C2)CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]31 ZINC000880964286 EF On-Demand Anodyne RBP4 55 41 C#C[C@H]1COCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880964287 CD On-Demand Mild RBP4 53 39 CO[C@@H]1[C@H]2C[C@@H]3CN(C(=O)Nc4cnccc4C(F)(F)F)[C@@H]1[C@H]3C2 ZINC000880964288 EF On-Demand Anodyne RBP4 55 41 CO[C@@H]1[C@@H]2C[C@@H]3[C@@H]1N(C(=O)Nc1cnccc1C(F)(F)F)C[C@@H]3C2 ZINC000880964290 EF On-Demand Anodyne RBP4 55 41 CC1(C)C[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964293 CG On-Demand Anodyne TRPV1 30 42 COC[C@@H](O)Cc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964303 EC On-Demand Anodyne DRD4 25 49 COC[C@@H](O)Cc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964303 EC On-Demand Anodyne TPP2 58 34 COC[C@@H](O)Cc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964309 EC On-Demand Anodyne DRD4 25 49 COC[C@@H](O)Cc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964309 EC On-Demand Anodyne TPP2 58 34 COC(=O)[C@@H]1C[C@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964321 ED On-Demand Anodyne RBP4 67 44 COC(=O)[C@H]1C[C@@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964322 ED On-Demand Anodyne RBP4 67 44 COC(=O)[C@H]1C[C@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964323 ED On-Demand Anodyne RBP4 67 44 COC(=O)[C@@H]1C[C@@H](O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964324 ED On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCSC1 ZINC000880964330 DG On-Demand Anodyne EPHX2 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCSC1 ZINC000880964331 DG On-Demand Anodyne EPHX2 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)c1ccc(Cl)cc1 ZINC000880964339 FH On-Demand Anodyne UTS2 43 33 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)c1ccc(Cl)cc1 ZINC000880964340 FH On-Demand Anodyne UTS2 43 33 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CC3)nn2)c1 ZINC000880964359 DD On-Demand Anodyne PLG 15 40 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CC3)nn2)c1 ZINC000880964359 DD On-Demand Anodyne FAAH 15 42 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CC3)nn2)c1 ZINC000880964359 DD On-Demand Anodyne FIMH 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC=C(c2ccco2)C1 ZINC000880964369 EI On-Demand Anodyne RBP4 54 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H](C1CC1)C(F)(F)F ZINC000880964376 EH On-Demand Anodyne TRPV1 18 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](C1CC1)C(F)(F)F ZINC000880964377 EH On-Demand Anodyne TRPV1 18 42 CC(C)(C#N)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964380 CF On-Demand Mild TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)[C@H](c2ccsc2)C1 ZINC000880964389 FG On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1ccc(F)cc1 ZINC000880964390 FH On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1ccc(F)cc1 ZINC000880964390 FH On-Demand Anodyne TRPM8 28 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1ccc(F)cc1 ZINC000880964391 FH On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1ccc(F)cc1 ZINC000880964391 FH On-Demand Anodyne TRPM8 28 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1ccc(F)cc1 ZINC000880964392 FH On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1ccc(F)cc1 ZINC000880964392 FH On-Demand Anodyne TRPM8 28 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1ccc(F)cc1 ZINC000880964393 FH On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1ccc(F)cc1 ZINC000880964393 FH On-Demand Anodyne TRPM8 28 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1cc(F)ccc1F ZINC000880964394 GH On-Demand Anodyne RBP4 43 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1cc(F)ccc1F ZINC000880964395 GH On-Demand Anodyne RBP4 43 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1cc(F)ccc1F ZINC000880964396 GH On-Demand Anodyne RBP4 43 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1cc(F)ccc1F ZINC000880964397 GH On-Demand Anodyne RBP4 43 38 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880964419 FE On-Demand Anodyne DPP8 18 43 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880964420 FE On-Demand Anodyne DPP8 18 43 C[C@@H]1CC(CCNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880964429 EH On-Demand Anodyne TRPV1 15 42 C[C@H]1CC(CCNC(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)O1 ZINC000880964430 EH On-Demand Anodyne TRPV1 15 42 C[C@H]1C[C@H](CCNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880964431 EH On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2(O)CC2)CC1 ZINC000880964436 EF On-Demand Anodyne RBP4 72 43 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)C(C)C ZINC000880964440 DG On-Demand Anodyne TRPV1 15 49 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)C(C)C ZINC000880964441 DG On-Demand Anodyne TRPV1 15 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880964443 GF On-Demand Anodyne DRD4 23 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2OCC[C@@H]2C1 ZINC000880964444 DF On-Demand Anodyne RBP4 88 47 CC(=O)N1CCN(Cc2cn(CC(=O)N3CCc4ccccc43)nn2)CC1 ZINC000880964447 FC On-Demand Anodyne DRD4 24 53 COCC(COC)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964448 GD On-Demand Anodyne RBP4 56 41 C=C[C@](C)(O)c1cn(CC(=O)N2CCc3ccccc32)nn1 ZINC000880964451 CD On-Demand Mild EIF2AK3 45 32 C=C[C@@](C)(O)c1cn(CC(=O)N2CCc3ccccc32)nn1 ZINC000880964452 CD On-Demand Mild EIF2AK3 45 32 COC(=O)C1CCC(c2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)CC1 ZINC000880964453 GF On-Demand Anodyne DRD4 26 49 COC(=O)C1CCC(c2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)CC1 ZINC000880964453 GF On-Demand Anodyne TPP2 53 31 COC(=O)C1CCC(c2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)CC1 ZINC000880964454 GF On-Demand Anodyne DRD4 26 49 COC(=O)C1CCC(c2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)CC1 ZINC000880964454 GF On-Demand Anodyne TPP2 53 31 CC(C)(C)OC(=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964455 EG On-Demand Anodyne TRPV1 17 45 CNC(=O)[C@]1(C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964457 GF On-Demand Anodyne RBP4 48 38 CCON(C)C(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964459 DD On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880964460 FH On-Demand Mild TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)C(F)(F)C2(F)F ZINC000880964460 FH On-Demand Mild RBP4 61 43 N#Cc1ccc2c(c1)CCC[C@@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964464 FI On-Demand Mild TRPV1 28 49 N#Cc1ccc2c(c1)CCC[C@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964465 FI On-Demand Mild TRPV1 28 49 O=C(NCc1ncc2c(n1)CCOC2)Nc1cnccc1C(F)(F)F ZINC000880964470 FE On-Demand Anodyne TRPV1 15 41 CC(C)(C)OC(=O)N1CC[C@H](c2cn(CC(=O)N3CCc4ccccc43)nn2)C1 ZINC000880964471 GF On-Demand Anodyne GPR119 28 41 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(CC(=O)N3CCc4ccccc43)nn2)C1 ZINC000880964472 GF On-Demand Anodyne GPR119 28 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)CC2(F)F ZINC000880964473 EH On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCSC2)C1 ZINC000880964485 EF On-Demand Anodyne EPHX2 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCSC2)C1 ZINC000880964485 EF On-Demand Anodyne RBP4 52 36 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCSC2)C1 ZINC000880964486 EF On-Demand Anodyne EPHX2 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCSC2)C1 ZINC000880964486 EF On-Demand Anodyne RBP4 52 36 Cc1nnc([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)o1 ZINC000880964492 FG On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCC(F)(F)C1 ZINC000880964493 DG On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(Cl)nnc2C1 ZINC000880964494 FG On-Demand Anodyne MAPK1 45 35 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(Cl)nnc2C1 ZINC000880964494 FG On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cn2cnnc2)CC1 ZINC000880964495 FF On-Demand Anodyne RBP4 69 41 CS(=O)(=O)C1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964500 DD On-Demand Anodyne RBP4 80 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)[C@H](C2CCCC2)C1 ZINC000880964502 FH On-Demand Anodyne RBP4 76 46 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880964504 GH On-Demand Anodyne RBP4 83 46 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880964504 GH On-Demand Anodyne SMO 18 42 COCCN1C(=O)N[C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@H]21 ZINC000880964507 GD On-Demand Anodyne RBP4 57 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@]1(F)c1ccccc1 ZINC000880964509 EH On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@]1(F)c1ccccc1 ZINC000880964510 EH On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@]1(F)c1ccccc1 ZINC000880964511 EH On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@]1(F)c1ccccc1 ZINC000880964512 EH On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)NC1(C2CCC2)CC1 ZINC000880964520 CH On-Demand Anodyne TRPV1 15 40 NC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964525 GF On-Demand Anodyne RBP4 64 45 NC(=O)[C@]1(c2ccccc2)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964526 GF On-Demand Anodyne RBP4 64 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880964527 GI On-Demand Anodyne CCR1 32 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880964527 GI On-Demand Anodyne EPHX2 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](O)(c2ccc(Cl)cc2)C1 ZINC000880964527 GI On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880964528 GI On-Demand Anodyne CCR1 32 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880964528 GI On-Demand Anodyne EPHX2 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](O)(c2ccc(Cl)cc2)C1 ZINC000880964528 GI On-Demand Anodyne RBP4 47 37 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCOC2)nn1 ZINC000880964532 DD On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCOC2)nn1 ZINC000880964532 DD On-Demand Anodyne TPP2 47 32 COCCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880964534 GH On-Demand Anodyne TRPV1 20 52 O=C(Nc1cnccc1C(F)(F)F)N1CC(O)(c2ccc(Cl)cc2)C1 ZINC000880964549 FG On-Demand Anodyne CCR1 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(O)(c2ccc(Cl)cc2)C1 ZINC000880964549 FG On-Demand Anodyne RBP4 42 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](F)C[C@H]1CO ZINC000880964550 DE On-Demand Anodyne RBP4 47 40 CN(C)CCCOc1cnccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964555 GG On-Demand Anodyne TRPV1 17 48 NC(=O)[C@H]1CCO[C@@H]1C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964558 GE On-Demand Anodyne RBP4 68 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880964567 GI On-Demand Anodyne EPHX2 28 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880964567 GI On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880964567 GI On-Demand Anodyne SCD1 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880964567 GI On-Demand Anodyne TRPM8 50 56 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880964568 GI On-Demand Anodyne EPHX2 28 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880964568 GI On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880964568 GI On-Demand Anodyne SCD1 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880964568 GI On-Demand Anodyne TRPM8 50 56 CN(C(=O)Nc1cnccc1C(F)(F)F)C1C[C@@H]2CC[C@H](C1)N2C ZINC000880964573 EG On-Demand Anodyne GLRA1 43 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2[C@@H](CO)[C@@H]2C1 ZINC000880964588 DD On-Demand Anodyne RBP4 81 46 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2cc(O)ccc2C1 ZINC000880964589 FG On-Demand Anodyne RBP4 53 39 Cn1nccc1C1=CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964590 FG On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1cccc(F)c1 ZINC000880964593 FH On-Demand Anodyne RBP4 42 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1cccc(F)c1 ZINC000880964594 FH On-Demand Anodyne RBP4 42 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1cccc(F)c1 ZINC000880964595 FH On-Demand Anodyne RBP4 42 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1cccc(F)c1 ZINC000880964596 FH On-Demand Anodyne RBP4 42 38 CN(C)S(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964597 GD On-Demand Anodyne EPHX2 31 40 CN(C)S(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964597 GD On-Demand Anodyne SFRP1 50 33 CN(C)S(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964597 GD On-Demand Anodyne WNT3 40 33 CCS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)C1 ZINC000880964598 GD On-Demand Anodyne RBP4 63 42 CO[C@@](C)(CNC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880964600 DG On-Demand Anodyne TRPV1 20 42 CCC1(O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964619 CE On-Demand Anodyne TRPV1 15 40 CCC1(O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964619 CE On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880964628 GH On-Demand Anodyne EPHX2 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@](CO)(Cc2ccccc2)C1 ZINC000880964628 GH On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880964629 GH On-Demand Anodyne EPHX2 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@](CO)(Cc2ccccc2)C1 ZINC000880964629 GH On-Demand Anodyne RBP4 65 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCOC2)nn1 ZINC000880964633 DD On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCOC2)nn1 ZINC000880964633 DD On-Demand Anodyne TPP2 47 32 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCC2)O1 ZINC000880964634 EG On-Demand Anodyne RBP4 55 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCC2)O1 ZINC000880964635 EG On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)NC1CC2(CCC2)C1 ZINC000880964636 CH On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)NC1CC2(CCC2)C1 ZINC000880964636 CH On-Demand Anodyne EPHX2 15 43 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCCCO2)nn1 ZINC000880964637 EE On-Demand Anodyne DRD4 25 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCCCO2)nn1 ZINC000880964637 EE On-Demand Anodyne TPP2 46 32 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCCCO2)nn1 ZINC000880964638 EE On-Demand Anodyne DRD4 25 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCCCO2)nn1 ZINC000880964638 EE On-Demand Anodyne TPP2 46 32 COC(=O)[C@H]1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964641 DE On-Demand Anodyne EPHX2 32 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2nnnn2CC1 ZINC000880964646 ED On-Demand Anodyne EPHX2 38 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2nnnn2CC1 ZINC000880964647 ED On-Demand Anodyne EPHX2 38 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](C)[C@@H]1C ZINC000880964648 DH On-Demand Anodyne RBP4 54 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)[C@H]1C ZINC000880964649 DH On-Demand Anodyne RBP4 54 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)[C@@H]1C ZINC000880964650 DH On-Demand Anodyne RBP4 54 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](C)[C@H]1C ZINC000880964651 DH On-Demand Anodyne RBP4 54 40 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)c1cccnc1 ZINC000880964652 EH On-Demand Anodyne TRPV1 32 50 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880964657 DD On-Demand Anodyne RBP4 57 41 CN1C(=O)CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880964658 ED On-Demand Anodyne TRPV1 26 43 CN1C(=O)CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880964659 ED On-Demand Anodyne TRPV1 26 43 O=C(Nc1cnccc1C(F)(F)F)N1CCOCCN1 ZINC000880964664 CD On-Demand Anodyne RBP4 41 39 NC(=O)[C@@H]1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964666 EF On-Demand Anodyne TRPV1 20 45 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC(F)F ZINC000880964667 DH On-Demand Anodyne TRPV1 20 47 COCC[C@@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964669 DF On-Demand Anodyne TRPV1 15 45 COCC[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964670 DF On-Demand Anodyne TRPV1 15 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880964675 FF On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880964675 FF On-Demand Anodyne TPP2 59 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880964677 FF On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880964677 FF On-Demand Anodyne TPP2 59 34 O=C(Nc1cnccc1C(F)(F)F)Nc1n[nH]cc1C1CC1 ZINC000880964679 DG On-Demand Anodyne RBP4 50 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCCC2)O1 ZINC000880964680 EH On-Demand Anodyne RBP4 55 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCCC2)O1 ZINC000880964681 EH On-Demand Anodyne RBP4 55 39 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@](=O)C1 ZINC000880964682 EE On-Demand Anodyne RBP4 60 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@](=O)C1 ZINC000880964683 EE On-Demand Anodyne RBP4 60 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@](=O)C1 ZINC000880964684 EE On-Demand Anodyne RBP4 60 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@](=O)C1 ZINC000880964685 EE On-Demand Anodyne RBP4 60 43 O=C(NC[C@H](CO)c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880964688 FG On-Demand Anodyne TRPV1 18 55 O=C(NC[C@@H](CO)c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880964689 FG On-Demand Anodyne TRPV1 18 55 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H]1O ZINC000880964693 CD On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H]1O ZINC000880964693 CD On-Demand Anodyne EPHX2 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880964698 GH On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880964698 GH On-Demand Anodyne TRPM8 41 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880964699 GH On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880964699 GH On-Demand Anodyne TRPM8 41 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880964700 GH On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880964700 GH On-Demand Anodyne TRPM8 41 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880964701 GH On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880964701 GH On-Demand Anodyne TRPM8 41 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]2C[C@H]21 ZINC000880964702 CG On-Demand Anodyne RBP4 57 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2C[C@@H]21 ZINC000880964703 CG On-Demand Anodyne RBP4 57 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]2C[C@@H]21 ZINC000880964704 CG On-Demand Anodyne RBP4 57 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2C[C@H]21 ZINC000880964705 CG On-Demand Anodyne RBP4 57 43 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@](C)(O)c1ccccc1 ZINC000880964708 FH On-Demand Anodyne TRPV1 21 48 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@](C)(O)c1ccccc1 ZINC000880964709 FH On-Demand Anodyne TRPV1 21 48 CCC1(c2ccccc2)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964710 EI On-Demand Anodyne TRPV1 26 43 CCC1(c2ccccc2)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964710 EI On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2COC[C@@H]21 ZINC000880964711 DF On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C2CCCC2)C1 ZINC000880964716 EI On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C2CCCC2)C1 ZINC000880964716 EI On-Demand Anodyne RBP4 91 50 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C2CCCC2)C1 ZINC000880964717 EI On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C2CCCC2)C1 ZINC000880964717 EI On-Demand Anodyne RBP4 91 50 COC(=O)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC1CC1 ZINC000880964719 EF On-Demand Anodyne TRPV1 19 42 COC(=O)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC1CC1 ZINC000880964720 EF On-Demand Anodyne TRPV1 19 42 COc1cccc([C@H](CO)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964726 FF On-Demand Anodyne TRPV1 23 51 COc1cccc([C@H](CO)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964726 FF On-Demand Anodyne ROCK1 25 46 COc1cccc([C@H](CO)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964726 FF On-Demand Anodyne RAF1 19 40 COc1cccc([C@H](CO)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964726 FF On-Demand Anodyne ROCK2 43 35 COc1cccc([C@H](CO)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964726 FF On-Demand Anodyne TAAR1 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](n2ccnn2)C1 ZINC000880964728 EF On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](n2ccnn2)C1 ZINC000880964729 EF On-Demand Anodyne RBP4 58 42 C#C[C@@H](CCC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880964734 CG On-Demand Mild TRPV1 15 44 CSC1(CNC(=O)Nc2cnccc2C(F)(F)F)CCN(C)CC1 ZINC000880964746 FG On-Demand Anodyne TRPV1 16 44 N#Cc1ccc(O[C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)nc1 ZINC000880964748 GG On-Demand Mild RBP4 60 40 N#Cc1ccc(O[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)nc1 ZINC000880964749 GG On-Demand Mild RBP4 60 40 Cn1nncc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964750 DD On-Demand Anodyne TRPV1 19 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CC(F)(F)F)CC1 ZINC000880964751 FI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CC(F)(F)F)CC1 ZINC000880964751 FI On-Demand Anodyne RBP4 73 43 COc1cccc([C@H]2C[C@H](O)CN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964757 GG On-Demand Anodyne RBP4 47 38 COc1cccc([C@H]2C[C@@H](O)CN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880964759 GG On-Demand Anodyne RBP4 47 38 O=C1C[C@@H]([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880964762 FE On-Demand Anodyne RBP4 65 45 O=C1C[C@H]([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880964763 FE On-Demand Anodyne RBP4 65 45 O=C1C[C@H]([C@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880964764 FE On-Demand Anodyne RBP4 65 45 O=C1C[C@@H]([C@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880964765 FE On-Demand Anodyne RBP4 65 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C1)Oc1ccccc1O2 ZINC000880964766 FH On-Demand Anodyne NPY5R 31 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C1)Oc1ccccc1O2 ZINC000880964766 FH On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C1)Oc1ccccc1O2 ZINC000880964766 FH On-Demand Anodyne TRPM8 23 40 COC1(c2ccccc2)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964772 FG On-Demand Anodyne RBP4 71 43 COC[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880964774 CD On-Demand Anodyne TRPV1 15 44 COC(=O)[C@@]1(C(F)(F)F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964779 GG On-Demand Anodyne RBP4 48 38 CN1C(=O)N[C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CC[C@@H]21 ZINC000880964783 ED On-Demand Anodyne RBP4 67 42 O=C(Nc1cnccc1C(F)(F)F)N1CC2(CCCOC2)C1 ZINC000880964786 DF On-Demand Anodyne RBP4 41 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCn2c(cc3ccccc32)C1 ZINC000880964788 FI On-Demand Anodyne RBP4 57 41 O=C(NC[C@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964792 GH On-Demand Anodyne TRPV1 21 41 O=C(NC[C@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964792 GH On-Demand Anodyne CCR3 17 41 O=C(NC[C@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964792 GH On-Demand Anodyne PIM1 22 41 O=C(NC[C@@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964793 GH On-Demand Anodyne TRPV1 21 41 O=C(NC[C@@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964793 GH On-Demand Anodyne CCR3 17 41 O=C(NC[C@@H]1CCN(c2ccccc2F)C1)Nc1cnccc1C(F)(F)F ZINC000880964793 GH On-Demand Anodyne PIM1 22 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne TRPV1 31 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne CCR3 16 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne EPHX2 60 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne RBP4 89 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne SFRP1 119 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne TRPM8 40 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964796 GH On-Demand Anodyne WNT3 82 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne TRPV1 31 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne CCR3 16 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne EPHX2 60 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne RBP4 89 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne SFRP1 119 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne TRPM8 40 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)Nc2ccccc2)C1 ZINC000880964797 GH On-Demand Anodyne WNT3 82 41 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1nc(C2CC2)no1 ZINC000880964801 GF On-Demand Anodyne RBP4 57 40 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1nc(C2CC2)no1 ZINC000880964802 GF On-Demand Anodyne RBP4 57 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)(F)F)CC1 ZINC000880964811 FG On-Demand Anodyne SLC6A5 29 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)(F)F)CC1 ZINC000880964811 FG On-Demand Anodyne EPHX2 45 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)(F)F)CC1 ZINC000880964811 FG On-Demand Anodyne CXCR3 20 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)(F)F)CC1 ZINC000880964811 FG On-Demand Anodyne HPGDS 44 47 CON(C)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964819 FE On-Demand Anodyne RBP4 66 43 CON(C)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964819 FE On-Demand Anodyne SFRP1 58 33 CON(C)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964819 FE On-Demand Anodyne WNT3 48 32 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCC1(F)F ZINC000880964820 DH On-Demand Anodyne RBP4 66 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCC1(F)F ZINC000880964821 DH On-Demand Anodyne RBP4 66 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](F)(CO)C1 ZINC000880964829 DE On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](F)(CO)C1 ZINC000880964830 DE On-Demand Anodyne RBP4 61 42 CN(C)S(=O)(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964831 GD On-Demand Anodyne RBP4 60 41 CN(C)S(=O)(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964831 GD On-Demand Anodyne SFRP1 60 33 CN(C)S(=O)(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964831 GD On-Demand Anodyne WNT3 56 33 CN(C)S(=O)(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964832 GD On-Demand Anodyne RBP4 60 41 CN(C)S(=O)(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964832 GD On-Demand Anodyne SFRP1 60 33 CN(C)S(=O)(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964832 GD On-Demand Anodyne WNT3 56 33 O=C(NCC1CCC(F)CC1)Nc1cnccc1C(F)(F)F ZINC000880964836 DH On-Demand Anodyne TRPV1 25 47 CN(C)C1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964841 EG On-Demand Anodyne EPHX2 47 45 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)N1CC#N ZINC000880964846 EF On-Demand Mild RBP4 78 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)N1CC#N ZINC000880964847 EF On-Demand Mild RBP4 78 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)N1CC#N ZINC000880964848 EF On-Demand Mild RBP4 78 47 O=C(NCCS(=O)(=O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880964850 ED On-Demand Anodyne TRPV1 17 44 CCOCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880964851 FF On-Demand Anodyne RBP4 54 39 CCOCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880964852 FF On-Demand Anodyne RBP4 54 39 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN2CCOC2=O)nn1 ZINC000880964854 ED On-Demand Anodyne DRD4 29 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN2CCOC2=O)nn1 ZINC000880964854 ED On-Demand Anodyne TPP2 43 32 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCC2)S(=O)(=O)CC1 ZINC000880964856 GF On-Demand Anodyne RBP4 48 38 C=C[C@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964857 DD On-Demand Mild DRD4 28 48 C=C[C@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964857 DD On-Demand Mild TPP2 51 33 C=C[C@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964858 DD On-Demand Mild DRD4 28 48 C=C[C@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964858 DD On-Demand Mild TPP2 51 33 C=C[C@@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964859 DD On-Demand Mild DRD4 28 48 C=C[C@@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880964859 DD On-Demand Mild TPP2 51 33 C=C[C@@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964860 DD On-Demand Mild DRD4 28 48 C=C[C@@](C)(O)c1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880964860 DD On-Demand Mild TPP2 51 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2CCCC[C@@H]21 ZINC000880964867 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)[C@H](CO)C1 ZINC000880964868 DD On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](O)[C@@H](CO)C1 ZINC000880964869 DD On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](O)[C@H](CO)C1 ZINC000880964870 DD On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)[C@@H](CO)C1 ZINC000880964871 DD On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)[C@H]1c1ccc(Cl)cc1 ZINC000880964872 GI On-Demand Anodyne RBP4 46 36 O=C1C[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964873 GH On-Demand Anodyne NPY5R 27 43 O=C1C[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964873 GH On-Demand Anodyne EPHX2 26 41 O=C1C[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964873 GH On-Demand Anodyne RBP4 55 38 O=C1C[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964873 GH On-Demand Anodyne TRPM8 32 44 O=C1C[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964874 GH On-Demand Anodyne NPY5R 27 43 O=C1C[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964874 GH On-Demand Anodyne EPHX2 26 41 O=C1C[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964874 GH On-Demand Anodyne RBP4 55 38 O=C1C[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)Oc2ccccc21 ZINC000880964874 GH On-Demand Anodyne TRPM8 32 44 CC(=O)c1cccc(OCc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)c1 ZINC000880964875 GG On-Demand Anodyne DRD4 28 46 CC(=O)c1cccc(OCc2cn(CC(=O)N3c4ccccc4C[C@@H]3C)nn2)c1 ZINC000880964875 GG On-Demand Anodyne TPP2 49 34 CC(=O)c1cccc(OCc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)c1 ZINC000880964876 GG On-Demand Anodyne DRD4 28 46 CC(=O)c1cccc(OCc2cn(CC(=O)N3c4ccccc4C[C@H]3C)nn2)c1 ZINC000880964876 GG On-Demand Anodyne TPP2 49 34 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880964877 EE On-Demand Anodyne RBP4 66 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880964885 FD On-Demand Anodyne ABL1 40 34 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880964885 FD On-Demand Anodyne ABL2 43 33 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2nc[nH]n2)CC1 ZINC000880964885 FD On-Demand Anodyne RBP4 41 38 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(CC3CC3)nnc2C1 ZINC000880964895 FF On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cccc(Cl)c2C1 ZINC000880964897 FI On-Demand Anodyne RBP4 61 44 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cccc(Cl)c2C1 ZINC000880964897 FI On-Demand Anodyne P2RY14 36 40 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964899 DD On-Demand Anodyne RBP4 75 44 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964899 DD On-Demand Anodyne SFRP1 75 35 CC(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964899 DD On-Demand Anodyne WNT3 61 33 CC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964901 DD On-Demand Anodyne RBP4 75 44 CC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964901 DD On-Demand Anodyne SFRP1 75 35 CC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964901 DD On-Demand Anodyne WNT3 61 33 CNC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964903 DD On-Demand Anodyne RBP4 75 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880964907 FD On-Demand Anodyne DRD4 28 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880964907 FD On-Demand Anodyne TPP2 56 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](O)CC1 ZINC000880964910 DF On-Demand Anodyne TRPV1 26 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](O)CC1 ZINC000880964910 DF On-Demand Anodyne EPHX2 45 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880964924 FF On-Demand Anodyne DRD4 28 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880964924 FF On-Demand Anodyne TPP2 59 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880964929 FF On-Demand Anodyne DRD4 28 49 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880964929 FF On-Demand Anodyne TPP2 59 34 COc1ccc(N2CC[C@H](CNC(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880964932 GH On-Demand Clean F10 17 47 COc1ccc(N2CC[C@H](CNC(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880964932 GH On-Demand Clean TRPV1 16 41 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880964937 FE On-Demand Clean DRD4 25 51 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880964937 FE On-Demand Clean TPP2 65 35 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(F)(F)F ZINC000880964954 DG On-Demand Anodyne TRPV1 23 49 COCC(C)(C)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880964955 FF On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)[C@@H](CO)C1 ZINC000880964957 DC On-Demand Anodyne RBP4 75 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)[C@H](CO)C1 ZINC000880964958 DC On-Demand Anodyne RBP4 75 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)[C@@H](CO)C1 ZINC000880964959 DC On-Demand Anodyne RBP4 75 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](CO)[C@@H](O)C1 ZINC000880964960 DC On-Demand Anodyne RBP4 75 45 Cn1ncc2c1CCCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880964962 EF On-Demand Anodyne RBP4 53 40 COC(=O)[C@H]1CN(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964963 FD On-Demand Anodyne RBP4 59 42 COC(=O)[C@@H]1CN(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880964964 FD On-Demand Anodyne RBP4 59 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880965058 DI On-Demand Anodyne TRPV1 24 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880965058 DI On-Demand Anodyne RBP4 86 46 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880965059 DI On-Demand Anodyne TRPV1 24 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)c2ccccc21 ZINC000880965059 DI On-Demand Anodyne RBP4 86 46 CC[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)C(=O)OC ZINC000880965061 DE On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCCS2(=O)=O)CC1 ZINC000880965062 GE On-Demand Anodyne RBP4 71 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCC2=O)CC1 ZINC000880965063 FG On-Demand Anodyne RBP4 58 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCC2=O)CC1 ZINC000880965064 FG On-Demand Anodyne RBP4 58 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2CCOCC2)CC1 ZINC000880965065 FH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2CCOCC2)CC1 ZINC000880965065 FH On-Demand Anodyne RBP4 73 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)C2CC2)nn1 ZINC000880965069 DD On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H](O)C2CC2)nn1 ZINC000880965069 DD On-Demand Anodyne TPP2 60 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)C2CC2)nn1 ZINC000880965071 DD On-Demand Anodyne DRD4 27 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H](O)C2CC2)nn1 ZINC000880965071 DD On-Demand Anodyne TPP2 60 34 O=C(NCc1nc(C(F)F)no1)Nc1cnccc1C(F)(F)F ZINC000880965075 EF On-Demand Anodyne TRPV1 16 48 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C(C)(C)NC(=O)OC(C)(C)C)nn1 ZINC000880965081 GG On-Demand Anodyne DRD4 25 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C(C)(C)NC(=O)OC(C)(C)C)nn1 ZINC000880965081 GG On-Demand Anodyne TPP2 54 32 COCC1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965083 EG On-Demand Anodyne TRPV1 27 40 COCC1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965083 EG On-Demand Anodyne EPHX2 45 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2CC3(C2)OCCO3)nn1 ZINC000880965088 FD On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2CC3(C2)OCCO3)nn1 ZINC000880965088 FD On-Demand Anodyne TPP2 47 32 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CCCCCCO)nn1 ZINC000880965093 EE On-Demand Anodyne DRD4 27 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CCCCCCO)nn1 ZINC000880965093 EE On-Demand Anodyne TPP2 60 39 COC(=O)Cc1cn(CC(=O)N2CCc3ccccc32)nn1 ZINC000880965094 DC On-Demand Anodyne EIF2AK3 50 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC12CC2 ZINC000880965097 CF On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC12CC2 ZINC000880965098 CF On-Demand Anodyne TRPV1 20 42 C[C@@H]1O[C@H](C)C[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965106 DG On-Demand Anodyne TRPV1 15 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CC(C)(C)O)nn1 ZINC000880965107 DD On-Demand Anodyne DRD4 28 51 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CC(C)(C)O)nn1 ZINC000880965107 DD On-Demand Anodyne TPP2 64 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C2CCC2)C1 ZINC000880965115 DH On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C2CCC2)C1 ZINC000880965115 DH On-Demand Anodyne RBP4 91 50 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C2CCC2)C1 ZINC000880965116 DH On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C2CCC2)C1 ZINC000880965116 DH On-Demand Anodyne RBP4 91 50 Cc1nnc(COC2CN(C(=O)Nc3cnccc3C(F)(F)F)C2)o1 ZINC000880965117 FE On-Demand Anodyne RBP4 56 41 C[C@@H](Cc1cccc(F)c1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880965119 FI On-Demand Anodyne TRPV1 25 46 C[C@@H](Cc1cccc(F)c1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880965119 FI On-Demand Anodyne NPY5R 16 42 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCOCC2)nn1 ZINC000880965125 ED On-Demand Anodyne DRD4 26 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(C2(O)CCOCC2)nn1 ZINC000880965125 ED On-Demand Anodyne TPP2 48 32 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1Cl ZINC000880965130 FI On-Demand Anodyne RAF1 31 42 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1Cl ZINC000880965130 FI On-Demand Anodyne PDE6A 43 33 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne TRPV1 19 40 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne CCR2 27 40 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne EPHX2 28 42 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne CYP2C9 22 40 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne RBP4 91 46 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne SFRP1 93 35 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne SCD 23 44 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne WNT3 70 33 O=C(NCc1ccccc1)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965133 GG On-Demand Anodyne NAMPT 93 38 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne TRPV1 19 40 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne CCR2 27 40 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne EPHX2 28 42 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne CYP2C9 22 40 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne RBP4 91 46 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne SFRP1 93 35 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne SCD 23 44 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne WNT3 70 33 O=C(NCc1ccccc1)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965134 GG On-Demand Anodyne NAMPT 93 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC2CCC2)CC1 ZINC000880965136 EH On-Demand Anodyne EPHX2 22 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC2CCC2)CC1 ZINC000880965136 EH On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1ccccc1 ZINC000880965141 FG On-Demand Anodyne RBP4 79 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1ccccc1 ZINC000880965142 FG On-Demand Anodyne RBP4 79 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1ccccc1 ZINC000880965143 FG On-Demand Anodyne RBP4 79 45 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1ccccc1 ZINC000880965144 FG On-Demand Anodyne RBP4 79 45 COc1ccc([C@@H](CO)CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965151 FG On-Demand Anodyne TRPV1 23 55 COc1ccc([C@H](CO)CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965153 FG On-Demand Anodyne TRPV1 23 55 C[C@H]1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965159 DH On-Demand Anodyne TRPV1 31 45 C[C@H]1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965160 DH On-Demand Anodyne TRPV1 31 45 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](CC)O1 ZINC000880965161 EH On-Demand Anodyne RBP4 75 45 N#Cc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880965164 GI On-Demand Mild EPHX2 27 46 N#Cc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880965164 GI On-Demand Mild RBP4 54 38 N#Cc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880965164 GI On-Demand Mild SCD1 17 41 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne DRD4 34 45 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne ACHE 45 48 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne HTR4 30 41 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne TRPV1 23 42 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne SIGMAR1 38 48 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne CCR3 78 46 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne CCR2 29 40 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne RBP4 53 38 O=C(NC[C@@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965166 GH On-Demand Anodyne CACNA1I 47 41 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne DRD4 34 45 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne ACHE 45 48 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne HTR4 30 41 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne TRPV1 23 42 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne SIGMAR1 38 48 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne CCR3 78 46 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne CCR2 29 40 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne RBP4 53 38 O=C(NC[C@H]1CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880965167 GH On-Demand Anodyne CACNA1I 47 41 O=C(c1ccc(CN2CCOCC2)o1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880965196 GE On-Demand Anodyne SIGMAR1 47 39 Cn1nccc1[C@@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880965197 FH On-Demand Anodyne RBP4 45 37 Cn1nccc1[C@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880965198 FH On-Demand Anodyne RBP4 45 37 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]2(CCO[C@@H]2C)O1 ZINC000880965199 FF On-Demand Anodyne RBP4 54 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]2(CCO[C@@H]2C)O1 ZINC000880965201 FF On-Demand Anodyne RBP4 54 39 C[C@@H]1OCC[C@]12CN(C(=O)Nc1cnccc1C(F)(F)F)C[C@@H](C)O2 ZINC000880965202 FF On-Demand Anodyne RBP4 54 39 O=C(c1cnc(CC2CC2)s1)N1CC(c2ccccc2)C1 ZINC000880965205 CG On-Demand Anodyne CCR5 20 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)CC1CC1 ZINC000880965206 DE On-Demand Anodyne TRPV1 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)CC1CC1 ZINC000880965207 DE On-Demand Anodyne TRPV1 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](c2ccccc2)C1 ZINC000880965218 EI On-Demand Anodyne TRPV1 27 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](c2ccccc2)C1 ZINC000880965218 EI On-Demand Anodyne EPHX2 22 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H](c2ccccc2)C1 ZINC000880965218 EI On-Demand Anodyne RBP4 67 42 O=C(Nc1cnccc1C(F)(F)F)NC1CC(c2ccccc2)C1 ZINC000880965219 EI On-Demand Anodyne TRPV1 27 45 O=C(Nc1cnccc1C(F)(F)F)NC1CC(c2ccccc2)C1 ZINC000880965219 EI On-Demand Anodyne EPHX2 22 43 O=C(Nc1cnccc1C(F)(F)F)NC1CC(c2ccccc2)C1 ZINC000880965219 EI On-Demand Anodyne RBP4 67 42 Cc1ccncc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965221 FG On-Demand Anodyne TRPV1 19 53 Cc1ccncc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965221 FG On-Demand Anodyne RBP4 59 44 O=C(c1cnc2cc[nH]c2c1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880965222 EF On-Demand Anodyne FAAH 19 47 O=C(c1cnc2cc[nH]c2c1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880965222 EF On-Demand Anodyne CCR8 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880965223 GG On-Demand Anodyne EPHX2 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880965223 GG On-Demand Anodyne RBP4 69 41 Cc1noc(C2CN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880965224 EE On-Demand Anodyne RBP4 67 44 Cc1noc(C2CN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880965224 EE On-Demand Anodyne SMO 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ncccc2F)CC1 ZINC000880965225 GH On-Demand Anodyne TRPV1 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ncccc2F)CC1 ZINC000880965225 GH On-Demand Anodyne EPHX2 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ncccc2F)CC1 ZINC000880965225 GH On-Demand Anodyne RBP4 66 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ncccc2F)CC1 ZINC000880965225 GH On-Demand Anodyne SCD 26 44 C[C@]1(O)CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965229 DF On-Demand Anodyne RBP4 60 41 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(N)=O ZINC000880965234 CD On-Demand Anodyne TRPV1 17 48 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCS1(=O)=O ZINC000880965240 FE On-Demand Anodyne RBP4 70 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCS1(=O)=O ZINC000880965241 FE On-Demand Anodyne RBP4 70 41 NOCc1cn(CC(=O)N2CCc3ccccc3C2)nn1 ZINC000880965243 CC On-Demand Anodyne DPP8 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cccc(F)c2C1 ZINC000880965244 EH On-Demand Anodyne RBP4 59 42 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](CC)O1 ZINC000880965253 EH On-Demand Anodyne RBP4 75 45 N#C[C@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965262 CF On-Demand Mild EPHX2 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CO)C1 ZINC000880965264 CD On-Demand Anodyne RBP4 81 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CO)C1 ZINC000880965265 CD On-Demand Anodyne RBP4 81 45 O=C(Nc1cnccc1C(F)(F)F)N1CC(N2CC[C@@H](O)C2)C1 ZINC000880965266 ED On-Demand Anodyne RBP4 76 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880965268 FE On-Demand Anodyne DRD4 24 46 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880965268 FE On-Demand Anodyne TPP2 52 33 COC(=O)[C@H]1CSCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965275 FE On-Demand Anodyne RBP4 57 41 COC(=O)[C@@H]1CSCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965276 FE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCS(=O)(=O)C2)C1 ZINC000880965280 GD On-Demand Anodyne EPHX2 16 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCS(=O)(=O)C2)C1 ZINC000880965280 GD On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCS(=O)(=O)C2)C1 ZINC000880965283 GD On-Demand Anodyne EPHX2 16 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCS(=O)(=O)C2)C1 ZINC000880965283 GD On-Demand Anodyne RBP4 40 37 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880965285 GF On-Demand Anodyne DRD4 24 44 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2c3ccccc3C[C@H]2C)nn1 ZINC000880965285 GF On-Demand Anodyne TPP2 52 33 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880965287 GF On-Demand Anodyne DRD4 24 44 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2c3ccccc3C[C@@H]2C)nn1 ZINC000880965287 GF On-Demand Anodyne TPP2 52 33 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880965293 CG On-Demand Anodyne TRPV1 24 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]2C[C@@H]2C1 ZINC000880965293 CG On-Demand Anodyne EPHX2 32 44 O=C(Nc1cnccc1C(F)(F)F)NC1C[C@H]2C[C@@H]2C1 ZINC000880965296 CG On-Demand Anodyne TRPV1 24 41 O=C(Nc1cnccc1C(F)(F)F)NC1C[C@H]2C[C@@H]2C1 ZINC000880965296 CG On-Demand Anodyne EPHX2 32 44 O=C(Nc1cnccc1C(F)(F)F)NC1C[C@@H]2C[C@H]2C1 ZINC000880965298 CG On-Demand Anodyne TRPV1 24 41 O=C(Nc1cnccc1C(F)(F)F)NC1C[C@@H]2C[C@H]2C1 ZINC000880965298 CG On-Demand Anodyne EPHX2 32 44 CN1CCO[C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]21 ZINC000880965314 ED On-Demand Anodyne RBP4 60 43 O=C(NCc1nnc(C2CC2)s1)Nc1cnccc1C(F)(F)F ZINC000880965316 EG On-Demand Anodyne TRPV1 15 45 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880965318 DI On-Demand Anodyne TRPV1 22 62 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880965318 DI On-Demand Anodyne TACR3 51 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](C2CCC2)C1 ZINC000880965325 EG On-Demand Anodyne RBP4 70 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](C2CCC2)C1 ZINC000880965327 EG On-Demand Anodyne RBP4 70 44 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)N1CCc2ccccc21 ZINC000880965339 GC On-Demand Anodyne DRD4 15 51 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@@H](O)CC[C@H]2C1 ZINC000880965342 EF On-Demand Anodyne RBP4 95 53 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CC[C@H](O)C[C@H]2C1 ZINC000880965343 EF On-Demand Anodyne RBP4 95 53 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CC[C@@H](O)C[C@H]2C1 ZINC000880965345 EF On-Demand Anodyne RBP4 95 53 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@H](O)CC[C@H]2C1 ZINC000880965347 EF On-Demand Anodyne RBP4 95 53 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CCO)CC1 ZINC000880965353 EG On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CCO)CC1 ZINC000880965354 EG On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880965365 FF On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880965365 FF On-Demand Anodyne EPHX2 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880965365 FF On-Demand Anodyne RBP4 79 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880965365 FF On-Demand Anodyne SFRP1 79 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ncccn2)C1 ZINC000880965365 FF On-Demand Anodyne WNT3 61 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880965367 FF On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880965367 FF On-Demand Anodyne EPHX2 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880965367 FF On-Demand Anodyne RBP4 79 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880965367 FF On-Demand Anodyne SFRP1 79 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ncccn2)C1 ZINC000880965367 FF On-Demand Anodyne WNT3 61 34 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@]2(O)CCOC2)nn1 ZINC000880965378 EC On-Demand Anodyne DRD4 25 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@]2(O)CCOC2)nn1 ZINC000880965378 EC On-Demand Anodyne TPP2 43 31 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@]2(O)CCOC2)nn1 ZINC000880965380 EC On-Demand Anodyne DRD4 25 44 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@]2(O)CCOC2)nn1 ZINC000880965380 EC On-Demand Anodyne TPP2 43 31 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CON)nn1 ZINC000880965383 CC On-Demand Anodyne DRD4 28 51 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CON)nn1 ZINC000880965383 CC On-Demand Anodyne TPP2 67 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOC1=O ZINC000880965384 CD On-Demand Anodyne TRPV1 29 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOC1=O ZINC000880965384 CD On-Demand Anodyne LUXR 77 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOC1=O ZINC000880965384 CD On-Demand Anodyne TRAR 93 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOC1=O ZINC000880965384 CD On-Demand Anodyne LASR 58 38 Cc1ccc2c(c1)[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880965385 EI On-Demand Anodyne TRPV1 32 51 Cc1ccc2c(c1)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880965386 EI On-Demand Anodyne TRPV1 32 51 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCCC(=O)C2)nn1 ZINC000880965393 EE On-Demand Anodyne DRD4 25 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@H]2CCCC(=O)C2)nn1 ZINC000880965393 EE On-Demand Anodyne TPP2 48 32 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCCC(=O)C2)nn1 ZINC000880965395 EE On-Demand Anodyne DRD4 25 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc([C@@H]2CCCC(=O)C2)nn1 ZINC000880965395 EE On-Demand Anodyne TPP2 48 32 N#CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965398 CF On-Demand Mild RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880965402 DF On-Demand Anodyne EPHX2 28 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@@H](CO)C1 ZINC000880965402 DF On-Demand Anodyne PTGES 17 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H](CO)C1 ZINC000880965403 DF On-Demand Anodyne EPHX2 28 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H](CO)C1 ZINC000880965403 DF On-Demand Anodyne PTGES 17 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@H](CO)C1 ZINC000880965404 DF On-Demand Anodyne EPHX2 28 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@H](CO)C1 ZINC000880965404 DF On-Demand Anodyne PTGES 17 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@@H](CO)C1 ZINC000880965405 DF On-Demand Anodyne EPHX2 28 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@@H](CO)C1 ZINC000880965405 DF On-Demand Anodyne PTGES 17 41 C[S@@](=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965407 CD On-Demand Anodyne TRPV1 17 47 NC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880965410 GF On-Demand Anodyne RBP4 84 48 NC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ccccc1 ZINC000880965410 GF On-Demand Anodyne SMO 29 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)CCF ZINC000880965412 CD On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)CCF ZINC000880965413 CD On-Demand Anodyne TRPV1 17 43 Cn1cc(CNC(=O)Nc2cnccc2C(F)(F)F)nn1 ZINC000880965416 DD On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COCc2ccccc21 ZINC000880965419 EG On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COCc2ccccc21 ZINC000880965419 EG On-Demand Anodyne RBP4 54 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COCc2ccccc21 ZINC000880965420 EG On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COCc2ccccc21 ZINC000880965420 EG On-Demand Anodyne RBP4 54 40 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)N2CCc3ccccc32)nn1 ZINC000880965423 FE On-Demand Anodyne EIF2AK3 43 33 O=C(CCCc1ccccc1)NCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965426 GG On-Demand Anodyne TRPV1 25 54 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN2CCS(=O)(=O)CC2)nn1 ZINC000880965428 GC On-Demand Anodyne DRD4 34 54 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN2CCS(=O)(=O)CC2)nn1 ZINC000880965428 GC On-Demand Anodyne TPP2 48 33 C[C@H]1C[C@H](CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965438 DF On-Demand Anodyne RBP4 79 47 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN(C)CC(=O)OC(C)(C)C)nn1 ZINC000880965443 GE On-Demand Anodyne DRD4 24 45 C[C@@H]1Cc2ccccc2N1C(=O)Cn1cc(CN(C)CC(=O)OC(C)(C)C)nn1 ZINC000880965443 GE On-Demand Anodyne TPP2 40 32 O=C(Nc1cnccc1C(F)(F)F)N1CCCN2c3ccccc3C[C@H]2C1 ZINC000880965457 GH On-Demand Anodyne RBP4 68 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCN2c3ccccc3C[C@@H]2C1 ZINC000880965458 GH On-Demand Anodyne RBP4 68 44 O=C(NCCC1(O)CCC1)Nc1cnccc1C(F)(F)F ZINC000880965464 DF On-Demand Anodyne TRPV1 15 47 CCc1nnc(CNC(=O)Nc2cnccc2C(F)(F)F)s1 ZINC000880965474 EF On-Demand Anodyne TRPV1 17 48 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2F)CC1 ZINC000880965475 GH On-Demand Anodyne KCNQ2 63 37 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2F)CC1 ZINC000880965475 GH On-Demand Anodyne TRPV1 18 57 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2F)CC1 ZINC000880965475 GH On-Demand Anodyne RBP4 62 47 O=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cnccc1C(F)(F)F ZINC000880965476 DF On-Demand Anodyne RBP4 40 38 O=C(NCC1(c2ccccn2)CCC1)Nc1cnccc1C(F)(F)F ZINC000880965477 FH On-Demand Anodyne TRPV1 23 48 O=C(NCC1(c2ccccn2)CCC1)Nc1cnccc1C(F)(F)F ZINC000880965477 FH On-Demand Anodyne NMBR 46 44 O=C(NCC1(c2ccccn2)CCC1)Nc1cnccc1C(F)(F)F ZINC000880965477 FH On-Demand Anodyne GRPR 24 44 CCOC(=O)C1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965481 FG On-Demand Anodyne EPHX2 48 41 Cn1ccnc(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)c1=O ZINC000880965496 GD On-Demand Anodyne TRPV1 19 41 Cn1ccnc(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)c1=O ZINC000880965496 GD On-Demand Anodyne EPHX2 43 40 O=C(NCCCCF)Nc1cnccc1C(F)(F)F ZINC000880965505 CF On-Demand Anodyne TRPV1 22 50 CS(=O)(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965510 GD On-Demand Anodyne RBP4 68 45 CS(=O)(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965510 GD On-Demand Anodyne SFRP1 64 34 CS(=O)(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965510 GD On-Demand Anodyne WNT3 51 32 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)c1ccccc1 ZINC000880965512 EG On-Demand Anodyne TRPV1 17 49 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)c1ccccc1 ZINC000880965513 EG On-Demand Anodyne TRPV1 17 49 CNC(=O)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1cnn(C)c1 ZINC000880965529 GD On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965536 GF On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965536 GF On-Demand Anodyne EPHX2 36 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965536 GF On-Demand Anodyne SFRP1 71 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965536 GF On-Demand Anodyne WNT3 61 34 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965537 GF On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965537 GF On-Demand Anodyne EPHX2 36 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965537 GF On-Demand Anodyne SFRP1 71 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(C(=O)N2CCCC2)C1 ZINC000880965537 GF On-Demand Anodyne WNT3 61 34 O=C(NCC(F)(F)Br)Nc1cnccc1C(F)(F)F ZINC000880965542 EG On-Demand Anodyne TRPV1 22 51 O=C(NC[C@@H](O)c1ccc(C(F)(F)F)cc1)Nc1cnccc1C(F)(F)F ZINC000880965543 GH On-Demand Anodyne TRPV1 24 56 O=C(NC[C@H](O)c1ccc(C(F)(F)F)cc1)Nc1cnccc1C(F)(F)F ZINC000880965544 GH On-Demand Anodyne TRPV1 24 56 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COc2ccccc2[C@H]1O ZINC000880965547 FF On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COc2ccccc2[C@@H]1O ZINC000880965548 FF On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COc2ccccc2[C@@H]1O ZINC000880965549 FF On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COc2ccccc2[C@H]1O ZINC000880965550 FF On-Demand Anodyne TRPV1 25 41 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ccc1F ZINC000880965555 GH On-Demand Anodyne CCR1 25 40 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ccc1F ZINC000880965555 GH On-Demand Anodyne RBP4 54 54 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ccc1F ZINC000880965555 GH On-Demand Anodyne DYRK1B 19 41 COC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965556 DG On-Demand Anodyne RBP4 59 41 C[S@@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965559 FG On-Demand Anodyne TRPV1 22 53 C[S@@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965559 FG On-Demand Anodyne FLT1 16 40 C[S@@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965559 FG On-Demand Anodyne NAMPT 54 36 C[S@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965560 FG On-Demand Anodyne TRPV1 22 53 C[S@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965560 FG On-Demand Anodyne FLT1 16 40 C[S@](=O)Cc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880965560 FG On-Demand Anodyne NAMPT 54 36 COCCCONC(=O)Nc1cnccc1C(F)(F)F ZINC000880965561 CE On-Demand Anodyne TRPV1 16 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@H]2COCC[C@H]21 ZINC000880965573 GI On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@H]2COCC[C@@H]21 ZINC000880965574 GI On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@@H]2COCC[C@H]21 ZINC000880965575 GI On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](c2ccccc2)[C@@H]2COCC[C@@H]21 ZINC000880965576 GI On-Demand Anodyne RBP4 53 38 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880965587 FE On-Demand Anodyne DPP8 18 44 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880965588 FE On-Demand Anodyne DPP8 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880965592 FG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C(F)(F)F)[C@H](CO)C1 ZINC000880965593 FG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C(F)(F)F)[C@H](CO)C1 ZINC000880965594 FG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C(F)(F)F)[C@@H](CO)C1 ZINC000880965595 FG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1c1ccc(F)c(F)c1 ZINC000880965596 GH On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1c1ccc(F)c(F)c1 ZINC000880965597 GH On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@@H]1c1ccc(F)c(F)c1 ZINC000880965598 GH On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@@H]1c1ccc(F)c(F)c1 ZINC000880965599 GH On-Demand Anodyne RBP4 40 37 C[C@@H]1[C@@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965600 CD On-Demand Anodyne CCR5 18 44 C[C@@H]1[C@@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965600 CD On-Demand Anodyne PREP 15 40 C[C@@H]1[C@@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965600 CD On-Demand Anodyne ADAM10 45 41 C[C@H]1[C@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965601 CD On-Demand Anodyne CCR5 18 44 C[C@H]1[C@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965601 CD On-Demand Anodyne PREP 15 40 C[C@H]1[C@H](C(=O)N2CC(c3ccccc3)C2)CCN1C ZINC000880965601 CD On-Demand Anodyne ADAM10 45 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C(=O)N2CCCC2)C1 ZINC000880965606 FF On-Demand Anodyne RBP4 73 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C(=O)N2CCCC2)C1 ZINC000880965606 FF On-Demand Anodyne SFRP1 74 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C(=O)N2CCCC2)C1 ZINC000880965606 FF On-Demand Anodyne WNT3 63 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C(=O)N2CCCC2)C1 ZINC000880965607 FF On-Demand Anodyne RBP4 73 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C(=O)N2CCCC2)C1 ZINC000880965607 FF On-Demand Anodyne SFRP1 74 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C(=O)N2CCCC2)C1 ZINC000880965607 FF On-Demand Anodyne WNT3 63 35 C[C@@H]1COCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965608 DF On-Demand Anodyne TRPV1 17 40 C[C@@H]1COCC[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965611 DF On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](F)(c2ccccc2)C1 ZINC000880965612 FI On-Demand Anodyne RBP4 66 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](F)(c2ccccc2)C1 ZINC000880965613 FI On-Demand Anodyne RBP4 66 45 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965619 GG On-Demand Anodyne RBP4 65 44 O=C(NC[C@H](O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965625 EF On-Demand Anodyne TRPV1 22 56 O=C(NC[C@H](O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965625 EF On-Demand Anodyne GPR142 55 33 O=C(NC[C@@H](O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965626 EF On-Demand Anodyne TRPV1 22 56 O=C(NC[C@@H](O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965626 EF On-Demand Anodyne GPR142 55 33 C[C@@H]1Oc2ccccc2[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965631 EH On-Demand Anodyne TRPV1 25 44 C[C@@H]1Oc2ccccc2[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965633 EH On-Demand Anodyne TRPV1 25 44 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)OCCO ZINC000880965641 DE On-Demand Anodyne TRPV1 17 44 NC(=O)C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965648 DD On-Demand Anodyne RBP4 70 43 NC(=O)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965649 DD On-Demand Anodyne RBP4 70 43 CN(C)S(=O)(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965683 GD On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CNC(=O)C(F)(F)F)C1 ZINC000880965685 GG On-Demand Anodyne RBP4 60 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CNC(=O)C(F)(F)F)C1 ZINC000880965686 GG On-Demand Anodyne RBP4 60 41 C[C@H]1C[C@H](c2ccccc2)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965689 EJ On-Demand Anodyne RBP4 72 44 C[C@@H]1C[C@H](c2ccccc2)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965691 EJ On-Demand Anodyne RBP4 72 44 CC(C)(C)OC(=O)N1CCCN(Cc2cn(CC(=O)NC3CC3)nn2)CC1 ZINC000880965693 GC On-Demand Anodyne KDM1A 19 44 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](C)O ZINC000880965697 CD On-Demand Anodyne TRPV1 17 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)C1CCCC1 ZINC000880965701 DF On-Demand Anodyne TRPV1 15 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)C1CCCC1 ZINC000880965702 DF On-Demand Anodyne TRPV1 15 49 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880965712 CE On-Demand Anodyne RBP4 78 45 O=C(Nc1cnccc1C(F)(F)F)N1CC(C2CC2)C1 ZINC000880965713 CF On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(C2CC2)C1 ZINC000880965713 CF On-Demand Anodyne RBP4 95 53 CCC[C@]1(CO)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965714 EG On-Demand Anodyne RBP4 57 41 Cn1nc(NC(=O)Nc2cnccc2C(F)(F)F)cc1C1CC1 ZINC000880965717 EG On-Demand Anodyne ABL2 40 43 CN(C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965718 GE On-Demand Anodyne RBP4 55 39 CN(C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965718 GE On-Demand Anodyne SFRP1 45 32 CN(C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965718 GE On-Demand Anodyne WNT3 46 32 CN(C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965719 GE On-Demand Anodyne RBP4 55 39 CN(C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965719 GE On-Demand Anodyne SFRP1 45 32 CN(C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1)S(C)(=O)=O ZINC000880965719 GE On-Demand Anodyne WNT3 46 32 C[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965720 ED On-Demand Anodyne TRPV1 16 43 C[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965720 ED On-Demand Anodyne RBP4 60 40 COc1cccc(C2(NC(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880965722 FH On-Demand Anodyne TRPV1 23 43 COc1cccc(C2(NC(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880965722 FH On-Demand Anodyne RAF1 19 40 COc1cccc(C2(NC(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880965722 FH On-Demand Anodyne TAAR1 25 41 C[C@H](CO)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880965730 CD On-Demand Anodyne TRPV1 17 42 C[C@@H](CO)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880965731 CD On-Demand Anodyne TRPV1 17 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](CO)(Cc2ccc(F)cc2)C1 ZINC000880965737 GH On-Demand Anodyne RBP4 54 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](CO)(Cc2ccc(F)cc2)C1 ZINC000880965738 GH On-Demand Anodyne RBP4 54 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC1(F)F ZINC000880965741 DG On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC1(F)F ZINC000880965742 DG On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(F)(c2ccccc2F)C1 ZINC000880965743 FH On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(O)(c2ccccc2)C1 ZINC000880965748 EF On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CC(O)(c2ccccc2)C1 ZINC000880965748 EF On-Demand Anodyne RBP4 81 46 O=C(NC[C@H]1COc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880965749 EG On-Demand Anodyne TRPV1 19 45 O=C(NC[C@@H]1COc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880965750 EG On-Demand Anodyne TRPV1 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCOCC2)CC1 ZINC000880965752 EH On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCCOC2)C1 ZINC000880965754 EF On-Demand Anodyne EPHX2 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCCOC2)C1 ZINC000880965754 EF On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCCOC2)C1 ZINC000880965755 EF On-Demand Anodyne EPHX2 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCCOC2)C1 ZINC000880965755 EF On-Demand Anodyne RBP4 40 37 NC(=O)C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965774 EF On-Demand Anodyne RBP4 62 40 NC(=O)C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965775 EF On-Demand Anodyne RBP4 62 40 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880965776 ED On-Demand Anodyne DPP8 21 45 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)N1CCc2ccccc2C1 ZINC000880965777 ED On-Demand Anodyne DPP8 21 45 C#CCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965787 FE On-Demand Mild EPHX2 19 41 C#CCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965787 FE On-Demand Mild RBP4 74 42 O=C(NC[C@]1(CO)C[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965790 FG On-Demand Anodyne TRPV1 26 51 O=C(NC[C@@]1(CO)C[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965791 FG On-Demand Anodyne TRPV1 26 51 O=C(NC[C@@]1(CO)C[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965792 FG On-Demand Anodyne TRPV1 26 51 O=C(NC[C@]1(CO)C[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880965793 FG On-Demand Anodyne TRPV1 26 51 CCC(CC)(CCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965801 DG On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880965809 FG On-Demand Anodyne EPHX2 32 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](CO)(c2ccccc2)C1 ZINC000880965809 FG On-Demand Anodyne RBP4 72 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880965810 FG On-Demand Anodyne EPHX2 32 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](CO)(c2ccccc2)C1 ZINC000880965810 FG On-Demand Anodyne RBP4 72 44 CN1CCO[C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]21 ZINC000880965811 EE On-Demand Anodyne RBP4 70 41 CN1CCO[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]21 ZINC000880965812 EE On-Demand Anodyne RBP4 70 41 CN1CCO[C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]21 ZINC000880965813 EE On-Demand Anodyne RBP4 70 41 CN1CCO[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]21 ZINC000880965814 EE On-Demand Anodyne RBP4 70 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](n2cc(Cl)cn2)C1 ZINC000880965817 FG On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](n2cc(Cl)cn2)C1 ZINC000880965818 FG On-Demand Anodyne RBP4 66 42 COC(=O)Cc1cn(CC(=O)N2CCc3ccccc3C2)nn1 ZINC000880965835 DC On-Demand Anodyne NOD2 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCCO2 ZINC000880965845 EE On-Demand Anodyne RBP4 57 41 C[C@@](CO)(NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(O)cc1 ZINC000880965846 FF On-Demand Anodyne TRPV1 19 47 O=C(Nc1cnccc1C(F)(F)F)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000880965851 FG On-Demand Anodyne EPHX2 49 47 CC[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880965854 CF On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@H]1CCCO1 ZINC000880965861 EG On-Demand Anodyne RBP4 50 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1[C@@H]1CCCO1 ZINC000880965862 EG On-Demand Anodyne RBP4 50 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@H]1CCCO1 ZINC000880965863 EG On-Demand Anodyne RBP4 50 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1[C@@H]1CCCO1 ZINC000880965864 EG On-Demand Anodyne RBP4 50 38 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880965868 EE On-Demand Anodyne TRPV1 15 42 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880965868 EE On-Demand Anodyne RBP4 68 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880965869 EE On-Demand Anodyne TRPV1 15 42 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880965869 EE On-Demand Anodyne RBP4 68 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880965870 EE On-Demand Anodyne TRPV1 15 42 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880965870 EE On-Demand Anodyne RBP4 68 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880965871 EE On-Demand Anodyne TRPV1 15 42 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880965871 EE On-Demand Anodyne RBP4 68 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1[C@H]2CCC[C@H]21 ZINC000880965875 CG On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1[C@H]2CCC[C@H]21 ZINC000880965875 CG On-Demand Anodyne EPHX2 16 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2CCC[C@H]21 ZINC000880965876 CG On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2CCC[C@H]21 ZINC000880965876 CG On-Demand Anodyne EPHX2 16 43 COCC[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965879 DD On-Demand Anodyne TRPV1 17 41 COCC[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965880 DD On-Demand Anodyne TRPV1 17 41 CCO[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880965906 FH On-Demand Anodyne TRPV1 20 46 CCO[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880965906 FH On-Demand Anodyne SOAT1 19 40 O=C(NCc1ccccc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880965926 FI On-Demand Anodyne KCNQ2 79 43 O=C(NCc1ccccc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880965926 FI On-Demand Anodyne TRPV1 33 59 O=C(NCc1ccccc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880965926 FI On-Demand Anodyne SCN2A 20 45 O=C(NCc1ccccc1N1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880965926 FI On-Demand Anodyne SCN10A 24 45 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NCCF ZINC000880965928 DD On-Demand Anodyne TRPV1 15 45 N#CC1(c2ccccn2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965929 GH On-Demand Mild NPY5R 16 40 N#CC1(c2ccccn2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965929 GH On-Demand Mild RBP4 61 41 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCCO1 ZINC000880965930 DG On-Demand Anodyne RBP4 83 44 O=C(Cn1cc([C@@H]2CCCCO2)nn1)N1CCc2ccccc2C1 ZINC000880965936 EE On-Demand Anodyne CPT1A 25 41 O=C(Cn1cc([C@H]2CCCCO2)nn1)N1CCc2ccccc2C1 ZINC000880965937 EE On-Demand Anodyne CPT1A 25 41 O=C(Nc1cnccc1C(F)(F)F)NC1(C(F)F)CC1 ZINC000880965938 CG On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1CO ZINC000880965940 CD On-Demand Anodyne TRPV1 23 41 O=C(NCC1CCC(F)(F)CC1)Nc1cnccc1C(F)(F)F ZINC000880965945 EI On-Demand Anodyne TRPV1 22 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880965946 GI On-Demand Anodyne TRPV1 21 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880965946 GI On-Demand Anodyne NPY5R 34 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880965946 GI On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880965946 GI On-Demand Anodyne TRPM8 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(n2cnnc2O)CC1 ZINC000880965947 FE On-Demand Anodyne RBP4 66 41 C[C@H]1CCC[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965950 DH On-Demand Anodyne TRPV1 22 43 C[C@H]1CCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965951 DH On-Demand Anodyne TRPV1 22 43 C[C@@H]1CCC[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880965952 DH On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2COC[C@@H](C1)O2 ZINC000880965955 DD On-Demand Anodyne RBP4 75 45 C[C@@H]1CN(CCCNC(=O)Nc2cnccc2C(F)(F)F)CCCO1 ZINC000880965957 FF On-Demand Anodyne CCR3 30 44 Cn1nccc1[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965961 FG On-Demand Anodyne RBP4 67 43 Cn1nccc1[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880965962 FG On-Demand Anodyne RBP4 67 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1NC(=O)OC(C)(C)C ZINC000880965965 GG On-Demand Anodyne RBP4 58 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1NC(=O)OC(C)(C)C ZINC000880965966 GG On-Demand Anodyne RBP4 58 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1NC(=O)OC(C)(C)C ZINC000880965967 GG On-Demand Anodyne RBP4 58 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1NC(=O)OC(C)(C)C ZINC000880965968 GG On-Demand Anodyne RBP4 58 41 Cc1csc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)n1 ZINC000880965969 FG On-Demand Anodyne RBP4 54 38 Cc1csc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)n1 ZINC000880965970 FG On-Demand Anodyne RBP4 54 38 O=C(Cn1cc([C@@H](O)c2ccc(F)cc2)nn1)N1CCc2ccccc2C1 ZINC000880965975 FE On-Demand Anodyne DPP8 21 42 O=C(Cn1cc([C@H](O)c2ccc(F)cc2)nn1)N1CCc2ccccc2C1 ZINC000880965976 FE On-Demand Anodyne DPP8 21 42 COC[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880965977 CE On-Demand Anodyne TRPV1 17 45 CNC(=O)[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880965978 DD On-Demand Anodyne TRPV1 16 46 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne MTOR 20 40 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne EPHX2 58 50 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne CXCR3 15 44 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne RBP4 54 42 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne SFRP1 83 36 COC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880965985 EE On-Demand Anodyne WNT3 65 33 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cncc3ncnn23)CC1 ZINC000880965988 GD On-Demand Anodyne RBP4 42 37 O=C(NCC1CCN(C2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880965991 EG On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cc3ccccc3[nH]2)CC1 ZINC000880965998 GJ On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cc3ccccc3[nH]2)CC1 ZINC000880965998 GJ On-Demand Anodyne RBP4 84 45 COCCONC(=O)Nc1cnccc1C(F)(F)F ZINC000880966000 CD On-Demand Anodyne TRPV1 20 42 O=C(NCC[C@@H](O)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880966001 EF On-Demand Anodyne TRPV1 15 47 O=C(NCC[C@H](O)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880966002 EF On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccnc(O)c2C1 ZINC000880966004 EF On-Demand Anodyne RBP4 55 40 O=C1CC[C@H](c2ccc(C(=O)N3CC(c4ccccc4)C3)cc2)N1 ZINC000880966010 DF On-Demand Anodyne SLC18A3 34 43 O=C1CC[C@H](c2ccc(C(=O)N3CC(c4ccccc4)C3)cc2)N1 ZINC000880966010 DF On-Demand Anodyne L3MBTL3 58 38 O=C1CC[C@@H](c2ccc(C(=O)N3CC(c4ccccc4)C3)cc2)N1 ZINC000880966011 DF On-Demand Anodyne SLC18A3 34 43 O=C1CC[C@@H](c2ccc(C(=O)N3CC(c4ccccc4)C3)cc2)N1 ZINC000880966011 DF On-Demand Anodyne L3MBTL3 58 38 C[C@@H]1OCC[C@]12CN(C(=O)Nc1cnccc1C(F)(F)F)CCO2 ZINC000880966012 EF On-Demand Anodyne RBP4 55 38 O=C(Nc1cnccc1C(F)(F)F)NC1CC(N2CCCCC2)C1 ZINC000880966018 EG On-Demand Anodyne EPHX2 31 43 CSC1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966026 DG On-Demand Anodyne TRPV1 23 48 CC(=O)N1CCN(Cc2cn(CC(=O)N3CCc4ccccc4C3)nn2)CC1 ZINC000880966029 GC On-Demand Anodyne NOD2 40 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC=C(Br)C1 ZINC000880966033 FH On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCS2(=O)=O)C1 ZINC000880966035 GE On-Demand Anodyne RBP4 63 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCS2(=O)=O)C1 ZINC000880966036 GE On-Demand Anodyne RBP4 63 42 N#CC1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966039 CF On-Demand Mild TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CC(C2CCOCC2)C1 ZINC000880966043 EF On-Demand Anodyne RBP4 81 49 N#CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966044 CE On-Demand Mild TRPV1 16 47 C[C@@H](CCCC(F)(F)F)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966048 EI On-Demand Anodyne TRPV1 17 45 COCCO[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966051 EF On-Demand Anodyne RBP4 58 41 COCCO[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966051 EF On-Demand Anodyne LIPG 34 40 COCCO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966052 EF On-Demand Anodyne RBP4 58 41 COCCO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966052 EF On-Demand Anodyne LIPG 34 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCC2)C1 ZINC000880966054 CH On-Demand Anodyne EPHX2 34 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCC2)C1 ZINC000880966054 CH On-Demand Anodyne RBP4 57 41 O=C(Cn1cc(CCCOc2cccnc2F)nn1)N1CCc2ccccc2C1 ZINC000880966056 GE On-Demand Anodyne MMP8 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne EPHX2 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne RBP4 105 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne SFRP1 67 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne SMO 20 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccn2)C1 ZINC000880966057 EH On-Demand Anodyne WNT3 55 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne EPHX2 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne RBP4 105 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne SFRP1 67 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne SMO 20 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccn2)C1 ZINC000880966058 EH On-Demand Anodyne WNT3 55 34 O=C([C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966065 FD On-Demand Anodyne SIGMAR1 30 42 O=C(COC1CC1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966066 CD On-Demand Anodyne CHRM2 15 40 O=C(COC1CC1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966066 CD On-Demand Anodyne CHRM3 15 40 O=C(COC1CC1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966066 CD On-Demand Anodyne SIGMAR1 45 46 CCSCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966067 DG On-Demand Anodyne TRPV1 17 44 C[C@@H](O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966077 CE On-Demand Anodyne TRPV1 18 45 O=C(NCc1nnc(C2CC2)o1)Nc1cnccc1C(F)(F)F ZINC000880966081 EF On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccc(F)c2)C1 ZINC000880966084 FI On-Demand Anodyne CCR5 74 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccc(F)c2)C1 ZINC000880966084 FI On-Demand Anodyne SLC9A1 37 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccc(F)c2)C1 ZINC000880966084 FI On-Demand Anodyne EPHX2 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2cccc(F)c2)C1 ZINC000880966084 FI On-Demand Anodyne RBP4 82 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccc(F)c2)C1 ZINC000880966085 FI On-Demand Anodyne CCR5 74 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccc(F)c2)C1 ZINC000880966085 FI On-Demand Anodyne SLC9A1 37 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccc(F)c2)C1 ZINC000880966085 FI On-Demand Anodyne EPHX2 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2cccc(F)c2)C1 ZINC000880966085 FI On-Demand Anodyne RBP4 82 45 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)C(F)(F)F ZINC000880966086 EH On-Demand Anodyne TRPV1 22 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccncc2)C1 ZINC000880966089 FG On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2COC[C@H]21 ZINC000880966096 CD On-Demand Anodyne TRPV1 21 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880966097 GH On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880966097 GH On-Demand Anodyne SIGMAR1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880966097 GH On-Demand Anodyne FAAH 21 53 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 ZINC000880966097 GH On-Demand Anodyne RBP4 96 55 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](O)C1 ZINC000880966099 CE On-Demand Anodyne RBP4 78 46 CC(C)(C)OC(=O)NC/C=C\CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966107 FG On-Demand Anodyne TRPV1 15 43 CC(C)(C)OC(=O)NC/C=C/CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966108 FG On-Demand Anodyne TRPV1 15 43 CO[C@@]1(C)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966119 DG On-Demand Anodyne RBP4 51 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Oc2ncccc2F)C1 ZINC000880966121 GH On-Demand Anodyne RBP4 60 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Oc2ncccc2F)C1 ZINC000880966122 GH On-Demand Anodyne RBP4 60 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)CC(F)F ZINC000880966125 DE On-Demand Anodyne TRPV1 16 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)CC(F)F ZINC000880966126 DE On-Demand Anodyne TRPV1 16 43 C[C@@H]1NC(=O)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966129 DD On-Demand Anodyne TRPV1 28 41 C[C@@H]1NC(=O)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966130 DD On-Demand Anodyne TRPV1 28 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCS1 ZINC000880966132 DG On-Demand Anodyne RBP4 68 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCS1 ZINC000880966133 DG On-Demand Anodyne RBP4 68 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cnccn2)CC1 ZINC000880966139 FF On-Demand Anodyne EPHX2 18 53 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cnccn2)CC1 ZINC000880966139 FF On-Demand Anodyne RBP4 66 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2cnccn2)CC1 ZINC000880966139 FF On-Demand Anodyne SCD 27 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCC2(CC1)CC2 ZINC000880966145 DH On-Demand Anodyne TRPV1 23 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCC2(CC1)CC2 ZINC000880966145 DH On-Demand Anodyne EPHX2 42 46 O=C(Nc1cnccc1C(F)(F)F)NC1(CO)Cc2ccccc2C1 ZINC000880966146 FF On-Demand Anodyne TRPV1 20 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966147 GI On-Demand Anodyne SLC18A3 34 46 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966147 GI On-Demand Anodyne RBP4 67 41 O=C(c1ccc(F)cc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966147 GI On-Demand Anodyne WNT3A 46 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CN2CCOCC2)C1 ZINC000880966150 FF On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CN2CCOCC2)C1 ZINC000880966151 FF On-Demand Anodyne RBP4 56 41 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild PGC 54 37 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild CCKAR 45 37 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild CTSK 24 40 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild REN 72 41 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild KLK5 22 40 C=CCOC(=O)[C@H](CC(=O)N1CC(c2ccccc2)C1)NC(=O)OC(C)(C)C ZINC000880966152 GF On-Demand Mild FPR1 48 41 O=C1C[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880966153 ED On-Demand Anodyne RBP4 41 38 O=C1C[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)CN1 ZINC000880966154 ED On-Demand Anodyne RBP4 41 38 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966167 GG On-Demand Anodyne TRPV1 24 48 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966167 GG On-Demand Anodyne FAAH 22 49 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966167 GG On-Demand Anodyne RBP4 94 46 O=C(Cc1ccccc1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966167 GG On-Demand Anodyne SFRP1 50 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ncc3n2CCCC3)CC1 ZINC000880966172 GI On-Demand Anodyne RBP4 66 41 COC[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966208 CD On-Demand Anodyne TRPV1 17 43 C[C@@](O)(CO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966209 CC On-Demand Anodyne TRPV1 20 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000880966213 DH On-Demand Anodyne TRPV1 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000880966213 DH On-Demand Anodyne EPHX2 27 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000880966213 DH On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000880966214 DH On-Demand Anodyne TRPV1 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000880966214 DH On-Demand Anodyne EPHX2 27 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000880966214 DH On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000880966215 DH On-Demand Anodyne TRPV1 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000880966215 DH On-Demand Anodyne EPHX2 27 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000880966215 DH On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000880966216 DH On-Demand Anodyne TRPV1 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000880966216 DH On-Demand Anodyne EPHX2 27 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000880966216 DH On-Demand Anodyne RBP4 47 40 O=C(NCc1ccncc1OCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880966218 GH On-Demand Anodyne TRPV1 19 53 O=C(NCCCc1ccccc1F)Nc1cnccc1C(F)(F)F ZINC000880966220 EH On-Demand Anodyne TRPV1 23 51 O=C(Nc1cnccc1C(F)(F)F)N1CCCC12CCC2 ZINC000880966223 CH On-Demand Anodyne RBP4 41 38 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CCS1(=O)=O ZINC000880966224 FF On-Demand Anodyne RBP4 55 39 O=C(NCCCCCO)Nc1cnccc1C(F)(F)F ZINC000880966225 CE On-Demand Anodyne TRPV1 19 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCC1=O ZINC000880966228 DF On-Demand Anodyne RBP4 70 45 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCC1=O ZINC000880966229 DF On-Demand Anodyne RBP4 70 45 CS(=O)(=O)[C@@H]1CCCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966235 FF On-Demand Anodyne RBP4 61 42 CS(=O)(=O)[C@@H]1CCCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966235 FF On-Demand Anodyne SFRP1 70 34 CS(=O)(=O)[C@@H]1CCCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966235 FF On-Demand Anodyne WNT3 64 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCc3ccccc32)CC1 ZINC000880966236 GI On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCc3ccccc32)CC1 ZINC000880966236 GI On-Demand Anodyne SCD1 20 55 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCc3ccccc32)CC1 ZINC000880966236 GI On-Demand Anodyne SFRP1 61 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCc3ccccc32)CC1 ZINC000880966236 GI On-Demand Anodyne WNT3 43 33 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)N1CCCC1 ZINC000880966237 EE On-Demand Anodyne TRPV1 15 44 O=C(NC[C@]1(CO)C[C@@H]1c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880966239 GH On-Demand Anodyne TRPV1 20 45 O=C(NC[C@@]1(CO)C[C@@H]1c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880966240 GH On-Demand Anodyne TRPV1 20 45 O=C(NC[C@@]1(CO)C[C@H]1c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880966241 GH On-Demand Anodyne TRPV1 20 45 O=C(NC[C@]1(CO)C[C@H]1c1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880966242 GH On-Demand Anodyne TRPV1 20 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880966243 GH On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)(Cc2ccccc2)CC1 ZINC000880966243 GH On-Demand Anodyne RBP4 73 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CC2)C(=O)C1 ZINC000880966247 ED On-Demand Anodyne RBP4 61 41 O=C(NCc1ccc2c(n1)CCCC2)Nc1cnccc1C(F)(F)F ZINC000880966250 FH On-Demand Anodyne TRPV1 20 46 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCS(=O)(=O)C1 ZINC000880966254 FD On-Demand Anodyne RBP4 60 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCS(=O)(=O)C1 ZINC000880966255 FD On-Demand Anodyne RBP4 60 43 O=C(Nc1cnccc1C(F)(F)F)N1CC(=O)N(C2CC2)C1 ZINC000880966257 DD On-Demand Anodyne RBP4 55 40 C[C@@H]1OCC[C@]1(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966261 DD On-Demand Anodyne TRPV1 19 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2cc(O)ccc2C1 ZINC000880966262 FG On-Demand Anodyne TRPV1 27 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2cc(O)ccc2C1 ZINC000880966263 FG On-Demand Anodyne TRPV1 27 41 O=C(NCCCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880966265 DH On-Demand Anodyne TRPV1 22 48 O=C1N[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]2CO1 ZINC000880966266 EE On-Demand Anodyne RBP4 81 46 O=C(NCCC1CC(O)C1)Nc1cnccc1C(F)(F)F ZINC000880966267 DE On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2nccs2)CC1 ZINC000880966269 FG On-Demand Anodyne TRPV1 17 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2nccs2)CC1 ZINC000880966269 FG On-Demand Anodyne EPHX2 42 42 O=C(C1CC1)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880966271 EE On-Demand Anodyne RBP4 68 42 O=C(C1CC1)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880966272 EE On-Demand Anodyne RBP4 68 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2ccccc2C1 ZINC000880966273 EI On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2ccccc2C1 ZINC000880966273 EI On-Demand Anodyne RBP4 71 45 CS(=O)(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CCC1 ZINC000880966278 FE On-Demand Anodyne TRPV1 17 45 C[C@@H]1CC[C@H](O)[C@@H]([C@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966279 FH On-Demand Anodyne RBP4 48 39 C[C@@H]1CC[C@H](O)[C@H]([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966280 FH On-Demand Anodyne RBP4 48 39 C[C@@H]1CC[C@H](O)[C@H]([C@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966281 FH On-Demand Anodyne RBP4 48 39 C[C@@H]1CC[C@H](O)[C@@H]([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966282 FH On-Demand Anodyne RBP4 48 39 O=C(Nc1cnccc1C(F)(F)F)NC1CC(F)(F)C1 ZINC000880966290 CG On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnccc1C(F)(F)F)NC1CC(F)(F)C1 ZINC000880966290 CG On-Demand Anodyne EPHX2 22 43 CN(C(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1)c1ccccc1 ZINC000880966292 GH On-Demand Anodyne RBP4 92 46 CN(C(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1)c1ccccc1 ZINC000880966292 GH On-Demand Anodyne SFRP1 96 36 CN(C(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1)c1ccccc1 ZINC000880966292 GH On-Demand Anodyne WNT3 77 36 O=C(COC1CC1)N1CC(c2ccccc2)C1 ZINC000880966295 BD On-Demand Anodyne SLC18A3 46 37 CC(C)(O)CONC(=O)Nc1cnccc1C(F)(F)F ZINC000880966296 CD On-Demand Anodyne TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H]1c1cccc(F)c1 ZINC000880966299 EH On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]1c1cccc(F)c1 ZINC000880966300 EH On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1c1cccc(F)c1 ZINC000880966301 EH On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]1c1cccc(F)c1 ZINC000880966302 EH On-Demand Anodyne TRPV1 37 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(C(F)(F)F)C1 ZINC000880966305 EF On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(C(F)(F)F)C1 ZINC000880966306 EF On-Demand Anodyne RBP4 57 41 NC(=O)[C@@H]1CC[C@H](C(=O)N2CC(c3ccccc3)C2)N1Cc1ccccc1 ZINC000880966309 FE On-Demand Anodyne PREP 56 39 C[C@H]1C[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880966313 EG On-Demand Anodyne TRPV1 19 43 C[C@@H]1CC(CNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880966314 EG On-Demand Anodyne TRPV1 19 43 C[C@H]1CC(CNC(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)O1 ZINC000880966315 EG On-Demand Anodyne TRPV1 19 43 Cc1nc(C(C)C)ncc1C(=O)N1CC(c2ccccc2)C1 ZINC000880966323 CG On-Demand Anodyne SORD 41 31 CCCc1cc(NC(=O)Nc2cnccc2C(F)(F)F)n[nH]1 ZINC000880966335 DG On-Demand Anodyne TRPV1 16 41 CCCc1cc(NC(=O)Nc2cnccc2C(F)(F)F)n[nH]1 ZINC000880966335 DG On-Demand Anodyne RIPK1 40 34 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1Cc2cccc(O)c2C1 ZINC000880966336 EG On-Demand Anodyne TRPV1 28 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1Cc2cccc(O)c2C1 ZINC000880966337 EG On-Demand Anodyne TRPV1 28 41 Cn1nnc(C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)n1 ZINC000880966338 CC On-Demand Anodyne FAAH 20 47 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1c1ccccc12 ZINC000880966341 EJ On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1c1ccccc12 ZINC000880966341 EJ On-Demand Anodyne RBP4 95 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2cccnn2)CC1 ZINC000880966342 FF On-Demand Anodyne TRPV1 22 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2cccnn2)CC1 ZINC000880966342 FF On-Demand Anodyne EPHX2 42 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCOCC2)O1 ZINC000880966343 FF On-Demand Anodyne RBP4 53 38 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC2(CCOCC2)O1 ZINC000880966344 FF On-Demand Anodyne RBP4 53 38 CC(C)(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966349 EI On-Demand Anodyne RBP4 73 44 CC(C)(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966349 EI On-Demand Anodyne SFRP1 59 33 CC(C)(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966349 EI On-Demand Anodyne WNT3 58 33 CC(C)C1(O)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966355 DE On-Demand Anodyne RBP4 59 40 O=C(c1ccc(CN2CCOCC2)o1)N1CC(c2ccccc2)C1 ZINC000880966356 EE On-Demand Anodyne CCR5 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(C2CCCC2)C1 ZINC000880966357 DH On-Demand Anodyne RBP4 92 52 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCCCC2)C1 ZINC000880966364 EH On-Demand Anodyne EPHX2 20 47 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCCCC2)C1 ZINC000880966364 EH On-Demand Anodyne RBP4 48 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)N1CCc2ccccc2C1 ZINC000880966367 DD On-Demand Anodyne DPP8 16 44 O=C(Cn1cc([C@H](O)C2CC2)nn1)N1CCc2ccccc2C1 ZINC000880966368 DD On-Demand Anodyne DPP8 16 44 NC(=O)CC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966371 DD On-Demand Anodyne RBP4 75 45 Cn1ccnc1[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966373 FG On-Demand Anodyne RBP4 66 42 Cn1ccnc1[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966374 FG On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1ccccc1 ZINC000880966378 EJ On-Demand Anodyne CPT1A 67 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1ccccc1 ZINC000880966378 EJ On-Demand Anodyne RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1ccccc1 ZINC000880966378 EJ On-Demand Anodyne SFRP1 79 37 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1ccccc1 ZINC000880966378 EJ On-Demand Anodyne WNT3 68 37 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1ccccc1 ZINC000880966379 EJ On-Demand Anodyne CPT1A 67 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1ccccc1 ZINC000880966379 EJ On-Demand Anodyne RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1ccccc1 ZINC000880966379 EJ On-Demand Anodyne SFRP1 79 37 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1ccccc1 ZINC000880966379 EJ On-Demand Anodyne WNT3 68 37 Cc1cnc(Cl)c(C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880966380 EG On-Demand Anodyne PLA2G2A 48 32 Cc1cnc(Cl)c(C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)c1 ZINC000880966380 EG On-Demand Anodyne FAAH 20 42 O=C(NCCF)Nc1cnccc1C(F)(F)F ZINC000880966381 CE On-Demand Anodyne TRPV1 22 51 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]2(CCOC2)O1 ZINC000880966388 EF On-Demand Anodyne RBP4 53 38 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]2(CCOC2)O1 ZINC000880966389 EF On-Demand Anodyne RBP4 53 38 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]2(CCOC2)O1 ZINC000880966390 EF On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2nnc3n2CCC3)C1 ZINC000880966451 GG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2nnc3n2CCC3)C1 ZINC000880966452 GG On-Demand Anodyne RBP4 59 42 CCC(CO)(CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966454 DD On-Demand Anodyne TRPV1 17 43 C[C@H]1CC[C@@H](C(F)(F)F)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966456 FI On-Demand Anodyne RBP4 40 38 C[C@H]1CC[C@H](C(F)(F)F)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966457 FI On-Demand Anodyne RBP4 40 38 C[C@@H]1CC[C@@H](C(F)(F)F)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966458 FI On-Demand Anodyne RBP4 40 38 C[C@@H]1CC[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1 ZINC000880966461 EI On-Demand Anodyne RBP4 55 39 C[C@H]1CC[C@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1 ZINC000880966463 EI On-Demand Anodyne RBP4 55 39 C[C@H]1CC[C@@]2(CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)C1 ZINC000880966464 EI On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](O)C1 ZINC000880966465 CD On-Demand Anodyne RBP4 90 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](O)C1 ZINC000880966466 CD On-Demand Anodyne RBP4 90 48 COC(=O)C1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966467 ED On-Demand Anodyne TRPV1 15 41 COC(=O)C1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966467 ED On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966476 GH On-Demand Anodyne TRPV1 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966476 GH On-Demand Anodyne FAAH 18 58 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966476 GH On-Demand Anodyne EPHX2 24 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966476 GH On-Demand Anodyne RBP4 54 37 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966477 GH On-Demand Anodyne TRPV1 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966477 GH On-Demand Anodyne FAAH 18 58 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966477 GH On-Demand Anodyne EPHX2 24 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(Cc2cccc(Cl)c2)C1 ZINC000880966477 GH On-Demand Anodyne RBP4 54 37 O=C(NC[C@H](O)CCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880966478 FG On-Demand Anodyne TRPV1 23 50 O=C(NC[C@@H](O)CCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880966479 FG On-Demand Anodyne TRPV1 23 50 Cc1noc(C2(C)CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880966485 FG On-Demand Anodyne RBP4 40 36 N#CCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966490 DG On-Demand Mild RBP4 67 41 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880966492 DF On-Demand Anodyne IMDH_CRYPV 39 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]2(CCOC2)O1 ZINC000880966495 EF On-Demand Anodyne RBP4 53 38 O=C(Cn1cc(CCCN2CCOCC2)nn1)N1CCc2ccccc2C1 ZINC000880966496 FD On-Demand Anodyne HTR7 17 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880966497 FG On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880966498 FG On-Demand Anodyne RBP4 48 38 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CC(F)(F)F ZINC000880966499 FG On-Demand Anodyne RBP4 59 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CC(F)(F)F ZINC000880966500 FG On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880966503 GI On-Demand Bother MMP8 30 43 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880966503 GI On-Demand Bother MMP9 15 43 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccc([N+](=O)[O-])cc1)C1CC1 ZINC000880966503 GI On-Demand Bother MMP1 22 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1c2ccccc2C[C@H]1O ZINC000880966505 EF On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1c2ccccc2C[C@H]1O ZINC000880966505 EF On-Demand Anodyne RBP4 49 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880966506 EF On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1c2ccccc2C[C@@H]1O ZINC000880966506 EF On-Demand Anodyne RBP4 49 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880966507 EF On-Demand Anodyne TRPV1 26 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1c2ccccc2C[C@H]1O ZINC000880966507 EF On-Demand Anodyne RBP4 49 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC12CCCC2 ZINC000880966508 CH On-Demand Anodyne TRPV1 16 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC12CCCC2 ZINC000880966509 CH On-Demand Anodyne TRPV1 16 40 CS(=O)(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966511 ED On-Demand Anodyne TRPV1 23 47 O=C(NCCCCO)Nc1cnccc1C(F)(F)F ZINC000880966515 CD On-Demand Anodyne TRPV1 19 48 COCC(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966517 CC On-Demand Reactive TRPV1 20 42 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCC2)C1 ZINC000880966524 DF On-Demand Anodyne EPHX2 22 48 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCC2)C1 ZINC000880966524 DF On-Demand Anodyne RBP4 54 39 NC(=O)C1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966527 CD On-Demand Anodyne TRPV1 17 45 O=C(NCc1cccnc1OCC(F)F)Nc1cnccc1C(F)(F)F ZINC000880966528 GG On-Demand Anodyne TRPV1 28 52 O=C(NCc1cccnc1OCC(F)F)Nc1cnccc1C(F)(F)F ZINC000880966528 GG On-Demand Anodyne SCN10A 18 42 N#Cc1cccc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)c1 ZINC000880966531 GH On-Demand Mild RBP4 55 39 N#Cc1cccc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)c1 ZINC000880966532 GH On-Demand Mild RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880966538 GG On-Demand Anodyne EPHX2 42 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880966538 GG On-Demand Anodyne SFRP1 70 36 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC[C@@H](C(=O)N2CCCCC2)C1 ZINC000880966538 GG On-Demand Anodyne WNT3 63 36 COCCO[C@H]1C[C@@H](CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966539 GD On-Demand Anodyne RBP4 56 41 COCCO[C@@H]1C[C@H](CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966540 GD On-Demand Anodyne RBP4 56 41 COCCO[C@H]1C[C@H](CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966541 GD On-Demand Anodyne RBP4 56 41 COCCO[C@@H]1C[C@@H](CO)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966542 GD On-Demand Anodyne RBP4 56 41 O=C(CC1CCCC1)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966547 EF On-Demand Reactive TRPV1 19 41 CC(CO)(CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966549 CC On-Demand Anodyne TRPV1 20 47 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CCOCC2)C1 ZINC000880966552 EH On-Demand Anodyne RBP4 48 38 C[C@@H]1C[C@@H](c2cccnc2)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966568 FI On-Demand Anodyne RBP4 48 40 C[C@@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966571 FI On-Demand Anodyne RBP4 48 40 COc1cnccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966572 GF On-Demand Anodyne PDGFRB 44 44 COc1cnccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966572 GF On-Demand Anodyne TRPV1 15 51 COc1cnccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966572 GF On-Demand Anodyne RBP4 60 53 C[C@H]1C[C@H](c2cccnc2)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966575 FI On-Demand Anodyne RBP4 48 40 O=C(NC[C@H]1CCC(F)(F)C1)Nc1cnccc1C(F)(F)F ZINC000880966576 DH On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880966579 GI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880966579 GI On-Demand Anodyne TRPM8 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880966581 GI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880966581 GI On-Demand Anodyne TRPM8 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880966583 GI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880966583 GI On-Demand Anodyne TRPM8 22 40 O=C([C@H]1CCc2nncn2CC1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966584 FD On-Demand Anodyne SIGMAR1 28 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880966585 GI On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880966585 GI On-Demand Anodyne TRPM8 22 40 O=C([C@@H]1CCc2nncn2CC1)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880966586 FD On-Demand Anodyne SIGMAR1 28 50 CN1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966587 DE On-Demand Anodyne RBP4 60 42 CC(=O)N1CCC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966589 EE On-Demand Anodyne TRPV1 16 40 CC(=O)N1CCC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966591 EE On-Demand Anodyne TRPV1 16 40 CSC1(CNC(=O)Nc2cnccc2C(F)(F)F)CCC1 ZINC000880966595 DH On-Demand Anodyne TRPV1 20 47 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NCC(F)F ZINC000880966601 ED On-Demand Anodyne TRPV1 15 46 CCn1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1=O ZINC000880966604 EF On-Demand Anodyne TRPV1 23 53 CCn1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1=O ZINC000880966604 EF On-Demand Anodyne P2RX7 47 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)Cc1ccccc1 ZINC000880966613 FG On-Demand Anodyne ANPEP 54 34 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)Cc1ccccc1 ZINC000880966613 FG On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)Cc1ccccc1 ZINC000880966613 FG On-Demand Anodyne GPR142 51 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)Cc1ccccc1 ZINC000880966614 FG On-Demand Anodyne ANPEP 54 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)Cc1ccccc1 ZINC000880966614 FG On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)Cc1ccccc1 ZINC000880966614 FG On-Demand Anodyne GPR142 51 34 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]2(CCCOC2)O1 ZINC000880966615 FF On-Demand Anodyne RBP4 40 37 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]2(CCCOC2)O1 ZINC000880966616 FF On-Demand Anodyne RBP4 40 37 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@]2(CCCOC2)O1 ZINC000880966617 FF On-Demand Anodyne RBP4 40 37 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@]2(CCCOC2)O1 ZINC000880966618 FF On-Demand Anodyne RBP4 40 37 COC(=O)[C@@]12CCOC[C@@H]1CN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880966623 FE On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N(CC1CCC1)CC1CC1 ZINC000880966629 EI On-Demand Anodyne TRPV1 15 40 N#CC1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966636 EH On-Demand Mild TRPV1 16 44 C[C@H]1C[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966641 CG On-Demand Anodyne TRPV1 17 43 C[C@H]1C[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966641 CG On-Demand Anodyne RBP4 70 44 CS(=O)(=O)C1CCC(C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CC1 ZINC000880966646 GD On-Demand Anodyne SIGMAR1 31 44 CN(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966648 EG On-Demand Anodyne RBP4 69 42 CN(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966648 EG On-Demand Anodyne SFRP1 83 35 CN(C)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966648 EG On-Demand Anodyne WNT3 75 35 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne GHRHR 44 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne P2RY12 160 38 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne PGC 52 33 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne PAPA1_CARPA 41 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne CTSK 29 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne CTSL 20 43 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne CCR1 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne TACR3 15 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne AMY2 43 29 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne REN 60 39 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966654 EF On-Demand Anodyne FPR1 51 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne GHRHR 44 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne P2RY12 160 38 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne PGC 52 33 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne PAPA1_CARPA 41 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne CTSK 29 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne CTSL 20 43 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne CCR1 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne TACR3 15 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne AMY2 43 29 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne REN 60 39 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC(c2ccccc2)C1 ZINC000880966655 EF On-Demand Anodyne FPR1 51 39 O=C(Cn1cc([C@H]2CCOC2)nn1)N1CCc2ccccc2C1 ZINC000880966666 DD On-Demand Anodyne CPT2 25 40 O=C(Cn1cc([C@@H]2CCOC2)nn1)N1CCc2ccccc2C1 ZINC000880966667 DD On-Demand Anodyne CPT2 25 40 CC(C)(C)CNC(=O)C(C)(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966674 FG On-Demand Anodyne TRPV1 17 43 C[C@H]1[C@H](C(F)(F)F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966676 EH On-Demand Anodyne RBP4 57 41 C[C@@H]1[C@@H](C(F)(F)F)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966677 EH On-Demand Anodyne RBP4 57 41 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)N1CCc2ccccc2C1 ZINC000880966682 GF On-Demand Anodyne DPP8 17 42 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)N1CCc2ccccc2C1 ZINC000880966683 GF On-Demand Anodyne DPP8 17 42 CC(C)(C)OC(=O)NCc1cn(CC(=O)N2CCCc3ccccc32)nn1 ZINC000880966688 FE On-Demand Anodyne AVPR2 35 42 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1Cl ZINC000880966692 FH On-Demand Anodyne TRPV1 25 49 O=C(NOCCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880966693 DG On-Demand Anodyne TRPV1 15 42 C[C@@H]1CN(CC(C)(C)O)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966696 FE On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cc(C3CC3)[nH]n2)CC1 ZINC000880966699 GG On-Demand Anodyne RBP4 57 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCOC2)C1 ZINC000880966709 EE On-Demand Anodyne EPHX2 21 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCOC2)C1 ZINC000880966709 EE On-Demand Anodyne RBP4 47 38 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCOC2)C1 ZINC000880966710 EE On-Demand Anodyne EPHX2 21 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCOC2)C1 ZINC000880966710 EE On-Demand Anodyne RBP4 47 38 CCOC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880966713 DG On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccn2)CC1 ZINC000880966716 FF On-Demand Anodyne TRPV1 21 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccn2)CC1 ZINC000880966716 FF On-Demand Anodyne ABL2 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccn2)CC1 ZINC000880966716 FF On-Demand Anodyne FAAH 26 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccccn2)CC1 ZINC000880966716 FF On-Demand Anodyne RBP4 72 43 CCOC(=O)C1CCN(C(=O)Cn2cc(C[C@@H](O)c3ccccc3)nn2)CC1 ZINC000880966719 GD On-Demand Anodyne FDFT1 22 46 CCOC(=O)C1CCN(C(=O)Cn2cc(C[C@H](O)c3ccccc3)nn2)CC1 ZINC000880966720 GD On-Demand Anodyne FDFT1 22 46 O=C(Nc1cnccc1C(F)(F)F)N1CCOCC2(CCCC2)C1 ZINC000880966727 EH On-Demand Anodyne RBP4 47 38 CC[C@@](C)(O)CN(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880966730 GI On-Demand Anodyne TRPV1 15 41 CC(C)c1cc(NC(=O)Nc2cnccc2C(F)(F)F)n[nH]1 ZINC000880966732 DH On-Demand Anodyne TRPV1 17 41 Cc1cc(C)c2c(c1)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880966733 EI On-Demand Anodyne RBP4 55 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880966734 EI On-Demand Anodyne TRPV1 23 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880966734 EI On-Demand Anodyne RBP4 83 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880966735 EI On-Demand Anodyne TRPV1 23 42 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880966735 EI On-Demand Anodyne RBP4 83 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880966736 EI On-Demand Anodyne TRPV1 23 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880966736 EI On-Demand Anodyne RBP4 83 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880966737 EI On-Demand Anodyne TRPV1 23 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880966737 EI On-Demand Anodyne RBP4 83 43 CN(CCNC(=O)Nc1cnccc1C(F)(F)F)C1CCCCC1 ZINC000880966738 EG On-Demand Anodyne TRPV1 22 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cn2cncn2)CC1 ZINC000880966739 FF On-Demand Anodyne RBP4 60 39 CCOC(=O)C1CCN(C(=O)Cn2cc(-c3ccc(Cl)cc3F)nn2)CC1 ZINC000880966742 GF On-Demand Anodyne IL2RA 53 35 CCOC(=O)C1CCN(C(=O)Cn2cc(-c3ccc(Cl)cc3F)nn2)CC1 ZINC000880966742 GF On-Demand Anodyne FDFT1 28 46 CN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966743 DE On-Demand Anodyne TRPV1 19 42 CN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966743 DE On-Demand Anodyne CCR3 25 42 CN1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966744 DE On-Demand Anodyne TRPV1 19 42 CN1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966744 DE On-Demand Anodyne CCR3 25 42 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N1CCCc2ccccc21 ZINC000880966748 FF On-Demand Anodyne AVPR2 26 42 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N1CCCc2ccccc21 ZINC000880966749 FF On-Demand Anodyne AVPR2 26 42 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966754 DF On-Demand Anodyne IMDH_CRYPV 18 40 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966755 DF On-Demand Anodyne IMDH_CRYPV 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCCn2ccnc2)CC1 ZINC000880966761 GI On-Demand Anodyne TBXAS1 31 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCCn2ccnc2)CC1 ZINC000880966761 GI On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Cc2ccncc2)C1 ZINC000880966764 FH On-Demand Anodyne CCR3 47 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Cc2ccncc2)C1 ZINC000880966764 FH On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880966765 FH On-Demand Anodyne CCR3 47 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Cc2ccncc2)C1 ZINC000880966765 FH On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)[C@H](O)C1 ZINC000880966766 CC On-Demand Anodyne TRPV1 19 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)[C@H](O)C1 ZINC000880966766 CC On-Demand Anodyne RBP4 90 51 CN1CCC(C)(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966767 EF On-Demand Anodyne TRPV1 18 45 CN1CC=C(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966768 DE On-Demand Anodyne TRPV1 18 45 O=C(Cn1cc(C(=O)C2CCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966770 EG On-Demand Anodyne IMDH_CRYPV 18 40 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccncc1 ZINC000880966771 EH On-Demand Anodyne TRPV1 26 49 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966777 FD On-Demand Anodyne IMDH_CRYPV 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cccnc2)CC1 ZINC000880966778 FH On-Demand Anodyne TRPV1 19 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cccnc2)CC1 ZINC000880966778 FH On-Demand Anodyne SLC9A1 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cccnc2)CC1 ZINC000880966778 FH On-Demand Anodyne CCR2 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cccnc2)CC1 ZINC000880966778 FH On-Demand Anodyne EPHX2 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cccnc2)CC1 ZINC000880966778 FH On-Demand Anodyne RBP4 92 48 O=C(NC[C@H](CO)Cc1ccc(F)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880966779 GG On-Demand Anodyne TRPV1 16 44 CCOC(=O)CC[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966781 EF On-Demand Anodyne TRPV1 15 45 CCOC(=O)CC[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880966782 EF On-Demand Anodyne TRPV1 15 45 O=C(NC[C@@H](CO)Cc1ccc(F)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880966785 GG On-Demand Anodyne TRPV1 16 44 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880966786 EH On-Demand Anodyne TRPV1 18 49 CNC(C)(C)c1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880966788 DF On-Demand Anodyne IMDH_CRYPV 37 41 C[C@@](CO)(NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880966790 EG On-Demand Anodyne TRPV1 24 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne TRPV1 17 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne CCR3 21 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne EPHX2 21 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne RBP4 95 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne SFRP1 80 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COc2ccccc2)C1 ZINC000880966805 FI On-Demand Anodyne WNT3 63 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne TRPV1 17 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne CCR3 21 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne EPHX2 21 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne RBP4 95 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne SFRP1 80 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COc2ccccc2)C1 ZINC000880966806 FI On-Demand Anodyne WNT3 63 33 O=C(NCCCO)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966807 FD On-Demand Anodyne RBP4 58 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne GRIN2B 49 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne TRPV1 27 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne CCR3 36 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne CHRNA7 54 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne C3AR1 43 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne RBP4 75 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne SCD 16 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne ACHP_LYMST 27 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cc2cccnc2)CC1 ZINC000880966809 FH On-Demand Anodyne NAMPT 44 38 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC12CCC2 ZINC000880966810 EI On-Demand Anodyne RBP4 65 40 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC12CCC2 ZINC000880966812 EI On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N1CC=CCC1 ZINC000880966814 CF On-Demand Anodyne RBP4 61 45 O=C(Cn1cc(CN2CCNCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966817 FD On-Demand Anodyne IMDH_CRYPV 20 43 NC1CCN(CCc2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)CC1 ZINC000880966823 GE On-Demand Anodyne DRD4 16 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne MME 49 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne ANPEP 70 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne TRPV1 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne AKT1 41 32 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne PIN1 15 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccccc1 ZINC000880966824 EF On-Demand Anodyne GPR142 57 35 CCC[C@@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966825 DI On-Demand Anodyne RBP4 47 38 CCC[C@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966826 DI On-Demand Anodyne RBP4 47 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne MME 49 36 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne ANPEP 70 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne TRPV1 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne AKT1 41 32 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne PIN1 15 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccccc1 ZINC000880966828 EF On-Demand Anodyne GPR142 57 35 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1(C)C ZINC000880966834 DI On-Demand Anodyne RBP4 68 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1(C)C ZINC000880966835 DI On-Demand Anodyne RBP4 68 41 NCCCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880966836 DE On-Demand Anodyne IMDH_CRYPV 24 42 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966844 FG On-Demand Anodyne CHRNA7 20 40 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966844 FG On-Demand Anodyne MCHR1 21 43 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966844 FG On-Demand Anodyne IMDH_CRYPV 16 41 COC[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)OC ZINC000880966868 DD On-Demand Anodyne TRPV1 15 44 O=C(CO)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966870 EC On-Demand Anodyne TRPV1 16 47 O=C(CO)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966870 EC On-Demand Anodyne RBP4 60 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCOC[C@@H]2C1 ZINC000880966874 ED On-Demand Anodyne RBP4 58 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCOC[C@H]2C1 ZINC000880966875 ED On-Demand Anodyne RBP4 58 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CCCC2)C1 ZINC000880966876 EI On-Demand Anodyne EPHX2 32 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CCCC2)C1 ZINC000880966876 EI On-Demand Anodyne RBP4 57 41 O=C(NOC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880966877 CG On-Demand Anodyne TRPV1 20 42 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880966878 DE On-Demand Anodyne IMDH_CRYPV 25 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(CO)C1 ZINC000880966880 CD On-Demand Anodyne RBP4 79 48 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccc(F)c(F)c2)C1 ZINC000880966883 FI On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCn2ncnc2C1 ZINC000880966884 DD On-Demand Anodyne RBP4 55 39 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966885 FF On-Demand Anodyne TRPV1 22 47 CC(C)(C)NC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880966885 FF On-Demand Anodyne RBP4 62 44 Cn1nccc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880966895 DE On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880966901 FH On-Demand Anodyne NPY5R 35 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000880966901 FH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880966904 FH On-Demand Anodyne NPY5R 35 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C1)OCc1ccccc12 ZINC000880966904 FH On-Demand Anodyne RBP4 55 39 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)CC)nn2)CC1 ZINC000880966914 DC On-Demand Anodyne FDFT1 15 40 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)CC)nn2)CC1 ZINC000880966917 DC On-Demand Anodyne FDFT1 15 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](CO)O1 ZINC000880966919 DD On-Demand Anodyne RBP4 62 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](CO)O1 ZINC000880966921 DD On-Demand Anodyne RBP4 62 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](CO)O1 ZINC000880966923 DD On-Demand Anodyne RBP4 62 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](CO)O1 ZINC000880966925 DD On-Demand Anodyne RBP4 62 43 C[C@]1(CO)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966932 DE On-Demand Anodyne RBP4 41 38 C[C@@]1(CO)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880966933 DE On-Demand Anodyne RBP4 41 38 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1cccc(Cl)c1 ZINC000880966938 FH On-Demand Anodyne TRPV1 29 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Nc2ccc3nccn3n2)C1 ZINC000880966940 GF On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Nc2ccc3nccn3n2)C1 ZINC000880966942 GF On-Demand Anodyne RBP4 68 43 CCc1nnc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)o1 ZINC000880966948 FF On-Demand Anodyne RBP4 53 38 CCc1nnc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)o1 ZINC000880966950 FF On-Demand Anodyne RBP4 53 38 COCCO[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966952 EE On-Demand Anodyne RBP4 67 42 COCCO[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966952 EE On-Demand Anodyne LIPG 39 43 COCCO[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966952 EE On-Demand Anodyne SCD 17 40 COCCO[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966954 EE On-Demand Anodyne RBP4 67 42 COCCO[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966954 EE On-Demand Anodyne LIPG 39 43 COCCO[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880966954 EE On-Demand Anodyne SCD 17 40 C[C@@](O)(CCNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880966973 FH On-Demand Anodyne TRPV1 25 48 CCOC(=O)C1CCN(C(=O)Cn2cc(C(C)(C)O)nn2)CC1 ZINC000880966993 DC On-Demand Anodyne FDFT1 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(C(F)F)CC1 ZINC000880966999 EF On-Demand Anodyne TRPV1 16 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(C(F)F)CC1 ZINC000880966999 EF On-Demand Anodyne RBP4 58 42 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCCC1 ZINC000880967001 EG On-Demand Anodyne TRPV1 20 43 O=C(NCC1(O)CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880967002 DD On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncc(F)cn2)CC1 ZINC000880967004 FE On-Demand Anodyne TRPV1 17 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncc(F)cn2)CC1 ZINC000880967004 FE On-Demand Anodyne RBP4 57 41 O=C(NOCCO)Nc1cnccc1C(F)(F)F ZINC000880967006 CD On-Demand Anodyne TRPV1 18 43 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)N2CCCc3ccccc32)nn1 ZINC000880967017 GF On-Demand Anodyne AVPR2 30 41 C[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967022 CG On-Demand Anodyne TRPV1 29 40 C[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967022 CG On-Demand Anodyne EPHX2 39 43 C[C@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967023 CG On-Demand Anodyne TRPV1 29 40 C[C@H]1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967023 CG On-Demand Anodyne EPHX2 39 43 C[C@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967024 CG On-Demand Anodyne TRPV1 29 40 C[C@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967024 CG On-Demand Anodyne EPHX2 39 43 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967030 FE On-Demand Anodyne TRPV1 18 40 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967030 FE On-Demand Anodyne EPHX2 47 45 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967030 FE On-Demand Anodyne RBP4 71 44 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967030 FE On-Demand Anodyne SFRP1 60 35 O=C(NC1CC1)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967030 FE On-Demand Anodyne WNT3 45 33 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967031 FE On-Demand Anodyne TRPV1 18 40 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967031 FE On-Demand Anodyne EPHX2 47 45 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967031 FE On-Demand Anodyne RBP4 71 44 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967031 FE On-Demand Anodyne SFRP1 60 35 O=C(NC1CC1)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967031 FE On-Demand Anodyne WNT3 45 33 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne TRPV1 23 41 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne CCR2 25 44 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne EPHX2 23 40 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne RBP4 87 50 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne MCHR1 23 41 COc1cccc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880967032 GJ On-Demand Anodyne TAAR1 26 40 CCC1(CC)CN(C(=O)Nc2cnccc2C(F)(F)F)CCS1 ZINC000880967038 EI On-Demand Anodyne RBP4 47 38 CCOC(=O)C1CCN(C(=O)Cn2cc(-c3cccnc3Cl)nn2)CC1 ZINC000880967045 GD On-Demand Anodyne IL2RA 40 33 CO[C@H]1CCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967047 DG On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCn2ccnc2C1 ZINC000880967048 EE On-Demand Anodyne EPHX2 32 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCn2ccnc2C1 ZINC000880967049 EE On-Demand Anodyne EPHX2 32 43 CCO[C@H]1C[C@H](O)C12CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967052 FF On-Demand Anodyne RBP4 55 39 CCO[C@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967053 FF On-Demand Anodyne RBP4 55 39 C[C@@]1(C#N)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967054 DG On-Demand Mild RBP4 50 38 CCO[C@@H]1C[C@H](O)C12CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967055 FF On-Demand Anodyne RBP4 55 39 CCO[C@@H]1C[C@@H](O)C12CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967056 FF On-Demand Anodyne RBP4 55 39 CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC12CCCCC2 ZINC000880967058 GG On-Demand Anodyne RBP4 42 37 COC(=O)CCCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967059 EG On-Demand Anodyne TRPV1 18 46 CC(C)(C)C(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967060 DE On-Demand Reactive TRPV1 19 43 O=C(Cn1cc([C@H]2CCCNC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967061 EF On-Demand Anodyne IMDH_CRYPV 15 41 O=C(Cn1cc([C@@H]2CCCNC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967062 EF On-Demand Anodyne IMDH_CRYPV 15 41 CCC[C@@H]1C(=O)NCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967065 EE On-Demand Anodyne RBP4 45 37 CCC[C@H]1C(=O)NCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967066 EE On-Demand Anodyne RBP4 45 37 O=C(NCC1(CO)CCC1)Nc1cnccc1C(F)(F)F ZINC000880967077 DE On-Demand Anodyne TRPV1 16 47 CC(=O)N1CCN(Cc2cn(CC(=O)N3CCCc4ccccc43)nn2)CC1 ZINC000880967078 GC On-Demand Anodyne DRD4 20 47 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967081 FD On-Demand Anodyne RBP4 66 41 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967081 FD On-Demand Anodyne SFRP1 51 35 CCNS(=O)(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967081 FD On-Demand Anodyne WNT3 43 34 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967082 FD On-Demand Anodyne RBP4 66 41 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967082 FD On-Demand Anodyne SFRP1 51 35 CCNS(=O)(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967082 FD On-Demand Anodyne WNT3 43 34 CC(C)(C)[C@@H](O)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967084 FG On-Demand Anodyne IMDH_CRYPV 23 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1N1CCN(C)CC1 ZINC000880967099 GF On-Demand Anodyne RBP4 65 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1N1CCN(C)CC1 ZINC000880967100 GF On-Demand Anodyne RBP4 65 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1N1CCN(C)CC1 ZINC000880967101 GF On-Demand Anodyne RBP4 65 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1N1CCN(C)CC1 ZINC000880967102 GF On-Demand Anodyne RBP4 65 41 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)c(F)c1 ZINC000880967104 GH On-Demand Anodyne TRPV1 22 51 COC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)c(F)c1 ZINC000880967105 GH On-Demand Anodyne TRPV1 22 51 CC(C)[C@H](O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967108 EG On-Demand Anodyne TRPV1 20 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)CC[C@@H]2C1 ZINC000880967109 ED On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)CC[C@@H]2C1 ZINC000880967109 ED On-Demand Anodyne SMO 17 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)CC[C@H]2C1 ZINC000880967110 ED On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)CC[C@H]2C1 ZINC000880967110 ED On-Demand Anodyne SMO 17 42 O=C(Cn1cc(C[C@@H](O)C2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967120 EE On-Demand Anodyne IMDH_CRYPV 15 41 O=C(Cn1cc(C[C@H](O)C2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967121 EE On-Demand Anodyne IMDH_CRYPV 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2nncn2C2CC2)C1 ZINC000880967123 GG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2nncn2C2CC2)C1 ZINC000880967124 GG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CCCC2)CC1 ZINC000880967132 FH On-Demand Anodyne EPHX2 48 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CCCC2)CC1 ZINC000880967132 FH On-Demand Anodyne CXCR3 20 52 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CCCC2)CC1 ZINC000880967132 FH On-Demand Anodyne SFRP1 55 35 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CCCC2)CC1 ZINC000880967132 FH On-Demand Anodyne WNT3 48 35 O=C(Cn1cc(CN2CCC[C@H]2CO)nn1)Nc1ccc2ccccc2c1 ZINC000880967133 FE On-Demand Anodyne SPHK1 28 42 O=C(Cn1cc(CN2CCC[C@@H]2CO)nn1)Nc1ccc2ccccc2c1 ZINC000880967134 FE On-Demand Anodyne SPHK1 28 42 N#CCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967135 CF On-Demand Mild TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@@H]2CCOC2)CC1 ZINC000880967150 FG On-Demand Anodyne RBP4 45 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@H]2CCOC2)CC1 ZINC000880967151 FG On-Demand Anodyne RBP4 45 37 O=C(Nc1cnccc1C(F)(F)F)N1CCOCC2(CCOCC2)C1 ZINC000880967153 FF On-Demand Anodyne RBP4 47 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1nc2ccccc2o1 ZINC000880967166 GK On-Demand Anodyne CPT1A 51 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1nc2ccccc2o1 ZINC000880967166 GK On-Demand Anodyne RBP4 40 36 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1nc2ccccc2o1 ZINC000880967167 GK On-Demand Anodyne CPT1A 51 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1nc2ccccc2o1 ZINC000880967167 GK On-Demand Anodyne RBP4 40 36 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](F)C[C@@H]1CO ZINC000880967168 DE On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](F)C[C@@H]1CO ZINC000880967169 DE On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](F)C[C@H]1CO ZINC000880967170 DE On-Demand Anodyne RBP4 47 40 CC(C)(C)OC(=O)N1CC(CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967176 FG On-Demand Anodyne TRPV1 15 40 CC(C)(C)OC(=O)N1CC(CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967176 FG On-Demand Anodyne GPR119 28 40 O=C(CC(F)(F)F)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967202 EE On-Demand Reactive TRPV1 22 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC12CCCCC2 ZINC000880967205 DH On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC12CCCCC2 ZINC000880967206 DH On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)CC(F)(F)C1 ZINC000880967207 EE On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(n2ccnn2)CC1 ZINC000880967209 EF On-Demand Anodyne RBP4 66 41 O=C(NCCCCCCO)Nc1cnccc1C(F)(F)F ZINC000880967210 DF On-Demand Anodyne TRPV1 19 47 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)CC(F)(F)C1 ZINC000880967211 EE On-Demand Anodyne RBP4 68 43 CCONC(=O)Nc1cnccc1C(F)(F)F ZINC000880967217 BE On-Demand Anodyne TRPV1 22 44 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967221 EF On-Demand Anodyne MCHR1 25 42 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967221 EF On-Demand Anodyne IMDH_CRYPV 25 42 C[C@H](CCO)N(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880967222 FH On-Demand Anodyne TRPV1 15 40 C[C@@H](CCO)N(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880967223 FH On-Demand Anodyne TRPV1 15 40 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880967228 GG On-Demand Anodyne TRPV1 18 42 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880967228 GG On-Demand Anodyne CCR3 34 44 O=C(NCC1CCN(CC(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880967228 GG On-Demand Anodyne CACNA1I 60 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOc2c(F)cccc21 ZINC000880967232 FH On-Demand Anodyne TRPV1 42 60 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOc2c(F)cccc21 ZINC000880967232 FH On-Demand Anodyne RBP4 45 39 Cc1ccccc1[C@@H]1C(=O)NCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967234 GG On-Demand Anodyne RBP4 73 41 Cc1ccccc1[C@@H]1C(=O)NCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967234 GG On-Demand Anodyne TRPM8 41 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1O ZINC000880967235 CD On-Demand Anodyne RBP4 78 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1O ZINC000880967237 CD On-Demand Anodyne RBP4 78 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1O ZINC000880967238 CD On-Demand Anodyne RBP4 78 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1O ZINC000880967239 CD On-Demand Anodyne RBP4 78 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2n[nH]c(C3CC3)n2)C1 ZINC000880967244 GH On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2n[nH]c(C3CC3)n2)C1 ZINC000880967245 GH On-Demand Anodyne RBP4 58 41 CC(C)[C@H]1CN(C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967256 EF On-Demand Anodyne RBP4 53 39 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967261 FG On-Demand Anodyne IMDH_CRYPV 21 40 Cn1cnc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880967262 DD On-Demand Anodyne TRPV1 19 48 COC(=O)[C@@H]1CCCN1Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967264 GE On-Demand Anodyne MCHR1 16 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCCC2)C1 ZINC000880967268 FG On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCCC2)C1 ZINC000880967268 FG On-Demand Anodyne SFRP1 82 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCCC2)C1 ZINC000880967268 FG On-Demand Anodyne WNT3 70 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880967272 FG On-Demand Anodyne RBP4 69 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880967272 FG On-Demand Anodyne SFRP1 82 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCCC2)C1 ZINC000880967272 FG On-Demand Anodyne WNT3 70 34 CC(C)(C)OC(=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967273 EF On-Demand Anodyne TRPV1 23 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967274 GG On-Demand Anodyne ACE 24 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967274 GG On-Demand Anodyne MME 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967274 GG On-Demand Anodyne TRPV1 28 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967274 GG On-Demand Anodyne RBP4 57 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967275 GG On-Demand Anodyne ACE 24 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967275 GG On-Demand Anodyne MME 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967275 GG On-Demand Anodyne TRPV1 28 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(Cc2ccccc2)C1=O ZINC000880967275 GG On-Demand Anodyne RBP4 57 39 O=C(Nc1cnccc1C(F)(F)F)N1CCOCC2(CCC2)C1 ZINC000880967277 EG On-Demand Anodyne RBP4 47 38 CCO[C@H]1COCC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967279 EE On-Demand Anodyne CCR2 25 40 CCO[C@H]1COCC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967280 EE On-Demand Anodyne CCR2 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2ncccc2C1 ZINC000880967283 EF On-Demand Anodyne TRPV1 16 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2ncccc2C1 ZINC000880967283 EF On-Demand Anodyne RBP4 55 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2)CC1 ZINC000880967286 FH On-Demand Anodyne OPRL1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2)CC1 ZINC000880967286 FH On-Demand Anodyne TRPV1 18 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2)CC1 ZINC000880967286 FH On-Demand Anodyne NPY5R 25 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(c2ccccc2)CC1 ZINC000880967286 FH On-Demand Anodyne RBP4 79 46 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](CCc2ccccc2)C1 ZINC000880967287 GH On-Demand Anodyne RBP4 89 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](CCc2ccccc2)C1 ZINC000880967288 GH On-Demand Anodyne RBP4 89 45 O=C(NC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1)C1CCC1 ZINC000880967296 EE On-Demand Anodyne RBP4 60 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](n2cncn2)C1 ZINC000880967297 EE On-Demand Anodyne RBP4 67 43 CN(C)C(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967300 FF On-Demand Anodyne RBP4 66 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](n2cncn2)C1 ZINC000880967301 EE On-Demand Anodyne RBP4 67 43 CC(C)(CS(C)(=O)=O)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967306 EE On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ncsc2C1 ZINC000880967307 EG On-Demand Anodyne RBP4 53 39 C#C[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967308 CE On-Demand Mild TRPV1 19 49 C#C[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967309 CE On-Demand Mild TRPV1 19 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880967314 GG On-Demand Anodyne TRPV1 24 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880967314 GG On-Demand Anodyne CCR3 49 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880967315 GG On-Demand Anodyne TRPV1 24 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccc(F)cc2)C1=O ZINC000880967315 GG On-Demand Anodyne CCR3 49 34 O=C(Nc1cnccc1C(F)(F)F)N1CCS(=O)(=O)c2ccccc2C1 ZINC000880967322 GF On-Demand Anodyne RBP4 58 42 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1ncc[nH]1 ZINC000880967325 FE On-Demand Anodyne RBP4 57 41 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1ncc[nH]1 ZINC000880967326 FE On-Demand Anodyne RBP4 57 41 C[C@@H](Cc1ccc(O)c(O)c1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967338 FG On-Demand Clean TRPV1 20 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967341 DE On-Demand Anodyne RBP4 80 45 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967341 DE On-Demand Anodyne SFRP1 55 34 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967341 DE On-Demand Anodyne WNT3 42 32 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967342 DE On-Demand Anodyne RBP4 80 45 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967342 DE On-Demand Anodyne SFRP1 55 34 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967342 DE On-Demand Anodyne WNT3 42 32 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967343 DE On-Demand Anodyne RBP4 80 45 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967343 DE On-Demand Anodyne SFRP1 55 34 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@@H]1O ZINC000880967343 DE On-Demand Anodyne WNT3 42 32 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967344 DE On-Demand Anodyne RBP4 80 45 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967344 DE On-Demand Anodyne SFRP1 55 34 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1O ZINC000880967344 DE On-Demand Anodyne WNT3 42 32 CN(C)c1noc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880967355 ED On-Demand Anodyne TRPV1 23 50 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCOCC2)C1 ZINC000880967356 FE On-Demand Anodyne RBP4 67 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCOCC2)C1 ZINC000880967357 FE On-Demand Anodyne RBP4 67 42 CCNC(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CCC1 ZINC000880967360 EF On-Demand Anodyne TRPV1 15 44 Cc1nc(CCNC(=O)Nc2cnccc2C(F)(F)F)n[nH]1 ZINC000880967362 DD On-Demand Anodyne TRPV1 19 47 CN1CN(C(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880967365 CD On-Demand Anodyne RBP4 54 40 COC1(C)CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967367 CE On-Demand Anodyne RBP4 55 40 O=C(NCCCc1cccs1)Nc1cnccc1C(F)(F)F ZINC000880967370 EH On-Demand Anodyne TRPV1 15 48 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967372 EF On-Demand Anodyne IMDH_CRYPV 19 41 CC[C@@H](C)C(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967373 DE On-Demand Reactive TRPV1 22 48 CC[C@@](C)(O)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967376 EF On-Demand Anodyne IMDH_CRYPV 43 44 CCC1(CO)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967379 EG On-Demand Anodyne RBP4 59 41 O=C(NCC1CCN(c2ccncc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880967384 GH On-Demand Anodyne TRPV1 19 43 O=C(Cn1cc(CN2CCSCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967387 FF On-Demand Anodyne IMDH_CRYPV 21 41 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880967404 FH On-Demand Anodyne TRPV1 28 40 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)[C@H]1c1ccccc1 ZINC000880967404 FH On-Demand Anodyne RBP4 61 39 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880967406 FH On-Demand Anodyne TRPV1 28 40 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)[C@@H]1c1ccccc1 ZINC000880967406 FH On-Demand Anodyne RBP4 61 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncccc2F)CC1 ZINC000880967407 FF On-Demand Anodyne TRPV1 43 55 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncccc2F)CC1 ZINC000880967407 FF On-Demand Anodyne RBP4 63 41 CC(C)(C)OC(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967409 DF On-Demand Reactive TRPV1 15 41 CN(C)CC1(CNC(=O)Nc2cnccc2C(F)(F)F)CCCC1 ZINC000880967414 EG On-Demand Anodyne TRPV1 17 46 C[C@@H]1C[C@H](O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967416 CE On-Demand Anodyne RBP4 61 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C ZINC000880967417 DH On-Demand Anodyne TRPV1 16 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C ZINC000880967417 DH On-Demand Anodyne RBP4 90 46 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C ZINC000880967417 DH On-Demand Anodyne SFRP1 91 37 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC[C@H]1C ZINC000880967417 DH On-Demand Anodyne WNT3 73 34 C[C@H]1C[C@H](O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967418 CE On-Demand Anodyne RBP4 61 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967419 DH On-Demand Anodyne TRPV1 16 43 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967419 DH On-Demand Anodyne RBP4 90 46 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967419 DH On-Demand Anodyne SFRP1 91 37 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967419 DH On-Demand Anodyne WNT3 73 34 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880967421 DH On-Demand Anodyne TRPV1 16 43 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880967421 DH On-Demand Anodyne RBP4 90 46 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880967421 DH On-Demand Anodyne SFRP1 91 37 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880967421 DH On-Demand Anodyne WNT3 73 34 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967422 DH On-Demand Anodyne TRPV1 16 43 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967422 DH On-Demand Anodyne RBP4 90 46 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967422 DH On-Demand Anodyne SFRP1 91 37 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880967422 DH On-Demand Anodyne WNT3 73 34 O=C(NCCc1ccc2c(c1)CCO2)Nc1cnccc1C(F)(F)F ZINC000880967425 FG On-Demand Anodyne RAF1 23 40 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(O)nnc2C1 ZINC000880967427 ED On-Demand Anodyne P2RX7 32 43 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(O)nnc2C1 ZINC000880967427 ED On-Demand Anodyne RBP4 54 40 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NCC1CC1 ZINC000880967432 DD On-Demand Anodyne TRPV1 24 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H]2CCCO2)CC1 ZINC000880967433 EH On-Demand Anodyne RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H]2CCCO2)CC1 ZINC000880967435 EH On-Demand Anodyne RBP4 72 43 Cc1nc2c(s1)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)CCC2 ZINC000880967436 FI On-Demand Anodyne TRPV1 26 41 N#C[C@]1(F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967437 DF On-Demand Mild RBP4 55 40 Cc1nc2c(s1)[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)CCC2 ZINC000880967438 FI On-Demand Anodyne TRPV1 26 41 N#C[C@@]1(F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967441 DF On-Demand Mild RBP4 55 40 CN1C(=O)NC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)C1=O ZINC000880967442 FD On-Demand Anodyne RBP4 50 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@@]2(CO)C1 ZINC000880967443 DD On-Demand Anodyne RBP4 65 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2C[C@]2(CO)C1 ZINC000880967444 DD On-Demand Anodyne RBP4 65 43 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@]2(CO)C1 ZINC000880967445 DD On-Demand Anodyne RBP4 65 43 CCC1(O)CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967446 EG On-Demand Anodyne TRPV1 26 40 CCC1(O)CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967446 EG On-Demand Anodyne EPHX2 39 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2C[C@@]2(CO)C1 ZINC000880967447 DD On-Demand Anodyne RBP4 65 43 O=C(Nc1cnccc1C(F)(F)F)NC1(Cc2ccccc2)CC1 ZINC000880967466 EH On-Demand Anodyne TRPV1 22 46 CCOCCOC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967467 EE On-Demand Anodyne RBP4 57 42 C[C@H]1[C@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967468 DD On-Demand Anodyne DRD4 43 40 C[C@H]1[C@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967468 DD On-Demand Anodyne ACHE 29 42 C[C@H]1[C@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967468 DD On-Demand Anodyne SIGMAR1 54 40 CN(C)c1nccc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880967469 EE On-Demand Anodyne TRPV1 27 50 C[C@@H]1[C@@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967471 DD On-Demand Anodyne DRD4 43 40 C[C@@H]1[C@@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967471 DD On-Demand Anodyne ACHE 29 42 C[C@@H]1[C@@H](C(=O)N2CC3(CN(Cc4ccccc4)C3)C2)CCN1C ZINC000880967471 DD On-Demand Anodyne SIGMAR1 54 40 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc2ccccc2c1 ZINC000880967472 EF On-Demand Anodyne HDAC1 15 52 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc2ccccc2c1 ZINC000880967472 EF On-Demand Anodyne IMDH_CRYPV 19 42 CN(CCO)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967474 ED On-Demand Anodyne IMDH_CRYPV 25 41 Cn1nc2c(cc1=O)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967475 FD On-Demand Anodyne RBP4 45 36 COC(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967476 EF On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCCNC1=O ZINC000880967477 DD On-Demand Anodyne TRPV1 26 41 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1C ZINC000880967478 EF On-Demand Anodyne RBP4 40 37 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCCNC1=O ZINC000880967479 DD On-Demand Anodyne TRPV1 26 41 COC(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1C ZINC000880967480 EF On-Demand Anodyne RBP4 40 37 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967482 EF On-Demand Anodyne RBP4 40 37 COC(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967487 DE On-Demand Anodyne TRPV1 26 49 CN1CCCC[C@H]1CCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880967491 EF On-Demand Anodyne SIGMAR1 46 40 CN1CCCC[C@H]1CCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880967491 EF On-Demand Anodyne ACKR3 54 36 CN1CCCC[C@@H]1CCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880967492 EF On-Demand Anodyne SIGMAR1 46 40 CN1CCCC[C@@H]1CCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880967492 EF On-Demand Anodyne ACKR3 54 36 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967495 DG On-Demand Anodyne RBP4 85 45 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967495 DG On-Demand Anodyne SFRP1 68 35 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967495 DG On-Demand Anodyne WNT3 64 35 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967497 DG On-Demand Anodyne RBP4 85 45 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967497 DG On-Demand Anodyne SFRP1 68 35 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967497 DG On-Demand Anodyne WNT3 64 35 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967498 DG On-Demand Anodyne RBP4 85 45 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967498 DG On-Demand Anodyne SFRP1 68 35 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1F ZINC000880967498 DG On-Demand Anodyne WNT3 64 35 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967500 DG On-Demand Anodyne RBP4 85 45 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967500 DG On-Demand Anodyne SFRP1 68 35 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1F ZINC000880967500 DG On-Demand Anodyne WNT3 64 35 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(Cl)c1 ZINC000880967511 FD On-Demand Anodyne EPHX2 25 49 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(Cl)c1 ZINC000880967511 FD On-Demand Anodyne MCHR1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCC2=O)C1 ZINC000880967514 EE On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCC2=O)C1 ZINC000880967517 EE On-Demand Anodyne RBP4 65 42 CC(=O)c1cccc(OCc2cn(CC(=O)N3CCCc4ccccc43)nn2)c1 ZINC000880967518 GG On-Demand Anodyne AVPR2 33 45 CN(C)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967525 DF On-Demand Anodyne RBP4 75 43 O=C(Nc1cc(C2CC2)[nH]n1)Nc1cnccc1C(F)(F)F ZINC000880967527 DG On-Demand Anodyne CDK2 17 52 O=C(Nc1cc(C2CC2)[nH]n1)Nc1cnccc1C(F)(F)F ZINC000880967527 DG On-Demand Anodyne PKNB 63 40 O=C(Nc1cc(C2CCCC2)[nH]n1)Nc1cnccc1C(F)(F)F ZINC000880967528 EI On-Demand Anodyne CDK2 15 48 O=C(Nc1cc(C2CCCC2)[nH]n1)Nc1cnccc1C(F)(F)F ZINC000880967528 EI On-Demand Anodyne PKNB 46 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880967529 GH On-Demand Anodyne CACNA1H 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880967529 GH On-Demand Anodyne S1PR2 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880967529 GH On-Demand Anodyne RBP4 55 38 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880967530 GF On-Demand Anodyne TRPV1 28 43 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880967530 GF On-Demand Anodyne SCN10A 18 40 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880967530 GF On-Demand Anodyne STAT6 55 35 O=C(NCc1cnc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880967530 GF On-Demand Anodyne NAMPT 46 39 N#Cc1cccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880967537 GF On-Demand Mild TRPV1 16 45 N#Cc1cccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880967537 GF On-Demand Mild RBP4 53 39 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967540 GD On-Demand Anodyne FDFT1 22 41 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967540 GD On-Demand Anodyne PDE6D 41 38 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967540 GD On-Demand Anodyne TIMP3 49 33 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967541 GD On-Demand Anodyne FDFT1 22 41 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967541 GD On-Demand Anodyne PDE6D 41 38 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)CC1 ZINC000880967541 GD On-Demand Anodyne TIMP3 49 33 CN(CC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)C1CCC1 ZINC000880967542 DD On-Demand Anodyne CHRM2 18 42 CN(CC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)C1CCC1 ZINC000880967542 DD On-Demand Anodyne ACE 41 35 CN(CC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)C1CCC1 ZINC000880967542 DD On-Demand Anodyne ACHE 20 41 CN(CC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)C1CCC1 ZINC000880967542 DD On-Demand Anodyne SIGMAR1 46 45 CN(CC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)C1CCC1 ZINC000880967542 DD On-Demand Anodyne SLC12A5 64 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccsc2)CC1 ZINC000880967543 FJ On-Demand Anodyne RBP4 76 46 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2cccc(Cl)c2)C1 ZINC000880967545 GI On-Demand Anodyne RBP4 60 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2cccc(Cl)c2)C1 ZINC000880967546 GI On-Demand Anodyne RBP4 60 41 COC(=O)C1=NOC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)C1 ZINC000880967547 GE On-Demand Anodyne RBP4 40 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(Cl)ccc2C1 ZINC000880967551 FI On-Demand Anodyne MAPK1 40 36 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(Cl)ccc2C1 ZINC000880967551 FI On-Demand Anodyne RBP4 55 38 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ncn1 ZINC000880967552 GE On-Demand Anodyne PDGFRB 55 39 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ncn1 ZINC000880967552 GE On-Demand Anodyne TRPV1 19 46 COc1cc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)ncn1 ZINC000880967552 GE On-Demand Anodyne RBP4 56 49 O=C(NC[C@@H](O)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880967554 DE On-Demand Anodyne TRPV1 22 48 O=C(NC[C@H](O)C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880967555 DE On-Demand Anodyne TRPV1 22 48 CS[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N(C)C ZINC000880967580 EF On-Demand Anodyne RBP4 62 43 CS[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N(C)C ZINC000880967581 EF On-Demand Anodyne RBP4 62 43 CS[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N(C)C ZINC000880967582 EF On-Demand Anodyne RBP4 62 43 CS[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N(C)C ZINC000880967583 EF On-Demand Anodyne RBP4 62 43 Cc1ccncc1[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967586 DH On-Demand Anodyne TRPV1 15 53 Cc1ccncc1[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967587 DH On-Demand Anodyne TRPV1 15 53 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967599 DH On-Demand Anodyne TRPV1 18 44 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967599 DH On-Demand Anodyne NPY5R 19 42 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967599 DH On-Demand Anodyne RBP4 69 43 CCOC(=O)c1cc(NC(=O)Nc2cnccc2C(F)(F)F)cn1C ZINC000880967600 FG On-Demand Anodyne P2RY1 43 36 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccc2ccccc2c1 ZINC000880967601 FG On-Demand Anodyne HDAC1 15 52 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccc2ccccc2c1 ZINC000880967601 FG On-Demand Anodyne IMDH_CRYPV 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(CC(F)F)CC1 ZINC000880967604 FF On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(F)cn2)CC1 ZINC000880967606 FF On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(F)cn2)CC1 ZINC000880967606 FF On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(F)cn2)CC1 ZINC000880967606 FF On-Demand Anodyne DGAT1 29 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H]2CCOC2)CC1 ZINC000880967607 EG On-Demand Anodyne RBP4 71 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H]2CCOC2)CC1 ZINC000880967608 EG On-Demand Anodyne RBP4 71 43 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880967611 DI On-Demand Anodyne KCNA5 19 41 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880967611 DI On-Demand Anodyne TRPV1 28 54 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880967611 DI On-Demand Anodyne SOAT1 23 45 Cn1nc2c(c1-c1cn(CC(=O)NCc3ccccc3)nn1)CCCC2 ZINC000880967615 FD On-Demand Anodyne ACHE 40 36 Cn1nc2c(c1-c1cn(CC(=O)NCc3ccccc3)nn1)CCCC2 ZINC000880967615 FD On-Demand Anodyne BCHE 70 32 O=C(NCC(F)(F)F)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967616 GF On-Demand Anodyne RBP4 69 43 O=C(NCC(F)(F)F)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967617 GF On-Demand Anodyne RBP4 69 43 O=C(NCC(=O)N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880967622 ED On-Demand Anodyne TRPV1 16 43 O=C(NCC1(CCO)CC1)Nc1cnccc1C(F)(F)F ZINC000880967625 DE On-Demand Anodyne TRPV1 17 47 CC(C)c1nnc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)o1 ZINC000880967626 GG On-Demand Anodyne RBP4 53 38 CC(C)c1nnc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)o1 ZINC000880967627 GG On-Demand Anodyne RBP4 53 38 O=C(Cn1cc(CN2CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967629 EG On-Demand Anodyne MCHR1 24 41 O=C(Cn1cc(CN2CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967629 EG On-Demand Anodyne IMDH_CRYPV 24 42 O=C(Cn1cc(CC2(O)CCCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967633 FG On-Demand Anodyne IMDH_CRYPV 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCCO)C1 ZINC000880967634 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCCO)C1 ZINC000880967634 EE On-Demand Anodyne LIPG 33 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCCO)C1 ZINC000880967635 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCCO)C1 ZINC000880967635 EE On-Demand Anodyne LIPG 33 41 COC(=O)[C@@H](C)OCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967639 FE On-Demand Anodyne IMDH_CRYPV 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880967641 GH On-Demand Anodyne S1PR2 27 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(Cc2ccc(F)cc2)CC1 ZINC000880967641 GH On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2F)CC1 ZINC000880967642 GI On-Demand Anodyne EPHX2 26 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2F)CC1 ZINC000880967642 GI On-Demand Anodyne RBP4 74 44 CO[C@@]1(C(F)(F)F)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967644 FH On-Demand Anodyne RBP4 45 38 Cc1nnc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)o1 ZINC000880967653 FE On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)C2CC2)CC1 ZINC000880967658 FF On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)C2CC2)CC1 ZINC000880967658 FF On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)C2CC2)CC1 ZINC000880967658 FF On-Demand Anodyne SFRP1 56 34 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)C2CC2)CC1 ZINC000880967658 FF On-Demand Anodyne WNT3 50 34 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(O)(c2cccnc2)CC1 ZINC000880967661 GG On-Demand Anodyne EPHX2 27 44 CCN(C)C(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967662 DD On-Demand Anodyne TRPV1 17 46 C[C@@H]1CCSCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967669 DG On-Demand Anodyne RBP4 45 38 C[C@H]1CCSCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967671 DG On-Demand Anodyne RBP4 45 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCOc2ccc(F)cc21 ZINC000880967674 FH On-Demand Anodyne TRPV1 31 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOc2ccc(F)cc21 ZINC000880967675 FH On-Demand Anodyne TRPV1 31 50 O=C(NCC1OCCCO1)Nc1cnccc1C(F)(F)F ZINC000880967680 DD On-Demand Anodyne TRPV1 18 45 Nc1ccc(OCc2cn(CC(=O)N3CCCc4ccccc43)nn2)cc1 ZINC000880967685 FE On-Demand Clean AVPR2 21 44 COC(=O)Cc1cn(CC(=O)N2CCCc3ccccc32)nn1 ZINC000880967697 DC On-Demand Anodyne AVPR2 39 42 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967698 FI On-Demand Anodyne RBP4 58 40 C[C@@H]1[C@@H](C(F)(F)F)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967698 FI On-Demand Anodyne WNT3 40 31 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967699 FI On-Demand Anodyne RBP4 58 40 C[C@H]1[C@H](C(F)(F)F)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967699 FI On-Demand Anodyne WNT3 40 31 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967706 EE On-Demand Anodyne EPHX2 50 43 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967706 EE On-Demand Anodyne CCR8 33 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967706 EE On-Demand Anodyne SFRP1 88 35 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967706 EE On-Demand Anodyne WNT3 70 33 CCOC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967707 EE On-Demand Anodyne EPHX2 50 43 CCOC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967707 EE On-Demand Anodyne CCR8 33 42 CCOC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967707 EE On-Demand Anodyne SFRP1 88 35 CCOC(=O)N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967707 EE On-Demand Anodyne WNT3 70 33 O=C(NNC(=O)C1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880967708 DE On-Demand Reactive TRPV1 20 41 O=C(NCCCNC(=O)C1CCC1)Nc1cnccc1C(F)(F)F ZINC000880967709 EF On-Demand Anodyne TRPV1 18 45 O=C(NCCCNC(=O)C1CCC1)Nc1cnccc1C(F)(F)F ZINC000880967709 EF On-Demand Anodyne TBK1 83 38 O=C(Nc1cnccc1C(F)(F)F)N1CCOCC2(CC2)C1 ZINC000880967711 DF On-Demand Anodyne RBP4 55 39 C[C@H]1[C@H](C)C[C@@H](C)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967713 DH On-Demand Anodyne RBP4 49 41 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967715 DH On-Demand Anodyne RBP4 49 41 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1C ZINC000880967716 DH On-Demand Anodyne RBP4 49 41 O=C(Cn1cc(CNC2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967717 DE On-Demand Anodyne NMT1 19 41 O=C(Cn1cc(CNC2CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967717 DE On-Demand Anodyne IMDH_CRYPV 20 42 O=C(NC[C@@H]1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967719 DE On-Demand Anodyne TRPV1 20 46 O=C(CC1CC1)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967720 DE On-Demand Reactive TRPV1 26 43 O=C(NC[C@H]1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967721 DE On-Demand Anodyne TRPV1 20 46 O=C(NC[C@H]1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967722 DE On-Demand Anodyne TRPV1 20 46 O=C(NNC(=O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880967723 CD On-Demand Reactive TRPV1 23 41 O=C(NNC(=O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880967723 CD On-Demand Reactive RBP4 42 38 O=C(NC[C@@H]1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967724 DE On-Demand Anodyne TRPV1 20 46 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccccc3)nn2)CC1 ZINC000880967726 FD On-Demand Anodyne FDFT1 31 44 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccccc3)nn2)CC1 ZINC000880967726 FD On-Demand Anodyne PDE6D 51 35 O=C(NCCC(=O)N1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880967727 EF On-Demand Anodyne TRPV1 23 48 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)CC1 ZINC000880967728 FD On-Demand Anodyne FDFT1 31 44 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)CC1 ZINC000880967728 FD On-Demand Anodyne PDE6D 51 35 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CC(C)(C)O ZINC000880967730 FE On-Demand Anodyne RBP4 59 42 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CC(C)(C)O ZINC000880967731 FE On-Demand Anodyne RBP4 59 42 CC[C@@H]1[C@H](C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967735 DH On-Demand Anodyne RBP4 40 38 CC[C@H]1[C@@H](C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967736 DH On-Demand Anodyne RBP4 40 38 CC[C@H]1[C@H](C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967739 DH On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCc2sccc21 ZINC000880967740 EI On-Demand Anodyne TRPV1 24 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCc2sccc21 ZINC000880967742 EI On-Demand Anodyne TRPV1 24 43 C[C@]1(O)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967747 DE On-Demand Anodyne RBP4 57 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nnc3n2CCCC3)CC1 ZINC000880967748 GG On-Demand Anodyne RBP4 69 41 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccc(C)cc3)nn2)CC1 ZINC000880967749 GD On-Demand Anodyne FDFT1 20 44 O=C(Cn1cc(CCN2CCNCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967750 FD On-Demand Anodyne IMDH_CRYPV 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880967752 GH On-Demand Anodyne TRPV1 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880967752 GH On-Demand Anodyne CCR3 33 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880967752 GH On-Demand Anodyne FAAH 40 60 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880967752 GH On-Demand Anodyne RBP4 57 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccc(F)c2)CC1 ZINC000880967752 GH On-Demand Anodyne CACNA1G 17 40 CC(C)(C)CC(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967756 DF On-Demand Reactive TRPV1 19 42 C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967759 DH On-Demand Anodyne RBP4 47 39 C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967759 DH On-Demand Anodyne SFRP1 44 35 C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967759 DH On-Demand Anodyne WNT3 46 35 C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880967759 DH On-Demand Anodyne TRPC6 50 36 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967762 DH On-Demand Anodyne RBP4 47 39 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967762 DH On-Demand Anodyne SFRP1 44 35 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967762 DH On-Demand Anodyne WNT3 46 35 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967762 DH On-Demand Anodyne TRPC6 50 36 NC(=O)CCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967763 EF On-Demand Anodyne RBP4 67 41 CN(C)CCCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967764 FH On-Demand Anodyne RBP4 70 40 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cc(F)ccc2C1 ZINC000880967765 EH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccc(O)cc1 ZINC000880967766 FF On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccc(O)cc1 ZINC000880967766 FF On-Demand Anodyne YARS 60 33 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880967770 GD On-Demand Anodyne DRD4 17 41 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880967770 GD On-Demand Anodyne FAAH 21 47 CC(C)(C)OC(=O)NCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967771 GG On-Demand Anodyne IMDH_CRYPV 23 40 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccc(C)cc3)nn2)CC1 ZINC000880967773 GD On-Demand Anodyne FDFT1 20 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CCO ZINC000880967774 ED On-Demand Anodyne RBP4 64 44 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CCO ZINC000880967775 ED On-Demand Anodyne RBP4 64 44 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccccc3)nn2)CC1 ZINC000880967776 FC On-Demand Anodyne SIGMAR1 25 42 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccccc3)nn2)CC1 ZINC000880967776 FC On-Demand Anodyne FAAH 19 41 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccccc3)nn2)CC1 ZINC000880967776 FC On-Demand Anodyne NPFFR1 42 36 COC[C@H](Cc1ccccc1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880967777 FH On-Demand Anodyne NPY5R 17 45 COC[C@@H](Cc1ccccc1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880967778 FH On-Demand Anodyne NPY5R 17 45 O=C(NCc1nc(C(F)(F)F)n[nH]1)Nc1cnccc1C(F)(F)F ZINC000880967782 FF On-Demand Anodyne TRPV1 22 51 O=C(NCC(F)(F)C(F)F)Nc1cnccc1C(F)(F)F ZINC000880967788 DG On-Demand Mild TRPV1 22 51 CCC1(CC)CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@@]1=O ZINC000880967789 FG On-Demand Anodyne RBP4 47 38 CCC1(CC)CN(C(=O)Nc2cnccc2C(F)(F)F)CC[S@]1=O ZINC000880967790 FG On-Demand Anodyne RBP4 47 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2c(F)cccc2F)C1 ZINC000880967792 FI On-Demand Anodyne RBP4 94 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2c(F)cccc2F)C1 ZINC000880967793 FI On-Demand Anodyne RBP4 94 47 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccc(F)cc2F)C1 ZINC000880967794 GH On-Demand Anodyne RBP4 60 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccc(F)cc2F)C1 ZINC000880967795 GH On-Demand Anodyne RBP4 60 41 O=C(CCCNC(=O)Nc1cnccc1C(F)(F)F)NC1CC1 ZINC000880967800 EE On-Demand Anodyne TRPV1 23 44 CC[C@@H](CC(F)(F)F)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880967801 EH On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC(F)F)C1 ZINC000880967810 EG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OC(F)F)C1 ZINC000880967810 EG On-Demand Anodyne PIM3 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC(F)F)C1 ZINC000880967812 EG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OC(F)F)C1 ZINC000880967812 EG On-Demand Anodyne PIM3 18 40 COC(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CCOCC1 ZINC000880967814 FE On-Demand Anodyne TRPV1 20 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](COc2ccccc2)C1 ZINC000880967823 GG On-Demand Anodyne RBP4 92 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCCO)CC1 ZINC000880967824 EG On-Demand Anodyne RBP4 68 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](COc2ccccc2)C1 ZINC000880967825 GG On-Demand Anodyne RBP4 92 45 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1cccc(Cl)c1 ZINC000880967833 DE On-Demand Anodyne MCHR1 17 40 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1cccc(Cl)c1 ZINC000880967835 DE On-Demand Anodyne MCHR1 17 40 Cc1cc(NC(=O)Nc2cnccc2C(F)(F)F)nn1C ZINC000880967837 CF On-Demand Anodyne TRPV1 15 40 Cc1cc(NC(=O)Nc2cnccc2C(F)(F)F)nn1C ZINC000880967837 CF On-Demand Anodyne ABL2 36 42 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1CO ZINC000880967838 DE On-Demand Anodyne RBP4 40 38 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1CO ZINC000880967840 DE On-Demand Anodyne RBP4 40 38 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1CO ZINC000880967841 DE On-Demand Anodyne RBP4 40 38 C[C@@H]1CCOCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967842 DF On-Demand Anodyne RBP4 43 38 C[C@H]1CCOCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967843 DF On-Demand Anodyne RBP4 43 38 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1CO ZINC000880967844 DE On-Demand Anodyne RBP4 40 38 CN(C)CCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967851 DE On-Demand Anodyne IMDH_CRYPV 26 42 O=C(Nc1cnccc1C(F)(F)F)N1CCSC2(CCOCC2)C1 ZINC000880967852 FG On-Demand Anodyne RBP4 40 37 O=C(NCCc1ccc(CO)cc1)Nc1cnccc1C(F)(F)F ZINC000880967855 EF On-Demand Anodyne TRPV1 21 60 O=C(NCCc1ccc(CO)cc1)Nc1cnccc1C(F)(F)F ZINC000880967855 EF On-Demand Anodyne RAF1 23 42 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)C1CCCCC1 ZINC000880967856 EH On-Demand Anodyne TRPV1 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(OCC(F)F)C1 ZINC000880967857 EF On-Demand Anodyne RBP4 77 46 O=C1NC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CO1 ZINC000880967859 EE On-Demand Anodyne RBP4 55 39 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967861 FD On-Demand Anodyne CASR 42 37 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967861 FD On-Demand Anodyne EPHX2 21 41 CN(C)CCc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880967862 FH On-Demand Anodyne TRPV1 24 53 CN(C)CCc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880967862 FH On-Demand Anodyne NAMPT 41 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C[C@H]2CCOC2)C1 ZINC000880967863 FH On-Demand Anodyne RBP4 54 39 CCc1cnc(CNC(=O)Nc2cnccc2C(F)(F)F)o1 ZINC000880967865 DF On-Demand Anodyne TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C[C@@H]2CCOC2)C1 ZINC000880967866 FH On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C[C@H]2CCOC2)C1 ZINC000880967868 FH On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccc(F)cc1 ZINC000880967869 FF On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)Cc1ccc(F)cc1 ZINC000880967869 FF On-Demand Anodyne AKT1 41 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C[C@@H]2CCOC2)C1 ZINC000880967870 FH On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccc(F)cc1 ZINC000880967871 FF On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)Cc1ccc(F)cc1 ZINC000880967871 FF On-Demand Anodyne AKT1 41 34 Cc1csc([C@H](C)CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880967872 EH On-Demand Anodyne TRPV1 15 43 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967876 GG On-Demand Anodyne CACNA1I 49 36 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967876 GG On-Demand Anodyne GPR119 45 45 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967876 GG On-Demand Anodyne SFRP1 68 40 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967876 GG On-Demand Anodyne WNT3 52 35 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967878 GG On-Demand Anodyne CACNA1I 49 36 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967878 GG On-Demand Anodyne GPR119 45 45 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967878 GG On-Demand Anodyne SFRP1 68 40 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880967878 GG On-Demand Anodyne WNT3 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cn[nH]c2)CC1 ZINC000880967881 EG On-Demand Anodyne RBP4 74 44 O=C(NC[C@H]1CCC=CO1)Nc1cnccc1C(F)(F)F ZINC000880967889 DF On-Demand Anodyne TRPV1 15 44 Cc1cc(NC(=O)Nc2cnccc2C(F)(F)F)c(C)c(C)c1O ZINC000880967897 EI On-Demand Anodyne TRPV1 21 42 O=C(NOCC(F)F)Nc1cnccc1C(F)(F)F ZINC000880967904 CE On-Demand Anodyne TRPV1 15 42 CC[C@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967905 EJ On-Demand Anodyne RBP4 75 42 CC[C@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967905 EJ On-Demand Anodyne TRPM8 45 49 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967906 EJ On-Demand Anodyne RBP4 75 42 CC[C@@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880967906 EJ On-Demand Anodyne TRPM8 45 49 CCOCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1CC ZINC000880967907 FG On-Demand Anodyne RBP4 54 39 CCOCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1CC ZINC000880967909 FG On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)NC12CCC(CC1)C2 ZINC000880967910 CH On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)NC12CCC(CC1)C2 ZINC000880967910 CH On-Demand Anodyne EPHX2 37 45 C[C@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880967914 EG On-Demand Anodyne TRPV1 18 41 C[C@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880967914 EG On-Demand Anodyne CCR5 17 41 C[C@@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880967916 EG On-Demand Anodyne TRPV1 18 41 C[C@@H](CCNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880967916 EG On-Demand Anodyne CCR5 17 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967918 GE On-Demand Anodyne CHRNA7 20 45 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967918 GE On-Demand Anodyne EPHX2 23 44 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)C(F)(F)F ZINC000880967921 EF On-Demand Anodyne TRPV1 22 47 C[C@@](O)(C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C(F)(F)F ZINC000880967925 GH On-Demand Anodyne RBP4 69 42 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880967930 GG On-Demand Anodyne HDAC10 18 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880967930 GG On-Demand Anodyne HDAC3 20 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880967930 GG On-Demand Anodyne HDAC6 15 40 CC(C)(C)OC(=O)CNCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880967932 GF On-Demand Anodyne IMDH_CRYPV 26 40 Cn1cc([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)cn1 ZINC000880967933 FG On-Demand Anodyne RBP4 69 43 CN(CCO)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880967934 EE On-Demand Anodyne RBP4 77 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2F)CC1 ZINC000880967937 GH On-Demand Anodyne TRPV1 21 56 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2F)CC1 ZINC000880967937 GH On-Demand Anodyne FAAH 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(F)c2F)CC1 ZINC000880967937 GH On-Demand Anodyne RBP4 59 46 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880967946 DF On-Demand Anodyne TRPV1 15 40 C[C@@H]1[C@@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880967946 DF On-Demand Anodyne RBP4 52 39 C[C@H]1[C@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880967947 DF On-Demand Anodyne TRPV1 15 40 C[C@H]1[C@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880967947 DF On-Demand Anodyne RBP4 52 39 O=C(NCC1(CO)CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880967952 EG On-Demand Anodyne TRPV1 16 47 COc1ccc([C@H](CCO)NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880967953 FG On-Demand Anodyne TRPV1 15 49 COc1ccc([C@@H](CCO)NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880967954 FG On-Demand Anodyne TRPV1 15 49 O=C(Cn1cc(C2CCNCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880967958 EF On-Demand Anodyne IMDH_CRYPV 28 44 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)C1 ZINC000880967959 EF On-Demand Anodyne HDAC10 16 42 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)C1 ZINC000880967959 EF On-Demand Anodyne HDAC3 18 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)C1 ZINC000880967960 EF On-Demand Anodyne HDAC10 16 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(Cl)c3)nn2)C1 ZINC000880967960 EF On-Demand Anodyne HDAC3 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CCOCC1 ZINC000880967962 EH On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CCOCC1 ZINC000880967963 EH On-Demand Anodyne RBP4 53 39 COC(=O)c1ccc2c(c1)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880967968 GG On-Demand Anodyne RBP4 45 36 O=C(Cn1cc(CN2CCCCC2=O)nn1)Nc1ccc2ccccc2c1 ZINC000880967969 FF On-Demand Anodyne IMDH_CRYPV 16 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](Cc2ccccc2)C1 ZINC000880967974 FH On-Demand Anodyne RBP4 91 46 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](Cc2ccccc2)C1 ZINC000880967975 FH On-Demand Anodyne RBP4 91 46 CCOC(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967979 CD On-Demand Reactive TRPV1 18 42 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967982 GF On-Demand Anodyne TRPV1 22 52 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967982 GF On-Demand Anodyne CCR3 23 40 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967982 GF On-Demand Anodyne ABL2 43 36 O=C(NCc1ccccc1CN1CC[C@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967982 GF On-Demand Anodyne MCHR1 18 42 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967983 GF On-Demand Anodyne TRPV1 22 52 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967983 GF On-Demand Anodyne CCR3 23 40 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967983 GF On-Demand Anodyne ABL2 43 36 O=C(NCc1ccccc1CN1CC[C@@H](O)C1)Nc1cnccc1C(F)(F)F ZINC000880967983 GF On-Demand Anodyne MCHR1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ncccc2F)CC1 ZINC000880967993 GG On-Demand Anodyne TRPV1 35 52 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ncccc2F)CC1 ZINC000880967993 GG On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)NC1Cc2ccccc2C1 ZINC000880967995 DG On-Demand Anodyne TRPV1 32 45 O=C(Nc1cnccc1C(F)(F)F)NC1Cc2ccccc2C1 ZINC000880967995 DG On-Demand Anodyne EPHX2 22 45 CC#CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880967997 CE On-Demand Mild TRPV1 22 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880967998 FG On-Demand Anodyne RBP4 73 44 CC(C)(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968001 EI On-Demand Anodyne TRPV1 22 43 CC(C)(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968001 EI On-Demand Anodyne RBP4 75 44 CC(C)(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968001 EI On-Demand Anodyne SFRP1 63 35 CC(C)(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968001 EI On-Demand Anodyne WNT3 53 33 O=C1NCC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)O1 ZINC000880968002 EE On-Demand Anodyne NPY5R 16 42 O=C1NCC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)O1 ZINC000880968002 EE On-Demand Anodyne RBP4 54 39 CCC[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CCOC ZINC000880968006 FG On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880968007 GG On-Demand Anodyne NPY5R 28 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(C1)C(=O)Nc1ccccc12 ZINC000880968007 GG On-Demand Anodyne RBP4 57 40 CCC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CCOC ZINC000880968008 FG On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880968009 GG On-Demand Anodyne NPY5R 28 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(C1)C(=O)Nc1ccccc12 ZINC000880968009 GG On-Demand Anodyne RBP4 57 40 CS[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)C(C)(C)C ZINC000880968010 EH On-Demand Anodyne TRPV1 15 44 CC(=O)CCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968013 EF On-Demand Anodyne HDAC1 15 52 CC(=O)CCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968013 EF On-Demand Anodyne IMDH_CRYPV 27 42 CC(=O)CCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968013 EF On-Demand Anodyne SUCNR1 59 35 C#CCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968020 CF On-Demand Mild TRPV1 16 48 CCC(=O)NNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968021 CD On-Demand Reactive TRPV1 22 44 CCOC(=O)CCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968027 FH On-Demand Anodyne RBP4 62 40 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CC1 ZINC000880968030 FF On-Demand Anodyne EPHX2 44 44 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CC1 ZINC000880968030 FF On-Demand Anodyne RBP4 68 42 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CC1 ZINC000880968030 FF On-Demand Anodyne SFRP1 94 37 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CC1 ZINC000880968030 FF On-Demand Anodyne WNT3 75 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCC2CC2)C1 ZINC000880968031 EH On-Demand Anodyne RBP4 63 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCC2CC2)C1 ZINC000880968031 EH On-Demand Anodyne LIPG 30 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCC2CC2)C1 ZINC000880968031 EH On-Demand Anodyne SFRP1 61 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCC2CC2)C1 ZINC000880968031 EH On-Demand Anodyne WNT3 58 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCC2CC2)C1 ZINC000880968032 EH On-Demand Anodyne RBP4 63 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCC2CC2)C1 ZINC000880968032 EH On-Demand Anodyne LIPG 30 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCC2CC2)C1 ZINC000880968032 EH On-Demand Anodyne SFRP1 61 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCC2CC2)C1 ZINC000880968032 EH On-Demand Anodyne WNT3 58 33 COCC1=CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968034 DF On-Demand Anodyne RBP4 59 40 COc1cccc([C@H]2C[C@@H](C)CN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968040 GJ On-Demand Anodyne RBP4 48 38 CCOC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccc(F)cc3)nn2)CC1 ZINC000880968041 GD On-Demand Anodyne FDFT1 20 44 COc1cccc([C@H]2C[C@H](C)CN2C(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968042 GJ On-Demand Anodyne RBP4 48 38 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(C)(C)C1 ZINC000880968043 DI On-Demand Anodyne RBP4 60 43 CCOC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccc(F)cc3)nn2)CC1 ZINC000880968044 GD On-Demand Anodyne FDFT1 20 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(C)(C)C1 ZINC000880968045 DI On-Demand Anodyne RBP4 60 43 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CC(F)F ZINC000880968047 FG On-Demand Anodyne RBP4 57 41 O=C(Cn1cc(CC2(O)CCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968053 EF On-Demand Anodyne IMDH_CRYPV 19 41 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968055 DF On-Demand Anodyne IMDH_CRYPV 31 40 C[C@@H](O)C(C)(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968059 CE On-Demand Anodyne TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)N1CCc2nnc(O)cc2C1 ZINC000880968061 EE On-Demand Anodyne RBP4 46 38 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1cccc(Cl)c1 ZINC000880968064 DF On-Demand Anodyne GRM5 15 40 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1cccc(Cl)c1 ZINC000880968066 DF On-Demand Anodyne GRM5 15 40 O=C(NCCOC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880968067 DF On-Demand Anodyne TRPV1 22 47 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968069 ED On-Demand Anodyne TRPV1 20 45 C[C@@H](O)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968069 ED On-Demand Anodyne RBP4 62 42 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880968070 DD On-Demand Anodyne TRPV1 27 43 CN1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880968070 DD On-Demand Anodyne RBP4 45 40 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccccc2)C1 ZINC000880968073 EH On-Demand Anodyne TRPV1 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccccc2)C1 ZINC000880968073 EH On-Demand Anodyne CCR3 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(Cc2ccccc2)C1 ZINC000880968073 EH On-Demand Anodyne RBP4 93 51 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OCC[C@@H]2C1 ZINC000880968075 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OCC[C@@H]2C1 ZINC000880968075 EE On-Demand Anodyne SMO 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OCC[C@H]2C1 ZINC000880968077 EE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OCC[C@H]2C1 ZINC000880968077 EE On-Demand Anodyne SMO 18 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1S(C)(=O)=O ZINC000880968078 FD On-Demand Anodyne HSD11B1 22 40 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1S(C)(=O)=O ZINC000880968078 FD On-Demand Anodyne RBP4 59 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(O)(c2ccccc2)CC1 ZINC000880968083 GI On-Demand Anodyne TRPV1 23 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(O)(c2ccccc2)CC1 ZINC000880968083 GI On-Demand Anodyne EPHX2 27 44 C/C=C/C[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968084 DF On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880968085 FG On-Demand Anodyne INHA 18 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880968085 FG On-Demand Anodyne EPHX2 17 44 C/C=C/C[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968086 DF On-Demand Anodyne TRPV1 15 43 C/C=C\C[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968087 DF On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880968088 FG On-Demand Anodyne INHA 18 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CC(=O)N(C2CCCCC2)C1 ZINC000880968088 FG On-Demand Anodyne EPHX2 17 44 C/C=C\C[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968089 DF On-Demand Anodyne TRPV1 15 43 COC(=O)N1CCC[C@@H]([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968095 FG On-Demand Anodyne WNT3 40 31 COC(=O)N1CCC[C@H]([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968097 FG On-Demand Anodyne WNT3 40 31 O=C1NC(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]12 ZINC000880968101 EC On-Demand Anodyne RBP4 59 43 O=C1NC(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]12 ZINC000880968101 EC On-Demand Anodyne SMO 25 44 COC(=O)N1CCC[C@@H]([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968102 FG On-Demand Anodyne WNT3 40 31 O=C1NC(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]12 ZINC000880968103 EC On-Demand Anodyne RBP4 59 43 O=C1NC(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]12 ZINC000880968103 EC On-Demand Anodyne SMO 25 44 O=C(Cn1cc(CN2CCCC2=O)nn1)Nc1ccc2ccccc2c1 ZINC000880968113 EE On-Demand Anodyne IMDH_CRYPV 20 41 O=C(NCc1cccc(N2CCOCC2)n1)Nc1cnccc1C(F)(F)F ZINC000880968116 GF On-Demand Anodyne TRPV1 28 48 O=C(NOC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880968125 DG On-Demand Anodyne TRPV1 17 42 CC1(CO)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968136 DF On-Demand Anodyne RBP4 63 43 CCOC(=O)C1CCN(C(=O)Cn2cc(-c3ccc(F)nc3)nn2)CC1 ZINC000880968148 FD On-Demand Anodyne PTR1 43 33 CCn1cc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)cn1 ZINC000880968154 FF On-Demand Anodyne RBP4 55 38 C[C@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968161 EI On-Demand Anodyne RBP4 86 44 C[C@H]1c2ccccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968161 EI On-Demand Anodyne TRPM8 53 52 O=C(NCC(F)(F)CO)Nc1cnccc1C(F)(F)F ZINC000880968168 CD On-Demand Anodyne TRPV1 20 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(C1)OCc1ccccc12 ZINC000880968169 GI On-Demand Anodyne NPY5R 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(C1)OCc1ccccc12 ZINC000880968169 GI On-Demand Anodyne RBP4 54 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(C1)OCc1ccccc12 ZINC000880968170 GI On-Demand Anodyne NPY5R 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(C1)OCc1ccccc12 ZINC000880968170 GI On-Demand Anodyne RBP4 54 38 O=C(NCCN1CCCOCC1)Nc1cnccc1C(F)(F)F ZINC000880968181 ED On-Demand Anodyne TRPV1 15 42 O=C(NCCN1CCCOCC1)Nc1cnccc1C(F)(F)F ZINC000880968181 ED On-Demand Anodyne EPHX2 25 48 O=C(NCCN1CCCOCC1)Nc1cnccc1C(F)(F)F ZINC000880968181 ED On-Demand Anodyne HPGDS 23 41 O=C(NCCN1CCCOCC1)Nc1cnccc1C(F)(F)F ZINC000880968181 ED On-Demand Anodyne NAMPT 21 41 Cn1cnc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880968185 EE On-Demand Anodyne RBP4 47 38 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1c1nccn1C ZINC000880968192 FE On-Demand Anodyne RBP4 57 41 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1c1nccn1C ZINC000880968193 FE On-Demand Anodyne RBP4 57 41 C[C@@H](CCC1CC1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968205 DH On-Demand Anodyne TRPV1 25 46 C=C(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968206 CF On-Demand Mild TRPV1 21 48 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CC2)C1 ZINC000880968213 CH On-Demand Anodyne EPHX2 32 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(CC2)C1 ZINC000880968213 CH On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CC(Oc2ccc([N+](=O)[O-])cc2)C1 ZINC000880968230 GG On-Demand Bother RBP4 55 41 C[C@H]1CCCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968235 DH On-Demand Anodyne RBP4 47 39 C[C@H]1CCCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968235 DH On-Demand Anodyne WNT3 40 31 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCOCC2)CC1 ZINC000880968238 FF On-Demand Anodyne EPHX2 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCOCC2)CC1 ZINC000880968238 FF On-Demand Anodyne RBP4 48 38 CN1CCC(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)CC1 ZINC000880968239 GF On-Demand Anodyne SLC6A5 30 47 CN1CCC(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)CC1 ZINC000880968239 GF On-Demand Anodyne EPHX2 43 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H]1c1ccco1 ZINC000880968241 EI On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1c1ccco1 ZINC000880968242 EI On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H](O)C[C@H]1CO ZINC000880968243 DD On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H](O)C[C@H]1CO ZINC000880968244 DD On-Demand Anodyne RBP4 47 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ncnn2C1 ZINC000880968247 ED On-Demand Anodyne EPHX2 19 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2ncnn2C1 ZINC000880968248 ED On-Demand Anodyne EPHX2 19 42 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)NCc1ccccc1 ZINC000880968249 FB On-Demand Anodyne SIGMAR1 18 42 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)NCc1ccccc1 ZINC000880968249 FB On-Demand Anodyne NPFFR1 42 36 CC(=O)Nc1ccn([C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880968250 GF On-Demand Anodyne RBP4 61 41 CC(=O)Nc1ccn([C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880968251 GF On-Demand Anodyne RBP4 61 41 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccccc3)nn2)CC1 ZINC000880968252 EC On-Demand Anodyne FAAH 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880968253 GH On-Demand Anodyne EPHX2 28 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880968253 GH On-Demand Anodyne RBP4 64 39 O=C(Nc1cc(C2CCOCC2)[nH]n1)Nc1cnccc1C(F)(F)F ZINC000880968254 FG On-Demand Anodyne PKNB 41 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC[C@@H]1O ZINC000880968256 DF On-Demand Anodyne EPHX2 15 44 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968258 FE On-Demand Anodyne ABL1 39 40 C[C@@H](CCN1CCN(C)CC1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968258 FE On-Demand Anodyne ABL2 43 40 CCC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880968261 DG On-Demand Anodyne RBP4 69 44 CCC[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880968262 DG On-Demand Anodyne RBP4 69 44 Cc1ccc2c(c1)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)CO2 ZINC000880968264 EH On-Demand Anodyne TRPV1 23 43 Cc1ccc2c(c1)[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)CO2 ZINC000880968265 EH On-Demand Anodyne TRPV1 23 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968268 FG On-Demand Anodyne EPHX2 47 50 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968268 FG On-Demand Anodyne RBP4 42 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968268 FG On-Demand Anodyne SFRP1 87 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968268 FG On-Demand Anodyne WNT3 71 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968269 FG On-Demand Anodyne EPHX2 47 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968269 FG On-Demand Anodyne RBP4 42 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968269 FG On-Demand Anodyne SFRP1 87 36 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(C(=O)C2CCCC2)C1 ZINC000880968269 FG On-Demand Anodyne WNT3 71 35 CC(C)(C)C[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968274 DG On-Demand Anodyne TRPV1 17 43 CC(C)(C)C[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968275 DG On-Demand Anodyne TRPV1 17 43 Cc1nc(CCNC(=O)Nc2cnccc2C(F)(F)F)sc1C ZINC000880968277 EH On-Demand Anodyne TRPV1 15 47 CS(=O)(=O)N1CCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968278 FD On-Demand Anodyne SFRP1 42 33 CS(=O)(=O)N1CCC[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968278 FD On-Demand Anodyne WNT3 53 33 O=C(NC[C@@]1(O)CCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880968279 FG On-Demand Anodyne TRPV1 23 49 O=C(NC[C@]1(O)CCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880968280 FG On-Demand Anodyne TRPV1 23 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCOC2(CCCC2)C1 ZINC000880968281 EH On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOC2(CCCC2)C1 ZINC000880968282 EH On-Demand Anodyne EPHX2 15 40 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968286 EF On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(cccc2[N+](=O)[O-])C1 ZINC000880968298 FH On-Demand Bother RBP4 54 39 O=C(NCC1([C@@H](O)c2ccccc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880968299 FH On-Demand Anodyne TRPV1 18 48 O=C(NCC1([C@H](O)c2ccccc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880968300 FH On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H](CO)CC1 ZINC000880968301 DF On-Demand Anodyne TRPV1 27 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@H](CO)CC1 ZINC000880968301 DF On-Demand Anodyne EPHX2 44 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880968302 DF On-Demand Anodyne TRPV1 27 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CC[C@@H](CO)CC1 ZINC000880968302 DF On-Demand Anodyne EPHX2 44 45 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1O ZINC000880968304 DE On-Demand Anodyne RBP4 76 45 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1O ZINC000880968306 DE On-Demand Anodyne RBP4 76 45 CC(C)(C(N)=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968312 FD On-Demand Anodyne TRPV1 19 46 CC(C)(C(N)=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968312 FD On-Demand Anodyne RBP4 61 45 Cc1c(NC(=O)Nc2cnccc2C(F)(F)F)cnn1C ZINC000880968314 CF On-Demand Anodyne TRPV1 17 40 Cc1c(NC(=O)Nc2cnccc2C(F)(F)F)cnn1C ZINC000880968314 CF On-Demand Anodyne FLT1 15 45 CCC(CC)C(=O)NCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968316 GG On-Demand Anodyne IMDH_CRYPV 18 40 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2F)nn1)NCC1CCCCC1 ZINC000880968317 GF On-Demand Anodyne CACNA1I 45 32 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2F)nn1)NCC1CCCCC1 ZINC000880968318 GF On-Demand Anodyne CACNA1I 45 32 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968319 FF On-Demand Anodyne RBP4 40 39 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968320 FF On-Demand Anodyne RBP4 40 39 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968321 FF On-Demand Anodyne RBP4 40 39 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968322 FF On-Demand Anodyne RBP4 40 39 CC(C)[C@H](O)C(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968336 EG On-Demand Anodyne TRPV1 18 44 C[C@@H]1N(C(=O)Nc2cnccc2C(F)(F)F)CCOC1(C)C ZINC000880968338 DG On-Demand Anodyne RBP4 54 39 COc1cccc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)c1 ZINC000880968340 GH On-Demand Anodyne RBP4 66 44 COCCCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968341 GH On-Demand Anodyne HRH2 27 41 COCCCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968341 GH On-Demand Anodyne TRPV1 30 52 COCCCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968341 GH On-Demand Anodyne ROCK2 48 54 COCCCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968341 GH On-Demand Anodyne NAMPT 41 38 COCCCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880968341 GH On-Demand Anodyne PDS 59 40 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1C1CC1 ZINC000880968342 DF On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1C1CC1 ZINC000880968343 DF On-Demand Anodyne RBP4 53 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(F)cccc2C1 ZINC000880968344 EH On-Demand Anodyne RBP4 58 42 Cn1ccnc1[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968345 EF On-Demand Anodyne RBP4 76 43 Cn1ccnc1[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968346 EF On-Demand Anodyne RBP4 76 43 O=C(NCc1nc(C2CC2)cs1)Nc1cnccc1C(F)(F)F ZINC000880968352 EH On-Demand Anodyne TRPV1 21 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1Cc1ccccc1 ZINC000880968358 EH On-Demand Anodyne TRPV1 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1Cc1ccccc1 ZINC000880968358 EH On-Demand Anodyne CHRNA7 46 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1Cc1ccccc1 ZINC000880968358 EH On-Demand Anodyne RBP4 77 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1Cc1ccccc1 ZINC000880968359 EH On-Demand Anodyne TRPV1 24 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1Cc1ccccc1 ZINC000880968359 EH On-Demand Anodyne CHRNA7 46 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1Cc1ccccc1 ZINC000880968359 EH On-Demand Anodyne RBP4 77 43 COc1cc(C)ccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968368 EH On-Demand Anodyne TRPV1 27 50 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne F2 15 44 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne GRIN2B 18 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne PREP 28 43 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne CAPN1 29 42 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne CAPN2 49 42 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCC1CCCCC1 ZINC000880968392 GE On-Demand Anodyne NPR 57 32 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccsc2)O1 ZINC000880968393 FI On-Demand Anodyne RBP4 57 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccsc2)O1 ZINC000880968394 FI On-Demand Anodyne RBP4 57 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccsc2)O1 ZINC000880968395 FI On-Demand Anodyne RBP4 57 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccsc2)O1 ZINC000880968396 FI On-Demand Anodyne RBP4 57 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCC1CCCCC1 ZINC000880968397 ED On-Demand Anodyne AVPR1B 25 40 Cc1ccccc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968408 DH On-Demand Anodyne TRPV1 26 52 Cc1ccccc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968408 DH On-Demand Anodyne RAF1 26 41 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCC2CCCCC2)nn1 ZINC000880968410 FE On-Demand Anodyne VCP 49 32 COCC1(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968411 CE On-Demand Anodyne TRPV1 17 44 CN1Cc2ccccc2[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968412 FG On-Demand Anodyne TRPV1 29 42 CN1Cc2ccccc2[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968412 FG On-Demand Anodyne RBP4 79 42 CN1Cc2ccccc2[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968413 FG On-Demand Anodyne TRPV1 29 42 CN1Cc2ccccc2[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968413 FG On-Demand Anodyne RBP4 79 42 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968414 FD On-Demand Anodyne EPHX2 19 40 CS(=O)(=O)N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968414 FD On-Demand Anodyne NAMPT 60 42 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968415 FD On-Demand Anodyne EPHX2 19 40 CS(=O)(=O)N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968415 FD On-Demand Anodyne NAMPT 60 42 COC(=O)C1CCC(c2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)CC1 ZINC000880968416 GH On-Demand Anodyne IMDH_CRYPV 23 42 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880968422 FH On-Demand Anodyne TRPV1 15 40 C[C@@H](Cc1ccc(O)cc1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880968422 FH On-Demand Anodyne NPY5R 17 43 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)CC1 ZINC000880968425 GD On-Demand Anodyne FAAH 17 42 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)CC1 ZINC000880968425 GD On-Demand Anodyne IMDH_CRYPV 21 40 O=C(NCC1(CO)COC1)Nc1cnccc1C(F)(F)F ZINC000880968430 DD On-Demand Anodyne TRPV1 18 47 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc2ccccc2c1 ZINC000880968432 EG On-Demand Anodyne IMDH_CRYPV 26 41 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc2ccccc2c1 ZINC000880968433 EG On-Demand Anodyne IMDH_CRYPV 26 41 O=C(Cn1cc(CN2CCS(=O)CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968437 GD On-Demand Anodyne IMDH_CRYPV 17 40 COCCC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968438 FE On-Demand Anodyne C3AR1 44 42 COCCC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968438 FE On-Demand Anodyne EPHX2 52 51 COCCC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968438 FE On-Demand Anodyne CCR8 42 37 COCCC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968438 FE On-Demand Anodyne SFRP1 50 35 COCCC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968438 FE On-Demand Anodyne WNT3 41 33 Cc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968439 EJ On-Demand Anodyne RBP4 88 44 Cc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968439 EJ On-Demand Anodyne SFRP1 77 36 Cc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968439 EJ On-Demand Anodyne WNT3 71 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC(F)(F)C1 ZINC000880968445 DG On-Demand Anodyne TRPV1 21 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC(F)(F)C1 ZINC000880968445 DG On-Demand Anodyne EPHX2 22 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC(F)(F)C1 ZINC000880968446 DG On-Demand Anodyne TRPV1 21 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC(F)(F)C1 ZINC000880968446 DG On-Demand Anodyne EPHX2 22 42 C=C[C@](C)(O)c1cn(CC(=O)NCC2CCCCC2)nn1 ZINC000880968447 CD On-Demand Mild CACNA1I 43 34 C=C[C@@](C)(O)c1cn(CC(=O)NCC2CCCCC2)nn1 ZINC000880968448 CD On-Demand Mild CACNA1I 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](C2CCOCC2)C1 ZINC000880968459 EG On-Demand Anodyne RBP4 88 48 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](C2CCOCC2)C1 ZINC000880968460 EG On-Demand Anodyne RBP4 88 48 CC(C)(C)OC(=O)C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968467 GI On-Demand Anodyne RBP4 55 39 CC(C)(C)OC(=O)C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968467 GI On-Demand Anodyne SFRP1 57 34 CC(C)(C)OC(=O)C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968467 GI On-Demand Anodyne WNT3 61 33 CC(C)(C)OC(=O)C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968468 GI On-Demand Anodyne RBP4 55 39 CC(C)(C)OC(=O)C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968468 GI On-Demand Anodyne SFRP1 57 34 CC(C)(C)OC(=O)C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968468 GI On-Demand Anodyne WNT3 61 33 O=C(Nc1cnccc1C(F)(F)F)N(CCO)CCO ZINC000880968470 CC On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCO[C@H](c2ccccc2)C1 ZINC000880968476 FI On-Demand Anodyne RBP4 92 47 O=C(Nc1cnccc1C(F)(F)F)N1CCCO[C@H](c2ccccc2)C1 ZINC000880968476 FI On-Demand Anodyne SMO 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCO[C@@H](c2ccccc2)C1 ZINC000880968477 FI On-Demand Anodyne RBP4 92 47 O=C(Nc1cnccc1C(F)(F)F)N1CCCO[C@@H](c2ccccc2)C1 ZINC000880968477 FI On-Demand Anodyne SMO 19 41 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968483 EF On-Demand Anodyne RBP4 58 41 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968483 EF On-Demand Anodyne SFRP1 60 33 CCOC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968483 EF On-Demand Anodyne WNT3 59 32 O=C(NCc1cccc2c1OCCCO2)Nc1cnccc1C(F)(F)F ZINC000880968484 FH On-Demand Anodyne TRPV1 26 54 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccsc2)C1 ZINC000880968491 FH On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccsc2)C1 ZINC000880968492 FH On-Demand Anodyne RBP4 58 42 O=C(Cn1cc(CN2CCS(=O)(=O)CC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968502 GD On-Demand Anodyne IMDH_CRYPV 15 40 O=C(NCc1ccc2c(c1)COC2)Nc1cnccc1C(F)(F)F ZINC000880968503 EG On-Demand Anodyne TRPV1 23 53 O=C(NCc1ccc2c(c1)COC2)Nc1cnccc1C(F)(F)F ZINC000880968503 EG On-Demand Anodyne NAMPT 55 35 CC[C@@H](C)c1ccc(NC(=O)Cn2cc([C@H](O)CC)nn2)cc1 ZINC000880968506 DF On-Demand Anodyne SCN2A 17 44 CC[C@H](O)c1cn(CC(=O)Nc2ccc([C@H](C)CC)cc2)nn1 ZINC000880968507 DF On-Demand Anodyne SCN2A 17 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880968508 FF On-Demand Anodyne EPHX2 47 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880968509 FF On-Demand Anodyne EPHX2 47 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880968510 FF On-Demand Anodyne EPHX2 47 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880968511 FF On-Demand Anodyne EPHX2 47 44 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccccc1[N+](=O)[O-])C1CC1 ZINC000880968512 GI On-Demand Bother COLA 120 43 C[C@H](O)CCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968533 DE On-Demand Anodyne IMDH_CRYPV 28 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCCCC2=O)CC1 ZINC000880968534 FG On-Demand Anodyne RBP4 61 40 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)Cc1ccccc1 ZINC000880968537 FG On-Demand Anodyne MME 48 35 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)Cc1ccccc1 ZINC000880968537 FG On-Demand Anodyne ANPEP 48 34 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)Cc1ccccc1 ZINC000880968537 FG On-Demand Anodyne TRPV1 20 45 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)Cc1ccccc1 ZINC000880968537 FG On-Demand Anodyne FPR1 40 37 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)Cc1ccccc1 ZINC000880968537 FG On-Demand Anodyne GPR142 63 34 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)Cc1ccccc1 ZINC000880968538 FG On-Demand Anodyne MME 48 35 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)Cc1ccccc1 ZINC000880968538 FG On-Demand Anodyne ANPEP 48 34 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)Cc1ccccc1 ZINC000880968538 FG On-Demand Anodyne TRPV1 20 45 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)Cc1ccccc1 ZINC000880968538 FG On-Demand Anodyne FPR1 40 37 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)Cc1ccccc1 ZINC000880968538 FG On-Demand Anodyne GPR142 63 34 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCCCC2)CC1 ZINC000880968539 FH On-Demand Anodyne HRH3 18 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCCCC2)CC1 ZINC000880968539 FH On-Demand Anodyne RBP4 67 43 O=C(NCCCF)Nc1cnccc1C(F)(F)F ZINC000880968540 CF On-Demand Anodyne TRPV1 21 50 CC(=O)c1ccc2c(c1)CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880968558 GH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1C[C@H](O)c1ccccc1 ZINC000880968561 GG On-Demand Anodyne RBP4 59 38 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880968562 GG On-Demand Anodyne RBP4 59 38 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880968563 GG On-Demand Anodyne RBP4 59 38 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880968564 GG On-Demand Anodyne RBP4 59 38 O=C(Cn1cc(CNC2CCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968568 EG On-Demand Anodyne NMT1 25 41 O=C(Cn1cc(CNC2CCCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968568 EG On-Demand Anodyne IMDH_CRYPV 18 43 O=C(NCc1cnn(CC(F)(F)F)c1)Nc1cnccc1C(F)(F)F ZINC000880968569 FG On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(F)F)CC1 ZINC000880968576 DH On-Demand Anodyne RBP4 74 44 CS[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968579 CF On-Demand Anodyne TRPV1 17 46 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NCC1CCCCC1 ZINC000880968585 GF On-Demand Anodyne MMP8 17 43 C[C@H](C[C@@H](O)c1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968590 FH On-Demand Anodyne TRPV1 17 47 C[C@@H](C[C@H](O)c1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968591 FH On-Demand Anodyne TRPV1 17 47 O=C(Cn1cc([C@@H]2COCCN2)nn1)Nc1ccc2ccccc2c1 ZINC000880968605 ED On-Demand Anodyne IMDH_CRYPV 19 41 O=C(Cn1cc([C@H]2COCCN2)nn1)Nc1ccc2ccccc2c1 ZINC000880968606 ED On-Demand Anodyne IMDH_CRYPV 19 41 O=C(NC[C@@H]1[C@H]2Cc3ccccc3[C@@H]21)Nc1cnccc1C(F)(F)F ZINC000880968607 EH On-Demand Anodyne TRPV1 22 46 O=C(NC[C@@H]1[C@@H]2Cc3ccccc3[C@@H]12)Nc1cnccc1C(F)(F)F ZINC000880968608 EH On-Demand Anodyne TRPV1 22 46 O=C(NC[C@@H]1[C@H]2Cc3ccccc3[C@H]21)Nc1cnccc1C(F)(F)F ZINC000880968609 EH On-Demand Anodyne TRPV1 22 46 O=C(NC[C@H]1[C@H]2c3ccccc3C[C@H]21)Nc1cnccc1C(F)(F)F ZINC000880968610 EH On-Demand Anodyne TRPV1 22 46 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968612 DF On-Demand Anodyne IMDH_CRYPV 17 41 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc2ccccc2c1 ZINC000880968613 DF On-Demand Anodyne IMDH_CRYPV 17 41 COCCCOC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968614 EE On-Demand Anodyne RBP4 65 42 CCc1nc([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)n[nH]1 ZINC000880968619 FE On-Demand Anodyne RBP4 48 38 C[C@@H](CCNC(=O)Nc1cnccc1C(F)(F)F)[S@@](C)=O ZINC000880968621 DE On-Demand Anodyne TRPV1 15 44 C[C@H](CCNC(=O)Nc1cnccc1C(F)(F)F)[S@@](C)=O ZINC000880968622 DE On-Demand Anodyne TRPV1 15 44 C[C@@H](CCNC(=O)Nc1cnccc1C(F)(F)F)[S@](C)=O ZINC000880968623 DE On-Demand Anodyne TRPV1 15 44 C[C@H](CCNC(=O)Nc1cnccc1C(F)(F)F)[S@](C)=O ZINC000880968624 DE On-Demand Anodyne TRPV1 15 44 CC(C)(C)C1=CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968626 EI On-Demand Anodyne RBP4 55 41 O=C(NCc1ccc2c(c1)CCS2(=O)=O)Nc1cnccc1C(F)(F)F ZINC000880968629 GF On-Demand Anodyne TRPV1 16 50 CCC(CC)(CO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968630 DG On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H](c1cccnc1)C1CC1 ZINC000880968631 EH On-Demand Anodyne TRPV1 19 60 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](c1cccnc1)C1CC1 ZINC000880968632 EH On-Demand Anodyne TRPV1 19 60 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2CCc3ccccc3[C@H]21 ZINC000880968650 EH On-Demand Anodyne TRPV1 23 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1[C@@H]2c3ccccc3CC[C@H]21 ZINC000880968651 EH On-Demand Anodyne TRPV1 23 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@@H]2CCc3ccccc3[C@@H]21 ZINC000880968652 EH On-Demand Anodyne TRPV1 23 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1[C@H]2CCc3ccccc3[C@@H]21 ZINC000880968653 EH On-Demand Anodyne TRPV1 23 44 CC(C)(C)N1C[C@H](NC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880968683 EF On-Demand Anodyne TRPV1 22 40 CC(C)(C)N1C[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)CC1=O ZINC000880968684 EF On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(F)ccc(F)c2C1 ZINC000880968686 FH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C2CCCCC2)CC1 ZINC000880968687 FI On-Demand Anodyne EPHX2 46 50 COC(=O)C1(CNC(=O)Nc2cnccc2C(F)(F)F)CCCC1 ZINC000880968694 EF On-Demand Anodyne TRPV1 22 48 CCCCCOC1CN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968695 EH On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CSc2ccccc2)C1 ZINC000880968714 GJ On-Demand Anodyne RBP4 90 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CSc2ccccc2)C1 ZINC000880968714 GJ On-Demand Anodyne SFRP1 61 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CSc2ccccc2)C1 ZINC000880968714 GJ On-Demand Anodyne WNT3 45 32 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CSc2ccccc2)C1 ZINC000880968715 GJ On-Demand Anodyne RBP4 90 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CSc2ccccc2)C1 ZINC000880968715 GJ On-Demand Anodyne SFRP1 61 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CSc2ccccc2)C1 ZINC000880968715 GJ On-Demand Anodyne WNT3 45 32 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCC2)C1 ZINC000880968718 DH On-Demand Anodyne EPHX2 34 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCC2)C1 ZINC000880968718 DH On-Demand Anodyne RBP4 57 41 C[C@H](C#N)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968725 CE On-Demand Mild TRPV1 15 45 CC[C@@H](C)c1ccc(NC(=O)Cn2cc(C(C)(C)O)nn2)cc1 ZINC000880968727 DF On-Demand Anodyne SCN2A 17 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCc2[nH]ccc21 ZINC000880968732 DH On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCc2[nH]ccc21 ZINC000880968733 DH On-Demand Anodyne TRPV1 24 42 O=C(Nc1cnn(CC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880968742 EG On-Demand Anodyne TRPV1 19 42 O=C(Nc1cnn(CC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880968742 EG On-Demand Anodyne PANC 40 31 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880968744 GD On-Demand Anodyne NOS2 95 37 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880968745 GD On-Demand Anodyne NOS2 95 37 O=C(NCC[C@H](O)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880968753 EG On-Demand Anodyne TRPV1 19 48 O=C(NCC[C@@H](O)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880968754 EG On-Demand Anodyne TRPV1 19 48 C[C@H]1[C@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968755 EJ On-Demand Anodyne RBP4 89 45 C[C@H]1[C@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968755 EJ On-Demand Anodyne SMO 17 40 C[C@H]1[C@@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968756 EJ On-Demand Anodyne RBP4 89 45 C[C@H]1[C@@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968756 EJ On-Demand Anodyne SMO 17 40 C[C@@H]1[C@@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968757 EJ On-Demand Anodyne RBP4 89 45 C[C@@H]1[C@@H](c2ccccc2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968757 EJ On-Demand Anodyne SMO 17 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880968761 GE On-Demand Anodyne EPHX2 45 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880968761 GE On-Demand Anodyne SFRP1 84 35 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(S(=O)(=O)C2CC2)CC1 ZINC000880968761 GE On-Demand Anodyne WNT3 42 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@@H]2CCCCO2)CC1 ZINC000880968767 GH On-Demand Anodyne RBP4 51 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC[C@H]2CCCCO2)CC1 ZINC000880968768 GH On-Demand Anodyne RBP4 51 38 O=C(NCCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880968769 CG On-Demand Anodyne TRPV1 29 50 O=C(NCC1(CCO)CCCC1)Nc1cnccc1C(F)(F)F ZINC000880968773 EG On-Demand Anodyne TRPV1 15 47 Cc1nsc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880968778 FF On-Demand Anodyne TRPV1 18 45 Cc1nsc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880968778 FF On-Demand Anodyne FAAH 15 49 Cc1nsc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880968778 FF On-Demand Anodyne RBP4 45 39 Cn1ccnc1[C@@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968785 GF On-Demand Anodyne RBP4 60 38 Cn1ccnc1[C@H](O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968786 GF On-Demand Anodyne RBP4 60 38 CCN(CC)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968787 EF On-Demand Anodyne IMDH_CRYPV 32 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCc1ccccc12 ZINC000880968800 GI On-Demand Anodyne NPY5R 38 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CC1)OCc1ccccc12 ZINC000880968800 GI On-Demand Anodyne RBP4 57 41 C[C@H]1CC[C@@H](C(N)=O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968802 EE On-Demand Anodyne RBP4 53 39 C[C@H]1CC[C@H](C(N)=O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968803 EE On-Demand Anodyne RBP4 53 39 C[C@@H]1CC[C@@H](C(N)=O)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968804 EE On-Demand Anodyne RBP4 53 39 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968808 FG On-Demand Anodyne RBP4 65 41 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968808 FG On-Demand Anodyne SFRP1 101 38 CC(C)(C)OC(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968808 FG On-Demand Anodyne WNT3 80 35 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968814 ED On-Demand Anodyne ENPP1 54 32 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880968814 ED On-Demand Anodyne IMDH_CRYPV 24 41 COC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968823 EF On-Demand Anodyne RBP4 74 46 COC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968823 EF On-Demand Anodyne SFRP1 50 34 COC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968823 EF On-Demand Anodyne WNT3 40 32 COC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968823 EF On-Demand Anodyne PTR1 45 32 O=C(NCC1(CO)CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880968826 EE On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2[C@@H](CCCN2C2CC2)C1 ZINC000880968827 FH On-Demand Anodyne RBP4 69 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2[C@@H](CCCN2C2CC2)C1 ZINC000880968828 FH On-Demand Anodyne RBP4 69 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]2[C@H](CCCN2C2CC2)C1 ZINC000880968829 FH On-Demand Anodyne RBP4 69 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]2[C@H](CCCN2C2CC2)C1 ZINC000880968830 FH On-Demand Anodyne RBP4 69 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC(F)(F)C1 ZINC000880968836 DH On-Demand Anodyne EPHX2 21 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC(F)(F)C1 ZINC000880968837 DH On-Demand Anodyne EPHX2 21 46 CC(C)CN1CCC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968842 FH On-Demand Anodyne CCR3 60 39 CC(C)CN1CCC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968843 FH On-Demand Anodyne CCR3 60 39 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCOCC2)C1 ZINC000880968844 EF On-Demand Anodyne EPHX2 23 47 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCOCC2)C1 ZINC000880968844 EF On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2O)CC1 ZINC000880968845 FG On-Demand Anodyne KCNQ2 44 33 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2O)CC1 ZINC000880968845 FG On-Demand Anodyne TRPV1 23 62 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2O)CC1 ZINC000880968845 FG On-Demand Anodyne FAAH 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2O)CC1 ZINC000880968845 FG On-Demand Anodyne RBP4 73 48 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880968848 GF On-Demand Anodyne MMP8 17 43 C[C@@H]1[C@@H](NC(=O)Cn2cc(CCCOc3cccnc3F)nn2)CCC[C@H]1C ZINC000880968850 GF On-Demand Anodyne MMP8 17 43 O=C(Cn1cc([C@@H]2CCCC[C@@H]2O)nn1)Nc1ccc2ccccc2c1 ZINC000880968860 FG On-Demand Anodyne IMDH_CRYPV 19 41 O=C(Cn1cc([C@H]2CCCC[C@H]2O)nn1)Nc1ccc2ccccc2c1 ZINC000880968861 FG On-Demand Anodyne IMDH_CRYPV 19 41 O=C(Cn1cc([C@H]2CCCC[C@@H]2O)nn1)Nc1ccc2ccccc2c1 ZINC000880968862 FG On-Demand Anodyne IMDH_CRYPV 19 41 O=C(Cn1cc([C@@H]2CCCC[C@H]2O)nn1)Nc1ccc2ccccc2c1 ZINC000880968863 FG On-Demand Anodyne IMDH_CRYPV 19 41 Cc1nc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)sc1C ZINC000880968873 GH On-Demand Anodyne TRPV1 16 45 Cc1nc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)sc1C ZINC000880968873 GH On-Demand Anodyne RBP4 46 41 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968882 EE On-Demand Anodyne SFRP1 48 38 O=C(NC1CC1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968882 EE On-Demand Anodyne WNT3 55 38 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968883 EE On-Demand Anodyne SFRP1 48 38 O=C(NC1CC1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968883 EE On-Demand Anodyne WNT3 55 38 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968894 FG On-Demand Anodyne MME 40 39 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968894 FG On-Demand Anodyne ANPEP 44 31 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968894 FG On-Demand Anodyne TRPV1 19 44 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968894 FG On-Demand Anodyne GPR142 49 35 COC[C@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968895 FG On-Demand Anodyne MME 40 39 COC[C@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968895 FG On-Demand Anodyne ANPEP 44 31 COC[C@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968895 FG On-Demand Anodyne TRPV1 19 44 COC[C@H](Cc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880968895 FG On-Demand Anodyne GPR142 49 35 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1F ZINC000880968901 GH On-Demand Clean RBP4 54 54 C[C@H]1[C@H](C)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968904 CG On-Demand Anodyne RBP4 59 40 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880968905 CG On-Demand Anodyne RBP4 59 40 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1C ZINC000880968906 CG On-Demand Anodyne RBP4 59 40 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880968907 CG On-Demand Anodyne RBP4 59 40 Cn1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1=O ZINC000880968908 GD On-Demand Anodyne TRPV1 19 48 Cn1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1=O ZINC000880968908 GD On-Demand Anodyne RBP4 46 46 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)(C)CN(C)C ZINC000880968910 EG On-Demand Anodyne TRPV1 16 43 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968916 DD On-Demand Anodyne UL80 25 41 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968916 DD On-Demand Anodyne RBP4 40 38 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968916 DD On-Demand Anodyne SFRP1 45 37 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968916 DD On-Demand Anodyne WNT3 50 37 CCc1cnc(CNC(=O)Nc2cnccc2C(F)(F)F)s1 ZINC000880968919 EG On-Demand Anodyne TRPV1 17 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N(C)C ZINC000880968920 DF On-Demand Anodyne RBP4 67 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N(C)C ZINC000880968921 DF On-Demand Anodyne RBP4 67 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N(C)C ZINC000880968922 DF On-Demand Anodyne RBP4 67 44 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N(C)C ZINC000880968923 DF On-Demand Anodyne RBP4 67 44 COC(=O)CCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880968931 FG On-Demand Anodyne RBP4 68 43 C[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880968933 EE On-Demand Anodyne RBP4 61 41 C[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880968934 EE On-Demand Anodyne RBP4 61 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C[C@@H](C)O ZINC000880968935 EE On-Demand Anodyne RBP4 61 41 CC[C@]1(C)CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880968938 DI On-Demand Anodyne RBP4 50 38 CC(C)(C)OC(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880968939 DF On-Demand Anodyne TRPV1 21 47 O=C(Cn1cc(C2(O)CCC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880968940 EC On-Demand Anodyne NOS2 100 39 C[C@@H]1C[C@H]2CCCC[C@@H]2N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968943 EI On-Demand Anodyne RBP4 47 39 C[C@@H]1C[C@H]2CCCC[C@H]2N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880968944 EI On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880968948 FG On-Demand Anodyne TRPV1 38 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ncccc2F)C1 ZINC000880968948 FG On-Demand Anodyne EPHX2 26 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880968949 FG On-Demand Anodyne TRPV1 38 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ncccc2F)C1 ZINC000880968949 FG On-Demand Anodyne EPHX2 26 42 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)c1c(F)cccc1F ZINC000880968962 GI On-Demand Anodyne TRPV1 19 52 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)c1c(F)cccc1F ZINC000880968963 GI On-Demand Anodyne TRPV1 19 52 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880968968 GC On-Demand Anodyne NOS2 102 40 C=C[C@](C)(O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880968978 EC On-Demand Mild NOS2 93 38 C=C[C@@](C)(O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880968979 EC On-Demand Mild NOS2 93 38 O=C(Nc1cnccc1C(F)(F)F)N(CCO)[C@H]1CCCc2ccccc21 ZINC000880968980 GI On-Demand Anodyne TRPM8 19 41 O=C(Nc1cnccc1C(F)(F)F)N(CCO)[C@@H]1CCCc2ccccc21 ZINC000880968981 GI On-Demand Anodyne TRPM8 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CC=CC2)CC1 ZINC000880968982 EF On-Demand Anodyne RBP4 71 43 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CNC(=O)OC(C)(C)C ZINC000880968997 GG On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCCNC2=O)CC1 ZINC000880969003 FF On-Demand Anodyne RBP4 62 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2cccs2)C1 ZINC000880969004 FH On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2cccs2)C1 ZINC000880969005 FH On-Demand Anodyne RBP4 65 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)C1 ZINC000880969006 EG On-Demand Anodyne IMDH_CRYPV 15 40 O=C1CCC[C@@H](c2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)C1 ZINC000880969007 EG On-Demand Anodyne IMDH_CRYPV 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCO)CC1 ZINC000880969008 EE On-Demand Anodyne RBP4 66 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCO)CC1 ZINC000880969008 EE On-Demand Anodyne LIPG 31 41 O=C(NC[C@H](O)CO)Nc1cnccc1C(F)(F)F ZINC000880969011 CC On-Demand Anodyne TRPV1 17 47 O=C(NC[C@@H](O)CO)Nc1cnccc1C(F)(F)F ZINC000880969012 CC On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccc(O)cc2)CC1 ZINC000880969014 GF On-Demand Anodyne RBP4 63 43 CN1[C@H]2CC[C@H]1CC(N1CCN(C(=O)Nc3cnccc3C(F)(F)F)CC1)C2 ZINC000880969015 GF On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccn2)C1 ZINC000880969016 FF On-Demand Anodyne TRPV1 25 61 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccn2)C1 ZINC000880969016 FF On-Demand Anodyne EPHX2 37 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccn2)C1 ZINC000880969017 FF On-Demand Anodyne TRPV1 25 61 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccn2)C1 ZINC000880969017 FF On-Demand Anodyne EPHX2 37 41 O=C(NCCS(=O)(=O)CC1CC1)Nc1cnccc1C(F)(F)F ZINC000880969022 FE On-Demand Anodyne TRPV1 18 44 C[C@H]1CC[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969025 CH On-Demand Anodyne TRPV1 21 43 C[C@H]1CC[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969025 CH On-Demand Anodyne RBP4 59 40 C[C@H]1CC[C@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969026 CH On-Demand Anodyne TRPV1 21 43 C[C@H]1CC[C@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969026 CH On-Demand Anodyne RBP4 59 40 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969027 CH On-Demand Anodyne TRPV1 21 43 C[C@@H]1CC[C@@H](C)N1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969027 CH On-Demand Anodyne RBP4 59 40 O=C(NCc1ccccc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880969038 GG On-Demand Anodyne KCNQ2 40 35 O=C(NCc1ccccc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880969038 GG On-Demand Anodyne TRPV1 28 53 O=C(NCc1ccccc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880969038 GG On-Demand Anodyne EPHX2 16 44 O=C(NCc1ccccc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880969038 GG On-Demand Anodyne SCN10A 22 49 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880969039 FG On-Demand Anodyne EPHX2 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880969039 FG On-Demand Anodyne RBP4 79 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880969039 FG On-Demand Anodyne SCD1 26 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880969039 FG On-Demand Anodyne SFRP1 53 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](Oc2ccccn2)C1 ZINC000880969039 FG On-Demand Anodyne SCD 29 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880969040 FG On-Demand Anodyne EPHX2 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880969040 FG On-Demand Anodyne RBP4 79 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880969040 FG On-Demand Anodyne SCD1 26 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880969040 FG On-Demand Anodyne SFRP1 53 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](Oc2ccccn2)C1 ZINC000880969040 FG On-Demand Anodyne SCD 29 43 O=C(NCCc1cnc(C2CC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880969054 FG On-Demand Anodyne TRPV1 16 49 O=C(NCCc1cnc(C2CC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880969054 FG On-Demand Anodyne RAF1 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880969055 FI On-Demand Anodyne TRPV1 21 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880969055 FI On-Demand Anodyne CCR2 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880969055 FI On-Demand Anodyne RBP4 94 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880969055 FI On-Demand Anodyne SFRP1 118 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Nc2ccccc2)C1 ZINC000880969055 FI On-Demand Anodyne WNT3 84 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880969056 FI On-Demand Anodyne TRPV1 21 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880969056 FI On-Demand Anodyne CCR2 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880969056 FI On-Demand Anodyne RBP4 94 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880969056 FI On-Demand Anodyne SFRP1 118 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Nc2ccccc2)C1 ZINC000880969056 FI On-Demand Anodyne WNT3 84 39 CCNC(=O)C(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969057 EE On-Demand Anodyne TRPV1 17 45 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969069 GH On-Demand Anodyne CCR3 15 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969069 GH On-Demand Anodyne EPHX2 23 44 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969070 GH On-Demand Anodyne CCR3 15 40 CC[C@H]1CN(C(=O)C(C)C)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969070 GH On-Demand Anodyne EPHX2 23 44 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCCC2)C1 ZINC000880969074 EG On-Demand Anodyne EPHX2 22 48 O=C(Nc1cnccc1C(F)(F)F)N1CCOC2(CCCC2)C1 ZINC000880969074 EG On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N[C@]1(CO)CCc2ccccc21 ZINC000880969075 FG On-Demand Anodyne TRPV1 20 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@]1(CO)CCc2ccccc21 ZINC000880969076 FG On-Demand Anodyne TRPV1 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CC=C(C(F)(F)F)CC1 ZINC000880969077 EH On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccccc2)C1 ZINC000880969078 FH On-Demand Anodyne RBP4 91 49 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccccc2)C1 ZINC000880969078 FH On-Demand Anodyne SMO 21 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccccc2)C1 ZINC000880969079 FH On-Demand Anodyne RBP4 91 49 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccccc2)C1 ZINC000880969079 FH On-Demand Anodyne SMO 21 42 O=C(Nc1cnccc1C(F)(F)F)N1CC(CC(F)(F)F)C1 ZINC000880969081 EH On-Demand Anodyne RBP4 77 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCN2CCCC2)CC1 ZINC000880969086 GG On-Demand Anodyne RBP4 58 39 COC(=O)[C@@H](C)[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969089 GH On-Demand Anodyne TRPV1 15 46 COC(=O)[C@@H](C)[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969090 GH On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCC2CCCCC2)CC1 ZINC000880969102 GJ On-Demand Anodyne RBP4 62 39 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969103 GI On-Demand Anodyne ACHE 42 44 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969103 GI On-Demand Anodyne SIGMAR1 35 43 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969103 GI On-Demand Anodyne CCR3 50 39 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969103 GI On-Demand Anodyne RBP4 51 36 CN(C[C@@H]1CCN(Cc2ccccc2)C1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969103 GI On-Demand Anodyne CACNA1G 34 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne HTR1A 42 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne DRD2 34 46 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne ADRA1D 42 46 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne ADRA1A 35 46 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne ADRA1B 30 46 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne DRD3 40 38 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne PDE3A 22 41 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne TRPV1 23 47 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne PIM1 18 44 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne EPHX2 40 39 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne RBP4 56 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne SCD1 29 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne SFRP1 47 33 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969111 GH On-Demand Anodyne SCD 25 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne HTR1A 42 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne DRD2 34 46 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne ADRA1D 42 46 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne ADRA1A 35 46 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne ADRA1B 30 46 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne DRD3 40 38 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne PDE3A 22 41 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne TRPV1 23 47 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne PIM1 18 44 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne EPHX2 40 39 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne RBP4 56 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne SCD1 29 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne SFRP1 47 33 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969112 GH On-Demand Anodyne SCD 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1c1ccc(Cl)cc1 ZINC000880969115 FJ On-Demand Anodyne RBP4 49 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1c1ccc(Cl)cc1 ZINC000880969116 FJ On-Demand Anodyne RBP4 49 38 CCC1(CNC(=O)Nc2cnccc2C(F)(F)F)CCC1 ZINC000880969117 DH On-Demand Anodyne TRPV1 20 49 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880969124 GG On-Demand Anodyne TRPV1 16 42 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880969124 GG On-Demand Anodyne EPHX2 25 47 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880969124 GG On-Demand Anodyne RBP4 54 43 CNC(=O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969129 EC On-Demand Anodyne RBP4 55 40 CC(C)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969131 DH On-Demand Anodyne RBP4 49 38 CC(C)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969131 DH On-Demand Anodyne WNT3 41 32 O=C1CCC[C@@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969135 FD On-Demand Anodyne NOS2 98 38 O=C1CCC[C@@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969135 FD On-Demand Anodyne MCHR1 22 42 O=C1CCC[C@@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969135 FD On-Demand Anodyne LUXR 29 41 O=C1CCC[C@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969136 FD On-Demand Anodyne NOS2 98 38 O=C1CCC[C@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969136 FD On-Demand Anodyne MCHR1 22 42 O=C1CCC[C@H](c2cn(CC(=O)NCc3ccc4c(c3)OCO4)nn2)C1 ZINC000880969136 FD On-Demand Anodyne LUXR 29 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](CO)C1 ZINC000880969137 DD On-Demand Anodyne RBP4 77 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](CO)C1 ZINC000880969138 DD On-Demand Anodyne RBP4 77 44 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C[C@@H](C)O ZINC000880969139 FE On-Demand Anodyne RBP4 56 40 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1C[C@H](C)O ZINC000880969141 FE On-Demand Anodyne RBP4 56 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969143 GG On-Demand Anodyne CCKAR 17 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969143 GG On-Demand Anodyne CCKBR 19 40 COc1ccccc1N1CC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969143 GG On-Demand Anodyne RBP4 63 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969144 GG On-Demand Anodyne CCKAR 17 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969144 GG On-Demand Anodyne CCKBR 19 40 COc1ccccc1N1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1=O ZINC000880969144 GG On-Demand Anodyne RBP4 63 40 CCC1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969147 CG On-Demand Anodyne TRPV1 23 51 COCCOc1cc(C)ccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969148 GH On-Demand Anodyne TRPV1 27 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CO ZINC000880969149 CE On-Demand Anodyne RBP4 41 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CO ZINC000880969149 CE On-Demand Anodyne SFRP1 46 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CO ZINC000880969149 CE On-Demand Anodyne WNT3 49 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CO ZINC000880969150 CE On-Demand Anodyne RBP4 41 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CO ZINC000880969150 CE On-Demand Anodyne SFRP1 46 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CO ZINC000880969150 CE On-Demand Anodyne WNT3 49 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCC2CC2)CC1 ZINC000880969161 EH On-Demand Anodyne RBP4 71 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCC2CC2)CC1 ZINC000880969161 EH On-Demand Anodyne LIPG 23 41 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne TRPV1 37 48 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne P2RY1 63 43 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne RAF1 66 46 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne KDR 53 41 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne EPHX2 34 46 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne TEK 48 39 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne BRAF 41 44 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne TAAR1 39 44 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne RIPK1 64 38 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne KCNK3 51 41 COCCCOc1cccc(NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880969164 FI On-Demand Anodyne KCNK9 42 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880969181 GI On-Demand Anodyne RBP4 63 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880969181 GI On-Demand Anodyne SFRP1 46 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@H](O)c1ccccc1 ZINC000880969181 GI On-Demand Anodyne WNT3 52 34 O=C(NC[C@@H]1CC(=O)N(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880969215 GG On-Demand Anodyne TRPV1 18 42 O=C(NC[C@H]1CC(=O)N(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880969216 GG On-Demand Anodyne TRPV1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(F)cc2C1 ZINC000880969218 EH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(F)cc2C1 ZINC000880969218 EH On-Demand Anodyne TRPM8 29 41 C=C[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969221 CF On-Demand Mild TRPV1 16 47 C=C[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969222 CF On-Demand Mild TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(O)CCCC[C@@H]2C1 ZINC000880969223 EG On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(O)CCCC[C@@H]2C1 ZINC000880969224 EG On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(O)CCCC[C@H]2C1 ZINC000880969225 EG On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(O)CCCC[C@H]2C1 ZINC000880969226 EG On-Demand Anodyne RBP4 58 42 C[C@@H]1CC[C@@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969227 DH On-Demand Anodyne RBP4 56 41 C[C@H]1CC[C@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969228 DH On-Demand Anodyne RBP4 56 41 C[C@H]1CC[C@@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969229 DH On-Demand Anodyne RBP4 56 41 C[C@H]1CC[C@@H](C)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969230 DH On-Demand Anodyne RBP4 56 41 COCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969242 EE On-Demand Anodyne S1PR2 26 40 COCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969242 EE On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(F)cc(F)cc2C1 ZINC000880969247 FH On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCc3ccccc32)C1 ZINC000880969258 GH On-Demand Anodyne NPY5R 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@]2(CCc3ccccc32)C1 ZINC000880969258 GH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCc3ccccc32)C1 ZINC000880969259 GH On-Demand Anodyne NPY5R 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@]2(CCc3ccccc32)C1 ZINC000880969259 GH On-Demand Anodyne RBP4 55 39 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1n1ccnc1 ZINC000880969266 FG On-Demand Anodyne RBP4 62 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1n1ccnc1 ZINC000880969267 FG On-Demand Anodyne RBP4 62 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1n1ccnc1 ZINC000880969268 FG On-Demand Anodyne RBP4 62 41 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1n1ccnc1 ZINC000880969269 FG On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OC[C@H]2C1 ZINC000880969271 ED On-Demand Anodyne RBP4 61 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN2C(=O)OC[C@@H]2C1 ZINC000880969272 ED On-Demand Anodyne RBP4 61 44 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N1CCOCC1 ZINC000880969281 FF On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880969282 GI On-Demand Anodyne RBP4 63 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880969282 GI On-Demand Anodyne SFRP1 46 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C[C@@H](O)c1ccccc1 ZINC000880969282 GI On-Demand Anodyne WNT3 52 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880969283 GI On-Demand Anodyne RBP4 63 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880969283 GI On-Demand Anodyne SFRP1 46 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@@H](O)c1ccccc1 ZINC000880969283 GI On-Demand Anodyne WNT3 52 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@H](O)c1ccccc1 ZINC000880969284 GI On-Demand Anodyne RBP4 63 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@H](O)c1ccccc1 ZINC000880969284 GI On-Demand Anodyne SFRP1 46 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C[C@H](O)c1ccccc1 ZINC000880969284 GI On-Demand Anodyne WNT3 52 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(F)(F)F)CC1 ZINC000880969285 EH On-Demand Anodyne TRPV1 16 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(F)(F)F)CC1 ZINC000880969285 EH On-Demand Anodyne RBP4 76 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CCO)CC1 ZINC000880969288 DD On-Demand Anodyne FAAH 15 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CCO)CC1 ZINC000880969288 DD On-Demand Anodyne RBP4 57 42 Cc1cnc(CNC(=O)Nc2cnccc2C(F)(F)F)o1 ZINC000880969299 DF On-Demand Anodyne TRPV1 21 48 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969302 ED On-Demand Anodyne NOS2 99 41 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969302 ED On-Demand Anodyne MCHR1 24 45 O=C(Cn1cc([C@H]2CCCCO2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969303 ED On-Demand Anodyne NOS2 99 41 O=C(Cn1cc([C@H]2CCCCO2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969303 ED On-Demand Anodyne MCHR1 24 45 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N1CCOCC1 ZINC000880969307 FF On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)C[C@H](O)c1ccccc1 ZINC000880969313 FF On-Demand Anodyne TRPV1 16 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)C[C@@H](O)c1ccccc1 ZINC000880969315 FF On-Demand Anodyne TRPV1 16 46 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969316 GH On-Demand Anodyne GPR119 39 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969316 GH On-Demand Anodyne SFRP1 82 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969316 GH On-Demand Anodyne WNT3 69 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)C[C@@H](O)c1ccccc1 ZINC000880969317 FF On-Demand Anodyne TRPV1 16 46 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969318 GH On-Demand Anodyne GPR119 39 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969318 GH On-Demand Anodyne SFRP1 82 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(C(=O)OC(C)(C)C)C1 ZINC000880969318 GH On-Demand Anodyne WNT3 69 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)C[C@H](O)c1ccccc1 ZINC000880969319 FF On-Demand Anodyne TRPV1 16 46 COCCNc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969321 FG On-Demand Anodyne TRPV1 30 57 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)S(C)(=O)=O ZINC000880969326 EE On-Demand Anodyne TRPV1 23 47 CC1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969339 CG On-Demand Anodyne RBP4 59 42 Cc1nc(CN(C)[C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)no1 ZINC000880969345 GF On-Demand Anodyne RBP4 54 38 CN(C)CC1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969347 EG On-Demand Anodyne TRPV1 25 40 CN(C)CC1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969347 EG On-Demand Anodyne EPHX2 42 42 Cc1nc(CN(C)[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)no1 ZINC000880969349 GF On-Demand Anodyne RBP4 54 38 CC(C)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969351 DH On-Demand Anodyne RBP4 85 45 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969354 GD On-Demand Anodyne EDNRA 27 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969354 GD On-Demand Anodyne BMP1 53 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969354 GD On-Demand Anodyne NOS2 95 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969354 GD On-Demand Anodyne MCHR1 15 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969357 GD On-Demand Anodyne EDNRA 27 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969357 GD On-Demand Anodyne BMP1 53 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969357 GD On-Demand Anodyne NOS2 95 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969357 GD On-Demand Anodyne MCHR1 15 40 O=C(Nc1cnccc1C(F)(F)F)N(Cc1cccc([N+](=O)[O-])c1)C1CC1 ZINC000880969365 GI On-Demand Bother CACNA1D 49 36 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ncccc2Cl)C1 ZINC000880969367 GH On-Demand Anodyne TRPV1 48 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ncccc2Cl)C1 ZINC000880969367 GH On-Demand Anodyne EPHX2 34 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ncccc2Cl)C1 ZINC000880969369 GH On-Demand Anodyne TRPV1 48 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ncccc2Cl)C1 ZINC000880969369 GH On-Demand Anodyne EPHX2 34 40 O=C(NCC1(C2CC2)CC1)Nc1cnccc1C(F)(F)F ZINC000880969374 CG On-Demand Anodyne TRPV1 21 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccn2)CC1 ZINC000880969377 FH On-Demand Anodyne TRPV1 23 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccn2)CC1 ZINC000880969377 FH On-Demand Anodyne EPHX2 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccn2)CC1 ZINC000880969377 FH On-Demand Anodyne RBP4 105 50 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccn2)CC1 ZINC000880969377 FH On-Demand Anodyne SFRP1 53 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccn2)CC1 ZINC000880969377 FH On-Demand Anodyne SMO 22 49 O=C(NCC1CCS(=O)(=O)CC1)Nc1cnccc1C(F)(F)F ZINC000880969379 FE On-Demand Anodyne TRPV1 16 44 CC(=O)N1CCN([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]2C)CC1 ZINC000880969384 GE On-Demand Anodyne RBP4 66 44 CS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969385 FE On-Demand Anodyne TRPV1 18 44 CS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969385 FE On-Demand Anodyne RBP4 75 45 CS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969385 FE On-Demand Anodyne SFRP1 82 36 CS(=O)(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969385 FE On-Demand Anodyne WNT3 69 33 CC(=O)N1CCN([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@@H]2C)CC1 ZINC000880969386 GE On-Demand Anodyne RBP4 66 44 CC(=O)N1CCN([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]2C)CC1 ZINC000880969388 GE On-Demand Anodyne RBP4 66 44 CC(=O)N1CCN([C@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)C[C@H]2C)CC1 ZINC000880969390 GE On-Demand Anodyne RBP4 66 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)c1ccc(C(F)(F)F)cc1 ZINC000880969391 GH On-Demand Anodyne TRPV1 21 53 CCc1nc([C@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)no1 ZINC000880969392 FG On-Demand Anodyne CPT1A 38 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)c1ccc(C(F)(F)F)cc1 ZINC000880969393 GH On-Demand Anodyne TRPV1 21 53 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)c1cccc(F)c1 ZINC000880969396 FG On-Demand Anodyne TRPV1 20 52 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)c1cccc(F)c1 ZINC000880969400 FG On-Demand Anodyne TRPV1 20 52 O=C(NCCOC1CCC1)Nc1cnccc1C(F)(F)F ZINC000880969422 DF On-Demand Anodyne TRPV1 20 45 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@@H]2CCCC[C@@H]2O)CC1 ZINC000880969423 GF On-Demand Anodyne EPHX2 45 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@H]2CCCC[C@@H]2O)CC1 ZINC000880969425 GF On-Demand Anodyne EPHX2 45 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@@H]2CCCC[C@H]2O)CC1 ZINC000880969426 GF On-Demand Anodyne EPHX2 45 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN([C@H]2CCCC[C@H]2O)CC1 ZINC000880969428 GF On-Demand Anodyne EPHX2 45 47 CCN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969430 DF On-Demand Anodyne TRPV1 21 40 CCN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969430 DF On-Demand Anodyne CCR2 17 41 CCN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969430 DF On-Demand Anodyne EPHX2 40 43 CCN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969430 DF On-Demand Anodyne BIRC2 29 41 CCN1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969431 DF On-Demand Anodyne TRPV1 21 40 CCN1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969431 DF On-Demand Anodyne CCR2 17 41 CCN1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969431 DF On-Demand Anodyne EPHX2 40 43 CCN1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969431 DF On-Demand Anodyne BIRC2 29 41 Cn1ncc(NC(=O)Nc2cnccc2C(F)(F)F)c1C(F)F ZINC000880969435 EG On-Demand Anodyne TRPV1 16 41 Cc1nc(CCNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880969443 EG On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCc2c[nH]nc21 ZINC000880969445 EG On-Demand Anodyne TRPV1 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCc2c[nH]nc21 ZINC000880969447 EG On-Demand Anodyne TRPV1 22 40 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne DRD4 38 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne ACHE 34 43 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne LTA4H 17 46 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne SIGMAR1 35 47 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne CCR5 29 44 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne RBP4 64 39 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne MCHR1 45 39 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(Cc2ccccc2)C1 ZINC000880969451 GH On-Demand Anodyne CACNA1G 27 41 CCC1(CC)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969452 DI On-Demand Anodyne RBP4 56 40 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne DRD4 38 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne ACHE 34 43 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne LTA4H 17 46 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne SIGMAR1 35 47 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne CCR5 29 44 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne RBP4 64 39 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne MCHR1 45 39 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880969453 GH On-Demand Anodyne CACNA1G 27 41 CCCN(C)C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969454 EG On-Demand Anodyne RBP4 59 42 CCCN(C)C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969456 EG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccco2)C1 ZINC000880969460 EG On-Demand Anodyne RBP4 65 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccco2)C1 ZINC000880969462 EG On-Demand Anodyne RBP4 65 42 O=C(Cn1cc([C@@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969464 EC On-Demand Anodyne NOS2 102 42 O=C(Cn1cc([C@@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969464 EC On-Demand Anodyne MCHR1 23 44 O=C(Cn1cc([C@@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969464 EC On-Demand Anodyne LUXR 26 43 O=C(Cn1cc([C@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969466 EC On-Demand Anodyne NOS2 102 42 O=C(Cn1cc([C@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969466 EC On-Demand Anodyne MCHR1 23 44 O=C(Cn1cc([C@H]2CCOC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969466 EC On-Demand Anodyne LUXR 26 43 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(F)c(F)c2C1 ZINC000880969470 FH On-Demand Anodyne RBP4 56 40 C[C@@H]1[C@@H](NC(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)CCC[C@H]1C ZINC000880969473 GF On-Demand Anodyne PREP 24 43 C[C@@H]1[C@@H](NC(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)CCC[C@H]1C ZINC000880969473 GF On-Demand Anodyne CAPN2 40 33 C[C@@H]1[C@@H](NC(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)CCC[C@H]1C ZINC000880969473 GF On-Demand Anodyne NPR 52 32 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880969475 GF On-Demand Anodyne PREP 24 43 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880969475 GF On-Demand Anodyne CAPN2 40 33 C[C@H]1[C@H](C)CCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880969475 GF On-Demand Anodyne NPR 52 32 O=C(Nc1cnccc1C(F)(F)F)N1CCS(=O)(=O)C2(CCCCC2)C1 ZINC000880969482 GG On-Demand Anodyne RBP4 48 38 CCC(CC)(CCO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969483 EG On-Demand Anodyne TRPV1 15 44 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880969486 EG On-Demand Anodyne HTR3A 33 42 CN1[C@H]2CCC[C@H]1CC(NC(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880969486 EG On-Demand Anodyne EPHX2 36 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(N2CCCCC2)CC1 ZINC000880969487 FI On-Demand Anodyne EPHX2 45 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(N2CCCCC2)CC1 ZINC000880969487 FI On-Demand Anodyne L3MBTL3 52 35 CC[C@@H](C)c1ccc(NC(=O)Cn2cc([C@H](C)N)nn2)cc1 ZINC000880969488 DE On-Demand Anodyne SCN2A 20 44 CC[C@@H](C)c1ccc(NC(=O)Cn2cc([C@@H](C)N)nn2)cc1 ZINC000880969491 DE On-Demand Anodyne SCN2A 20 44 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969492 EE On-Demand Anodyne RBP4 54 39 COC(=O)C[C@@H](C)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969494 FE On-Demand Anodyne RBP4 43 41 CCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969509 DF On-Demand Anodyne TRPV1 17 42 CCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969509 DF On-Demand Anodyne S1PR2 26 41 CCC1(O)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969509 DF On-Demand Anodyne RBP4 57 41 CO[C@@H](C)c1nc(CNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880969511 FH On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C2CCCC2)CC1 ZINC000880969512 FH On-Demand Anodyne EPHX2 47 48 O=C(NC[C@]1(O)CCSC1)Nc1cnccc1C(F)(F)F ZINC000880969516 DE On-Demand Anodyne TRPV1 17 45 O=C(NC[C@@]1(O)CCSC1)Nc1cnccc1C(F)(F)F ZINC000880969518 DE On-Demand Anodyne TRPV1 17 45 Cc1ccccc1[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969530 EG On-Demand Anodyne TRPV1 16 47 Cc1ccccc1[C@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969530 EG On-Demand Anodyne CTSA 47 32 Cc1ccccc1[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969532 EG On-Demand Anodyne TRPV1 16 47 Cc1ccccc1[C@@H](CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969532 EG On-Demand Anodyne CTSA 47 32 CC[C@@H](C)c1ccc(NC(=O)Cn2cc(CN3CCN(C(C)=O)CC3)nn2)cc1 ZINC000880969535 GE On-Demand Anodyne SCN2A 15 40 O=C(NCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1)c1ccc(O)cc1 ZINC000880969536 FD On-Demand Anodyne SIGMAR1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2CCC[C@@H]21 ZINC000880969537 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]2CCC[C@H]21 ZINC000880969538 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]2CCC[C@@H]21 ZINC000880969540 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]2CCC[C@H]21 ZINC000880969541 DH On-Demand Anodyne RBP4 56 41 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969543 FC On-Demand Anodyne NOS2 103 38 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969543 FC On-Demand Anodyne MCHR1 20 43 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969543 FC On-Demand Anodyne LUXR 15 43 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCC1CCCCC1 ZINC000880969549 EE On-Demand Anodyne REN 75 36 O=C(NC[C@H]1CCCS1)Nc1cnccc1C(F)(F)F ZINC000880969550 DG On-Demand Anodyne TRPV1 15 43 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCC1CCCCC1 ZINC000880969552 EE On-Demand Anodyne REN 75 36 COCC(C)(C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969554 CF On-Demand Anodyne TRPV1 18 46 O=C(Nc1cnccc1C(F)(F)F)N(CCCO)Cc1cccc(Cl)c1 ZINC000880969555 GI On-Demand Anodyne TRPV1 15 41 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969556 CF On-Demand Anodyne TRPV1 20 44 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969556 CF On-Demand Anodyne EPHX2 18 44 C[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969556 CF On-Demand Anodyne RBP4 87 48 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969557 CF On-Demand Anodyne TRPV1 20 44 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969557 CF On-Demand Anodyne EPHX2 18 44 C[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969557 CF On-Demand Anodyne RBP4 87 48 CCC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969558 DI On-Demand Anodyne RBP4 73 44 CCC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969559 DI On-Demand Anodyne RBP4 73 44 O=C(Nc1cnccc1C(F)(F)F)NC1(C2CC2)CC1 ZINC000880969561 CG On-Demand Anodyne TRPV1 18 42 CNc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880969562 EF On-Demand Anodyne TRPV1 20 49 CNc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880969562 EF On-Demand Anodyne ROCK1 17 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(O)(C(F)(F)F)CC1 ZINC000880969568 FG On-Demand Anodyne RBP4 59 42 Cn1c(S)nnc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969582 ED On-Demand Anodyne TRPV1 17 47 CCC(CC)(CNC(=O)Nc1cnccc1C(F)(F)F)C(=O)OC ZINC000880969584 EG On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC[C@H]1CO ZINC000880969587 DF On-Demand Anodyne TRPV1 22 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC[C@@H]1CO ZINC000880969588 DF On-Demand Anodyne TRPV1 22 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCC[C@@H]1CO ZINC000880969589 DF On-Demand Anodyne TRPV1 22 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCC[C@H]1CO ZINC000880969590 DF On-Demand Anodyne TRPV1 22 42 O=C1CCC(c2cn(CC(=O)Nc3ccc4ccccc4c3)nn2)CC1 ZINC000880969592 EG On-Demand Anodyne IMDH_CRYPV 35 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880969595 GI On-Demand Anodyne GRIN2B 43 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880969595 GI On-Demand Anodyne CCR3 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880969595 GI On-Demand Anodyne RBP4 93 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](COCc2ccccc2)C1 ZINC000880969595 GI On-Demand Anodyne SFRP1 47 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880969597 GI On-Demand Anodyne GRIN2B 43 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880969597 GI On-Demand Anodyne CCR3 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880969597 GI On-Demand Anodyne RBP4 93 47 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](COCc2ccccc2)C1 ZINC000880969597 GI On-Demand Anodyne SFRP1 47 33 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc2ccccc2c1 ZINC000880969598 FE On-Demand Anodyne IMDH_CRYPV 22 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCCC2)C1 ZINC000880969599 EI On-Demand Anodyne EPHX2 33 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCCCC2)C1 ZINC000880969599 EI On-Demand Anodyne RBP4 56 41 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)(N2CCCCC2)CC1 ZINC000880969601 GG On-Demand Anodyne HCN1 58 38 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)(N2CCCCC2)CC1 ZINC000880969601 GG On-Demand Anodyne HCN4 48 31 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CCC[C@H]21 ZINC000880969605 CG On-Demand Anodyne RBP4 59 42 Cc1cnc(CN(C)[C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)o1 ZINC000880969606 GG On-Demand Anodyne RBP4 56 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CCC[C@@H]21 ZINC000880969607 CG On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1C[C@@H]2CCC[C@@H]21 ZINC000880969608 CG On-Demand Anodyne RBP4 59 42 Cc1cnc(CN(C)[C@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)o1 ZINC000880969609 GG On-Demand Anodyne RBP4 56 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CCC[C@H]21 ZINC000880969610 CG On-Demand Anodyne RBP4 59 42 COC(=O)C[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969611 EF On-Demand Anodyne RBP4 44 39 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969613 EF On-Demand Anodyne RBP4 44 39 CCn1nc2c(cc1=O)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880969614 FE On-Demand Anodyne P2RY14 49 36 COCCNCCc1cn(CC(=O)Nc2ccc3ccccc3c2)nn1 ZINC000880969615 FD On-Demand Anodyne IMDH_CRYPV 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCCC2(C1)OCCO2 ZINC000880969617 EE On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c[nH]nc2C1 ZINC000880969618 DE On-Demand Anodyne RBP4 46 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC12CCCCC2 ZINC000880969619 EI On-Demand Anodyne RBP4 40 38 O=C(Nc1cnn(CCO)c1)Nc1cnccc1C(F)(F)F ZINC000880969640 DD On-Demand Anodyne TRPV1 16 42 COc1cc(NCCNC(=O)Nc2cnccc2C(F)(F)F)cc(OC)c1 ZINC000880969644 GG On-Demand Anodyne TRPV1 23 42 COc1cc(NCCNC(=O)Nc2cnccc2C(F)(F)F)cc(OC)c1 ZINC000880969644 GG On-Demand Anodyne RAF1 48 39 C[C@@H](CO)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969653 DF On-Demand Anodyne TRPV1 15 44 C[C@H](CO)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969654 DF On-Demand Anodyne TRPV1 15 44 CC[C@]1(C)CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969666 DH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H]1c1cccc(F)c1 ZINC000880969672 EI On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H]1c1cccc(F)c1 ZINC000880969673 EI On-Demand Anodyne RBP4 48 38 CC[C@H]1CN(C(=O)C2CC2)CC[C@@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969675 GG On-Demand Anodyne EPHX2 29 42 CC[C@H]1CN(C(=O)C2CC2)CC[C@H]1NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969677 GG On-Demand Anodyne EPHX2 29 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCCN2CCCC2)CC1 ZINC000880969681 GI On-Demand Anodyne CCR3 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCCN2CCCC2)CC1 ZINC000880969681 GI On-Demand Anodyne RBP4 65 40 CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)C1 ZINC000880969686 EE On-Demand Anodyne TRPV1 15 45 CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](C)C1 ZINC000880969686 EE On-Demand Anodyne RBP4 63 42 CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](C)C1 ZINC000880969687 EE On-Demand Anodyne TRPV1 15 45 CC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](C)C1 ZINC000880969687 EE On-Demand Anodyne RBP4 63 42 CNC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969689 CE On-Demand Anodyne TRPV1 23 47 CC(=O)OC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969690 EF On-Demand Anodyne EPHX2 22 41 CC(=O)OC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969690 EF On-Demand Anodyne RBP4 70 43 CC[C@@H](O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969691 CE On-Demand Anodyne TRPV1 17 46 CC[C@H](O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880969692 CE On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)NC1(CO)CC1 ZINC000880969693 CD On-Demand Anodyne TRPV1 18 45 CCOC(=O)CC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969696 FH On-Demand Anodyne RBP4 54 38 CCOC(=O)CC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969697 FH On-Demand Anodyne RBP4 54 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](Cn2ccnn2)C1 ZINC000880969698 FF On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](Cn2ccnn2)C1 ZINC000880969699 FF On-Demand Anodyne RBP4 55 39 O=C(NCc1ccco1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969700 GG On-Demand Anodyne WNT3 42 35 O=C(NCc1ccco1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969701 GG On-Demand Anodyne WNT3 42 35 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880969702 GG On-Demand Clean TRPV1 20 46 COc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880969702 GG On-Demand Clean RBP4 56 46 O=C(NCC1(C2CC2)CCC1)Nc1cnccc1C(F)(F)F ZINC000880969705 DH On-Demand Anodyne TRPV1 19 46 Cn1ccnc1[C@H](O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969709 GF On-Demand Anodyne RBP4 54 38 Cn1ccnc1[C@@H](O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969710 GF On-Demand Anodyne RBP4 54 38 Cn1ccnc1[C@@H](O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969711 GF On-Demand Anodyne RBP4 54 38 Cn1ccnc1[C@H](O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880969712 GF On-Demand Anodyne RBP4 54 38 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)cc1 ZINC000880969714 FG On-Demand Anodyne TRPV1 23 44 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1ccc2ccccc2c1 ZINC000880969722 FF On-Demand Anodyne IMDH_CRYPV 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2[C@@H]1CO ZINC000880969723 FG On-Demand Anodyne RBP4 78 43 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2[C@@H]1CO ZINC000880969723 FG On-Demand Anodyne TRPM8 46 51 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2[C@H]1CO ZINC000880969724 FG On-Demand Anodyne RBP4 78 43 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2[C@H]1CO ZINC000880969724 FG On-Demand Anodyne TRPM8 46 51 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)C(F)(F)F)CC1 ZINC000880969725 FG On-Demand Anodyne RBP4 72 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)C(F)(F)F)CC1 ZINC000880969726 FG On-Demand Anodyne RBP4 72 43 C[C@@H](CNc1ccccc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969730 EH On-Demand Anodyne TRPV1 22 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne TRPV1 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne EPHX2 28 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne RBP4 75 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne SCD1 61 60 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne SFRP1 51 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Oc2ccccc2Cl)CC1 ZINC000880969731 GJ On-Demand Anodyne SCD 44 48 CN(C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1)c1cccnn1 ZINC000880969732 GE On-Demand Anodyne RBP4 53 38 CC[C@@H]1C[C@@H](C)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969799 DH On-Demand Anodyne RBP4 47 39 CC[C@H]1C[C@H](C)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880969800 DH On-Demand Anodyne RBP4 47 39 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N1CCOCC1 ZINC000880969803 FE On-Demand Anodyne RBP4 65 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N1CCOCC1 ZINC000880969804 FE On-Demand Anodyne RBP4 65 44 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1N1CCOCC1 ZINC000880969805 FE On-Demand Anodyne RBP4 65 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1N1CCOCC1 ZINC000880969806 FE On-Demand Anodyne RBP4 65 44 O=C(Cn1c(=O)nc(O)c2ccccc21)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880969807 GD On-Demand Anodyne FABI 47 35 O=C(NCCc1nc(C(F)(F)F)cs1)Nc1cnccc1C(F)(F)F ZINC000880969808 GH On-Demand Anodyne TRPV1 16 48 CC[C@@](C)(CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969827 CE On-Demand Anodyne TRPV1 16 45 N#CCCN(CCN1CCOCC1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969828 FE On-Demand Mild CASR 59 47 O=C(NCCC1CCN(CC(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880969835 GH On-Demand Anodyne TRPV1 15 42 O=C(NCCC1CCN(CC(F)(F)F)CC1)Nc1cnccc1C(F)(F)F ZINC000880969835 GH On-Demand Anodyne CCR3 31 48 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H]([C@H]2CCCO2)C1 ZINC000880969839 EF On-Demand Anodyne RBP4 70 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H]([C@H]2CCCO2)C1 ZINC000880969840 EF On-Demand Anodyne RBP4 70 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H]([C@@H]2CCCO2)C1 ZINC000880969841 EF On-Demand Anodyne RBP4 70 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H]([C@@H]2CCCO2)C1 ZINC000880969842 EF On-Demand Anodyne RBP4 70 42 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969845 FD On-Demand Anodyne NOS2 98 39 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969846 FD On-Demand Anodyne NOS2 98 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCOC2)C1 ZINC000880969847 DF On-Demand Anodyne EPHX2 33 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@]2(CCOC2)C1 ZINC000880969847 DF On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCOC2)C1 ZINC000880969848 DF On-Demand Anodyne EPHX2 33 40 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@]2(CCOC2)C1 ZINC000880969848 DF On-Demand Anodyne RBP4 54 39 CS(=O)(=O)CC1(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969849 FE On-Demand Anodyne TRPV1 17 45 O=C(NCC1(CO)CC1)Nc1cnccc1C(F)(F)F ZINC000880969850 CD On-Demand Anodyne TRPV1 21 49 O=C(NC[C@H](CO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880969852 EF On-Demand Anodyne TRPV1 23 54 O=C(NC[C@H](CO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880969852 EF On-Demand Anodyne SOAT1 15 41 O=C(NC[C@@H](CO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880969853 EF On-Demand Anodyne TRPV1 23 54 O=C(NC[C@@H](CO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880969853 EF On-Demand Anodyne SOAT1 15 41 C[S@@](=O)C[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969856 FG On-Demand Anodyne TRPV1 15 49 C[S@@](=O)C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969857 FG On-Demand Anodyne TRPV1 15 49 C[S@](=O)C[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969858 FG On-Demand Anodyne TRPV1 15 49 C[S@](=O)C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880969859 FG On-Demand Anodyne TRPV1 15 49 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)N1CCS(=O)CC1 ZINC000880969860 GE On-Demand Anodyne TRPV1 15 42 C[C@@H](Cc1ccncc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969861 DG On-Demand Anodyne TRPV1 19 47 C[C@@H](Cc1ccncc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969861 DG On-Demand Anodyne FLT1 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ncc[nH]2)CC1 ZINC000880969868 EG On-Demand Anodyne RBP4 74 44 O=C1CC2(CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)CN1 ZINC000880969874 EE On-Demand Anodyne RBP4 54 39 O=C(Cn1cc(CCCCCCO)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969876 FD On-Demand Anodyne NOS2 101 37 CCC(CC)c1cc(CNC(=O)Nc2cnccc2C(F)(F)F)on1 ZINC000880969877 FI On-Demand Anodyne TRPV1 19 47 CN(CCOCc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880969878 FH On-Demand Anodyne RBP4 17 47 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CCCC[C@@H]1O ZINC000880969884 EG On-Demand Anodyne TRPV1 17 43 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CCCC[C@H]1O ZINC000880969885 EG On-Demand Anodyne TRPV1 17 43 CNC(=O)[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969887 CD On-Demand Anodyne TRPV1 21 48 O=C(Nc1cnccc1C(F)(F)F)NC(CO)CO ZINC000880969890 CC On-Demand Anodyne TRPV1 21 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nccs2)CC1 ZINC000880969891 FH On-Demand Anodyne RBP4 75 45 Cn1cc([C@@H]2CN(C(=O)Nc3cnccc3C(F)(F)F)CCO2)cn1 ZINC000880969895 FE On-Demand Anodyne RBP4 56 40 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)NC(=O)OC(C)(C)C ZINC000880969901 GH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H]2CCOC2)CC1 ZINC000880969908 FE On-Demand Anodyne CCR2 23 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H]2CCOC2)CC1 ZINC000880969908 FE On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H]2CCOC2)CC1 ZINC000880969909 FE On-Demand Anodyne CCR2 23 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H]2CCOC2)CC1 ZINC000880969909 FE On-Demand Anodyne RBP4 54 39 C[C@H](N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C(F)(F)F ZINC000880969911 FG On-Demand Anodyne TRPV1 16 44 C[C@H](N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C(F)(F)F ZINC000880969911 FG On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880969912 GH On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880969912 GH On-Demand Anodyne SMO 33 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2noc(C3CC3)n2)C1 ZINC000880969912 GH On-Demand Anodyne ETHR 59 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880969913 GH On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880969913 GH On-Demand Anodyne SMO 33 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2noc(C3CC3)n2)C1 ZINC000880969913 GH On-Demand Anodyne ETHR 59 43 O=C(Cn1cc(C2(O)CCCCC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880969914 FD On-Demand Anodyne NOS2 95 37 O=C(NCc1nncn1C1CC1)Nc1cnccc1C(F)(F)F ZINC000880969915 EE On-Demand Anodyne TRPV1 16 45 O=C(NCC(C1CC1)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880969922 DH On-Demand Anodyne TRPV1 22 46 C[C@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969924 GE On-Demand Anodyne TRPV1 15 42 C[C@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969924 GE On-Demand Anodyne RBP4 54 39 C[C@@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969925 GE On-Demand Anodyne TRPV1 15 42 C[C@@H](C(=O)N1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969925 GE On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCOCC1 ZINC000880969926 CE On-Demand Anodyne RBP4 58 42 CNC(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969927 EE On-Demand Anodyne RBP4 73 41 NC(=O)NCCCCCC(=O)N1CC2(CN(Cc3ccccc3)C2)C1 ZINC000880969944 ED On-Demand Anodyne NPFFR1 43 38 CCCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969951 EG On-Demand Anodyne CCR3 25 42 CCCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969951 EG On-Demand Anodyne EPHX2 51 45 CCCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969951 EG On-Demand Anodyne CXCR3 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCC2)C1 ZINC000880969952 EG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCC2)C1 ZINC000880969952 EG On-Demand Anodyne SFRP1 87 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CN2CCCC2)C1 ZINC000880969952 EG On-Demand Anodyne WNT3 73 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCC2)C1 ZINC000880969953 EG On-Demand Anodyne RBP4 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCC2)C1 ZINC000880969953 EG On-Demand Anodyne SFRP1 87 35 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CN2CCCC2)C1 ZINC000880969953 EG On-Demand Anodyne WNT3 73 35 O=C(NCc1nnnn1C1CC1)Nc1cnccc1C(F)(F)F ZINC000880969954 ED On-Demand Anodyne TRPV1 15 45 C[C@@H](CCCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969956 CE On-Demand Anodyne TRPV1 16 45 Cc1cnc(CNC(=O)Nc2cnccc2C(F)(F)F)s1 ZINC000880969957 DG On-Demand Anodyne TRPV1 20 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](n2cncn2)C1 ZINC000880969964 EF On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](n2cncn2)C1 ZINC000880969965 EF On-Demand Anodyne RBP4 61 42 O=C(NC[C@H]1CCC[C@H]1O)Nc1cnccc1C(F)(F)F ZINC000880969967 DE On-Demand Anodyne TRPV1 19 44 CN(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969971 GI On-Demand Anodyne TRPV1 23 44 CN(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969971 GI On-Demand Anodyne RBP4 100 48 CN(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969971 GI On-Demand Anodyne SFRP1 121 38 CN(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969971 GI On-Demand Anodyne SMO 18 44 CN(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880969971 GI On-Demand Anodyne WNT3 85 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCOCC2)C1 ZINC000880969972 EG On-Demand Anodyne EPHX2 36 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(CCOCC2)C1 ZINC000880969972 EG On-Demand Anodyne RBP4 55 39 CCC(CC)(CO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880969998 DF On-Demand Anodyne TRPV1 17 43 CC[C@H](O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970001 DC On-Demand Anodyne EDNRB 30 40 CC[C@H](O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970001 DC On-Demand Anodyne EDNRA 27 40 CC[C@H](O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970001 DC On-Demand Anodyne BMP1 55 36 CC[C@H](O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970001 DC On-Demand Anodyne NOS2 99 39 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970004 GD On-Demand Anodyne BMP1 52 41 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970004 GD On-Demand Anodyne NOS2 95 40 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970004 GD On-Demand Anodyne MCHR1 16 40 CCC(CC)(CNC(=O)Nc1cnccc1C(F)(F)F)SC ZINC000880970008 EI On-Demand Anodyne TRPV1 17 46 COC(=O)C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880970016 ED On-Demand Anodyne RBP4 61 43 COC(=O)C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880970017 ED On-Demand Anodyne RBP4 61 43 Cc1cc(F)ccc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970018 EH On-Demand Anodyne TRPV1 26 45 Cc1cc(F)ccc1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970018 EH On-Demand Anodyne RAF1 25 40 Cc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)sc1C ZINC000880970023 EG On-Demand Anodyne TRPV1 22 50 Cn1nc2c(c1-c1cn(CC(=O)NCc3ccc4c(c3)OCO4)nn1)CCCC2 ZINC000880970024 GD On-Demand Anodyne NOS2 95 37 CCOC(=O)[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970030 DE On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CCC[C@H]1CC2 ZINC000880970033 CH On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@H]1c1ccccc1 ZINC000880970044 FH On-Demand Anodyne RBP4 60 42 O=C(Nc1cnccc1C(F)(F)F)N1CCOC[C@@H]1c1ccccc1 ZINC000880970045 FH On-Demand Anodyne RBP4 60 42 CCC1(NC(=O)Nc2cnccc2C(F)(F)F)CCC1 ZINC000880970048 CH On-Demand Anodyne TRPV1 16 43 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@@H](O)c1c(F)cccc1Cl ZINC000880970051 GI On-Demand Anodyne TRPV1 19 48 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)[C@H](O)c1c(F)cccc1Cl ZINC000880970052 GI On-Demand Anodyne TRPV1 19 48 CC[C@@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970065 EE On-Demand Anodyne RBP4 54 39 CC[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970066 EE On-Demand Anodyne RBP4 54 39 N#C[C@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970076 FI On-Demand Mild PTAFR 17 40 N#C[C@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970076 FI On-Demand Mild RBP4 60 39 N#C[C@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970076 FI On-Demand Mild SFRP1 42 34 N#C[C@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970076 FI On-Demand Mild WNT3 41 34 N#C[C@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970077 FI On-Demand Mild PTAFR 17 40 N#C[C@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970077 FI On-Demand Mild RBP4 60 39 N#C[C@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970077 FI On-Demand Mild SFRP1 42 34 N#C[C@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970077 FI On-Demand Mild WNT3 41 34 N#C[C@@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970078 FI On-Demand Mild PTAFR 17 40 N#C[C@@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970078 FI On-Demand Mild RBP4 60 39 N#C[C@@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970078 FI On-Demand Mild SFRP1 42 34 N#C[C@@H](c1ccccc1)[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970078 FI On-Demand Mild WNT3 41 34 N#C[C@@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970079 FI On-Demand Mild PTAFR 17 40 N#C[C@@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970079 FI On-Demand Mild RBP4 60 39 N#C[C@@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970079 FI On-Demand Mild SFRP1 42 34 N#C[C@@H](c1ccccc1)[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970079 FI On-Demand Mild WNT3 41 34 COc1ccccc1C[C@@H](C)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970084 FI On-Demand Anodyne TRPV1 17 42 COc1ccccc1C[C@@H](C)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970084 FI On-Demand Anodyne NPY5R 21 42 COc1ccccc1C[C@H](C)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970085 FI On-Demand Anodyne TRPV1 17 42 COc1ccccc1C[C@H](C)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970085 FI On-Demand Anodyne NPY5R 21 42 CSC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970091 DG On-Demand Anodyne TRPV1 20 47 CS[C@@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970093 DH On-Demand Anodyne EPHX2 29 41 CS[C@H]1CC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970094 DH On-Demand Anodyne EPHX2 29 41 O=C(NCC(=O)OC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970096 EG On-Demand Anodyne TRPV1 18 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccs2)CC1 ZINC000880970097 FH On-Demand Anodyne TRPV1 18 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccs2)CC1 ZINC000880970097 FH On-Demand Anodyne RBP4 62 41 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970104 GI On-Demand Anodyne ABL1 45 38 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970104 GI On-Demand Anodyne TRPV1 22 40 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970104 GI On-Demand Anodyne ABL2 45 38 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970104 GI On-Demand Anodyne RBP4 58 39 CN1CCC(N(Cc2ccccc2)C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970104 GI On-Demand Anodyne SFRP1 40 32 C[C@@](CO)(NC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880970115 DE On-Demand Anodyne TRPV1 19 43 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970117 EC On-Demand Anodyne NOS2 97 38 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc3c(c2)OCO3)nn1 ZINC000880970117 EC On-Demand Anodyne MCHR1 18 41 CC[C@H]1CN(C(C)=O)[C@H](CC)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970125 FG On-Demand Anodyne RBP4 40 38 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](CC)CN1C(C)=O ZINC000880970126 FG On-Demand Anodyne RBP4 40 38 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](CC)CN1C(C)=O ZINC000880970127 FG On-Demand Anodyne RBP4 40 38 O=C(Nc1cnccc1C(F)(F)F)N(CCO)[C@H]1CCc2ccccc21 ZINC000880970128 FH On-Demand Anodyne TRPM8 20 42 O=C(Nc1cnccc1C(F)(F)F)N(CCO)[C@@H]1CCc2ccccc21 ZINC000880970129 FH On-Demand Anodyne TRPM8 20 42 O=C(Cn1cc([C@@H](O)C2CC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880970130 EC On-Demand Anodyne NOS2 101 39 O=C(Cn1cc([C@@H](O)C2CC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880970130 EC On-Demand Anodyne MCHR1 21 41 O=C(Cn1cc([C@H](O)C2CC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880970131 EC On-Demand Anodyne NOS2 101 39 O=C(Cn1cc([C@H](O)C2CC2)nn1)NCc1ccc2c(c1)OCO2 ZINC000880970131 EC On-Demand Anodyne MCHR1 21 41 C[C@H](CCO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970132 CE On-Demand Anodyne TRPV1 17 45 C[C@@H](CCO)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970133 CE On-Demand Anodyne TRPV1 17 45 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880970137 CG On-Demand Anodyne TRPV1 19 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880970137 CG On-Demand Anodyne RBP4 85 49 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880970138 CG On-Demand Anodyne TRPV1 19 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H]1C ZINC000880970138 CG On-Demand Anodyne RBP4 85 49 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880970139 CG On-Demand Anodyne TRPV1 19 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H]1C ZINC000880970139 CG On-Demand Anodyne RBP4 85 49 CCC(C)(CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970140 CH On-Demand Anodyne TRPV1 23 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880970142 FG On-Demand Anodyne RBP4 66 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C(F)(F)F)O1 ZINC000880970143 FG On-Demand Anodyne RBP4 66 43 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880970144 FG On-Demand Anodyne RBP4 66 43 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C(F)(F)F)O1 ZINC000880970145 FG On-Demand Anodyne RBP4 66 43 O=C(Nc1cnccc1C(F)(F)F)N(CCO)CCN1CCOCC1 ZINC000880970154 FD On-Demand Anodyne CASR 62 49 CC(C)(C)OC(=O)NC[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970157 GH On-Demand Anodyne SFRP1 43 33 CC(C)(C)OC(=O)NC[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970157 GH On-Demand Anodyne WNT3 51 33 CC(C)(C)OC(=O)NC[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970158 GH On-Demand Anodyne SFRP1 43 33 CC(C)(C)OC(=O)NC[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970158 GH On-Demand Anodyne WNT3 51 33 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCOCC2)CC1 ZINC000880970160 FE On-Demand Anodyne CCR2 16 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCOCC2)CC1 ZINC000880970160 FE On-Demand Anodyne RBP4 65 41 O=C(NCCOCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970161 EG On-Demand Anodyne TRPV1 24 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cnc[nH]2)CC1 ZINC000880970164 EG On-Demand Anodyne RBP4 78 44 Cn1cc([C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)cn1 ZINC000880970171 EF On-Demand Anodyne RBP4 83 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nc3ccccc3o2)CC1 ZINC000880970172 GH On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nc3ccccc3o2)CC1 ZINC000880970172 GH On-Demand Anodyne FAAH 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nc3ccccc3o2)CC1 ZINC000880970172 GH On-Demand Anodyne SORD 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nc3ccccc3o2)CC1 ZINC000880970172 GH On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2nc3ccccc3o2)CC1 ZINC000880970172 GH On-Demand Anodyne DGAT1 20 42 CC(C)c1ccccc1NC(=O)Cn1cc(CCCCCCO)nn1 ZINC000880970176 EG On-Demand Anodyne SOAT1 21 42 O=C(NC[C@@H](CCO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970179 FG On-Demand Anodyne TRPV1 19 52 O=C(NC[C@H](CCO)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970180 FG On-Demand Anodyne TRPV1 19 52 O=C(NCCCCN1CCC[C@@H]1CO)Nc1cnccc1C(F)(F)F ZINC000880970182 FE On-Demand Anodyne CCR3 29 44 O=C(NCCCCN1CCC[C@H]1CO)Nc1cnccc1C(F)(F)F ZINC000880970183 FE On-Demand Anodyne CCR3 29 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H](O)c2ccccc2)CC1 ZINC000880970184 GF On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H](O)c2ccccc2)CC1 ZINC000880970184 GF On-Demand Anodyne FAAH 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H](O)c2ccccc2)CC1 ZINC000880970184 GF On-Demand Anodyne RBP4 83 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H](O)c2ccccc2)CC1 ZINC000880970185 GF On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H](O)c2ccccc2)CC1 ZINC000880970185 GF On-Demand Anodyne FAAH 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H](O)c2ccccc2)CC1 ZINC000880970185 GF On-Demand Anodyne RBP4 83 44 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](C)O1 ZINC000880970187 DG On-Demand Anodyne RBP4 58 42 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880970189 DG On-Demand Anodyne RBP4 58 42 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880970194 DE On-Demand Anodyne TRPV1 25 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880970199 FF On-Demand Anodyne RBP4 71 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880970199 FF On-Demand Anodyne SFRP1 74 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCCC2)C1 ZINC000880970199 FF On-Demand Anodyne WNT3 64 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880970200 FF On-Demand Anodyne RBP4 71 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880970200 FF On-Demand Anodyne SFRP1 74 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCCC2)C1 ZINC000880970200 FF On-Demand Anodyne WNT3 64 35 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880970202 EG On-Demand Anodyne TRPV1 28 50 CCN(CC)C(=O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970206 GE On-Demand Anodyne RBP4 55 40 CCOC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880970211 ED On-Demand Anodyne RBP4 57 40 CCC(CC)[C@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970216 DG On-Demand Anodyne TRPV1 15 45 CCC(CC)[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970217 DG On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)NC1(c2ccccc2F)CC1 ZINC000880970218 EI On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cncnc2C1 ZINC000880970227 DE On-Demand Anodyne MAPK1 45 38 O=C(Nc1cnccc1C(F)(F)F)N1CCc2cncnc2C1 ZINC000880970227 DE On-Demand Anodyne RBP4 54 39 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)Cc1cccs1 ZINC000880970230 EI On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880970231 GE On-Demand Anodyne ABL2 43 36 O=C(Nc1cnn(CCN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880970231 GE On-Demand Anodyne EPHX2 30 46 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970239 EI On-Demand Anodyne RBP4 55 39 C[C@H]1Cc2ccccc2CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970240 EI On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCCCC[C@H]1c1ccco1 ZINC000880970241 FJ On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCCC[C@@H]1c1ccco1 ZINC000880970242 FJ On-Demand Anodyne RBP4 53 38 CC[C@@H]1CCCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970243 DI On-Demand Anodyne WNT3 40 32 CC[C@H]1CCCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970244 DI On-Demand Anodyne WNT3 40 32 C[C@H]1C[C@H](NC(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880970248 DF On-Demand Anodyne SFRP1 49 34 C[C@H]1C[C@H](NC(=O)Nc2cnccc2C(F)(F)F)CCN1C ZINC000880970248 DF On-Demand Anodyne WNT3 40 34 CN1CCN(C)[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970253 ED On-Demand Anodyne TRPV1 15 41 CN1CCN(C)[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970254 ED On-Demand Anodyne TRPV1 15 41 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne TRPV1 20 42 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne P2RY1 57 43 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne RAF1 51 42 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne KDR 18 43 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne MTOR 50 35 O=C(Nc1ccc(OCC2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880970261 GJ On-Demand Anodyne EPHX2 43 43 C[C@H]1C[C@@H](C)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970263 CG On-Demand Anodyne RBP4 57 42 C[C@H]1C[C@@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970264 CG On-Demand Anodyne RBP4 57 42 COc1cc(C)nc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880970277 GF On-Demand Anodyne RBP4 43 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@@H]1Cc1ccccc1 ZINC000880970278 EH On-Demand Anodyne TRPV1 27 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@@H]1Cc1ccccc1 ZINC000880970279 EH On-Demand Anodyne TRPV1 27 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1C[C@H]1Cc1ccccc1 ZINC000880970280 EH On-Demand Anodyne TRPV1 27 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1C[C@H]1Cc1ccccc1 ZINC000880970281 EH On-Demand Anodyne TRPV1 27 49 CC(C)(C)C[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970284 DG On-Demand Anodyne TRPV1 17 45 CC(C)(C)C[C@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970285 DG On-Demand Anodyne TRPV1 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCn2cnnc2C1 ZINC000880970292 DD On-Demand Anodyne RBP4 55 39 O=C(NCc1nc(C(F)(F)F)cs1)Nc1cnccc1C(F)(F)F ZINC000880970293 FH On-Demand Anodyne TRPV1 23 51 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)c1cccs1 ZINC000880970295 EI On-Demand Anodyne TRPV1 21 47 COC(=O)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC(C)C ZINC000880970296 EG On-Demand Anodyne TRPV1 15 44 COC(=O)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CC(C)C ZINC000880970297 EG On-Demand Anodyne TRPV1 15 44 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970303 FG On-Demand Anodyne TRPV1 29 44 C[S@@](=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970308 DD On-Demand Anodyne TRPV1 16 47 CC[C@@H](C)[C@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970314 DG On-Demand Anodyne TRPV1 15 44 CC[C@@H](C)[C@@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970315 DG On-Demand Anodyne TRPV1 15 44 CC[C@H](C)[C@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970316 DG On-Demand Anodyne TRPV1 15 44 CC[C@H](C)[C@@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970317 DG On-Demand Anodyne TRPV1 15 44 NC(=O)c1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880970318 GF On-Demand Anodyne RBP4 54 39 O=C(NCC1(O)CCCC1)Nc1cnccc1C(F)(F)F ZINC000880970321 DF On-Demand Anodyne TRPV1 20 49 O=C(NCCCc1ccc(O)cc1)Nc1cnccc1C(F)(F)F ZINC000880970322 EH On-Demand Anodyne TRPV1 23 53 O=C(NCCCc1ccc(O)cc1)Nc1cnccc1C(F)(F)F ZINC000880970322 EH On-Demand Anodyne SLC6A5 16 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](c1ccccc1)C1CCOCC1 ZINC000880970327 GI On-Demand Anodyne TRPV1 15 56 O=C(Nc1cnccc1C(F)(F)F)N[C@H](c1ccccc1)C1CCOCC1 ZINC000880970328 GI On-Demand Anodyne TRPV1 15 56 CC[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCN1CCOC ZINC000880970332 FF On-Demand Anodyne RBP4 54 39 O=C(NCCOC1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970334 EH On-Demand Anodyne TRPV1 19 44 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970335 EF On-Demand Anodyne RBP4 64 43 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970335 EF On-Demand Anodyne SFRP1 74 36 COC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970335 EF On-Demand Anodyne WNT3 70 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(F)(F)F)(C(F)(F)F)C1 ZINC000880970340 GI On-Demand Mild RBP4 58 42 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970342 GI On-Demand Mild TRPV1 25 50 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970342 GI On-Demand Mild ROCK1 16 41 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970342 GI On-Demand Mild ROCK2 29 44 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970342 GI On-Demand Mild CARM1 41 34 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970342 GI On-Demand Mild PDS 62 36 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970343 GI On-Demand Mild TRPV1 25 50 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970343 GI On-Demand Mild ROCK1 16 41 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970343 GI On-Demand Mild ROCK2 29 44 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970343 GI On-Demand Mild CARM1 41 34 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970343 GI On-Demand Mild PDS 62 36 C[C@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970345 EJ On-Demand Anodyne TRPV1 15 40 C[C@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970345 EJ On-Demand Anodyne RBP4 89 48 C[C@@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970346 EJ On-Demand Anodyne TRPV1 15 40 C[C@@H]1C[C@H](c2ccccc2)CN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970346 EJ On-Demand Anodyne RBP4 89 48 CC[C@@H]1CN(CCn2cccn2)CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970356 GF On-Demand Anodyne ABL2 44 35 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970359 GG On-Demand Anodyne NPY5R 26 42 NC(=O)C1(c2ccccc2)CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970359 GG On-Demand Anodyne RBP4 66 46 NC(=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970364 CD On-Demand Anodyne TRPV1 26 54 O=C(Nc1ccc(NC[C@H]2CCCO2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880970365 GI On-Demand Anodyne TNK2 29 46 O=C(Nc1ccc(NC[C@@H]2CCCO2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880970366 GI On-Demand Anodyne TNK2 29 46 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCN(c2ccccc2)C1=O ZINC000880970369 GG On-Demand Anodyne RBP4 49 38 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCN(c2ccccc2)C1=O ZINC000880970370 GG On-Demand Anodyne RBP4 49 38 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCN(C)CC1 ZINC000880970372 FE On-Demand Anodyne ABL1 34 40 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCN(C)CC1 ZINC000880970372 FE On-Demand Anodyne TRPV1 15 40 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCN(C)CC1 ZINC000880970372 FE On-Demand Anodyne ABL2 38 40 COC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880970388 DF On-Demand Anodyne TRPV1 20 46 COC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880970389 DF On-Demand Anodyne TRPV1 20 46 O=C(NCCCNC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970391 EH On-Demand Anodyne TRPV1 20 47 O=C(NCC1Cc2ccccc2C1)Nc1cnccc1C(F)(F)F ZINC000880970407 EH On-Demand Anodyne TRPV1 26 49 O=C(NCCN1CCSCC1)Nc1cnccc1C(F)(F)F ZINC000880970410 EE On-Demand Anodyne UTS2R 16 40 CCN(CCNC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880970424 DF On-Demand Anodyne TRPV1 16 43 CC[C@H](CCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970429 CE On-Demand Anodyne TRPV1 15 48 CC[C@@H](CCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970430 CE On-Demand Anodyne TRPV1 15 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC2CCOCC2)CC1 ZINC000880970443 FF On-Demand Anodyne RBP4 58 40 O=C(NCCCC(=O)N1CCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970451 GH On-Demand Anodyne TRPV1 20 46 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccco1 ZINC000880970457 EF On-Demand Anodyne TRPV1 17 44 CCC[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970464 CE On-Demand Anodyne TRPV1 15 45 CCC[C@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970465 CE On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(nnc2C2CC2)C1 ZINC000880970468 FF On-Demand Anodyne P2RX7 26 41 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(nnc2C2CC2)C1 ZINC000880970468 FF On-Demand Anodyne RBP4 61 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccc(F)cc2)O1 ZINC000880970473 GI On-Demand Anodyne RBP4 58 41 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccc(F)cc2)O1 ZINC000880970474 GI On-Demand Anodyne RBP4 58 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccc(F)cc2)O1 ZINC000880970475 GI On-Demand Anodyne RBP4 58 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccc(F)cc2)O1 ZINC000880970476 GI On-Demand Anodyne RBP4 58 41 C=CC[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970479 CG On-Demand Mild TRPV1 15 47 C=CC[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970480 CG On-Demand Mild TRPV1 15 47 CC(=O)NC[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880970482 ED On-Demand Anodyne RBP4 60 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2cc[nH]n2)C1 ZINC000880970498 EG On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2cc[nH]n2)C1 ZINC000880970499 EG On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCS(=O)(=O)c2ccccc21 ZINC000880970500 GG On-Demand Anodyne TRPV1 26 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCS(=O)(=O)c2ccccc21 ZINC000880970500 GG On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCS(=O)(=O)c2ccccc21 ZINC000880970501 GG On-Demand Anodyne TRPV1 26 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCS(=O)(=O)c2ccccc21 ZINC000880970501 GG On-Demand Anodyne RBP4 58 42 Cc1ccccc1[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970507 EG On-Demand Anodyne TRPV1 21 48 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C2CCCC2)CC1 ZINC000880970509 FH On-Demand Anodyne HRH3 22 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C2CCCC2)CC1 ZINC000880970509 FH On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C2CCCC2)CC1 ZINC000880970509 FH On-Demand Anodyne L3MBTL3 45 35 C[C@H]1c2c(F)cccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970510 FI On-Demand Anodyne RBP4 45 37 C[C@H]1c2c(F)cccc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970510 FI On-Demand Anodyne TRPM8 47 46 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970522 GH On-Demand Anodyne RBP4 55 39 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970522 GH On-Demand Anodyne F13A1 23 41 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970522 GH On-Demand Anodyne GPR119 34 43 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](C(F)(F)F)C1 ZINC000880970525 EF On-Demand Anodyne RBP4 70 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](C(F)(F)F)C1 ZINC000880970526 EF On-Demand Anodyne RBP4 70 45 CCC[C@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970530 DF On-Demand Anodyne TRPV1 17 45 CC(C)(C)C(=O)NC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970532 GH On-Demand Anodyne RBP4 60 41 CC(C)(C)C(=O)NC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970533 GH On-Demand Anodyne RBP4 60 41 COCc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1F ZINC000880970534 FH On-Demand Anodyne TRPV1 29 51 COCc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1F ZINC000880970534 FH On-Demand Anodyne ROCK2 34 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCOCC2)CC1 ZINC000880970539 GE On-Demand Anodyne EPHX2 25 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCOCC2)CC1 ZINC000880970539 GE On-Demand Anodyne RBP4 70 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCOCC2)CC1 ZINC000880970539 GE On-Demand Anodyne SFRP1 49 36 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](Cn2cncn2)C1 ZINC000880970544 FD On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](Cn2cncn2)C1 ZINC000880970545 FD On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne TRPV1 17 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne EPHX2 20 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne RBP4 80 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne SFRP1 52 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne SCD 21 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCCc2ccccc2)CC1 ZINC000880970556 GI On-Demand Anodyne WNT3 40 32 O=C(NCC1(O)CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970557 EG On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cn1cccn1 ZINC000880970564 EF On-Demand Anodyne SFRP1 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cn1cccn1 ZINC000880970564 EF On-Demand Anodyne WNT3 49 34 O=C(Cn1cc(C(=O)c2ccc(C(F)(F)F)cc2)nn1)NC1CCCC1 ZINC000880970572 FF On-Demand Anodyne CCR2 41 36 O=C(Cn1cc(COc2ccc(Br)nc2)nn1)NC1CCCC1 ZINC000880970573 GE On-Demand Anodyne FIMH 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCC2)C1 ZINC000880970575 EF On-Demand Anodyne RBP4 72 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCC2)C1 ZINC000880970575 EF On-Demand Anodyne SFRP1 50 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCC2)C1 ZINC000880970575 EF On-Demand Anodyne L3MBTL3 89 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCC2)C1 ZINC000880970576 EF On-Demand Anodyne RBP4 72 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCC2)C1 ZINC000880970576 EF On-Demand Anodyne SFRP1 50 34 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCC2)C1 ZINC000880970576 EF On-Demand Anodyne L3MBTL3 89 43 O=C(NCc1ccc2c(c1)OCCCO2)Nc1cnccc1C(F)(F)F ZINC000880970577 FH On-Demand Anodyne TRPV1 24 52 O=C(NCc1ccc2c(c1)OCCCO2)Nc1cnccc1C(F)(F)F ZINC000880970577 FH On-Demand Anodyne NOS2 86 35 O=C(NCc1ccc2c(c1)OCCCO2)Nc1cnccc1C(F)(F)F ZINC000880970577 FH On-Demand Anodyne NAMPT 45 34 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)N1CCCC[C@H]1C ZINC000880970579 FG On-Demand Anodyne WNT3 40 33 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)N1CCCC[C@@H]1C ZINC000880970580 FG On-Demand Anodyne WNT3 40 33 C[C@H]1CCCCN1C(=O)[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970581 FG On-Demand Anodyne WNT3 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2nccs2)C1 ZINC000880970584 FG On-Demand Anodyne RBP4 59 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2nccs2)C1 ZINC000880970585 FG On-Demand Anodyne RBP4 59 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@H]2CCCO2)CC1 ZINC000880970586 FE On-Demand Anodyne RBP4 67 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C[C@@H]2CCCO2)CC1 ZINC000880970587 FE On-Demand Anodyne RBP4 67 40 O=C(CC1CCCC1)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970590 GH On-Demand Anodyne RBP4 59 40 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)c2ccsc2)CC1 ZINC000880970591 GH On-Demand Anodyne RBP4 54 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C2OCCO2)CC1 ZINC000880970598 EF On-Demand Anodyne RBP4 74 44 O=C(Cn1cc(CN2CCCC2)nn1)NC1CCCCCCC1 ZINC000880970602 DE On-Demand Anodyne SIGMAR1 15 47 O=C(Cn1cc(CN2CCCC2)nn1)NC1CCCCCCC1 ZINC000880970602 DE On-Demand Anodyne EPHX2 20 42 CN(C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)S(C)(=O)=O ZINC000880970603 GD On-Demand Anodyne RBP4 71 45 CN(C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)S(C)(=O)=O ZINC000880970603 GD On-Demand Anodyne SFRP1 77 35 CN(C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)S(C)(=O)=O ZINC000880970603 GD On-Demand Anodyne WNT3 64 34 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccccc2Cl)C1 ZINC000880970605 GI On-Demand Anodyne RBP4 93 48 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccccc2Cl)C1 ZINC000880970606 GI On-Demand Anodyne RBP4 93 48 CC(=O)N1CCN(C(=O)CCNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970611 GD On-Demand Anodyne TRPV1 27 48 CC[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970614 CH On-Demand Anodyne RBP4 46 38 CC[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970614 CH On-Demand Anodyne WNT3 41 33 CC[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970615 CH On-Demand Anodyne RBP4 46 38 CC[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880970615 CH On-Demand Anodyne WNT3 41 33 CN(CCN1CCOCC1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970624 ED On-Demand Anodyne CASR 53 42 O=C(NCCCNc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970626 EH On-Demand Anodyne TRPV1 31 53 C[C@H](O)c1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880970627 EG On-Demand Anodyne TRPV1 44 54 C[C@H](O)c1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880970627 EG On-Demand Anodyne NAMPT 58 36 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@@H]2C1 ZINC000880970634 EF On-Demand Anodyne HRH3 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@@H]2C1 ZINC000880970634 EF On-Demand Anodyne RBP4 66 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@@H]2C1 ZINC000880970634 EF On-Demand Anodyne L3MBTL3 48 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@H]2C1 ZINC000880970635 EF On-Demand Anodyne HRH3 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@H]2C1 ZINC000880970635 EF On-Demand Anodyne RBP4 66 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCCC[C@H]2C1 ZINC000880970635 EF On-Demand Anodyne L3MBTL3 48 37 N#Cc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970638 GG On-Demand Mild TRPV1 19 58 N#Cc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970638 GG On-Demand Mild RBP4 61 46 O=C(Nc1cnccc1C(F)(F)F)N1CCS(=O)CC1 ZINC000880970644 DD On-Demand Anodyne RBP4 60 44 CCN(CCNC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880970655 DF On-Demand Anodyne TRPV1 18 42 O=C(Cn1cc(CN2CCCCC2)nn1)NC1CCCCCCC1 ZINC000880970659 EE On-Demand Anodyne SIGMAR1 15 47 O=C(Cn1cc(CN2CCCCC2)nn1)NC1CCCCCCC1 ZINC000880970659 EE On-Demand Anodyne EPHX2 20 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccccc2C1 ZINC000880970660 EH On-Demand Anodyne TRPV1 29 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccccc2C1 ZINC000880970660 EH On-Demand Anodyne EPHX2 20 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2ccccc2C1 ZINC000880970661 EH On-Demand Anodyne TRPV1 29 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2ccccc2C1 ZINC000880970661 EH On-Demand Anodyne EPHX2 20 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CN2CCCCCC2)C1 ZINC000880970662 GI On-Demand Anodyne CCR3 16 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CN2CCCCCC2)C1 ZINC000880970662 GI On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CN2CCCCCC2)C1 ZINC000880970662 GI On-Demand Anodyne SFRP1 74 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CN2CCCCCC2)C1 ZINC000880970662 GI On-Demand Anodyne WNT3 59 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CN2CCCCCC2)C1 ZINC000880970663 GI On-Demand Anodyne CCR3 16 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CN2CCCCCC2)C1 ZINC000880970663 GI On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CN2CCCCCC2)C1 ZINC000880970663 GI On-Demand Anodyne SFRP1 74 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CN2CCCCCC2)C1 ZINC000880970663 GI On-Demand Anodyne WNT3 59 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cn1cccn1 ZINC000880970670 EF On-Demand Anodyne SFRP1 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cn1cccn1 ZINC000880970670 EF On-Demand Anodyne WNT3 49 34 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)cc1F ZINC000880970672 GG On-Demand Anodyne TRPV1 17 43 O=C(Nc1cnn(CC(F)F)c1)Nc1cnccc1C(F)(F)F ZINC000880970673 EG On-Demand Anodyne TRPV1 16 41 O=C(NCC[S@@](=O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970674 FG On-Demand Anodyne TRPV1 19 47 O=C(NCC[S@](=O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880970675 FG On-Demand Anodyne TRPV1 19 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc(F)c(F)c1 ZINC000880970677 FJ On-Demand Anodyne SFRP1 41 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc(F)c(F)c1 ZINC000880970677 FJ On-Demand Anodyne WNT3 46 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc(F)c(F)c1 ZINC000880970678 FJ On-Demand Anodyne SFRP1 41 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc(F)c(F)c1 ZINC000880970678 FJ On-Demand Anodyne WNT3 46 36 CN(CCNC(=O)Nc1cnccc1C(F)(F)F)C1CCCC1 ZINC000880970679 EG On-Demand Anodyne TRPV1 21 44 COc1ccc(CN(CCO)C(=O)Nc2cnccc2C(F)(F)F)c(OC)c1 ZINC000880970681 GG On-Demand Anodyne ROCK2 22 42 C[C@@H](O)CC(C)(C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970685 DG On-Demand Anodyne TRPV1 20 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](Cn2cccn2)C1 ZINC000880970728 FE On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](Cn2cccn2)C1 ZINC000880970733 FE On-Demand Anodyne RBP4 57 41 COCCCOC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970740 FG On-Demand Anodyne RBP4 66 42 O=C(NC[C@@H]1OCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970756 FH On-Demand Anodyne TRPV1 18 43 O=C(NC[C@H]1OCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970761 FH On-Demand Anodyne TRPV1 18 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@]2(CC=CCC2)C1 ZINC000880970770 EI On-Demand Anodyne RBP4 48 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@]2(CC=CCC2)C1 ZINC000880970774 EI On-Demand Anodyne RBP4 48 38 CC(C)c1ccccc1NC(=O)Cn1cc([C@@H](O)c2ccccc2)nn1 ZINC000880970779 FG On-Demand Anodyne SOAT1 44 36 CC(C)c1ccccc1NC(=O)Cn1cc([C@H](O)c2ccccc2)nn1 ZINC000880970784 FG On-Demand Anodyne SOAT1 44 36 Cn1cc(CN2CCCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cn1 ZINC000880970787 GF On-Demand Anodyne FAAH 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nnc3n2CCC3)CC1 ZINC000880970794 GG On-Demand Anodyne RBP4 71 42 COC(=O)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(C)cc1 ZINC000880970809 GG On-Demand Anodyne TRPV1 15 43 C[C@@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970810 GI On-Demand Anodyne RBP4 54 39 C[C@@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970810 GI On-Demand Anodyne SFRP1 47 36 C[C@@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970810 GI On-Demand Anodyne WNT3 46 36 COC(=O)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(C)cc1 ZINC000880970811 GG On-Demand Anodyne TRPV1 15 43 C[C@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970812 GI On-Demand Anodyne RBP4 54 39 C[C@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970812 GI On-Demand Anodyne SFRP1 47 36 C[C@H]1CCCCN1C[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970812 GI On-Demand Anodyne WNT3 46 36 O=C(NCc1nnc2n1CCCCC2)Nc1cnccc1C(F)(F)F ZINC000880970813 FF On-Demand Anodyne TRPV1 15 42 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1cnccc1C(F)(F)F ZINC000880970814 GH On-Demand Anodyne TRPV1 30 51 O=C(NCc1cccc(CN2CCCC2=O)c1)Nc1cnccc1C(F)(F)F ZINC000880970814 GH On-Demand Anodyne NAMPT 59 41 C[C@@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970815 GI On-Demand Anodyne RBP4 54 39 C[C@@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970815 GI On-Demand Anodyne SFRP1 47 36 C[C@@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970815 GI On-Demand Anodyne WNT3 46 36 CC(C)(C)OC(=O)N1CCC(c2cn(CC(=O)NC3CCCC3)nn2)CC1 ZINC000880970816 GE On-Demand Anodyne GPR119 44 42 C[C@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970817 GI On-Demand Anodyne RBP4 54 39 C[C@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970817 GI On-Demand Anodyne SFRP1 47 36 C[C@H]1CCCCN1C[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970817 GI On-Demand Anodyne WNT3 46 36 CC(C)(C)OC(=O)N1CCN(Cc2cn(CC(=O)NC3CCCC3)nn2)CC1 ZINC000880970818 GD On-Demand Anodyne KDM1A 19 44 O=C(NCc1cn2c(n1)CCCC2)Nc1cnccc1C(F)(F)F ZINC000880970823 EF On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)NC1(c2ccccc2)CC1 ZINC000880970826 DH On-Demand Anodyne TRPV1 21 47 CC(=O)N(Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1)C(C)C ZINC000880970829 GJ On-Demand Anodyne TRPV1 19 44 CCc1nnc2n1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880970831 EE On-Demand Anodyne P2RX7 27 41 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2CC1 ZINC000880970833 EH On-Demand Anodyne TRPV1 22 49 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2CC1 ZINC000880970833 EH On-Demand Anodyne RBP4 90 48 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2CC1 ZINC000880970833 EH On-Demand Anodyne TRPM8 55 44 O=C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CCN1 ZINC000880970834 DD On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2ncc[nH]2)C1 ZINC000880970842 EG On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2ncc[nH]2)C1 ZINC000880970844 EG On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880970848 GI On-Demand Anodyne PRCP 50 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000880970848 GI On-Demand Anodyne RBP4 43 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880970850 GI On-Demand Anodyne PRCP 50 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000880970850 GI On-Demand Anodyne RBP4 43 37 O=C(Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCC1 ZINC000880970860 FE On-Demand Anodyne CCR2 64 41 O=C(Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCC1 ZINC000880970862 FE On-Demand Anodyne CCR2 64 41 Cn1cc(CNC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880970864 CE On-Demand Anodyne TRPV1 25 49 Cn1cc(CNC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880970864 CE On-Demand Anodyne FLT1 22 41 Cn1cc(CNC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880970864 CE On-Demand Anodyne NAMPT 56 46 O=C(NCCCCNc1ccccn1)Nc1cnccc1C(F)(F)F ZINC000880970872 FH On-Demand Anodyne TRPV1 20 47 O=C(NCc1ccnc(OC2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880970873 GG On-Demand Anodyne TRPV1 16 45 C[C@@H]1SCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H]1C ZINC000880970875 DG On-Demand Anodyne RBP4 40 38 Cc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880970876 EH On-Demand Anodyne RBP4 57 42 Cc1cccc2c1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880970876 EH On-Demand Anodyne P2RY14 51 38 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970879 GH On-Demand Anodyne TRPV1 26 51 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970879 GH On-Demand Anodyne ROCK2 44 39 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970879 GH On-Demand Anodyne CARM1 40 35 CC[C@H](C)NC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970879 GH On-Demand Anodyne NAMPT 40 37 C[C@@H]1SCCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H]1C ZINC000880970880 DG On-Demand Anodyne RBP4 40 38 O=C(Cn1cc(-c2ccc(Cl)cc2F)nn1)NC1CCCC1 ZINC000880970883 DF On-Demand Anodyne CNR1 28 53 Cc1nc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)oc1C ZINC000880970887 GG On-Demand Anodyne ABL1 42 35 CC(C)n1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)n1 ZINC000880970890 EG On-Demand Anodyne TRPV1 17 47 CN1CCC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880970895 DF On-Demand Anodyne TRPV1 17 41 O=C(CC1CCCCC1)NCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970902 FG On-Demand Anodyne TRPV1 16 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000880970903 FE On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000880970904 FE On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000880970905 FE On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000880970906 FE On-Demand Anodyne RBP4 66 42 CC[C@@](C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880970910 CE On-Demand Anodyne TRPV1 22 47 O=C(NCC(=O)N1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970912 EE On-Demand Anodyne TRPV1 19 44 O=C(NCC(=O)N1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970912 EE On-Demand Anodyne PRMT3 18 47 O=C(NCC(=O)N1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880970912 EE On-Demand Anodyne NAMPT 16 40 CC(C)(C)OC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970914 GH On-Demand Anodyne RBP4 66 41 CC(C)(C)OC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970914 GH On-Demand Anodyne SFRP1 103 37 CC(C)(C)OC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880970914 GH On-Demand Anodyne WNT3 81 35 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(Cl)cccc2C1 ZINC000880970917 FI On-Demand Anodyne RBP4 60 44 O=C(Nc1cnccc1C(F)(F)F)N1CCc2c(Cl)cccc2C1 ZINC000880970917 FI On-Demand Anodyne TRPM8 28 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CCC1 ZINC000880970918 DH On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CCC1 ZINC000880970920 DH On-Demand Anodyne RBP4 56 41 C[C@@H](Cn1cncn1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880970924 DD On-Demand Anodyne HIS3 81 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccnn2)CC1 ZINC000880970925 FE On-Demand Anodyne TRPV1 20 56 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccnn2)CC1 ZINC000880970925 FE On-Demand Anodyne RBP4 59 41 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970930 GH On-Demand Anodyne BMP1 50 38 COCCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880970930 GH On-Demand Anodyne NOS2 50 33 O=C(NC[C@@]1(O)CCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970931 FG On-Demand Anodyne TRPV1 18 47 O=C(NC[C@]1(O)CCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970932 FG On-Demand Anodyne TRPV1 18 47 O=C(NC[C@H]1CCOc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970934 FH On-Demand Anodyne TRPV1 23 44 O=C(NC[C@@H]1CCOc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880970935 FH On-Demand Anodyne TRPV1 23 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccco1 ZINC000880970947 EI On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccco1 ZINC000880970949 EI On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880970950 EF On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880970950 EF On-Demand Anodyne CXCR3 15 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC2CC2)C1 ZINC000880970950 EF On-Demand Anodyne RBP4 52 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC2CC2)C1 ZINC000880970952 EF On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC2CC2)C1 ZINC000880970952 EF On-Demand Anodyne CXCR3 15 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC2CC2)C1 ZINC000880970952 EF On-Demand Anodyne RBP4 52 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)c2ccc(F)cc2)CC1 ZINC000880970953 GI On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)c2ccc(F)cc2)CC1 ZINC000880970955 GI On-Demand Anodyne RBP4 65 40 O=C(NCc1ccc(OCC2CC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880970957 FH On-Demand Anodyne TRPV1 22 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC(F)(F)F)CC1 ZINC000880970958 FF On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC(F)(F)F)CC1 ZINC000880970958 FF On-Demand Anodyne RBP4 59 43 O=C(NC[C@H]1CCN(c2ccc(F)cc2)C1)Nc1cnccc1C(F)(F)F ZINC000880970959 GH On-Demand Anodyne TRPV1 15 40 O=C(NC[C@@H]1CCN(c2ccc(F)cc2)C1)Nc1cnccc1C(F)(F)F ZINC000880970960 GH On-Demand Anodyne TRPV1 15 40 C[C@H]1C[C@H]1c1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)o1 ZINC000880970964 EI On-Demand Anodyne TRPV1 17 42 C[C@@H]1C[C@H]1c1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)o1 ZINC000880970966 EI On-Demand Anodyne TRPV1 17 42 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne KCNQ2 32 40 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne TRPV1 24 60 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne ROCK1 18 57 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne RAF1 20 41 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne ROCK2 22 43 COc1cccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970969 EH On-Demand Anodyne TAAR1 23 42 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne KCNQ2 32 40 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne TRPV1 24 60 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne ROCK1 18 57 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne RAF1 20 41 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne ROCK2 22 43 COc1cccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880970970 EH On-Demand Anodyne TAAR1 23 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)NC1CCCCCCC1 ZINC000880970972 FD On-Demand Anodyne EPHX2 16 46 O=C1C[C@@H](c2ccccc2)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1 ZINC000880970974 GG On-Demand Anodyne RBP4 58 41 O=C1C[C@H](c2ccccc2)N(C(=O)Nc2cnccc2C(F)(F)F)CCN1 ZINC000880970975 GG On-Demand Anodyne RBP4 58 41 Cc1ccc(N2CCCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880970977 GI On-Demand Anodyne RBP4 53 38 O=C(Cn1cc(COc2ccc(CO)cc2)nn1)NC1CCCCCCC1 ZINC000880970978 FF On-Demand Anodyne FIMH 15 42 O=C(NCCOc1ccc2c(c1)OCO2)Nc1cnccc1C(F)(F)F ZINC000880970980 FG On-Demand Anodyne HRH2 20 46 O=C(NC[C@H]1CC=CCC1)Nc1cnccc1C(F)(F)F ZINC000880970982 CH On-Demand Anodyne TRPV1 15 45 O=C(NC[C@@H]1CC=CCC1)Nc1cnccc1C(F)(F)F ZINC000880970983 CH On-Demand Anodyne TRPV1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CC2C[C@H]3CC1C[C@@H](C2)C3 ZINC000880970984 EI On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccsc2)CC1 ZINC000880970985 GG On-Demand Anodyne RBP4 58 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880970986 FF On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880970986 FF On-Demand Anodyne EPHX2 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880970986 FF On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880970986 FF On-Demand Anodyne SFRP1 74 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCC2)CC1 ZINC000880970986 FF On-Demand Anodyne WNT3 67 36 Nc1cccc(OCc2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880970987 FF On-Demand Anodyne FAAH 25 45 O=C(CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)NC1CCCC1 ZINC000880970988 GH On-Demand Anodyne RBP4 61 39 O=C(Cn1cc(C(=O)c2ccccc2)nn1)NC1CCCCCCC1 ZINC000880970990 EF On-Demand Anodyne EPHX2 15 43 O=C(Cn1cc(C(=O)c2ccccc2)nn1)NC1CCCCCCC1 ZINC000880970990 EF On-Demand Anodyne SCARB1 32 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC2CC2)CC1 ZINC000880970995 EF On-Demand Anodyne TRPV1 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC2CC2)CC1 ZINC000880970995 EF On-Demand Anodyne RBP4 72 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne GRIN2B 35 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne TRPV1 20 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne FAAH 18 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne EPHX2 28 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne RBP4 89 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne SFRP1 87 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne DGAT1 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(COc2ccccc2)CC1 ZINC000880970996 GI On-Demand Anodyne WNT3 68 33 COCCNC(=O)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880971001 EC On-Demand Anodyne LGALS3 36 45 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971003 GG On-Demand Clean TRPV1 21 50 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971003 GG On-Demand Clean STAT6 62 42 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971003 GG On-Demand Clean NAMPT 82 43 CC(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971009 EE On-Demand Anodyne EPHX2 25 40 CC(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971009 EE On-Demand Anodyne RBP4 70 42 CC(=O)NCC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971009 EE On-Demand Anodyne CACNA1I 40 33 O=C(NCC(=O)N1CCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880971016 GG On-Demand Anodyne AVPR2 32 40 O=C(NCC(=O)N1CCCc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880971016 GG On-Demand Anodyne TRPV1 24 45 CS(=O)(=O)c1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971017 GF On-Demand Anodyne HDAC10 18 41 CS(=O)(=O)c1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971017 GF On-Demand Anodyne HDAC3 18 41 CS(=O)(=O)c1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971017 GF On-Demand Anodyne HDAC6 15 41 CS(=O)(=O)c1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971017 GF On-Demand Anodyne FAAH 23 47 CS(=O)(=O)c1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971017 GF On-Demand Anodyne EPHX2 20 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880971020 GG On-Demand Anodyne TRPV1 29 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1=O ZINC000880971020 GG On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880971021 GG On-Demand Anodyne TRPV1 29 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1=O ZINC000880971021 GG On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)N1CCc2sccc2C1 ZINC000880971022 EH On-Demand Anodyne RBP4 57 42 O=C(NCCS(=O)(=O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880971027 GF On-Demand Anodyne TRPV1 21 47 O=C(NCCS(=O)(=O)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880971027 GF On-Demand Anodyne NAMPT 47 38 O=C(Nc1cnccc1C(F)(F)F)N1C2CCC1CC2 ZINC000880971028 CG On-Demand Anodyne RBP4 60 41 Nc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971033 EF On-Demand Anodyne HDAC10 20 41 Nc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971033 EF On-Demand Anodyne HDAC3 21 41 Nc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971033 EF On-Demand Anodyne HDAC6 17 41 Nc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880971033 EF On-Demand Anodyne FAAH 25 48 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880971036 FF On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880971036 FF On-Demand Anodyne CXCR3 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(CC(F)(F)F)C1 ZINC000880971036 FF On-Demand Anodyne HPGDS 40 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880971037 FF On-Demand Anodyne TRPV1 19 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880971037 FF On-Demand Anodyne CXCR3 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(CC(F)(F)F)C1 ZINC000880971037 FF On-Demand Anodyne HPGDS 40 43 N[C@@H](Cc1cn(CC(=O)NC2CCCCCCC2)nn1)c1ccccc1 ZINC000880971043 FF On-Demand Anodyne SCARB1 33 40 N[C@H](Cc1cn(CC(=O)NC2CCCCCCC2)nn1)c1ccccc1 ZINC000880971044 FF On-Demand Anodyne SCARB1 33 40 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NCC(F)(F)F ZINC000880971049 ED On-Demand Anodyne TRPV1 16 47 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880971054 CG On-Demand Anodyne TRPV1 23 44 CC(C)(O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971061 CD On-Demand Anodyne TRPV1 26 49 O=C(Nc1cnccc1C(F)(F)F)NC1(c2ccccc2)CCC1 ZINC000880971067 EI On-Demand Anodyne TRPV1 15 44 COC(=O)C1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971068 EF On-Demand Anodyne EPHX2 47 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000880971072 GE On-Demand Anodyne RBP4 63 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000880971072 GE On-Demand Anodyne SFRP1 49 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C(=O)N2CCOCC2)C1 ZINC000880971072 GE On-Demand Anodyne WNT3 41 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCOCC2)C1 ZINC000880971073 GE On-Demand Anodyne RBP4 63 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCOCC2)C1 ZINC000880971073 GE On-Demand Anodyne SFRP1 49 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C(=O)N2CCOCC2)C1 ZINC000880971073 GE On-Demand Anodyne WNT3 41 37 CCS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971074 FD On-Demand Anodyne TRPV1 17 44 CCS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971074 FD On-Demand Anodyne RBP4 70 45 CC(C)(C)OC(=O)NCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971077 FG On-Demand Anodyne TRPV1 19 47 O=C(Cn1cc(-c2ccccn2)nn1)NC1CCCCCCC1 ZINC000880971080 DF On-Demand Anodyne EPHX2 16 42 O=C(NC[C@H](O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880971081 CD On-Demand Anodyne TRPV1 20 45 O=C(NC[C@@H](O)C1CC1)Nc1cnccc1C(F)(F)F ZINC000880971082 CD On-Demand Anodyne TRPV1 20 45 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)Oc1ccccc1 ZINC000880971088 EH On-Demand Anodyne TRPV1 23 48 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)Oc1ccccc1 ZINC000880971088 EH On-Demand Anodyne SOAT1 15 40 CN(C)C(=O)c1cccc(CCNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880971089 GG On-Demand Anodyne TRPV1 27 57 CN(C)C(=O)c1cccc(CCNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880971089 GG On-Demand Anodyne RAF1 34 41 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971090 GH On-Demand Anodyne EPHX2 54 45 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971090 GH On-Demand Anodyne GPR119 51 45 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971090 GH On-Demand Anodyne SFRP1 110 45 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971090 GH On-Demand Anodyne WNT3 82 39 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne CTSB 35 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne CTSK 29 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne PREP 31 45 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne CAPNS1 47 32 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne CAPN1 57 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne CAPN2 96 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCC1 ZINC000880971092 FD On-Demand Anodyne NPR 59 33 C[C@@]1(CNC(=O)Nc2cnccc2C(F)(F)F)CCOC1 ZINC000880971093 DF On-Demand Anodyne TRPV1 16 45 COC(=O)[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880971094 ED On-Demand Anodyne RBP4 69 42 COC(=O)[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880971096 ED On-Demand Anodyne RBP4 69 42 O=C(Nc1cnccc1C(F)(F)F)NC1(c2cccc(F)c2)CC1 ZINC000880971100 EI On-Demand Anodyne TRPV1 22 43 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971101 FF On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971101 FF On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971101 FF On-Demand Anodyne SCARB1 32 41 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971103 FF On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971103 FF On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971103 FF On-Demand Anodyne SCARB1 32 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@H]2CCOC2)CC1 ZINC000880971106 FF On-Demand Anodyne CXCR3 16 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@@H]2CCOC2)CC1 ZINC000880971108 FF On-Demand Anodyne CXCR3 16 46 Cc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)no1 ZINC000880971128 DE On-Demand Anodyne TRPV1 23 50 CC1(C)C[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971129 CG On-Demand Anodyne TRPV1 25 47 Cn1nccc1C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971135 FG On-Demand Anodyne RBP4 75 44 N#Cc1cccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971136 GI On-Demand Mild CCR3 25 40 N#Cc1cccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971136 GI On-Demand Mild EPHX2 25 51 N#Cc1cccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971136 GI On-Demand Mild RBP4 61 38 N#Cc1cccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971136 GI On-Demand Mild SCD1 20 42 CCOC[C@H](O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971145 GD On-Demand Anodyne RBP4 46 38 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)c(C)c1 ZINC000880971149 FI On-Demand Anodyne RAF1 48 41 COc1nc(C)cc(C)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971150 FG On-Demand Anodyne TRPV1 22 46 CC(C)c1nnc2n1CCN(C(=O)Nc1cnccc1C(F)(F)F)C2 ZINC000880971155 FF On-Demand Anodyne P2RX7 28 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCO)CC1 ZINC000880971164 ED On-Demand Anodyne CCR3 20 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCO)CC1 ZINC000880971164 ED On-Demand Anodyne SLC6A5 31 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCO)CC1 ZINC000880971164 ED On-Demand Anodyne EPHX2 45 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCO)CC1 ZINC000880971164 ED On-Demand Anodyne CXCR3 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](C2OCCO2)C1 ZINC000880971170 EF On-Demand Anodyne RBP4 85 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C2OCCO2)C1 ZINC000880971172 EF On-Demand Anodyne RBP4 85 46 CSC[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971175 CF On-Demand Anodyne TRPV1 17 46 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccc(F)c(F)c2)C1 ZINC000880971176 GH On-Demand Anodyne RBP4 57 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccc(F)c(F)c2)C1 ZINC000880971178 GH On-Demand Anodyne RBP4 57 40 COc1ccccc1[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971179 FF On-Demand Anodyne TRPV1 20 46 COc1ccccc1[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971179 FF On-Demand Anodyne SOAT1 21 40 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCC3)nn2)c1 ZINC000880971180 EE On-Demand Anodyne FAAH 22 45 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCC3)nn2)c1 ZINC000880971180 EE On-Demand Anodyne SCARB1 31 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CC=CC2)C1 ZINC000880971181 EF On-Demand Anodyne RBP4 68 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CC=CC2)C1 ZINC000880971183 EF On-Demand Anodyne RBP4 68 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880971184 GE On-Demand Anodyne TRPV1 22 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880971184 GE On-Demand Anodyne GRM4 38 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880971184 GE On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880971184 GE On-Demand Anodyne SCD1 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccn2)CC1 ZINC000880971184 GE On-Demand Anodyne SFRP1 22 44 C#CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971187 CE On-Demand Mild TRPV1 17 50 O=C(NCCn1cccn1)Nc1cnccc1C(F)(F)F ZINC000880971189 CE On-Demand Anodyne TRPV1 19 47 CCOc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1OC ZINC000880971190 FH On-Demand Anodyne TRPV1 28 50 CCOc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1OC ZINC000880971190 FH On-Demand Anodyne SSTR5 40 38 CCOc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1OC ZINC000880971190 FH On-Demand Anodyne RAF1 31 41 CCOc1cc(CNC(=O)Nc2cnccc2C(F)(F)F)ccc1OC ZINC000880971190 FH On-Demand Anodyne ROCK2 24 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccccc2F)C1 ZINC000880971195 FH On-Demand Anodyne RBP4 94 49 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccccc2F)C1 ZINC000880971197 FH On-Demand Anodyne RBP4 94 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Cn2cccn2)CC1 ZINC000880971202 FG On-Demand Anodyne RBP4 70 42 C[C@H](O)c1ccc(OCc2cn(CC(=O)NC3CCCC3)nn2)cc1 ZINC000880971205 ED On-Demand Anodyne ALOX5 23 40 COc1ccc([C@@H]2CCN(C(=O)Nc3cnccc3C(F)(F)F)C2)cc1 ZINC000880971207 FI On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Nc2cccnn2)CC1 ZINC000880971208 FF On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Nc2cccnn2)CC1 ZINC000880971208 FF On-Demand Anodyne SFRP1 58 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC(Nc2cccnn2)CC1 ZINC000880971208 FF On-Demand Anodyne WNT3 40 33 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971211 GG On-Demand Anodyne RBP4 57 39 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971211 GG On-Demand Anodyne CACNA1I 46 32 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971211 GG On-Demand Anodyne WNT3 40 31 CC(=O)N(Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1)C1CC1 ZINC000880971212 GI On-Demand Anodyne TRPV1 27 44 CC(=O)N(Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1)C1CC1 ZINC000880971212 GI On-Demand Anodyne RAF1 40 39 CC(=O)N(Cc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1)C1CC1 ZINC000880971212 GI On-Demand Anodyne MTOR 40 31 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971213 GG On-Demand Anodyne RBP4 57 39 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971213 GG On-Demand Anodyne CACNA1I 46 32 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971213 GG On-Demand Anodyne WNT3 40 31 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880971215 GF On-Demand Anodyne TRPV1 20 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880971215 GF On-Demand Anodyne SLC9A1 23 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880971215 GF On-Demand Anodyne EPHX2 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(O)c2)CC1 ZINC000880971215 GF On-Demand Anodyne RBP4 69 43 O=C(Cn1cc(C[C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971221 FF On-Demand Anodyne PGC 41 30 O=C(Cn1cc(C[C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971221 FF On-Demand Anodyne REN 64 34 O=C(Cn1cc(C[C@@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971221 FF On-Demand Anodyne SCARB1 34 41 O=C(NCCCC(=O)N1Cc2ccccc2C1)Nc1cnccc1C(F)(F)F ZINC000880971222 GH On-Demand Anodyne TRPV1 20 48 O=C(Cn1cc(C[C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971223 FF On-Demand Anodyne PGC 41 30 O=C(Cn1cc(C[C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971223 FF On-Demand Anodyne REN 64 34 O=C(Cn1cc(C[C@H](O)Cc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971223 FF On-Demand Anodyne SCARB1 34 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc3nncn3n2)CC1 ZINC000880971235 GD On-Demand Anodyne RBP4 48 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCC2)CC1 ZINC000880971237 EF On-Demand Anodyne HRH3 22 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCC2)CC1 ZINC000880971237 EF On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880971238 GI On-Demand Anodyne TRPV1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880971238 GI On-Demand Anodyne CCR2 18 52 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ncccc23)CC1 ZINC000880971238 GI On-Demand Anodyne RBP4 82 47 CN(C)C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880971240 ED On-Demand Anodyne RBP4 65 41 Nc1cccc(OCc2cn(CC(=O)NC3CCCC3)nn2)c1 ZINC000880971243 DD On-Demand Anodyne FAAH 22 44 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880971246 GF On-Demand Anodyne P2RX7 31 43 O=C(Nc1cnccc1C(F)(F)F)N1CCn2c(nnc2C(F)(F)F)C1 ZINC000880971246 GF On-Demand Anodyne RBP4 57 41 CC(C)c1ccccc1NC(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880971253 FG On-Demand Anodyne SOAT1 47 37 CC(C)c1ccccc1NC(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880971254 FG On-Demand Anodyne SOAT1 47 37 CCOc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971255 GF On-Demand Anodyne TRPV1 15 42 CCOc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971255 GF On-Demand Anodyne RBP4 41 41 O=C(NC[C@H]1CCCCO1)Nc1cnccc1C(F)(F)F ZINC000880971260 DF On-Demand Anodyne TRPV1 15 42 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971262 GH On-Demand Anodyne PRKD1 23 40 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971262 GH On-Demand Anodyne EPHX2 47 47 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971262 GH On-Demand Anodyne RBP4 66 40 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971262 GH On-Demand Anodyne SFRP1 57 34 O=C(NC1CCCCC1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971262 GH On-Demand Anodyne WNT3 46 33 O=C(Cn1cc(-c2cccnc2Cl)nn1)NC1CCCCCCC1 ZINC000880971271 EG On-Demand Anodyne CNR1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC2CCCC2)CC1 ZINC000880971272 FI On-Demand Anodyne EPHX2 17 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OC2CCCC2)CC1 ZINC000880971272 FI On-Demand Anodyne RBP4 73 43 O=C(Cn1cc([C@@H](O)c2ccc(F)cc2)nn1)NC1CCCCCCC1 ZINC000880971273 FF On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@H](O)c2ccc(F)cc2)nn1)NC1CCCCCCC1 ZINC000880971274 FF On-Demand Anodyne SCARB1 29 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971282 GE On-Demand Anodyne RBP4 67 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971282 GE On-Demand Anodyne CCR8 81 39 CCS(=O)(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971282 GE On-Demand Anodyne SFRP1 132 41 CCS(=O)(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971282 GE On-Demand Anodyne WNT3 91 38 O=C(Nc1cnccc1C(F)(F)F)N1C[C@H]2CC[C@H]1C2 ZINC000880971285 CG On-Demand Anodyne RBP4 62 42 Cc1noc(C)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971286 DG On-Demand Anodyne TRPV1 19 48 Cc1noc(C)c1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971286 DG On-Demand Anodyne P2RX7 15 51 O=C(NCCN1CCc2sccc2C1)Nc1cnccc1C(F)(F)F ZINC000880971291 FG On-Demand Anodyne UTS2R 16 43 O=C(NCCOCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880971296 EF On-Demand Anodyne TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cscn2)CC1 ZINC000880971299 FF On-Demand Anodyne RBP4 54 39 CS(=O)(=O)N1CCN(CCNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971300 GC On-Demand Anodyne TRPV1 21 40 CS(=O)(=O)N1CCN(CCNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971300 GC On-Demand Anodyne CCR3 19 42 CS(=O)(=O)N1CCN(CCNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971300 GC On-Demand Anodyne ABL2 42 35 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CCCCC1 ZINC000880971301 GH On-Demand Anodyne C3AR1 41 39 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CCCCC1 ZINC000880971301 GH On-Demand Anodyne EPHX2 44 43 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CCCCC1 ZINC000880971301 GH On-Demand Anodyne RBP4 65 40 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CCCCC1 ZINC000880971301 GH On-Demand Anodyne SFRP1 82 36 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)C1CCCCC1 ZINC000880971301 GH On-Demand Anodyne WNT3 71 35 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1O ZINC000880971302 FG On-Demand Anodyne TRPV1 15 42 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880971303 GF On-Demand Mild RBP4 42 37 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880971303 GF On-Demand Mild DGAT1 20 40 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)C(C)C ZINC000880971305 CH On-Demand Anodyne TRPV1 18 49 CN(C(=O)Nc1cnccc1C(F)(F)F)C1Cc2ccccc2C1 ZINC000880971312 EH On-Demand Anodyne TRPV1 21 40 O=C(NCCCS(=O)(=O)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880971315 GG On-Demand Anodyne TRPV1 20 47 O=C(NCCCS(=O)(=O)c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880971315 GG On-Demand Anodyne NAMPT 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccn1 ZINC000880971320 EH On-Demand Anodyne RBP4 70 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccn1 ZINC000880971320 EH On-Demand Anodyne SFRP1 49 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccn1 ZINC000880971320 EH On-Demand Anodyne WNT3 49 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccn1 ZINC000880971321 EH On-Demand Anodyne RBP4 70 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccn1 ZINC000880971321 EH On-Demand Anodyne SFRP1 49 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccn1 ZINC000880971321 EH On-Demand Anodyne WNT3 49 35 O=C(Cn1cc(CNCc2ccc(F)cc2)nn1)NC1CCCCCCC1 ZINC000880971322 FF On-Demand Anodyne SCARB1 28 40 CS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971325 FD On-Demand Anodyne TRPV1 15 45 CS(=O)(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971325 FD On-Demand Anodyne RBP4 72 46 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(S(C)(=O)=O)cc1 ZINC000880971326 GG On-Demand Anodyne TRPV1 50 33 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(S(C)(=O)=O)cc1 ZINC000880971326 GG On-Demand Anodyne CTSF 52 37 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne HTR1A 65 43 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne DRD2 52 51 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne DRD4 33 41 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne ADRA1D 65 51 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne ADRA1A 55 51 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne ADRA1B 48 51 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne DRD3 56 43 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne PDE3A 19 40 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne HTR7 45 39 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne TRPV1 27 43 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne EPHX2 48 42 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne RBP4 60 43 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne SCD1 33 41 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne SFRP1 71 34 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne SCD 27 41 COc1ccccc1N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971337 GH On-Demand Anodyne WNT3 43 32 O=C(NCCCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880971338 EF On-Demand Anodyne TBXAS1 48 56 O=C(NCCCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880971338 EF On-Demand Anodyne QPCT 44 53 C[C@@H]1CCCN(C(=O)C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)C1 ZINC000880971339 GH On-Demand Anodyne RBP4 73 42 C[C@@H]1CCCN(C(=O)C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)C1 ZINC000880971339 GH On-Demand Anodyne SFRP1 68 33 C[C@@H]1CCCN(C(=O)C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)C1 ZINC000880971339 GH On-Demand Anodyne WNT3 59 33 COCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971342 EE On-Demand Anodyne CCR3 25 40 COCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971342 EE On-Demand Anodyne SLC6A5 32 41 COCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971342 EE On-Demand Anodyne EPHX2 51 41 COCCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971342 EE On-Demand Anodyne CXCR3 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)N2CCCC2)CC1 ZINC000880971349 FE On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)N2CCCC2)CC1 ZINC000880971349 FE On-Demand Anodyne RBP4 60 44 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccccc2)O1 ZINC000880971353 FI On-Demand Anodyne RBP4 86 47 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccccc2)O1 ZINC000880971354 FI On-Demand Anodyne RBP4 86 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@H](c2ccccc2)O1 ZINC000880971355 FI On-Demand Anodyne RBP4 86 47 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)C[C@@H](c2ccccc2)O1 ZINC000880971356 FI On-Demand Anodyne RBP4 86 47 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne HTR1A 54 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne DRD2 39 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne ADRA1D 43 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne ADRA1A 38 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne DRD3 48 38 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne PDE3A 24 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne HTR7 40 40 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne TRPV1 17 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne CCR3 22 41 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne PIM1 19 42 COc1ccccc1N1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971359 GH On-Demand Anodyne RBP4 48 38 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne HTR1A 54 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne DRD2 39 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne ADRA1D 43 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne ADRA1A 38 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne DRD3 48 38 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne PDE3A 24 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne HTR7 40 40 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne TRPV1 17 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne CCR3 22 41 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne PIM1 19 42 COc1ccccc1N1CC[C@@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971360 GH On-Demand Anodyne RBP4 48 38 O=C(NCc1ccc2c(c1)CCO2)Nc1cnccc1C(F)(F)F ZINC000880971361 EG On-Demand Anodyne TRPV1 21 51 O=C(NCc1ccc2c(c1)CCO2)Nc1cnccc1C(F)(F)F ZINC000880971361 EG On-Demand Anodyne NAMPT 40 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CC1 ZINC000880971376 CH On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CC1 ZINC000880971376 CH On-Demand Anodyne SFRP1 42 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CC1 ZINC000880971376 CH On-Demand Anodyne WNT3 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CC1 ZINC000880971377 CH On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CC1 ZINC000880971377 CH On-Demand Anodyne SFRP1 42 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CC1 ZINC000880971377 CH On-Demand Anodyne WNT3 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](n2ccnc2)C1 ZINC000880971380 EG On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](n2ccnc2)C1 ZINC000880971381 EG On-Demand Anodyne RBP4 61 42 COc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971384 GE On-Demand Anodyne TRPV1 17 43 COc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971384 GE On-Demand Anodyne RBP4 50 46 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971385 FI On-Demand Anodyne RBP4 80 43 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971385 FI On-Demand Anodyne SFRP1 42 34 COc1ccccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971385 FI On-Demand Anodyne WNT3 41 32 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971386 FI On-Demand Anodyne RBP4 80 43 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971386 FI On-Demand Anodyne SFRP1 42 34 COc1ccccc1[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880971386 FI On-Demand Anodyne WNT3 41 32 CCC(CC)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971389 CH On-Demand Anodyne TRPV1 21 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCC[C@H]2C1 ZINC000880971390 DE On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN2CCC[C@@H]2C1 ZINC000880971391 DE On-Demand Anodyne RBP4 67 44 Cc1noc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971393 FG On-Demand Anodyne RBP4 72 42 Cc1noc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971393 FG On-Demand Anodyne SMO 42 56 Cc1noc(C2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)n1 ZINC000880971393 FG On-Demand Anodyne ETHR 64 38 O=C(Cn1cc(C(=O)c2ccc(Cl)cc2)nn1)NC1CCCC1 ZINC000880971394 EE On-Demand Anodyne CNR1 21 45 O=C(Cn1cc(C(=O)c2ccc(Cl)cc2)nn1)NC1CCCC1 ZINC000880971394 EE On-Demand Anodyne SCARB1 30 41 O=C(NCCCN1CCOC1=O)Nc1cnccc1C(F)(F)F ZINC000880971403 EE On-Demand Anodyne CCR3 15 43 C=C(C)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971407 EG On-Demand Mild EPHX2 43 43 C=C(C)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971407 EG On-Demand Mild CXCR3 20 45 O=C(Cn1cc(COc2cccc(CO)c2)nn1)NC1CCCCCCC1 ZINC000880971409 FF On-Demand Anodyne HRH2 27 43 O=C(Cn1cc(COc2cccc(CO)c2)nn1)NC1CCCCCCC1 ZINC000880971409 FF On-Demand Anodyne FAAH 29 49 O=C(Cn1cc(COc2cccc(CO)c2)nn1)NC1CCCCCCC1 ZINC000880971409 FF On-Demand Anodyne FIMH 18 41 O=C(NCC(=O)N1CCc2ccccc2C1)Nc1cnccc1C(F)(F)F ZINC000880971410 GF On-Demand Anodyne TRPV1 17 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2ccc(F)cc21 ZINC000880971412 EI On-Demand Anodyne TRPV1 32 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2ccc(F)cc21 ZINC000880971413 EI On-Demand Anodyne TRPV1 32 49 CC(C)(C)NC(=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971414 EF On-Demand Anodyne TRPV1 25 51 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCN2CCOCC2)CC1 ZINC000880971416 GG On-Demand Anodyne RBP4 64 39 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971419 FF On-Demand Anodyne SCARB1 33 40 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NC1CCCCCCC1 ZINC000880971420 FF On-Demand Anodyne SCARB1 33 40 O=C(NCCOCCO)Nc1cnccc1C(F)(F)F ZINC000880971421 CD On-Demand Anodyne TRPV1 15 46 Cc1ccccc1CN(C(=O)Nc1cnccc1C(F)(F)F)C1CC1 ZINC000880971424 EJ On-Demand Anodyne TRPV1 21 42 COC(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971427 EE On-Demand Anodyne TRPV1 19 40 COC(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971427 EE On-Demand Anodyne EPHX2 41 43 COC(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971427 EE On-Demand Anodyne RBP4 44 37 COC(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971427 EE On-Demand Anodyne SFRP1 72 34 COC(=O)N1CCC[C@@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971427 EE On-Demand Anodyne WNT3 64 33 COC(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971428 EE On-Demand Anodyne TRPV1 19 40 COC(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971428 EE On-Demand Anodyne EPHX2 41 43 COC(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971428 EE On-Demand Anodyne RBP4 44 37 COC(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971428 EE On-Demand Anodyne SFRP1 72 34 COC(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971428 EE On-Demand Anodyne WNT3 64 33 O=C(NCC1(O)CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880971429 DF On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880971430 GG On-Demand Anodyne C3AR1 42 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880971430 GG On-Demand Anodyne EPHX2 51 62 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880971430 GG On-Demand Anodyne RBP4 39 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880971430 GG On-Demand Anodyne SFRP1 67 35 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)CC(F)(F)F)CC1 ZINC000880971430 GG On-Demand Anodyne WNT3 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCS(=O)(=O)CC1 ZINC000880971439 ED On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000880971440 GG On-Demand Anodyne CASR 45 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000880971442 GG On-Demand Anodyne CASR 45 41 O=C(Nc1ccc(O[C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971443 FH On-Demand Anodyne P2RY1 43 36 O=C(Nc1ccc(O[C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971443 FH On-Demand Anodyne RAF1 45 43 O=C(Nc1ccc(O[C@@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971443 FH On-Demand Anodyne EPHX2 46 42 O=C(Nc1ccc(O[C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971445 FH On-Demand Anodyne P2RY1 43 36 O=C(Nc1ccc(O[C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971445 FH On-Demand Anodyne RAF1 45 43 O=C(Nc1ccc(O[C@H]2CCOC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880971445 FH On-Demand Anodyne EPHX2 46 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCc2ccccc2C1 ZINC000880971447 EI On-Demand Anodyne TRPV1 17 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCc2ccccc2C1 ZINC000880971449 EI On-Demand Anodyne TRPV1 17 41 N#CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971453 EE On-Demand Mild EPHX2 42 42 N#CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971453 EE On-Demand Mild CXCR3 19 42 COc1ccc(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880971462 GH On-Demand Clean TRPV1 21 41 COc1ccc(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880971462 GH On-Demand Clean EPHX2 58 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccco2)C1 ZINC000880971464 EH On-Demand Anodyne RBP4 89 46 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccco2)C1 ZINC000880971467 EH On-Demand Anodyne RBP4 89 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2cc[nH]n2)CC1 ZINC000880971468 EG On-Demand Anodyne RBP4 75 44 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971469 GH On-Demand Anodyne C3AR1 40 38 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971469 GH On-Demand Anodyne RBP4 58 39 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971469 GH On-Demand Anodyne SFRP1 61 33 O=C(CC1CCCC1)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971469 GH On-Demand Anodyne WNT3 55 33 CC[C@@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccncc1 ZINC000880971475 DH On-Demand Anodyne TRPV1 17 61 CCOC(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971476 FG On-Demand Anodyne RBP4 65 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)c1ccccc1 ZINC000880971479 EG On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC2(C1)OCCO2 ZINC000880971481 DE On-Demand Anodyne RBP4 55 40 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne DRD4 17 42 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne TRPV1 22 43 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne CHRNA7 18 40 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne SLC6A5 30 41 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne EPHX2 40 42 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne RBP4 92 46 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne MCHR1 15 41 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne SFRP1 123 43 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne SMO 21 43 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne WNT3 83 38 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccccc1 ZINC000880971486 GH On-Demand Anodyne HPGDS 37 43 CC(C)c1ccccc1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880971488 GH On-Demand Anodyne MMP13 18 48 CC(C)c1ccccc1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880971488 GH On-Demand Anodyne MMP8 26 47 O=C(NCCN1Cc2ccccc2C1)Nc1cnccc1C(F)(F)F ZINC000880971490 FG On-Demand Anodyne TRPV1 26 48 O=C(Nc1cnccc1C(F)(F)F)N(CCO)CCc1ccccc1 ZINC000880971492 FG On-Demand Anodyne TRPV1 17 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CO)C1CC1 ZINC000880971497 CD On-Demand Anodyne TRPV1 18 48 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CO)C1CC1 ZINC000880971498 CD On-Demand Anodyne TRPV1 18 48 C[C@H]1CCC[C@H](C)N(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971501 DI On-Demand Anodyne RBP4 42 38 CCOC(=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971503 DE On-Demand Anodyne TRPV1 23 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC(F)(F)C(F)F)CC1 ZINC000880971505 GG On-Demand Mild RBP4 55 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](CCO)C1 ZINC000880971524 DE On-Demand Anodyne RBP4 77 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](CCO)C1 ZINC000880971525 DE On-Demand Anodyne RBP4 77 44 C[C@H](CCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971532 CD On-Demand Anodyne TRPV1 19 47 C[C@@H](CCO)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971533 CD On-Demand Anodyne TRPV1 19 47 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880971537 FF On-Demand Anodyne RBP4 59 40 CCc1nccn1[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971539 FH On-Demand Anodyne RBP4 55 38 CCc1nccn1[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971540 FH On-Demand Anodyne RBP4 55 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](CCO)C1CC1 ZINC000880971541 DE On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H](CCO)C1CC1 ZINC000880971542 DE On-Demand Anodyne TRPV1 15 46 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne TRPV1 31 47 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne P2RY1 81 45 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne RAF1 74 49 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne KDR 51 39 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne EPHX2 33 45 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne CA12 18 40 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne PDGFRA 47 36 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne TEK 47 39 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne CA9 18 40 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne BRAF 20 44 COCCOc1ccc(NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971546 FH On-Demand Anodyne MTCA1 15 40 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971549 GF On-Demand Anodyne TRPV1 19 44 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971549 GF On-Demand Anodyne SIGMAR1 15 40 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971549 GF On-Demand Anodyne NPFFR2 40 41 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971549 GF On-Demand Anodyne UTS2R 16 42 O=C(NC[C@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971549 GF On-Demand Anodyne NPFFR1 50 41 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971550 GF On-Demand Anodyne TRPV1 19 44 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971550 GF On-Demand Anodyne SIGMAR1 15 40 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971550 GF On-Demand Anodyne NPFFR2 40 41 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971550 GF On-Demand Anodyne UTS2R 16 42 O=C(NC[C@@]1(O)CCN(Cc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971550 GF On-Demand Anodyne NPFFR1 50 41 C[C@@](O)(CNC(=O)Nc1cnccc1C(F)(F)F)c1cccs1 ZINC000880971556 EG On-Demand Anodyne TRPV1 17 44 O=C(NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)c1ccsc1 ZINC000880971558 GH On-Demand Anodyne RBP4 59 40 C[C@@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(C)(C)O1 ZINC000880971559 DG On-Demand Anodyne RBP4 56 41 C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CC(C)(C)O1 ZINC000880971560 DG On-Demand Anodyne RBP4 56 41 O=C(NCC1CCN(Cc2cccs2)CC1)Nc1cnccc1C(F)(F)F ZINC000880971563 GI On-Demand Anodyne CCR3 27 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C(=O)N2CCCC2)CC1 ZINC000880971568 GD On-Demand Anodyne TRPV1 16 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C(=O)N2CCCC2)CC1 ZINC000880971568 GD On-Demand Anodyne RBP4 61 44 CCC[C@@H](CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971573 CH On-Demand Anodyne TRPV1 16 48 CCC[C@H](CC)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971574 CH On-Demand Anodyne TRPV1 16 48 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne MAPK11 31 41 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne MAPK14 40 43 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne TRPV1 37 54 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne RAF1 32 41 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne MAPK13 55 35 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne ROCK2 43 39 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne CCR2 58 39 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne EPHX2 15 45 O=C(NCc1cccc(C(=O)NC2CC2)c1)Nc1cnccc1C(F)(F)F ZINC000880971580 GG On-Demand Anodyne NAMPT 55 40 O=C(NCCOC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880971583 DG On-Demand Anodyne TRPV1 20 45 Cc1ccc(C(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)s1 ZINC000880971585 GG On-Demand Anodyne RBP4 60 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CC(F)F)CC1 ZINC000880971590 EF On-Demand Anodyne RBP4 57 42 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(N2CCOCC2)cc1 ZINC000880971592 GH On-Demand Clean STAT6 46 31 CCN(Cc1ccc(OC)cc1OC)C(=O)Nc1cnccc1C(F)(F)F ZINC000880971601 GI On-Demand Anodyne RAF1 15 40 CCOC(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971604 FF On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](OCC(F)(F)F)C1 ZINC000880971605 FH On-Demand Anodyne RBP4 59 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](OCC(F)(F)F)C1 ZINC000880971606 FH On-Demand Anodyne RBP4 59 42 O=C(NCCO)Nc1cnccc1C(F)(F)F ZINC000880971611 BD On-Demand Anodyne TRPV1 23 51 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971613 DE On-Demand Anodyne RBP4 79 44 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971613 DE On-Demand Anodyne SFRP1 79 39 COC(=O)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971613 DE On-Demand Anodyne WNT3 67 33 COC(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971614 DE On-Demand Anodyne RBP4 79 44 COC(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971614 DE On-Demand Anodyne SFRP1 79 39 COC(=O)[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971614 DE On-Demand Anodyne WNT3 67 33 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)Cn1cccn1 ZINC000880971616 EF On-Demand Anodyne TRPV1 17 43 O=C(NCCCOC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880971619 EH On-Demand Anodyne TRPV1 15 44 COC(=O)CCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971622 EF On-Demand Anodyne TRPV1 18 46 O=C(Cn1cc(-c2cnccc2Cl)nn1)NC1CCCCCCC1 ZINC000880971623 EG On-Demand Anodyne CNR1 17 44 CC[C@H](C)NC(=O)[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971629 EF On-Demand Anodyne TRPV1 15 48 CC[C@H](C)NC(=O)[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971630 EF On-Demand Anodyne TRPV1 15 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne DRD4 22 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne KCNH2 18 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne TRPV1 25 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne SIGMAR1 33 52 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne SSTR5 50 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne CCR3 99 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne CCR2 17 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne SLC6A5 31 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne EPHX2 44 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne CXCR3 31 45 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne MCHR1 62 51 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccc(F)cc2)CC1 ZINC000880971633 GI On-Demand Anodyne CACNA1G 44 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCNC2=O)CC1 ZINC000880971638 FE On-Demand Anodyne RBP4 66 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCNC2=O)CC1 ZINC000880971638 FE On-Demand Anodyne CALCRL 24 42 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCCCC1 ZINC000880971641 EG On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880971650 GG On-Demand Anodyne FAAH 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880971650 GG On-Demand Anodyne RBP4 86 46 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880971650 GG On-Demand Anodyne SCD1 15 45 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(C(=O)c2ccccc2)CC1 ZINC000880971650 GG On-Demand Anodyne SFRP1 37 41 COc1ccc2c(c1)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880971651 FH On-Demand Anodyne RBP4 49 37 CCN(Cc1ccccc1)C(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971652 GG On-Demand Anodyne TRPV1 21 48 CC(C)(C)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971654 EG On-Demand Anodyne TRPV1 28 40 CC(C)(C)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971654 EG On-Demand Anodyne EPHX2 48 45 CC(C)(C)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971654 EG On-Demand Anodyne SFRP1 72 35 CC(C)(C)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971654 EG On-Demand Anodyne WNT3 47 33 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971655 GD On-Demand Anodyne RBP4 59 41 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971655 GD On-Demand Anodyne SFRP1 56 33 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971655 GD On-Demand Anodyne WNT3 56 32 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971656 GD On-Demand Anodyne RBP4 59 41 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971656 GD On-Demand Anodyne SFRP1 56 33 CS(=O)(=O)NC[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971656 GD On-Demand Anodyne WNT3 56 32 O=C(Nc1cnccc1C(F)(F)F)N(Cc1cccnc1)C1CC1 ZINC000880971658 EH On-Demand Anodyne CHRNA7 41 40 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880971662 FH On-Demand Anodyne TRPV1 16 48 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)Cc2ccccc21 ZINC000880971662 FH On-Demand Anodyne RBP4 67 43 CC(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971663 EF On-Demand Anodyne TRPV1 15 41 CC(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971663 EF On-Demand Anodyne RBP4 73 43 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCC1 ZINC000880971664 EE On-Demand Anodyne CNR1 18 44 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCC1 ZINC000880971665 EE On-Demand Anodyne CNR1 18 44 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971666 FG On-Demand Anodyne RBP4 65 42 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971666 FG On-Demand Anodyne SFRP1 65 35 CC(C)(C)C(=O)N[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971666 FG On-Demand Anodyne WNT3 59 33 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971667 FG On-Demand Anodyne RBP4 65 42 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971667 FG On-Demand Anodyne SFRP1 65 35 CC(C)(C)C(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971667 FG On-Demand Anodyne WNT3 59 33 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC2CCCC2)nn1 ZINC000880971674 ED On-Demand Anodyne SIGMAR1 15 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCC1 ZINC000880971678 DD On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCC1 ZINC000880971679 DD On-Demand Anodyne SIGMAR1 15 43 O=C(NCCCc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880971682 EH On-Demand Anodyne TRPV1 31 55 O=C(NCCCc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880971682 EH On-Demand Anodyne CCR3 15 41 COc1ccc(N2CCCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880971684 GH On-Demand Clean RBP4 48 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCO)CC1 ZINC000880971686 DF On-Demand Anodyne EPHX2 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CCO)CC1 ZINC000880971686 DF On-Demand Anodyne RBP4 73 43 CN(C)CCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971687 GH On-Demand Anodyne TRPV1 15 50 CN(C)CCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971687 GH On-Demand Anodyne RAF1 23 42 CN(C)CCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971687 GH On-Demand Anodyne ROCK2 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCC2=O)C1 ZINC000880971694 FF On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCC2=O)C1 ZINC000880971695 FF On-Demand Anodyne RBP4 58 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)CC1 ZINC000880971696 EE On-Demand Anodyne TRPV1 22 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)CC1 ZINC000880971696 EE On-Demand Anodyne EPHX2 20 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)CC1 ZINC000880971696 EE On-Demand Anodyne RBP4 74 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CC2)CC1 ZINC000880971696 EE On-Demand Anodyne SFRP1 51 34 CCS(=O)(=O)C[C@@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971703 EE On-Demand Anodyne TRPV1 17 46 CCS(=O)(=O)C[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971704 EE On-Demand Anodyne TRPV1 17 46 CCOCCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971705 EE On-Demand Anodyne RBP4 50 38 CC(C)(C)[C@@H](O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971708 DF On-Demand Anodyne TRPV1 21 47 CCC(CC)[C@H](CNC(=O)Nc1cnccc1C(F)(F)F)N(C)C ZINC000880971711 EH On-Demand Anodyne TRPV1 15 45 CCC(CC)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N(C)C ZINC000880971712 EH On-Demand Anodyne TRPV1 15 45 CC[C@@H](C)[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971719 CH On-Demand Anodyne TRPV1 18 49 CC[C@H](C)[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971722 CH On-Demand Anodyne TRPV1 18 49 N#Cc1ccc(N2CCC(NC(=O)Nc3cnccc3C(F)(F)F)CC2)nc1 ZINC000880971727 GG On-Demand Mild HPGDS 24 41 CCC[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccccn1 ZINC000880971731 EI On-Demand Anodyne TRPV1 16 48 O=C(Cn1cc(-c2ccc(F)cn2)nn1)NC1CCCCCCC1 ZINC000880971733 EF On-Demand Anodyne SCARB1 31 40 N#C[C@H]1CN(C(=O)Nc2cnccc2C(F)(F)F)CCO1 ZINC000880971743 DD On-Demand Mild RBP4 61 43 O=C(NCC1(O)CCC1)Nc1cnccc1C(F)(F)F ZINC000880971746 CE On-Demand Anodyne TRPV1 20 49 O=C(Nc1cnccc1C(F)(F)F)N(CCc1ccccc1)C1CC1 ZINC000880971749 EI On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)N(CCc1ccccc1)C1CC1 ZINC000880971749 EI On-Demand Anodyne RBP4 49 40 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971757 FI On-Demand Anodyne TRPV1 17 43 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971757 FI On-Demand Anodyne SLC9A1 37 40 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971757 FI On-Demand Anodyne RBP4 111 54 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971757 FI On-Demand Anodyne SFRP1 41 32 O=C(CN1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971758 GD On-Demand Anodyne RBP4 55 41 COc1ccccc1[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971759 FI On-Demand Anodyne TRPV1 17 43 COc1ccccc1[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971759 FI On-Demand Anodyne SLC9A1 37 40 COc1ccccc1[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971759 FI On-Demand Anodyne RBP4 111 54 COc1ccccc1[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971759 FI On-Demand Anodyne SFRP1 41 32 O=C(NCCOCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880971762 DF On-Demand Anodyne TRPV1 21 45 CN(C)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971764 DE On-Demand Anodyne RBP4 84 46 CN(C)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971764 DE On-Demand Anodyne MCHR1 15 43 CN(C)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971764 DE On-Demand Anodyne SFRP1 64 35 CN(C)[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971764 DE On-Demand Anodyne WNT3 54 33 O=C(Cn1cc(CCCN2CCOCC2)nn1)NC1CCCC1 ZINC000880971767 DC On-Demand Anodyne EPHX2 16 45 C[C@H](O)CN(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880971773 FH On-Demand Anodyne TRPV1 15 41 CCCCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971774 FG On-Demand Anodyne RBP4 65 41 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971775 FD On-Demand Anodyne EPHX2 18 40 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971775 FD On-Demand Anodyne RBP4 69 43 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971775 FD On-Demand Anodyne SFRP1 124 40 CS(=O)(=O)N[C@@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971775 FD On-Demand Anodyne WNT3 85 37 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971776 FD On-Demand Anodyne EPHX2 18 40 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971776 FD On-Demand Anodyne RBP4 69 43 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971776 FD On-Demand Anodyne SFRP1 124 40 CS(=O)(=O)N[C@H]1CCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971776 FD On-Demand Anodyne WNT3 85 37 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCc2nc(O)ccc21 ZINC000880971777 FG On-Demand Anodyne TRPV1 35 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCc2nc(O)ccc21 ZINC000880971779 FG On-Demand Anodyne TRPV1 35 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CC2)CC1 ZINC000880971782 DE On-Demand Anodyne TRPV1 15 46 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CC2)CC1 ZINC000880971782 DE On-Demand Anodyne RBP4 70 45 CCN(CC)C(=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971784 EF On-Demand Anodyne TRPV1 16 45 O=C(NCc1nccn1CC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880971787 FG On-Demand Anodyne TRPV1 15 47 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccccc1)C1CC1 ZINC000880971792 EI On-Demand Anodyne TRPV1 24 44 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCC1 ZINC000880971793 FE On-Demand Anodyne CNR1 19 45 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCC1 ZINC000880971794 FE On-Demand Anodyne CNR1 19 45 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880971802 FF On-Demand Anodyne EPHX2 38 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880971802 FF On-Demand Anodyne CXCR3 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880971803 FH On-Demand Anodyne TRPV1 28 52 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880971803 FH On-Demand Anodyne EPHX2 41 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880971803 FH On-Demand Anodyne RBP4 65 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880971803 FH On-Demand Anodyne SFRP1 99 38 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(c2ccccc2)C1 ZINC000880971803 FH On-Demand Anodyne WNT3 63 34 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880971804 FF On-Demand Anodyne EPHX2 38 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880971804 FF On-Demand Anodyne CXCR3 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2)C1 ZINC000880971805 FH On-Demand Anodyne TRPV1 28 52 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2)C1 ZINC000880971805 FH On-Demand Anodyne EPHX2 41 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2)C1 ZINC000880971805 FH On-Demand Anodyne RBP4 65 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2)C1 ZINC000880971805 FH On-Demand Anodyne SFRP1 99 38 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(c2ccccc2)C1 ZINC000880971805 FH On-Demand Anodyne WNT3 63 34 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880971806 GG On-Demand Anodyne FAAH 28 53 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880971806 GG On-Demand Anodyne RBP4 48 39 O=C(Nc1cnccc1C(F)(F)F)N1[C@H]2CC[C@H]1CC(O)C2 ZINC000880971809 DF On-Demand Anodyne RBP4 48 40 O=C(Cn1cc(-c2cccnc2)nn1)NC1CCCCCCC1 ZINC000880971810 DF On-Demand Anodyne C3AR1 41 39 O=C(Cn1cc(-c2cccnc2)nn1)NC1CCCCCCC1 ZINC000880971810 DF On-Demand Anodyne FIMH 17 51 O=C(Cn1cc(-c2cccnc2)nn1)NC1CCCCCCC1 ZINC000880971810 DF On-Demand Anodyne VCP 51 35 O=C(NCCNc1nccc(C(F)(F)F)n1)Nc1cnccc1C(F)(F)F ZINC000880971811 GG On-Demand Anodyne TRPV1 18 44 CN(CCNC(=O)Nc1cnccc1C(F)(F)F)CC(F)(F)F ZINC000880971822 EF On-Demand Anodyne TRPV1 17 45 O=C(c1ccc(F)cc1)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971827 GI On-Demand Anodyne SLC18A3 16 40 O=C(c1ccc(F)cc1)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971827 GI On-Demand Anodyne RBP4 58 41 O=C(c1ccc(F)cc1)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971828 GI On-Demand Anodyne SLC18A3 16 40 O=C(c1ccc(F)cc1)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880971828 GI On-Demand Anodyne RBP4 58 41 O=C(NCC1(O)Cc2ccccc2C1)Nc1cnccc1C(F)(F)F ZINC000880971829 FF On-Demand Anodyne TRPV1 34 54 Cc1cc([C@@](C)(O)CNC(=O)Nc2cnccc2C(F)(F)F)c(C)o1 ZINC000880971831 FG On-Demand Anodyne TRPV1 19 43 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne ABL1 44 36 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne DRD2 15 43 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne DRD4 41 43 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne ACHE 47 46 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne LTA4H 19 46 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne SIGMAR1 45 50 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne CCR3 38 42 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne CCR5 20 45 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne ABL2 42 34 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne FAAH 23 49 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne CXCR3 15 42 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne RBP4 58 38 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne MCHR1 54 42 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne CACNA1G 33 43 CN(C(=O)Nc1cnccc1C(F)(F)F)C1CCN(Cc2ccccc2)CC1 ZINC000880971833 GI On-Demand Anodyne SFRP1 42 33 O=C(Nc1cnccc1C(F)(F)F)N1CCSC[C@H]1c1ccccc1 ZINC000880971835 FI On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CCSC[C@@H]1c1ccccc1 ZINC000880971836 FI On-Demand Anodyne RBP4 61 42 CCc1csc([C@@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880971838 GJ On-Demand Anodyne RBP4 60 40 CCc1csc([C@H]2CCCN(C(=O)Nc3cnccc3C(F)(F)F)C2)n1 ZINC000880971839 GJ On-Demand Anodyne RBP4 60 40 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c(F)c1 ZINC000880971865 GG On-Demand Mild NPY2R 41 38 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c(F)c1 ZINC000880971865 GG On-Demand Mild SLC6A9 22 44 N#Cc1ccc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c(F)c1 ZINC000880971865 GG On-Demand Mild RBP4 52 36 CN(C)CCOc1ccc(CCNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880971870 GG On-Demand Anodyne RAF1 33 52 CCCO[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971874 EH On-Demand Anodyne RBP4 62 40 CCCO[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971874 EH On-Demand Anodyne SFRP1 47 32 CCCO[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971874 EH On-Demand Anodyne WNT3 51 32 CCCO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971875 EH On-Demand Anodyne RBP4 62 40 CCCO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971875 EH On-Demand Anodyne SFRP1 47 32 CCCO[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971875 EH On-Demand Anodyne WNT3 51 32 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc2c(c1)OCO2 ZINC000880971877 GI On-Demand Anodyne NOS2 45 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc2c(c1)OCO2 ZINC000880971878 GI On-Demand Anodyne NOS2 45 33 Cc1cccc2c1CC[C@@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971879 EI On-Demand Anodyne TRPV1 42 58 Cc1cccc2c1CC[C@@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971879 EI On-Demand Anodyne RBP4 40 39 Cc1cccc2c1CC[C@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971880 EI On-Demand Anodyne TRPV1 42 58 Cc1cccc2c1CC[C@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971880 EI On-Demand Anodyne RBP4 40 39 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne ACHE 21 40 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne HTR4 19 43 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne TRPV1 18 41 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne SIGMAR1 19 41 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne CCR3 68 46 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne CCR2 27 42 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne RBP4 54 39 O=C(NC[C@@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971882 GH On-Demand Anodyne NAMPT 40 37 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne ACHE 21 40 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne HTR4 19 43 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne TRPV1 18 41 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne SIGMAR1 19 41 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne CCR3 68 46 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne CCR2 27 42 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne RBP4 54 39 O=C(NC[C@H]1CCN(CCc2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880971883 GH On-Demand Anodyne NAMPT 40 37 C=CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971885 EF On-Demand Mild EPHX2 41 41 C=CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971885 EF On-Demand Mild CXCR3 19 42 C[C@@H](c1cccc(O)c1)N(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880971887 EI On-Demand Anodyne TRPV1 18 43 Cn1cc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cn1 ZINC000880971893 FE On-Demand Anodyne ABL2 44 36 Cn1cc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cn1 ZINC000880971893 FE On-Demand Anodyne FAAH 20 50 Cn1cc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cn1 ZINC000880971893 FE On-Demand Anodyne RBP4 43 38 O=C(Cn1cc(-c2cncc(Cl)c2)nn1)NC1CCCCCCC1 ZINC000880971894 EG On-Demand Anodyne CNR1 15 46 C[C@@H](Cc1cccs1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880971898 EH On-Demand Anodyne TRPV1 15 45 O=C(NC[C@@H](O)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880971900 EG On-Demand Anodyne TRPV1 17 43 O=C(NC[C@@H](O)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880971900 EG On-Demand Anodyne PRMT3 26 48 O=C(NC[C@H](O)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880971901 EG On-Demand Anodyne TRPV1 17 43 O=C(NC[C@H](O)C1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880971901 EG On-Demand Anodyne PRMT3 26 48 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NC1CCCC1 ZINC000880971903 ED On-Demand Anodyne MMP8 25 45 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2cccc(F)c2)C1 ZINC000880971905 FH On-Demand Anodyne RBP4 59 41 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2cccc(F)c2)C1 ZINC000880971906 FH On-Demand Anodyne RBP4 59 41 Cc1ncc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)s1 ZINC000880971911 GG On-Demand Anodyne ABL1 41 34 Cc1ncc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)s1 ZINC000880971911 GG On-Demand Anodyne ABL2 42 33 Cc1ncc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)s1 ZINC000880971911 GG On-Demand Anodyne RBP4 45 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccc2c1OCCO2 ZINC000880971912 GI On-Demand Anodyne RBP4 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccc2c1OCCO2 ZINC000880971913 GI On-Demand Anodyne RBP4 53 38 COc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971920 GF On-Demand Anodyne TRPV1 17 44 COc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880971920 GF On-Demand Anodyne RBP4 53 48 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(O)cc2C1 ZINC000880971923 EG On-Demand Anodyne RBP4 57 41 O=C(Nc1cnccc1C(F)(F)F)N1CCCc2sccc2C1 ZINC000880971939 EI On-Demand Anodyne RBP4 59 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CCO)C1 ZINC000880971942 DF On-Demand Anodyne RBP4 67 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CCO)C1 ZINC000880971943 DF On-Demand Anodyne RBP4 67 43 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971947 DF On-Demand Anodyne TRPV1 23 43 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971947 DF On-Demand Anodyne CCR3 25 42 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971947 DF On-Demand Anodyne ABL2 40 37 CN1CCC(CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971947 DF On-Demand Anodyne CACNA1I 59 39 O=C(NCc1nccn1C(F)F)Nc1cnccc1C(F)(F)F ZINC000880971952 EG On-Demand Anodyne TRPV1 16 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880971969 GG On-Demand Anodyne TRPV1 18 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880971969 GG On-Demand Anodyne P2RX7 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880971969 GG On-Demand Anodyne SLC9A1 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880971969 GG On-Demand Anodyne EPHX2 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2cccc(F)c2)CC1 ZINC000880971969 GG On-Demand Anodyne RBP4 64 41 Cc1ncsc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880971970 DG On-Demand Anodyne TRPV1 18 48 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971976 GE On-Demand Anodyne RBP4 72 43 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971976 GE On-Demand Anodyne SFRP1 71 35 CCS(=O)(=O)N(C)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971976 GE On-Demand Anodyne WNT3 62 35 N#Cc1ccccc1N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971978 GH On-Demand Mild KCNQ2 44 33 N#Cc1ccccc1N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971978 GH On-Demand Mild TRPV1 15 54 N#Cc1ccccc1N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880971978 GH On-Demand Mild RBP4 58 43 O=C(NC[C@@H](O)COc1ccc(F)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880971983 GF On-Demand Anodyne ADRB1 43 34 O=C(NC[C@H](O)COc1ccc(F)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880971984 GF On-Demand Anodyne ADRB1 43 34 COc1ccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)cn1 ZINC000880971987 EF On-Demand Anodyne PDE5A 41 37 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H](N2CCCC2)C1 ZINC000880971989 FH On-Demand Anodyne RBP4 66 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@@H](N2CCCC2)C1 ZINC000880971989 FH On-Demand Anodyne L3MBTL3 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H](N2CCCC2)C1 ZINC000880971990 FH On-Demand Anodyne RBP4 66 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCC[C@H](N2CCCC2)C1 ZINC000880971990 FH On-Demand Anodyne L3MBTL3 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(N2CCCC2=O)CC1 ZINC000880971992 FF On-Demand Anodyne RBP4 66 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCOc2ccccc21 ZINC000880971993 FI On-Demand Anodyne TRPV1 33 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCOc2ccccc21 ZINC000880971993 FI On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCOc2ccccc21 ZINC000880971994 FI On-Demand Anodyne TRPV1 33 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCOc2ccccc21 ZINC000880971994 FI On-Demand Anodyne RBP4 57 42 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(O)cc2CC1 ZINC000880971998 FG On-Demand Anodyne TRPV1 16 41 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccc(O)cc2CC1 ZINC000880971998 FG On-Demand Anodyne RBP4 59 42 C[C@H]1CC[C@@H](C)N1CCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972003 GG On-Demand Anodyne RBP4 58 40 C[C@H]1CC[C@H](C)N1CCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972004 GG On-Demand Anodyne RBP4 58 40 C[C@@H]1CC[C@@H](C)N1CCN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972005 GG On-Demand Anodyne RBP4 58 40 O=C(CC1CCCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972009 GH On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CN1CCCC1 ZINC000880972010 EG On-Demand Anodyne SFRP1 70 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1CN1CCCC1 ZINC000880972010 EG On-Demand Anodyne WNT3 71 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CN1CCCC1 ZINC000880972011 EG On-Demand Anodyne SFRP1 70 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1CN1CCCC1 ZINC000880972011 EG On-Demand Anodyne WNT3 71 36 CCc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880972012 EG On-Demand Anodyne TRPV1 21 49 O=C(NCCCN1CCCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880972013 EF On-Demand Anodyne CCR3 20 43 O=C(NCCCN1CCCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880972013 EF On-Demand Anodyne TYRO3 20 40 CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972016 EH On-Demand Anodyne TRPV1 29 57 CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972016 EH On-Demand Anodyne P2RY1 41 39 CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972016 EH On-Demand Anodyne CARM1 15 40 CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972016 EH On-Demand Anodyne KCNK3 20 44 CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972016 EH On-Demand Anodyne KCNK9 19 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCCC2)C1 ZINC000880972018 EG On-Demand Anodyne RBP4 71 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCCC2)C1 ZINC000880972018 EG On-Demand Anodyne SFRP1 44 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](N2CCCCC2)C1 ZINC000880972018 EG On-Demand Anodyne L3MBTL3 87 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCCC2)C1 ZINC000880972019 EG On-Demand Anodyne RBP4 71 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCCC2)C1 ZINC000880972019 EG On-Demand Anodyne SFRP1 44 33 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](N2CCCCC2)C1 ZINC000880972019 EG On-Demand Anodyne L3MBTL3 87 43 C[C@H](O)c1ccc(OCc2cn(CC(=O)NC3CCCCCCC3)nn2)cc1 ZINC000880972020 GG On-Demand Anodyne SCARB1 40 39 O=C(NC[C@@H](O)c1ccccc1C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880972027 GH On-Demand Anodyne TRPV1 22 52 O=C(NC[C@@H](O)c1ccccc1C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880972027 GH On-Demand Anodyne SOAT1 15 43 O=C(NC[C@H](O)c1ccccc1C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880972028 GH On-Demand Anodyne TRPV1 22 52 O=C(NC[C@H](O)c1ccccc1C(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880972028 GH On-Demand Anodyne SOAT1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(n2ccnc2)CC1 ZINC000880972029 EG On-Demand Anodyne RBP4 67 41 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCC1 ZINC000880972036 EE On-Demand Anodyne TRPV1 23 44 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCC1 ZINC000880972036 EE On-Demand Anodyne CCR2 43 40 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCC1 ZINC000880972036 EE On-Demand Anodyne EPHX2 22 46 Cc1cc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)on1 ZINC000880972039 EH On-Demand Anodyne RBP4 46 36 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972040 GG On-Demand Clean TRPV1 23 48 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972040 GG On-Demand Clean NPY2R 45 34 O=C(NCc1ccc(N2CCOCC2)c(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972040 GG On-Demand Clean NAMPT 55 39 O=C(NCc1nc(C2CC2)no1)Nc1cnccc1C(F)(F)F ZINC000880972045 EF On-Demand Anodyne TRPV1 21 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne SIGMAR1 15 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne SLC6A5 28 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne EPHX2 49 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne CXCR3 20 53 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC2CC2)CC1 ZINC000880972046 EG On-Demand Anodyne SFRP1 47 34 O=C(NCC1CC1)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972048 FF On-Demand Anodyne RBP4 62 42 O=C(NCC1CC1)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972049 FF On-Demand Anodyne RBP4 62 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1C1CCCC1 ZINC000880972050 EI On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1C1CCCC1 ZINC000880972051 EI On-Demand Anodyne RBP4 56 41 O=C(Nc1cnccc1C(F)(F)F)N1CCOc2ccccc2C1 ZINC000880972052 EH On-Demand Anodyne RBP4 58 42 COCCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972059 DG On-Demand Anodyne TRPV1 18 44 O=C(Nc1cnccc1C(F)(F)F)N(CCO)Cc1ccccc1 ZINC000880972069 EG On-Demand Anodyne TRPV1 15 43 CCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972070 FH On-Demand Anodyne TRPV1 35 52 CCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972070 FH On-Demand Anodyne P2RY1 48 41 CCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972070 FH On-Demand Anodyne SCN10A 20 42 N[C@@H](c1ccc(F)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972071 FF On-Demand Anodyne SCARB1 28 40 N[C@H](c1ccc(F)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972072 FF On-Demand Anodyne SCARB1 28 40 CCN(Cc1ccc(OC)cc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880972077 FI On-Demand Anodyne ROCK2 21 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccc(F)c1 ZINC000880972078 FJ On-Demand Anodyne RBP4 53 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccc(F)c1 ZINC000880972078 FJ On-Demand Anodyne SFRP1 44 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccc(F)c1 ZINC000880972078 FJ On-Demand Anodyne WNT3 43 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccc(F)c1 ZINC000880972079 FJ On-Demand Anodyne RBP4 53 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccc(F)c1 ZINC000880972079 FJ On-Demand Anodyne SFRP1 44 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccc(F)c1 ZINC000880972079 FJ On-Demand Anodyne WNT3 43 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCc2occc21 ZINC000880972081 EH On-Demand Anodyne TRPV1 25 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCc2occc21 ZINC000880972082 EH On-Demand Anodyne TRPV1 25 42 O=C(Nc1cnn(C[C@H]2CCCO2)c1)Nc1cnccc1C(F)(F)F ZINC000880972083 FG On-Demand Anodyne PANC 51 34 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)Nc1cnccc1C(F)(F)F ZINC000880972084 FG On-Demand Anodyne PANC 51 34 C[C@@H](Cc1ccc(O)cc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880972087 EH On-Demand Anodyne TRPV1 20 44 C[C@@H](Cc1ccc(O)cc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880972087 EH On-Demand Anodyne GRIA1 42 35 CC(C)(C)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972097 EG On-Demand Anodyne RBP4 57 41 Cc1ccc([C@@H](C)NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880972098 DI On-Demand Anodyne TRPV1 15 60 Cc1ccc([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880972099 DI On-Demand Anodyne TRPV1 15 60 NCc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880972103 EF On-Demand Anodyne HDAC10 20 40 NCc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880972103 EF On-Demand Anodyne HDAC3 19 40 NCc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880972103 EF On-Demand Anodyne HDAC6 16 40 NCc1cccc(-c2cn(CC(=O)NC3CCCCCCC3)nn2)c1 ZINC000880972103 EF On-Demand Anodyne FAAH 26 42 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972105 FF On-Demand Anodyne ADRB2 15 42 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972105 FF On-Demand Anodyne ADRB1 53 36 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972105 FF On-Demand Anodyne TRPV1 20 43 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972105 FF On-Demand Anodyne P2RY1 15 41 O=C(NC[C@@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972105 FF On-Demand Anodyne PDS 43 38 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972106 FF On-Demand Anodyne ADRB2 15 42 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972106 FF On-Demand Anodyne ADRB1 53 36 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972106 FF On-Demand Anodyne TRPV1 20 43 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972106 FF On-Demand Anodyne P2RY1 15 41 O=C(NC[C@H](O)COc1cccc(F)c1)Nc1cnccc1C(F)(F)F ZINC000880972106 FF On-Demand Anodyne PDS 43 38 O=C(NCCCNc1ccccn1)Nc1cnccc1C(F)(F)F ZINC000880972110 EG On-Demand Anodyne TRPV1 22 49 O=C(CCNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCCC1 ZINC000880972113 FG On-Demand Anodyne TRPV1 32 47 O=C(CCNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCCC1 ZINC000880972113 FG On-Demand Anodyne EPHX2 25 47 O=C(NC[C@H]1Cc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880972121 DH On-Demand Anodyne TRPV1 23 47 O=C(NC[C@@H]1Cc2ccccc21)Nc1cnccc1C(F)(F)F ZINC000880972122 DH On-Demand Anodyne TRPV1 23 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)F)CC1 ZINC000880972123 FF On-Demand Anodyne EPHX2 47 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CC(F)F)CC1 ZINC000880972123 FF On-Demand Anodyne CXCR3 20 45 CN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972130 DE On-Demand Anodyne TRPV1 21 42 CN1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972130 DE On-Demand Anodyne EPHX2 40 45 CC[C@H](C)NC(=O)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972132 EF On-Demand Anodyne TRPV1 22 48 CN(C)C(=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972135 DE On-Demand Anodyne TRPV1 20 49 N#Cc1ccc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972137 GG On-Demand Mild FAAH 25 51 N#Cc1ccc(CN2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972137 GG On-Demand Mild RBP4 42 37 CS(=O)(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972138 GE On-Demand Anodyne SFRP1 49 34 CS(=O)(=O)NC[C@@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972138 GE On-Demand Anodyne WNT3 54 34 CS(=O)(=O)NC[C@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972139 GE On-Demand Anodyne SFRP1 49 34 CS(=O)(=O)NC[C@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972139 GE On-Demand Anodyne WNT3 54 34 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)c(OC)c1 ZINC000880972142 FH On-Demand Anodyne TSPO 41 33 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)c(OC)c1 ZINC000880972142 FH On-Demand Anodyne RAF1 19 41 O=C(NCCSC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880972145 EG On-Demand Anodyne TRPV1 17 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2ccccc2)CC1 ZINC000880972148 FH On-Demand Anodyne TRPV1 32 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2ccccc2)CC1 ZINC000880972148 FH On-Demand Anodyne EPHX2 49 45 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2ccccc2)CC1 ZINC000880972148 FH On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2ccccc2)CC1 ZINC000880972148 FH On-Demand Anodyne SFRP1 113 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(c2ccccc2)CC1 ZINC000880972148 FH On-Demand Anodyne WNT3 74 35 CC(C)(C)OC(=O)NCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972151 EF On-Demand Anodyne TRPV1 20 46 O=C(NCCCCOCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880972156 FI On-Demand Anodyne TRPV1 20 46 CN1CCN(c2ncccc2CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972178 GF On-Demand Anodyne TRPV1 63 52 CN1CCN(c2ncccc2CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972178 GF On-Demand Anodyne P2RX7 47 42 CN1CCN(c2ncccc2CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972178 GF On-Demand Anodyne SCN10A 25 40 CN1CCN(c2ncccc2CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972178 GF On-Demand Anodyne NAMPT 44 35 COc1ccc(C)cc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972179 EH On-Demand Anodyne TRPV1 25 50 COc1ccc(C)cc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972179 EH On-Demand Anodyne RAF1 27 40 CCN(CC)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972187 FG On-Demand Anodyne RBP4 66 40 O=C(NCc1ccc(CN2CCCC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880972190 GH On-Demand Anodyne TRPV1 20 49 O=C(NCc1ccc(CN2CCCC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880972190 GH On-Demand Anodyne NAMPT 70 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne TRPV1 19 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne FAAH 21 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne RBP4 55 39 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne SCD1 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne SCD 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(Cl)cn2)CC1 ZINC000880972191 GH On-Demand Anodyne DGAT1 23 44 N#Cc1c(F)cccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972192 GG On-Demand Mild RBP4 54 38 COC[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972197 CF On-Demand Anodyne TRPV1 18 47 COC[C@@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972198 CF On-Demand Anodyne TRPV1 18 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2cc(F)ccc21 ZINC000880972199 EI On-Demand Anodyne TRPV1 39 58 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2cc(F)ccc21 ZINC000880972200 EI On-Demand Anodyne TRPV1 39 58 O=C(NCCC(=O)N1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972205 FG On-Demand Anodyne TRPV1 23 48 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)C(=O)NC(C)(C)C ZINC000880972207 EF On-Demand Anodyne TRPV1 15 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880972208 GF On-Demand Anodyne TRPV1 15 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880972208 GF On-Demand Anodyne RBP4 81 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880972208 GF On-Demand Anodyne SCD1 21 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2O)CC1 ZINC000880972208 GF On-Demand Anodyne SCD 22 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne TRPV1 23 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne SLC9A1 29 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne EPHX2 61 56 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne RBP4 70 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne SFRP1 129 50 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne WNT3 84 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000880972209 GH On-Demand Anodyne L3MBTL3 41 32 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2)CC1 ZINC000880972213 FH On-Demand Anodyne TRPV1 21 52 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2)CC1 ZINC000880972213 FH On-Demand Anodyne FAAH 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2)CC1 ZINC000880972213 FH On-Demand Anodyne RBP4 73 46 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2ccccc2)CC1 ZINC000880972213 FH On-Demand Anodyne DGAT1 17 40 CCn1cc(NC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880972219 CF On-Demand Anodyne TRPV1 20 42 CCn1cc(NC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880972219 CF On-Demand Anodyne BRAF 15 40 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCCC1 ZINC000880972220 EF On-Demand Anodyne TRPV1 22 43 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCCC1 ZINC000880972220 EF On-Demand Anodyne CCR2 41 39 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CCCCC1 ZINC000880972220 EF On-Demand Anodyne EPHX2 24 48 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972222 EE On-Demand Anodyne RBP4 61 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1COc2ccccc2C1 ZINC000880972223 EG On-Demand Anodyne TRPV1 22 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1COc2ccccc2C1 ZINC000880972224 EG On-Demand Anodyne TRPV1 22 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCCC2)CC1 ZINC000880972236 GG On-Demand Anodyne EPHX2 21 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCCC2)CC1 ZINC000880972236 GG On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCCC2)CC1 ZINC000880972236 GG On-Demand Anodyne SFRP1 74 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(C(=O)N2CCCCC2)CC1 ZINC000880972236 GG On-Demand Anodyne WNT3 64 35 NC(=O)c1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880972238 GG On-Demand Anodyne GCGR 25 41 NC(=O)c1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880972238 GG On-Demand Anodyne GIPR 39 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CTSB 34 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CTSK 28 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CTSL 32 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne PREP 30 44 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CAPNS1 42 32 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CAPN1 53 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne CAPN2 94 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne EPHX2 17 42 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972246 GF On-Demand Anodyne NPR 59 32 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)cc1 ZINC000880972247 FH On-Demand Anodyne TRPV1 15 49 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccc(F)cc1 ZINC000880972256 EI On-Demand Anodyne TRPV1 24 50 COCCN(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880972258 FH On-Demand Anodyne ROCK2 20 40 N[C@@H](c1ccc(Cl)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972264 GG On-Demand Anodyne CNR1 22 45 N[C@@H](c1ccc(Cl)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972264 GG On-Demand Anodyne SCARB1 28 41 N[C@H](c1ccc(Cl)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972265 GG On-Demand Anodyne CNR1 22 45 N[C@H](c1ccc(Cl)cc1)c1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972265 GG On-Demand Anodyne SCARB1 28 41 COc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972266 GI On-Demand Anodyne EPHX2 40 38 COc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972266 GI On-Demand Anodyne RBP4 67 43 COc1ccc(OC2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972266 GI On-Demand Anodyne SCD1 28 43 N[C@H](Cc1ccccc1)Cc1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972269 FF On-Demand Anodyne OPRM1 30 40 N[C@H](Cc1ccccc1)Cc1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972269 FF On-Demand Anodyne SCARB1 32 41 N[C@@H](Cc1ccccc1)Cc1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972270 FF On-Demand Anodyne OPRM1 30 40 N[C@@H](Cc1ccccc1)Cc1cn(CC(=O)NC2CCCCCCC2)nn1 ZINC000880972270 FF On-Demand Anodyne SCARB1 32 41 CC(C)(C)CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972276 CH On-Demand Anodyne TRPV1 23 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(CCc2cccs2)CC1 ZINC000880972278 GH On-Demand Anodyne RBP4 55 39 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972281 FD On-Demand Anodyne TRPV1 16 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972281 FD On-Demand Anodyne EPHX2 44 42 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972281 FD On-Demand Anodyne SFRP1 72 33 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972281 FD On-Demand Anodyne WNT3 55 33 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972287 GH On-Demand Anodyne EPHX2 56 53 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972287 GH On-Demand Anodyne SFRP1 51 33 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)N2CCCCC2)CC1 ZINC000880972289 GF On-Demand Anodyne RBP4 59 43 COc1cc2c(cc1OC)CCN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880972296 GH On-Demand Anodyne RBP4 60 47 O=C(Cn1cc(CNCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972300 FF On-Demand Anodyne SIGMAR1 16 46 O=C(Cn1cc(CNCc2ccccc2)nn1)NC1CCCCCCC1 ZINC000880972300 FF On-Demand Anodyne EPHX2 15 46 O=C(NCCOC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972307 EH On-Demand Anodyne TRPV1 19 44 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880972309 EG On-Demand Anodyne TRPV1 16 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2c(F)cccc21 ZINC000880972314 EI On-Demand Anodyne TRPV1 40 56 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCc2c(F)cccc21 ZINC000880972314 EI On-Demand Anodyne RBP4 48 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2c(F)cccc21 ZINC000880972315 EI On-Demand Anodyne TRPV1 40 56 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCc2c(F)cccc21 ZINC000880972315 EI On-Demand Anodyne RBP4 48 40 CCOCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972316 DG On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne TRPV1 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne EPHX2 28 51 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne RBP4 108 53 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne ADAM10 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne SFRP1 96 37 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne SMO 33 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@@H](c2ccccc2)C1 ZINC000880972319 EI On-Demand Anodyne WNT3 80 36 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne TRPV1 19 43 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne EPHX2 28 51 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne RBP4 108 53 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne ADAM10 19 41 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne SFRP1 96 37 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne SMO 33 45 O=C(Nc1cnccc1C(F)(F)F)N1CC[C@H](c2ccccc2)C1 ZINC000880972320 EI On-Demand Anodyne WNT3 80 36 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CCCCC2)CC1 ZINC000880972324 GG On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CCCCC2)CC1 ZINC000880972324 GG On-Demand Anodyne EPHX2 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CCCCC2)CC1 ZINC000880972324 GG On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CCCCC2)CC1 ZINC000880972324 GG On-Demand Anodyne SFRP1 57 36 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)C2CCCCC2)CC1 ZINC000880972324 GG On-Demand Anodyne WNT3 51 36 C[C@@H](Cc1ccccc1F)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880972327 EH On-Demand Anodyne TRPV1 25 50 C[C@H](Cc1ccccc1F)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880972328 EH On-Demand Anodyne TRPV1 25 50 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)CN1CCCC1 ZINC000880972341 EF On-Demand Anodyne TRPV1 17 42 O=C(NCC(F)(F)F)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972350 GG On-Demand Anodyne RBP4 69 41 O=C(NCC(F)(F)F)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972350 GG On-Demand Anodyne SFRP1 42 33 O=C(Cn1cc(CN2C(=O)C(=O)c3ccccc32)nn1)NC1CCCCCCC1 ZINC000880972351 GE On-Demand Anodyne CASP3 15 41 O=C(Cn1cc(CN2C(=O)C(=O)c3ccccc32)nn1)NC1CCCCCCC1 ZINC000880972351 GE On-Demand Anodyne ALDH1A1 45 39 O=C(Cn1cc(CN2C(=O)C(=O)c3ccccc32)nn1)NC1CCCCCCC1 ZINC000880972351 GE On-Demand Anodyne CASP7 15 41 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880972360 GH On-Demand Anodyne TRPV1 18 50 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880972360 GH On-Demand Anodyne MLYCD 18 42 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880972360 GH On-Demand Anodyne NAMPT 93 58 CCC(=O)N1CCCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972361 EF On-Demand Anodyne RBP4 58 41 C[C@@H]1C[C@@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972364 CF On-Demand Anodyne TRPV1 25 46 C[C@@H]1C[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972366 CF On-Demand Anodyne TRPV1 25 46 C[C@H]1C[C@H]1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972367 CF On-Demand Anodyne TRPV1 25 46 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880972368 FF On-Demand Anodyne ADRB2 22 40 O=C(NC[C@@H](O)COc1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880972368 FF On-Demand Anodyne ADRB1 55 40 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880972369 FF On-Demand Anodyne ADRB2 22 40 O=C(NC[C@H](O)COc1ccc(F)cc1)Nc1cnccc1C(F)(F)F ZINC000880972369 FF On-Demand Anodyne ADRB1 55 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880972370 GI On-Demand Anodyne TRPV1 19 45 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880972370 GI On-Demand Anodyne RBP4 45 37 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880972371 GI On-Demand Anodyne TRPV1 19 45 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880972371 GI On-Demand Anodyne RBP4 45 37 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972374 FF On-Demand Anodyne RBP4 58 42 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880972375 FF On-Demand Anodyne RBP4 58 42 CN(C)CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972379 GG On-Demand Anodyne TRPV1 21 52 CN(C)CCOc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972379 GG On-Demand Anodyne ROCK2 18 42 Cc1ccc(C(=O)N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)cc1 ZINC000880972386 GG On-Demand Anodyne RBP4 61 41 O=C(NCC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880972391 CG On-Demand Anodyne TRPV1 26 47 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880972398 GI On-Demand Anodyne TRPV1 36 54 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880972398 GI On-Demand Anodyne CARM1 53 34 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880972398 GI On-Demand Anodyne NAMPT 44 38 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880972398 GI On-Demand Anodyne PDS 52 35 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2nccs2)CC1 ZINC000880972400 FG On-Demand Anodyne TRPV1 16 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(c2nccs2)CC1 ZINC000880972400 FG On-Demand Anodyne RBP4 50 37 O=C(CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)N1CCCC1 ZINC000880972409 GG On-Demand Anodyne RBP4 69 41 O=C(CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)N1CCCC1 ZINC000880972409 GG On-Demand Anodyne SFRP1 47 38 O=C(CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)N1CCCC1 ZINC000880972409 GG On-Demand Anodyne WNT3 48 33 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCCC1 ZINC000880972411 GG On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCCC1 ZINC000880972411 GG On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCCC1 ZINC000880972412 GG On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCCC1 ZINC000880972412 GG On-Demand Anodyne SCARB1 29 41 CNC(=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972417 DD On-Demand Anodyne TRPV1 18 47 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880972423 GH On-Demand Anodyne SOAT1 49 40 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880972424 GH On-Demand Anodyne SOAT1 49 40 C=C[C@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972439 ED On-Demand Mild ENPP1 87 41 C=C[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972440 ED On-Demand Mild ENPP1 87 41 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972442 CD On-Demand Anodyne TRPV1 21 48 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972442 CD On-Demand Anodyne RBP4 71 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@@H](O)c1ccco1 ZINC000880972444 EH On-Demand Anodyne SOAT1 15 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@@H](O)c1ccco1 ZINC000880972444 EH On-Demand Anodyne CCR2 20 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@H](O)c1ccco1 ZINC000880972445 EH On-Demand Anodyne SOAT1 15 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@H](O)c1ccco1 ZINC000880972445 EH On-Demand Anodyne CCR2 20 42 COC[C@@H](O)Cc1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880972448 ED On-Demand Anodyne SOAT1 36 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne TBXAS1 39 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne PTAFR 25 46 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne TRPV1 16 52 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne CHRNA7 18 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne RAF1 26 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1cccnc1 ZINC000880972452 EI On-Demand Anodyne NAMPT 49 45 C=C[C@@](C)(O)c1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880972457 EF On-Demand Mild SOAT1 31 40 C=C[C@](C)(O)c1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880972458 EF On-Demand Mild SOAT1 31 40 CC[C@@](C)(O)c1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880972461 EF On-Demand Anodyne SOAT1 45 45 COC(=O)N1CCC(NC(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880972470 FH On-Demand Anodyne EPHX2 60 53 COC(=O)N1CCC(NC(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880972470 FH On-Demand Anodyne CXCR3 15 51 CCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972495 CG On-Demand Anodyne TRPV1 24 47 CCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972495 CG On-Demand Anodyne ASAH1 81 40 O=C(NCCCO)Nc1cnccc1C(F)(F)F ZINC000880972520 CD On-Demand Anodyne TRPV1 21 49 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NCCCc1ccccc1 ZINC000880972528 FE On-Demand Anodyne AMP1_PLAFQ 21 40 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NCCCc1ccccc1 ZINC000880972529 FE On-Demand Anodyne AMP1_PLAFQ 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(O)cc2)CC1 ZINC000880972530 FG On-Demand Anodyne TRPV1 18 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(O)cc2)CC1 ZINC000880972530 FG On-Demand Anodyne RBP4 60 43 NOCc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880972531 CC On-Demand Anodyne SCNN1A 42 38 COCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972538 CE On-Demand Anodyne TRPV1 20 46 Nc1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972553 FE On-Demand Anodyne HRH2 42 38 Nc1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972553 FE On-Demand Anodyne SCNN1A 46 36 Nc1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972553 FE On-Demand Anodyne MTNR1A 16 41 Nc1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972553 FE On-Demand Anodyne MTNR1B 17 41 Nc1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972553 FE On-Demand Anodyne CRTM 40 40 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](O)c2ccccc2)nn1 ZINC000880972554 FG On-Demand Anodyne SOAT1 64 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](O)c2ccccc2)nn1 ZINC000880972555 FG On-Demand Anodyne SOAT1 64 41 CC(C)(C)OC(=O)NCc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880972625 FE On-Demand Anodyne TACR3 15 41 CC(C)(C)OC(=O)NCc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880972625 FE On-Demand Anodyne GHSR 20 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(C(=O)NCC(C)C)CC1 ZINC000880972635 GI On-Demand Anodyne EPHX2 34 47 CC[C@H](O)c1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880972649 DF On-Demand Anodyne SOAT1 46 44 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972657 ED On-Demand Anodyne PDGFRB 28 41 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972657 ED On-Demand Anodyne FLT4 28 41 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972657 ED On-Demand Anodyne ENPP1 86 41 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972657 ED On-Demand Anodyne DRTS_TRYCR 43 30 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(Cl)cc3)nn2)CC1 ZINC000880972660 GD On-Demand Anodyne FAAH 17 46 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880972714 GH On-Demand Anodyne SOAT1 52 42 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880972715 GH On-Demand Anodyne SOAT1 52 42 Nc1ccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)cc1 ZINC000880972728 FE On-Demand Clean SCNN1A 65 37 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3c(C)cccc3C(C)C)nn2)CC1 ZINC000880972734 GE On-Demand Anodyne SOAT1 21 40 COC(=O)C1CCC(c2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880972735 GE On-Demand Anodyne PREP 35 42 COC(=O)C1CCC(c2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880972735 GE On-Demand Anodyne MTNR1A 23 40 COC(=O)C1CCC(c2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880972735 GE On-Demand Anodyne MTNR1B 22 40 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880972740 GF On-Demand Anodyne SOAT1 23 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(CCCCCCO)nn1 ZINC000880972768 FG On-Demand Anodyne SOAT1 47 48 CC(=O)c1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972782 GF On-Demand Anodyne HRH2 43 38 CC(=O)c1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972782 GF On-Demand Anodyne MTNR1A 28 42 CC(=O)c1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972782 GF On-Demand Anodyne MTNR1B 31 42 CC(=O)c1cccc(OCc2cn(CC(=O)NCCCc3ccccc3)nn2)c1 ZINC000880972782 GF On-Demand Anodyne CRTM 44 39 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2C1 ZINC000880972801 DH On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2C1 ZINC000880972801 DH On-Demand Anodyne RBP4 71 45 O=C(Nc1cnccc1C(F)(F)F)N1CCc2ccccc2C1 ZINC000880972801 DH On-Demand Anodyne TRPM8 39 41 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)NCCCc1ccccc1 ZINC000880972806 FE On-Demand Anodyne AMP1_PLAFQ 20 40 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)NCCCc1ccccc1 ZINC000880972807 FE On-Demand Anodyne AMP1_PLAFQ 20 40 CC[C@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972808 DH On-Demand Anodyne WNT3 41 33 CC[C@@H]1CCCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880972809 DH On-Demand Anodyne WNT3 41 33 O=C(NCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880972819 CE On-Demand Anodyne TBXAS1 43 47 O=C(NCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880972819 CE On-Demand Anodyne QPCT 34 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne GRIN2B 32 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne TRPV1 18 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne FAAH 17 47 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne EPHX2 29 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne TGM2 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne RBP4 87 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne F13A1 27 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne LIPG 43 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne SFRP1 79 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne SCD 39 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(OCc2ccccc2)CC1 ZINC000880972825 GI On-Demand Anodyne WNT3 63 33 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N1CCC[C@@H](C)C1 ZINC000880972833 EG On-Demand Anodyne TRPV1 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccncc1 ZINC000880972841 EH On-Demand Anodyne RBP4 47 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccncc1 ZINC000880972842 EH On-Demand Anodyne RBP4 47 39 CC(=O)NCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972845 DD On-Demand Anodyne TRPV1 22 50 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880972850 GF On-Demand Anodyne TRPV1 18 46 O=C(NCc1ccnc(N2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880972850 GF On-Demand Anodyne NAMPT 49 41 O=C(NCCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880972851 DF On-Demand Anodyne TBXAS1 48 54 O=C(NCCCn1ccnc1)Nc1cnccc1C(F)(F)F ZINC000880972851 DF On-Demand Anodyne QPCT 55 55 O=C(NCCCOC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972852 EH On-Demand Anodyne TRPV1 15 43 O=C(NCCC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880972856 DH On-Demand Anodyne TRPV1 25 46 O=C(NCCC1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880972856 DH On-Demand Anodyne PRMT3 18 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880972857 FF On-Demand Anodyne TRPV1 29 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880972857 FF On-Demand Anodyne PIM1 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880972857 FF On-Demand Anodyne EPHX2 33 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCCN(c2ncccn2)C1 ZINC000880972857 FF On-Demand Anodyne RBP4 43 39 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880972858 FF On-Demand Anodyne TRPV1 29 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880972858 FF On-Demand Anodyne PIM1 18 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880972858 FF On-Demand Anodyne EPHX2 33 45 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCCN(c2ncccn2)C1 ZINC000880972858 FF On-Demand Anodyne RBP4 43 39 CCOC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972861 FF On-Demand Anodyne EPHX2 61 50 CCOC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972861 FF On-Demand Anodyne CXCR3 16 45 CCOC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972861 FF On-Demand Anodyne CCR8 30 43 CCOC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972861 FF On-Demand Anodyne SFRP1 64 34 CCOC(=O)N1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972861 FF On-Demand Anodyne WNT3 51 32 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne TRPV1 23 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne EPHX2 31 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne RBP4 108 54 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne SFRP1 95 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne SMO 33 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2ccccc2)CC1 ZINC000880972862 EJ On-Demand Anodyne WNT3 75 35 COC(=O)Cc1cn(CC(=O)NC[C@@H]2CCCO2)nn1 ZINC000880972863 CB On-Demand Anodyne PDE8B 21 40 COC(=O)Cc1cn(CC(=O)NC[C@H]2CCCO2)nn1 ZINC000880972864 CB On-Demand Anodyne PDE8B 21 40 C[C@@H](Cn1cccn1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880972867 DF On-Demand Anodyne TRPV1 16 45 O=C(NC[C@H]1CCN(CC(F)(F)F)C1)Nc1cnccc1C(F)(F)F ZINC000880972869 FG On-Demand Anodyne CCR3 29 42 O=C(NC[C@@H]1CCN(CC(F)(F)F)C1)Nc1cnccc1C(F)(F)F ZINC000880972870 FG On-Demand Anodyne CCR3 29 42 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880972872 FG On-Demand Anodyne TRPV1 21 47 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880972872 FG On-Demand Anodyne SCD1 15 44 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880972872 FG On-Demand Anodyne SCD 15 44 O=C(NCc1ccc(N2CCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880972872 FG On-Demand Anodyne NAMPT 72 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972875 FG On-Demand Anodyne TRPV1 18 47 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972875 FG On-Demand Anodyne RBP4 57 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972875 FG On-Demand Anodyne F13A1 24 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972875 FG On-Demand Anodyne GPR119 38 45 CCOC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972876 EF On-Demand Anodyne RBP4 67 41 CCOC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972876 EF On-Demand Anodyne PTR1 44 32 COc1cccc([C@H](CNC(=O)Nc2cnccc2C(F)(F)F)N(C)C)c1 ZINC000880972879 GH On-Demand Anodyne TRPV1 24 46 COc1cccc([C@H](CNC(=O)Nc2cnccc2C(F)(F)F)N(C)C)c1 ZINC000880972879 GH On-Demand Anodyne ROCK2 43 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCC2)C1 ZINC000880972882 EG On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCC2)C1 ZINC000880972882 EG On-Demand Anodyne SFRP1 41 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](N2CCCC2)C1 ZINC000880972882 EG On-Demand Anodyne L3MBTL3 53 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCC2)C1 ZINC000880972883 EG On-Demand Anodyne RBP4 67 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCC2)C1 ZINC000880972883 EG On-Demand Anodyne SFRP1 41 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](N2CCCC2)C1 ZINC000880972883 EG On-Demand Anodyne L3MBTL3 53 38 O=C(NC[C@H]1CN(Cc2ccccc2)CCO1)Nc1cnccc1C(F)(F)F ZINC000880972889 GG On-Demand Anodyne DRD4 20 44 O=C(NC[C@H]1CN(Cc2ccccc2)CCO1)Nc1cnccc1C(F)(F)F ZINC000880972889 GG On-Demand Anodyne TRPV1 16 40 O=C(NC[C@@H]1CN(Cc2ccccc2)CCO1)Nc1cnccc1C(F)(F)F ZINC000880972890 GG On-Demand Anodyne DRD4 20 44 O=C(NC[C@@H]1CN(Cc2ccccc2)CCO1)Nc1cnccc1C(F)(F)F ZINC000880972890 GG On-Demand Anodyne TRPV1 16 40 O=C(NCC1(c2ccccc2)CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880972893 GH On-Demand Anodyne TRPV1 18 48 O=C(NCCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972894 EG On-Demand Anodyne HRH2 25 43 O=C(NCCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972894 EG On-Demand Anodyne TRPV1 15 43 O=C(NCCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972894 EG On-Demand Anodyne CCR3 27 52 O=C(NCCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972894 EG On-Demand Anodyne CHRNA7 24 54 O=C(NCCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880972894 EG On-Demand Anodyne HNMT 63 36 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccs2)CC1 ZINC000880972895 FH On-Demand Anodyne FAAH 17 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccs2)CC1 ZINC000880972895 FH On-Demand Anodyne RBP4 56 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](CO)C1 ZINC000880972896 DE On-Demand Anodyne RBP4 75 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](CO)C1 ZINC000880972897 DE On-Demand Anodyne RBP4 75 44 CCCCCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972903 GH On-Demand Anodyne EPHX2 17 41 CCCCCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972903 GH On-Demand Anodyne RBP4 58 40 CCCCCNC(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972903 GH On-Demand Anodyne ASAH1 57 36 O=C(Nc1cnccc1C(F)(F)F)NC1CCC(C(F)(F)F)CC1 ZINC000880972904 FI On-Demand Anodyne EPHX2 43 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc([N+](=O)[O-])cc2)CC1 ZINC000880972906 GG On-Demand Bother RBP4 49 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nc3ccccc3[nH]2)CC1 ZINC000880972907 GI On-Demand Anodyne RBP4 82 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nc3ccccc3[nH]2)CC1 ZINC000880972907 GI On-Demand Anodyne SMO 33 48 Cn1nccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972917 CE On-Demand Anodyne TRPV1 21 49 Cn1nccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880972917 CE On-Demand Anodyne FLT1 17 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(-c2cnc(Cl)nc2)nn1 ZINC000880972929 FG On-Demand Anodyne SOAT1 25 41 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne HTR1A 84 54 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne DRD2 58 46 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne DRD4 32 41 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne ADRA1D 66 45 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne HTR1D 16 54 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne HTR1B 19 54 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne HTR2A 21 46 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne ADRA1A 59 45 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne ADRA1B 50 42 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne DRD3 65 41 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne PDGFRB 46 44 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne HTR7 57 47 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne TRPV1 22 59 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne FAAH 16 46 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne RBP4 85 61 COc1ccccc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880972935 GG On-Demand Anodyne TAAR1 25 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCC(C)(O)CC1 ZINC000880972947 EI On-Demand Anodyne EPHX2 40 43 C#CCNC(=O)C1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880972949 GG On-Demand Mild EPHX2 32 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880972969 GI On-Demand Anodyne EPHX2 45 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCN(C[C@@H]2CCCO2)CC1 ZINC000880972969 GI On-Demand Anodyne CXCR3 22 52 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880972970 GI On-Demand Anodyne EPHX2 45 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCN(C[C@H]2CCCO2)CC1 ZINC000880972970 GI On-Demand Anodyne CXCR3 22 52 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](O)C2CC2)nn1 ZINC000880972983 EF On-Demand Anodyne SOAT1 29 40 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](O)C2CC2)nn1 ZINC000880972984 EF On-Demand Anodyne SOAT1 29 40 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972987 DD On-Demand Anodyne PDGFRB 32 42 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972987 DD On-Demand Anodyne FLT4 30 42 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC)c(OC)c2)nn1 ZINC000880972987 DD On-Demand Anodyne ENPP1 87 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880973001 FH On-Demand Anodyne SOAT1 22 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(Cl)cc1 ZINC000880973007 FD On-Demand Anodyne CHRNA7 17 47 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(Cl)cc1 ZINC000880973007 FD On-Demand Anodyne EPHX2 25 52 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880973014 EF On-Demand Anodyne SOAT1 30 40 COC[C@@H](O)Cc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880973015 EC On-Demand Anodyne GHSR 16 40 O=C(NC1CC1)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973020 GD On-Demand Anodyne RBP4 66 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C2CC2)CC1 ZINC000880973021 EF On-Demand Anodyne TRPV1 20 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C2CC2)CC1 ZINC000880973021 EF On-Demand Anodyne EPHX2 46 45 CCCN(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973022 EJ On-Demand Anodyne TRPV1 17 42 CCN(Cc1ccc(OC)c(OC)c1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973023 GI On-Demand Anodyne ROCK2 20 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccncc2)CC1 ZINC000880973024 FF On-Demand Anodyne TRPV1 20 52 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccncc2)CC1 ZINC000880973024 FF On-Demand Anodyne RBP4 60 43 O=C(NCC1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973025 DH On-Demand Anodyne TRPV1 24 46 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne HRH2 25 40 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne TRPV1 29 52 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne AURKB 16 40 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne FAAH 20 52 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne CCR2 16 40 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne EPHX2 23 44 O=C(NCc1cccc(CN2CCOCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973032 GG On-Demand Anodyne NAMPT 72 44 O=C(NCc1nnc2n1CCC2)Nc1cnccc1C(F)(F)F ZINC000880973033 ED On-Demand Anodyne TRPV1 18 45 COCC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973038 FD On-Demand Anodyne RBP4 66 43 COCC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973038 FD On-Demand Anodyne SFRP1 62 33 COCC(=O)NC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973038 FD On-Demand Anodyne WNT3 48 31 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne DRD4 16 55 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne TRPV1 25 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne SIGMAR1 16 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne SSTR5 40 35 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne CCR3 24 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne SLC6A5 29 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne EPHX2 43 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne CXCR3 22 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne MCHR1 29 45 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne SFRP1 41 34 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccn2)CC1 ZINC000880973043 GG On-Demand Anodyne HPGDS 36 40 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973045 GF On-Demand Anodyne RAF1 27 40 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973045 GF On-Demand Anodyne MTNR1A 16 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)[C@H]2CCCO2)CC1 ZINC000880973052 FD On-Demand Anodyne RBP4 73 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)[C@@H]2CCCO2)CC1 ZINC000880973053 FD On-Demand Anodyne RBP4 73 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000880973056 FI On-Demand Anodyne EPHX2 25 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@H](C(F)(F)F)C1 ZINC000880973057 FI On-Demand Anodyne EPHX2 25 46 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H](C(F)(F)F)C1 ZINC000880973058 FI On-Demand Anodyne EPHX2 25 46 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@@H](C(F)(F)F)C1 ZINC000880973059 FI On-Demand Anodyne EPHX2 25 46 N#Cc1cccnc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973060 GF On-Demand Mild P2RY12 16 43 N#Cc1cccnc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973060 GF On-Demand Mild TRPV1 36 56 N#Cc1cccnc1N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973060 GF On-Demand Mild RBP4 54 39 COCC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973066 ED On-Demand Anodyne TRPV1 17 44 COCC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973066 ED On-Demand Anodyne RBP4 62 43 CCOC(=O)CCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973067 DF On-Demand Anodyne TRPV1 18 45 COc1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880973069 FI On-Demand Anodyne GCGR 26 42 COc1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880973069 FI On-Demand Anodyne TRPV1 21 44 COc1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880973069 FI On-Demand Anodyne ROCK2 15 44 COc1ccc(CN(C(=O)Nc2cnccc2C(F)(F)F)C2CC2)cc1 ZINC000880973069 FI On-Demand Anodyne GIPR 38 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000880973070 GG On-Demand Bother TRPV1 20 58 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2[N+](=O)[O-])CC1 ZINC000880973070 GG On-Demand Bother RBP4 59 44 CCCN(CCC)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973076 CH On-Demand Anodyne TRPV1 17 41 CNC(=O)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973079 CC On-Demand Anodyne TRPV1 21 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2F)CC1 ZINC000880973082 FH On-Demand Anodyne KCNQ2 43 35 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2F)CC1 ZINC000880973082 FH On-Demand Anodyne TRPV1 24 61 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2F)CC1 ZINC000880973082 FH On-Demand Anodyne NPY2R 53 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2F)CC1 ZINC000880973082 FH On-Demand Anodyne FAAH 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2F)CC1 ZINC000880973082 FH On-Demand Anodyne RBP4 73 50 CC(C)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973083 EF On-Demand Anodyne TRPV1 20 44 CC(C)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973083 EF On-Demand Anodyne RBP4 61 41 NOCc1cn(CC(=O)Nc2ccc(C(F)(F)F)cc2)nn1 ZINC000880973087 DD On-Demand Anodyne EPHX2 17 40 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NC[C@@H]1CCCO1 ZINC000880973091 CC On-Demand Anodyne PDE8B 43 36 O=C(Cn1cc([C@H]2CCCCO2)nn1)NC[C@H]1CCCO1 ZINC000880973092 CC On-Demand Anodyne PDE8B 43 36 O=C(Cn1cc([C@H]2CCCCO2)nn1)NC[C@@H]1CCCO1 ZINC000880973093 CC On-Demand Anodyne PDE8B 43 36 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NC[C@H]1CCCO1 ZINC000880973094 CC On-Demand Anodyne PDE8B 43 36 O=C(NCc1ccc(N2CCSCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880973095 GH On-Demand Clean TRPV1 20 50 O=C(NCc1ccc(N2CCSCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880973095 GH On-Demand Clean NAMPT 71 38 O=C(NC[C@@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973100 FF On-Demand Anodyne ADRB2 35 42 O=C(NC[C@@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973100 FF On-Demand Anodyne ADRB1 61 49 O=C(NC[C@@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973100 FF On-Demand Anodyne ADRB3 34 43 O=C(NC[C@@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973100 FF On-Demand Anodyne TRPV1 19 47 O=C(NC[C@@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973100 FF On-Demand Anodyne PDS 42 33 O=C(NC[C@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973101 FF On-Demand Anodyne ADRB2 35 42 O=C(NC[C@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973101 FF On-Demand Anodyne ADRB1 61 49 O=C(NC[C@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973101 FF On-Demand Anodyne ADRB3 34 43 O=C(NC[C@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973101 FF On-Demand Anodyne TRPV1 19 47 O=C(NC[C@H](O)COc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973101 FF On-Demand Anodyne PDS 42 33 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](c1ccccc1)C1CC1 ZINC000880973107 EI On-Demand Anodyne TRPV1 21 64 O=C(Nc1cnccc1C(F)(F)F)N[C@@H](c1ccccc1)C1CC1 ZINC000880973107 EI On-Demand Anodyne RBP4 46 37 O=C(Nc1cnccc1C(F)(F)F)N[C@H](c1ccccc1)C1CC1 ZINC000880973108 EI On-Demand Anodyne TRPV1 21 64 O=C(Nc1cnccc1C(F)(F)F)N[C@H](c1ccccc1)C1CC1 ZINC000880973108 EI On-Demand Anodyne RBP4 46 37 C[C@@H]1CN(CCCNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880973114 FF On-Demand Anodyne CCR3 23 46 C[C@@H]1CN(CCCNC(=O)Nc2cnccc2C(F)(F)F)C[C@@H](C)O1 ZINC000880973114 FF On-Demand Anodyne NAMPT 20 44 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)N1CCCCC1 ZINC000880973115 EG On-Demand Anodyne TRPV1 19 44 O=C(NCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880973118 FG On-Demand Anodyne TRPV1 29 53 O=C(NCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880973118 FG On-Demand Anodyne NOS2 91 35 O=C(NCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880973118 FG On-Demand Anodyne NAMPT 51 34 CC(=O)N1CCN(Cc2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880973119 GC On-Demand Anodyne SIGMAR1 26 42 CC(=O)N1CCN(Cc2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880973119 GC On-Demand Anodyne SCN2A 16 43 CC(=O)N1CCN(Cc2cn(CC(=O)NCCCc3ccccc3)nn2)CC1 ZINC000880973119 GC On-Demand Anodyne PREP 27 42 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(CC(C)(C)O)nn1 ZINC000880973130 EF On-Demand Anodyne SOAT1 40 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@@H]1C(=O)N(C)C ZINC000880973133 FG On-Demand Anodyne WNT3 41 32 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](C)N)nn1 ZINC000880973156 DE On-Demand Anodyne SOAT1 49 43 Cc1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](C)N)nn1 ZINC000880973157 DE On-Demand Anodyne SOAT1 49 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2)CC1 ZINC000880973160 FG On-Demand Anodyne TRPV1 25 55 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2)CC1 ZINC000880973160 FG On-Demand Anodyne FAAH 22 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2)CC1 ZINC000880973160 FG On-Demand Anodyne RBP4 92 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccc2)CC1 ZINC000880973160 FG On-Demand Anodyne SCD1 21 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C[C@H](O)c2ccccn2)nn1 ZINC000880973164 GG On-Demand Anodyne SOAT1 34 42 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C[C@@H](O)c2ccccn2)nn1 ZINC000880973165 GG On-Demand Anodyne SOAT1 34 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CC1)OCCO2 ZINC000880973169 FH On-Demand Anodyne TRPM8 23 40 COC(=O)Cc1cn(CC(=O)Nc2c(C)cccc2C(C)C)nn1 ZINC000880973170 EE On-Demand Anodyne SOAT1 45 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCCCc1ccccc1 ZINC000880973182 FD On-Demand Anodyne SIGMAR1 26 40 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCCCc1ccccc1 ZINC000880973182 FD On-Demand Anodyne EPHX2 17 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(CON)nn1 ZINC000880973193 DD On-Demand Anodyne SOAT1 46 41 Cn1nc2c(c1-c1cn(CC(=O)NCCCc3ccccc3)nn1)CCCC2 ZINC000880973199 GE On-Demand Anodyne BCHE 65 35 COC(=O)Cc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880973207 DC On-Demand Anodyne MTNR1A 25 41 COC(=O)Cc1cn(CC(=O)NCCCc2ccccc2)nn1 ZINC000880973207 DC On-Demand Anodyne MTNR1B 29 41 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C(C)(C)O)nn1 ZINC000880973212 DF On-Demand Anodyne SOAT1 47 43 COCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cn1 ZINC000880973219 FF On-Demand Anodyne TRPV1 18 47 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973226 FG On-Demand Anodyne BMP1 45 36 CN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973226 FG On-Demand Anodyne NOS2 63 32 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccnc1 ZINC000880973236 EH On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccnc1 ZINC000880973236 EH On-Demand Anodyne CHRNA7 17 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccnc1 ZINC000880973236 EH On-Demand Anodyne RBP4 54 39 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(NC2CCOCC2)CC1 ZINC000880973237 GI On-Demand Anodyne CCR2 51 48 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(NC2CCOCC2)CC1 ZINC000880973237 GI On-Demand Anodyne EPHX2 27 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccnc1 ZINC000880973238 EH On-Demand Anodyne TRPV1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccnc1 ZINC000880973238 EH On-Demand Anodyne CHRNA7 17 48 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccnc1 ZINC000880973238 EH On-Demand Anodyne RBP4 54 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880973241 GG On-Demand Anodyne EPHX2 45 51 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880973241 GG On-Demand Anodyne RBP4 29 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccoc2)CC1 ZINC000880973241 GG On-Demand Anodyne SFRP1 42 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CHRM2 16 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CHRM1 15 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne DRD2 19 60 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne DRD4 45 60 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne ACHE 44 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne DRD3 15 60 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CHRM3 22 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne LTA4H 19 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne TRPV1 31 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne SIGMAR1 49 63 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne SSTR5 54 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CCR3 53 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CHRNA7 41 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne C3AR1 41 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne ABL2 42 35 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne FAAH 23 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CCR2 27 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne SLC6A5 31 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne EPHX2 47 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CXCR3 33 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne RBP4 57 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne MCHR1 61 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CACNA1G 28 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne CCR8 16 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne SFRP1 98 36 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne WNT3 62 36 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccccc2)CC1 ZINC000880973242 GH On-Demand Anodyne HPGDS 39 41 O=C(NCCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973245 EG On-Demand Anodyne HRH2 25 43 O=C(NCCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973245 EG On-Demand Anodyne TRPV1 15 43 O=C(NCCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973245 EG On-Demand Anodyne CCR3 27 52 O=C(NCCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973245 EG On-Demand Anodyne CHRNA7 24 54 O=C(NCCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973245 EG On-Demand Anodyne HNMT 63 36 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880973249 GE On-Demand Anodyne CHRNA7 15 47 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880973249 GE On-Demand Anodyne EPHX2 37 55 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880973249 GE On-Demand Anodyne MCHR1 15 41 O=C(NCc1ccccc1CN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973261 GG On-Demand Anodyne TRPV1 25 54 O=C(NCc1ccccc1CN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973261 GG On-Demand Anodyne ABL2 44 37 O=C(NCc1ccccc1CN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973261 GG On-Demand Anodyne EPHX2 26 41 O=C(NCc1ccccc1CN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973261 GG On-Demand Anodyne NAMPT 38 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccc1 ZINC000880973269 EI On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccc1 ZINC000880973269 EI On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccc1 ZINC000880973269 EI On-Demand Anodyne SFRP1 93 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccccc1 ZINC000880973269 EI On-Demand Anodyne WNT3 76 38 COC(=O)[C@@]1(C)CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880973273 EE On-Demand Anodyne MTNR1A 17 42 COC(=O)[C@@]1(C)CN(C(=O)[C@@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880973273 EE On-Demand Anodyne MTNR1B 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccc1 ZINC000880973274 EI On-Demand Anodyne TRPV1 15 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccc1 ZINC000880973274 EI On-Demand Anodyne RBP4 73 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccc1 ZINC000880973274 EI On-Demand Anodyne SFRP1 93 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccccc1 ZINC000880973274 EI On-Demand Anodyne WNT3 76 38 C[C@H](Cc1ccco1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880973275 DG On-Demand Anodyne TRPV1 15 44 COC(=O)[C@@]1(C)CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880973276 EE On-Demand Anodyne MTNR1A 17 42 COC(=O)[C@@]1(C)CN(C(=O)[C@H]2CCc3cc(OC)ccc3C2)C[C@@H]1C ZINC000880973276 EE On-Demand Anodyne MTNR1B 19 42 C[C@@H](Cc1ccco1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880973277 DG On-Demand Anodyne TRPV1 15 44 O=C(NCCCN1CCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880973283 EE On-Demand Anodyne CCR3 19 43 O=C(NCCCN1CCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880973283 EE On-Demand Anodyne TYRO3 20 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCOc2ccccc21 ZINC000880973284 EH On-Demand Anodyne TRPV1 38 56 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCOc2ccccc21 ZINC000880973284 EH On-Demand Anodyne RBP4 63 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOc2ccccc21 ZINC000880973285 EH On-Demand Anodyne TRPV1 38 56 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCOc2ccccc21 ZINC000880973285 EH On-Demand Anodyne RBP4 63 43 CC(C)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973287 EG On-Demand Anodyne EPHX2 51 46 CC(C)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973287 EG On-Demand Anodyne CXCR3 21 45 CC(C)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973287 EG On-Demand Anodyne MCHR1 17 41 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc(NC(=O)C2CC2)cc1 ZINC000880973289 GI On-Demand Anodyne TRPV1 18 52 COc1ccc(CN(CCO)C(=O)Nc2cscc2Cl)cc1 ZINC000880973291 EG On-Demand Anodyne ROCK2 17 42 COc1ccccc1NC(=O)Cn1cc(CCCCCCO)nn1 ZINC000880973292 EE On-Demand Anodyne SOAT1 19 43 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@H](c2ccccc2)C1 ZINC000880973294 FH On-Demand Anodyne RBP4 79 44 CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)[C@@H](c2ccccc2)C1 ZINC000880973296 FH On-Demand Anodyne RBP4 79 44 O=C(NCc1cccnc1OCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880973299 GH On-Demand Anodyne TRPV1 30 54 O=C(NCc1cccnc1OCC(F)(F)F)Nc1cnccc1C(F)(F)F ZINC000880973299 GH On-Demand Anodyne SCN10A 17 52 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCc2ccccc21 ZINC000880973300 EI On-Demand Anodyne TRPV1 23 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCc2ccccc21 ZINC000880973300 EI On-Demand Anodyne RBP4 71 44 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCc2ccccc21 ZINC000880973300 EI On-Demand Anodyne TRPM8 33 45 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCc2ccccc21 ZINC000880973302 EI On-Demand Anodyne TRPV1 23 41 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCc2ccccc21 ZINC000880973302 EI On-Demand Anodyne RBP4 71 44 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCc2ccccc21 ZINC000880973302 EI On-Demand Anodyne TRPM8 33 45 CCCNC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973306 GH On-Demand Anodyne TRPV1 31 53 CCCNC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973306 GH On-Demand Anodyne ROCK2 48 41 CCCNC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973306 GH On-Demand Anodyne NR1H3 17 46 CCCNC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973306 GH On-Demand Anodyne NR1H2 29 46 CCCNC(=O)c1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880973306 GH On-Demand Anodyne NAMPT 51 38 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@H](CF)C1 ZINC000880973311 EJ On-Demand Anodyne CCR2 27 42 CCNC(=O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973312 FD On-Demand Anodyne RBP4 54 39 O=C(NCC1(c2ccccc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880973317 EH On-Demand Anodyne TRPV1 27 52 O=C(NCC1(c2ccccc2)CC1)Nc1cnccc1C(F)(F)F ZINC000880973317 EH On-Demand Anodyne KCNA3 41 40 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc2c(c1)OCCO2 ZINC000880973318 FH On-Demand Anodyne TRPV1 18 58 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@@H](CF)C1 ZINC000880973319 EJ On-Demand Anodyne CCR2 27 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880973321 GG On-Demand Anodyne RBP4 51 32 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne CHRM2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne DRD4 41 54 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne ACHE 34 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne CHRM3 21 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne TRPV1 28 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne SIGMAR1 37 55 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne SSTR5 40 36 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne CCR3 55 50 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne FAAH 15 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne CCR2 39 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne SLC6A5 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne MCHR1 40 49 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne BIRC2 26 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne SFRP1 93 35 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000880973322 FG On-Demand Anodyne WNT3 56 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880973323 GG On-Demand Anodyne RBP4 51 32 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne CHRM2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne DRD4 41 54 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne ACHE 34 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne CHRM3 21 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne TRPV1 28 43 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne SIGMAR1 37 55 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne SSTR5 40 36 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne CCR3 55 50 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne FAAH 15 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne CCR2 39 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne SLC6A5 25 44 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne RBP4 64 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne MCHR1 40 49 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne BIRC2 26 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne SFRP1 93 35 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000880973324 FG On-Demand Anodyne WNT3 56 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H]2CS(=O)(=O)C[C@H]2C1 ZINC000880973325 GG On-Demand Anodyne RBP4 51 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H]2CS(=O)(=O)C[C@@H]2C1 ZINC000880973328 GG On-Demand Anodyne RBP4 51 32 O=C(NCc1ccc(OCC(F)(F)F)nc1)Nc1cnccc1C(F)(F)F ZINC000880973332 GH On-Demand Anodyne TRPV1 17 49 CN(CCNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880973333 EG On-Demand Anodyne TRPV1 22 48 O=C(NC[C@H](CO)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973334 FG On-Demand Anodyne TRPV1 22 54 O=C(NC[C@H](CO)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973334 FG On-Demand Anodyne GPR142 49 33 O=C(NC[C@@H](CO)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973335 FG On-Demand Anodyne TRPV1 22 54 O=C(NC[C@@H](CO)Cc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973335 FG On-Demand Anodyne GPR142 49 33 COCc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973336 EH On-Demand Anodyne TRPV1 31 59 COCc1ccccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973336 EH On-Demand Anodyne NAMPT 20 40 O=C(NCc1ccc(N2CCCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880973341 FI On-Demand Clean TRPV1 23 52 O=C(NCc1ccc(N2CCCC2)cc1)Nc1cnccc1C(F)(F)F ZINC000880973341 FI On-Demand Clean NAMPT 100 43 O=C(NCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973342 DF On-Demand Anodyne HRH2 22 40 O=C(NCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973342 DF On-Demand Anodyne TRPV1 21 44 O=C(NCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973342 DF On-Demand Anodyne CCR3 17 44 O=C(NCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973342 DF On-Demand Anodyne CHRNA7 17 48 O=C(NCCN1CCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973342 DF On-Demand Anodyne HNMT 45 34 O=C(CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)N1CCCCC1 ZINC000880973344 GE On-Demand Anodyne RBP4 54 39 O=C(NCCCN1CCCCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880973345 FG On-Demand Anodyne CCR3 20 43 O=C(NCCCN1CCCCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880973345 FG On-Demand Anodyne TYRO3 19 40 O=C(NCc1cccc(N2CCCC2=O)c1)Nc1cnccc1C(F)(F)F ZINC000880973351 GH On-Demand Anodyne TRPV1 27 51 O=C(NCc1cccc(N2CCCC2=O)c1)Nc1cnccc1C(F)(F)F ZINC000880973351 GH On-Demand Anodyne CARM1 51 34 O=C(NCc1cccc(N2CCCC2=O)c1)Nc1cnccc1C(F)(F)F ZINC000880973351 GH On-Demand Anodyne NAMPT 43 38 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000880973354 FF On-Demand Anodyne TRPV1 21 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000880973354 FF On-Demand Anodyne CHRNA7 41 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000880973354 FF On-Demand Anodyne FAAH 35 56 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2cccnc2)CC1 ZINC000880973354 FF On-Demand Anodyne RBP4 58 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H]2[C@@H](CCN2C)C1 ZINC000880973360 FH On-Demand Anodyne RBP4 51 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H]2[C@H](CCN2C)C1 ZINC000880973361 FH On-Demand Anodyne RBP4 51 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H]2[C@H](CCN2C)C1 ZINC000880973362 FH On-Demand Anodyne RBP4 51 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H]2[C@@H](CCN2C)C1 ZINC000880973363 FH On-Demand Anodyne RBP4 51 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2nccs2)C1 ZINC000880973404 FJ On-Demand Anodyne RBP4 39 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2nccs2)C1 ZINC000880973405 FJ On-Demand Anodyne RBP4 39 40 CC(=O)C1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880973415 EI On-Demand Anodyne EPHX2 25 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N(C)Cc1cccc(C(N)=O)c1 ZINC000880973429 GI On-Demand Anodyne TACR1 28 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccncc2)CC1 ZINC000880973452 FF On-Demand Anodyne TRPV1 19 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccncc2)CC1 ZINC000880973452 FF On-Demand Anodyne FAAH 31 57 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccncc2)CC1 ZINC000880973452 FF On-Demand Anodyne RBP4 57 41 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne TRPV1 50 53 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne PIK3CA 35 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne MTOR 50 40 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne EPHX2 18 42 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne SCN10A 29 51 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne STAT6 53 33 O=C(NCc1cccnc1N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973453 GF On-Demand Anodyne NAMPT 52 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)CC1 ZINC000880973454 DE On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)CC1 ZINC000880973454 DE On-Demand Anodyne EPHX2 15 51 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CO)CC1 ZINC000880973454 DE On-Demand Anodyne RBP4 76 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2nnc3ccccn23)CC1 ZINC000880973455 GH On-Demand Anodyne RBP4 96 47 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880973460 GH On-Demand Anodyne SOAT1 59 40 Cc1cccc(C(C)C)c1NC(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880973461 GH On-Demand Anodyne SOAT1 59 40 COc1ccccc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880973481 FD On-Demand Anodyne HTR1A 46 41 COc1ccccc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880973481 FD On-Demand Anodyne DRD2 39 47 COc1ccccc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880973481 FD On-Demand Anodyne DRD4 25 41 COc1ccccc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880973481 FD On-Demand Anodyne DRD3 53 47 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@@H]1CC[C@H](O)CC1 ZINC000880973484 EH On-Demand Anodyne EPHX2 44 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCC2(CC1)OCCO2 ZINC000880973486 EF On-Demand Anodyne EPHX2 30 43 Cn1ncc2c1CCC[C@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880973488 EG On-Demand Anodyne TRPV1 26 43 Cn1ncc2c1CCC[C@@H]2NC(=O)Nc1cnccc1C(F)(F)F ZINC000880973490 EG On-Demand Anodyne TRPV1 26 43 CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973492 DF On-Demand Anodyne TRPV1 26 40 CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973492 DF On-Demand Anodyne SLC6A5 29 40 CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973492 DF On-Demand Anodyne EPHX2 55 45 CCN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973492 DF On-Demand Anodyne CXCR3 22 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne DRD4 22 50 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne SIGMAR1 24 53 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne SSTR5 50 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne SLC6A5 32 49 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne EPHX2 43 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne CXCR3 27 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(Cc2ccncc2)CC1 ZINC000880973496 GG On-Demand Anodyne MCHR1 51 47 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880973499 FF On-Demand Anodyne EPHX2 57 63 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880973499 FF On-Demand Anodyne RBP4 49 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880973499 FF On-Demand Anodyne SFRP1 108 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)C2CC2)CC1 ZINC000880973499 FF On-Demand Anodyne WNT3 82 37 O=C(NCc1ccc(N2CCCC2=O)cc1)Nc1cnccc1C(F)(F)F ZINC000880973504 GH On-Demand Anodyne NAMPT 57 39 O=C(CCC1CCCC1)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973507 GH On-Demand Anodyne RBP4 62 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCc2ncncc2C1 ZINC000880973509 FH On-Demand Anodyne P2RY14 44 37 O=C(NCCCOCC1CC1)Nc1cnccc1C(F)(F)F ZINC000880973510 DG On-Demand Anodyne TRPV1 18 44 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCCc2ccccc21 ZINC000880973515 EJ On-Demand Anodyne RBP4 56 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@H]1CCCc2ccccc21 ZINC000880973515 EJ On-Demand Anodyne TRPM8 29 43 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCCc2ccccc21 ZINC000880973517 EJ On-Demand Anodyne RBP4 56 42 CN(C(=O)Nc1cnccc1C(F)(F)F)[C@@H]1CCCc2ccccc21 ZINC000880973517 EJ On-Demand Anodyne TRPM8 29 43 CCS(=O)(=O)N1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880973529 GF On-Demand Anodyne EPHX2 17 45 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880973534 EF On-Demand Anodyne EPHX2 33 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCC[C@@H]2C1 ZINC000880973534 EF On-Demand Anodyne WNT3 40 34 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880973536 EF On-Demand Anodyne EPHX2 33 41 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCC[C@H]2C1 ZINC000880973536 EF On-Demand Anodyne WNT3 40 34 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880973538 EF On-Demand Anodyne EPHX2 33 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCC[C@H]2C1 ZINC000880973538 EF On-Demand Anodyne WNT3 40 34 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880973540 EF On-Demand Anodyne EPHX2 33 41 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCC[C@@H]2C1 ZINC000880973540 EF On-Demand Anodyne WNT3 40 34 CNC(=O)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973545 FD On-Demand Anodyne DRD4 15 40 CNC(=O)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973545 FD On-Demand Anodyne EPHX2 45 41 CNC(=O)CN1CCC(NC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973545 FD On-Demand Anodyne CXCR3 20 43 COc1ccc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)cc1OC ZINC000880973551 GI On-Demand Anodyne RBP4 33 40 O=C(NC[C@@H](c1ccccc1)N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973555 GG On-Demand Anodyne TRPV1 15 44 O=C(NC[C@H](c1ccccc1)N1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880973557 GG On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880973562 GI On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880973562 GI On-Demand Anodyne RBP4 94 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880973562 GI On-Demand Anodyne SFRP1 66 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880973562 GI On-Demand Anodyne WNT3 48 33 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880973563 GI On-Demand Anodyne TRPV1 15 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880973563 GI On-Demand Anodyne RBP4 94 46 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880973563 GI On-Demand Anodyne SFRP1 66 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880973563 GI On-Demand Anodyne WNT3 48 33 COc1ccccc1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880973566 GE On-Demand Anodyne MMP13 15 49 COc1ccccc1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880973566 GE On-Demand Anodyne MMP8 25 44 Cc1ccccc1CN(C)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973571 DI On-Demand Anodyne TRPV1 15 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccco2)CC1 ZINC000880973572 FG On-Demand Anodyne FAAH 15 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccco2)CC1 ZINC000880973572 FG On-Demand Anodyne RBP4 59 42 O=C(NC[C@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973574 FH On-Demand Anodyne TRPV1 23 43 O=C(NC[C@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973574 FH On-Demand Anodyne CCR3 19 41 O=C(NC[C@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973574 FH On-Demand Anodyne RBP4 54 39 O=C(NC[C@@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973576 FH On-Demand Anodyne TRPV1 23 43 O=C(NC[C@@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973576 FH On-Demand Anodyne CCR3 19 41 O=C(NC[C@@H]1CCN(c2ccccc2)C1)Nc1cnccc1C(F)(F)F ZINC000880973576 FH On-Demand Anodyne RBP4 54 39 O=C(Nc1cscc1Cl)N1CC[C@@]2(CCc3ccccc32)C1 ZINC000880973577 EJ On-Demand Anodyne NPY5R 38 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CHRM1 15 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne DRD2 17 48 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne DRD4 27 50 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne HTR2A 16 50 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CHRM3 20 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne SIGMAR1 40 50 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CCR3 48 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CHRNA7 46 43 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne C3AR1 41 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne SLC6A5 31 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne EPHX2 44 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CXCR3 20 41 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne RBP4 63 39 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne MCHR1 36 44 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne CACNA1G 25 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne BIRC2 29 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne SFRP1 90 37 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne WNT3 56 33 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne ACHP_LYMST 28 42 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(CCc2ccccc2)CC1 ZINC000880973578 GH On-Demand Anodyne HPGDS 34 40 O=C(Nc1cscc1Cl)N1CC[C@]2(CCc3ccccc32)C1 ZINC000880973581 EJ On-Demand Anodyne NPY5R 38 48 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccccc2)CC1 ZINC000880973582 GH On-Demand Anodyne ACHE 19 46 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccccc2)CC1 ZINC000880973582 GH On-Demand Anodyne TRPV1 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccccc2)CC1 ZINC000880973582 GH On-Demand Anodyne SIGMAR1 25 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccccc2)CC1 ZINC000880973582 GH On-Demand Anodyne FAAH 40 56 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccccc2)CC1 ZINC000880973582 GH On-Demand Anodyne RBP4 70 44 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880973587 FH On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@H](c2ccc(F)cc2)C1 ZINC000880973587 FH On-Demand Anodyne TRPM8 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880973588 FH On-Demand Anodyne RBP4 61 42 O=C(Nc1cnccc1C(F)(F)F)N1CCO[C@@H](c2ccc(F)cc2)C1 ZINC000880973588 FH On-Demand Anodyne TRPM8 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1nc2ccccc2s1 ZINC000880973592 GK On-Demand Anodyne RBP4 46 37 CCN(Cc1ccccc1)C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880973593 GF On-Demand Anodyne TSPO 18 40 CCN(Cc1ccccc1)C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880973596 GF On-Demand Anodyne TSPO 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1nc2ccccc2s1 ZINC000880973597 GK On-Demand Anodyne RBP4 46 37 CN(C)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973603 EE On-Demand Anodyne RBP4 69 42 CN(C)C(=O)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973603 EE On-Demand Anodyne SFRP1 41 34 O=C(Nc1cnccc1C(F)(F)F)N(Cc1ccncc1)C1CC1 ZINC000880973610 EH On-Demand Anodyne TRPV1 18 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@H](O)C1 ZINC000880973611 DF On-Demand Anodyne TRPV1 32 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@H](O)C1 ZINC000880973611 DF On-Demand Anodyne EPHX2 32 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@@H](O)C1 ZINC000880973613 DF On-Demand Anodyne TRPV1 32 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@@H](O)C1 ZINC000880973613 DF On-Demand Anodyne EPHX2 32 47 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H](O)C1 ZINC000880973615 DF On-Demand Anodyne TRPV1 32 42 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCC[C@H](O)C1 ZINC000880973615 DF On-Demand Anodyne EPHX2 32 47 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@@H](O)C1 ZINC000880973616 DF On-Demand Anodyne TRPV1 32 42 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCC[C@@H](O)C1 ZINC000880973616 DF On-Demand Anodyne EPHX2 32 47 CCN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880973619 DF On-Demand Anodyne TRPV1 16 40 CCN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880973619 DF On-Demand Anodyne CCR3 40 42 CCN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880973619 DF On-Demand Anodyne CACNA1I 57 37 CCN1CC[C@H](CNC(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880973619 DF On-Demand Anodyne NAMPT 22 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1cccs1 ZINC000880973621 EJ On-Demand Anodyne RBP4 46 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1cccs1 ZINC000880973623 EJ On-Demand Anodyne RBP4 46 37 O=C(c1ccc(O)cc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973624 GH On-Demand Anodyne RBP4 68 43 CCN(Cc1ccccc1)C(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880973626 DD On-Demand Anodyne TSPO 20 41 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880973635 FD On-Demand Anodyne EPHX2 25 41 O=C(NCCCn1cccn1)Nc1cnccc1C(F)(F)F ZINC000880973636 DF On-Demand Anodyne TRPV1 16 45 O=C(Cn1cc(CC2(O)CCOCC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880973640 GE On-Demand Anodyne EPHX2 24 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccco2)CC1 ZINC000880973642 FF On-Demand Anodyne RBP4 69 49 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCCCc1ccccc1 ZINC000880973645 FE On-Demand Anodyne AMP1_PLAFQ 39 47 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCCCc1ccccc1 ZINC000880973645 FE On-Demand Anodyne NPFFR1 47 31 CONC(=O)C1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880973646 FG On-Demand Anodyne TACR1 25 41 CONC(=O)C1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880973646 FG On-Demand Anodyne EPHX2 27 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCCCc1ccccc1 ZINC000880973647 FE On-Demand Anodyne AMP1_PLAFQ 39 47 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCCCc1ccccc1 ZINC000880973647 FE On-Demand Anodyne NPFFR1 47 31 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CCCCO2)CC1 ZINC000880973676 FJ On-Demand Anodyne EPHX2 20 46 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CCCCO2)CC1 ZINC000880973676 FJ On-Demand Anodyne TRPM8 29 42 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1c(C)cc(C(F)(F)F)cc1C ZINC000880973687 FH On-Demand Anodyne SLC6A3 30 42 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1c(C)cc(C(F)(F)F)cc1C ZINC000880973688 FH On-Demand Anodyne SLC6A3 30 42 Cn1ncc(Br)c1CC(=O)NCc1ccc(C(C)(C)C)nc1O ZINC000880973708 GE On-Demand Anodyne P2RX7 17 46 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(C1)OCCO2 ZINC000880973724 EG On-Demand Anodyne EPHX2 35 43 O=C(NCc1cccc(NC(=O)C2CCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973763 GI On-Demand Anodyne TRPV1 34 52 O=C(NCc1cccc(NC(=O)C2CCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973763 GI On-Demand Anodyne ROCK2 25 40 O=C(NCc1cccc(NC(=O)C2CCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973763 GI On-Demand Anodyne EPHX2 15 45 O=C(NCc1cccc(NC(=O)C2CCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973763 GI On-Demand Anodyne NAMPT 61 39 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne TACR1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne TRPV1 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne CHRNA7 42 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne PREP 69 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne RBP4 76 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne SFRP1 78 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1Cc1ccccc1 ZINC000880973764 EI On-Demand Anodyne WNT3 69 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne TACR1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne TRPV1 19 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne CHRNA7 42 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne PREP 69 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne RBP4 76 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne SFRP1 78 36 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1Cc1ccccc1 ZINC000880973765 EI On-Demand Anodyne WNT3 69 36 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000880973770 GH On-Demand Anodyne CCR3 27 44 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000880973770 GH On-Demand Anodyne FAAH 26 51 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000880973770 GH On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccsc2)CC1 ZINC000880973771 FH On-Demand Anodyne FAAH 21 50 O=C(Nc1cnccc1C(F)(F)F)N1CCN(Cc2ccsc2)CC1 ZINC000880973771 FH On-Demand Anodyne RBP4 54 40 O=C(NCc1ccccc1CN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880973773 GI On-Demand Anodyne ABL1 43 38 O=C(NCc1ccccc1CN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880973773 GI On-Demand Anodyne TRPV1 28 57 O=C(NCc1ccccc1CN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880973773 GI On-Demand Anodyne ABL2 45 38 O=C(NCc1ccccc1CN1CCCC1)Nc1cnccc1C(F)(F)F ZINC000880973773 GI On-Demand Anodyne NAMPT 42 38 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc(F)cc1 ZINC000880973774 FJ On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H]1c1ccc(F)cc1 ZINC000880973774 FJ On-Demand Anodyne TRPM8 35 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000880973775 FJ On-Demand Anodyne RBP4 47 37 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000880973775 FJ On-Demand Anodyne TRPM8 35 45 COc1ccccc1NC(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880973776 EE On-Demand Anodyne HCN1 40 33 O=C(NCc1ccccc1CN1CCCC1=O)Nc1cnccc1C(F)(F)F ZINC000880973779 GH On-Demand Anodyne TRPV1 25 53 CN(CCOc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973785 EH On-Demand Anodyne LTA4H 20 40 CN(CCOc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880973785 EH On-Demand Anodyne RBP4 17 57 CN(C)CCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973794 GG On-Demand Anodyne TRPV1 15 51 CN(C)CCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973794 GG On-Demand Anodyne RAF1 22 44 CN(C)CCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973794 GG On-Demand Anodyne ROCK2 15 43 CN(C)CCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973794 GG On-Demand Anodyne DDR2 15 41 COc1ccc(CN(C)C(=O)Nc2cnccc2C(F)(F)F)cc1OC ZINC000880973797 FH On-Demand Anodyne MT-ND1 19 44 COc1ccc([C@@H](O)CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973802 FF On-Demand Anodyne TRPV1 21 54 CN1CCN(C(C)(C)CNC(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973806 FE On-Demand Anodyne TRPV1 17 43 COc1ccc(OCCNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973808 FG On-Demand Anodyne TRPV1 23 52 COc1ccc(OCCNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973808 FG On-Demand Anodyne P2RY1 15 40 COc1ccc(OCCNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973808 FG On-Demand Anodyne RAF1 42 41 COc1ccc(OCCNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973808 FG On-Demand Anodyne MTNR1A 21 40 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1cccs1 ZINC000880973810 FH On-Demand Anodyne TRPV1 15 43 O=C(NCCCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973811 DH On-Demand Anodyne TRPV1 28 57 O=C(NCCCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973811 DH On-Demand Anodyne CES1 41 37 O=C(NCCCc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973811 DH On-Demand Anodyne AMP1_PLAFQ 24 41 O=C(NCCCOc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973812 EH On-Demand Anodyne HRH2 23 42 O=C(NCCCOc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973812 EH On-Demand Anodyne TRPV1 23 49 O=C(NCCCOc1ccccc1)Nc1cnccc1C(F)(F)F ZINC000880973812 EH On-Demand Anodyne EPHX2 15 43 O=C(NCc1ccc(N2CCCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880973814 GH On-Demand Anodyne TRPV1 19 46 O=C(NCc1ccc(N2CCCCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880973814 GH On-Demand Anodyne NAMPT 71 42 Cc1nc(CNC(=O)Nc2cnccc2C(F)(F)F)cs1 ZINC000880973816 DG On-Demand Anodyne TRPV1 24 51 O=C(NCc1ccnc(OCC(F)(F)F)c1)Nc1cnccc1C(F)(F)F ZINC000880973817 GH On-Demand Anodyne TRPV1 20 51 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880973818 GF On-Demand Anodyne TRPV1 16 45 O=C(NCc1ccc(N2CCOCC2)nc1)Nc1cnccc1C(F)(F)F ZINC000880973818 GF On-Demand Anodyne NAMPT 65 49 O=C(NCc1ccnc(N2CCCCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973819 GH On-Demand Anodyne TRPV1 21 48 O=C(NCc1ccnc(N2CCCCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880973819 GH On-Demand Anodyne NAMPT 51 39 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1C ZINC000880973820 EG On-Demand Anodyne TRPV1 24 42 C[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)N1CCCC[C@H]1C ZINC000880973820 EG On-Demand Anodyne NAMPT 15 40 C[C@H]1CCCCN1[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973821 EG On-Demand Anodyne TRPV1 24 42 C[C@H]1CCCCN1[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973821 EG On-Demand Anodyne NAMPT 15 40 C[C@H]1CCCCN1[C@@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973822 EG On-Demand Anodyne TRPV1 24 42 C[C@H]1CCCCN1[C@@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973822 EG On-Demand Anodyne NAMPT 15 40 C[C@@H]1CCCCN1[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973823 EG On-Demand Anodyne TRPV1 24 42 C[C@@H]1CCCCN1[C@H](C)CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880973823 EG On-Demand Anodyne NAMPT 15 40 O=C(CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)NC1CC1 ZINC000880973836 FD On-Demand Anodyne CCR2 19 41 O=C(CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)NC1CC1 ZINC000880973836 FD On-Demand Anodyne RBP4 58 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncccn2)CC1 ZINC000880973844 FE On-Demand Anodyne TRPV1 30 53 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ncccn2)CC1 ZINC000880973844 FE On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(O)c2)CC1 ZINC000880973845 FG On-Demand Anodyne TRPV1 26 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc(O)c2)CC1 ZINC000880973845 FG On-Demand Anodyne RBP4 61 43 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@@H](O)[C@H](C)O ZINC000880973851 DE On-Demand Anodyne SOAT1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne TRPV1 20 50 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne NPY2R 24 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne FAAH 17 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne EPHX2 23 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne RBP4 95 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne SCD1 21 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne SFRP1 39 43 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccccc2)CC1 ZINC000880973852 GG On-Demand Anodyne SMO 29 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@H](O)[C@@H](C)O ZINC000880973854 DE On-Demand Anodyne SOAT1 15 42 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CN2CCCCCC2)CC1 ZINC000880973856 GI On-Demand Anodyne RBP4 67 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CN2CCCCCC2)CC1 ZINC000880973856 GI On-Demand Anodyne SFRP1 88 35 O=C(Nc1cnccc1C(F)(F)F)N1CCC(CN2CCCCCC2)CC1 ZINC000880973856 GI On-Demand Anodyne WNT3 73 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@@H](O)[C@@H](C)O ZINC000880973857 DE On-Demand Anodyne SOAT1 15 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC[C@H](O)[C@H](C)O ZINC000880973858 DE On-Demand Anodyne SOAT1 15 42 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CC1 ZINC000880973866 DD On-Demand Anodyne TRPV1 27 45 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CC1 ZINC000880973866 DD On-Demand Anodyne CCR2 44 41 O=C(CNC(=O)Nc1cnccc1C(F)(F)F)NC1CC1 ZINC000880973866 DD On-Demand Anodyne EPHX2 25 40 COc1ccc(OC)c2c1CN(C(=O)Nc1cnccc1C(F)(F)F)C[C@H]2O ZINC000880973868 GG On-Demand Anodyne RBP4 52 38 COc1ccc(OC)c2c1CN(C(=O)Nc1cnccc1C(F)(F)F)C[C@@H]2O ZINC000880973869 GG On-Demand Anodyne RBP4 52 38 CCOC(=O)CC1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973871 FG On-Demand Anodyne RBP4 65 40 COCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973873 FG On-Demand Anodyne TRPV1 23 53 COCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973873 FG On-Demand Anodyne RAF1 42 38 COCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973873 FG On-Demand Anodyne ROCK2 17 45 COCCOc1ccc(CNC(=O)Nc2cnccc2C(F)(F)F)cc1 ZINC000880973873 FG On-Demand Anodyne NAMPT 49 39 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCc2cc(Cl)nnc2C1 ZINC000880973882 GI On-Demand Anodyne MAPK1 41 34 CC(=O)[C@@H]1CCCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)C1 ZINC000880973891 EI On-Demand Anodyne EPHX2 18 40 CC(=O)[C@H]1CCCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)C1 ZINC000880973892 EI On-Demand Anodyne EPHX2 18 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CC1)COCCO2 ZINC000880973899 FH On-Demand Anodyne EPHX2 23 46 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CC1)COCCO2 ZINC000880973899 FH On-Demand Anodyne TRPM8 29 42 CCN(Cc1ccccc1)C(=O)Cn1cc([C@@H](O)c2ccc(C)cc2)nn1 ZINC000880973901 FF On-Demand Anodyne TSPO 21 40 CCN(Cc1ccccc1)C(=O)Cn1cc([C@H](O)c2ccc(C)cc2)nn1 ZINC000880973902 FF On-Demand Anodyne TSPO 21 40 O=C(Nc1cscc1Cl)N1CCn2c(CCc3ccccc3)nnc2C1 ZINC000880973905 GH On-Demand Anodyne P2RX7 23 40 COC(=O)[C@@]1(C)CN(C(=O)CC[C@H]2CCc3ccccc32)C[C@@H]1C ZINC000880973906 EG On-Demand Anodyne EBP 20 44 COC(=O)[C@@]1(C)CN(C(=O)CC[C@@H]2CCc3ccccc32)C[C@@H]1C ZINC000880973907 EG On-Demand Anodyne EBP 20 44 CCN(Cc1ccccc1)C(=O)Cn1cc(CON)nn1 ZINC000880973908 CC On-Demand Anodyne TSPO 20 41 C[C@H]1CN(C(=O)Nc2cscc2Cl)Cc2ccccc21 ZINC000880973917 DJ On-Demand Anodyne RBP4 52 33 C[C@@H]1CN(C(=O)Nc2cscc2Cl)Cc2ccccc21 ZINC000880973918 DJ On-Demand Anodyne RBP4 52 33 CO[C@H]1COCC[C@@H]1N(C)C(=O)Nc1c(C)cc(C(F)(F)F)cc1C ZINC000880973922 FH On-Demand Anodyne CCR2 34 43 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](O)[C@@H](O)C1 ZINC000880973956 EE On-Demand Anodyne RBP4 42 33 O=C(NC[C@H]1COc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880973965 FG On-Demand Anodyne ADRA2B 15 41 O=C(NC[C@H]1COc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880973965 FG On-Demand Anodyne TRPV1 16 45 O=C(NC[C@@H]1COc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880973966 FG On-Demand Anodyne ADRA2B 15 41 O=C(NC[C@@H]1COc2ccccc2O1)Nc1cnccc1C(F)(F)F ZINC000880973966 FG On-Demand Anodyne TRPV1 16 45 O=C(NCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973968 EG On-Demand Anodyne HRH2 22 40 O=C(NCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973968 EG On-Demand Anodyne TRPV1 21 44 O=C(NCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973968 EG On-Demand Anodyne CCR3 17 44 O=C(NCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973968 EG On-Demand Anodyne CHRNA7 17 48 O=C(NCCN1CCCCCC1)Nc1cnccc1C(F)(F)F ZINC000880973968 EG On-Demand Anodyne HNMT 45 34 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2nc3ccccc3o2)C1 ZINC000880973969 GJ On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@@H](c2nc3ccccc3o2)C1 ZINC000880973969 GJ On-Demand Anodyne SMO 21 45 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2nc3ccccc3o2)C1 ZINC000880973970 GJ On-Demand Anodyne RBP4 74 44 O=C(Nc1cnccc1C(F)(F)F)N1CCC[C@H](c2nc3ccccc3o2)C1 ZINC000880973970 GJ On-Demand Anodyne SMO 21 45 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cnccc2C(F)(F)F)C1 ZINC000880973978 FF On-Demand Anodyne RBP4 56 39 Cn1cccc1[C@@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880973982 EH On-Demand Anodyne RBP4 48 37 Cn1cccc1[C@H]1CCCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880973983 EH On-Demand Anodyne RBP4 48 37 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)C(N)=O ZINC000880973984 DD On-Demand Anodyne TRPV1 20 47 Cn1cnnc1C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973986 FF On-Demand Anodyne RBP4 74 43 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne HTR1D 23 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne HTR1B 21 49 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne HTR1F 74 40 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne TRPV1 18 41 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne CCR2 32 55 O=C(Nc1cnccc1C(F)(F)F)N1CCC(c2c[nH]c3ccccc23)CC1 ZINC000880973990 GJ On-Demand Anodyne RBP4 99 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(F)cc2)CC1 ZINC000880973991 FH On-Demand Anodyne TRPV1 17 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccc(F)cc2)CC1 ZINC000880973991 FH On-Demand Anodyne RBP4 59 41 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne TRPV1 27 48 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne EPHX2 40 38 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne RBP4 93 47 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne SCD1 15 40 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne SFRP1 110 38 O=C(Nc1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880973993 GH On-Demand Anodyne WNT3 80 38 COc1ccc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)c(OC)c1 ZINC000880973994 GI On-Demand Anodyne RAF1 21 43 COc1ccc([C@@H]2CCCN2C(=O)Nc2cnccc2C(F)(F)F)c(OC)c1 ZINC000880973994 GI On-Demand Anodyne TAAR1 21 40 COC(=O)Cc1cn(CC(=O)Nc2ccc(C(F)(F)F)cc2)nn1 ZINC000880973999 ED On-Demand Anodyne EPHX2 18 40 O=C(Nc1cnccc1C(F)(F)F)N1CCCN(CC(F)(F)F)CC1 ZINC000880974004 FG On-Demand Anodyne RBP4 55 41 O=C(NC[C@@H]1CC1(Cl)Cl)Nc1cnccc1C(F)(F)F ZINC000880974009 EG On-Demand Anodyne TRPV1 21 47 O=C(NC[C@H]1CC1(Cl)Cl)Nc1cnccc1C(F)(F)F ZINC000880974010 EG On-Demand Anodyne TRPV1 21 47 Cn1cnnc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974011 DD On-Demand Anodyne TRPV1 19 48 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974013 FF On-Demand Anodyne TRPV1 21 47 CC(C)(C)C(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974013 FF On-Demand Anodyne RBP4 61 43 CC[C@H](C)NC(=O)CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974015 GE On-Demand Anodyne RBP4 40 37 C[C@@H]1CCCCN1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974023 EG On-Demand Anodyne TRPV1 15 43 C[C@H]1CCCCN1CCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974024 EG On-Demand Anodyne TRPV1 15 43 O=C(CN1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1)N1CCCC1 ZINC000880974025 GD On-Demand Anodyne RBP4 55 40 COc1ccc(OC)c([C@H](C)NC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974026 FI On-Demand Anodyne RAF1 23 42 N#Cc1ccnc(N2CCN(C(=O)Nc3cnccc3C(F)(F)F)CC2)c1 ZINC000880974030 GF On-Demand Mild RBP4 46 37 COCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974031 FF On-Demand Anodyne TRPV1 35 52 COCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974031 FF On-Demand Anodyne P2RY1 42 39 COCCOc1ncccc1CNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974031 FF On-Demand Anodyne SCN10A 21 44 O=C(NCc1ccnc(N2CCCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880974032 FG On-Demand Anodyne TRPV1 22 49 O=C(NCc1ccnc(N2CCCC2)c1)Nc1cnccc1C(F)(F)F ZINC000880974032 FG On-Demand Anodyne NAMPT 55 38 O=C(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974035 GI On-Demand Anodyne TRPV1 17 44 O=C(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974035 GI On-Demand Anodyne SLC18A3 35 41 O=C(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974035 GI On-Demand Anodyne RBP4 94 48 O=C(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974035 GI On-Demand Anodyne SFRP1 117 42 O=C(c1ccccc1)C1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974035 GI On-Demand Anodyne WNT3 81 38 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880974040 FH On-Demand Anodyne KCNA5 21 42 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880974040 FH On-Demand Anodyne TRPV1 22 48 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1ccccc1 ZINC000880974040 FH On-Demand Anodyne SOAT1 19 42 O=C(Nc1cnccc1C(F)(F)F)N1CCCCC[C@H]1c1ccncc1 ZINC000880974042 FJ On-Demand Anodyne RBP4 43 38 O=C(Nc1cnccc1C(F)(F)F)N1CCCCC[C@@H]1c1ccncc1 ZINC000880974043 FJ On-Demand Anodyne RBP4 43 38 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974044 EE On-Demand Anodyne MCHR1 17 41 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974044 EE On-Demand Anodyne LUXR 15 40 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974044 EE On-Demand Anodyne TRAR 18 40 CCN(Cc1ccccc1)C(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1 ZINC000880974045 FF On-Demand Anodyne PLA2G7 79 36 CCN(Cc1ccccc1)C(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1 ZINC000880974045 FF On-Demand Anodyne TSPO 21 40 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974046 EE On-Demand Anodyne MCHR1 17 41 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974046 EE On-Demand Anodyne LUXR 15 40 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974046 EE On-Demand Anodyne TRAR 18 40 CCN(Cc1ccccc1)C(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1 ZINC000880974047 FF On-Demand Anodyne PLA2G7 79 36 CCN(Cc1ccccc1)C(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1 ZINC000880974047 FF On-Demand Anodyne TSPO 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc([N+](=O)[O-])c2)CC1 ZINC000880974055 GG On-Demand Bother TRPV1 15 51 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc([N+](=O)[O-])c2)CC1 ZINC000880974055 GG On-Demand Bother SERPINE1 21 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc([N+](=O)[O-])c2)CC1 ZINC000880974055 GG On-Demand Bother MET 16 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cccc([N+](=O)[O-])c2)CC1 ZINC000880974055 GG On-Demand Bother RBP4 54 38 CN(C)CCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974062 GG On-Demand Anodyne TRPV1 28 52 CN(C)CCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974062 GG On-Demand Anodyne ROCK1 24 47 CN(C)CCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974062 GG On-Demand Anodyne RAF1 25 42 CN(C)CCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974062 GG On-Demand Anodyne ROCK2 42 53 CN(C)CCOc1cccc(CNC(=O)Nc2cnccc2C(F)(F)F)c1 ZINC000880974062 GG On-Demand Anodyne PDS 55 40 O=C(NCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974064 DD On-Demand Anodyne TRPV1 18 43 O=C(NCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974064 DD On-Demand Anodyne EPHX2 27 51 O=C(NCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974064 DD On-Demand Anodyne HPGDS 23 41 O=C(NCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974064 DD On-Demand Anodyne NAMPT 16 41 COc1ccccc1NC(=O)Cn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880974065 FC On-Demand Anodyne DRD2 25 48 COc1ccccc1NC(=O)Cn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880974065 FC On-Demand Anodyne DRD4 29 44 COc1ccccc1NC(=O)Cn1cc(CN2CCN(C(C)=O)CC2)nn1 ZINC000880974065 FC On-Demand Anodyne DRD3 30 48 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCCC2)CC1 ZINC000880974066 EG On-Demand Anodyne HRH3 20 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C2CCCC2)CC1 ZINC000880974066 EG On-Demand Anodyne RBP4 68 43 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCCC[C@@H]12 ZINC000880974067 EF On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCCC[C@H]12 ZINC000880974068 EF On-Demand Anodyne EPHX2 15 40 C=C[C@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974071 DC On-Demand Mild CA9 15 42 C=C[C@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974071 DC On-Demand Mild PROKR1 63 35 C=C[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974072 DC On-Demand Mild CA9 15 42 C=C[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974072 DC On-Demand Mild PROKR1 63 35 CCN(Cc1ccccc1)C(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880974107 EE On-Demand Anodyne TSPO 19 40 O=C(Nc1cscc1Cl)N1CCC(Oc2ccc(Cl)cn2)CC1 ZINC000880974185 FJ On-Demand Anodyne EPHX2 18 42 O=C(NCCCCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974193 GE On-Demand Anodyne PREP 42 49 O=C(NCCCCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974193 GE On-Demand Anodyne CAPN1 40 34 O=C(NCCCCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974193 GE On-Demand Anodyne CAPN2 66 38 O=C(NCCCCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974193 GE On-Demand Anodyne TGM2 22 44 O=C(NCCCCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974193 GE On-Demand Anodyne NPR 54 36 CN(C(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1)C1CCCCC1 ZINC000880974198 EE On-Demand Anodyne SCARB1 29 40 CN(C(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1)C1CCCCC1 ZINC000880974199 EE On-Demand Anodyne SCARB1 29 40 O=C(Nc1cscc1Cl)N[C@H]1CCCC[C@H]1F ZINC000880974219 CH On-Demand Anodyne SSTR3 15 41 COC(=O)c1cccc(C#Cc2cccc(NC(=O)c3ccccc3SCC#N)c2)c1 ZINC000880974228 IJ On-Demand Mild KCNK3 108 43 COC(=O)c1cccc(C#Cc2cccc(NC(=O)c3ccccc3SCC#N)c2)c1 ZINC000880974228 IJ On-Demand Mild KCNK9 82 42 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974233 ED On-Demand Anodyne KLK3 46 32 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974233 ED On-Demand Anodyne PREP 49 48 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974233 ED On-Demand Anodyne CAPN1 45 36 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974233 ED On-Demand Anodyne CAPN2 70 36 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)OCc1ccccc1 ZINC000880974233 ED On-Demand Anodyne NPR 60 35 O=C(Nc1cscc1Cl)N1CCC(c2nccc(-c3cccnc3)n2)CC1 ZINC000880974241 GJ On-Demand Anodyne CALCRL 17 41 O=C(Cn1cc(-c2ccc(Cl)cc2F)nn1)N1CCCC1 ZINC000880974246 DE On-Demand Anodyne DPP9 15 40 O=C(NCc1cn(CC(=O)N2CCCC2)nn1)c1cccnc1Cl ZINC000880974252 EC On-Demand Anodyne G2YM83_BOTF4 67 34 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NOCc1cccnc1 ZINC000880974344 EH On-Demand Anodyne CHRNA7 22 40 O=C(Nc1cnccc1C(F)(F)F)N[C@H]1CCN2CCCC[C@H]12 ZINC000880974368 EF On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)N[C@@H]1CCN2CCCC[C@@H]12 ZINC000880974371 EF On-Demand Anodyne EPHX2 15 40 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880974375 GG On-Demand Anodyne C3AR1 40 37 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880974375 GG On-Demand Anodyne EPHX2 44 46 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880974375 GG On-Demand Anodyne RBP4 45 52 O=C(Nc1cnccc1C(F)(F)F)NC1CCN(C(=O)c2ccco2)CC1 ZINC000880974375 GG On-Demand Anodyne SFRP1 58 38 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880974384 GH On-Demand Clean EPHB4 45 32 CN(Cc1ccc(N2CCOCC2)cc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880974384 GH On-Demand Clean STAT6 52 33 C[C@H](CCc1ccc(O)cc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880974387 FH On-Demand Anodyne TRPV1 22 43 C[C@@H](CCc1ccc(O)cc1)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880974389 FH On-Demand Anodyne TRPV1 22 43 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC2(CC1)CNC(=O)O2 ZINC000880974401 FG On-Demand Anodyne TRPM8 31 43 C[C@H](N)c1cn(CC(=O)Nc2ccc(C(F)(F)F)cc2)nn1 ZINC000880974410 DD On-Demand Anodyne EPHX2 18 40 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NC1CCCCCC1 ZINC000880974412 EE On-Demand Anodyne SCARB1 33 40 CN(C)[C@@H](CNC(=O)Nc1cnccc1C(F)(F)F)c1cccc(F)c1 ZINC000880974413 FH On-Demand Anodyne TRPV1 25 46 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NC1CCCCCC1 ZINC000880974418 EE On-Demand Anodyne SCARB1 33 40 CC[C@H](O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974419 DD On-Demand Anodyne PROKR1 59 32 COCCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974422 CF On-Demand Anodyne TRPV1 18 45 COc1cc2c(cc1OC)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880974432 GH On-Demand Anodyne ABCB1 21 41 COc1cc2c(cc1OC)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880974432 GH On-Demand Anodyne RBP4 50 43 COc1cc2c(cc1OC)CN(C(=O)Nc1cnccc1C(F)(F)F)CC2 ZINC000880974432 GH On-Demand Anodyne ABCG2 32 40 O=C(NCCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974440 ED On-Demand Anodyne CCR3 25 50 O=C(NCCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974440 ED On-Demand Anodyne EPHX2 28 45 O=C(NCCCN1CCOCC1)Nc1cnccc1C(F)(F)F ZINC000880974440 ED On-Demand Anodyne NAMPT 24 45 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@](O)(C(F)F)C1 ZINC000880974452 FH On-Demand Anodyne EPHX2 23 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@](O)(C(F)F)C1 ZINC000880974456 FH On-Demand Anodyne EPHX2 23 40 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC[C@H]2CCCO2)nn1 ZINC000880974459 ED On-Demand Anodyne TNK2 42 36 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NC[C@@H]2CCCO2)nn1 ZINC000880974462 ED On-Demand Anodyne TNK2 42 36 O=C(Cn1cc(CNC(=O)C(F)(F)F)nn1)Nc1ccc(C(F)(F)F)cc1 ZINC000880974469 GE On-Demand Anodyne EPHX2 16 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880974478 FG On-Demand Anodyne CCR2 37 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880974478 FG On-Demand Anodyne EPHX2 33 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCN(CC(C)(C)O)C1 ZINC000880974478 FG On-Demand Anodyne CXCR3 19 48 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1ccncc1 ZINC000880974489 EI On-Demand Anodyne RAF1 25 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1ccncc1 ZINC000880974489 EI On-Demand Anodyne FLT1 31 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCCc1ccncc1 ZINC000880974489 EI On-Demand Anodyne KDR 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880974490 GG On-Demand Anodyne NPY2R 15 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880974490 GG On-Demand Anodyne SLC9A1 27 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000880974490 GG On-Demand Anodyne RBP4 62 41 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cnccn2)CC1 ZINC000880974492 FE On-Demand Anodyne TRPV1 18 49 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2cnccn2)CC1 ZINC000880974492 FE On-Demand Anodyne RBP4 58 41 Cc1ccccc1[C@H](C)NC(=O)Nc1cnccc1C(F)(F)F ZINC000880974499 DI On-Demand Anodyne TRPV1 19 53 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(CC(=O)N2CCCC2)nn1 ZINC000880974500 ED On-Demand Anodyne PREP 25 47 O=C(NCCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880974502 FG On-Demand Anodyne TRPV1 22 51 O=C(NCCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880974502 FG On-Demand Anodyne RAF1 25 41 O=C(NCCc1ccc2c(c1)OCCO2)Nc1cnccc1C(F)(F)F ZINC000880974502 FG On-Demand Anodyne NOS2 48 36 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(CC(=O)N2CCCC2)nn1 ZINC000880974503 ED On-Demand Anodyne PREP 25 47 CCOCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974524 CF On-Demand Anodyne TRPV1 17 44 CC(C)(CNC(=O)Nc1cnccc1C(F)(F)F)N1CCOCC1 ZINC000880974526 EE On-Demand Anodyne TRPV1 17 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@H](NC2CCOCC2)C1 ZINC000880974540 GI On-Demand Anodyne CCR2 55 47 CCN(Cc1ccc2c(c1)OCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880974543 FH On-Demand Anodyne NOS2 76 33 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@@H](NC2CCOCC2)C1 ZINC000880974545 GI On-Demand Anodyne CCR2 55 47 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccn2)CC1 ZINC000880974548 FF On-Demand Anodyne TRPV1 26 63 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccn2)CC1 ZINC000880974548 FF On-Demand Anodyne FAAH 19 45 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccn2)CC1 ZINC000880974548 FF On-Demand Anodyne RBP4 72 44 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccn2)CC1 ZINC000880974548 FF On-Demand Anodyne SCD1 25 40 O=C(Nc1cnccc1C(F)(F)F)N1CCN(c2ccccn2)CC1 ZINC000880974548 FF On-Demand Anodyne DGAT1 22 42 CCOC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974556 EE On-Demand Anodyne TRPV1 18 44 CCOC(=O)N1CCN(C(=O)Nc2cnccc2C(F)(F)F)CC1 ZINC000880974556 EE On-Demand Anodyne RBP4 57 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC2(CC2)C1 ZINC000880974559 CH On-Demand Anodyne EPHX2 23 40 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880974560 FJ On-Demand Anodyne RBP4 40 38 CC[C@@H]1c2ccsc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880974560 FJ On-Demand Anodyne TRPM8 29 50 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880974563 FJ On-Demand Anodyne RBP4 40 38 CC[C@H]1c2ccsc2CCN1C(=O)Nc1cnccc1C(F)(F)F ZINC000880974563 FJ On-Demand Anodyne TRPM8 29 50 O=C(NCCc1ccc2c(c1)OCO2)Nc1cnccc1C(F)(F)F ZINC000880974567 FG On-Demand Anodyne TRPV1 19 51 O=C(NCCc1ccc2c(c1)OCO2)Nc1cnccc1C(F)(F)F ZINC000880974567 FG On-Demand Anodyne RAF1 24 41 O=C(NCCc1ccc2c(c1)OCO2)Nc1cnccc1C(F)(F)F ZINC000880974567 FG On-Demand Anodyne NOS2 94 41 O=C(Nc1cscc1Cl)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880974569 EI On-Demand Anodyne HRH1 27 41 O=C(Nc1cscc1Cl)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880974569 EI On-Demand Anodyne CCR3 35 41 O=C(Nc1cscc1Cl)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880974569 EI On-Demand Anodyne EPHX2 29 49 O=C(Nc1cscc1Cl)N1CC[C@H](Oc2ccc(F)cc2)C1 ZINC000880974569 EI On-Demand Anodyne SCD1 19 42 C[C@@H]1CCCCN1CCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974570 FH On-Demand Anodyne CCR3 26 42 C[C@H]1CCCCN1CCCCNC(=O)Nc1cnccc1C(F)(F)F ZINC000880974574 FH On-Demand Anodyne CCR3 26 42 CN(C(=O)Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)C1CCCCC1 ZINC000880974599 FF On-Demand Anodyne SCARB1 27 40 CN(C(=O)Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)C1CCCCC1 ZINC000880974603 FF On-Demand Anodyne SCARB1 27 40 O=C(Cn1cc(-c2cccnc2Cl)nn1)NC1CCCCCC1 ZINC000880974614 EF On-Demand Anodyne CNR1 15 43 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc2c(c1)OCO2 ZINC000880974615 FH On-Demand Anodyne KCNQ2 30 43 C[C@H](NC(=O)Nc1cnccc1C(F)(F)F)c1ccc2c(c1)OCO2 ZINC000880974615 FH On-Demand Anodyne TRPV1 15 58 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)n1cc(CC(C)(C)O)nn1 ZINC000880974616 FF On-Demand Anodyne PDS 41 35 CCN(Cc1ccccc1)C(=O)Nc1cnccc1C(F)(F)F ZINC000880974618 DI On-Demand Anodyne TRPV1 18 44 O=C(Cn1cc(CCCN2CCOCC2)nn1)NC1CCCCC1 ZINC000880974636 EC On-Demand Anodyne EPHX2 16 46 O=C(Nc1cscc1Cl)N1CC[C@@H]2CSC[C@@H]2C1 ZINC000880974637 DH On-Demand Anodyne RBP4 44 32 COC[C@@H](O)Cc1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974641 EC On-Demand Anodyne CA9 15 40 COC[C@@H](O)Cc1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880974641 EC On-Demand Anodyne PROKR1 47 31 O=C(Nc1cscc1Cl)N1CC[C@H]2CSC[C@H]2C1 ZINC000880974642 DH On-Demand Anodyne RBP4 44 32 O=C(Nc1cscc1Cl)N1CC[C@H]2CSC[C@@H]2C1 ZINC000880974644 DH On-Demand Anodyne RBP4 44 32 COC(=O)C1CCC(c2cn(CC(=O)NCc3ccc(OC)cc3)nn2)CC1 ZINC000880974646 GE On-Demand Anodyne PROKR1 42 30 O=C(Nc1cscc1Cl)N1CC[C@@H]2CSC[C@H]2C1 ZINC000880974647 DH On-Demand Anodyne RBP4 44 32 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974657 EE On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974657 EE On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974657 EE On-Demand Anodyne SCARB1 32 41 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974661 EE On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974661 EE On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCCC1 ZINC000880974661 EE On-Demand Anodyne SCARB1 32 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(C)(N2CCC2)CC1 ZINC000880974668 FI On-Demand Anodyne CCR5 25 44 CN(Cc1ccc2c(c1)OCCO2)C(=O)Nc1cnccc1C(F)(F)F ZINC000880974683 FH On-Demand Anodyne TRPV1 16 41 O=C(Cn1cc(CCCOc2cccnc2F)nn1)N1CCCC1 ZINC000880974701 ED On-Demand Anodyne MMP8 18 45 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCCCC1 ZINC000880974706 GF On-Demand Anodyne CNR1 22 46 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCCCC1 ZINC000880974707 GF On-Demand Anodyne CNR1 22 46 CN(C(=O)Cn1cc(CCCOc2cccnc2F)nn1)C1CCCCC1 ZINC000880974712 GF On-Demand Anodyne MMP8 25 45 O=C(Nc1cscc1Cl)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880974717 FI On-Demand Anodyne SMO 41 48 O=C(Nc1cscc1Cl)N1CCC(c2nc(C3CCC3)no2)CC1 ZINC000880974717 FI On-Demand Anodyne ETHR 62 47 CC(C)(C)OC(=O)N1CCN(Cc2cn(CC(=O)N3CCCC3)nn2)CC1 ZINC000880974729 GC On-Demand Anodyne KDM1A 21 48 CC[C@H](O)c1cn(CC(=O)Nc2cc(OC)cc(OC)c2)nn1 ZINC000880974757 DD On-Demand Anodyne PDGFRB 23 40 CC[C@H](O)c1cn(CC(=O)Nc2cc(OC)cc(OC)c2)nn1 ZINC000880974757 DD On-Demand Anodyne FLT4 20 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@@H](CO)CC1 ZINC000880974763 EH On-Demand Anodyne CCR2 21 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@H](CO)CC1 ZINC000880974764 EH On-Demand Anodyne CCR2 21 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NNC(=O)C1CC1 ZINC000880974778 DF On-Demand Reactive EPHX2 24 41 COc1cccc([C@H](O)C2CCN(C(=O)Nc3cscc3Cl)CC2)c1 ZINC000880974784 GI On-Demand Anodyne DRD4 40 31 Cc1nc(NC2CC2)sc1C(=O)NCc1ccc(C(C)(C)C)nc1O ZINC000880974791 FG On-Demand Anodyne SCD1 24 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880974798 DF On-Demand Anodyne LUXR 80 54 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880974798 DF On-Demand Anodyne TRAR 97 54 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCOC1=O ZINC000880974798 DF On-Demand Anodyne LASR 64 40 N#Cc1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880974803 FD On-Demand Mild EPHX2 19 43 COc1ccccc1[C@@H]1CN(C(=O)Nc2cscc2Cl)CCO1 ZINC000880974808 FI On-Demand Anodyne RBP4 48 41 CN(C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1)C1CCCCC1 ZINC000880974814 GE On-Demand Anodyne G2YM83_BOTF4 68 35 O=C(Cn1cc([C@H](O)c2ccc(F)cc2)nn1)NC1CCCCCC1 ZINC000880974825 EE On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@@H](O)c2ccc(F)cc2)nn1)NC1CCCCCC1 ZINC000880974829 EE On-Demand Anodyne SCARB1 29 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@@H]1C[C@@H](S(C)(=O)=O)C1 ZINC000880974919 FG On-Demand Anodyne EPHX2 18 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1CCC2(CC1)COC2 ZINC000880974926 FI On-Demand Anodyne EPHX2 32 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@@]2(C1)CC2(F)F ZINC000880974930 FJ On-Demand Anodyne EPHX2 23 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC[C@]2(C1)CC2(F)F ZINC000880974935 FJ On-Demand Anodyne EPHX2 23 40 O=C(Cn1cc(COc2ccc(Br)nc2)nn1)NC1CCCCC1 ZINC000880974940 GE On-Demand Anodyne FIMH 19 40 O=C(Cn1cc(C[C@H](O)c2ccccc2)nn1)NC1CCCCC1 ZINC000880974952 EE On-Demand Anodyne SCARB1 33 40 O=C(Cn1cc(C[C@@H](O)c2ccccc2)nn1)NC1CCCCC1 ZINC000880974954 EE On-Demand Anodyne SCARB1 33 40 CN(C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1)C1CCCCC1 ZINC000880974958 GE On-Demand Anodyne PREP 25 41 CN(C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1)C1CCCCC1 ZINC000880974958 GE On-Demand Anodyne CAPN1 43 36 CN(C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1)C1CCCCC1 ZINC000880974958 GE On-Demand Anodyne CAPN2 69 35 CN(C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1)C1CCCCC1 ZINC000880974958 GE On-Demand Anodyne NPR 61 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NC1COC(C)(C)OC1 ZINC000880974996 EH On-Demand Anodyne EPHX2 15 40 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccccc1C(F)(F)F ZINC000880975022 EE On-Demand Anodyne RBP4 41 33 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccccc1C(F)(F)F ZINC000880975025 EE On-Demand Anodyne RBP4 41 33 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(F)CC1 ZINC000880975036 DI On-Demand Anodyne EPHX2 28 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(F)CC1 ZINC000880975036 DI On-Demand Anodyne RBP4 40 37 CN(C(=O)Cn1cc(COc2cccc(N)c2)nn1)C1CCCCC1 ZINC000880975049 EE On-Demand Anodyne SCARB1 29 40 O=C(Nc1cscc1Cl)N1C[C@H]2CC=CC[C@H]2C1 ZINC000880975055 CH On-Demand Anodyne RBP4 47 34 CC(C)(C)OC(=O)N1CCCN(Cc2cn(CC(=O)N3CCCC3)nn2)CC1 ZINC000880975060 GD On-Demand Anodyne KDM1A 20 46 COc1cc2c(cc1OC)[C@H](C)N(C(=O)Nc1cscc1Cl)CC2 ZINC000880975090 FJ On-Demand Anodyne SLC18A2 40 33 COc1cc2c(cc1OC)[C@@H](C)N(C(=O)Nc1cscc1Cl)CC2 ZINC000880975094 FJ On-Demand Anodyne SLC18A2 40 33 O=C(Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCCCC1 ZINC000880975101 GG On-Demand Anodyne CCR2 63 40 O=C(Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCCCC1 ZINC000880975103 GG On-Demand Anodyne CCR2 63 40 O=C(Cn1cc(C(=O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975115 EF On-Demand Anodyne CNR1 25 47 O=C(Cn1cc(C(=O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975115 EF On-Demand Anodyne SCARB1 31 42 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880975119 DD On-Demand Anodyne CA9 18 44 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880975119 DD On-Demand Anodyne PROKR1 66 36 O=C(Nc1cscc1Cl)N1[C@H]2CC[C@H]1CC(O)(c1ccccc1)C2 ZINC000880975132 FI On-Demand Anodyne OPRL1 19 47 CCN(Cc1ccccc1)C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880975133 FF On-Demand Anodyne TSPO 21 41 CCN(Cc1ccccc1)C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880975135 FF On-Demand Anodyne TSPO 21 41 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NC1CCCCC1 ZINC000880975147 FE On-Demand Anodyne MMP8 18 44 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne DRD4 19 42 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne GRIN2B 29 40 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne SIGMAR1 16 41 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne CTSB 15 51 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne CTSK 19 51 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne CTSL 25 51 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne EPHX2 47 40 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne TGM2 36 48 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne DPP7 15 48 O=C(NC1CCN(C(=O)Nc2cscc2Cl)CC1)OCc1ccccc1 ZINC000880975158 GI On-Demand Anodyne F13A1 29 48 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1ccccc1C(F)(F)F ZINC000880975171 EE On-Demand Anodyne RBP4 44 34 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1ccccc1C(F)(F)F ZINC000880975172 EE On-Demand Anodyne RBP4 44 34 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NC1CCCCCC1 ZINC000880975191 GF On-Demand Anodyne MMP8 18 44 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975230 EE On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975230 EE On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975232 EE On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCC1 ZINC000880975232 EE On-Demand Anodyne SCARB1 29 41 Nc1cccc(OCc2cn(CC(=O)NC3CCCCCC3)nn2)c1 ZINC000880975263 EE On-Demand Anodyne FAAH 25 45 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCc1cnc(Cl)cn1 ZINC000880975272 FI On-Demand Anodyne ATF1 45 33 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCc1cnc(Cl)cn1 ZINC000880975272 FI On-Demand Anodyne NFKB1 41 33 COC(=O)Cc1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880975277 DC On-Demand Anodyne CA9 19 46 COC(=O)Cc1cn(CC(=O)NCc2ccc(OC)cc2)nn1 ZINC000880975277 DC On-Demand Anodyne PROKR1 55 33 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCCC2(C1)OCCO2 ZINC000880975289 FH On-Demand Anodyne EPHX2 31 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H]1CCCC2(C1)OCCO2 ZINC000880975294 FI On-Demand Anodyne EPHX2 15 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@@H]1CCCC2(C1)OCCO2 ZINC000880975296 FI On-Demand Anodyne EPHX2 15 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(N2CCN(C)CC2)CC1 ZINC000880975325 GH On-Demand Anodyne L3MBTL3 58 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(C(=O)NCCO)CC1 ZINC000880975342 GF On-Demand Anodyne EPHX2 33 40 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1cscc1Cl ZINC000880975344 GH On-Demand Anodyne SIGMAR1 42 39 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1cscc1Cl ZINC000880975344 GH On-Demand Anodyne NPFFR2 36 41 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1cscc1Cl ZINC000880975344 GH On-Demand Anodyne UTS2R 19 46 O=C(NCCC1(O)CCN(Cc2ccccc2)CC1)Nc1cscc1Cl ZINC000880975344 GH On-Demand Anodyne NPFFR1 48 41 CC(=O)N1CCN(Cc2cn(Cc3cc(Cl)ccc3OC(F)F)nn2)CC1 ZINC000880975386 GE On-Demand Anodyne KDM1A 16 40 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)n1cc(C(C)(C)O)nn1 ZINC000880975389 EF On-Demand Anodyne KCNK3 18 41 CC(C)(C)OC(=O)N1CCC(c2cn(CC(=O)N3CCCC3)nn2)CC1 ZINC000880975424 FE On-Demand Anodyne GPR119 41 41 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975429 EE On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975429 EE On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975429 EE On-Demand Anodyne SCARB1 32 41 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975431 EE On-Demand Anodyne SIGMAR1 15 43 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975431 EE On-Demand Anodyne REN 48 34 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NC1CCCCC1 ZINC000880975431 EE On-Demand Anodyne SCARB1 32 41 CON(C)C(=O)C1CCN(C(=O)Nc2c(C)cc(C(F)(F)F)cc2C)CC1 ZINC000880975446 GH On-Demand Anodyne TACR1 29 40 CCN(Cc1ccccc1)C(=O)Cn1cc(CNC(=O)OC(C)(C)C)nn1 ZINC000880975458 FE On-Demand Anodyne CTSB 15 45 O=C(Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCCC1 ZINC000880975485 GF On-Demand Anodyne CCR2 63 40 O=C(Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1)NC1CCCCC1 ZINC000880975486 GF On-Demand Anodyne CCR2 63 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CTSB 34 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CTSK 28 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CTSL 32 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne PREP 30 44 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CAPNS1 42 32 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CAPN1 53 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne CAPN2 94 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne EPHX2 17 42 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCCC1 ZINC000880975491 GF On-Demand Anodyne NPR 59 32 C[C@H](O)c1ccc(OCc2cn(CC(=O)NC3CCCCCC3)nn2)cc1 ZINC000880975497 FF On-Demand Anodyne SCARB1 40 39 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCCCC3)nn2)c1 ZINC000880975499 FF On-Demand Anodyne FAAH 24 47 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCCCC3)nn2)c1 ZINC000880975499 FF On-Demand Anodyne SCARB1 34 42 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(F)(F)CC1 ZINC000880975517 EJ On-Demand Anodyne TRPM8 25 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(CCCO)CC1 ZINC000880975538 FI On-Demand Anodyne EPHX2 15 41 O=C(Nc1cscc1Cl)N1CC(CNC(=O)C(F)(F)F)C1 ZINC000880975547 EF On-Demand Anodyne RBP4 44 32 COC(=O)c1cccc(C#Cc2cccc(NC(=O)c3cc(S(=O)(=O)N(C)C)ccc3F)c2)c1 ZINC000880975570 JH On-Demand Mild KCNK3 88 38 COC(=O)c1cccc(C#Cc2cccc(NC(=O)c3cc(S(=O)(=O)N(C)C)ccc3F)c2)c1 ZINC000880975570 JH On-Demand Mild KCNK9 68 36 O=C(Nc1cscc1Cl)N1CCC[C@](CO)(c2ccccc2)C1 ZINC000880975578 FH On-Demand Anodyne EPHX2 19 57 O=C(Nc1cscc1Cl)N1CCC[C@@](CO)(c2ccccc2)C1 ZINC000880975579 FH On-Demand Anodyne EPHX2 19 57 Cc1cccc2c1OCC[C@@H]2NC(=O)Nc1cscc1Cl ZINC000880975589 DI On-Demand Anodyne TRPV1 18 48 O=C(Nc1cscc1Cl)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880975590 FG On-Demand Anodyne SMO 20 42 O=C(Nc1cscc1Cl)N1CCO[C@@H](c2noc(C3CC3)n2)C1 ZINC000880975590 FG On-Demand Anodyne ETHR 41 34 O=C(Nc1cscc1Cl)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880975591 FG On-Demand Anodyne SMO 20 42 O=C(Nc1cscc1Cl)N1CCO[C@H](c2noc(C3CC3)n2)C1 ZINC000880975591 FG On-Demand Anodyne ETHR 41 34 O=C(Nc1cscc1Cl)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880975600 EJ On-Demand Anodyne RBP4 66 39 O=C(Nc1cscc1Cl)N1C[C@@H]2[C@@H](C[C@H]2c2ccccc2)C1 ZINC000880975600 EJ On-Demand Anodyne SMO 34 40 O=C(Nc1cscc1Cl)N1CCC[C@@](O)(c2ccccc2)C1 ZINC000880975621 EH On-Demand Anodyne EPHX2 18 48 O=C(Nc1cscc1Cl)N1CCC[C@](O)(c2ccccc2)C1 ZINC000880975622 EH On-Demand Anodyne EPHX2 18 48 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)n1cc([C@@H](O)C2CC2)nn1 ZINC000880975641 FF On-Demand Anodyne CCR2 46 36 C[C@H](C(=O)Nc1cccc(C(F)(F)F)c1)n1cc([C@H](O)C2CC2)nn1 ZINC000880975643 FF On-Demand Anodyne CCR2 46 36 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCC1 ZINC000880975672 FF On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCC1 ZINC000880975672 FF On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCC1 ZINC000880975673 FF On-Demand Anodyne CNR1 22 45 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2)nn1)NC1CCCCCC1 ZINC000880975673 FF On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CTSB 34 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CTSK 28 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CTSL 32 40 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne PREP 30 44 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CAPNS1 42 32 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CAPN1 53 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne CAPN2 94 38 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne EPHX2 17 42 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NC1CCCCC1 ZINC000880975695 FE On-Demand Anodyne NPR 59 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne TACR1 42 36 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne TRPV1 18 57 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne CCR2 65 38 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne EPHX2 25 48 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne RBP4 79 38 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](c2ccccn2)C1 ZINC000880975697 FJ On-Demand Anodyne MAP3K12 47 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne TACR1 42 36 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne TRPV1 18 57 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne CCR2 65 38 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne EPHX2 25 48 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne RBP4 79 38 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](c2ccccn2)C1 ZINC000880975698 FJ On-Demand Anodyne MAP3K12 47 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)NCc1cccc(F)n1 ZINC000880975710 EI On-Demand Anodyne TRPV1 17 42 CCOC(=O)N1CCC(C(=O)Nc2cccc(C#Cc3cccc(C(=O)OC)c3)c2)CC1 ZINC000880975748 IH On-Demand Mild P2RY12 69 38 CCOC(=O)N1CCC(C(=O)Nc2cccc(C#Cc3cccc(C(=O)OC)c3)c2)CC1 ZINC000880975748 IH On-Demand Mild EPHX2 22 42 CN1CCN(C2CCN(C(=O)Nc3cscc3Cl)CC2)CC1 ZINC000880975784 EF On-Demand Anodyne L3MBTL3 61 42 CN(C(=O)Cn1cc(Cn2cnc(-c3ccccc3)c2N)nn1)C1CCCCC1 ZINC000880975832 GF On-Demand Anodyne SCARB1 32 43 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCCC3)nn2)c1 ZINC000880975849 FF On-Demand Anodyne FAAH 24 47 CC(=O)c1cccc(OCc2cn(CC(=O)NC3CCCCC3)nn2)c1 ZINC000880975849 FF On-Demand Anodyne SCARB1 34 42 O=C(Cn1cc([C@@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCCC1 ZINC000880975851 FF On-Demand Anodyne CNR1 22 46 O=C(Cn1cc([C@H](O)c2ccc(Cl)cc2F)nn1)NC1CCCCC1 ZINC000880975852 FF On-Demand Anodyne CNR1 22 46 O=C(Cn1cc([C@@H](O)c2ccc(F)cc2)nn1)NC1CCCCC1 ZINC000880975854 ED On-Demand Anodyne SCARB1 29 41 O=C(Cn1cc([C@H](O)c2ccc(F)cc2)nn1)NC1CCCCC1 ZINC000880975855 ED On-Demand Anodyne SCARB1 29 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H]2NC(=O)OC[C@H]2C1 ZINC000880975862 FG On-Demand Anodyne RBP4 44 32 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@@H](OC(=O)N(C)C)C1 ZINC000880975875 FH On-Demand Anodyne LIPG 45 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CC[C@H](OC(=O)N(C)C)C1 ZINC000880975876 FH On-Demand Anodyne LIPG 45 35 C[C@H](O)c1ccc(OCc2cn(CC(=O)NC3CCCCC3)nn2)cc1 ZINC000880975902 FE On-Demand Anodyne SCARB1 40 39 Cn1cnc(-c2nnc3n2CCN(C(=O)Nc2cscc2Cl)C3)c1 ZINC000880975916 FE On-Demand Anodyne P2RX7 24 46 CC(=O)c1cccc(OCc2cn(CC(=O)N(C)C3CCCCC3)nn2)c1 ZINC000880975932 FF On-Demand Anodyne SCARB1 32 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne OPRL1 21 49 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne TACR1 50 44 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne CCR1 28 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne CCR2 22 40 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne EPHX2 39 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne RBP4 54 34 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCC(O)(c2ccccc2)CC1 ZINC000880975936 GJ On-Demand Anodyne TRPM8 41 44 O=C(Cn1cc(-c2cccnc2Cl)nn1)NC1CCCCC1 ZINC000880975939 DE On-Demand Anodyne CNR1 15 43 O=C(Cn1cc(CCCN2CCOCC2)nn1)NC1CCCCCC1 ZINC000880975940 ED On-Demand Anodyne EPHX2 16 46 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H](CO)C[C@@H](O)c1ccccc1 ZINC000880975960 GH On-Demand Anodyne MTTP 43 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@@H](CO)C[C@@H](O)c1ccccc1 ZINC000880975961 GH On-Demand Anodyne MTTP 43 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@H](CO)C[C@H](O)c1ccccc1 ZINC000880975962 GH On-Demand Anodyne MTTP 43 35 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N[C@@H](CO)C[C@H](O)c1ccccc1 ZINC000880975963 GH On-Demand Anodyne MTTP 43 35 CCNc1nc(C)c(C(=O)NCc2ccc(C(C)(C)C)nc2O)s1 ZINC000880975970 EG On-Demand Anodyne SCD1 29 47 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(CC(=O)Nc3ccccc3F)nn2)C1 ZINC000880975982 GF On-Demand Anodyne GPR119 36 43 CC(C)(C)OC(=O)N1CC[C@H](c2cn(CC(=O)Nc3ccccc3F)nn2)C1 ZINC000880975983 GF On-Demand Anodyne GPR119 36 43 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCOC[C@@H](C)C1 ZINC000880975984 EH On-Demand Anodyne EPHX2 20 41 Cc1cc(C(F)(F)F)cc(C)c1NC(=O)N1CCOC[C@H](C)C1 ZINC000880975985 EH On-Demand Anodyne EPHX2 20 41 CC(C)(C)OC(=O)N1CCC(c2cn(CC(=O)NC3CCCCC3)nn2)CC1 ZINC000880976006 GF On-Demand Anodyne GPR119 43 41 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)c3cccnc3Cl)nn2)C1 ZINC000880976011 GD On-Demand Anodyne G2YM83_BOTF4 68 38 CNc1nc(C(=O)N2C[C@@H](C)[C@](C)(C(=O)OC)C2)cs1 ZINC000880976048 CD On-Demand Anodyne TRPC6 60 43 CNc1nc(C(=O)N2C[C@@H](C)[C@](C)(C(=O)OC)C2)cs1 ZINC000880976048 CD On-Demand Anodyne TRPC3 53 43 O=C(NCc1cn(Cc2cccc(C(F)(F)F)c2)nn1)C(F)(F)F ZINC000880976069 FF On-Demand Anodyne SCD1 23 42 COC(=O)Cc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880976074 CE On-Demand Anodyne SCD1 24 41 COC(=O)Cc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880976074 CE On-Demand Anodyne PDS 42 34 CC(C)(C)OC(=O)NCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880976085 FG On-Demand Anodyne SCD1 24 40 CC(C)(C)OC(=O)NCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880976085 FG On-Demand Anodyne PDS 44 39 O=C(Nc1cscc1Cl)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880976117 FH On-Demand Anodyne EPHX2 19 41 O=C(Nc1cscc1Cl)N1CC[C@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880976117 FH On-Demand Anodyne TRPM8 26 47 O=C(Nc1cscc1Cl)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880976118 FH On-Demand Anodyne EPHX2 19 41 O=C(Nc1cscc1Cl)N1CC[C@@]2(C[C@@H](O)c3ccccc3O2)C1 ZINC000880976118 FH On-Demand Anodyne TRPM8 26 47 O=C(Nc1cscc1Cl)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880976119 FH On-Demand Anodyne EPHX2 19 41 O=C(Nc1cscc1Cl)N1CC[C@@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880976119 FH On-Demand Anodyne TRPM8 26 47 O=C(Nc1cscc1Cl)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880976120 FH On-Demand Anodyne EPHX2 19 41 O=C(Nc1cscc1Cl)N1CC[C@]2(C[C@H](O)c3ccccc3O2)C1 ZINC000880976120 FH On-Demand Anodyne TRPM8 26 47 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880976121 GE On-Demand Anodyne PREP 29 42 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880976121 GE On-Demand Anodyne CAPNS1 42 32 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880976121 GE On-Demand Anodyne CAPN1 50 36 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880976121 GE On-Demand Anodyne CAPN2 84 35 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880976121 GE On-Demand Anodyne NPR 60 34 COc1ccc([C@@H](O)C2CCN(C(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880976182 GI On-Demand Anodyne NPBWR1 40 35 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880976233 GF On-Demand Anodyne MMP8 25 44 O=C(Nc1cscc1Cl)NN1CCCC1 ZINC000880976253 BF On-Demand Anodyne CNR1 40 31 CC(=O)N1CCN(Cc2cn(Cc3cccc(C(F)(F)F)c3)nn2)CC1 ZINC000880976271 FE On-Demand Anodyne FAAH 23 54 CC(=O)N1CCN(Cc2cn(Cc3cccc(C(F)(F)F)c3)nn2)CC1 ZINC000880976271 FE On-Demand Anodyne SCD1 20 40 O=C(Nc1cscc1Cl)N1CCC([C@H](O)c2cc(F)ccc2F)CC1 ZINC000880976278 GJ On-Demand Anodyne CACNA1H 49 36 O=C(Nc1cscc1Cl)N1CCC([C@@H](O)c2cc(F)ccc2F)CC1 ZINC000880976279 GJ On-Demand Anodyne CACNA1H 49 36 O=C(Nc1cscc1Cl)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880976321 FI On-Demand Anodyne CACNA1H 52 35 O=C(Nc1cscc1Cl)N1CCC(O)(c2c(F)cccc2F)CC1 ZINC000880976321 FI On-Demand Anodyne EPHX2 15 43 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cscc2Cl)C1 ZINC000880976377 DF On-Demand Anodyne EPHX2 36 44 CCOC(=O)N1CC[C@H](NC(=O)Nc2cscc2Cl)C1 ZINC000880976379 DF On-Demand Anodyne EPHX2 36 44 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1ccc(F)cc1 ZINC000880976427 FC On-Demand Anodyne EPHX2 15 42 O=C(Nc1cscc1Cl)N1CCC(C(=O)C(F)(F)F)CC1 ZINC000880976439 EH On-Demand Anodyne RBP4 46 38 O=C(Nc1cscc1Cl)N1CC[C@@](O)(c2ccc(F)cc2)C1 ZINC000880976462 EH On-Demand Anodyne CCR1 22 40 O=C(Nc1cscc1Cl)N1CC[C@](O)(c2ccc(F)cc2)C1 ZINC000880976463 EH On-Demand Anodyne CCR1 22 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCCc1ccc(F)cc1 ZINC000880976483 FE On-Demand Anodyne AMP1_PLAFQ 25 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCCc1ccc(F)cc1 ZINC000880976484 FE On-Demand Anodyne AMP1_PLAFQ 25 40 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NCc1ccc(F)cc1 ZINC000880976561 DD On-Demand Anodyne SSTR3 27 41 O=C(Cn1cc([C@H]2CCCCO2)nn1)NCc1ccc(F)cc1 ZINC000880976562 DD On-Demand Anodyne SSTR3 27 41 O=C(Nc1cscc1Cl)N1CCN(c2nc(F)c(F)cc2F)CC1 ZINC000880976573 GH On-Demand Anodyne RBP4 18 41 O=C(Nc1cscc1Cl)N1CC[C@@H](c2c(F)cccc2F)C1 ZINC000880976576 EJ On-Demand Anodyne RBP4 55 38 O=C(Nc1cscc1Cl)N1CC[C@H](c2c(F)cccc2F)C1 ZINC000880976577 EJ On-Demand Anodyne RBP4 55 38 COC(=O)N1CCC(NC(=O)Nc2cscc2Cl)CC1 ZINC000880976611 DF On-Demand Anodyne EPHX2 51 46 C[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)c3ccc(F)cc3)nn2)C1 ZINC000880976695 ED On-Demand Anodyne CCR3 44 31 C[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)c3ccc(F)cc3)nn2)C1 ZINC000880976697 ED On-Demand Anodyne CCR3 44 31 CC(=O)N1CCN(Cc2cn([C@H](C)C(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880976730 GD On-Demand Anodyne MCHR1 21 41 CC(=O)N1CCN(Cc2cn([C@@H](C)C(=O)Nc3cccc(Cl)c3)nn2)CC1 ZINC000880976731 GD On-Demand Anodyne MCHR1 21 41 C[C@H](O)c1cn(CC(=O)N2N=C(c3ccc(Cl)cc3)C[C@H]2c2ccco2)nn1 ZINC000880976782 GF On-Demand Anodyne GRIN2D 78 34 C[C@H](O)c1cn(CC(=O)N2N=C(c3ccc(Cl)cc3)C[C@@H]2c2ccco2)nn1 ZINC000880976784 GF On-Demand Anodyne GRIN2D 78 34 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cscc2Cl)C1 ZINC000880976846 FH On-Demand Anodyne EPHX2 20 41 COC(=O)[C@@]1(c2ccccc2)CCN(C(=O)Nc2cscc2Cl)C1 ZINC000880976846 FH On-Demand Anodyne RBP4 44 31 C[C@H]1CCC[C@H](C)N1C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880976852 GE On-Demand Anodyne G2YM83_BOTF4 76 41 C[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)c3ccc(Cl)cc3F)nn2)C1 ZINC000880976876 FE On-Demand Anodyne FDFT1 22 40 C[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)c3ccc(Cl)cc3F)nn2)C1 ZINC000880976878 FE On-Demand Anodyne FDFT1 22 40 O=C(Nc1cscc1Cl)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880977010 GG On-Demand Anodyne RBP4 60 38 O=C(Nc1cscc1Cl)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880977011 GG On-Demand Anodyne RBP4 60 38 O=C(Nc1cscc1Cl)N1CC[C@H]2CN(C(=O)C(F)(F)F)C[C@@H]2C1 ZINC000880977012 GG On-Demand Anodyne RBP4 60 38 O=C(Nc1cscc1Cl)N1CC[C@@H]2CN(C(=O)C(F)(F)F)C[C@H]2C1 ZINC000880977013 GG On-Demand Anodyne RBP4 60 38 O=C(Nc1cscc1Cl)N[C@H](CCO)Cc1ccccc1 ZINC000880977120 DH On-Demand Anodyne MME 72 40 O=C(Nc1cscc1Cl)N[C@H](CCO)Cc1ccccc1 ZINC000880977120 DH On-Demand Anodyne ANPEP 71 33 O=C(Nc1cscc1Cl)N[C@H](CCO)Cc1ccccc1 ZINC000880977120 DH On-Demand Anodyne GPR142 50 32 O=C(Nc1cscc1Cl)N[C@@H](CCO)Cc1ccccc1 ZINC000880977121 DH On-Demand Anodyne MME 72 40 O=C(Nc1cscc1Cl)N[C@@H](CCO)Cc1ccccc1 ZINC000880977121 DH On-Demand Anodyne ANPEP 71 33 O=C(Nc1cscc1Cl)N[C@@H](CCO)Cc1ccccc1 ZINC000880977121 DH On-Demand Anodyne GPR142 50 32 CC(C)(C)OC(=O)N1C[C@@H]2CN(C(=O)Nc3cscc3Cl)C[C@@H]2C1 ZINC000880977148 FH On-Demand Anodyne RBP4 45 33 C[C@@H]1CCCN(C(=O)Cn2cc(CCCOc3cccnc3F)nn2)C1 ZINC000880977219 FE On-Demand Anodyne MMP8 18 44 CC(=O)NCCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880977239 DE On-Demand Anodyne MTNR1A 39 46 CC(=O)NCCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880977239 DE On-Demand Anodyne MTNR1B 39 46 CC(=O)NCCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880977239 DE On-Demand Anodyne SCD1 21 40 CC(=O)NCCc1cn(Cc2cccc(C(F)(F)F)c2)nn1 ZINC000880977239 DE On-Demand Anodyne SCD 27 40 O=C(Nc1cscc1Cl)N1CCCN(c2ncccc2F)CC1 ZINC000880977276 FH On-Demand Anodyne TRPV1 15 54 O=C(Nc1cscc1Cl)N1CCCN(c2ncccc2F)CC1 ZINC000880977276 FH On-Demand Anodyne RBP4 25 52 O=C(Nc1cscc1Cl)N1CCC(O)(c2ccccc2)CC1 ZINC000880977278 EH On-Demand Anodyne OPRL1 17 42 O=C(Nc1cscc1Cl)N1CCC(O)(c2ccccc2)CC1 ZINC000880977278 EH On-Demand Anodyne CCR1 46 41 C[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)C1 ZINC000880977321 ED On-Demand Anodyne TRY1_BOVIN 42 33 C[C@@H]1CCCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)C1 ZINC000880977321 ED On-Demand Anodyne PREP 44 35 C[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)C1 ZINC000880977323 ED On-Demand Anodyne TRY1_BOVIN 42 33 C[C@@H]1CCCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)C1 ZINC000880977323 ED On-Demand Anodyne PREP 44 35 COC(=O)Cc1cn(CC(=O)Nc2cccc(SC)c2)nn1 ZINC000880977355 DD On-Demand Anodyne ENPP1 61 32 NC(=O)c1cc(OC2CCN(C(=O)Nc3cscc3Cl)CC2)ccn1 ZINC000880977366 GF On-Demand Anodyne EPHX2 20 44 NC(=O)c1cc(OC2CCN(C(=O)Nc3cscc3Cl)CC2)ccn1 ZINC000880977366 GF On-Demand Anodyne SCD1 20 45 O=C(Nc1cscc1Cl)NC12CCC(CC1)C2 ZINC000880977430 CH On-Demand Anodyne EPHX2 51 44 O=C(Nc1cscc1Cl)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880977484 EI On-Demand Anodyne EPHX2 26 48 O=C(Nc1cscc1Cl)N1CC[C@@]2(CCc3ccccc3O2)C1 ZINC000880977484 EI On-Demand Anodyne TRPM8 32 50 O=C(Nc1cscc1Cl)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880977485 EI On-Demand Anodyne EPHX2 26 48 O=C(Nc1cscc1Cl)N1CC[C@]2(CCc3ccccc3O2)C1 ZINC000880977485 EI On-Demand Anodyne TRPM8 32 50 CC(C)(C)OC(=O)N1CC(CNC(=O)Nc2cscc2Cl)C1 ZINC000880977540 EG On-Demand Anodyne CACNA1I 50 36 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880977541 GJ On-Demand Anodyne SIRT3 30 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880977541 GJ On-Demand Anodyne SIRT2 30 44 CC(C)(C)OC(=O)NCCC1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880977541 GJ On-Demand Anodyne SIRT1 30 44 O=C(Nc1cscc1Cl)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880977556 FI On-Demand Anodyne EPHX2 23 43 O=C(Nc1cscc1Cl)N1CCC(Oc2ccc(F)nc2)CC1 ZINC000880977556 FI On-Demand Anodyne SCD1 15 42 C[C@H](C(=O)Nc1cccc(Cl)c1)n1cc(CCCN2CCOCC2)nn1 ZINC000880977576 GE On-Demand Anodyne CASR 43 38 C[C@H](C(=O)Nc1cccc(Cl)c1)n1cc(CCCN2CCOCC2)nn1 ZINC000880977576 GE On-Demand Anodyne EPHX2 25 44 C[C@H](C(=O)Nc1cccc(Cl)c1)n1cc(CCCN2CCOCC2)nn1 ZINC000880977576 GE On-Demand Anodyne MCHR1 26 41 COCC(COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880977622 EE On-Demand Anodyne PDGFRB 30 40 COCC(COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880977622 EE On-Demand Anodyne KDR 56 38 COCC(COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880977622 EE On-Demand Anodyne PDGFRA 55 40 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977624 FF On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977624 FF On-Demand Anodyne CTSK 17 41 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977624 FF On-Demand Anodyne CTSL 24 42 COCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977624 FF On-Demand Anodyne CTSS 19 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977625 FF On-Demand Anodyne PAPA1_CARPA 38 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977625 FF On-Demand Anodyne CTSK 17 41 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977625 FF On-Demand Anodyne CTSL 24 42 COCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(OC)cc1F ZINC000880977625 FF On-Demand Anodyne CTSS 19 42 C=C[C@](C)(O)c1cn(CC(=O)Nc2nc3ccc(C)cc3s2)nn1 ZINC000880977626 EE On-Demand Mild CSNK1D 46 46 C=C[C@@](C)(O)c1cn(CC(=O)Nc2nc3ccc(C)cc3s2)nn1 ZINC000880977627 EE On-Demand Mild CSNK1D 46 46 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCCc1ccc(Cl)cc1 ZINC000880977668 GD On-Demand Anodyne MRGPRX1 22 40 CNC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880977678 FD On-Demand Anodyne PDGFRA 46 38 O=C(Nc1cscc1Cl)N[C@H]1CCOC1=O ZINC000880977736 CD On-Demand Anodyne LUXR 75 43 O=C(Nc1cscc1Cl)N[C@H]1CCOC1=O ZINC000880977736 CD On-Demand Anodyne TRAR 91 43 O=C(Nc1cscc1Cl)N[C@H]1CCOC1=O ZINC000880977736 CD On-Demand Anodyne LASR 63 39 CN1CC[C@@H](CNC(=O)Nc2cscc2Cl)[C@@H]1c1cccnc1 ZINC000880977747 FH On-Demand Anodyne NAMPT 40 36 O=C(Nc1cscc1Cl)NN1CCCCC1 ZINC000880977749 CF On-Demand Anodyne CNR1 51 32 O=C(NCc1cn(Cc2cccc(C(F)(F)F)c2)nn1)OCC(F)(F)F ZINC000880977764 GG On-Demand Anodyne PDS 43 44 COC(=O)CCCCCCCNC(=O)Nc1cscc1Cl ZINC000880977771 EI On-Demand Anodyne EPHX2 15 45 O=C(Nc1cscc1Cl)N1CCC(CNC(=O)C(F)(F)F)CC1 ZINC000880977787 FG On-Demand Anodyne CACNA1I 57 34 C[C@@H](C[C@H](O)c1ccccc1)NC(=O)Nc1cscc1Cl ZINC000880977796 DI On-Demand Anodyne CAPN2 49 38 C[C@H](C[C@@H](O)c1ccccc1)NC(=O)Nc1cscc1Cl ZINC000880977800 DI On-Demand Anodyne CAPN2 49 38 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(OC)cc2OC)nn1 ZINC000880977820 ED On-Demand Anodyne SOAT1 22 41 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne F2 41 38 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne ACE 24 41 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne ELANE 23 40 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne CTRA_BOVIN 52 30 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne KLK3 68 33 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne TRY1_BOVIN 68 38 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne CTSK 31 40 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne PREP 56 47 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne CAPNS1 46 32 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne CAPN1 56 37 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne CAPN2 80 37 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne NPR 62 35 C[C@@H]1CCCN(C(=O)Cn2cc(CNC(=O)OCc3ccccc3)nn2)C1 ZINC000880977866 FD On-Demand Anodyne TMPRSS11D 43 37 O=C(Nc1cscc1Cl)N1CCC(O)(Cc2cccc(F)c2)CC1 ZINC000880977876 FI On-Demand Anodyne CACNA1H 61 37 CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)Nc2cscc2Cl)C1 ZINC000880977879 FH On-Demand Anodyne CACNA1I 73 40 CC(C)(C)OC(=O)N1CC[C@H](CNC(=O)Nc2cscc2Cl)C1 ZINC000880977883 FH On-Demand Anodyne CACNA1I 73 40 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3cscc3Cl)C2)CC1 ZINC000880977908 GJ On-Demand Anodyne EPHX2 25 41 CC(C)(C)OC(=O)N1CCC2(CCN(C(=O)Nc3cscc3Cl)C2)CC1 ZINC000880977908 GJ On-Demand Anodyne GPR119 16 48 CCOC(=O)N1CCCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880977919 EG On-Demand Anodyne P2RY12 25 41 O=C(NCc1ccccc1N1CCOCC1)Nc1cscc1Cl ZINC000880977948 FH On-Demand Anodyne KCNQ2 53 44 O=C(NCc1ccccc1N1CCOCC1)Nc1cscc1Cl ZINC000880977948 FH On-Demand Anodyne P2RX7 20 45 O=C(NCc1ccccc1N1CCOCC1)Nc1cscc1Cl ZINC000880977948 FH On-Demand Anodyne SCN2A 17 40 O=C(NCc1ccccc1N1CCOCC1)Nc1cscc1Cl ZINC000880977948 FH On-Demand Anodyne SCN10A 22 52 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCCc1ccc(F)cc1 ZINC000880977950 GD On-Demand Anodyne EPHX2 15 42 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccc(F)c3)nn2)CC1 ZINC000880977957 FC On-Demand Anodyne AURKB 16 40 Cc1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1F ZINC000880978005 FD On-Demand Anodyne CHRNA7 18 43 Cc1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)cc1F ZINC000880978005 FD On-Demand Anodyne EPHX2 24 44 CCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978018 FE On-Demand Anodyne PDGFRB 51 38 CCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978018 FE On-Demand Anodyne KDR 40 36 CCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978018 FE On-Demand Anodyne PDGFRA 50 35 O=C(Cn1cc(C2(O)CCC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978031 ED On-Demand Anodyne BDKRB1 47 41 O=C(Cn1cc(C2(O)CCC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978032 ED On-Demand Anodyne BDKRB1 47 41 O=C(Cn1cc(-c2cccnc2F)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978040 FF On-Demand Anodyne BDKRB1 43 39 O=C(Cn1cc(-c2cccnc2F)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978041 FF On-Demand Anodyne BDKRB1 43 39 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCCc1ccc(Cl)cc1 ZINC000880978047 GF On-Demand Anodyne BRS3 19 41 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)NCCc1ccc(Cl)cc1 ZINC000880978047 GF On-Demand Anodyne AMP1_PLAFQ 26 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCCc1ccc(Cl)cc1 ZINC000880978048 GF On-Demand Anodyne BRS3 19 41 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)NCCc1ccc(Cl)cc1 ZINC000880978048 GF On-Demand Anodyne AMP1_PLAFQ 26 40 CC[C@@](C)(O)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978053 EE On-Demand Anodyne BDKRB1 55 41 CC[C@@](C)(O)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978054 EE On-Demand Anodyne BDKRB1 55 41 C[C@H](N)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978084 CD On-Demand Anodyne BDKRB1 59 40 C[C@H](N)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978084 CD On-Demand Anodyne XIAP 29 40 C[C@H](N)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978084 CD On-Demand Anodyne BIRC3 34 41 C[C@H](N)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978084 CD On-Demand Anodyne BIRC2 42 40 C[C@H](N)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978086 CD On-Demand Anodyne BDKRB1 59 40 C[C@H](N)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978086 CD On-Demand Anodyne XIAP 29 40 C[C@H](N)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978086 CD On-Demand Anodyne BIRC3 34 41 C[C@H](N)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978086 CD On-Demand Anodyne BIRC2 42 40 C[C@H](C(=O)Nc1cccc(Cl)c1)n1cc(C(C)(C)O)nn1 ZINC000880978096 DE On-Demand Anodyne IMDH_CRYPV 23 40 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NCc1ccc(F)cc1 ZINC000880978101 GE On-Demand Anodyne MMP8 17 43 O=C(Cn1cc(CCCOc2cccnc2F)nn1)NCc1ccc(F)cc1 ZINC000880978101 GE On-Demand Anodyne SUCNR1 54 38 O=C(Nc1cscc1Cl)N1CC[C@H](c2ccccn2)C1 ZINC000880978120 DH On-Demand Anodyne GRM4 40 38 O=C(Nc1cscc1Cl)N1CC[C@H](c2ccccn2)C1 ZINC000880978120 DH On-Demand Anodyne RBP4 61 38 O=C(Nc1cscc1Cl)N1CC[C@H](c2ccccn2)C1 ZINC000880978120 DH On-Demand Anodyne SMO 26 40 O=C(Nc1cscc1Cl)N1CC[C@@H](c2ccccn2)C1 ZINC000880978121 DH On-Demand Anodyne GRM4 40 38 O=C(Nc1cscc1Cl)N1CC[C@@H](c2ccccn2)C1 ZINC000880978121 DH On-Demand Anodyne RBP4 61 38 O=C(Nc1cscc1Cl)N1CC[C@@H](c2ccccn2)C1 ZINC000880978121 DH On-Demand Anodyne SMO 26 40 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cscc1Cl ZINC000880978158 FG On-Demand Anodyne EPHX2 17 52 O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)Nc1cscc1Cl ZINC000880978158 FG On-Demand Anodyne CACNA1I 62 36 CC(=O)c1ccc(NC(=O)[C@H](C)n2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880978161 GD On-Demand Anodyne CHRNA7 17 40 CC(=O)c1ccc(NC(=O)[C@H](C)n2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880978161 GD On-Demand Anodyne EPHX2 21 40 CC(=O)c1ccc(NC(=O)[C@@H](C)n2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880978163 GD On-Demand Anodyne CHRNA7 17 40 CC(=O)c1ccc(NC(=O)[C@@H](C)n2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880978163 GD On-Demand Anodyne EPHX2 21 40 O=C(NCC1CCN(S(=O)(=O)C(F)F)CC1)Nc1cscc1Cl ZINC000880978167 GF On-Demand Anodyne CACNA1I 45 33 CC(C)(C)OC(=O)NC[C@@H]1CCN(C(=O)Nc2cscc2Cl)C1 ZINC000880978176 FH On-Demand Anodyne CACNA1I 61 38 CC(C)(C)OC(=O)NC[C@H]1CCN(C(=O)Nc2cscc2Cl)C1 ZINC000880978179 FH On-Demand Anodyne CACNA1I 61 38 Cc1cccc2c1CCN(C(=O)Nc1cscc1Cl)C2 ZINC000880978211 DI On-Demand Anodyne P2RY14 48 35 O=C(Nc1cscc1Cl)N1CCC(O)(c2ccccc2Cl)CC1 ZINC000880978216 FJ On-Demand Anodyne NPY5R 36 45 COC(=O)CCCCCCNC(=O)Nc1cscc1Cl ZINC000880978253 DH On-Demand Anodyne EPHX2 15 45 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(F)c1 ZINC000880978259 DE On-Demand Anodyne AURKB 24 40 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(F)c1 ZINC000880978259 DE On-Demand Anodyne HDAC10 24 41 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(F)c1 ZINC000880978259 DE On-Demand Anodyne HDAC3 29 41 O=C(Cn1cc(CCCCCCO)nn1)Nc1cccc(F)c1 ZINC000880978259 DE On-Demand Anodyne HDAC6 24 41 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880978264 EG On-Demand Anodyne F13A1 16 42 CC(C)(C)OC(=O)N1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880978264 EG On-Demand Anodyne GPR119 33 44 CN(C(=O)Nc1cscc1Cl)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000880978285 FI On-Demand Anodyne GPR119 41 41 COc1ccc(NC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)c(F)c1 ZINC000880978369 EE On-Demand Anodyne MTNR1A 17 41 COc1ccc(NC(=O)[C@H]2C[C@@H]3CC[C@H](C2)S3(=O)=O)c(F)c1 ZINC000880978369 EE On-Demand Anodyne MTNR1B 18 41 Cc1nc(C(C)C)ncc1C(=O)Nc1cc(F)cc(C#N)c1 ZINC000880978383 CG On-Demand Mild JUN 20 43 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978419 GF On-Demand Anodyne BDKRB1 54 39 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978420 GF On-Demand Anodyne BDKRB1 54 39 COCCO[C@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978430 GF On-Demand Anodyne PDGFRB 41 34 COCCO[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978431 GF On-Demand Anodyne PDGFRB 41 34 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(F)c1 ZINC000880978441 ED On-Demand Anodyne CHRNA7 15 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(F)c1 ZINC000880978441 ED On-Demand Anodyne EPHX2 24 49 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cccc(F)c1 ZINC000880978441 ED On-Demand Anodyne AURKA 26 43 CCOC(=O)CCCCCCNC(=O)Nc1cscc1Cl ZINC000880978449 EI On-Demand Anodyne EPHX2 18 48 CC[C@@](C)(O)c1cn(CC(=O)Nc2nc(-c3ccccc3)cs2)nn1 ZINC000880978458 FF On-Demand Anodyne ROCK1 20 41 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne PIK3CA 33 40 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne CHRNA7 15 47 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne PRNP 41 37 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne MTOR 52 40 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne EPHX2 16 42 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978481 GE On-Demand Anodyne PIK3CG 30 40 Cc1c(NC(=O)[C@@H](C)n2cc([C@H]3CCOC3)nn2)c(=O)n(-c2ccccc2)n1C ZINC000880978506 GD On-Demand Anodyne FPR2 43 39 Cc1c(NC(=O)[C@H](C)n2cc([C@H]3CCOC3)nn2)c(=O)n(-c2ccccc2)n1C ZINC000880978507 GD On-Demand Anodyne FPR2 43 39 Cc1c(NC(=O)[C@@H](C)n2cc([C@@H]3CCOC3)nn2)c(=O)n(-c2ccccc2)n1C ZINC000880978508 GD On-Demand Anodyne FPR2 43 39 Cc1c(NC(=O)[C@H](C)n2cc([C@@H]3CCOC3)nn2)c(=O)n(-c2ccccc2)n1C ZINC000880978509 GD On-Demand Anodyne FPR2 43 39 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(F)c3)nn2)CC1 ZINC000880978519 FF On-Demand Anodyne AURKB 17 42 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(F)c3)nn2)CC1 ZINC000880978519 FF On-Demand Anodyne HDAC10 19 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(F)c3)nn2)CC1 ZINC000880978519 FF On-Demand Anodyne HDAC3 21 40 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccc(F)c3)nn2)CC1 ZINC000880978519 FF On-Demand Anodyne HDAC6 18 40 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cscc1Cl ZINC000880978522 FH On-Demand Anodyne L3MBTL3 47 38 O=C(NCc1ccc(C(=O)N2CCCC2)cc1)Nc1cscc1Cl ZINC000880978522 FH On-Demand Anodyne NAMPT 26 51 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc([C@@H](C)O)nn2)c1 ZINC000880978523 DD On-Demand Anodyne KCNK3 43 32 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc([C@H](C)O)nn2)c1 ZINC000880978524 DD On-Demand Anodyne KCNK3 43 32 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc([C@@H](C)O)nn2)c1 ZINC000880978525 DD On-Demand Anodyne KCNK3 43 32 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc([C@H](C)O)nn2)c1 ZINC000880978526 DD On-Demand Anodyne KCNK3 43 32 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880978538 FE On-Demand Anodyne SLC12A5 20 42 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880978539 FE On-Demand Anodyne SLC12A5 20 42 COCCCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978547 EE On-Demand Anodyne KDR 65 38 COCCCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978547 EE On-Demand Anodyne PDGFRA 53 39 O=C(Cn1cc([C@@H]2CCCCO2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978568 EF On-Demand Anodyne BDKRB1 46 38 O=C(Cn1cc([C@H]2CCCCO2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978569 EF On-Demand Anodyne BDKRB1 46 38 O=C(Cn1cc([C@H]2CCCCO2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978570 EF On-Demand Anodyne BDKRB1 46 38 O=C(Cn1cc([C@@H]2CCCCO2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978571 EF On-Demand Anodyne BDKRB1 46 38 COC(=O)Cc1cn(CC(=O)Nc2nc3ccc(C)cc3s2)nn1 ZINC000880978578 ED On-Demand Anodyne CSNK1D 52 54 O=C(Cn1cc(CN2CCOC2=O)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978589 FD On-Demand Anodyne BDKRB1 49 36 O=C(Cn1cc(CN2CCOC2=O)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978590 FD On-Demand Anodyne BDKRB1 49 36 O=C(Cn1cc(C2(O)CCCCC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978599 FF On-Demand Anodyne BDKRB1 43 39 O=C(Cn1cc(C2(O)CCCCC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978600 FF On-Demand Anodyne BDKRB1 43 39 CC#CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978601 DF On-Demand Mild KDR 59 37 CC#CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978601 DF On-Demand Mild PDGFRA 54 40 COC(=O)Cc1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978608 ED On-Demand Anodyne BDKRB1 45 39 COC(=O)Cc1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978608 ED On-Demand Anodyne BIRC3 26 40 COC(=O)Cc1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978608 ED On-Demand Anodyne BIRC2 41 37 COC(=O)Cc1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978609 ED On-Demand Anodyne BDKRB1 45 39 COC(=O)Cc1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978609 ED On-Demand Anodyne BIRC3 26 40 COC(=O)Cc1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978609 ED On-Demand Anodyne BIRC2 41 37 COCC[C@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978612 FE On-Demand Anodyne KDR 56 36 COCC[C@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978612 FE On-Demand Anodyne PDGFRA 51 38 COCC[C@@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978613 FE On-Demand Anodyne KDR 56 36 COCC[C@@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978613 FE On-Demand Anodyne PDGFRA 51 38 N#Cc1cc(F)cc(NC(=O)[C@H]2CC[C@@H](C(N)=O)N2Cc2ccccc2)c1 ZINC000880978615 FE On-Demand Mild CCR3 24 41 CC[C@H](O)c1cn(CC(=O)Nc2nc3ccc(C)cc3s2)nn1 ZINC000880978618 EE On-Demand Anodyne CSNK1D 46 48 CC(=O)N1CCN(Cc2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)CC1 ZINC000880978630 GD On-Demand Anodyne HTR7 15 47 CC(=O)N1CCN(Cc2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)CC1 ZINC000880978630 GD On-Demand Anodyne BDKRB1 56 39 CC(=O)N1CCN(Cc2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)CC1 ZINC000880978631 GD On-Demand Anodyne HTR7 15 47 CC(=O)N1CCN(Cc2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)CC1 ZINC000880978631 GD On-Demand Anodyne BDKRB1 56 39 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccccc3)cs2)nn1 ZINC000880978652 EE On-Demand Anodyne ROCK1 21 46 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccccc3)cs2)nn1 ZINC000880978652 EE On-Demand Anodyne TRPA1 15 48 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccccc3)cs2)nn1 ZINC000880978652 EE On-Demand Anodyne SLC12A5 17 45 COc1ccc(N2CCCN(C(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880978679 FI On-Demand Clean RBP4 20 42 COc1ccc(N2CCCN(C(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880978679 FI On-Demand Clean NPBWR1 69 34 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cscc2Cl)CC1 ZINC000880978680 FH On-Demand Anodyne EPHX2 49 43 CC(C)(C)OC(=O)N1CCC(NC(=O)Nc2cscc2Cl)CC1 ZINC000880978680 FH On-Demand Anodyne GPR119 44 41 COc1ccc(OC)c([C@H](O)CNC(=O)Nc2cscc2Cl)c1 ZINC000880978688 FG On-Demand Anodyne MTNR1A 19 43 CN(Cc1cn(CC(=O)Nc2cccc(F)c2)nn1)C(=O)OC(C)(C)C ZINC000880978690 FE On-Demand Anodyne AURKB 19 42 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc(C(C)(C)O)nn2)c1 ZINC000880978698 DD On-Demand Anodyne IMDH_CRYPV 49 34 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc(C(C)(C)O)nn2)c1 ZINC000880978699 DD On-Demand Anodyne IMDH_CRYPV 49 34 CC[C@H](O)c1cn(CC(=O)Nc2ccc(OC)cc2OC)nn1 ZINC000880978704 DD On-Demand Anodyne PDGFRB 42 39 O=C(Cn1cc(CCN2CCNCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978709 GE On-Demand Anodyne CHRNA7 17 45 CC(C)(C)OC(=O)NCc1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880978729 EE On-Demand Anodyne AURKB 19 43 CC[C@@H](CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12)OC ZINC000880978757 EF On-Demand Anodyne KDR 40 39 CC[C@@H](CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12)OC ZINC000880978757 EF On-Demand Anodyne PDGFRA 56 40 COC(=O)c1cccc(C#Cc2cccc(NC(=O)CN(C)C3=NS(=O)(=O)c4ccccc43)c2)c1 ZINC000880978758 JF On-Demand Mild KCNA3 20 42 CCc1nc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)co1 ZINC000880978768 FG On-Demand Anodyne PDGFRA 44 37 O=C1CCC[C@@H](c2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)C1 ZINC000880978772 FF On-Demand Anodyne BDKRB1 50 39 O=C1CCC[C@@H](c2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)C1 ZINC000880978772 FF On-Demand Anodyne BIRC3 31 41 O=C1CCC[C@H](c2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)C1 ZINC000880978773 FF On-Demand Anodyne BDKRB1 50 39 O=C1CCC[C@H](c2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)C1 ZINC000880978773 FF On-Demand Anodyne BIRC3 31 41 O=C1CCC[C@@H](c2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)C1 ZINC000880978774 FF On-Demand Anodyne BDKRB1 50 39 O=C1CCC[C@@H](c2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)C1 ZINC000880978774 FF On-Demand Anodyne BIRC3 31 41 O=C1CCC[C@H](c2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)C1 ZINC000880978775 FF On-Demand Anodyne BDKRB1 50 39 O=C1CCC[C@H](c2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)C1 ZINC000880978775 FF On-Demand Anodyne BIRC3 31 41 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880978779 FH On-Demand Anodyne PDGFRB 56 38 COC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978780 DE On-Demand Anodyne PDGFRB 30 41 COC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978780 DE On-Demand Anodyne KDR 52 38 COC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978780 DE On-Demand Anodyne PDGFRA 53 41 COC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978781 DE On-Demand Anodyne PDGFRB 30 41 COC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978781 DE On-Demand Anodyne KDR 52 38 COC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978781 DE On-Demand Anodyne PDGFRA 53 41 C=C[C@@H]1OCC[C@H]1NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978784 EF On-Demand Mild PDGFRA 47 38 O=C(Cn1cc([C@@H]2CCOC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978785 ED On-Demand Anodyne BDKRB1 40 37 O=C(Cn1cc([C@H]2CCOC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978786 ED On-Demand Anodyne BDKRB1 40 37 O=C(Cn1cc([C@H]2CCOC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978787 ED On-Demand Anodyne BDKRB1 40 37 O=C(Cn1cc([C@@H]2CCOC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978788 ED On-Demand Anodyne BDKRB1 40 37 COCC1(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCC1 ZINC000880978794 EF On-Demand Anodyne KDR 40 36 COCC1(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCC1 ZINC000880978794 EF On-Demand Anodyne PDGFRA 51 37 C=CCC[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978816 EF On-Demand Mild PDGFRA 48 37 C=CCC[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978817 EF On-Demand Mild PDGFRA 48 37 N#Cc1cc(F)cc(NC(=O)CN2CCCCS2(=O)=O)c1 ZINC000880978827 DD On-Demand Mild MCHR1 22 40 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@H](C)O ZINC000880978829 EF On-Demand Anodyne PDGFRB 31 40 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@H](C)O ZINC000880978829 EF On-Demand Anodyne KDR 44 37 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@H](C)O ZINC000880978829 EF On-Demand Anodyne PDGFRA 52 40 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@@H](C)O ZINC000880978831 EF On-Demand Anodyne PDGFRB 31 40 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@@H](C)O ZINC000880978831 EF On-Demand Anodyne KDR 44 37 CC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@@H](C)O ZINC000880978831 EF On-Demand Anodyne PDGFRA 52 40 N#Cc1cc(F)cc(NC(=O)c2ccc(CN3CCOCC3)o2)c1 ZINC000880978837 EE On-Demand Mild CSF1R 25 42 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880978859 GG On-Demand Anodyne ROCK1 20 41 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880978859 GG On-Demand Anodyne SLC12A5 15 40 O=C(NCc1ccc(N2CCOCC2)cc1)Nc1cscc1Cl ZINC000880978860 FH On-Demand Clean STAT6 53 36 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978863 EI On-Demand Mild ROCK1 17 40 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978863 EI On-Demand Mild ROCK2 28 44 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978863 EI On-Demand Mild PDS 56 38 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978864 EI On-Demand Mild ROCK1 17 40 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978864 EI On-Demand Mild ROCK2 28 44 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cscc2Cl)c1 ZINC000880978864 EI On-Demand Mild PDS 56 38 CC(C)(C)OC(=O)NC[C@H]1CCCN(C(=O)Nc2cscc2Cl)C1 ZINC000880978865 FI On-Demand Anodyne CACNA1I 44 35 CC(C)(C)OC(=O)NC[C@@H]1CCCN(C(=O)Nc2cscc2Cl)C1 ZINC000880978866 FI On-Demand Anodyne CACNA1I 44 35 COc1ccc(N2CCC(NC(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880978867 FI On-Demand Clean EPHX2 48 39 COc1ccc(N2CCC(NC(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880978867 FI On-Demand Clean PDK1 49 35 COc1ccc(N2CCC(NC(=O)Nc3cscc3Cl)CC2)cc1 ZINC000880978867 FI On-Demand Clean NPBWR1 51 34 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978896 FG On-Demand Anodyne HDAC10 36 41 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978896 FG On-Demand Anodyne HDAC1 18 53 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978896 FG On-Demand Anodyne HDAC2 18 44 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978896 FG On-Demand Anodyne HDAC3 29 43 O=C(Cn1cc(CCCCCO)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880978896 FG On-Demand Anodyne HDAC6 28 44 O=C(Nc1cscc1Cl)NC1CCC(N2CCCCC2)CC1 ZINC000880978903 EI On-Demand Anodyne EPHX2 21 40 O=C(Nc1cscc1Cl)NC1CCC(N2CCCCC2)CC1 ZINC000880978903 EI On-Demand Anodyne L3MBTL3 54 35 O=C(Nc1cscc1Cl)N1CCCN(C(=O)Oc2ccccc2)CC1 ZINC000880978906 GI On-Demand Anodyne FAAH 23 42 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880978935 FH On-Demand Anodyne F13A1 16 40 CC(C)(C)OC(=O)N1CCCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880978935 FH On-Demand Anodyne GPR119 28 42 COC[C@@]1(C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978942 FG On-Demand Anodyne PDGFRA 41 33 COC[C@]1(C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978943 FG On-Demand Anodyne PDGFRA 41 33 COc1ccc(NC(=O)[C@H]2CCc3nncn3CC2)c(F)c1 ZINC000880978947 DE On-Demand Anodyne MTNR1B 15 40 COc1ccc(NC(=O)[C@@H]2CCc3nncn3CC2)c(F)c1 ZINC000880978948 DE On-Demand Anodyne MTNR1B 15 40 O=C(Cn1cc(CCCN2CCOCC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880978953 GD On-Demand Anodyne HTR7 15 52 O=C(Cn1cc(CCCN2CCOCC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880978954 GD On-Demand Anodyne HTR7 15 52 CCc1nnc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)s1 ZINC000880978962 FF On-Demand Anodyne PDGFRA 50 36 CCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978963 EE On-Demand Anodyne PDGFRB 48 39 CCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978963 EE On-Demand Anodyne KDR 48 35 CCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880978963 EE On-Demand Anodyne PDGFRA 51 36 C=C[C@@](C)(O)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978966 ED On-Demand Mild BDKRB1 56 39 C=C[C@@](C)(O)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978967 ED On-Demand Mild BDKRB1 56 39 C=C[C@](C)(O)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880978968 ED On-Demand Mild BDKRB1 56 39 C=C[C@](C)(O)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880978969 ED On-Demand Mild BDKRB1 56 39 Cc1ccc(NC(=O)Cn2cc([C@@](C)(O)Cc3ccccc3)nn2)cc1F ZINC000880978979 FF On-Demand Anodyne FPR2 25 40 Cc1ccc(NC(=O)Cn2cc([C@](C)(O)Cc3ccccc3)nn2)cc1F ZINC000880978980 FF On-Demand Anodyne FPR2 25 40 COCC[C@@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978981 EG On-Demand Anodyne KDR 47 36 COCC[C@@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978981 EG On-Demand Anodyne PDGFRA 50 37 COCC[C@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978982 EG On-Demand Anodyne KDR 47 36 COCC[C@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880978982 EG On-Demand Anodyne PDGFRA 50 37 CC[C@@](C)(O)c1cn(CC(=O)Nc2nc3ccc(C)cc3s2)nn1 ZINC000880979021 EE On-Demand Anodyne CSNK1D 47 47 Nc1cccc(OCc2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)c1 ZINC000880979022 GF On-Demand Anodyne BDKRB1 45 35 Nc1cccc(OCc2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)c1 ZINC000880979023 GF On-Demand Anodyne BDKRB1 45 35 CC[C@H](O)c1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1 ZINC000880979028 DD On-Demand Anodyne BDKRB1 47 39 CC[C@H](O)c1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1 ZINC000880979029 DD On-Demand Anodyne BDKRB1 47 39 C=CCN(CCC#N)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979036 EG On-Demand Mild PDGFRA 40 34 CC(C)(C)N1CCC(NC(=O)Nc2cscc2Cl)CC1 ZINC000880979141 DH On-Demand Anodyne EPHX2 41 41 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880979145 FG On-Demand Anodyne CPT1A 34 43 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880979146 FG On-Demand Anodyne CPT1A 34 43 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc2c(c1)OCCO2 ZINC000880979149 GC On-Demand Anodyne EPHX2 21 46 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979189 EG On-Demand Anodyne CA4 15 40 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979189 EG On-Demand Anodyne HDAC3 22 40 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979189 EG On-Demand Anodyne HDAC6 19 41 CC[C@@](C)(N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979189 EG On-Demand Anodyne SLC1A2 21 40 N#Cc1cc(NC(=O)Nc2cscc2Cl)ccc1N1CCC(O)CC1 ZINC000880979190 GH On-Demand Mild NPY2R 50 37 COC[C@@H](O)Cc1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979200 DC On-Demand Anodyne AURKB 22 44 COCCCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979240 EG On-Demand Anodyne KDR 66 36 COCCCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979240 EG On-Demand Anodyne PDGFRA 53 39 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979254 GF On-Demand Anodyne ACE 34 42 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979254 GF On-Demand Anodyne BDKRB1 49 38 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979254 GF On-Demand Anodyne BIRC3 28 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979254 GF On-Demand Anodyne BIRC2 28 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979255 GF On-Demand Anodyne ACE 34 42 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979255 GF On-Demand Anodyne BDKRB1 49 38 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979255 GF On-Demand Anodyne BIRC3 28 40 O=C(Cn1cc([C@@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979255 GF On-Demand Anodyne BIRC2 28 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979256 GF On-Demand Anodyne ACE 34 42 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979256 GF On-Demand Anodyne BDKRB1 49 38 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979256 GF On-Demand Anodyne BIRC3 28 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979256 GF On-Demand Anodyne BIRC2 28 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979257 GF On-Demand Anodyne ACE 34 42 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979257 GF On-Demand Anodyne BDKRB1 49 38 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979257 GF On-Demand Anodyne BIRC3 28 40 O=C(Cn1cc([C@H](O)Cc2ccccc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979257 GF On-Demand Anodyne BIRC2 28 40 O=C(Cn1cc([C@H](O)C2CC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979287 ED On-Demand Anodyne BDKRB1 40 38 O=C(Cn1cc([C@H](O)C2CC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979288 ED On-Demand Anodyne BDKRB1 40 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979289 ED On-Demand Anodyne BDKRB1 40 38 O=C(Cn1cc([C@@H](O)C2CC2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979290 ED On-Demand Anodyne BDKRB1 40 38 COC(=O)C1CCC(c2cn(CC(=O)N[C@@H]3CCCc4ccccc43)nn2)CC1 ZINC000880979297 GF On-Demand Anodyne BDKRB1 53 39 COC(=O)C1CCC(c2cn(CC(=O)N[C@H]3CCCc4ccccc43)nn2)CC1 ZINC000880979298 GF On-Demand Anodyne BDKRB1 53 39 COc1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979317 EH On-Demand Anodyne NQO2 26 41 COc1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979317 EH On-Demand Anodyne MTNR1A 24 40 COc1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979317 EH On-Demand Anodyne MTNR1B 23 40 COc1ccc(NC(=O)[C@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979317 EH On-Demand Anodyne ROCK2 22 42 COc1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979318 EH On-Demand Anodyne NQO2 26 41 COc1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979318 EH On-Demand Anodyne MTNR1A 24 40 COc1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979318 EH On-Demand Anodyne MTNR1B 23 40 COc1ccc(NC(=O)[C@@H]2CCc3cc(OC)ccc3C2)c(F)c1 ZINC000880979318 EH On-Demand Anodyne ROCK2 22 42 CC(C)(C)OC(=O)NC(C)(C)c1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979327 GF On-Demand Anodyne AURKB 17 43 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880979328 EE On-Demand Anodyne HDAC10 17 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880979328 EE On-Demand Anodyne HDAC3 20 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880979329 EE On-Demand Anodyne HDAC10 17 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880979329 EE On-Demand Anodyne HDAC3 20 40 CC(C)(C)OC(=O)NCC1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880979333 FI On-Demand Anodyne CACNA1I 54 37 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979341 GG On-Demand Anodyne CCR3 34 41 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979341 GG On-Demand Anodyne AURKB 20 40 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979342 GG On-Demand Anodyne CCR3 34 41 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(CC(=O)Nc2cccc(F)c2)nn1 ZINC000880979342 GG On-Demand Anodyne AURKB 20 40 O=C(Nc1cscc1Cl)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880979384 FH On-Demand Anodyne FAAH 26 47 O=C(Nc1cscc1Cl)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880979384 FH On-Demand Anodyne Q8WSF8_APLCA 42 39 O=C(Nc1cscc1Cl)N1CCN(Cc2ccc(Cl)nc2)CC1 ZINC000880979384 FH On-Demand Anodyne NACHRBETA2 48 39 O=C(Nc1cscc1Cl)N1CCN(C[C@H](O)c2ccccc2)CC1 ZINC000880979388 FG On-Demand Anodyne FAAH 19 42 O=C(Nc1cscc1Cl)N1CCN(C[C@@H](O)c2ccccc2)CC1 ZINC000880979389 FG On-Demand Anodyne FAAH 19 42 O=C(Cn1cc(C[C@H](O)C2CC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979393 FF On-Demand Anodyne PRNP 41 35 O=C(Cn1cc(C[C@@H](O)C2CC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979394 FF On-Demand Anodyne PRNP 41 35 CC(=O)c1ccc(N2CCN(C(=O)Nc3cscc3Cl)CC2)c(F)c1 ZINC000880979398 GI On-Demand Anodyne NPY2R 80 42 CC(=O)c1ccc(N2CCN(C(=O)Nc3cscc3Cl)CC2)c(F)c1 ZINC000880979398 GI On-Demand Anodyne SLC6A9 23 45 CC(=O)c1ccc(N2CCN(C(=O)Nc3cscc3Cl)CC2)c(F)c1 ZINC000880979398 GI On-Demand Anodyne RBP4 19 44 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880979419 FE On-Demand Anodyne ROCK1 20 42 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880979419 FE On-Demand Anodyne HDAC9 15 46 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1nc(-c2ccccc2)cs1 ZINC000880979419 FE On-Demand Anodyne SLC12A5 16 41 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979420 FG On-Demand Anodyne CHRNA7 20 52 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979420 FG On-Demand Anodyne HDAC6 16 42 O=C(Cn1cc(CN2CCCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979420 FG On-Demand Anodyne MCHR1 15 45 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979426 DE On-Demand Anodyne HDAC10 18 42 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979426 DE On-Demand Anodyne HDAC3 20 42 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979426 DE On-Demand Anodyne HDAC6 16 42 CN(Cc1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1)C(=O)OC(C)(C)C ZINC000880979441 GF On-Demand Anodyne XIAP 27 40 CN(Cc1cn(CC(=O)N[C@@H]2CCCc3ccccc32)nn1)C(=O)OC(C)(C)C ZINC000880979441 GF On-Demand Anodyne BIRC2 47 34 CN(Cc1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1)C(=O)OC(C)(C)C ZINC000880979442 GF On-Demand Anodyne XIAP 27 40 CN(Cc1cn(CC(=O)N[C@H]2CCCc3ccccc32)nn1)C(=O)OC(C)(C)C ZINC000880979442 GF On-Demand Anodyne BIRC2 47 34 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979445 FF On-Demand Anodyne BDKRB1 41 36 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979446 FF On-Demand Anodyne BDKRB1 41 36 CCC1(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)COC1 ZINC000880979472 EF On-Demand Anodyne KDR 52 36 CCC1(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)COC1 ZINC000880979472 EF On-Demand Anodyne PDGFRA 53 37 O=C(Cn1cc(-c2ccc(F)nc2)nn1)N[C@H]1CCCc2ccccc21 ZINC000880979492 FF On-Demand Anodyne BDKRB1 42 38 O=C(Cn1cc(-c2ccc(F)nc2)nn1)N[C@@H]1CCCc2ccccc21 ZINC000880979493 FF On-Demand Anodyne BDKRB1 42 38 COCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880979512 ED On-Demand Anodyne PDGFRB 55 39 COCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880979512 ED On-Demand Anodyne KDR 43 35 COCC1(O)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880979512 ED On-Demand Anodyne PDGFRA 50 35 COCC1(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCOCC1 ZINC000880979526 GF On-Demand Anodyne PDGFRA 47 36 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979537 EG On-Demand Anodyne SLC1A2 18 40 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979538 EG On-Demand Anodyne SLC1A2 18 40 COC[C@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CCOCC1 ZINC000880979542 GF On-Demand Anodyne PDGFRA 44 36 COC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CCOCC1 ZINC000880979543 GF On-Demand Anodyne PDGFRA 44 36 CC#CC[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979549 EE On-Demand Mild PDGFRA 49 38 CC#CC[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979550 EE On-Demand Mild PDGFRA 49 38 CCNCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979551 CD On-Demand Anodyne G2YM83_BOTF4 66 34 CNC(C)(C)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979557 DD On-Demand Anodyne G2YM83_BOTF4 57 33 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1cccnc1Cl ZINC000880979558 DD On-Demand Anodyne G2YM83_BOTF4 65 33 COC(=O)C1CCC(c2cn(CC(=O)Nc3cccnc3Cl)nn2)CC1 ZINC000880979568 GE On-Demand Anodyne G2YM83_BOTF4 51 32 CN(Cc1cn(CC(=O)Nc2cccnc2Cl)nn1)C1CCCCC1 ZINC000880979571 FF On-Demand Anodyne G2YM83_BOTF4 58 33 O=C1CCC[C@H](c2cn(CC(=O)Nc3ccc(Cl)cn3)nn2)C1 ZINC000880979572 EE On-Demand Anodyne F10 47 31 O=C1CCC[C@@H](c2cn(CC(=O)Nc3ccc(Cl)cn3)nn2)C1 ZINC000880979573 EE On-Demand Anodyne F10 47 31 C#CC[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979582 ED On-Demand Mild KDR 54 38 C#CC[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979582 ED On-Demand Mild PDGFRA 52 39 C#CC[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979583 ED On-Demand Mild KDR 54 38 C#CC[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979583 ED On-Demand Mild PDGFRA 52 39 C[C@H](O)CCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979603 DD On-Demand Anodyne G2YM83_BOTF4 49 30 CN(C)CCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979607 DD On-Demand Anodyne G2YM83_BOTF4 56 31 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979608 DE On-Demand Anodyne HDAC10 18 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979608 DE On-Demand Anodyne HDAC3 20 42 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979608 DE On-Demand Anodyne HDAC6 16 42 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1cccc(Cl)c1 ZINC000880979614 GD On-Demand Anodyne AVPR1B 30 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)NCc1cccc(Cl)c1 ZINC000880979614 GD On-Demand Anodyne CCR4 20 49 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3cccc(Cl)c3)nn2)CC1 ZINC000880979633 GC On-Demand Anodyne CHRM3 15 43 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3cccc(Cl)c3)nn2)CC1 ZINC000880979633 GC On-Demand Anodyne FAAH 25 46 O=C(Cn1cc(CN[C@H]2CCc3ccccc32)nn1)Nc1cccnc1Cl ZINC000880979639 GF On-Demand Anodyne G2YM83_BOTF4 52 36 O=C(Cn1cc(CN[C@@H]2CCc3ccccc32)nn1)Nc1cccnc1Cl ZINC000880979641 GF On-Demand Anodyne G2YM83_BOTF4 52 36 C[C@H](O)CCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979643 FF On-Demand Anodyne SLC1A2 21 40 O=C(Nc1cscc1Cl)NC1CCN(S(=O)(=O)C(F)(F)F)CC1 ZINC000880979667 GF On-Demand Anodyne EPHX2 43 46 CC[C@@](C)(N)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979669 DD On-Demand Anodyne G2YM83_BOTF4 63 32 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979670 GD On-Demand Anodyne CASR 45 47 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979670 GD On-Demand Anodyne CCR3 30 41 CC(=O)c1cccc(NC(=O)[C@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979670 GD On-Demand Anodyne EPHX2 25 42 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979671 GD On-Demand Anodyne CASR 45 47 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979671 GD On-Demand Anodyne CCR3 30 41 CC(=O)c1cccc(NC(=O)[C@@H](C)n2cc(CCCN3CCOCC3)nn2)c1 ZINC000880979671 GD On-Demand Anodyne EPHX2 25 42 O=C(Nc1cscc1Cl)N1CCC([C@@H](O)c2ccccc2)CC1 ZINC000880979683 FI On-Demand Anodyne RBP4 47 38 O=C(Nc1cscc1Cl)N1CCC([C@H](O)c2ccccc2)CC1 ZINC000880979684 FI On-Demand Anodyne RBP4 47 38 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@@H]3CCOC3)nn2)c1 ZINC000880979695 ED On-Demand Anodyne HDAC10 16 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@@H]3CCOC3)nn2)c1 ZINC000880979695 ED On-Demand Anodyne HDAC3 20 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@H]3CCOC3)nn2)c1 ZINC000880979696 ED On-Demand Anodyne HDAC10 16 40 CC(=O)Nc1cccc(NC(=O)Cn2cc([C@H]3CCOC3)nn2)c1 ZINC000880979696 ED On-Demand Anodyne HDAC3 20 40 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979721 FG On-Demand Anodyne HDAC10 21 40 C[C@@H](O)CCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979721 FG On-Demand Anodyne HDAC6 16 40 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979724 GF On-Demand Anodyne CCR3 34 40 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979724 GF On-Demand Anodyne GPR119 34 45 CC(C)(C)OC(=O)N1CC[C@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979725 GF On-Demand Anodyne CCR3 34 40 CC(C)(C)OC(=O)N1CC[C@H](c2cn(CC(=O)Nc3cccc(F)c3)nn2)C1 ZINC000880979725 GF On-Demand Anodyne GPR119 34 45 Cn1nc2c(c1-c1cn(CC(=O)Nc3cccc(F)c3)nn1)CCCC2 ZINC000880979730 FE On-Demand Anodyne HDAC10 19 40 Cn1nc2c(c1-c1cn(CC(=O)Nc3cccc(F)c3)nn1)CCCC2 ZINC000880979730 FE On-Demand Anodyne HDAC3 21 40 Cn1nc2c(c1-c1cn(CC(=O)Nc3cccc(F)c3)nn1)CCCC2 ZINC000880979730 FE On-Demand Anodyne HDAC6 18 40 N[C@@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)[C@H]1CCCO1 ZINC000880979752 GF On-Demand Anodyne SLC1A2 21 40 N[C@@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)[C@@H]1CCCO1 ZINC000880979753 GF On-Demand Anodyne SLC1A2 21 40 N[C@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)[C@@H]1CCCO1 ZINC000880979754 GF On-Demand Anodyne SLC1A2 21 40 N[C@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)[C@H]1CCCO1 ZINC000880979755 GF On-Demand Anodyne SLC1A2 21 40 O=C(Cn1cc(C2(F)COC2)nn1)Nc1cccnc1Cl ZINC000880979765 DD On-Demand Anodyne G2YM83_BOTF4 65 32 O=C(Cn1cc(C2CCCCCC2)nn1)Nc1cccnc1Cl ZINC000880979766 EG On-Demand Anodyne G2YM83_BOTF4 58 33 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1cccnc1Cl ZINC000880979767 DD On-Demand Anodyne G2YM83_BOTF4 57 33 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1cccnc1Cl ZINC000880979768 DD On-Demand Anodyne G2YM83_BOTF4 57 33 O=C(Nc1cscc1Cl)N1CCC2(CCCC2)C1 ZINC000880979771 CI On-Demand Anodyne EPHX2 26 40 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979799 GE On-Demand Anodyne CASR 46 39 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979799 GE On-Demand Anodyne CHRNA7 21 50 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979799 GE On-Demand Anodyne MTOR 51 39 O=C(Cn1cc(CCN2CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979799 GE On-Demand Anodyne EPHX2 21 45 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1ccc(Cl)cn1 ZINC000880979824 DE On-Demand Anodyne F10 40 31 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1ccc(Cl)cn1 ZINC000880979825 DE On-Demand Anodyne F10 40 31 C=C(C)CONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979829 DF On-Demand Mild KDR 62 38 C=C(C)CONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979829 DF On-Demand Mild PDGFRA 53 39 O=C(Cn1cc(CNC2CCCC2)nn1)Nc1cccnc1Cl ZINC000880979834 ED On-Demand Anodyne G2YM83_BOTF4 45 32 C=CCOCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979840 EF On-Demand Mild PDGFRA 50 37 O=C(Cn1cc(CN2CCCCC2)nn1)Nc1cccnc1Cl ZINC000880979844 ED On-Demand Anodyne G2YM83_BOTF4 49 30 COC(=O)C1CCC(c2cn(CC(=O)Nc3ccc(Cl)cn3)nn2)CC1 ZINC000880979845 GE On-Demand Anodyne F10 50 33 C#C[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979849 DD On-Demand Mild KDR 42 37 C#C[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979849 DD On-Demand Mild PDGFRA 52 38 C#C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979850 DD On-Demand Mild KDR 42 37 C#C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979850 DD On-Demand Mild PDGFRA 52 38 C#C[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880979852 EG On-Demand Mild PDGFRA 46 38 C#C[C@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880979853 EG On-Demand Mild PDGFRA 46 38 C#CC[C@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979866 EE On-Demand Mild KDR 50 36 C#CC[C@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979866 EE On-Demand Mild PDGFRA 49 38 C#CC[C@@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979867 EE On-Demand Mild KDR 50 36 C#CC[C@@H](COC)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979867 EE On-Demand Mild PDGFRA 49 38 CCOC(=O)N1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880979874 DF On-Demand Anodyne P2RY12 38 42 CCOC(=O)N1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880979874 DF On-Demand Anodyne TGM2 21 40 CCOC(=O)N1CCN(C(=O)Nc2cscc2Cl)CC1 ZINC000880979874 DF On-Demand Anodyne F13A1 19 40 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979881 EF On-Demand Anodyne HDAC10 17 42 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979881 EF On-Demand Anodyne HDAC6 17 42 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880979881 EF On-Demand Anodyne SLC1A2 18 41 C=C[C@H](C)ONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979884 DF On-Demand Mild KDR 53 39 C=C[C@H](C)ONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979884 DF On-Demand Mild PDGFRA 53 41 C=C[C@@H](C)ONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979885 DF On-Demand Mild KDR 53 39 C=C[C@@H](C)ONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979885 DF On-Demand Mild PDGFRA 53 41 O=C(Cn1cc(C2CCC(C3OCCO3)CC2)nn1)Nc1cccnc1Cl ZINC000880979894 GF On-Demand Anodyne G2YM83_BOTF4 43 31 C#CCCN(CCOC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979895 FF On-Demand Mild PDGFRA 47 36 CCNCc1cn(CC(=O)Nc2cc3oc4ccccc4c3cc2OC)nn1 ZINC000880979896 GF On-Demand Anodyne PTPN22 41 39 COC(=O)C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979898 EE On-Demand Anodyne PDGFRB 28 41 COC(=O)C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979898 EE On-Demand Anodyne KDR 49 37 COC(=O)C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979898 EE On-Demand Anodyne PDGFRA 52 41 O=C(Cn1cc([C@@H]2CCCC[C@@H]2O)nn1)Nc1cccnc1Cl ZINC000880979911 ED On-Demand Anodyne G2YM83_BOTF4 65 34 O=C(Cn1cc([C@@H]2CCCC[C@H]2O)nn1)Nc1cccnc1Cl ZINC000880979912 ED On-Demand Anodyne G2YM83_BOTF4 65 34 O=C(Cn1cc([C@H]2CCCC[C@@H]2O)nn1)Nc1cccnc1Cl ZINC000880979913 ED On-Demand Anodyne G2YM83_BOTF4 65 34 O=C(Cn1cc([C@H]2CCCC[C@H]2O)nn1)Nc1cccnc1Cl ZINC000880979914 ED On-Demand Anodyne G2YM83_BOTF4 65 34 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1cccnc1Cl ZINC000880979915 EE On-Demand Anodyne G2YM83_BOTF4 58 33 O=C(Cn1cc(CCCCCCO)nn1)Nc1ccc(Cl)cn1 ZINC000880979916 EE On-Demand Anodyne F10 46 31 O=C(Cn1cc(CC2(O)CCCCC2)nn1)Nc1cccnc1Cl ZINC000880979919 EE On-Demand Anodyne G2YM83_BOTF4 57 32 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3ccc(Cl)cn3)nn2)CC1 ZINC000880979921 GC On-Demand Anodyne F10 49 33 C#CCC(CC#C)C(=O)Nc1ccc(OC)cc1F ZINC000880979935 CE On-Demand Mild MTNR1B 24 40 COC(=O)Cc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880979940 DC On-Demand Anodyne G2YM83_BOTF4 64 32 CCCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979947 DF On-Demand Anodyne KDR 67 39 CCCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880979947 DF On-Demand Anodyne PDGFRA 55 40 O=C(Cn1cc(CCCCCCO)nn1)NCc1cccc(Cl)c1 ZINC000880979951 FE On-Demand Anodyne SUCNR1 44 40 C#CC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880979960 EG On-Demand Mild PDGFRB 41 38 C#CC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880979960 EG On-Demand Mild KDR 40 38 C#CC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880979960 EG On-Demand Mild PDGFRA 49 36 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1cccnc1Cl ZINC000880979961 DE On-Demand Anodyne G2YM83_BOTF4 56 32 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1cccnc1Cl ZINC000880979962 DE On-Demand Anodyne G2YM83_BOTF4 56 32 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880979981 FE On-Demand Anodyne ACOX1 22 40 O=C1CCC(c2cn(CC(=O)Nc3cccnc3Cl)nn2)CC1 ZINC000880980067 EE On-Demand Anodyne G2YM83_BOTF4 52 34 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@H]1C ZINC000880980068 FF On-Demand Anodyne KDR 54 34 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@H]1C ZINC000880980068 FF On-Demand Anodyne PDGFRA 46 34 CNC(C)(C)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980089 EG On-Demand Anodyne HDAC10 15 40 COC(=O)[C@@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980092 GF On-Demand Anodyne PDGFRA 40 33 COC(=O)[C@H]1C[C@H]2CC[C@H]1N2C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980093 GF On-Demand Anodyne PDGFRA 40 33 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980102 GH On-Demand Anodyne PDGFRB 50 37 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980102 GH On-Demand Anodyne KDR 43 37 CCC1(N(C)C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980102 GH On-Demand Anodyne PDGFRA 45 34 CC#CCNCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980109 DD On-Demand Mild G2YM83_BOTF4 56 32 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980111 GE On-Demand Anodyne KDR 40 35 COC(=O)[C@@]1(OC)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980111 GE On-Demand Anodyne PDGFRA 44 33 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(Cl)cn1 ZINC000880980112 FD On-Demand Anodyne F10 48 33 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(Cl)cn1 ZINC000880980112 FD On-Demand Anodyne EPHX2 19 42 COCCNCCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980113 EC On-Demand Anodyne G2YM83_BOTF4 62 31 COC(=O)Cc1cn(CC(=O)Nc2ccc(Cl)cn2)nn1 ZINC000880980117 DC On-Demand Anodyne F10 55 36 C[C@H](N)c1cn(CC(=O)NCc2cccc(Cl)c2)nn1 ZINC000880980122 CD On-Demand Anodyne CARM1 41 36 O=C(Cn1cc(CC2(O)CCC2)nn1)Nc1cccnc1Cl ZINC000880980125 DD On-Demand Anodyne G2YM83_BOTF4 58 32 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1cccnc1Cl ZINC000880980134 ED On-Demand Anodyne G2YM83_BOTF4 68 34 O=C(Cn1cc(CCN2CCCCC2)nn1)Nc1cccnc1Cl ZINC000880980139 ED On-Demand Anodyne HNMT 46 32 CC[C@@](C)(O)c1cn(CC(=O)Nc2ccc(Cl)cn2)nn1 ZINC000880980141 DD On-Demand Anodyne F10 47 33 CC[C@H](O)c1cn(CC(=O)NCc2cccc(Cl)c2)nn1 ZINC000880980144 DD On-Demand Anodyne PDS 54 38 CCN1CC[C@@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1=O ZINC000880980153 FD On-Demand Anodyne PDGFRA 45 38 CCN1CC[C@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1=O ZINC000880980154 FD On-Demand Anodyne PDGFRA 45 38 COC[C@@H]1CCCN1C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980156 EF On-Demand Anodyne PDGFRA 49 37 COC[C@@H]1CCCN1C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980156 EF On-Demand Anodyne ACKR3 50 31 O=C(Cn1cc(C[C@@H](O)C2CC2)nn1)Nc1cccnc1Cl ZINC000880980157 DD On-Demand Anodyne G2YM83_BOTF4 44 32 O=C(Cn1cc(C[C@H](O)C2CC2)nn1)Nc1cccnc1Cl ZINC000880980158 DD On-Demand Anodyne G2YM83_BOTF4 44 32 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@@H]1C ZINC000880980175 GF On-Demand Anodyne KDR 41 35 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@@H]1C ZINC000880980175 GF On-Demand Anodyne PDGFRA 42 33 COC[C@@H]1CCCN1NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980177 FE On-Demand Anodyne PDGFRA 49 36 CC[C@H](O)c1cn(CC(=O)Nc2ccc(Cl)cn2)nn1 ZINC000880980183 CD On-Demand Anodyne F10 51 33 N[C@@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)C1CCOCC1 ZINC000880980197 GG On-Demand Anodyne SLC1A2 21 41 N[C@H](c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1)C1CCOCC1 ZINC000880980198 GG On-Demand Anodyne SLC1A2 21 41 CCOC1CC2(C1)C[C@@H]2NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980203 FG On-Demand Anodyne PDGFRA 47 36 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1cc(F)ccc1F ZINC000880980204 FD On-Demand Anodyne EPHX2 18 42 CC[C@H](C[C@H](C)O)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980219 EF On-Demand Anodyne PDGFRA 49 39 CCC[C@@H](N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980236 EG On-Demand Anodyne SLC1A1 27 44 CCC[C@@H](N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980236 EG On-Demand Anodyne SLC1A2 40 44 CCC[C@H](N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980237 EG On-Demand Anodyne SLC1A1 27 44 CCC[C@H](N)c1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980237 EG On-Demand Anodyne SLC1A2 40 44 CC[C@@](C)(O)Cc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980240 DD On-Demand Anodyne G2YM83_BOTF4 50 32 C=C(C)CN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980253 DG On-Demand Mild KDR 64 37 C=C(C)CN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980253 DG On-Demand Mild PDGFRA 55 41 O=C(Cn1cc(C2CCNCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980254 FG On-Demand Anodyne HDAC6 20 40 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@@H](C)O1 ZINC000880980332 GE On-Demand Anodyne PDGFRA 41 33 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@H](C)O1 ZINC000880980333 GE On-Demand Anodyne PDGFRA 41 33 CCn1ncc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1C ZINC000880980338 FG On-Demand Anodyne PDGFRB 48 45 CCn1ncc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1C ZINC000880980338 FG On-Demand Anodyne KDR 63 40 CCn1ncc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1C ZINC000880980338 FG On-Demand Anodyne PDGFRA 57 42 CCn1ncc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1C ZINC000880980338 FG On-Demand Anodyne CSF1R 20 45 O=C1CCC(c2cn(CC(=O)Nc3ccc(-c4ccccc4)cc3)nn2)CC1 ZINC000880980339 FH On-Demand Anodyne HDAC6 19 40 CCN(CC)C(=O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980348 FE On-Demand Anodyne KDR 44 37 CCN(CC)C(=O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980348 FE On-Demand Anodyne PDGFRA 52 38 O=C(Cn1cc(C2CCCCC2)nn1)Nc1cccnc1Cl ZINC000880980355 DG On-Demand Anodyne G2YM83_BOTF4 58 33 C[C@@](O)(Cc1cn(CC(=O)Nc2ccc(Cl)cn2)nn1)c1cccs1 ZINC000880980369 GE On-Demand Anodyne F10 48 32 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)NCc2cccc(Cl)c2)nn1 ZINC000880980372 GF On-Demand Anodyne F2 15 43 O=C(Cn1cc(CN2CCCC2)nn1)Nc1cccnc1Cl ZINC000880980376 DD On-Demand Anodyne G2YM83_BOTF4 50 31 C[C@H](N)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980385 CC On-Demand Anodyne G2YM83_BOTF4 64 32 C[C@H](N)c1cn(CC(=O)Nc2ccc(Cl)cn2)nn1 ZINC000880980394 CC On-Demand Anodyne F10 49 34 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3cccnc3Cl)nn2)CC1 ZINC000880980404 GC On-Demand Anodyne G2YM83_BOTF4 50 31 CC[C@H](O)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980408 CD On-Demand Anodyne G2YM83_BOTF4 65 33 O=C(Cn1cc([C@H]2CCCC[C@@H]2O)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980414 GH On-Demand Anodyne HDAC6 18 40 O=C(Cn1cc([C@@H]2CCCC[C@@H]2O)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980415 GH On-Demand Anodyne HDAC6 18 40 O=C(Cn1cc([C@@H]2CCCC[C@H]2O)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980416 GH On-Demand Anodyne HDAC6 18 40 O=C(Cn1cc([C@H]2CCCC[C@H]2O)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980417 GH On-Demand Anodyne HDAC6 18 40 CN(CCO)Cc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980419 DC On-Demand Anodyne G2YM83_BOTF4 44 32 CCC(C)(C)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980425 DF On-Demand Anodyne G2YM83_BOTF4 68 35 CCN(CC)Cc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980427 DD On-Demand Anodyne G2YM83_BOTF4 63 33 CC[C@@H](N)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980446 CD On-Demand Anodyne G2YM83_BOTF4 64 33 COC[C@@H](CCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12)OC ZINC000880980453 FE On-Demand Anodyne PDGFRA 50 37 CC[C@@](C)(O)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980456 DD On-Demand Anodyne G2YM83_BOTF4 63 33 CC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980462 DE On-Demand Anodyne KDR 53 39 CC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980462 DE On-Demand Anodyne PDGFRA 54 39 O=C(Cn1cc(C[C@@]2(O)CCSC2)nn1)Nc1cccnc1Cl ZINC000880980466 FD On-Demand Anodyne G2YM83_BOTF4 49 31 O=C(Cn1cc(C[C@]2(O)CCSC2)nn1)Nc1cccnc1Cl ZINC000880980467 FD On-Demand Anodyne G2YM83_BOTF4 49 31 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccc(Cl)cn1 ZINC000880980469 DD On-Demand Anodyne F10 46 30 CCOC(=O)N1CCC(NC(=O)Nc2cscc2Cl)CC1 ZINC000880980477 EG On-Demand Anodyne EPHX2 50 48 O=C1CCC[C@H](c2cn(CC(=O)Nc3cccnc3Cl)nn2)C1 ZINC000880980478 EE On-Demand Anodyne G2YM83_BOTF4 44 32 O=C1CCC[C@@H](c2cn(CC(=O)Nc3cccnc3Cl)nn2)C1 ZINC000880980479 EE On-Demand Anodyne G2YM83_BOTF4 44 32 NCCCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980480 EF On-Demand Anodyne HDAC1 15 53 NCCCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980480 EF On-Demand Anodyne HDAC3 22 41 NCCCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980480 EF On-Demand Anodyne HDAC6 21 42 NCCCCc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980480 EF On-Demand Anodyne SLC1A2 18 41 CC(=O)CCCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980491 DD On-Demand Anodyne SUCNR1 44 34 CC(=O)CCCc1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980491 DD On-Demand Anodyne G2YM83_BOTF4 62 31 COC[C@@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980492 FE On-Demand Anodyne SLC1A1 18 42 COC[C@@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980492 FE On-Demand Anodyne SLC1A2 26 42 COC[C@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980493 FE On-Demand Anodyne SLC1A1 18 42 COC[C@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980493 FE On-Demand Anodyne SLC1A2 26 42 C=C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980494 DD On-Demand Mild PDGFRA 52 39 O=C(Cn1cc(CN[C@H]2CCCc3ccccc32)nn1)Nc1cccnc1Cl ZINC000880980495 GG On-Demand Anodyne G2YM83_BOTF4 44 33 O=C(Cn1cc(CN[C@@H]2CCCc3ccccc32)nn1)Nc1cccnc1Cl ZINC000880980496 GG On-Demand Anodyne G2YM83_BOTF4 44 33 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1cccnc1Cl ZINC000880980497 DD On-Demand Anodyne G2YM83_BOTF4 50 32 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1cccnc1Cl ZINC000880980498 DD On-Demand Anodyne G2YM83_BOTF4 50 32 C#CCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980499 FF On-Demand Mild PDGFRB 52 37 C#CCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980499 FF On-Demand Mild PDGFRA 42 33 O=C(Cn1cc(CN2CCOCC2)nn1)Nc1cccnc1Cl ZINC000880980500 EC On-Demand Anodyne G2YM83_BOTF4 43 30 COC(=O)C1(Cc2cn(CC(=O)Nc3cccnc3Cl)nn2)CCCCC1 ZINC000880980503 GF On-Demand Anodyne G2YM83_BOTF4 50 32 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1cccnc1Cl ZINC000880980507 ED On-Demand Anodyne G2YM83_BOTF4 45 34 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1cccnc1Cl ZINC000880980508 ED On-Demand Anodyne G2YM83_BOTF4 45 34 CCC[C@@H](N)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980509 DD On-Demand Anodyne G2YM83_BOTF4 51 33 CCC[C@H](N)c1cn(CC(=O)Nc2cccnc2Cl)nn1 ZINC000880980510 DD On-Demand Anodyne G2YM83_BOTF4 51 33 C#CC1(F)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980521 EE On-Demand Mild KDR 42 36 C#CC1(F)CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980521 EE On-Demand Mild PDGFRA 49 35 O=C(Cn1cc(C2(O)CCOCC2)nn1)Nc1ccc(-c2ccccc2)cc1 ZINC000880980527 GF On-Demand Anodyne HDAC6 15 40 C=C(C)C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980530 EF On-Demand Mild PDGFRA 51 38 C=C(C)C[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980531 EF On-Demand Mild PDGFRA 51 38 O=C(Cn1cc(C(=O)C2CCC2)nn1)Nc1cccnc1Cl ZINC000880980534 DD On-Demand Anodyne G2YM83_BOTF4 58 33 O=C(Cn1cc(C2CCNCC2)nn1)Nc1cccnc1Cl ZINC000880980538 DD On-Demand Anodyne G2YM83_BOTF4 44 32 O=C(Cn1cc(CNC2CC2)nn1)Nc1cccnc1Cl ZINC000880980541 DD On-Demand Anodyne G2YM83_BOTF4 51 33 COCC[C@@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980542 GE On-Demand Anodyne SLC1A2 22 41 COCC[C@H](N)Cc1cn(CC(=O)Nc2ccc(-c3ccccc3)cc2)nn1 ZINC000880980543 GE On-Demand Anodyne SLC1A2 22 41 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980638 ED On-Demand Anodyne TRPV1 16 41 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980638 ED On-Demand Anodyne MT-ND1 25 45 CC[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980638 ED On-Demand Anodyne DRTS_TRYCR 47 32 Cc1ccc(NC(=O)Cn2cc(CCCN3CCOCC3)nn2)c(F)c1 ZINC000880980653 FD On-Demand Anodyne EPHX2 15 40 CCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980676 CE On-Demand Anodyne KDR 70 40 CCONC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980676 CE On-Demand Anodyne PDGFRA 57 42 COC[C@@H](CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12)OC ZINC000880980702 EE On-Demand Anodyne PDGFRA 55 39 C=C[C@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980713 ED On-Demand Mild MT-ND1 23 42 C=C[C@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980713 ED On-Demand Mild DRTS_TRYCR 45 31 C=C[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980714 ED On-Demand Mild MT-ND1 23 42 C=C[C@@](C)(O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980714 ED On-Demand Mild DRTS_TRYCR 45 31 CCN(C)C(=O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980730 ED On-Demand Anodyne PDGFRA 50 37 COCCOC1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980735 FE On-Demand Anodyne PDGFRB 41 35 COCCOC1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980735 FE On-Demand Anodyne KDR 54 34 COCCOC1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980735 FE On-Demand Anodyne PDGFRA 46 34 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1ccccc1-c1ccccc1 ZINC000880980736 EG On-Demand Anodyne CHRM3 16 41 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1ccccc1-c1ccccc1 ZINC000880980737 EG On-Demand Anodyne CHRM3 16 41 Cc1ccc(NC(=O)Cn2cc(CCCOc3cccnc3F)nn2)c(F)c1 ZINC000880980749 GF On-Demand Anodyne MMP8 24 44 COCCO[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980758 GF On-Demand Anodyne PDGFRB 40 35 COCCO[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980758 GF On-Demand Anodyne PDGFRA 44 34 COCCO[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980759 GF On-Demand Anodyne PDGFRB 40 35 COCCO[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980759 GF On-Demand Anodyne PDGFRA 44 34 COC(=O)[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)[C@H]1C ZINC000880980782 FF On-Demand Anodyne PDGFRA 42 34 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)[C@@H]1C ZINC000880980783 FF On-Demand Anodyne PDGFRA 42 34 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)[C@H]1C ZINC000880980784 FF On-Demand Anodyne PDGFRA 42 34 COC(=O)[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)[C@@H]1C ZINC000880980785 FF On-Demand Anodyne PDGFRA 42 34 CCO[C@H]1COCC[C@H]1NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980831 GF On-Demand Anodyne PDGFRA 41 36 CCO[C@H]1COCC[C@@H]1NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980834 GF On-Demand Anodyne PDGFRA 41 36 COCC1=CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880980844 FG On-Demand Anodyne PDGFRA 41 33 C#CCC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980880 EE On-Demand Mild KDR 43 35 C#CCC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980880 EE On-Demand Mild PDGFRA 49 36 C#CCC[C@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980881 EE On-Demand Mild KDR 43 35 C#CCC[C@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980881 EE On-Demand Mild PDGFRA 49 36 C#C[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980901 CE On-Demand Mild PDGFRB 27 42 C#C[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980901 CE On-Demand Mild KDR 56 38 C#C[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980901 CE On-Demand Mild PDGFRA 54 42 C#C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980902 CE On-Demand Mild PDGFRB 27 42 C#C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980902 CE On-Demand Mild KDR 56 38 C#C[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980902 CE On-Demand Mild PDGFRA 54 42 COC[C@@H]1CCCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980906 FH On-Demand Anodyne PDGFRB 55 36 COC[C@@H]1CCCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880980906 FH On-Demand Anodyne PDGFRA 48 39 CNC(C)(C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980925 EE On-Demand Anodyne KDR 55 37 CNC(C)(C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980925 EE On-Demand Anodyne PDGFRA 54 38 O=C(Cn1cc([C@@H]2CCOC2)nn1)NCCc1ccc(Cl)cc1 ZINC000880980934 ED On-Demand Anodyne LUXR 18 41 O=C(Cn1cc([C@H]2CCOC2)nn1)NCCc1ccc(Cl)cc1 ZINC000880980935 ED On-Demand Anodyne LUXR 18 41 C=CCN(CCOC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880980943 EF On-Demand Mild PDGFRA 46 36 C[C@H](N)c1cn(CC(=O)NCCC(c2ccccc2)c2ccccc2)nn1 ZINC000880980959 FF On-Demand Anodyne C3AR1 47 35 CC[C@H](O)c1cn(CC(=O)NCc2ccc(OC)c(OC)c2)nn1 ZINC000880980983 ED On-Demand Anodyne DRTS_TRYCR 45 31 COC[C@@H](C)n1ccc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)n1 ZINC000880980992 GG On-Demand Anodyne PDGFRA 50 37 COC[C@@H](C)n1ccc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)n1 ZINC000880980992 GG On-Demand Anodyne GCK 15 40 CCn1cccc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1=O ZINC000880981032 GF On-Demand Anodyne PDGFRB 39 41 CCn1cccc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1=O ZINC000880981032 GF On-Demand Anodyne KDR 54 35 CCn1cccc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1=O ZINC000880981032 GF On-Demand Anodyne PDGFRA 46 39 CCn1cccc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1=O ZINC000880981032 GF On-Demand Anodyne CSF1R 16 41 CCc1cnc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)o1 ZINC000880981126 FG On-Demand Anodyne PDGFRB 32 41 CCc1cnc(CNC(=O)Nc2cc(OC)cc3c(OC)ccnc23)o1 ZINC000880981126 FG On-Demand Anodyne PDGFRA 45 35 COCCCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981130 GF On-Demand Anodyne KDR 58 35 COCCCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981130 GF On-Demand Anodyne PDGFRA 51 38 COC[C@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CC1 ZINC000880981135 EF On-Demand Anodyne KDR 45 35 COC[C@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CC1 ZINC000880981135 EF On-Demand Anodyne PDGFRA 52 38 COC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CC1 ZINC000880981136 EF On-Demand Anodyne KDR 45 35 COC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)C1CC1 ZINC000880981136 EF On-Demand Anodyne PDGFRA 52 38 CCC1(CO)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880981149 FG On-Demand Anodyne PDGFRB 45 38 CCC1(CO)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880981149 FG On-Demand Anodyne PDGFRA 42 34 COCCn1ccc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)n1 ZINC000880981160 FF On-Demand Anodyne KDR 57 36 COCCn1ccc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)n1 ZINC000880981160 FF On-Demand Anodyne PDGFRA 51 39 C#CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981216 CE On-Demand Mild KDR 65 38 C#CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981216 CE On-Demand Mild PDGFRA 56 41 COC[C@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@H]1CCCO1 ZINC000880981227 GF On-Demand Anodyne PDGFRA 40 35 COC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@H]1CCCO1 ZINC000880981228 GF On-Demand Anodyne PDGFRA 40 35 COC[C@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@@H]1CCCO1 ZINC000880981229 GF On-Demand Anodyne PDGFRA 40 35 COC[C@@H](NC(=O)Nc1cc(OC)cc2c(OC)ccnc12)[C@@H]1CCCO1 ZINC000880981230 GF On-Demand Anodyne PDGFRA 40 35 CC[C@@H](CC#N)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981236 EG On-Demand Mild PDGFRA 49 37 O=C(Cn1cc(CNC(=O)OCc2ccccc2)nn1)NCCC1=CCCCC1 ZINC000880981238 GF On-Demand Anodyne CAPN2 58 33 CCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981239 EF On-Demand Anodyne KDR 59 36 CCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981239 EF On-Demand Anodyne PDGFRA 53 39 CC[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@@H]1O ZINC000880981242 EE On-Demand Anodyne KDR 44 35 CC[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@@H]1O ZINC000880981242 EE On-Demand Anodyne PDGFRA 48 35 CC[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@H]1O ZINC000880981243 EE On-Demand Anodyne KDR 44 35 CC[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C[C@H]1O ZINC000880981243 EE On-Demand Anodyne PDGFRA 48 35 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1ccccc1-c1ccccc1 ZINC000880981278 EF On-Demand Anodyne PTPN22 21 40 CC[C@@](C)(O)c1cn(CC(=O)NCCC(c2ccccc2)c2ccccc2)nn1 ZINC000880981282 GG On-Demand Anodyne C3AR1 45 33 CCN(C)C(=O)[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981300 FE On-Demand Anodyne PDGFRA 49 38 CCN(C)C(=O)[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981301 FE On-Demand Anodyne PDGFRA 49 38 CCOCCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981306 GF On-Demand Anodyne KDR 51 35 CCOCCOCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981306 GF On-Demand Anodyne PDGFRA 52 38 CNC(=O)CCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981412 FE On-Demand Anodyne KDR 51 37 CNC(=O)CCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981412 FE On-Demand Anodyne PDGFRA 52 38 C#CCOCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981450 EE On-Demand Mild PDGFRA 50 37 C/C=C/C[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981454 EF On-Demand Anodyne PDGFRA 49 38 C/C=C\C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981455 EF On-Demand Anodyne PDGFRA 49 38 C/C=C\C[C@@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981456 EF On-Demand Anodyne PDGFRA 49 38 C/C=C/C[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981457 EF On-Demand Anodyne PDGFRA 49 38 C#CCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981460 DF On-Demand Mild KDR 41 37 C#CCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981460 DF On-Demand Mild PDGFRA 53 38 C=CCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981476 DG On-Demand Mild KDR 57 36 C=CCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981476 DG On-Demand Mild PDGFRA 53 39 C=CC[C@H](CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981492 EE On-Demand Mild PDGFRA 51 38 COCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880981532 GE On-Demand Anodyne PDGFRB 60 38 COCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880981532 GE On-Demand Anodyne PDGFRA 48 35 C=CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981569 DF On-Demand Mild KDR 64 37 C=CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981569 DF On-Demand Mild PDGFRA 55 41 CCN(Cc1ccncc1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981644 FH On-Demand Anodyne KDR 41 36 CCN(Cc1ccncc1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981644 FH On-Demand Anodyne ROCK2 21 40 CCN(Cc1ccncc1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981644 FH On-Demand Anodyne PDGFRA 51 37 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne PDGFRB 52 46 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne KDR 47 39 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne FLT4 30 44 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne PDGFRA 57 42 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne FLT3 15 44 COCCn1cc(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)cn1 ZINC000880981682 FF On-Demand Anodyne CSF1R 20 46 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H]2CCOC2)nn1 ZINC000880981694 FH On-Demand Anodyne SOAT1 47 42 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H]2CCOC2)nn1 ZINC000880981696 FH On-Demand Anodyne SOAT1 47 42 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(CC(C)(C)O)nn1 ZINC000880981721 FG On-Demand Anodyne SOAT1 60 46 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(C(C)(C)O)nn1 ZINC000880981746 EG On-Demand Anodyne SOAT1 60 48 CCC[C@@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981789 CG On-Demand Anodyne NQO2 18 41 CCC[C@@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981789 CG On-Demand Anodyne MTNR1A 15 41 CCC[C@@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981789 CG On-Demand Anodyne MTNR1B 15 41 CCC[C@@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981790 CG On-Demand Anodyne NQO2 18 41 CCC[C@@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981790 CG On-Demand Anodyne MTNR1A 15 41 CCC[C@@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981790 CG On-Demand Anodyne MTNR1B 15 41 CCC[C@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981791 CG On-Demand Anodyne NQO2 18 41 CCC[C@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981791 CG On-Demand Anodyne MTNR1A 15 41 CCC[C@H](CCO)NC(=O)CC[C@H]1CCc2ccccc21 ZINC000880981791 CG On-Demand Anodyne MTNR1B 15 41 CCC[C@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981792 CG On-Demand Anodyne NQO2 18 41 CCC[C@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981792 CG On-Demand Anodyne MTNR1A 15 41 CCC[C@H](CCO)NC(=O)CC[C@@H]1CCc2ccccc21 ZINC000880981792 CG On-Demand Anodyne MTNR1B 15 41 CS(=O)(=O)C1CCC(C(=O)Nc2ccc([C@H](O)C(F)(F)F)cc2)CC1 ZINC000880981807 GF On-Demand Anodyne EPHX2 17 40 CS(=O)(=O)C1CCC(C(=O)Nc2ccc([C@@H](O)C(F)(F)F)cc2)CC1 ZINC000880981808 GF On-Demand Anodyne EPHX2 17 40 COCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981812 DE On-Demand Anodyne KDR 60 38 COCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880981812 DE On-Demand Anodyne PDGFRA 55 39 N#Cc1c(NC(=O)Cn2cc(-c3ccc(F)nc3)nn2)sc2c1CCCCC2 ZINC000880981849 GG On-Demand Mild VIPR1 31 49 N#Cc1c(NC(=O)Cn2cc(-c3cccnc3F)nn2)sc2c1CCCCC2 ZINC000880981877 GG On-Demand Mild VIPR1 30 49 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(CN2CCOC2=O)nn1 ZINC000880981898 GG On-Demand Anodyne SOAT1 44 41 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880981945 GI On-Demand Anodyne SOAT1 50 45 C[C@H]1c2ccccc2CCN1C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880981960 GF On-Demand Anodyne TRPM8 33 40 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@]2(O)CCOC2)nn1 ZINC000880981969 FF On-Demand Anodyne SOAT1 48 42 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@]2(O)CCOC2)nn1 ZINC000880981970 FF On-Demand Anodyne SOAT1 48 42 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H]2CCCC(=O)C2)nn1 ZINC000880981975 GI On-Demand Anodyne SOAT1 45 41 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H]2CCCC(=O)C2)nn1 ZINC000880981976 GI On-Demand Anodyne SOAT1 45 41 COCCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982028 EF On-Demand Anodyne KDR 60 37 COCCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982028 EF On-Demand Anodyne PDGFRA 53 39 Cc1cc(C)c2c(c1)CN(C(=O)Nc1ccc3c(c1)S(=O)(=O)CC(=O)N3)CC2 ZINC000880982082 GF On-Demand Anodyne P2RY14 43 33 Fc1ccccc1OCCn1cc(CCCN2CCOCC2)nn1 ZINC000880982102 ED On-Demand Anodyne DRD3 15 45 COC[C@@H](O)Cc1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880982145 FF On-Demand Anodyne SOAT1 59 45 COC(=O)Cc1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880982153 FF On-Demand Anodyne SOAT1 64 46 C=C[C@](C)(O)c1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880982154 FH On-Demand Mild SOAT1 52 44 C=C[C@@](C)(O)c1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880982155 FH On-Demand Mild SOAT1 52 44 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(C2(O)CCCCC2)nn1 ZINC000880982157 GI On-Demand Anodyne SOAT1 55 44 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880982177 GI On-Demand Anodyne SOAT1 36 40 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1 ZINC000880982178 GI On-Demand Anodyne SOAT1 36 40 COC(=O)C[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCO1 ZINC000880982307 GE On-Demand Anodyne KDR 40 39 COC(=O)C[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCO1 ZINC000880982311 GE On-Demand Anodyne KDR 40 39 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccc(C)cc3)cs2)nn1 ZINC000880982313 FF On-Demand Anodyne ROCK1 19 40 COC(=O)[C@@]1(F)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982324 GE On-Demand Anodyne PDGFRA 42 33 CCC[C@H](CCO)NC(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880982333 DG On-Demand Anodyne MTTP 50 33 CCC[C@H](CCO)NC(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880982333 DG On-Demand Anodyne UTS2 55 33 CCC[C@@H](CCO)NC(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880982334 DG On-Demand Anodyne MTTP 50 33 CCC[C@@H](CCO)NC(=O)c1ccc2nc(Cl)ccc2c1 ZINC000880982334 DG On-Demand Anodyne UTS2 55 33 CCC[C@H](CCO)NC(=O)c1cccnc1I ZINC000880982374 ED On-Demand Anodyne G2YM83_BOTF4 50 32 CC[C@@](C)(O)c1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880982377 FH On-Demand Anodyne SOAT1 63 50 CCC[C@@H](CCO)NC(=O)c1cccnc1I ZINC000880982392 ED On-Demand Anodyne G2YM83_BOTF4 50 32 COC(OC)c1ccc(C(=O)Nc2ccc([C@@H](O)C(F)(F)F)cc2)o1 ZINC000880982401 FG On-Demand Anodyne SCN10A 18 40 COCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982402 ED On-Demand Anodyne KDR 51 34 COCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982402 ED On-Demand Anodyne ROCK2 15 41 COCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982402 ED On-Demand Anodyne PDGFRA 50 37 COC(OC)c1ccc(C(=O)Nc2ccc([C@H](O)C(F)(F)F)cc2)o1 ZINC000880982403 FG On-Demand Anodyne SCN10A 18 40 COCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982412 GD On-Demand Anodyne PDGFRB 62 41 COCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982412 GD On-Demand Anodyne KDR 44 37 COCC(=O)N1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982412 GD On-Demand Anodyne PDGFRA 50 36 C[C@@H]1CCCN(C(=O)Nc2ccc3c(c2)S(=O)(=O)CC(=O)N3)[C@@H]1C ZINC000880982444 FE On-Demand Anodyne TRPC6 46 35 C[C@H]1[C@H](C)CCCN1C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880982447 FE On-Demand Anodyne TRPC6 46 35 O=C(CCc1cn[nH]c1)Nc1ccc([C@@H](O)C(F)(F)F)cc1 ZINC000880982459 DF On-Demand Anodyne ROCK2 19 55 O=C(CCc1cn[nH]c1)Nc1ccc([C@H](O)C(F)(F)F)cc1 ZINC000880982460 DF On-Demand Anodyne ROCK2 19 55 C[C@H](O)c1ccc(OCc2cn(CCOc3ccccc3F)nn2)cc1 ZINC000880982500 FG On-Demand Anodyne MMP13 22 40 C[C@H](O)c1ccc(OCc2cn(CCOc3ccccc3F)nn2)cc1 ZINC000880982500 FG On-Demand Anodyne MMP8 34 40 CC(=O)N1CCN(Cc2cn(CCOc3ccccc3F)nn2)CC1 ZINC000880982525 ED On-Demand Anodyne DRD3 15 48 CC(C)(C)OC(=O)N1CCN(Cc2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880982526 GE On-Demand Mild GPR119 23 41 CC(C)(C)OC(=O)N1CCN(Cc2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880982526 GE On-Demand Mild KDM1A 22 47 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(C2CC3(C2)OCCO3)nn1 ZINC000880982527 GH On-Demand Anodyne SOAT1 41 41 CC(C)(C)OC(=O)N1CC[C@H](c2cn(Cc3ccccc3C#N)nn2)C1 ZINC000880982536 FF On-Demand Mild GPR119 31 40 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(Cc3ccccc3C#N)nn2)C1 ZINC000880982537 FF On-Demand Mild GPR119 31 40 CCC[C@@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982563 DE On-Demand Anodyne NQO2 27 43 CCC[C@@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982563 DE On-Demand Anodyne MTNR1A 48 39 CCC[C@@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982563 DE On-Demand Anodyne MTNR1B 44 39 CCOC(=O)CCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982564 EE On-Demand Anodyne KDR 49 38 CCOC(=O)CCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982564 EE On-Demand Anodyne PDGFRA 51 38 CCC[C@@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982565 DE On-Demand Anodyne NQO2 27 43 CCC[C@@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982565 DE On-Demand Anodyne MTNR1A 48 39 CCC[C@@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982565 DE On-Demand Anodyne MTNR1B 44 39 CCC[C@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982566 DE On-Demand Anodyne NQO2 27 43 CCC[C@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982566 DE On-Demand Anodyne MTNR1A 48 39 CCC[C@H](CCO)NC(=O)[C@@H]1CCc2cc(OC)ccc2C1 ZINC000880982566 DE On-Demand Anodyne MTNR1B 44 39 CCC[C@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982567 DE On-Demand Anodyne NQO2 27 43 CCC[C@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982567 DE On-Demand Anodyne MTNR1A 48 39 CCC[C@H](CCO)NC(=O)[C@H]1CCc2cc(OC)ccc2C1 ZINC000880982567 DE On-Demand Anodyne MTNR1B 44 39 CC[C@@](C)(CCO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982573 EF On-Demand Anodyne PDGFRA 50 37 O=C(Cn1cc([C@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1nccs1 ZINC000880982579 DD On-Demand Anodyne MAP1 59 36 O=C(Cn1cc([C@@]2(O)C[C@H]3CC[C@H]2C3)nn1)Nc1nccs1 ZINC000880982582 DD On-Demand Anodyne MAP1 59 36 O=C(Nc1ccc([C@@H](O)C(F)(F)F)cc1)c1ncsc1C1CC1 ZINC000880982591 EH On-Demand Anodyne MAP1 59 35 O=C(Nc1ccc([C@H](O)C(F)(F)F)cc1)c1ncsc1C1CC1 ZINC000880982593 EH On-Demand Anodyne MAP1 59 35 CC[C@@](C)(CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982600 EF On-Demand Anodyne KDR 42 37 CC[C@@](C)(CO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982600 EF On-Demand Anodyne PDGFRA 51 38 O=C1CCC[C@@H](c2cn(CC(=O)Nc3nc(-c4ccc(F)cc4)cs3)nn2)C1 ZINC000880982625 GG On-Demand Anodyne MAOB 15 41 O=C1CCC[C@H](c2cn(CC(=O)Nc3nc(-c4ccc(F)cc4)cs3)nn2)C1 ZINC000880982628 GG On-Demand Anodyne MAOB 15 41 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1nccs1 ZINC000880982643 CC On-Demand Anodyne MAP1 87 43 COCCN(CCOC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982649 FE On-Demand Anodyne PDGFRB 40 36 COCCN(CCOC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982649 FE On-Demand Anodyne KDR 63 36 COCCN(CCOC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982649 FE On-Demand Anodyne PDGFRA 54 40 O=C(Cc1ccccc1N1CCCC1=O)Nc1ccc([C@H](O)C(F)(F)F)cc1 ZINC000880982661 GH On-Demand Anodyne KCNQ2 69 38 O=C(Cc1ccccc1N1CCCC1=O)Nc1ccc([C@@H](O)C(F)(F)F)cc1 ZINC000880982662 GH On-Demand Anodyne KCNQ2 69 38 N#Cc1c(NC(=O)Cn2cc([C@@H]3CCCCO3)nn2)sc2c1CCCCC2 ZINC000880982665 GG On-Demand Mild VIPR1 29 46 N#Cc1c(NC(=O)Cn2cc([C@H]3CCCCO3)nn2)sc2c1CCCCC2 ZINC000880982666 GG On-Demand Mild VIPR1 29 46 O=C(Cn1cc(CCCOc2cccnc2F)nn1)Nc1nccs1 ZINC000880982671 FD On-Demand Anodyne MAP1 105 41 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne HTR4 49 38 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne CCR3 18 43 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne KDR 41 36 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne SLC9A1 40 33 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne MET 48 35 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne PDGFRA 53 43 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne PDK1 45 32 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne MCHR1 20 42 COCCN1CCC(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880982697 GE On-Demand Anodyne EHMT2 49 30 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982706 FD On-Demand Anodyne KDR 62 36 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982706 FD On-Demand Anodyne PDGFRA 55 39 O=C(Cn1cc(C2(O)CCCCC2)nn1)Nc1nccs1 ZINC000880982715 DD On-Demand Anodyne MAP1 85 42 O=C(Cn1cc(C2CC3(C2)OCCO3)nn1)Nc1nccs1 ZINC000880982719 DC On-Demand Anodyne MAP1 61 37 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982723 FE On-Demand Anodyne PDGFRA 50 37 COC(=O)[C@@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982723 FE On-Demand Anodyne PTR1 45 32 COC(=O)[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982724 FE On-Demand Anodyne PDGFRA 50 37 COC(=O)[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982724 FE On-Demand Anodyne PTR1 45 32 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(CON)nn1 ZINC000880982771 EF On-Demand Anodyne SOAT1 62 46 CC(C)(C)OC(=O)N1CC[C@H](c2cn(CC(=O)c3c[nH]c4ccccc34)nn2)C1 ZINC000880982784 GG On-Demand Anodyne SSTR2 64 37 CC(C)(C)OC(=O)N1CC[C@@H](c2cn(CC(=O)c3c[nH]c4ccccc34)nn2)C1 ZINC000880982785 GG On-Demand Anodyne SSTR2 64 37 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(-c2cccnc2Cl)nn1 ZINC000880982810 GJ On-Demand Anodyne SOAT1 51 43 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](O)c2ccccc2)nn1 ZINC000880982824 GI On-Demand Anodyne SOAT1 78 45 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](O)c2ccccc2)nn1 ZINC000880982825 GI On-Demand Anodyne SOAT1 78 45 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H]2CCCCO2)nn1 ZINC000880982837 FI On-Demand Anodyne SOAT1 45 44 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H]2CCCCO2)nn1 ZINC000880982838 FI On-Demand Anodyne SOAT1 45 44 CCOCCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982927 EG On-Demand Anodyne PDGFRA 51 39 CCS(=O)(=O)C[C@@H](C)N(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982929 GF On-Demand Anodyne PDGFRA 50 37 CCS(=O)(=O)C[C@H](C)N(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982931 GF On-Demand Anodyne PDGFRA 50 37 CCOCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982936 DE On-Demand Anodyne KDR 51 38 CCOCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982936 DE On-Demand Anodyne PDGFRA 53 39 CCN(Cc1ccccn1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982969 FH On-Demand Anodyne KDR 42 38 CCN(Cc1ccccn1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880982969 FH On-Demand Anodyne PDGFRA 49 38 CCOC[C@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880982994 FH On-Demand Anodyne PDGFRB 51 36 O=C(Cn1cc(C2CCC(C3OCCO3)CC2)nn1)Nc1nccs1 ZINC000880983003 FE On-Demand Anodyne MAP1 56 36 CNC(=O)CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983008 ED On-Demand Anodyne KDR 58 36 CNC(=O)CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983008 ED On-Demand Anodyne PDGFRA 53 39 CCC[C@@H](CCO)NC(=O)c1cc2ccccc2cc1F ZINC000880983017 CG On-Demand Anodyne PYGL 22 40 CCC[C@H](CCO)NC(=O)c1cc2ccccc2cc1F ZINC000880983020 CG On-Demand Anodyne PYGL 22 40 COCC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983029 FG On-Demand Anodyne PDGFRB 56 38 COCC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983029 FG On-Demand Anodyne PDGFRA 49 35 CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983031 CF On-Demand Anodyne PDGFRB 40 39 CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983031 CF On-Demand Anodyne KDR 72 40 CCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983031 CF On-Demand Anodyne PDGFRA 59 43 CC(=O)NCCc1cn(Cc2ccccc2C#N)nn1 ZINC000880983057 CC On-Demand Mild MTNR1A 40 36 Cc1nc(C(C)C)ncc1C(=O)Nc1ccc([C@H](O)C(F)(F)F)cc1 ZINC000880983084 FH On-Demand Anodyne JUN 21 43 Cc1nc(C(C)C)ncc1C(=O)Nc1ccc([C@H](O)C(F)(F)F)cc1 ZINC000880983084 FH On-Demand Anodyne ATF1 41 39 Cc1nc(C(C)C)ncc1C(=O)Nc1ccc([C@@H](O)C(F)(F)F)cc1 ZINC000880983085 FH On-Demand Anodyne JUN 21 43 Cc1nc(C(C)C)ncc1C(=O)Nc1ccc([C@@H](O)C(F)(F)F)cc1 ZINC000880983085 FH On-Demand Anodyne ATF1 41 39 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(C2(O)CCOCC2)nn1 ZINC000880983087 GG On-Demand Anodyne SOAT1 52 43 Oc1nc(Cn2cc(CCCN3CCOCC3)nn2)nc2ccccc12 ZINC000880983115 FD On-Demand Anodyne HNMT 42 31 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(-c2cccnc2F)nn1 ZINC000880983135 GI On-Demand Anodyne SOAT1 52 43 CCN(CC(C)(C)O)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983200 EF On-Demand Anodyne PDGFRA 50 37 COC(=O)[C@@]1(C)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983201 FF On-Demand Anodyne PDGFRA 43 34 COC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983203 FF On-Demand Anodyne PDGFRB 43 41 COC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983203 FF On-Demand Anodyne KDR 44 37 COC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983203 FF On-Demand Anodyne PDGFRA 50 36 COC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983203 FF On-Demand Anodyne PTR1 47 34 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983212 FE On-Demand Anodyne EPHX2 28 51 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983212 FE On-Demand Anodyne PDGFRA 46 41 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983213 FE On-Demand Anodyne EPHX2 28 51 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983213 FE On-Demand Anodyne PDGFRA 46 41 CCCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983253 EF On-Demand Anodyne PDGFRA 49 37 O=C1CCC[C@@H](c2cn(CC(=O)Nc3nccs3)nn2)C1 ZINC000880983272 DD On-Demand Anodyne MAP1 59 39 O=C1CCC[C@H](c2cn(CC(=O)Nc3nccs3)nn2)C1 ZINC000880983274 DD On-Demand Anodyne MAP1 59 39 CCCC[C@@H](C)N(C)C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880983286 FE On-Demand Anodyne SLC10A2 40 34 CCCC[C@H](C)N(C)C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880983291 FE On-Demand Anodyne SLC10A2 40 34 COCCN(CCC#N)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983295 FF On-Demand Mild PDGFRA 45 35 CCC(=O)N1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983301 GF On-Demand Anodyne PDGFRB 59 39 CCC(=O)N1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983301 GF On-Demand Anodyne PDGFRA 48 35 CCC(=O)N1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983301 GF On-Demand Anodyne RBP4 19 42 CC(C)(C)OC(=O)N1CCC(c2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880983305 FG On-Demand Mild GPR119 43 41 N#Cc1c(NC(=O)Cn2cc([C@@H]3CCOC3)nn2)sc2c1CCCCC2 ZINC000880983306 FF On-Demand Mild VIPR1 29 46 N#Cc1c(NC(=O)Cn2cc([C@H]3CCOC3)nn2)sc2c1CCCCC2 ZINC000880983308 FF On-Demand Mild VIPR1 29 46 C[C@@](O)(Cc1ccccc1)c1cn(CC(=O)Nc2nccs2)nn1 ZINC000880983315 ED On-Demand Anodyne MAP1 104 43 COc1ccc(-c2csc(NC(=O)Cn3cc([C@@H]4CCCCO4)nn3)n2)cc1 ZINC000880983321 GG On-Demand Anodyne CPT1A 21 41 COc1ccc(-c2csc(NC(=O)Cn3cc([C@H]4CCCCO4)nn3)n2)cc1 ZINC000880983322 GG On-Demand Anodyne CPT1A 21 41 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccccc2C#N)nn1 ZINC000880983326 FG On-Demand Mild DPP4 29 41 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2ccccc2C#N)nn1 ZINC000880983326 FG On-Demand Mild DPP9 22 41 CC[C@H](O)c1cn(CC(=O)Nc2c(C(C)C)cccc2C(C)C)nn1 ZINC000880983330 EH On-Demand Anodyne SOAT1 61 49 COCCCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983351 EG On-Demand Anodyne KDR 53 37 COCCCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983351 EG On-Demand Anodyne PDGFRA 53 38 C#CCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983355 CE On-Demand Mild KDR 51 38 C#CCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983355 CE On-Demand Mild PDGFRA 54 39 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(-c2cnc(Cl)nc2)nn1 ZINC000880983366 GI On-Demand Anodyne SOAT1 52 46 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880983385 GF On-Demand Mild SSTR5 43 36 CC(C)(C)OC(=O)NC1CCN(Cc2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880983385 GF On-Demand Mild MCHR1 19 40 CC(C)(C)OC(=O)N1CCCN(Cc2cn(Cc3ccccc3C#N)nn2)CC1 ZINC000880983386 GF On-Demand Mild KDM1A 21 45 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](O)C2CC2)nn1 ZINC000880983419 FH On-Demand Anodyne SOAT1 55 45 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](O)C2CC2)nn1 ZINC000880983420 FH On-Demand Anodyne SOAT1 55 45 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc(C2(O)CCC2)nn1 ZINC000880983421 FH On-Demand Anodyne SOAT1 57 45 O=C(Cn1cc(CCCN2CCOCC2)nn1)c1c[nH]c2ccccc12 ZINC000880983461 FD On-Demand Anodyne HTR1D 29 41 O=C(Cn1cc(CCCN2CCOCC2)nn1)c1c[nH]c2ccccc12 ZINC000880983461 FD On-Demand Anodyne HTR1B 24 41 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@@H](C)N)nn1 ZINC000880983462 EG On-Demand Anodyne SOAT1 62 48 CC(C)c1cccc(C(C)C)c1NC(=O)Cn1cc([C@H](C)N)nn1 ZINC000880983463 EG On-Demand Anodyne SOAT1 62 48 CCC[C@@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983486 ED On-Demand Anodyne CAPN1 48 35 CCC[C@@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983486 ED On-Demand Anodyne CAPN2 45 38 CCC[C@@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983486 ED On-Demand Anodyne XIAP 68 36 CCC[C@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983487 ED On-Demand Anodyne CAPN1 48 35 CCC[C@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983487 ED On-Demand Anodyne CAPN2 45 38 CCC[C@H](CCO)NC(=O)[C@@H]1CC[C@H](C(N)=O)N1Cc1ccccc1 ZINC000880983487 ED On-Demand Anodyne XIAP 68 36 CCC[C@@H](CCO)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880983494 EG On-Demand Anodyne ACACB 26 40 CCC[C@H](CCO)NC(=O)c1ccc(Oc2ccc(C)cn2)cc1 ZINC000880983495 EG On-Demand Anodyne ACACB 26 40 O=C(Cn1cc([C@@H]2CCOC2)nn1)Nc1nccs1 ZINC000880983607 CC On-Demand Anodyne MAP1 87 38 O=C(Cn1cc([C@H]2CCOC2)nn1)Nc1nccs1 ZINC000880983608 CC On-Demand Anodyne MAP1 87 38 COc1ccc(-c2csc(NC(=O)Cn3cc([C@@H]4CCOC4)nn3)n2)cc1 ZINC000880983610 GF On-Demand Anodyne SPHK2 23 40 COc1ccc(-c2csc(NC(=O)Cn3cc([C@@H]4CCOC4)nn3)n2)cc1 ZINC000880983610 GF On-Demand Anodyne SPHK1 25 40 COc1ccc(-c2csc(NC(=O)Cn3cc([C@H]4CCOC4)nn3)n2)cc1 ZINC000880983611 GF On-Demand Anodyne SPHK2 23 40 COc1ccc(-c2csc(NC(=O)Cn3cc([C@H]4CCOC4)nn3)n2)cc1 ZINC000880983611 GF On-Demand Anodyne SPHK1 25 40 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983645 GE On-Demand Anodyne PDGFRB 53 40 CC[C@H](O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983645 GE On-Demand Anodyne PDGFRA 44 35 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983646 GE On-Demand Anodyne PDGFRB 53 40 CC[C@@H](O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983646 GE On-Demand Anodyne PDGFRA 44 35 CCC[C@H](CCO)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880983682 DE On-Demand Anodyne MPO 64 37 CCC[C@@H](CCO)NC(=O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880983683 DE On-Demand Anodyne MPO 64 37 COCCn1nc(C)c(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)c1C ZINC000880983691 GG On-Demand Anodyne PDGFRA 49 38 CCOC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983719 GG On-Demand Anodyne PDGFRB 44 38 CCOC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983719 GG On-Demand Anodyne PDGFRA 44 34 CCOC(=O)C1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983719 GG On-Demand Anodyne PTR1 49 35 COCCN(Cc1ccccn1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983724 GG On-Demand Anodyne PDGFRA 44 37 C[C@]1(C(F)(F)F)CCN(C(=O)Nc2ccc3c(c2)S(=O)(=O)CC(=O)N3)C1 ZINC000880983727 GE On-Demand Anodyne EPHX2 31 41 C[C@H]1c2sccc2CCN1C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880983729 GF On-Demand Anodyne TRPM8 17 42 O=C(Nc1ccc([C@H](O)C(F)(F)F)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880983731 GF On-Demand Anodyne EPHX2 21 41 O=C(Nc1ccc([C@@H](O)C(F)(F)F)cc1)c1ccc(CN2CCOCC2)o1 ZINC000880983732 GF On-Demand Anodyne EPHX2 21 41 Cn1ncc(Br)c1CC(=O)Nc1ccc([C@@H](O)C(F)(F)F)cc1 ZINC000880983750 GF On-Demand Anodyne HTR2A 21 40 Cn1ncc(Br)c1CC(=O)Nc1ccc([C@H](O)C(F)(F)F)cc1 ZINC000880983751 GF On-Demand Anodyne HTR2A 21 40 COC[C@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983758 EF On-Demand Anodyne KDR 40 37 COC[C@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983758 EF On-Demand Anodyne PDGFRA 52 38 COC[C@@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983759 EF On-Demand Anodyne KDR 40 37 COC[C@@H](C)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983759 EF On-Demand Anodyne PDGFRA 52 38 CCC[C@@H](CCO)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880983765 DE On-Demand Anodyne KCNQ2 64 38 CCC[C@H](CCO)NC(=O)Cc1ccccc1N1CCCC1=O ZINC000880983766 DE On-Demand Anodyne KCNQ2 64 38 CCOCCCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983777 EF On-Demand Anodyne PDGFRA 52 39 CCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983787 EE On-Demand Anodyne KDR 41 35 CCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983787 EE On-Demand Anodyne ROCK2 18 40 CCCN(CCO)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983787 EE On-Demand Anodyne PDGFRA 51 38 COCCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983800 EF On-Demand Anodyne KDR 67 37 COCCCN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983800 EF On-Demand Anodyne PDGFRA 54 40 CC(=O)N1CCN(Cc2cn(Cc3ccc(C)cc3)nn2)CC1 ZINC000880983815 DD On-Demand Anodyne KDM1A 17 52 CNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983822 FE On-Demand Anodyne PDGFRA 45 41 CNC(=O)[C@@H](C)CN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983827 FE On-Demand Anodyne KDR 67 39 CNC(=O)[C@@H](C)CN(C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983827 FE On-Demand Anodyne PDGFRA 55 40 C=C[C@@](C)(O)c1cn(CC(=O)Nc2nccs2)nn1 ZINC000880983867 CC On-Demand Mild MAP1 91 39 C=C[C@](C)(O)c1cn(CC(=O)Nc2nccs2)nn1 ZINC000880983868 CC On-Demand Mild MAP1 91 39 COCC(C)(C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983877 EF On-Demand Anodyne KDR 57 38 COCC(C)(C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983877 EF On-Demand Anodyne PDGFRA 54 39 CC[C@@](C)(O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983885 EF On-Demand Anodyne KDR 45 37 CC[C@@](C)(O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983885 EF On-Demand Anodyne PDGFRA 53 38 COC(=O)[C@@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCO1 ZINC000880983896 GD On-Demand Anodyne PDGFRA 42 33 COC(=O)[C@H]1CN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CCO1 ZINC000880983897 GD On-Demand Anodyne PDGFRA 42 33 CCOCCN(CC)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983898 EG On-Demand Anodyne PDGFRA 50 37 CCC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983901 EF On-Demand Anodyne KDR 48 36 CCC[C@@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983901 EF On-Demand Anodyne PDGFRA 50 37 CCC[C@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983902 EF On-Demand Anodyne KDR 48 36 CCC[C@H](O)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880983902 EF On-Demand Anodyne PDGFRA 50 37 O=C(Cn1cc(CCCCCCO)nn1)Nc1nccs1 ZINC000880983908 DD On-Demand Anodyne MAP1 119 40 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983911 FG On-Demand Anodyne PDGFRB 54 37 COC[C@@H]1CCCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880983911 FG On-Demand Anodyne PDGFRA 48 38 CNC(=O)CC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983964 GF On-Demand Anodyne PDGFRB 49 36 CNC(=O)CC1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880983964 GF On-Demand Anodyne PDGFRA 42 34 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1nccs1 ZINC000880983968 EC On-Demand Anodyne MAP1 58 40 O=C(Cn1cc([C@@H]2CCCCO2)nn1)Nc1nccs1 ZINC000880983975 CD On-Demand Anodyne MAP1 79 39 O=C(Cn1cc([C@H]2CCCCO2)nn1)Nc1nccs1 ZINC000880983976 CD On-Demand Anodyne MAP1 79 39 O=C(Cn1cc(CN[C@H]2CCCc3ccccc32)nn1)Nc1nccs1 ZINC000880983981 FF On-Demand Anodyne MAP1 51 35 O=C(Cn1cc(CN[C@@H]2CCCc3ccccc32)nn1)Nc1nccs1 ZINC000880983982 FF On-Demand Anodyne MAP1 51 35 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880983987 FF On-Demand Anodyne ROCK1 19 42 CC[C@@](C)(O)c1cn(CC(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880983991 GF On-Demand Anodyne ROCK1 19 41 COCC1(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984008 EF On-Demand Anodyne KDR 54 37 COCC1(NC(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984008 EF On-Demand Anodyne PDGFRA 53 38 C[C@@](O)(Cc1cn(CC(=O)Nc2nccs2)nn1)c1cccs1 ZINC000880984016 ED On-Demand Anodyne MAP1 95 37 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984029 GD On-Demand Anodyne PDGFRB 59 39 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984029 GD On-Demand Anodyne MET 18 43 CNC(=O)CN1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984029 GD On-Demand Anodyne PDGFRA 46 35 CC(=O)N1CCN(Cc2cn(CC(=O)Nc3nccs3)nn2)CC1 ZINC000880984037 EC On-Demand Anodyne MAP1 86 42 COC(=O)[C@@H]1CC12CCN(C(=O)Nc1cc(OC)cc3c(OC)ccnc13)CC2 ZINC000880984055 GG On-Demand Anodyne PDGFRA 43 33 CC(C)(C)NC(=O)Cn1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880984061 EF On-Demand Anodyne MAP3K5 47 35 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CASP3 17 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne BMP1 21 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne KLK3 77 36 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CTSB 67 45 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne PAPA1_CARPA 73 36 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CYSP_TRYCR 50 38 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CTSK 37 42 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CTSL 43 38 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne PREP 15 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CAPNS1 65 38 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CTSS 16 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne GHSR 32 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CAPN1 87 45 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne CAPN2 138 45 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne NPR 77 41 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne PSMB5 43 37 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne Q6PRC7_IXORI 41 33 CC[C@H](C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880984075 ED On-Demand Anodyne PDS 50 34 CC(C)(C)NC(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880984080 FE On-Demand Anodyne GPR119 42 41 CC[C@H](C)NC(=O)Cn1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880984111 GD On-Demand Anodyne KDM1A 21 47 O=C(N[C@@H](CCc1ccccc1)c1ccccn1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880984117 GG On-Demand Anodyne F11 37 40 O=C(N[C@H](CCc1ccccc1)c1ccccn1)[C@H]1C[C@@H]2CC[C@H](C1)S2(=O)=O ZINC000880984118 GG On-Demand Anodyne F11 37 40 Cc1cccc2c1CCN(C(=O)Nc1ccc3c(c1)S(=O)(=O)CC(=O)N3)C2 ZINC000880984139 GE On-Demand Anodyne P2RY14 52 37 CC(C)(C)NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880984140 ED On-Demand Anodyne MMP8 18 46 Cn1nc2c(c1-c1cn(CC(=O)Nc3nccs3)nn1)CCCC2 ZINC000880984221 ED On-Demand Anodyne MAP1 51 37 CC[C@H](CCO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984227 EF On-Demand Anodyne PDGFRA 51 38 CC[C@@H](CCO)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984228 EF On-Demand Anodyne PDGFRA 51 38 CC[C@H](CCO)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984238 EF On-Demand Anodyne PDGFRA 51 37 CC[C@@H](CCO)CNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984239 EF On-Demand Anodyne PDGFRA 51 37 O=C(Cn1cc(C2(O)CCC2)nn1)Nc1nc(-c2ccc(F)cc2)cs1 ZINC000880984243 FF On-Demand Anodyne ROCK1 18 43 CC[C@@H](O)CCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984246 EF On-Demand Anodyne PDGFRA 53 38 CC[C@H](O)CCNC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984247 EF On-Demand Anodyne PDGFRA 53 38 COC(=O)Cc1cn(CC(=O)Nc2nccs2)nn1 ZINC000880984250 CC On-Demand Anodyne MAP1 125 41 COCC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984261 EF On-Demand Anodyne PDGFRB 29 41 COCC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984261 EF On-Demand Anodyne KDR 65 37 COCC[C@@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984261 EF On-Demand Anodyne PDGFRA 53 41 COCC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984262 EF On-Demand Anodyne PDGFRB 29 41 COCC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984262 EF On-Demand Anodyne KDR 65 37 COCC[C@H](C)NC(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984262 EF On-Demand Anodyne PDGFRA 53 41 CCOC[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880984264 FG On-Demand Anodyne PDGFRB 45 35 CCOC[C@H]1CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)C1 ZINC000880984264 FG On-Demand Anodyne PDGFRA 43 34 COC(=O)C1CCC(c2cn(CC(=O)Nc3nccs3)nn2)CC1 ZINC000880984276 ED On-Demand Anodyne MAP1 108 39 CCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984279 FG On-Demand Anodyne PDGFRB 56 38 CCC1(O)CCN(C(=O)Nc2cc(OC)cc3c(OC)ccnc23)CC1 ZINC000880984279 FG On-Demand Anodyne PDGFRA 47 35 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1nc(-c2ccc(F)cc2)cs1 ZINC000880984287 FF On-Demand Anodyne ROCK1 17 41 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1nc(-c2ccc(F)cc2)cs1 ZINC000880984291 FF On-Demand Anodyne ROCK1 17 41 CC[C@H](C)NC(=O)Cn1cc([C@@H]2CCN(C(=O)OC(C)(C)C)C2)nn1 ZINC000880984377 FD On-Demand Anodyne GPR119 29 40 CC[C@H](C)NC(=O)Cn1cc([C@H]2CCN(C(=O)OC(C)(C)C)C2)nn1 ZINC000880984378 FD On-Demand Anodyne GPR119 29 40 CC(C)(C)N(Cc1ccccc1)C(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880984379 GE On-Demand Anodyne CYP2J2 45 32 CC(C)(C)NC(=O)Cn1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880984387 GD On-Demand Anodyne KDM1A 21 48 COCCN(CCN(C)C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984403 GE On-Demand Anodyne KDR 48 34 COCCN(CCN(C)C)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984403 GE On-Demand Anodyne PDGFRA 49 37 O=C(Cn1cc([C@@H](O)C2CC2)nn1)Nc1nccs1 ZINC000880984406 CC On-Demand Anodyne MAP1 105 40 O=C(Cn1cc([C@H](O)C2CC2)nn1)Nc1nccs1 ZINC000880984407 CC On-Demand Anodyne MAP1 105 40 COCCN(Cc1cccnc1)C(=O)Nc1cc(OC)cc2c(OC)ccnc12 ZINC000880984425 GG On-Demand Anodyne ROCK2 35 44 O=C(Cn1cc(CCCN2CCOCC2)nn1)Nc1ccc(OC(F)F)cc1 ZINC000880984442 GD On-Demand Anodyne EPHX2 22 45 CC(C)(C)NC(=O)Cn1cc(CN2CCCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880984497 GD On-Demand Anodyne KDM1A 20 45 CC(=O)N1CCN(C(=O)Cn2cc(-c3ccc(Cl)cc3F)nn2)CC1 ZINC000880984562 FD On-Demand Anodyne IL2RA 49 33 C[C@@H]1Cc2ccccc2CN1C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880984693 GE On-Demand Anodyne CFTR 43 32 C[C@H]1Cc2ccccc2CN1C(=O)Nc1ccc2c(c1)S(=O)(=O)CC(=O)N2 ZINC000880984694 GE On-Demand Anodyne CFTR 43 32 CC(C)(C)NC(=O)Cn1cc(-c2ccc(Cl)cc2F)nn1 ZINC000880984699 DF On-Demand Anodyne ALPL 34 43 CCCCNC(=O)Cn1cc([C@@H](O)c2ccc(F)cc2)nn1 ZINC000880984788 DD On-Demand Anodyne ASAH1 46 31 CCCCNC(=O)Cn1cc([C@H](O)c2ccc(F)cc2)nn1 ZINC000880984789 DD On-Demand Anodyne ASAH1 46 31 C#CC1(F)CN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880984848 CE On-Demand Mild CSNK2A1 24 40 CN1CCN(C(=O)Nc2ccc3c(c2)S(=O)(=O)CC(=O)N3)CC1 ZINC000880984866 EC On-Demand Anodyne HTR1B 15 43 Brc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880984912 GE On-Demand Anodyne LTA4H 28 43 Brc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880984912 GE On-Demand Anodyne HRH3 41 46 CC[C@H](C)NC(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880984927 FE On-Demand Anodyne GPR119 41 42 CC(=O)Nc1cccc2c1CN(C(=O)Nc1cc(C#N)c(F)cc1C)CC2 ZINC000880985007 FH On-Demand Mild CSNK2A1 43 40 COCCCNC(=O)Cn1cc(-c2ccc(Cl)cc2F)nn1 ZINC000880985016 ED On-Demand Anodyne ALPL 53 41 CC(=O)NC[C@@H]1CCCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880985030 EF On-Demand Mild CSNK2A1 37 43 C#C[C@@H]1CC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880985042 CG On-Demand Mild CSNK2A1 27 42 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne KLK3 44 33 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne CTSB 40 39 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne CTSK 22 42 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne CAPNS1 49 36 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne GHSR 21 44 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne CAPN1 63 41 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne CAPN2 106 43 CCCCNC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985047 ED On-Demand Anodyne NPR 66 46 Cc1csc([C@H]2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)C2)n1 ZINC000880985052 EH On-Demand Mild CSNK2A1 21 40 CS[C@@H]1C[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880985113 CG On-Demand Mild CSNK2A1 27 41 CCCCNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985152 DD On-Demand Anodyne GRIA1 41 33 CCCCNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985152 DD On-Demand Anodyne PLM2_PLAFA 23 40 CCCCNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985152 DD On-Demand Anodyne NPFFR1 41 33 CCCCNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985153 DD On-Demand Anodyne GRIA1 41 33 CCCCNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985153 DD On-Demand Anodyne PLM2_PLAFA 23 40 CCCCNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985153 DD On-Demand Anodyne NPFFR1 41 33 CCCCNC(=O)Cn1cc(-c2cccnc2F)nn1 ZINC000880985154 CD On-Demand Anodyne ASAH1 45 31 CC[C@H](C)NC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985211 DD On-Demand Anodyne MME 57 38 CC[C@H](C)NC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985211 DD On-Demand Anodyne FCER2 49 34 CC[C@H](C)NC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985211 DD On-Demand Anodyne CAPNS1 42 30 CC[C@H](C)NC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985211 DD On-Demand Anodyne ACE2 47 36 CC[C@H](C)NC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985212 DD On-Demand Anodyne MME 57 38 CC[C@H](C)NC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985212 DD On-Demand Anodyne FCER2 49 34 CC[C@H](C)NC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985212 DD On-Demand Anodyne CAPNS1 42 30 CC[C@H](C)NC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985212 DD On-Demand Anodyne ACE2 47 36 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne PREP 17 44 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne CAPNS1 53 33 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne GHSR 33 42 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne CAPN1 60 37 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne CAPN2 98 37 CC(C)(C)NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880985222 ED On-Demand Anodyne NPR 64 37 CC[C@H](C)NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880985255 ED On-Demand Anodyne MMP13 21 51 CC[C@H](C)NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880985255 ED On-Demand Anodyne MMP8 27 49 CCCCNC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880985292 ED On-Demand Anodyne MMP8 18 45 CCCCNC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880985292 ED On-Demand Anodyne ASAH1 41 31 CCCCNC(=O)Cn1cc(CN2CCCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880985326 GD On-Demand Anodyne KDM1A 19 42 CC(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880985404 DF On-Demand Mild CSNK2A1 27 42 O=C(COC1CC1)N[C@H](CCc1ccccc1)c1ccccn1 ZINC000880985476 DG On-Demand Anodyne TIMP3 76 40 O=C(COC1CC1)N[C@@H](CCc1ccccc1)c1ccccn1 ZINC000880985477 DG On-Demand Anodyne TIMP3 76 40 COCCCNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880985570 DC On-Demand Anodyne NPFFR1 40 30 COCCCNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880985571 DC On-Demand Anodyne NPFFR1 40 30 CC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880985625 DF On-Demand Mild CSNK2A1 24 41 CC(=O)[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880985626 DF On-Demand Mild CSNK2A1 24 41 CO[C@@H]1C[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880985640 CE On-Demand Mild CSNK2A1 27 40 CC[C@H](C)NC(=O)Cn1cc(CN[C@@H]2CCCc3ccccc32)nn1 ZINC000880985737 EE On-Demand Anodyne BIRC2 40 37 CC[C@H](C)NC(=O)Cn1cc(CN[C@H]2CCCc3ccccc32)nn1 ZINC000880985740 EE On-Demand Anodyne BIRC2 40 37 CC[C@H](C)NC(=O)Cn1cc(CN2CCCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880985764 GD On-Demand Anodyne KDM1A 20 45 CC(=O)N1CCN(C(=O)Cn2cc(CCCOc3cccnc3F)nn2)CC1 ZINC000880985801 GC On-Demand Anodyne MMP13 15 48 CC(=O)N1CCN(C(=O)Cn2cc(CCCOc3cccnc3F)nn2)CC1 ZINC000880985801 GC On-Demand Anodyne MMP8 26 47 CCCCNC(=O)Cn1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880985804 GD On-Demand Anodyne KDM1A 20 44 Cc1cncc([C@H]2CCCN2C(=O)Nc2cc(C#N)c(F)cc2C)c1 ZINC000880985828 EI On-Demand Mild CSNK2A1 21 40 Cc1cncc([C@@H]2CCCN2C(=O)Nc2cc(C#N)c(F)cc2C)c1 ZINC000880985830 EI On-Demand Mild CSNK2A1 21 40 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880985834 DG On-Demand Mild CSNK2A1 24 41 CCCCNC(=O)Cn1cc(CNC(=O)C(F)(F)F)nn1 ZINC000880985848 DC On-Demand Anodyne ASAH1 51 31 COc1cccc([C@H](O)C2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)c1 ZINC000880985895 GH On-Demand Mild TAAR1 23 43 CCCCNC(=O)Cn1cc([C@@H](O)c2ccc(Cl)cc2F)nn1 ZINC000880985903 EE On-Demand Anodyne ASAH1 41 31 CCCCNC(=O)Cn1cc([C@H](O)c2ccc(Cl)cc2F)nn1 ZINC000880985904 EE On-Demand Anodyne ASAH1 41 31 C=C1C[C@@H]2CC[C@H](C1)N2C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880985940 CH On-Demand Mild CSNK2A1 21 40 COCCCNC(=O)Cn1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880985949 FD On-Demand Anodyne MAP3K5 44 33 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccccn3)nn2)CC1 ZINC000880985959 EC On-Demand Anodyne P2RY12 52 40 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccccn3)nn2)CC1 ZINC000880985959 EC On-Demand Anodyne METAP1 21 42 CNC(=O)Cn1cc(CN2CCCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880985979 FC On-Demand Anodyne KDM1A 21 46 CNC(=O)Cn1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880986001 EC On-Demand Anodyne KDM1A 22 49 CNC(=O)Cn1cc(C(=O)c2ccc(C(C)(C)C)cc2)nn1 ZINC000880986005 DD On-Demand Anodyne MAP3K5 48 36 CCOC(=O)N1CCN(C(=O)Cn2cc(CN(C)c3ccccc3)nn2)CC1 ZINC000880986085 GD On-Demand Anodyne P2RY12 47 39 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccc(OC)cc3)nn2)CC1 ZINC000880986088 FD On-Demand Anodyne P2RY12 74 46 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne CTSB 41 38 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne PAPA1_CARPA 43 31 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne CYSP_TRYCR 46 40 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne CAPNS1 58 34 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne HDAC1 15 45 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne GHSR 22 43 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne CAPN1 60 40 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne CAPN2 98 40 CNC(=O)Cn1cc(CCCCNC(=O)OCc2ccccc2)nn1 ZINC000880986089 ED On-Demand Anodyne NPR 64 39 COCCCNC(=O)Cn1cc(COc2cccc(C(C)=O)c2)nn1 ZINC000880986094 ED On-Demand Anodyne DRD4 41 31 CNC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880986144 CC On-Demand Anodyne MMP13 15 49 CNC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880986144 CC On-Demand Anodyne MMP8 26 48 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cc(F)cc(F)c3)nn2)CC1 ZINC000880986230 GD On-Demand Anodyne P2RY12 37 40 CCOC(=O)N1CCN(C(=O)Cn2cc(Cn3cnc4ccccc43)nn2)CC1 ZINC000880986295 GC On-Demand Anodyne PKM 18 41 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(COC)c3)nn2)CC1 ZINC000880986296 GD On-Demand Anodyne P2RY12 60 40 COCCCNC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880986366 EB On-Demand Anodyne DRD3 21 41 COC[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880986412 CF On-Demand Mild LGMN 57 34 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccnc3)nn2)CC1 ZINC000880986418 EC On-Demand Anodyne P2RY12 51 41 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccccc3F)nn2)CC1 ZINC000880986421 FD On-Demand Anodyne GABRA3 45 39 CCOC(=O)N1CCN(C(=O)Cn2cc(CCOc3ccccc3)nn2)CC1 ZINC000880986437 GD On-Demand Anodyne P2RY12 64 38 CO[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880986445 DG On-Demand Mild CSNK2A1 25 42 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(C)n3)nn2)CC1 ZINC000880986465 FC On-Demand Anodyne P2RY12 43 40 CC[C@@H](O)CNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880986476 CD On-Demand Mild ADRB1 40 34 CNC(=O)Cn1cc(CN[C@H]2CCCc3ccccc32)nn1 ZINC000880986525 CD On-Demand Anodyne BIRC3 34 41 CNC(=O)Cn1cc(CN[C@H]2CCCc3ccccc32)nn1 ZINC000880986525 CD On-Demand Anodyne BIRC2 42 41 CNC(=O)Cn1cc(CN[C@@H]2CCCc3ccccc32)nn1 ZINC000880986527 CD On-Demand Anodyne BIRC3 34 41 CNC(=O)Cn1cc(CN[C@@H]2CCCc3ccccc32)nn1 ZINC000880986527 CD On-Demand Anodyne BIRC2 42 41 COC[C@@H](NC(=O)Nc1cc(C#N)c(F)cc1C)c1cccc(OC)c1 ZINC000880986561 FH On-Demand Mild TAAR1 17 45 COC[C@H](NC(=O)Nc1cc(C#N)c(F)cc1C)c1cccc(OC)c1 ZINC000880986562 FH On-Demand Mild TAAR1 17 45 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccncc3)nn2)CC1 ZINC000880986620 EC On-Demand Anodyne P2RY12 36 43 CCOC(=O)N1CCN(C(=O)Cn2cc(COc3ccc(C)cc3)nn2)CC1 ZINC000880986624 GD On-Demand Anodyne KDM1A 15 41 CNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880986677 CC On-Demand Anodyne MME 57 37 CNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880986677 CC On-Demand Anodyne FCER2 67 36 CNC(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880986677 CC On-Demand Anodyne AMP1_PLAFQ 41 35 CNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880986678 CC On-Demand Anodyne MME 57 37 CNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880986678 CC On-Demand Anodyne FCER2 67 36 CNC(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880986678 CC On-Demand Anodyne AMP1_PLAFQ 41 35 CNC(=O)Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 ZINC000880986743 DD On-Demand Anodyne GPR119 46 42 CC(=O)Nc1cccc2c1CCN(C(=O)Nc1cc(C#N)c(F)cc1C)C2 ZINC000880986774 FH On-Demand Mild CSNK2A1 51 42 CCNc1cccc(-c2cn(CC(=O)N3CCN(C(=O)OCC)CC3)nn2)c1 ZINC000880986859 GD On-Demand Anodyne P2RY12 86 42 CCNc1cccc(-c2cn(CC(=O)N3CCN(C(=O)OCC)CC3)nn2)c1 ZINC000880986859 GD On-Demand Anodyne HDAC10 19 40 CCNc1cccc(-c2cn(CC(=O)N3CCN(C(=O)OCC)CC3)nn2)c1 ZINC000880986859 GD On-Demand Anodyne HDAC3 22 41 CCNc1cccc(-c2cn(CC(=O)N3CCN(C(=O)OCC)CC3)nn2)c1 ZINC000880986859 GD On-Demand Anodyne HDAC6 17 41 C[C@@H]1CCCCN1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880986940 EE On-Demand Anodyne CPT1A 76 36 C[C@@H]1CCCCN1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880986941 EE On-Demand Anodyne CPT1A 76 36 C[C@H]1CCCCN1C(=O)Cn1cc([C@](C)(O)Cc2ccccc2)nn1 ZINC000880986943 EE On-Demand Anodyne CPT1A 76 36 C[C@H]1CCCCN1C(=O)Cn1cc([C@@](C)(O)Cc2ccccc2)nn1 ZINC000880986945 EE On-Demand Anodyne CPT1A 76 36 C[C@H]1CCCCN1C(=O)Cn1cc(-c2cnc(Cl)nc2)nn1 ZINC000880986955 DD On-Demand Anodyne CPT1A 47 36 C[C@@H]1CCCCN1C(=O)Cn1cc(-c2cnc(Cl)nc2)nn1 ZINC000880986957 DD On-Demand Anodyne CPT1A 47 36 CC(=O)N[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880986970 DD On-Demand Mild CSNK2A1 39 44 CC(=O)N[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880986972 DD On-Demand Mild CSNK2A1 39 44 CCOC(=O)N1CCN(C(=O)Cn2cc(C(=O)CCc3ccccc3)nn2)CC1 ZINC000880986981 GD On-Demand Anodyne P2RY12 84 41 CCOC(=O)N1CCN(C(=O)Cn2cc(C(=O)CCc3ccccc3)nn2)CC1 ZINC000880986981 GD On-Demand Anodyne FAAH 27 41 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2CCCC[C@H]2C)nn1 ZINC000880987007 FE On-Demand Anodyne CPT1A 42 34 C[C@H](O)c1ccccc1OCc1cn(CC(=O)N2CCCC[C@@H]2C)nn1 ZINC000880987009 FE On-Demand Anodyne CPT1A 42 34 C[C@H]1CCCCN1C(=O)Cn1cc(COc2ccccc2[C@@H](C)O)nn1 ZINC000880987013 FE On-Demand Anodyne CPT1A 42 34 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccsc3)nn2)CC1 ZINC000880987083 ED On-Demand Anodyne P2RY12 17 45 CCOC(=O)N1CCN(C(=O)Cn2cc(CSC)nn2)CC1 ZINC000880987109 EC On-Demand Anodyne KDM1A 17 42 C[C@H]1CCCCN1C(=O)Cn1cc(Cn2cnc(-c3ccccc3)c2N)nn1 ZINC000880987148 GE On-Demand Anodyne CPT1A 73 35 C[C@@H]1CCCCN1C(=O)Cn1cc(Cn2cnc(-c3ccccc3)c2N)nn1 ZINC000880987149 GE On-Demand Anodyne CPT1A 73 35 CON(C)C(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880987153 EE On-Demand Mild CSNK2A1 27 40 CCOC(=O)N1CCN(C(=O)Cn2cc(CNCc3ccccc3)nn2)CC1 ZINC000880987185 GC On-Demand Anodyne P2RY12 55 40 CCOC(=O)N1CCN(C(=O)Cn2cc(CNCc3ccccc3)nn2)CC1 ZINC000880987185 GC On-Demand Anodyne CCR8 16 42 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3CCCC[C@H]3C)nn2)cc1 ZINC000880987189 FE On-Demand Anodyne CPT1A 58 37 C[C@H](O)c1ccc(OCc2cn(CC(=O)N3CCCC[C@@H]3C)nn2)cc1 ZINC000880987190 FE On-Demand Anodyne CPT1A 58 37 C[C@H]1CCCCN1C(=O)Cn1cc(COc2ccc([C@@H](C)O)cc2)nn1 ZINC000880987192 FE On-Demand Anodyne CPT1A 58 37 C[C@@H]1CCCCN1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880987226 ED On-Demand Anodyne CPT1A 105 41 C[C@H]1CCCCN1C(=O)Cn1cc(COc2cccc(N)c2)nn1 ZINC000880987227 ED On-Demand Anodyne CPT1A 105 41 C#CCN(C(=O)Nc1cc(C#N)c(F)cc1C)C1CC1 ZINC000880987246 CF On-Demand Mild CSNK2A1 24 40 C[C@@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987248 ED On-Demand Anodyne ACE 33 41 C[C@@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987248 ED On-Demand Anodyne MME 20 41 C[C@@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987248 ED On-Demand Anodyne CPT1A 60 36 C[C@@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987248 ED On-Demand Anodyne PREP 54 35 C[C@@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987249 ED On-Demand Anodyne ACE 33 41 C[C@@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987249 ED On-Demand Anodyne MME 20 41 C[C@@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987249 ED On-Demand Anodyne CPT1A 60 36 C[C@@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987249 ED On-Demand Anodyne PREP 54 35 C[C@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987250 ED On-Demand Anodyne ACE 33 41 C[C@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987250 ED On-Demand Anodyne MME 20 41 C[C@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987250 ED On-Demand Anodyne CPT1A 60 36 C[C@H]1CCCCN1C(=O)Cn1cc([C@H](O)Cc2ccccc2)nn1 ZINC000880987250 ED On-Demand Anodyne PREP 54 35 C[C@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987251 ED On-Demand Anodyne ACE 33 41 C[C@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987251 ED On-Demand Anodyne MME 20 41 C[C@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987251 ED On-Demand Anodyne CPT1A 60 36 C[C@H]1CCCCN1C(=O)Cn1cc([C@@H](O)Cc2ccccc2)nn1 ZINC000880987251 ED On-Demand Anodyne PREP 54 35 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(NC)c3)nn2)CC1 ZINC000880987301 FD On-Demand Anodyne P2RY12 95 43 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(NC)c3)nn2)CC1 ZINC000880987301 FD On-Demand Anodyne HDAC10 18 40 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(NC)c3)nn2)CC1 ZINC000880987301 FD On-Demand Anodyne HDAC3 21 42 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cccc(NC)c3)nn2)CC1 ZINC000880987301 FD On-Demand Anodyne HDAC6 17 42 C#C[C@@H]1COCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880987312 CD On-Demand Mild CSNK2A1 29 43 C#C[C@H]1COCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880987313 CD On-Demand Mild CSNK2A1 29 43 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cnc4ccccc4c3)nn2)CC1 ZINC000880987321 GD On-Demand Anodyne P2RY12 106 43 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3cnc4ccccc4c3)nn2)CC1 ZINC000880987321 GD On-Demand Anodyne CCKAR 42 40 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA2 54 52 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA1 45 43 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA5B 48 38 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA4 44 52 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA5A 49 35 Cc1nc(CCNC(=O)c2cc(S(N)(=O)=O)ccc2F)cs1 ZINC000880987410 ED On-Demand Anodyne CA9 33 43 C[C@@H]1CCCCN1C(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880987549 ED On-Demand Anodyne CPT1A 49 35 C[C@@H]1CCCCN1C(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880987551 ED On-Demand Anodyne CPT1A 49 35 C[C@H]1CCCCN1C(=O)Cn1cc(C[C@@H](O)c2ccccc2)nn1 ZINC000880987552 ED On-Demand Anodyne CPT1A 49 35 C[C@H]1CCCCN1C(=O)Cn1cc(C[C@H](O)c2ccccc2)nn1 ZINC000880987553 ED On-Demand Anodyne CPT1A 49 35 CCOC(=O)N1CCN(C(=O)Cn2cc(C(=O)Cc3ccccc3)nn2)CC1 ZINC000880987554 GD On-Demand Anodyne P2RY12 60 41 C[C@@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2F)nn1 ZINC000880987627 DD On-Demand Anodyne CPT1A 55 36 C[C@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2F)nn1 ZINC000880987628 DD On-Demand Anodyne CPT1A 55 36 CCOC(=O)N1CCN(C(=O)Cn2cc(C(=O)c3ccccc3)nn2)CC1 ZINC000880987788 FC On-Demand Anodyne P2RY12 87 42 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880987797 GD On-Demand Anodyne G2YM83_BOTF4 69 36 C#C[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880987799 CF On-Demand Mild CSNK2A1 24 41 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880987800 GD On-Demand Anodyne G2YM83_BOTF4 69 36 C#C[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880987801 CF On-Demand Mild CSNK2A1 24 41 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)nc1 ZINC000880987964 FF On-Demand Mild P2RY12 22 42 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)nc1 ZINC000880987964 FF On-Demand Mild PDGFRB 50 37 COc1ccc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)nc1 ZINC000880987964 FF On-Demand Mild DGAT1 25 49 C[C@@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2Cl)nn1 ZINC000880987969 DE On-Demand Anodyne CPT1A 69 36 C[C@H]1CCCCN1C(=O)Cn1cc(-c2cccnc2Cl)nn1 ZINC000880987970 DE On-Demand Anodyne CPT1A 69 36 C#CC1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880988001 CF On-Demand Mild CSNK2A1 25 42 CCOC(=O)N1CCN(C(=O)Cn2cc(-c3ccc4ccccc4n3)nn2)CC1 ZINC000880988188 GD On-Demand Anodyne P2RY12 110 43 C[C@@H]1CCCCN1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880988274 ED On-Demand Clean CPT1A 78 38 C[C@H]1CCCCN1C(=O)Cn1cc(COc2ccc(N)cc2)nn1 ZINC000880988275 ED On-Demand Clean CPT1A 78 38 COCC1(O)CN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880988327 CD On-Demand Mild TRPV4 44 36 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1 ZINC000880988354 GG On-Demand Anodyne CCR2 48 39 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1 ZINC000880988355 GG On-Demand Anodyne CCR2 48 39 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc([C@H](O)c2cccc(C(F)(F)F)c2)nn1 ZINC000880988356 GG On-Demand Anodyne CCR2 48 39 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc([C@@H](O)c2cccc(C(F)(F)F)c2)nn1 ZINC000880988357 GG On-Demand Anodyne CCR2 48 39 COc1cccc(C2(NC(=O)Nc3cc(C#N)c(F)cc3C)CC2)c1 ZINC000880988461 EH On-Demand Mild TAAR1 21 46 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne ACE 26 41 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne FKBP1A 35 43 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne ELANE 27 41 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne CTRA_BOVIN 52 31 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne TRY1_BOVIN 57 33 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne CTSG 40 31 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne CPT1A 81 38 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne PREP 66 46 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne CAPN1 43 36 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne CAPN2 63 35 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne NPR 60 33 C[C@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988526 FE On-Demand Anodyne TMPRSS11D 46 36 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne ACE 26 41 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne FKBP1A 35 43 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne ELANE 27 41 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne CTRA_BOVIN 52 31 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne TRY1_BOVIN 57 33 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne CTSG 40 31 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne CPT1A 81 38 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne PREP 66 46 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne CAPN1 43 36 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne CAPN2 63 35 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne NPR 60 33 C[C@@H]1CCCCN1C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880988527 FE On-Demand Anodyne TMPRSS11D 46 36 COCCO[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880988653 EF On-Demand Mild CSNK2A1 24 42 COCCO[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880988654 EF On-Demand Mild CSNK2A1 24 42 C[C@H]1CCCCN1C(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880988671 FE On-Demand Anodyne MMP8 17 42 C[C@@H]1CCCCN1C(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880988672 FE On-Demand Anodyne MMP8 17 42 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880988685 GF On-Demand Anodyne MMP8 25 44 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc(CCCOc2cccnc2F)nn1 ZINC000880988688 GF On-Demand Anodyne MMP8 25 44 CCS(=O)(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)[C@H](C)C1 ZINC000880988911 FD On-Demand Mild LIMK2 43 35 CCCN(CCN1CCCC1)C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880988916 EG On-Demand Mild CASR 41 37 C[C@@H]1CCCCN1C(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880988934 DD On-Demand Anodyne CPT1A 58 36 C[C@H]1CCCCN1C(=O)Cn1cc(-c2ccc(F)nc2)nn1 ZINC000880988935 DD On-Demand Anodyne CPT1A 58 36 CC(=O)N(C[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C)C1CC1 ZINC000880989022 FG On-Demand Mild CSNK2A1 21 40 CC(=O)N(C[C@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C)C1CC1 ZINC000880989024 FG On-Demand Mild CSNK2A1 21 40 CNC(=O)OC[C@@H]1CCCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880989047 EF On-Demand Mild LGMN 61 34 CC(=O)N1CCN(Cc2cn(CC(=O)NCc3ccc(C)cc3)nn2)CC1 ZINC000880989101 FC On-Demand Anodyne KDM1A 15 42 CCC1(O)CN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880989551 CD On-Demand Mild CSNK2A1 21 40 C[C@@H]1CCCCN1C(=O)Cn1cc(COc2ccc(Br)nc2)nn1 ZINC000880989568 GE On-Demand Anodyne CPT1A 41 35 C[C@H]1CCCCN1C(=O)Cn1cc(COc2ccc(Br)nc2)nn1 ZINC000880989569 GE On-Demand Anodyne CPT1A 41 35 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989570 GE On-Demand Anodyne PREP 27 45 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989570 GE On-Demand Anodyne CAPN2 63 36 C[C@@H]1CCCC[C@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989570 GE On-Demand Anodyne NPR 58 33 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989572 GE On-Demand Anodyne PREP 27 45 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989572 GE On-Demand Anodyne CAPN2 63 36 C[C@@H]1CCCC[C@@H]1NC(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880989572 GE On-Demand Anodyne NPR 58 33 CC(=O)c1cccc(OCc2cn(CC(=O)N3CCCC[C@@H]3C)nn2)c1 ZINC000880989576 FE On-Demand Anodyne CPT1A 108 40 CC(=O)c1cccc(OCc2cn(CC(=O)N3CCCC[C@H]3C)nn2)c1 ZINC000880989577 FE On-Demand Anodyne CPT1A 108 40 COC[C@@H](O)CNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880989587 CD On-Demand Mild ADRB1 46 38 C=C(C)CN(CC)C(=O)Cn1cc(CNC(=O)c2cccnc2Cl)nn1 ZINC000880989652 GD On-Demand Mild G2YM83_BOTF4 64 33 COC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880989856 EE On-Demand Mild EPHX2 43 39 C=C(C)CN(CC)C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880990117 FE On-Demand Mild CAPNS1 48 34 C=C(C)CN(CC)C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880990117 FE On-Demand Mild CAPN1 45 37 C=C(C)CN(CC)C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880990117 FE On-Demand Mild CAPN2 80 37 C=C(C)CN(CC)C(=O)Cn1cc(CNC(=O)OCc2ccccc2)nn1 ZINC000880990117 FE On-Demand Mild NPR 64 36 COCCO[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880990292 DE On-Demand Mild CSNK2A1 21 40 COCCO[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880990293 DE On-Demand Mild CSNK2A1 21 40 CC(=O)c1ccccc1NC(=O)Cn1cc(CCCN2CCOCC2)nn1 ZINC000880990366 FD On-Demand Anodyne PRKDC 44 33 COc1cnccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880990418 FF On-Demand Mild HTR1B 15 42 COc1cnccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880990418 FF On-Demand Mild PDGFRB 41 41 COc1cnccc1N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880990418 FF On-Demand Mild RBP4 18 43 C[C@H](C(=O)Nc1nc(-c2ccc(F)c(F)c2)cs1)n1cc(C(C)(C)O)nn1 ZINC000880990614 GG On-Demand Anodyne MPL 15 41 CC[C@H](O)c1cn(CC(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880990626 GF On-Demand Anodyne MPL 17 42 CCOC(=O)N1CC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880990964 EE On-Demand Mild CCR8 47 38 CCOC(=O)N1CC[C@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880990965 EE On-Demand Mild CCR8 47 38 COC1(C)CN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880990977 CE On-Demand Mild CSNK2A1 24 40 CO[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991047 CF On-Demand Mild CSNK2A1 25 43 COCCOC1CN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991329 DD On-Demand Mild CSNK2A1 21 40 COc1cc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)ncn1 ZINC000880991347 FE On-Demand Mild PDGFRB 38 41 C[C@H](O)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991390 GF On-Demand Anodyne MPL 23 43 C[C@H](O)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991392 GF On-Demand Anodyne MPL 23 43 C[C@H](N)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991398 GF On-Demand Anodyne MPL 24 43 C[C@H](N)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991399 GF On-Demand Anodyne MPL 24 43 CC[C@H](O)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991429 GG On-Demand Anodyne MPL 17 41 CC[C@H](O)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)nn1 ZINC000880991431 GG On-Demand Anodyne MPL 17 41 CC(=O)OC1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880991450 DF On-Demand Mild CSNK2A1 27 42 CCN1CCC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991563 DF On-Demand Mild CSNK2A1 26 41 CCN1CCC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991563 DF On-Demand Mild CCR3 36 40 CCN1CCC[C@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991564 DF On-Demand Mild CSNK2A1 26 41 CCN1CCC[C@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880991564 DF On-Demand Mild CCR3 36 40 CCOc1ccnc(N2CCCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)n1 ZINC000880991568 GF On-Demand Mild P2RY12 28 41 CC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)[C@H](C)C1 ZINC000880991650 DE On-Demand Mild CSNK2A1 24 40 CC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)[C@@H](C)C1 ZINC000880991651 DE On-Demand Mild CSNK2A1 24 40 CC[C@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991712 EF On-Demand Mild CCR3 37 40 CC[C@@H]1CN(C(C)=O)CC[C@@H]1NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991713 EF On-Demand Mild CCR3 37 40 CC[C@@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991714 EF On-Demand Mild CCR3 37 40 CC[C@H]1CN(C(C)=O)CC[C@H]1NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991715 EF On-Demand Mild CCR3 37 40 COCC1(O)CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880991724 DE On-Demand Mild S1PR2 27 40 CNC(=O)[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991812 DD On-Demand Mild LGMN 77 39 COC(=O)C[C@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991826 DF On-Demand Mild LGMN 50 33 COC(=O)C[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991827 DF On-Demand Mild LGMN 50 33 CC[C@@H]1COCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880991936 CF On-Demand Mild CSNK2A1 18 40 CCn1nc2c(cc1=O)CN(C(=O)Nc1cc(C#N)c(F)cc1C)CC2 ZINC000880991968 FE On-Demand Mild P2RY14 44 36 CN(Cc1cn(CC(=O)NNC(=O)c2ccc(F)cc2)nn1)C1CCCCC1 ZINC000880991973 GD On-Demand Reactive SCARB1 30 41 Cc1cccc(C(=O)NNC(=O)Cn2cc(CN3CCCC3)nn2)c1 ZINC000880991992 EC On-Demand Reactive KCNK3 48 36 CCC1(O)CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880992022 DF On-Demand Mild S1PR2 27 41 CN1CCCC[C@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992087 DE On-Demand Anodyne HDAC10 15 40 CN1CCCC[C@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992087 DE On-Demand Anodyne HDAC3 21 40 CN1CCCC[C@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992087 DE On-Demand Anodyne HDAC6 17 40 CN1CCCC[C@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992087 DE On-Demand Anodyne ACKR3 43 31 CN1CCCC[C@@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992088 DE On-Demand Anodyne HDAC10 15 40 CN1CCCC[C@@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992088 DE On-Demand Anodyne HDAC3 21 40 CN1CCCC[C@@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992088 DE On-Demand Anodyne HDAC6 17 40 CN1CCCC[C@@H]1CCC(=O)Nc1cccc(-n2nccn2)c1 ZINC000880992088 DE On-Demand Anodyne ACKR3 43 31 CC[C@@H](C#N)Oc1cccc(CNC(=O)Nc2cc(C#N)c(F)cc2C)c1 ZINC000880992299 FI On-Demand Mild ROCK2 18 43 CC[C@H](C#N)Oc1cccc(CNC(=O)Nc2cc(C#N)c(F)cc2C)c1 ZINC000880992300 FI On-Demand Mild ROCK2 18 43 CC(=O)N(Cc1ccc(NC(=O)Nc2cc(C#N)c(F)cc2C)cc1)C1CC1 ZINC000880992345 GI On-Demand Mild CSNK2A1 51 38 Cc1ncc2c(n1)CCC[C@H]2NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880992393 EG On-Demand Mild CSNK2A1 27 41 CC[C@@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880992525 CE On-Demand Mild ADRB1 42 35 CC[C@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880992526 CE On-Demand Mild ADRB1 42 35 COCCC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880992546 FE On-Demand Mild EPHX2 35 41 COCCC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880992546 FE On-Demand Mild CCR8 51 35 CC(=O)NC[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880992661 EE On-Demand Mild CSNK2A1 44 42 COc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)c1 ZINC000880992675 FF On-Demand Mild P2RY12 18 41 Cc1cccc(C(=O)NNC(=O)Cn2cc(C3(F)COC3)nn2)c1 ZINC000880992682 EC On-Demand Reactive KCNK3 47 35 COC[C@@H](O)CCNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880992726 CD On-Demand Mild ADRB1 45 37 COc1cccc([C@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3C)CCO2)c1 ZINC000880992751 FH On-Demand Mild TAAR1 15 41 CC(=O)N1CCN([C@@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3C)C[C@H]2C)CC1 ZINC000880992760 GE On-Demand Mild CSNK2A1 24 40 CC(=O)N1CCN([C@@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3C)C[C@@H]2C)CC1 ZINC000880992761 GE On-Demand Mild CSNK2A1 24 40 CC(=O)N1CCN([C@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3C)C[C@H]2C)CC1 ZINC000880992762 GE On-Demand Mild CSNK2A1 24 40 CC(=O)N1CCN([C@H]2CN(C(=O)Nc3cc(C#N)c(F)cc3C)C[C@@H]2C)CC1 ZINC000880992763 GE On-Demand Mild CSNK2A1 24 40 CCC(=O)N1CC[C@@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880992791 DE On-Demand Mild EPHX2 31 45 CCC(=O)N1CC[C@H](NC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880992793 DE On-Demand Mild EPHX2 31 45 CC[C@@H](O)CCCNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993077 CF On-Demand Mild ADRB1 41 34 CC[C@H](O)CCCNC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993078 CF On-Demand Mild ADRB1 41 34 CCCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880993080 EG On-Demand Mild CCR3 36 41 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NNC(=O)c1ccc(F)cc1 ZINC000880993088 ED On-Demand Reactive SSTR3 23 41 O=C(Cn1cc([C@H]2CCCCO2)nn1)NNC(=O)c1ccc(F)cc1 ZINC000880993089 ED On-Demand Reactive SSTR3 23 41 Cc1cccc(C(=O)NNC(=O)Cn2cc(CN3CCCCC3)nn2)c1 ZINC000880993095 FD On-Demand Reactive KCNK3 48 35 CC(=O)NC[C@@H]1CN(C(=O)Nc2cc(C#N)c(F)cc2C)CCO1 ZINC000880993140 ED On-Demand Mild CSNK2A1 26 40 Cc1cccc(C(=O)NNC(=O)Cn2cc(C3CCCCC3)nn2)c1 ZINC000880993225 EE On-Demand Reactive KCNK3 50 35 Cc1ccc(N2CCC[C@@H](NC(=O)Nc3cc(C#N)c(F)cc3C)C2)nn1 ZINC000880993331 FF On-Demand Mild CSNK2A1 29 40 CCC(C)(C)c1cn(CC(=O)NNC(=O)c2ccccc2Cl)nn1 ZINC000880993333 EE On-Demand Reactive ECR 42 36 COC[C@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993347 EG On-Demand Mild MME 41 37 COC[C@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993347 EG On-Demand Mild ANPEP 45 31 COC[C@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993347 EG On-Demand Mild CTSB 43 35 COC[C@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993347 EG On-Demand Mild PAPA1_CARPA 54 38 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993348 EG On-Demand Mild MME 41 37 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993348 EG On-Demand Mild ANPEP 45 31 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993348 EG On-Demand Mild CTSB 43 35 COC[C@@H](Cc1ccccc1)NC(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993348 EG On-Demand Mild PAPA1_CARPA 54 38 Cc1cccc(C(=O)NNC(=O)Cn2cc(C(C)(C)C)nn2)c1 ZINC000880993410 DD On-Demand Reactive KCNK3 55 41 Cc1cccc(C(=O)NNC(=O)Cn2cc(C(C)(C)C)nn2)c1 ZINC000880993410 DD On-Demand Reactive KCNK9 44 38 COc1ccccc1[C@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880993428 FI On-Demand Mild RBP4 59 47 COc1ccccc1[C@@H]1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880993429 FI On-Demand Mild RBP4 59 47 Cc1cccc(C(=O)NNC(=O)Cn2cc(CN3CCN(C)CC3)nn2)c1 ZINC000880993462 FB On-Demand Reactive DRD4 42 34 Cc1cccc(C(=O)NNC(=O)Cn2cc(CN3CCN(C)CC3)nn2)c1 ZINC000880993462 FB On-Demand Reactive KCNK3 45 34 CCCO[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880993470 EH On-Demand Mild CSNK2A1 19 40 CCCO[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880993471 EH On-Demand Mild CSNK2A1 19 40 COc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)n1 ZINC000880993503 FE On-Demand Mild FAAH 22 40 CCOC(=O)N1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880993552 EF On-Demand Mild P2RY12 30 41 CCCNC(=O)[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880993593 EF On-Demand Mild GPBAR1 20 40 CCCNC(=O)[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880993594 EF On-Demand Mild GPBAR1 20 40 CC(=O)N(C)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880993633 EE On-Demand Mild CSNK2A1 32 42 Cc1cccc(C(=O)NNC(=O)Cn2cc(CCN3CCCCC3)nn2)c1 ZINC000880993708 FD On-Demand Reactive DRD4 42 33 Cc1cccc(C(=O)NNC(=O)Cn2cc(CCN3CCCCC3)nn2)c1 ZINC000880993708 FD On-Demand Reactive KCNK3 40 33 Cc1noc(C2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)n1 ZINC000880993714 EG On-Demand Mild SMO 40 49 Cc1noc(C2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)n1 ZINC000880993714 EG On-Demand Mild ETHR 57 36 CCOc1ccnc(N2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)n1 ZINC000880993855 GF On-Demand Mild P2RY12 34 43 CC[C@@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993866 CG On-Demand Mild LGMN 43 33 CC[C@H]1CCCN1C(=O)Nc1cc(C#N)c(F)cc1C ZINC000880993867 CG On-Demand Mild LGMN 43 33 Cc1cccc(C(=O)NNC(=O)Cn2cc(/C=C/C(C)C)nn2)c1 ZINC000880993891 ED On-Demand Reactive KCNK3 50 36 Cc1cccc(C(=O)NNC(=O)Cn2cc(/C=C\C(C)C)nn2)c1 ZINC000880993892 ED On-Demand Reactive KCNK3 50 36 Cc1cccc(C(=O)NNC(=O)Cn2cc(CCN(C)C)nn2)c1 ZINC000880993951 EC On-Demand Reactive KCNK3 49 37 Cc1cccc(C(=O)NNC(=O)Cn2cc(CN3CCSCC3)nn2)c1 ZINC000880993988 FC On-Demand Reactive KCNK3 42 34 CCC(C)(C)c1cn(CC(=O)NNC(=O)c2cccc(C)c2)nn1 ZINC000880994074 ED On-Demand Reactive KCNK3 52 37 CCC(C)(C)c1cn(CC(=O)NNC(=O)c2cccc(C)c2)nn1 ZINC000880994074 ED On-Demand Reactive KCNK9 42 36 CCOC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994102 EF On-Demand Mild P2RY12 19 41 CCOC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994102 EF On-Demand Mild EPHX2 44 39 CCOC(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994102 EF On-Demand Mild CCR8 40 39 C[C@H](N)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994104 FF On-Demand Anodyne ROCK1 20 43 C[C@H](N)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994105 FF On-Demand Anodyne ROCK1 20 43 CCN(CC)C(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994142 FG On-Demand Mild CSNK2A1 34 41 CCN(CC)Cc1cn(CC(=O)NNC(=O)c2cccc(C)c2)nn1 ZINC000880994166 EC On-Demand Reactive KCNK3 52 36 CCN(CC)Cc1cn(CC(=O)NNC(=O)c2cccc(C)c2)nn1 ZINC000880994166 EC On-Demand Reactive KCNK9 41 36 C[C@H](C(=O)Nc1nc(-c2ccc(F)cc2)cs1)n1cc(CC(C)(C)O)nn1 ZINC000880994182 GG On-Demand Anodyne ROCK1 20 43 COc1ccc([C@@H]2CCCN2C(=O)Nc2cc(C#N)c(F)cc2C)cc1OC ZINC000880994220 GI On-Demand Mild LGMN 43 33 C[C@H](C(=O)Nc1nc(-c2ccc(F)cc2)cs1)n1cc([C@@H](O)C2CC2)nn1 ZINC000880994227 GG On-Demand Anodyne ROCK1 18 40 C[C@H](C(=O)Nc1nc(-c2ccc(F)cc2)cs1)n1cc([C@H](O)C2CC2)nn1 ZINC000880994230 GG On-Demand Anodyne ROCK1 18 40 CCO[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994270 DG On-Demand Mild CSNK2A1 22 41 CN(C(=O)c1ccc(OC(F)F)c(Cl)c1)[C@@H]1CCCC[C@H]1O ZINC000880994303 EG On-Demand Anodyne PDE4D 15 44 COc1ccc2c(c1)CN(C(=O)Nc1cc(C#N)c(F)cc1C)CC2 ZINC000880994313 EH On-Demand Mild HDAC6 31 41 COc1ccc2c(c1)CN(C(=O)Nc1cc(C#N)c(F)cc1C)CC2 ZINC000880994313 EH On-Demand Mild AKR1C3 19 43 CCCNC(=O)c1cccc(CNC(=O)Nc2cc(C#N)c(F)cc2C)c1 ZINC000880994319 FG On-Demand Mild ROCK2 17 45 COCCn1cc(NC(=O)Nc2cc(C#N)c(F)cc2C)cn1 ZINC000880994327 DE On-Demand Mild CSNK2A1 41 35 C[C@H](C(=O)Nc1nc(-c2ccc(F)cc2)cs1)n1cc(C2(O)CCC2)nn1 ZINC000880994337 GG On-Demand Anodyne ROCK1 18 42 CCN1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994341 DE On-Demand Mild CCR3 44 40 CCN1CC[C@H](CNC(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994341 DE On-Demand Mild CACNA1I 57 34 CN(C(=O)Cc1ccccc1N1CCCC1=O)[C@@H]1CCCC[C@H]1O ZINC000880994371 EE On-Demand Anodyne OPRK1 19 43 CC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994441 DD On-Demand Mild CSNK2A1 37 43 Cc1ccc(NC(=O)N2CCC[C@H](N3CCOCC3)CC2)cc1-c1ccsc1 ZINC000880994447 GI On-Demand Anodyne L3MBTL3 42 35 Cc1ccc(NC(=O)N2CCC[C@@H](N3CCOCC3)CC2)cc1-c1ccsc1 ZINC000880994450 GI On-Demand Anodyne L3MBTL3 42 35 Cc1ccc(NC(=O)N2CCOC3(CCN(C)CC3)C2)cc1-c1ccsc1 ZINC000880994452 GI On-Demand Anodyne EPHX2 19 45 CCC(CC)C(=O)N1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994502 FH On-Demand Mild EPHX2 36 43 Cc1ccc(NC(=O)N2CCC3=C(CCC(=O)N3)C2)cc1-c1ccsc1 ZINC000880994514 FI On-Demand Anodyne P2RY14 53 34 COc1ccc(CN(C)C(=O)Nc2cc(C#N)c(F)cc2C)cc1OC ZINC000880994558 FH On-Demand Mild MT-ND1 18 43 CCOC(=O)N[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994567 EF On-Demand Mild CSNK2A1 18 40 COCCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994647 EE On-Demand Mild CCR3 35 41 COc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)cc1 ZINC000880994699 GI On-Demand Mild PRSS2 70 34 COc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)cc1 ZINC000880994699 GI On-Demand Mild CSNK2A1 24 41 COc1ccc(OC2CCN(C(=O)Nc3cc(C#N)c(F)cc3C)CC2)cc1 ZINC000880994699 GI On-Demand Mild EPHX2 23 45 CCN1CCC(NC(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994705 DF On-Demand Mild CXCR3 19 40 CCc1noc([C@]2(O)CCN(C(=O)Nc3ccc(C)c(-c4ccsc4)c3)C2)n1 ZINC000880994728 GH On-Demand Anodyne P2RY14 43 34 CCc1noc([C@@]2(O)CCN(C(=O)Nc3ccc(C)c(-c4ccsc4)c3)C2)n1 ZINC000880994729 GH On-Demand Anodyne P2RY14 43 34 C[C@H](O)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994824 FF On-Demand Anodyne ROCK1 20 44 C[C@H](O)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994826 FF On-Demand Anodyne ROCK1 20 44 CC(=O)NCC1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994828 EE On-Demand Mild CSNK2A1 33 43 CC(=O)NCC1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994828 EE On-Demand Mild CACNA1I 44 31 CCCCCNC(=O)C1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880994849 FH On-Demand Mild ASAH1 49 35 CC[C@H](O)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994879 GG On-Demand Anodyne ROCK1 20 43 CC[C@H](O)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994880 GG On-Demand Anodyne ROCK1 20 43 Cc1ncc2c(n1)CC[C@H](NC(=O)Nc1cc(C#N)c(F)cc1C)C2 ZINC000880994909 EF On-Demand Mild CSNK2A1 33 41 Cc1ncc2c(n1)CC[C@@H](NC(=O)Nc1cc(C#N)c(F)cc1C)C2 ZINC000880994910 EF On-Demand Mild CSNK2A1 33 41 C[C@H](C(=O)Nc1nc(-c2ccc(F)cc2)cs1)n1cc(C(C)(C)O)nn1 ZINC000880994926 GF On-Demand Anodyne ROCK1 19 42 CC(=O)N[C@@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994969 DE On-Demand Mild CSNK2A1 34 46 CC(=O)N[C@H]1CCCN(C(=O)Nc2cc(C#N)c(F)cc2C)C1 ZINC000880994970 DE On-Demand Mild CSNK2A1 34 46 O=C(COC1CC1)N1CCC[C@H]1c1ccc(F)c(C(F)(F)F)c1 ZINC000880994971 EH On-Demand Anodyne CPT1A 49 36 O=C(COC1CC1)N1CCC[C@@H]1c1ccc(F)c(C(F)(F)F)c1 ZINC000880994972 EH On-Demand Anodyne CPT1A 49 36 CC[C@@](C)(O)c1cn([C@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994974 GG On-Demand Anodyne ROCK1 19 43 CC[C@@](C)(O)c1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(F)cc3)cs2)nn1 ZINC000880994975 GG On-Demand Anodyne ROCK1 19 43 Cc1ccc(NC(=O)N2CCN(C)C(=O)C2)cc1-c1ccsc1 ZINC000880995034 EG On-Demand Anodyne P2RY14 49 33 COC(=O)Cc1cn([C@H](C)C(=O)Nc2nc(-c3ccc(C)cc3)cs2)nn1 ZINC000880995089 GF On-Demand Anodyne ROCK1 20 41 COC(=O)Cc1cn([C@@H](C)C(=O)Nc2nc(-c3ccc(C)cc3)cs2)nn1 ZINC000880995090 GF On-Demand Anodyne ROCK1 20 41 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880995212 FH On-Demand Anodyne EPHX2 17 44 CCC(=O)N1CCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880995229 EH On-Demand Anodyne P2RY14 46 33 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1-c1ccsc1 ZINC000880995287 GH On-Demand Anodyne L3MBTL3 46 38 Cc1ccc(NC(=O)N2CCN(C(=O)CC#N)CC2)cc1-c1ccsc1 ZINC000880995314 FG On-Demand Mild P2RY14 49 34 Cc1ccc(NC(=O)N2CCC(=O)N(C)CC2)cc1-c1ccsc1 ZINC000880995354 EG On-Demand Anodyne P2RY14 49 33 Cc1ccc(NC(=O)N2CCCNC(=O)C2)cc1-c1ccsc1 ZINC000880995449 EG On-Demand Anodyne P2RY14 55 36 Cc1nc(CN2CCN(C(=O)Nc3ccc(C)c(-c4ccsc4)c3)CC2)n[nH]1 ZINC000880995468 GG On-Demand Anodyne P2RY14 42 32 CCOC(=O)N1CCN(C(=O)Nc2cc(C#N)c(F)cc2C)CC1 ZINC000880995497 EE On-Demand Mild P2RY12 40 43 Cc1ccc(NC(=O)N2CCC3(CCCC3=O)CC2)cc1-c1ccsc1 ZINC000880995502 FK On-Demand Anodyne P2RY14 45 32 Cc1ccc(NC(=O)N2CCC(CO)(CO)C2)cc1-c1ccsc1 ZINC000880995518 EF On-Demand Anodyne P2RY14 45 34 Cc1ccc(NC(=O)N2CCCc3n[nH]cc3C2)cc1-c1ccsc1 ZINC000880995519 FI On-Demand Anodyne P2RY14 55 35 Cc1ccc(NC(=O)N2CCCN(C=O)CC2)cc1-c1ccsc1 ZINC000880995539 EG On-Demand Anodyne P2RY14 40 32 Cc1ccc(NC(=O)N2CC[C@@H](C(=O)N3CCCC3)C2)cc1-c1ccsc1 ZINC000880995547 GI On-Demand Anodyne P2RY14 51 33 COC(=O)Cc1cn(CCOc2ccc(F)cc2)nn1 ZINC000880995553 CD On-Demand Anodyne MMP13 23 43 Cc1ccc(NC(=O)N2CCC[C@H](CO)CC2)cc1-c1ccsc1 ZINC000880995567 EI On-Demand Anodyne P2RY14 42 33 Cc1ccc(NC(=O)N2CCC[C@@H](CO)CC2)cc1-c1ccsc1 ZINC000880995568 EI On-Demand Anodyne P2RY14 42 33 COC(=O)[C@@H]1CCCN(Cc2cn(Cc3cc(F)cc(C(C)=O)c3O)nn2)C1 ZINC000880995596 GD On-Demand Clean SLC6A1 48 35 CCC1(O)CN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880995617 DH On-Demand Anodyne P2RY14 45 32 CC(C)(C)OC(=O)NCc1cn(CCOc2ccc(F)cc2)nn1 ZINC000880995743 EF On-Demand Anodyne MMP13 22 43 Cc1ccc(NC(=O)N2CCO[C@@]3(CCCOC3)C2)cc1-c1ccsc1 ZINC000880995746 FI On-Demand Anodyne EPHX2 19 40 Cc1ccc(NC(=O)N2CCO[C@]3(CCCOC3)C2)cc1-c1ccsc1 ZINC000880995747 FI On-Demand Anodyne EPHX2 19 40 O=S1(=O)CCN(Cc2cn(CCOc3ccc(Cl)cc3)nn2)CC1 ZINC000880995753 FD On-Demand Anodyne LTA4H 19 42 Cc1ccc(NC(=O)N2CCCc3c(cnn3C)C2)cc1-c1ccsc1 ZINC000880996012 FI On-Demand Anodyne P2RY14 56 36 CC(=O)N1CCN(Cc2cn(CCOc3ccc(Cl)cc3)nn2)CC1 ZINC000880996017 FD On-Demand Anodyne LTA4H 25 40 CC(=O)N1CCN(Cc2cn(CCOc3ccc(Cl)cc3)nn2)CC1 ZINC000880996017 FD On-Demand Anodyne HRH3 29 41 O=C(N[C@H]1COC[C@H]1O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880996183 FD On-Demand Anodyne OPRD1 53 34 O=C(N[C@H]1COC[C@H]1O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880996183 FD On-Demand Anodyne CFTR 79 47 O=C(N[C@H]1COC[C@H]1O)[C@@H]1Cc2ccccc2CN1C(=O)c1ccccc1 ZINC000880996183 FD On-Demand Anodyne ADAM9 42 34 C[C@H](O)c1ccccc1OCc1cn(CCOc2ccc(F)cc2)nn1 ZINC000880996207 FG On-Demand Anodyne MMP13 24 43 C[C@H](O)c1ccccc1OCc1cn(CCOc2ccc(F)cc2)nn1 ZINC000880996207 FG On-Demand Anodyne MMP8 36 42 CC(=O)N1CCN(Cc2cn(CCOc3cccc(C)c3)nn2)CC1 ZINC000880996250 ED On-Demand Anodyne DRD4 40 33 Cc1ccc(NC(=O)N2CCCC[C@H]2c2nc[nH]n2)cc1-c1ccsc1 ZINC000880996377 FJ On-Demand Anodyne CPT1A 55 38 Cc1ccc(NC(=O)N2CCCC[C@@H]2c2nc[nH]n2)cc1-c1ccsc1 ZINC000880996378 FJ On-Demand Anodyne CPT1A 55 38 COC[C@]1(CO)CCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880996419 FH On-Demand Anodyne EPHX2 17 40 C[C@H](O)c1ccc(OCc2cn(CCOc3ccc(F)cc3)nn2)cc1 ZINC000880996426 FG On-Demand Anodyne MMP13 24 44 O=C(N[C@H]1COC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880996456 CC On-Demand Anodyne GABRA1 19 44 O=C(N[C@H]1COC[C@H]1O)C(=O)c1c[nH]c2cc(F)ccc12 ZINC000880996456 CC On-Demand Anodyne GABRA2 17 44 O=C(N[C@H]1COC[C@H]1O)c1ccc(OC(F)F)c(Cl)c1 ZINC000880996474 DD On-Demand Anodyne PDE4D 20 43 COC[C@@H](O)CCNC(=O)Nc1ccc(C)c(-c2ccsc2)c1 ZINC000880996500 EG On-Demand Anodyne ADRB1 40 30 COCCn1nnc2c1CCN(C(=O)Nc1ccc(C)c(-c3ccsc3)c1)C2 ZINC000880996548 GH On-Demand Anodyne P2RY14 55 35 Cc1ccc(NC(=O)N2CCN(CC(N)=O)C(=O)C2)cc1-c1ccsc1 ZINC000880996607 FD On-Demand Anodyne P2RY14 46 32 O[C@@]1(c2cn(CCOc3ccc(Cl)cc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880996620 EG On-Demand Anodyne ALOX5AP 32 43 O[C@]1(c2cn(CCOc3ccc(Cl)cc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880996621 EG On-Demand Anodyne ALOX5AP 32 43 Cc1ccc(NC(=O)N2CCOC3(CCC3)C2)cc1-c1ccsc1 ZINC000880996723 EJ On-Demand Anodyne EPHX2 21 44 Cc1ccc(NC(=O)N2CCN(C(=O)CO)CC2)cc1-c1ccsc1 ZINC000880996732 FE On-Demand Anodyne P2RY14 42 34 Cc1ccc(NC(=O)N(C)CCCn2ccnc2)cc1-c1ccsc1 ZINC000880996754 FI On-Demand Anodyne QPCT 39 41 O=C(Cc1ccccc1N1CCCC1=O)N[C@H]1COC[C@H]1O ZINC000880996860 DC On-Demand Anodyne KCNQ2 44 39 Cc1ccc(NC(=O)N(CCC#N)CCN2CCOCC2)cc1-c1ccsc1 ZINC000880996883 GH On-Demand Mild CASR 61 46 Cc1ccc(NC(=O)N2CCOC3(CCOCC3)C2)cc1-c1ccsc1 ZINC000880996928 FI On-Demand Anodyne EPHX2 19 44 CC[C@H]1CN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C[C@@H]1O ZINC000880996944 EH On-Demand Anodyne P2RY14 46 33 CC[C@H]1CN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)C[C@H]1O ZINC000880996945 EH On-Demand Anodyne P2RY14 46 33 CCC(=O)N1CC[C@H](NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880996959 FH On-Demand Anodyne EPHX2 36 52 CCC(=O)N1CC[C@@H](NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)C1 ZINC000880996960 FH On-Demand Anodyne EPHX2 36 52 O=C(N[C@H]1COC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880996975 FC On-Demand Anodyne PREP 25 42 O=C(N[C@H]1COC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880996975 FC On-Demand Anodyne KLK5 41 40 O=C(N[C@H]1COC[C@H]1O)[C@H]1C[C@@H](F)CN1C(=O)OCc1ccccc1 ZINC000880996975 FC On-Demand Anodyne Q9NAW4_PLAFA 41 48 Cc1ccc(NC(=O)N(CCCCO)C2CC2)cc1-c1ccsc1 ZINC000880996989 EI On-Demand Anodyne MCHR1 15 40 Cc1ccc(NC(=O)N(CCCO)C2CC2)cc1-c1ccsc1 ZINC000880997001 EI On-Demand Anodyne MCHR1 17 40 Cc1ccc(NC(=O)N2CCCN(C)CC2)cc1-c1ccsc1 ZINC000880997011 EH On-Demand Anodyne P2RY14 42 32 Cc1ccc(NC(=O)N2CCC(NC(=O)C3CC3)CC2)cc1-c1ccsc1 ZINC000880997094 GI On-Demand Anodyne MAPK14 15 42 COc1ccc(OCCn2cc(CNC(=O)OC(C)(C)C)nn2)cc1 ZINC000880997096 EE On-Demand Anodyne PROKR1 41 30 COC[C@@H](O)CNC(=O)Nc1ccc(C)c(-c2ccsc2)c1 ZINC000880997098 DF On-Demand Anodyne ADRB1 43 33 Fc1ccc(OCCn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880997138 FG On-Demand Anodyne HRH3 17 47 Fc1ccc(OCCn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880997138 FG On-Demand Anodyne MMP13 16 51 Fc1ccc(OCCn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880997138 FG On-Demand Anodyne MMP8 19 51 O=C(N[C@H]1COC[C@H]1O)c1ccc(OC(F)F)c(Br)c1 ZINC000880997143 FD On-Demand Anodyne PDE4D 17 42 CCn1nc2c(cc1=O)CN(C(=O)Nc1ccc(C)c(-c3ccsc3)c1)CC2 ZINC000880997144 GH On-Demand Anodyne P2RY14 63 41 CC(=O)N1CCN(Cc2cn(CCOc3cccc(Cl)c3)nn2)CC1 ZINC000880997180 FD On-Demand Anodyne DRD4 42 34 CC(=O)N1CCN(Cc2cn(CCOc3cccc(Cl)c3)nn2)CC1 ZINC000880997180 FD On-Demand Anodyne HRH3 17 41 CC(=O)N1CCN(Cc2cn(CCOc3cccc(Cl)c3)nn2)CC1 ZINC000880997180 FD On-Demand Anodyne FAAH 27 41 NOCc1cn(CCOc2cccc(Br)c2)nn1 ZINC000880997185 DD On-Demand Anodyne HMOX2 20 44 COc1ccc(OCCn2cc(C3(O)CCCCC3)nn2)cc1 ZINC000880997194 DF On-Demand Anodyne LTA4H 19 40 Cc1ccc(NC(=O)N2CCC3(CCOCC3)C2)cc1-c1ccsc1 ZINC000880997236 FJ On-Demand Anodyne EPHX2 31 40 COc1ccc(OCCn2cc(COc3ccccc3[C@H](C)O)nn2)cc1 ZINC000880997241 FF On-Demand Anodyne MMP13 24 42 COc1ccc(OCCn2cc(COc3ccccc3[C@H](C)O)nn2)cc1 ZINC000880997241 FF On-Demand Anodyne MMP8 39 40 COc1ccc(OCCn2cc(COc3ccccc3[C@H](C)O)nn2)cc1 ZINC000880997241 FF On-Demand Anodyne MMP9 19 40 COc1ccc(OCCn2cc(COc3ccccc3[C@@H](C)O)nn2)cc1 ZINC000880997243 FF On-Demand Anodyne MMP13 24 42 COc1ccc(OCCn2cc(COc3ccccc3[C@@H](C)O)nn2)cc1 ZINC000880997243 FF On-Demand Anodyne MMP8 39 40 COc1ccc(OCCn2cc(COc3ccccc3[C@@H](C)O)nn2)cc1 ZINC000880997243 FF On-Demand Anodyne MMP9 19 40 CCC1(O)CCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880997250 EI On-Demand Anodyne P2RY14 40 32 Brc1cccc(OCCn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880997261 GE On-Demand Anodyne HRH3 18 44 Brc1cccc(OCCn2cc(CCCN3CCOCC3)nn2)c1 ZINC000880997261 GE On-Demand Anodyne HMOX2 19 40 COc1ccc(OCCn2cc(CN3CCS(=O)(=O)CC3)nn2)cc1 ZINC000880997268 FC On-Demand Anodyne LTA4H 23 41 O=[N+]([O-])c1ccccc1Cn1cc(C2(O)CCC2)nn1 ZINC000880997289 CD On-Demand Bother COLA 45 33 Cc1ccc(NC(=O)N2CCC[C@@](C)(O)C2)cc1-c1ccsc1 ZINC000880997290 EI On-Demand Anodyne EPHX2 19 43 Cc1ccc(NC(=O)N2CCC[C@](C)(O)C2)cc1-c1ccsc1 ZINC000880997291 EI On-Demand Anodyne EPHX2 19 43 Cc1ccc(NC(=O)N(CCO)CCN2CCOCC2)cc1-c1ccsc1 ZINC000880997311 GF On-Demand Anodyne CASR 64 49 Cc1ccc(NC(=O)N(CCO)CCN2CCOCC2)cc1-c1ccsc1 ZINC000880997311 GF On-Demand Anodyne PRKDC 43 34 Cc1ccc(NC(=O)N(CCO)CCN2CCOCC2)cc1-c1ccsc1 ZINC000880997311 GF On-Demand Anodyne PIK3CA 16 40 Cc1ccc(NC(=O)N2CC(C)C2)cc1-c1ccsc1 ZINC000880997343 CI On-Demand Anodyne P2RY14 42 33 COc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880997344 ED On-Demand Anodyne DRD3 18 42 COc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880997344 ED On-Demand Anodyne LTA4H 35 44 COc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880997344 ED On-Demand Anodyne HRH3 62 47 COc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880997344 ED On-Demand Anodyne SIGMAR1 17 53 COc1ccc(OCCn2cc(C3(O)CCC3)nn2)cc1 ZINC000880997395 CD On-Demand Anodyne LTA4H 19 41 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne LTA4H 46 36 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne KLK3 57 32 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CTSB 46 43 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne PAPA1_CARPA 44 33 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CYSP_TRYCR 42 41 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CTSK 32 44 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CAPNS1 54 34 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne MMP2 15 40 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CTSS 15 42 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne GHSR 40 39 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CAPN1 70 40 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne MMP9 22 40 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne CAPN2 113 43 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne TPSAB1 36 41 COc1ccc(OCCn2cc(CNC(=O)OCc3ccccc3)nn2)cc1 ZINC000880997397 GF On-Demand Anodyne NPR 63 35 Cc1ccc(NC(=O)N2CCOC3(CCOCC3)CC2)cc1-c1ccsc1 ZINC000880997460 GJ On-Demand Anodyne EPHX2 15 40 O=[N+]([O-])c1ccccc1Cn1cc([C@H](O)C2CC2)nn1 ZINC000880997505 CD On-Demand Bother COLA 42 31 O=[N+]([O-])c1ccccc1Cn1cc([C@@H](O)C2CC2)nn1 ZINC000880997506 CD On-Demand Bother COLA 42 31 Cc1ccc(NC(=O)N2CCC(Cc3nccs3)CC2)cc1N1CCCC1 ZINC000880997539 GJ On-Demand Anodyne HTR1B 18 41 Cc1ccc(NC(=O)N2CCC[C@@H](CF)C2)cc1N1CCCC1 ZINC000880997543 DH On-Demand Anodyne HTR1B 17 43 Cc1ccc(NC(=O)N2CCC[C@@H](CF)C2)cc1N1CCCC1 ZINC000880997543 DH On-Demand Anodyne KCNQ2 48 31 Cc1ccc(NC(=O)N2CCC[C@@H](CF)C2)cc1N1CCCC1 ZINC000880997543 DH On-Demand Anodyne NPY2R 52 35 Cc1ccc(NC(=O)N2CCC[C@@H](CF)C2)cc1N1CCCC1 ZINC000880997543 DH On-Demand Anodyne EPHX2 22 48 Cc1ccc(NC(=O)N2CCC[C@H](CF)C2)cc1N1CCCC1 ZINC000880997544 DH On-Demand Anodyne HTR1B 17 43 Cc1ccc(NC(=O)N2CCC[C@H](CF)C2)cc1N1CCCC1 ZINC000880997544 DH On-Demand Anodyne KCNQ2 48 31 Cc1ccc(NC(=O)N2CCC[C@H](CF)C2)cc1N1CCCC1 ZINC000880997544 DH On-Demand Anodyne NPY2R 52 35 Cc1ccc(NC(=O)N2CCC[C@H](CF)C2)cc1N1CCCC1 ZINC000880997544 DH On-Demand Anodyne EPHX2 22 48 COCC(C)(C)CCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997545 EH On-Demand Anodyne NPY2R 41 34 COCC(C)(C)CCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997545 EH On-Demand Anodyne EPHX2 16 43 Cc1ccc(NC(=O)N2CCN(C)c3ncccc3C2)cc1N1CCCC1 ZINC000880997552 FG On-Demand Anodyne HTR1D 15 46 Cc1ccc(NC(=O)N2CCN(C)c3ncccc3C2)cc1N1CCCC1 ZINC000880997552 FG On-Demand Anodyne HTR1B 19 46 Cc1ccc(NC(=O)N2CCN(C)c3ncccc3C2)cc1N1CCCC1 ZINC000880997552 FG On-Demand Anodyne PDGFRB 41 36 Cc1ccc(NC(=O)N2CCN(C)c3ncccc3C2)cc1N1CCCC1 ZINC000880997552 FG On-Demand Anodyne TRPV1 20 48 Cc1ccc(NC(=O)N2CCC(C(=O)NCCO)CC2)cc1N1CCCC1 ZINC000880997555 FD On-Demand Anodyne EPHX2 44 40 COC(=O)[C@@]1(O)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880997560 ED On-Demand Anodyne EPHX2 33 40 CSCC[C@H](NC(=O)Nc1ccc(C)c(N2CCCC2)c1)C(N)=O ZINC000880997564 FE On-Demand Anodyne FPR1 38 40 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne HTR1D 15 48 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne HTR1B 21 48 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne KCNQ2 70 36 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne NPY2R 69 38 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne RBP4 54 34 Cc1ccc(NC(=O)N2CC(c3ccccc3)C2)cc1N1CCCC1 ZINC000880997574 EI On-Demand Anodyne MCHR1 16 43 O=C(Cn1cc(CC2(O)CCOCC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880997576 FD On-Demand Anodyne HSD11B1 20 41 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne HTR1D 17 46 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne HTR1B 20 46 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne KCNQ2 57 33 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne TRPV1 15 44 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne NPY2R 54 36 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne CCR2 15 43 Cc1ccc(NC(=O)N2CCC(CCF)CC2)cc1N1CCCC1 ZINC000880997577 EI On-Demand Anodyne EPHX2 45 47 Cc1ccc(NC(=O)N2CC(=O)N(C)c3ccccc3C2)cc1N1CCCC1 ZINC000880997579 GH On-Demand Anodyne HTR1D 16 50 Cc1ccc(NC(=O)N2CC(=O)N(C)c3ccccc3C2)cc1N1CCCC1 ZINC000880997579 GH On-Demand Anodyne HTR1B 22 50 Cc1ccc(NC(=O)N2CC(=O)N(C)c3ccccc3C2)cc1N1CCCC1 ZINC000880997579 GH On-Demand Anodyne KCNQ2 67 33 Cc1ccc(NC(=O)N2CCC(NC3CCOCC3)CC2)cc1N1CCCC1 ZINC000880997584 GG On-Demand Anodyne HTR1B 15 42 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880997586 GF On-Demand Anodyne HTR1D 21 52 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880997586 GF On-Demand Anodyne HTR1B 26 52 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880997586 GF On-Demand Anodyne NPY2R 26 42 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880997586 GF On-Demand Anodyne SCD1 16 40 Cc1ccc(NC(=O)N2CCC(N3CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880997586 GF On-Demand Anodyne L3MBTL3 105 45 Cc1ccc(NC(=O)N2CCN(C)[C@@H](C(C)C)C2)cc1N1CCCC1 ZINC000880997606 EG On-Demand Anodyne HTR1B 16 46 Cc1ccc(NC(=O)N2CCS(=O)(=O)[C@@H](C)C2)cc1N1CCCC1 ZINC000880997610 FE On-Demand Anodyne HTR1B 17 46 Cc1ccc(NC(=O)N2CCS(=O)(=O)[C@@H](C)C2)cc1N1CCCC1 ZINC000880997610 FE On-Demand Anodyne KCNQ2 50 31 Cc1ccc(NC(=O)N2CCS(=O)(=O)[C@H](C)C2)cc1N1CCCC1 ZINC000880997611 FE On-Demand Anodyne HTR1B 17 46 Cc1ccc(NC(=O)N2CCS(=O)(=O)[C@H](C)C2)cc1N1CCCC1 ZINC000880997611 FE On-Demand Anodyne KCNQ2 50 31 O=C(Cn1cc([C@H](O)C2CC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880997614 ED On-Demand Anodyne HSD11B1 41 32 O=C(Cn1cc([C@@H](O)C2CC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880997615 ED On-Demand Anodyne HSD11B1 41 32 CC(=O)Nc1ccc2c(c1)CN(C(=O)Nc1ccc(C)c(N3CCCC3)c1)CC2 ZINC000880997618 GI On-Demand Anodyne P2RY14 44 32 CC(=O)C1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880997631 EG On-Demand Anodyne HTR1B 15 47 CC(=O)C1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880997631 EG On-Demand Anodyne NPY2R 40 35 CC(=O)C1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880997631 EG On-Demand Anodyne EPHX2 36 41 COc1ccc(OCCn2cc(COc3ccc([C@H](C)O)cc3)nn2)cc1 ZINC000880997661 FF On-Demand Anodyne MMP13 24 41 COc1ccc(OCCn2cc(COc3ccc([C@H](C)O)cc3)nn2)cc1 ZINC000880997661 FF On-Demand Anodyne MMP8 38 41 COc1ccc(OCCn2cc(COc3ccc([C@H](C)O)cc3)nn2)cc1 ZINC000880997661 FF On-Demand Anodyne MMP9 20 41 COc1ccc(OCCn2cc(COc3ccc([C@@H](C)O)cc3)nn2)cc1 ZINC000880997662 FF On-Demand Anodyne MMP13 24 41 COc1ccc(OCCn2cc(COc3ccc([C@@H](C)O)cc3)nn2)cc1 ZINC000880997662 FF On-Demand Anodyne MMP8 38 41 COc1ccc(OCCn2cc(COc3ccc([C@@H](C)O)cc3)nn2)cc1 ZINC000880997662 FF On-Demand Anodyne MMP9 20 41 O=C(NCc1cn(CCOc2cccc(Cl)c2)nn1)OCC(F)(F)F ZINC000880997669 GF On-Demand Anodyne PDS 64 41 COc1ccc(OCCn2cc([C@]3(O)C[C@H]4CC[C@H]3C4)nn2)cc1 ZINC000880997678 EE On-Demand Anodyne ALOX5AP 35 41 COc1ccc(OCCn2cc([C@@]3(O)C[C@H]4CC[C@H]3C4)nn2)cc1 ZINC000880997679 EE On-Demand Anodyne ALOX5AP 35 41 OC1(c2cn(CCOc3cccc(Br)c3)nn2)CCC1 ZINC000880997687 EE On-Demand Anodyne HMOX2 19 41 COc1ccc(OCCn2cc(COc3cccc(C(C)=O)c3)nn2)cc1 ZINC000880997689 FG On-Demand Anodyne DRD4 40 30 COCC1=CCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880997712 EJ On-Demand Anodyne P2RY14 51 34 CC(=O)N1CCN(Cc2cn(CCOc3ccc(F)cc3)nn2)CC1 ZINC000880997729 ED On-Demand Anodyne LTA4H 23 40 CC(=O)N1CCN(Cc2cn(CCOc3ccc(F)cc3)nn2)CC1 ZINC000880997729 ED On-Demand Anodyne MMP13 22 42 COC(=O)C1CCC(c2cn(CC(=O)NCc3cccc(OC)c3)nn2)CC1 ZINC000880997750 GE On-Demand Anodyne MTNR1A 45 39 COC(=O)C1CCC(c2cn(CC(=O)NCc3cccc(OC)c3)nn2)CC1 ZINC000880997750 GE On-Demand Anodyne MTNR1B 43 39 COC(=O)C1CCC(c2cn(CC(=O)NCc3cccc(OC)c3)nn2)CC1 ZINC000880997750 GE On-Demand Anodyne ROCK2 42 39 O=C(Cn1cc(C2(O)CCOCC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880997762 FD On-Demand Anodyne HSD11B1 28 40 COC(=O)C[C@H](O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997766 ED On-Demand Anodyne KCNQ2 49 32 COC(=O)C[C@@H](O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997767 ED On-Demand Anodyne KCNQ2 49 32 COC(=O)C1CCN(C(=O)Cn2cc(-c3ccc(Cl)cc3F)nn2)CC1 ZINC000880997771 GE On-Demand Anodyne IL2RA 55 36 COC(=O)C1CCN(C(=O)Cn2cc(-c3ccc(Cl)cc3F)nn2)CC1 ZINC000880997771 GE On-Demand Anodyne PTR1 44 31 Cc1ccc(NC(=O)N2CCCN(C(=O)CC(C)C)CC2)cc1N1CCCC1 ZINC000880997775 GH On-Demand Anodyne KCNQ2 57 32 CO[C@@H]1CC[C@@H](C)N(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880997781 EH On-Demand Anodyne HTR1B 16 42 C/C=C\CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997784 CG On-Demand Anodyne KCNQ2 57 33 C/C=C\CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997784 CG On-Demand Anodyne EPHX2 18 42 C/C=C/CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997785 CG On-Demand Anodyne KCNQ2 57 33 C/C=C/CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880997785 CG On-Demand Anodyne EPHX2 18 42 Cc1ccc(NC(=O)N2CC=C[C@H]2CO)cc1N1CCCC1 ZINC000880997790 DE On-Demand Anodyne KCNQ2 65 32 Cc1ccc(NC(=O)N2CC=C[C@@H]2CO)cc1N1CCCC1 ZINC000880997791 DE On-Demand Anodyne KCNQ2 65 32 Cc1ccc(NC(=O)N2CCC3(CC2)COCCO3)cc1N1CCCC1 ZINC000880997796 FG On-Demand Anodyne EPHX2 22 40 Cc1ccc(NC(=O)N2CCC3(CC2)COCCO3)cc1N1CCCC1 ZINC000880997796 FG On-Demand Anodyne TRPM8 30 41 CC(=O)[C@H]1CCCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880997807 EG On-Demand Anodyne EPHX2 17 43 CC(=O)[C@@H]1CCCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880997808 EG On-Demand Anodyne EPHX2 17 43 Cc1ccc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)cc1N1CCCC1 ZINC000880997828 FF On-Demand Anodyne KCNQ2 41 31 Cc1ccc(NC(=O)N2CCC([C@H](F)C(N)=O)CC2)cc1N1CCCC1 ZINC000880997828 FF On-Demand Anodyne NPY2R 42 34 Cc1ccc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)cc1N1CCCC1 ZINC000880997829 FF On-Demand Anodyne KCNQ2 41 31 Cc1ccc(NC(=O)N2CCC([C@@H](F)C(N)=O)CC2)cc1N1CCCC1 ZINC000880997829 FF On-Demand Anodyne NPY2R 42 34 COC[C@@H](O)Cc1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880997833 EC On-Demand Anodyne ROCK2 42 39 Cc1ccc(NC(=O)N2CCC(C)(N3CCC3)CC2)cc1N1CCCC1 ZINC000880997838 FH On-Demand Anodyne CCR5 21 42 Cc1ccc(NC(=O)N2CCC([C@H](C)O)CC2)cc1N1CCCC1 ZINC000880997847 EG On-Demand Anodyne HTR1B 17 44 Cc1ccc(NC(=O)N2CCC([C@H](C)O)CC2)cc1N1CCCC1 ZINC000880997847 EG On-Demand Anodyne KCNQ2 51 34 Cc1ccc(NC(=O)N2CCC([C@H](C)O)CC2)cc1N1CCCC1 ZINC000880997847 EG On-Demand Anodyne NPY2R 59 36 Cc1ccc(NC(=O)N2CCC([C@@H](C)O)CC2)cc1N1CCCC1 ZINC000880997848 EG On-Demand Anodyne HTR1B 17 44 Cc1ccc(NC(=O)N2CCC([C@@H](C)O)CC2)cc1N1CCCC1 ZINC000880997848 EG On-Demand Anodyne KCNQ2 51 34 Cc1ccc(NC(=O)N2CCC([C@@H](C)O)CC2)cc1N1CCCC1 ZINC000880997848 EG On-Demand Anodyne NPY2R 59 36 Cc1ccc(NC(=O)N2CCO[C@@]3(CCOC3)C2)cc1-c1ccsc1 ZINC000880997956 FH On-Demand Anodyne EPHX2 17 41 Cc1ccc(NC(=O)N2CCO[C@]3(CCOC3)C2)cc1-c1ccsc1 ZINC000880997957 FH On-Demand Anodyne EPHX2 17 41 OC1(c2cn(CCOc3ccc(F)cc3)nn2)CCC1 ZINC000880997960 CD On-Demand Anodyne LTA4H 15 42 COC(=O)Cc1cn(CCOc2ccc(OC)cc2)nn1 ZINC000880998008 CD On-Demand Anodyne MMP13 23 41 COC(=O)Cc1cn(CCOc2ccc(OC)cc2)nn1 ZINC000880998008 CD On-Demand Anodyne MMP8 37 41 COC(=O)Cc1cn(CCOc2ccc(OC)cc2)nn1 ZINC000880998008 CD On-Demand Anodyne MMP9 19 41 COc1ccc(OCCn2cc([C@@H](O)Cc3ccccc3)nn2)cc1 ZINC000880998011 EF On-Demand Anodyne LTA4H 45 38 COc1ccc(OCCn2cc([C@H](O)Cc3ccccc3)nn2)cc1 ZINC000880998012 EF On-Demand Anodyne LTA4H 45 38 COC(=O)C1=NO[C@@]2(CCN(C(=O)Nc3ccc(C)c(N4CCCC4)c3)C2)C1 ZINC000880998033 GF On-Demand Anodyne EPHX2 31 40 O=S1(=O)CCN(Cc2cn(CCOc3ccc(F)cc3)nn2)CC1 ZINC000880998034 FC On-Demand Anodyne LTA4H 19 42 COC(=O)C1=NO[C@]2(CCN(C(=O)Nc3ccc(C)c(N4CCCC4)c3)C2)C1 ZINC000880998035 GF On-Demand Anodyne EPHX2 31 40 Cc1ccc(NC(=O)N2CCC(C)(CO)CC2)cc1-c1ccsc1 ZINC000880998040 EI On-Demand Anodyne P2RY14 43 34 CONC(=O)C1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880998048 FF On-Demand Anodyne HTR1B 15 48 CONC(=O)C1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880998048 FF On-Demand Anodyne EPHX2 37 42 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne HTR1A 16 43 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne HTR1D 19 41 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne HTR1B 29 43 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne HTR2A 20 41 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne DRD3 15 41 Cc1ccc(NC(=O)N2CCN(CCc3cnccn3)CC2)cc1N1CCCC1 ZINC000880998050 GF On-Demand Anodyne PDGFRB 44 36 Brc1cccc(OCCn2cc([C@@H]3CCCCO3)nn2)c1 ZINC000880998062 FG On-Demand Anodyne HMOX2 19 40 Brc1cccc(OCCn2cc([C@H]3CCCCO3)nn2)c1 ZINC000880998065 FG On-Demand Anodyne HMOX2 19 40 Cc1ccc(NC(=O)N2CC3(CCCO3)C2)cc1N1CCCC1 ZINC000880998072 DF On-Demand Anodyne EPHX2 30 45 COCC1CC(NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998082 DG On-Demand Anodyne KCNQ2 41 32 COCC1CC(NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998082 DG On-Demand Anodyne EPHX2 43 46 O=C(Cn1cc(-c2cnc(Cl)nc2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998089 FE On-Demand Anodyne HSD11B1 15 43 O=C(Cn1cc(C2(O)CCC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998094 ED On-Demand Anodyne HSD11B1 45 36 O=C(NCc1cn(CCOc2cccc(Br)c2)nn1)C(F)(F)F ZINC000880998099 GE On-Demand Anodyne HMOX2 19 40 COC(=O)C1CCN(C(=O)Cn2cc(C[C@H](O)c3ccccc3)nn2)CC1 ZINC000880998116 FC On-Demand Anodyne PTR1 44 31 COC(=O)C1CCN(C(=O)Cn2cc(C[C@@H](O)c3ccccc3)nn2)CC1 ZINC000880998117 FC On-Demand Anodyne PTR1 44 31 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998121 GG On-Demand Anodyne HTR1D 16 43 COCCN(CC1CCN(C)CC1)C(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998121 GG On-Demand Anodyne HTR1B 20 43 C[C@H](N)c1cn(CC(=O)NC2C3CC4CC(C3)CC2C4)nn1 ZINC000880998126 DD On-Demand Anodyne HSD11B1 40 35 Cc1ccc(NC(=O)N2CCC(OC[C@@H]3CCCO3)CC2)cc1N1CCCC1 ZINC000880998133 GH On-Demand Anodyne HTR1B 16 41 Cc1ccc(NC(=O)N2CCC(OC[C@H]3CCCO3)CC2)cc1N1CCCC1 ZINC000880998134 GH On-Demand Anodyne HTR1B 16 41 Cc1ccc(NC(=O)N2CCCC(F)(F)CC2)cc1N1CCCC1 ZINC000880998135 EI On-Demand Anodyne HTR1B 15 44 CNS(=O)(=O)CCCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998137 FD On-Demand Anodyne HRH2 21 40 CNS(=O)(=O)CCCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998137 FD On-Demand Anodyne KCNQ2 55 32 CNS(=O)(=O)CCCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998137 FD On-Demand Anodyne EPHX2 31 45 Cc1ccc(NC(=O)N(C)CC2(C)COC2)cc1N1CCCC1 ZINC000880998138 DG On-Demand Anodyne KCNQ2 62 32 O=C(Cn1cc(CNC(=O)C(F)(F)F)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998142 GD On-Demand Anodyne HSD11B1 19 42 CCn1ncc(NC(=O)Nc2ccc(C)c(N3CCCC3)c2)c1C ZINC000880998185 EH On-Demand Anodyne KCNQ2 68 36 Cc1ccc(NC(=O)N2CCC[C@H](C(F)(F)F)C2)cc1N1CCCC1 ZINC000880998202 FI On-Demand Anodyne EPHX2 31 47 Cc1ccc(NC(=O)N2CCC[C@H](C(F)(F)F)C2)cc1N1CCCC1 ZINC000880998202 FI On-Demand Anodyne TAAR1 23 41 Cc1ccc(NC(=O)N2CCC[C@@H](C(F)(F)F)C2)cc1N1CCCC1 ZINC000880998203 FI On-Demand Anodyne EPHX2 31 47 Cc1ccc(NC(=O)N2CCC[C@@H](C(F)(F)F)C2)cc1N1CCCC1 ZINC000880998203 FI On-Demand Anodyne TAAR1 23 41 Cc1ccc(NC(=O)N2CCN(CCC#N)CC2)cc1N1CCCC1 ZINC000880998207 EF On-Demand Mild HTR1A 18 47 Cc1ccc(NC(=O)N2CCN(CCC#N)CC2)cc1N1CCCC1 ZINC000880998207 EF On-Demand Mild HTR1D 19 47 Cc1ccc(NC(=O)N2CCN(CCC#N)CC2)cc1N1CCCC1 ZINC000880998207 EF On-Demand Mild HTR1B 29 47 Cc1ccc(NC(=O)N2CCN(CCC#N)CC2)cc1N1CCCC1 ZINC000880998207 EF On-Demand Mild HTR2A 18 41 Cc1ccc(NC(=O)N2CCN(CCC#N)CC2)cc1N1CCCC1 ZINC000880998207 EF On-Demand Mild HTR2C 18 40 Cc1ccc(NC(=O)N2CCCCCCNC(=O)CC2)cc1N1CCCC1 ZINC000880998210 FH On-Demand Anodyne P2RY14 42 31 Cc1ccc(NC(=O)N2CC(Cc3ccco3)C2)cc1N1CCCC1 ZINC000880998225 EH On-Demand Anodyne HTR1B 18 41 COC(=O)C1(O)CN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998227 ED On-Demand Anodyne HTR1B 15 47 Cc1ccc(NC(=O)N2CCC3(CCCCO3)CC2)cc1N1CCCC1 ZINC000880998237 FI On-Demand Anodyne EPHX2 26 42 Cc1ccc(NC(=O)N2CCC3(CCCCO3)CC2)cc1N1CCCC1 ZINC000880998237 FI On-Demand Anodyne TRPM8 31 42 COC(=O)[C@@]1(C)CN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C[C@@H]1C ZINC000880998244 FG On-Demand Anodyne HTR1B 16 47 COC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccccc3)nn2)CC1 ZINC000880998253 FC On-Demand Anodyne PTR1 43 30 COC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccccc3)nn2)CC1 ZINC000880998256 FC On-Demand Anodyne PTR1 43 30 Fc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880998278 ED On-Demand Anodyne DRD3 15 46 Fc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880998278 ED On-Demand Anodyne LTA4H 31 43 Fc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880998278 ED On-Demand Anodyne HRH3 48 46 Fc1ccc(OCCn2cc(CCCN3CCOCC3)nn2)cc1 ZINC000880998278 ED On-Demand Anodyne SIGMAR1 15 49 Cc1ccc(NC(=O)N(C)OCC(F)(F)F)cc1N1CCCC1 ZINC000880998284 EH On-Demand Anodyne KCNQ2 60 35 Cc1ccc(NC(=O)N(C)OCC(F)(F)F)cc1N1CCCC1 ZINC000880998284 EH On-Demand Anodyne NPY2R 58 35 Cc1ccc(NC(=O)N(C)OCC(F)(F)F)cc1N1CCCC1 ZINC000880998284 EH On-Demand Anodyne MCHR1 17 40 Cc1ccc(NC(=O)N(C)OCC(F)(F)F)cc1N1CCCC1 ZINC000880998284 EH On-Demand Anodyne TAAR1 27 41 COc1ccc(OCCn2cc(CON)nn2)cc1 ZINC000880998286 CC On-Demand Anodyne FIMH 18 42 O=C(Cn1cc([C@@H](O)c2ccccc2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998289 FE On-Demand Anodyne HSD11B1 20 46 O=C(Cn1cc([C@H](O)c2ccccc2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998291 FE On-Demand Anodyne HSD11B1 20 46 COC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)Cc3ccccc3)nn2)CC1 ZINC000880998302 FC On-Demand Anodyne PTR1 43 30 COC(=O)C1CCN(C(=O)Cn2cc([C@H](O)Cc3ccccc3)nn2)CC1 ZINC000880998304 FC On-Demand Anodyne PTR1 43 30 Cc1ccc(NC(=O)N2CCN([S@@](C)(=N)=O)CC2)cc1N1CCCC1 ZINC000880998305 FE On-Demand Anodyne KCNQ2 46 31 Cc1ccc(NC(=O)N2CCN([S@](C)(=N)=O)CC2)cc1N1CCCC1 ZINC000880998306 FE On-Demand Anodyne KCNQ2 46 31 Cc1ccc(NC(=O)N2CCC(C)(F)CC2)cc1N1CCCC1 ZINC000880998315 DH On-Demand Anodyne HTR1B 15 46 Cc1ccc(NC(=O)N2CCC(C)(F)CC2)cc1N1CCCC1 ZINC000880998315 DH On-Demand Anodyne KCNQ2 55 32 COC(=O)Cc1cn(CCOc2cccc(Br)c2)nn1 ZINC000880998320 ED On-Demand Anodyne HMOX2 20 42 Cc1ccc(NC(=O)N2CCC(F)CC2)cc1N1CCCC1 ZINC000880998325 DH On-Demand Anodyne HTR1B 17 47 Cc1ccc(NC(=O)N2CCC(F)CC2)cc1N1CCCC1 ZINC000880998325 DH On-Demand Anodyne KCNQ2 57 32 Cc1ccc(NC(=O)N2CCC(F)CC2)cc1N1CCCC1 ZINC000880998325 DH On-Demand Anodyne TRPV1 16 46 Cc1ccc(NC(=O)N2CCC(F)CC2)cc1N1CCCC1 ZINC000880998325 DH On-Demand Anodyne NPY2R 55 36 Cc1ccc(NC(=O)N2CCC(F)CC2)cc1N1CCCC1 ZINC000880998325 DH On-Demand Anodyne EPHX2 42 44 CS[C@@H]1C[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998335 DH On-Demand Anodyne EPHX2 37 48 COc1ccc(OCCn2cc(CN3CCN(C(C)=O)CC3)nn2)cc1 ZINC000880998337 FD On-Demand Anodyne LTA4H 30 40 COc1ccc(OCCn2cc(CN3CCN(C(C)=O)CC3)nn2)cc1 ZINC000880998337 FD On-Demand Anodyne HRH3 31 42 COc1ccc(OCCn2cc(CN3CCN(C(C)=O)CC3)nn2)cc1 ZINC000880998337 FD On-Demand Anodyne MMP9 21 40 O=C(NCc1cn(CCOc2ccc(F)cc2)nn1)C(F)(F)F ZINC000880998341 ED On-Demand Anodyne MMP13 19 43 Cc1ccc(NC(=O)N2CCC(=O)[C@H](C)C2)cc1-c1ccsc1 ZINC000880998349 EI On-Demand Anodyne P2RY14 46 33 Cc1ccc(NC(=O)N2CCC(=O)[C@@H](C)C2)cc1-c1ccsc1 ZINC000880998350 EI On-Demand Anodyne P2RY14 46 33 COc1ccc(OCCn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880998367 FF On-Demand Anodyne MMP13 22 55 COc1ccc(OCCn2cc(CCCOc3cccnc3F)nn2)cc1 ZINC000880998367 FF On-Demand Anodyne MMP8 37 52 O=C(Cn1cc([C@H]2CCOC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998425 ED On-Demand Anodyne HSD11B1 42 32 O=C(Cn1cc([C@@H]2CCOC2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880998426 ED On-Demand Anodyne HSD11B1 42 32 Cc1ccc(NC(=O)N2CC(NS(C)(=O)=O)C2)cc1N1CCCC1 ZINC000880998430 FD On-Demand Anodyne EPHX2 19 40 Cc1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998433 GI On-Demand Anodyne HTR1B 15 42 Cc1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998433 GI On-Demand Anodyne KCNQ2 62 33 Cc1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998433 GI On-Demand Anodyne NPY2R 43 38 Cc1ccc(NC(=O)N2CCC[C@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998433 GI On-Demand Anodyne EPHX2 36 57 Cc1ccc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998434 GI On-Demand Anodyne HTR1B 15 42 Cc1ccc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998434 GI On-Demand Anodyne KCNQ2 62 33 Cc1ccc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998434 GI On-Demand Anodyne NPY2R 43 38 Cc1ccc(NC(=O)N2CCC[C@@](CO)(c3ccccc3)C2)cc1N1CCCC1 ZINC000880998434 GI On-Demand Anodyne EPHX2 36 57 COC(=O)Cc1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998444 DC On-Demand Anodyne ROCK1 42 42 COC(=O)Cc1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998444 DC On-Demand Anodyne MTNR1A 56 41 COC(=O)Cc1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998444 DC On-Demand Anodyne MTNR1B 55 41 COC(=O)Cc1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998444 DC On-Demand Anodyne ROCK2 48 42 C=C(C)C[C@@H](CO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998476 DG On-Demand Mild KCNQ2 57 32 C=C(C)C[C@H](CO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998480 DG On-Demand Mild KCNQ2 57 32 O[C@H](c1cn(CCOc2cccc(Br)c2)nn1)C1CC1 ZINC000880998516 EF On-Demand Anodyne HMOX2 19 40 O[C@@H](c1cn(CCOc2cccc(Br)c2)nn1)C1CC1 ZINC000880998517 EF On-Demand Anodyne HMOX2 19 40 CCOCCOC[C@@H](O)CNC(=O)Nc1ccc(C)c(-c2ccsc2)c1 ZINC000880998547 GG On-Demand Anodyne ADRB1 40 31 CCOCCOC[C@H](O)CNC(=O)Nc1ccc(C)c(-c2ccsc2)c1 ZINC000880998548 GG On-Demand Anodyne ADRB1 40 31 O=C(N[C@H]1COC[C@H]1O)c1cccnc1I ZINC000880998550 EC On-Demand Anodyne G2YM83_BOTF4 58 33 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PLG 22 45 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne ACE 66 46 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne TYR 40 46 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne OPRM1 62 44 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne OPRD1 57 44 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CELA1 23 41 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MME 125 44 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne ANPEP 65 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne TACR1 16 63 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PGC 52 31 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTRA_BOVIN 57 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne FCER2 79 35 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CASP3 35 61 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne BMP1 21 46 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CASP8 19 49 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne KLK3 86 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTSB 102 61 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PAPA1_CARPA 105 48 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CYSP_TRYCR 81 60 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CCKAR 22 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTSG 46 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTSK 56 60 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTSL 76 60 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PGA 37 40 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne NPFFR2 46 33 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne TIMP3 81 39 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CAPNS1 85 48 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MMP2 17 40 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MMP3 18 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne GRIA1 48 36 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne ECE1 30 43 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne HLA-DRB1 72 39 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CELA2A 54 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne REN 71 45 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne REN1 18 40 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MMP11 67 34 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne YARS 78 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CTSS 37 60 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CAPN1 133 52 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MMP9 23 41 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CASP1 44 61 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CAPN2 174 61 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne ACE2 69 36 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PLAU 20 45 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CASP6 37 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne CASP9 29 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne TGM2 27 41 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne LAP3 40 35 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne KLK5 42 38 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne TPSAB1 41 35 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne MMP1 23 41 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne FPR1 64 40 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne NPR 84 42 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne NAAA 70 46 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PSMB5 51 46 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne PSMB8 41 31 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne KDM1A 16 54 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne NPFFR1 55 31 O=C(N[C@H](Cc1ccccc1)C(=O)N[C@H]1COC[C@H]1O)OCc1ccccc1 ZINC000880998714 GD On-Demand Anodyne Q9NAW4_PLAFA 38 43 COc1ccc(OCCn2cc(CCNC(C)=O)nn2)cc1 ZINC000880998726 DD On-Demand Anodyne NQO2 58 46 COc1ccc(OCCn2cc(CCNC(C)=O)nn2)cc1 ZINC000880998726 DD On-Demand Anodyne MMP13 23 40 COc1ccc(OCCn2cc(CCNC(C)=O)nn2)cc1 ZINC000880998726 DD On-Demand Anodyne MTNR1A 115 46 COc1ccc(OCCn2cc(CCNC(C)=O)nn2)cc1 ZINC000880998726 DD On-Demand Anodyne MTNR1B 100 46 COc1ccc(OCCn2cc(CCNC(C)=O)nn2)cc1 ZINC000880998726 DD On-Demand Anodyne MMP9 19 40 COc1ccc(OCCn2cc(CN(C)C(=O)OC(C)(C)C)nn2)cc1 ZINC000880998727 FF On-Demand Anodyne MMP13 25 42 COc1ccc(OCCn2cc(CN(C)C(=O)OC(C)(C)C)nn2)cc1 ZINC000880998727 FF On-Demand Anodyne MMP8 38 42 COc1ccc(OCCn2cc(CN(C)C(=O)OC(C)(C)C)nn2)cc1 ZINC000880998727 FF On-Demand Anodyne MMP9 20 42 O[C@@]1(c2cn(CCOc3ccc(F)cc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880998740 DF On-Demand Anodyne ALOX5AP 34 43 O[C@]1(c2cn(CCOc3ccc(F)cc3)nn2)C[C@H]2CC[C@H]1C2 ZINC000880998741 DF On-Demand Anodyne ALOX5AP 34 43 Cc1ccc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)cc1N1CCCC1 ZINC000880998812 GG On-Demand Mild HTR1B 15 43 Cc1ccc(NC(=O)N2CCN(c3ccc(C#N)nc3)CC2)cc1N1CCCC1 ZINC000880998812 GG On-Demand Mild PDGFRB 43 39 Cc1ccc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880998829 EH On-Demand Anodyne NPY2R 43 38 Cc1ccc(NC(=O)N2CCC[C@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880998829 EH On-Demand Anodyne EPHX2 22 44 Cc1ccc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880998831 EH On-Demand Anodyne NPY2R 43 38 Cc1ccc(NC(=O)N2CCC[C@@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880998831 EH On-Demand Anodyne EPHX2 22 44 Cc1ccc(NC(=O)N(C)C[C@@H]2CN(C)CCO2)cc1N1CCCC1 ZINC000880998833 EE On-Demand Anodyne HTR1B 15 41 Cc1ccc(NC(=O)N(C)C[C@H]2CN(C)CCO2)cc1N1CCCC1 ZINC000880998835 EE On-Demand Anodyne HTR1B 15 41 O=C1CCC[C@@H](c2cn(CC(=O)NC3C4CC5CC(C4)CC3C5)nn2)C1 ZINC000880998837 FE On-Demand Anodyne HSD11B1 40 31 O=C1CCC[C@H](c2cn(CC(=O)NC3C4CC5CC(C4)CC3C5)nn2)C1 ZINC000880998839 FE On-Demand Anodyne HSD11B1 40 31 COC[C@H](C)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998841 CF On-Demand Anodyne KCNQ2 64 33 Cc1ccc(NC(=O)N2CCNC(=O)C2)cc1-c1ccsc1 ZINC000880998849 DF On-Demand Anodyne P2RY14 52 33 Cc1ccc(NC(=O)N2CCO[C@@H](c3noc(C4CC4)n3)C2)cc1N1CCCC1 ZINC000880998859 GG On-Demand Anodyne ETHR 45 35 Cc1ccc(NC(=O)N2CCO[C@H](c3noc(C4CC4)n3)C2)cc1N1CCCC1 ZINC000880998861 GG On-Demand Anodyne ETHR 45 35 COC(=O)C1CCN(C(=O)Cn2cc(-c3cccnc3F)nn2)CC1 ZINC000880998863 EC On-Demand Anodyne PTR1 44 31 Cc1ccc(NC(=O)N2CCC(CO)(CO)CC2)cc1N1CCCC1 ZINC000880998867 EE On-Demand Anodyne HTR1D 15 45 Cc1ccc(NC(=O)N2CCC(CO)(CO)CC2)cc1N1CCCC1 ZINC000880998867 EE On-Demand Anodyne HTR1B 21 45 Cc1ccc(NC(=O)N2CCC(CO)(CO)CC2)cc1N1CCCC1 ZINC000880998867 EE On-Demand Anodyne KCNQ2 60 33 Cc1ccc(NC(=O)N2CCC[C@H](NS(C)(=O)=O)C2)cc1N1CCCC1 ZINC000880998873 GE On-Demand Anodyne EPHX2 20 49 Cc1ccc(NC(=O)N2CCC[C@@H](NS(C)(=O)=O)C2)cc1N1CCCC1 ZINC000880998875 GE On-Demand Anodyne EPHX2 20 49 CCN1CC[C@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998881 EE On-Demand Anodyne CCKAR 32 44 CCN1CC[C@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998881 EE On-Demand Anodyne CCKBR 53 44 CCN1CC[C@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998881 EE On-Demand Anodyne EPHX2 30 42 CCN1CC[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998883 EE On-Demand Anodyne CCKAR 32 44 CCN1CC[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998883 EE On-Demand Anodyne CCKBR 53 44 CCN1CC[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1=O ZINC000880998883 EE On-Demand Anodyne EPHX2 30 42 Cc1ccc(NC(=O)N2CCC[C@H](CO)C2)cc1-c1ccsc1 ZINC000880998893 EH On-Demand Anodyne P2RY14 45 32 Cc1ccc(NC(=O)N2CCC[C@@H](CO)C2)cc1-c1ccsc1 ZINC000880998894 EH On-Demand Anodyne P2RY14 45 32 Cc1ccc(NC(=O)N2CCC(NC(=O)C(C)C)CC2)cc1-c1ccsc1 ZINC000880998898 GI On-Demand Anodyne MAPK14 18 42 C=CC[C@H]1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998899 DI On-Demand Mild HTR1B 16 40 C=CC[C@@H]1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880998901 DI On-Demand Mild HTR1B 16 40 CCN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880998920 EI On-Demand Anodyne MAPK14 20 45 CCN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880998920 EI On-Demand Anodyne EPHX2 46 46 CCN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880998920 EI On-Demand Anodyne CXCR3 21 47 Cc1ccc(NC(=O)N2CCC[C@H](C3OCCO3)C2)cc1-c1ccsc1 ZINC000880998930 FI On-Demand Anodyne P2RY14 42 32 Cc1ccc(NC(=O)N2CCC[C@@H](C3OCCO3)C2)cc1-c1ccsc1 ZINC000880998931 FI On-Demand Anodyne P2RY14 42 32 COC(=O)Cc1cn(CC(=O)NC2C3CC4CC(C3)CC2C4)nn1 ZINC000880998943 EC On-Demand Anodyne HSD11B1 41 32 Cc1ccc(NC(=O)N2CCC(C)(N3CCOCC3)CC2)cc1N1CCCC1 ZINC000880998947 GG On-Demand Anodyne HTR1B 16 42 COc1ccc(CN(CCO)C(=O)Nc2ccc(C)c(N3CCCC3)c2)cc1 ZINC000880998949 GH On-Demand Anodyne BMP1 21 40 COc1ccc(CN(CCO)C(=O)Nc2ccc(C)c(N3CCCC3)c2)cc1 ZINC000880998949 GH On-Demand Anodyne ROCK2 17 44 COc1ccc(CN(CCO)C(=O)Nc2ccc(C)c(N3CCCC3)c2)cc1 ZINC000880998949 GH On-Demand Anodyne GALR2 40 33 COc1ccc(CN(CCO)C(=O)Nc2ccc(C)c(N3CCCC3)c2)cc1 ZINC000880998949 GH On-Demand Anodyne MCHR1 25 41 C=C[C@](C)(O)c1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998963 DC On-Demand Mild ROCK2 31 40 C=C[C@@](C)(O)c1cn(CC(=O)NCc2cccc(OC)c2)nn1 ZINC000880998964 DC On-Demand Mild ROCK2 31 40 Cc1ccc(NC(=O)N2CCC(F)(F)CC2)cc1N1CCCC1 ZINC000880998967 DH On-Demand Anodyne HTR1B 15 47 Cc1ccc(NC(=O)N2CCC(F)(F)CC2)cc1N1CCCC1 ZINC000880998967 DH On-Demand Anodyne KCNQ2 47 33 COC(=O)C[C@@H](C)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998980 DF On-Demand Anodyne KCNQ2 63 33 COC[C@@H]1CCCN1C(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880998992 DG On-Demand Anodyne HTR1B 15 40 Cc1ccc(NC(=O)N2CCC3(CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880998995 FH On-Demand Anodyne HTR1D 17 53 Cc1ccc(NC(=O)N2CCC3(CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880998995 FH On-Demand Anodyne HTR1B 21 53 Cc1ccc(NC(=O)N2CCC3(CCN(C)CC3)CC2)cc1N1CCCC1 ZINC000880998995 FH On-Demand Anodyne TRPM8 27 40 Cc1ccc(NC(=O)N2CCC(C(C)(C)O)CC2)cc1N1CCCC1 ZINC000880999038 EH On-Demand Anodyne HTR1B 15 44 Cc1ccc(NC(=O)N2CCC(C(C)(C)O)CC2)cc1N1CCCC1 ZINC000880999038 EH On-Demand Anodyne NPY2R 61 37 Cc1ccc(NC(=O)N2CCC(C(C)(C)O)CC2)cc1N1CCCC1 ZINC000880999038 EH On-Demand Anodyne EPHX2 32 41 COC(=O)C1CCN(C(=O)Cn2cc(-c3cccnc3Cl)nn2)CC1 ZINC000880999042 FD On-Demand Anodyne IL2RA 50 34 COC(=O)C1CCN(C(=O)Cn2cc(-c3cccnc3Cl)nn2)CC1 ZINC000880999042 FD On-Demand Anodyne PTR1 44 32 COC[C@@H](O)Cc1cn(CC(=O)Nc2ccc3c(c2)CCC3)nn1 ZINC000880999064 EC On-Demand Anodyne ACOX1 19 44 Cc1ccc(NC(=O)N2CCO[C@@H](Cn3cccn3)C2)cc1-c1ccsc1 ZINC000880999094 GH On-Demand Anodyne P2RY14 45 32 Cc1ccc(NC(=O)N2CCO[C@H](Cn3cccn3)C2)cc1-c1ccsc1 ZINC000880999095 GH On-Demand Anodyne P2RY14 45 32 CCc1nnc2n1CCN(C(=O)Nc1ccc(C)c(-c3ccsc3)c1)C2 ZINC000880999103 FH On-Demand Anodyne P2RY14 55 36 C[C@H](O)c1ccc(OCc2cn(CC(=O)Nc3ccc4c(c3)CCC4)nn2)cc1 ZINC000880999119 GG On-Demand Anodyne ACOX1 18 43 Cc1ccc(NC(=O)N2CCN(c3cnccn3)CC2)cc1-c1ccsc1 ZINC000880999126 GH On-Demand Anodyne KARS 46 33 CNc1nc(C(=O)Nc2ccn(C3CCSCC3)n2)cs1 ZINC000880999132 DF On-Demand Anodyne TRPC6 44 36 Cc1ccc(NC(=O)N2CCN(CC(=O)NC3CC3)CC2)cc1-c1ccsc1 ZINC000880999133 GG On-Demand Anodyne MAPK14 25 44 Cc1ccc(NC(=O)N2CCCO[C@@H](C)C2)cc1-c1ccsc1 ZINC000880999134 EI On-Demand Anodyne P2RY14 45 32 Cc1ccc(NC(=O)N2CCCO[C@H](C)C2)cc1-c1ccsc1 ZINC000880999135 EI On-Demand Anodyne P2RY14 45 32 COC(=O)Cc1cn(Cc2ccc(C(C)(C)C)cc2)nn1 ZINC000880999137 CE On-Demand Anodyne KDM1A 15 42 Cc1ccc(NC(=O)N2CCCSCC2)cc1-c1ccsc1 ZINC000880999148 EJ On-Demand Anodyne P2RY14 42 32 Cc1ccc(NC(=O)N2CCC(C)(N3CCCC3)CC2)cc1N1CCCC1 ZINC000880999157 FI On-Demand Anodyne CCR5 23 42 Cc1ccc(NC(=O)N2CCC[C@H]2C(=O)N(C)C)cc1N1CCCC1 ZINC000880999158 EF On-Demand Anodyne AVPR2 22 46 Cc1ccc(NC(=O)N2CCC[C@H]2C(=O)N(C)C)cc1N1CCCC1 ZINC000880999158 EF On-Demand Anodyne UL80 40 42 Cc1ccc(NC(=O)N2CCCNC(=O)C2)cc1N1CCCC1 ZINC000880999165 DD On-Demand Anodyne P2RY14 46 32 Cc1ccc(NC(=O)N2CCC(O)CC2)cc1N1CCCC1 ZINC000880999170 DF On-Demand Anodyne HTR1D 17 47 Cc1ccc(NC(=O)N2CCC(O)CC2)cc1N1CCCC1 ZINC000880999170 DF On-Demand Anodyne HTR1B 20 47 Cc1ccc(NC(=O)N2CCC(O)CC2)cc1N1CCCC1 ZINC000880999170 DF On-Demand Anodyne KCNQ2 51 32 Cc1ccc(NC(=O)N2CCC(O)CC2)cc1N1CCCC1 ZINC000880999170 DF On-Demand Anodyne EPHX2 30 42 CCN(CC)C(=O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999172 EF On-Demand Anodyne KCNQ2 61 33 CCN(CC)C(=O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999172 EF On-Demand Anodyne NPY2R 59 36 Cc1ccc(NC(=O)N2CCC(c3nnnn3C)CC2)cc1N1CCCC1 ZINC000880999173 FF On-Demand Anodyne HTR1B 15 42 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc(C)c(N3CCCC3)c1)CC2 ZINC000880999174 GI On-Demand Anodyne KCNQ2 61 34 CC(=O)Nc1cccc2c1CN(C(=O)Nc1ccc(C)c(N3CCCC3)c1)CC2 ZINC000880999174 GI On-Demand Anodyne P2RY14 51 36 CCC[C@@H](CCO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999181 DG On-Demand Anodyne KCNQ2 62 38 CCC[C@H](CCO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999182 DG On-Demand Anodyne KCNQ2 62 38 COC(=O)[C@@]12C[C@@H](NC(=O)Nc3ccc(C)c(N4CCCC4)c3)C[C@@H]1C2 ZINC000880999183 FG On-Demand Anodyne EPHX2 38 43 CC[C@@H](NC(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@H]1CCCOC1 ZINC000880999185 EH On-Demand Anodyne KCNQ2 40 32 CC[C@@H](NC(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@H]1CCCOC1 ZINC000880999185 EH On-Demand Anodyne NPY2R 29 40 CC[C@@H](NC(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@@H]1CCCOC1 ZINC000880999186 EH On-Demand Anodyne KCNQ2 40 32 CC[C@@H](NC(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@@H]1CCCOC1 ZINC000880999186 EH On-Demand Anodyne NPY2R 29 40 Cc1ccc(NC(=O)N2CCC3(CCNC3=O)CC2)cc1N1CCCC1 ZINC000880999193 FF On-Demand Anodyne HTR1B 15 42 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999196 FH On-Demand Anodyne HTR1B 15 43 CO[C@@]1(C(F)(F)F)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999196 FH On-Demand Anodyne EPHX2 35 41 Cc1ccc(NC(=O)N(C2CC2)C2CC2)cc1N1CCCC1 ZINC000880999206 CH On-Demand Anodyne KCNQ2 60 32 Cc1ccc(NC(=O)N(C2CC2)C2CC2)cc1N1CCCC1 ZINC000880999206 CH On-Demand Anodyne NPY2R 49 37 Cc1ccc(NC(=O)N(C2CC2)C2CC2)cc1N1CCCC1 ZINC000880999206 CH On-Demand Anodyne TAAR1 26 40 Cc1ccc(NC(=O)N2CCN(C)C(C)(C)CC2)cc1N1CCCC1 ZINC000880999207 EH On-Demand Anodyne HTR1B 15 48 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999210 FG On-Demand Anodyne HTR1B 16 41 CCOC(=O)[C@H](C)C1CN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999210 FG On-Demand Anodyne KCNQ2 53 34 O=C(Cn1cc([C@H]2CCCCO2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880999217 EE On-Demand Anodyne HSD11B1 42 33 O=C(Cn1cc([C@@H]2CCCCO2)nn1)NC1C2CC3CC(C2)CC1C3 ZINC000880999218 EE On-Demand Anodyne HSD11B1 42 33 Cc1ccc(NC(=O)N2CCC(CCO)(CCO)CC2)cc1N1CCCC1 ZINC000880999231 GF On-Demand Anodyne KCNQ2 45 30 CO[C@@H]1C[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999238 DF On-Demand Anodyne HTR1B 15 40 CO[C@@H]1C[C@@H](NC(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999238 DF On-Demand Anodyne EPHX2 46 48 CCC1(N(C)C)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999254 FH On-Demand Anodyne HTR1B 18 48 CCC1(N(C)C)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999254 FH On-Demand Anodyne KCNQ2 54 32 CCC1(N(C)C)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999254 FH On-Demand Anodyne NPY2R 42 32 Cc1ccc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)cc1N1CCCC1 ZINC000880999255 FJ On-Demand Anodyne HTR1B 16 46 Cc1ccc(NC(=O)N2CCC[C@H](OC3CCC3)CC2)cc1N1CCCC1 ZINC000880999255 FJ On-Demand Anodyne EPHX2 29 42 Cc1ccc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)cc1N1CCCC1 ZINC000880999256 FJ On-Demand Anodyne HTR1B 16 46 Cc1ccc(NC(=O)N2CCC[C@@H](OC3CCC3)CC2)cc1N1CCCC1 ZINC000880999256 FJ On-Demand Anodyne EPHX2 29 42 Cc1ccc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880999265 EG On-Demand Anodyne NPY2R 61 37 Cc1ccc(NC(=O)N2CC[C@@H](C(C)(C)O)C2)cc1N1CCCC1 ZINC000880999265 EG On-Demand Anodyne EPHX2 25 40 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999276 GG On-Demand Anodyne DRD4 15 40 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999276 GG On-Demand Anodyne MAPK14 19 44 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999276 GG On-Demand Anodyne EPHX2 36 43 CNC(=O)CN1CCC(NC(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999276 GG On-Demand Anodyne CXCR3 20 44 O=C(Cn1cc(CCCOc2cccnc2F)nn1)Nc1ccc2c(c1)CCC2 ZINC000880999484 GF On-Demand Anodyne MMP8 17 43 CC(=O)N1CCN(Cc2cn(Cc3ccccc3[N+](=O)[O-])nn2)CC1 ZINC000880999502 EC On-Demand Bother COLA 81 32 Cc1ccc(NC(=O)N2CCN(c3ncccn3)CC2)cc1-c1ccsc1 ZINC000880999529 GH On-Demand Anodyne PDGFRB 45 38 Cc1ccc(NC(=O)N2CCN(c3ncccn3)CC2)cc1-c1ccsc1 ZINC000880999529 GH On-Demand Anodyne P2RY14 48 34 Cc1ccc(NC(=O)N2CCN(Cc3cnn(C)c3)CC2)cc1-c1ccsc1 ZINC000880999533 GH On-Demand Anodyne P2RY14 45 32 CCC(=O)N1CCCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999537 FI On-Demand Anodyne P2RY14 50 34 COC[C@@H]1CCCN1NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999562 EF On-Demand Anodyne CASP7 40 35 COC(=O)CNC(=O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999565 ED On-Demand Anodyne KCNQ2 66 35 Cc1ccc(NC(=O)N2CCN(C)C(=O)C2)cc1N1CCCC1 ZINC000880999569 DD On-Demand Anodyne HTR1B 16 48 COC(=O)C1CCN(C(=O)Cn2cc(CCCCCCO)nn2)CC1 ZINC000880999575 FC On-Demand Anodyne PTR1 45 33 C=CCOCCNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999636 DF On-Demand Mild HRH2 23 41 Cc1ccc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)cc1N1CCCC1 ZINC000880999668 GG On-Demand Anodyne HTR1D 15 40 Cc1ccc(NC(=O)N2CCC([C@H](O)c3ccnn3C)CC2)cc1N1CCCC1 ZINC000880999668 GG On-Demand Anodyne HTR1B 21 40 Cc1ccc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)cc1N1CCCC1 ZINC000880999673 GG On-Demand Anodyne HTR1D 15 40 Cc1ccc(NC(=O)N2CCC([C@@H](O)c3ccnn3C)CC2)cc1N1CCCC1 ZINC000880999673 GG On-Demand Anodyne HTR1B 21 40 COC[C@@H](O)Cc1cn(Cc2ccc(F)cc2Cl)nn1 ZINC000880999689 CD On-Demand Anodyne P2RX7 46 37 Cc1noc(C2CCN(C(=O)Nc3ccc(C)c(-c4ccsc4)c3)CC2)n1 ZINC000880999702 GJ On-Demand Anodyne SMO 35 43 Cc1noc(C2CCN(C(=O)Nc3ccc(C)c(-c4ccsc4)c3)CC2)n1 ZINC000880999702 GJ On-Demand Anodyne ETHR 53 36 Cc1ccc(NC(=O)N2CCOC3(CCN(C)CC3)C2)cc1N1CCCC1 ZINC000880999704 FF On-Demand Anodyne HTR1B 18 45 Cc1ccc(NC(=O)N2CCOC3(CCN(C)CC3)C2)cc1N1CCCC1 ZINC000880999704 FF On-Demand Anodyne EPHX2 31 51 CC(=O)N1CCN(C(=O)Nc2ccc(C)c(-c3ccsc3)c2)CC1 ZINC000880999714 EG On-Demand Anodyne P2RY14 52 34 COC1(CO)CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999731 EF On-Demand Anodyne HTR1B 18 47 Cc1ccc(NC(=O)N(C)[C@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999733 FH On-Demand Anodyne KCNQ2 69 38 Cc1ccc(NC(=O)N(C)[C@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999733 FH On-Demand Anodyne NPY2R 79 34 Cc1ccc(NC(=O)N(C)[C@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999733 FH On-Demand Anodyne NPY5R 35 48 Cc1ccc(NC(=O)N(C)[C@@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999735 FH On-Demand Anodyne KCNQ2 69 38 Cc1ccc(NC(=O)N(C)[C@@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999735 FH On-Demand Anodyne NPY2R 79 34 Cc1ccc(NC(=O)N(C)[C@@H](CO)Cc2ccccc2)cc1N1CCCC1 ZINC000880999735 FH On-Demand Anodyne NPY5R 35 48 COC(=O)C1CCN(C(=O)Cn2cc(-c3c4c(nn3C)CCCC4)nn2)CC1 ZINC000880999738 GC On-Demand Anodyne IL2RA 40 31 Cc1ccc(NC(=O)N2CCN(C)CC2)cc1-c1ccsc1 ZINC000880999747 DH On-Demand Anodyne HTR1B 17 46 Cc1ccc(NC(=O)N2CCN(C)CC2)cc1-c1ccsc1 ZINC000880999747 DH On-Demand Anodyne P2RY14 42 34 CCNC(=O)CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999824 DD On-Demand Anodyne KCNQ2 64 34 Cc1ccc(NC(=O)N2CCCC(F)(F)C2)cc1N1CCCC1 ZINC000880999831 DH On-Demand Anodyne EPHX2 37 42 COC(=O)c1occc1CNC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999836 FG On-Demand Anodyne NPY1R 23 40 C#CC1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999841 DG On-Demand Mild HTR1B 16 48 C#CC1CCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)CC1 ZINC000880999841 DG On-Demand Mild EPHX2 20 40 C#C[C@H](CO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999859 CD On-Demand Mild KCNQ2 64 33 C#C[C@@H](CO)NC(=O)Nc1ccc(C)c(N2CCCC2)c1 ZINC000880999860 CD On-Demand Mild KCNQ2 64 33 Cc1cncc(CCNC(=O)Nc2ccc(C)c(N3CCCC3)c2)n1 ZINC000880999862 EG On-Demand Anodyne HTR1D 19 40 Cc1cncc(CCNC(=O)Nc2ccc(C)c(N3CCCC3)c2)n1 ZINC000880999862 EG On-Demand Anodyne HTR1B 25 40 Cc1ccc(NC(=O)N(C)CCN2CCCCC2)cc1N1CCCC1 ZINC000880999870 EH On-Demand Anodyne DRD2 15 43 Cc1ccc(NC(=O)N(C)CCN2CCCCC2)cc1N1CCCC1 ZINC000880999870 EH On-Demand Anodyne HTR2A 27 43 Cc1ccc(NC(=O)N(C)CCN2CCCCC2)cc1N1CCCC1 ZINC000880999870 EH On-Demand Anodyne DRD3 29 43 Cc1ccc(NC(=O)N(C)CCN2CCCCC2)cc1N1CCCC1 ZINC000880999870 EH On-Demand Anodyne KCNQ2 50 33 Cc1ccc(NC(=O)N2CCC3(CC2)CC3(F)F)cc1N1CCCC1 ZINC000880999879 EI On-Demand Anodyne HTR1B 15 44 Cc1ccc(NC(=O)N2CCC3(CC2)CC3(F)F)cc1N1CCCC1 ZINC000880999879 EI On-Demand Anodyne TRPV1 15 40 CC(C)(C)OC(=O)NCC(=O)NCc1cn(Cc2ccc(F)cc2Cl)nn1 ZINC000880999880 GE On-Demand Anodyne P2RX7 60 44 Cc1ccc(NC(=O)N2CCC[C@@H](O)C2)cc1N1CCCC1 ZINC000880999882 DF On-Demand Anodyne HTR1B 15 44 Cc1ccc(NC(=O)N2CCC[C@@H](O)C2)cc1N1CCCC1 ZINC000880999882 DF On-Demand Anodyne EPHX2 21 44 Cc1ccc(NC(=O)N(CCN2CCOCC2)CC2CC2)cc1N1CCCC1 ZINC000880999891 GG On-Demand Anodyne CASR 64 47 OC1(c2cn(Cc3ccc(F)cc3Cl)nn2)CCCCC1 ZINC000880999894 DG On-Demand Anodyne P2RX7 47 37 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999896 EF On-Demand Anodyne HTR1B 15 43 CO[C@]1(CO)CCCN(C(=O)Nc2ccc(C)c(N3CCCC3)c2)C1 ZINC000880999896 EF On-Demand Anodyne EPHX2 29 41 Cc1ccc(NC(=O)N2CCN(Cc3nc[nH]n3)CC2)cc1N1CCCC1 ZINC000880999897 FE On-Demand Anodyne HTR1D 19 44 Cc1ccc(NC(=O)N2CCN(Cc3nc[nH]n3)CC2)cc1N1CCCC1 ZINC000880999897 FE On-Demand Anodyne HTR1B 28 44 Cc1ccc(NC(=O)N2CCN(Cc3nc[nH]n3)CC2)cc1N1CCCC1 ZINC000880999897 FE On-Demand Anodyne PDGFRB 47 35 CC(=O)N1CCN(Cc2cn(Cc3ccc(F)cc3Cl)nn2)CC1 ZINC000880999898 FD On-Demand Anodyne P2RX7 71 42 C=CCN(C(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@@H](C)COC ZINC000880999899 EH On-Demand Mild KCNQ2 43 33 C=CCN(C(=O)Nc1ccc(C)c(N2CCCC2)c1)[C@H](C)COC ZINC000880999900 EH On-Demand Mild KCNQ2 43 33 Cc1ccc(NC(=O)N2CCC(O)(CO)CC2)cc1N1CCCC1 ZINC000880999905 ED On-Demand Anodyne HTR1B 20 44 Cc1ccc(NC(=O)N2CCC(O)(CO)CC2)cc1N1CCCC1 ZINC000880999905 ED On-Demand Anodyne KCNQ2 50 33 Cc1ccc(NC(=O)N2CCC(O)(CO)CC2)cc1N1CCCC1 ZINC000880999905 ED On-Demand Anodyne S1PR2 28 41 COC(=O)C1CCN(C(=O)Cn2cc([C@H](O)c3ccc(C)cc3)nn2)CC1 ZINC000880999912 FD On-Demand Anodyne PTR1 43 30 COC(=O)C1CCN(C(=O)Cn2cc([C@@H](O)c3ccc(C)cc3)nn2)CC1 ZINC000880999913 FD On-Demand Anodyne PTR1 43 30 CC(C)(C)OC(=O)N1CCC[C@H]1c1cn(Cc2nnc(-c3ccccc3)o2)nn1 ZINC000880999943 GG On-Demand Anodyne CPT1A 63 34 CC(C)(C)OC(=O)N1CCC[C@@H]1c1cn(Cc2nnc(-c3ccccc3)o2)nn1 ZINC000880999944 GG On-Demand Anodyne CPT1A 63 34 Cc1ccc(NC(=O)N2CCNC(=O)CC2)cc1-c1ccsc1 ZINC000880999970 EG On-Demand Anodyne P2RY14 52 33 CN(C(=O)Cn1cc([C@H]2CCOC2)nn1)C(c1ccccc1)c1ccccc1 ZINC000880999980 GG On-Demand Anodyne OPRK1 24 40 CN(C(=O)Cn1cc([C@@H]2CCOC2)nn1)C(c1ccccc1)c1ccccc1 ZINC000880999981 GG On-Demand Anodyne OPRK1 24 40 CC(=O)N1CCN(Cc2cn(Cc3ccc(C(C)(C)C)cc3)nn2)CC1 ZINC000880999995 FE On-Demand Anodyne KDM1A 17 46